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Discovery of N-substituted-2-oxoindolin benzoylhydrazines as c-MET/SMO modulators in EGFRi-resistant non-small cell lung cancer.
RSC Med Chem 16: 77-97 (0)
University of Campania
New anti-ovarian cancer quinolone derivatives acting by modulating microRNA processing machinery.
RSC Med Chem 16: 98-124 (0)
University of Perugia
Design, synthesis, and structure-activity relationship studies of 6H-benzo[b]indeno[1,2-d]thiophen-6-one derivatives as DYRK1A/CLK1/CLK4/haspin inhibitors.
RSC Med Chem 16: 179-99 (0)
Universite Claude Bernard Lyon 1
Design, synthesis, and evaluation of benzhydrylpiperazine-based novel dual COX-2/5-LOX inhibitors with anti-inflammatory and anti-cancer activity.
RSC Med Chem 16: 200-20 (0)
India Institute of Technology (Banaras Hindu University)
Inhibition of monoamine oxidases by heterocyclic derived conjugated dienones: synthesis and in vitro and in silico investigations.
RSC Med Chem 16: 221-31 (0)
Amrita School of Pharmacy
Development, biological evaluation, and molecular modelling of some benzene-sulfonamide derivatives as protein tyrosine phosphatase-1B inhibitors for managing diabetes mellitus and associated metabolic disorders.
RSC Med Chem 16: 247-73 (0)
Suez Canal University
Breaking boundaries in diabetic nephropathy treatment: design and synthesis of novel steroidal SGLT2 inhibitors.
RSC Med Chem 16: 296-311 (0)
Institute of Advanced Study in Science and Technology
Novel benzenesulfonamides containing a dual triazole moiety with selective carbonic anhydrase inhibition and anticancer activity.
RSC Med Chem 16: 324-45 (0)
University of Prishtina
Ligand-centred phenotype-driven development of potent kinase inhibitors against oesophageal cancer.
RSC Med Chem 16: 379-91 (0)
University of Edinburgh
Medicinal chemistry-based perspectives on thiophene and its derivatives: exploring structural insights to discover plausible druggable leads.
RSC Med Chem 16: 481-510 (0)
Birla Institute of Technology and Sciences Pilani Pilani Campus
Distinctive roles of aquaporins and novel therapeutic opportunities against cancer.
RSC Med Chem 16: 640-651 (0)
Gachon University
Synthesis, in silico and bio-evaluation studies of new isothiocyanate derivatives with respect to COX inhibition and H2S release profiles.
RSC Med Chem 16: 732-746 (0)
Canakkale Onsekiz Mart University
Design and synthesis of novel cathepsin C inhibitors with anti-inflammatory activity.
RSC Med Chem 16: 876-891 (0)
Fuyang Normal University
Novel rhodanine-thiazole hybrids as potential antidiabetic agents: a structure-based drug design approach.
RSC Med Chem 16: 927-944 (0)
KLE Academy of Higher education and Research Belagavi
3-Thio-3,4,5-trisubstituted-1,2,4-triazoles: high affinity somatostatin receptor-4 agonist synthesis and structure-activity relationships.
RSC Med Chem 16: 945-960 (0)
Southern Illinois University
Novel sigma 1-antagonists with cis-(+)-normetazocine scaffold: synthesis, molecular modeling, and antinociceptive effect.
RSC Med Chem 16: 1172-1187 (0)
University of Catania
Probing structural requirements for thiazole-based mimetics of sunitinib as potent VEGFR-2 inhibitors.
RSC Med Chem 16: 1329-1349 (0)
Department of Medicinal Chemistry, Faculty of Pharmacy, Mansoura University Mansoura