Report error Found 33 Enz. Inhib. hit(s) with all data for entry = 50023603
TargetHigh affinity nerve growth factor receptor(Human)
University of British Columbia
Curated by ChEMBL
University of British Columbia
Curated by ChEMBL
Affinity DataIC50: 1nMAssay Description:Inhibition of TRKA (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:Inhibition of TRKB (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 5nMAssay Description:Inhibition of TRKC (unknown origin)More data for this Ligand-Target Pair
TargetHigh affinity nerve growth factor receptor(Human)
University of British Columbia
Curated by ChEMBL
University of British Columbia
Curated by ChEMBL
Affinity DataIC50: 6.5nMAssay Description:Inhibition of TRKA (unknown origin)More data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase ROS(Human)
University of British Columbia
Curated by ChEMBL
University of British Columbia
Curated by ChEMBL
Affinity DataIC50: 7nMAssay Description:Inhibition of ROS1 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 8.10nMAssay Description:Inhibition of TRKB (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 11nMAssay Description:Inhibition of TRKC (unknown origin)More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase receptor R3(Human)
University of British Columbia
Curated by ChEMBL
University of British Columbia
Curated by ChEMBL
Affinity DataIC50: 12nMAssay Description:Inhibition of ALK1 (unknown origin)More data for this Ligand-Target Pair
TargetHigh affinity nerve growth factor receptor(Human)
University of British Columbia
Curated by ChEMBL
University of British Columbia
Curated by ChEMBL
Affinity DataKd: 31nMAssay Description:Binding affinity to TRKA (unknown origin) assessed as dissociation constant by KINOMEscan assayMore data for this Ligand-Target Pair
Ligand Info
TargetHigh affinity nerve growth factor receptor(Human)
University of British Columbia
Curated by ChEMBL
University of British Columbia
Curated by ChEMBL
Affinity DataKd: 36nMAssay Description:Binding affinity to TRKA (unknown origin) assessed as dissociation constantMore data for this Ligand-Target Pair
Ligand Info
TargetHigh affinity nerve growth factor receptor(Human)
University of British Columbia
Curated by ChEMBL
University of British Columbia
Curated by ChEMBL
Affinity DataKd: 52nMAssay Description:Binding affinity to TRKA (unknown origin) assessed as dissociation constant by KINOMEscan assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataKd: 60nMAssay Description:Binding affinity to TRKB (unknown origin) assessed as dissociation constant by KINOMEscan assayMore data for this Ligand-Target Pair
Ligand Info
TargetReceptor-type tyrosine-protein kinase FLT3(Human)
University of British Columbia
Curated by ChEMBL
University of British Columbia
Curated by ChEMBL
Affinity DataIC50: 70nMAssay Description:Inhibition of FLT3 (unknown origin)More data for this Ligand-Target Pair
Ligand Info
Affinity DataKd: 150nMAssay Description:Binding affinity to TRKB (unknown origin) assessed as dissociation constant by KINOMEscan assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 177nMAssay Description:Inhibition of JAK2 (unknown origin) by Z-LYTE Kinase assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataKd: 180nMAssay Description:Binding affinity to TRKB (unknown origin) assessed as dissociation constant by KINOMEscan assayMore data for this Ligand-Target Pair
Ligand Info
TargetHigh affinity nerve growth factor receptor(Human)
University of British Columbia
Curated by ChEMBL
University of British Columbia
Curated by ChEMBL
Affinity DataKd: 220nMAssay Description:Binding affinity to TRKA (unknown origin) assessed as dissociation constant by KINOMEscan assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataKd: 230nMAssay Description:Binding affinity to TRKC (unknown origin) assessed as dissociation constant by KINOMEscan assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataKd: 280nMAssay Description:Binding affinity to TRKC (unknown origin) assessed as dissociation constant by KINOMEscan assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 361nMAssay Description:Inhibition of JAK2 (unknown origin) by Z-LYTE Kinase assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataKd: 470nMAssay Description:Binding affinity to TRKC (unknown origin) assessed as dissociation constant by KINOMEscan assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 530nMAssay Description:Inhibition of JAK2 (unknown origin) by Z-LYTE Kinase assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 576nMAssay Description:Inhibition of TNK2 (unknown origin)More data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Human)
University of British Columbia
Curated by ChEMBL
University of British Columbia
Curated by ChEMBL
Affinity DataKd: 640nMAssay Description:Binding affinity to SRC (unknown origin) assessed as dissociation constantMore data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 663nMAssay Description:Inhibition of JAK2 (unknown origin) by Z-LYTE Kinase assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 750nMAssay Description:Inhibition of MK2 (unknown origin)More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 870nMAssay Description:Inhibition of NEK2 (unknown origin)More data for this Ligand-Target Pair
Ligand Info
Affinity DataKd: 1.10E+3nMAssay Description:Binding affinity to JAK2 (unknown origin) assessed as dissociation constantMore data for this Ligand-Target Pair
Ligand Info
TargetProto-oncogene tyrosine-protein kinase Src(Human)
University of British Columbia
Curated by ChEMBL
University of British Columbia
Curated by ChEMBL
Affinity DataIC50: 1.11E+3nMAssay Description:Inhibition of SRC (unknown origin) by Z-LYTE Kinase assayMore data for this Ligand-Target Pair
Ligand Info
TargetProto-oncogene tyrosine-protein kinase Src(Human)
University of British Columbia
Curated by ChEMBL
University of British Columbia
Curated by ChEMBL
Affinity DataIC50: 1.56E+3nMAssay Description:Inhibition of SRC (unknown origin) by Z-LYTE Kinase assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 4.00E+3nMAssay Description:Inhibition of LDHA (unknown origin)More data for this Ligand-Target Pair
Ligand Info
TargetProto-oncogene tyrosine-protein kinase Src(Human)
University of British Columbia
Curated by ChEMBL
University of British Columbia
Curated by ChEMBL
Affinity DataIC50: 4.52E+3nMAssay Description:Inhibition of SRC (unknown origin) by Z-LYTE Kinase assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataKd: 5.30E+3nMAssay Description:Binding affinity to ABL1 (unknown origin) assessed as dissociation constantMore data for this Ligand-Target Pair
Ligand Info

3D Structure (crystal)





