Report error Found 4 Enz. Inhib. hit(s) with all data for entry = 50023812
Affinity DataIC50: 5.70nMAssay Description:Antagonist activity at human CCR6 expressed in CHO-K1 cells incubated for 4 hrsMore data for this Ligand-Target Pair
Ligand InfoPDB
Affinity DataIC50: 13nMAssay Description:Antagonist activity at CXCR2 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 16nMAssay Description:Antagonist activity at CXCR2 (unknown origin)More data for this Ligand-Target Pair
Affinity DataKd: 4.55E+3nMAssay Description:Competitive binding affinity to full length CCR5 (unknown origin) expressed in HEK293F cells assessed as dissociation constant incubated for 3 hrs by...More data for this Ligand-Target Pair
Ligand Info

3D Structure (crystal)

