Compile Data Set for Download or QSAR
Report error Found 5 Enz. Inhib. hit(s) with all data for entry = 50023318
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
University of Auckland

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 100152BDBM100152(cid_5359389 | SMR001233259 | HARMINE | 7-methoxy-1...)
Affinity DataIC50: 9nMAssay Description:Inhibition of DYRK1A (unknown origin) incubated for 2 hrs in presence of [gamma-33P]-ATP by radioactivity based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2026
Entry Details
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
University of Auckland

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50047009BDBM50047009(CHEMBL1535235 | 1-methyl-9H-pyrido[3,4-b]indol-7-o...)
Affinity DataIC50: 16nMAssay Description:Inhibition of DYRK1A (unknown origin) incubated for 2 hrs in presence of [gamma-33P]-ATP by radioactivity based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2026
Entry Details
PubMed
TargetAmine oxidase [flavin-containing] A(Human)
University of Auckland

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 100152BDBM100152(cid_5359389 | SMR001233259 | HARMINE | 7-methoxy-1...)
Affinity DataIC50: 60nMAssay Description:Inhibition of MAO-A (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2026
Entry Details
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
University of Auckland

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50047009BDBM50047009(CHEMBL1535235 | 1-methyl-9H-pyrido[3,4-b]indol-7-o...)
Affinity DataIC50: 70nMAssay Description:Inhibition of DYRK1A (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2026
Entry Details
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
University of Auckland

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 100152BDBM100152(cid_5359389 | SMR001233259 | HARMINE | 7-methoxy-1...)
Affinity DataIC50: 100nMAssay Description:Inhibition of DYRK1A (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2026
Entry Details
PubMed