Report error Found 28 Enz. Inhib. hit(s) with all data for entry = 50023138
TargetATP-dependent Clp protease proteolytic subunit, mitochondrial(Human)
University of Bari Aldo Moro
Curated by ChEMBL
University of Bari Aldo Moro
Curated by ChEMBL
Affinity DataEC50: 130nMAssay Description:Activation of recombinant human ClpP using Ac-WLA-AMC as substrate by plate reader analysisMore data for this Ligand-Target Pair
3D Structure (crystal)TargetATP-dependent Clp protease proteolytic subunit, mitochondrial(Human)
University of Bari Aldo Moro
Curated by ChEMBL
University of Bari Aldo Moro
Curated by ChEMBL
Affinity DataEC50: 140nMAssay Description:Activation of recombinant human ClpP using casein-FITC as substrate preincubated for 30 mins followed by substrate addition by fluorescence based ana...More data for this Ligand-Target Pair
TargetATP-dependent Clp protease proteolytic subunit, mitochondrial(Human)
University of Bari Aldo Moro
Curated by ChEMBL
University of Bari Aldo Moro
Curated by ChEMBL
Affinity DataEC50: 1.18E+3nMAssay Description:Activation of human ClpP using FITC-casein as substrate assessed as increase in proteolytic activity preincubated for 15 mins followed by substrate a...More data for this Ligand-Target Pair
TargetATP-dependent Clp protease proteolytic subunit, mitochondrial(Human)
University of Bari Aldo Moro
Curated by ChEMBL
University of Bari Aldo Moro
Curated by ChEMBL
Affinity DataEC50: 2.00E+3nMAssay Description:Activation of human ClpP using FITC-casein as substrate assessed as increase in proteolytic activity preincubated for 15 mins followed by substrate a...More data for this Ligand-Target Pair
TargetATP-dependent Clp protease proteolytic subunit, mitochondrial(Human)
University of Bari Aldo Moro
Curated by ChEMBL
University of Bari Aldo Moro
Curated by ChEMBL
Affinity DataEC50: 2.00E+3nMAssay Description:Activation of human ClpPMore data for this Ligand-Target Pair
TargetATP-dependent Clp protease proteolytic subunit, mitochondrial(Human)
University of Bari Aldo Moro
Curated by ChEMBL
University of Bari Aldo Moro
Curated by ChEMBL
Affinity DataEC50: 2.88E+3nMAssay Description:Activation of human ClpP using FITC-casein as substrate assessed as increase in proteolytic activity preincubated for 15 mins followed by substrate a...More data for this Ligand-Target Pair
TargetATP-dependent Clp protease proteolytic subunit, mitochondrial(Human)
University of Bari Aldo Moro
Curated by ChEMBL
University of Bari Aldo Moro
Curated by ChEMBL
Affinity DataEC50: 3.80E+3nMAssay Description:Activation of human ClpP using FITC-casein as substrate assessed as increase in proteolytic activity preincubated for 15 mins followed by substrate a...More data for this Ligand-Target Pair
TargetATP-dependent Clp protease proteolytic subunit, mitochondrial(Human)
University of Bari Aldo Moro
Curated by ChEMBL
University of Bari Aldo Moro
Curated by ChEMBL
Affinity DataEC50: 3.99E+3nMAssay Description:Activation of human ClpP using FITC-casein as substrate assessed as increase in proteolytic activity preincubated for 15 mins followed by substrate a...More data for this Ligand-Target Pair
Affinity DataKi: 4.09E+3nMAssay Description:Displacement of [3H]-N-methylspiperone from human D3 receptor extracted from HEK293 cell membrane assessed as inhibition constant incubated for 60 mi...More data for this Ligand-Target Pair
TargetATP-dependent Clp protease proteolytic subunit, mitochondrial(Human)
University of Bari Aldo Moro
Curated by ChEMBL
University of Bari Aldo Moro
Curated by ChEMBL
Affinity DataEC50: 4.20E+3nMAssay Description:Activation of human ClpP using FITC-casein as substrate assessed as increase in proteolytic activity preincubated for 15 mins followed by substrate a...More data for this Ligand-Target Pair
TargetATP-dependent Clp protease proteolytic subunit, mitochondrial(Human)
University of Bari Aldo Moro
Curated by ChEMBL
University of Bari Aldo Moro
Curated by ChEMBL
Affinity DataEC50: 4.70E+3nMAssay Description:Activation of human ClpP using FITC-casein as substrate assessed as increase in proteolytic activity preincubated for 15 mins followed by substrate a...More data for this Ligand-Target Pair
TargetATP-dependent Clp protease proteolytic subunit, mitochondrial(Human)
University of Bari Aldo Moro
Curated by ChEMBL
University of Bari Aldo Moro
Curated by ChEMBL
Affinity DataEC50: 5.90E+3nMAssay Description:Activation of human ClpP using FITC-casein as substrate assessed as increase in proteolytic activity preincubated for 15 mins followed by substrate a...More data for this Ligand-Target Pair
TargetATP-dependent Clp protease proteolytic subunit, mitochondrial(Human)
University of Bari Aldo Moro
Curated by ChEMBL
University of Bari Aldo Moro
Curated by ChEMBL
Affinity DataEC50: 7.70E+3nMAssay Description:Activation of human ClpP using FITC-casein as substrate assessed as increase in proteolytic activity preincubated for 15 mins followed by substrate a...More data for this Ligand-Target Pair
TargetATP-dependent Clp protease proteolytic subunit, mitochondrial(Human)
University of Bari Aldo Moro
Curated by ChEMBL
University of Bari Aldo Moro
Curated by ChEMBL
Affinity DataEC50: 9.00E+3nMAssay Description:Activation of human ClpP using FITC-casein as substrate assessed as increase in proteolytic activity preincubated for 15 mins followed by substrate a...More data for this Ligand-Target Pair
TargetATP-dependent Clp protease proteolytic subunit, mitochondrial(Human)
University of Bari Aldo Moro
Curated by ChEMBL
University of Bari Aldo Moro
Curated by ChEMBL
Affinity DataEC50: 1.00E+4nMAssay Description:Activation of human ClpP using FITC-casein as substrate assessed as increase in proteolytic activity preincubated for 15 mins followed by substrate a...More data for this Ligand-Target Pair
Affinity DataKi: 1.48E+4nMAssay Description:Displacement of [3H]-N-methylspiperone from human D2L receptor extracted from HEK293 cell membrane assessed as inhibition constant incubated for 60 m...More data for this Ligand-Target Pair
TargetATP-dependent Clp protease proteolytic subunit, mitochondrial(Human)
University of Bari Aldo Moro
Curated by ChEMBL
University of Bari Aldo Moro
Curated by ChEMBL
Affinity DataEC50: 1.60E+4nMAssay Description:Activation of human ClpP using FITC-casein as substrate assessed as increase in proteolytic activity preincubated for 15 mins followed by substrate a...More data for this Ligand-Target Pair
TargetATP-dependent Clp protease proteolytic subunit, mitochondrial(Human)
University of Bari Aldo Moro
Curated by ChEMBL
University of Bari Aldo Moro
Curated by ChEMBL
Affinity DataEC50: 2.20E+4nMAssay Description:Activation of human ClpP using FITC-casein as substrate assessed as increase in proteolytic activity preincubated for 15 mins followed by substrate a...More data for this Ligand-Target Pair
Affinity DataKi: 2.67E+4nMAssay Description:Displacement of [3H]-N-methylspiperone from human D3 receptor extracted from HEK293 cell membrane assessed as inhibition constant incubated for 60 mi...More data for this Ligand-Target Pair
Affinity DataKi: 3.14E+4nMAssay Description:Displacement of [3H]-N-methylspiperone from human D3 receptor extracted from HEK293 cell membrane assessed as inhibition constant incubated for 60 mi...More data for this Ligand-Target Pair
TargetATP-dependent Clp protease proteolytic subunit, mitochondrial(Human)
University of Bari Aldo Moro
Curated by ChEMBL
University of Bari Aldo Moro
Curated by ChEMBL
Affinity DataEC50: 3.47E+4nMAssay Description:Activation of human ClpP using FITC-casein as substrate assessed as increase in proteolytic activity preincubated for 15 mins followed by substrate a...More data for this Ligand-Target Pair
Affinity DataKi: 3.64E+4nMAssay Description:Displacement of [3H]-N-methylspiperone from human D3 receptor extracted from HEK293 cell membrane assessed as inhibition constant incubated for 60 mi...More data for this Ligand-Target Pair
Affinity DataKi: 5.11E+4nMAssay Description:Displacement of [3H]-N-methylspiperone from human D3 receptor extracted from HEK293 cell membrane assessed as inhibition constant incubated for 60 mi...More data for this Ligand-Target Pair
TargetATP-dependent Clp protease proteolytic subunit, mitochondrial(Human)
University of Bari Aldo Moro
Curated by ChEMBL
University of Bari Aldo Moro
Curated by ChEMBL
Affinity DataEC50: >1.00E+5nMAssay Description:Activation of human ClpP using FITC-casein as substrate assessed as increase in proteolytic activity preincubated for 15 mins followed by substrate a...More data for this Ligand-Target Pair
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]-N-methylspiperone from human D2L receptor extracted from HEK293 cell membrane assessed as inhibition constant incubated for 60 m...More data for this Ligand-Target Pair
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]-N-methylspiperone from human D2L receptor extracted from HEK293 cell membrane assessed as inhibition constant incubated for 60 m...More data for this Ligand-Target Pair
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]-N-methylspiperone from human D2L receptor extracted from HEK293 cell membrane assessed as inhibition constant incubated for 60 m...More data for this Ligand-Target Pair
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]-N-methylspiperone from human D2L receptor extracted from HEK293 cell membrane assessed as inhibition constant incubated for 60 m...More data for this Ligand-Target Pair
