Report error Found 32 Enz. Inhib. hit(s) with all data for entry = 50023289
Affinity DataIC50: 2.32E+3nMAssay Description:Inhibition of ALKBH5 (unknown origin) using 5'-ATTGTCA(m6A)CAGCAGA-FAM-3' as substrate measured after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 5.34E+3nMAssay Description:Inhibition of ALKBH5 (unknown origin) using 5'-ATTGTCA(m6A)CAGCAGA-FAM-3' as substrate measured after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 9.57E+3nMAssay Description:Inhibition of ALKBH5 (unknown origin) using 5'-ATTGTCA(m6A)CAGCAGA-FAM-3' as substrate measured after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 1.12E+4nMAssay Description:Inhibition of ALKBH5 (unknown origin) using 5'-TAGACATTGCCATTCTCGATAGG (m6A) TCCGGTCAAACCTAGAC GAATTCCA-3' as substrate measured after 2 hrs in prese...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 1.65E+4nMAssay Description:Inhibition of ALKBH5 (unknown origin) using 5'-ATTGTCA(m6A)CAGCAGA-FAM-3' as substrate measured after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 1.69E+4nMAssay Description:Inhibition of ALKBH5 (unknown origin) using 5'-ATTGTCA(m6A)CAGCAGA-FAM-3' as substrate measured after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 1.74E+4nMAssay Description:Inhibition of ALKBH5 (unknown origin) using 5'-ATTGTCA(m6A)CAGCAGA-FAM-3' as substrate measured after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 1.87E+4nMAssay Description:Inhibition of ALKBH5 (unknown origin) using 5'-ATTGTCA(m6A)CAGCAGA-FAM-3' as substrate measured after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 2.06E+4nMAssay Description:Inhibition of ALKBH5 (unknown origin) using 5'-ATTGTCA(m6A)CAGCAGA-FAM-3' as substrate measured after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 2.13E+4nMAssay Description:Inhibition of ALKBH5 (unknown origin) using 5'-ATTGTCA(m6A)CAGCAGA-FAM-3' as substrate measured after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 2.59E+4nMAssay Description:Inhibition of ALKBH5 (unknown origin) using 5'-TAGACATTGCCATTCTCGATAGG (m6A) TCCGGTCAAACCTAGAC GAATTCCA-3' as substrate measured after 2 hrs in prese...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 2.96E+4nMAssay Description:Inhibition of ALKBH5 (unknown origin) using 5'-ATTGTCA(m6A)CAGCAGA-FAM-3' as substrate measured after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 3.29E+4nMAssay Description:Inhibition of ALKBH5 (unknown origin) using 5'-ATTGTCA(m6A)CAGCAGA-FAM-3' as substrate measured after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 3.41E+4nMAssay Description:Inhibition of ALKBH5 (unknown origin) using 5'-ATTGTCA(m6A)CAGCAGA-FAM-3' as substrate measured after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 3.70E+4nMAssay Description:Inhibition of ALKBH5 (unknown origin) using 5'-ATTGTCA(m6A)CAGCAGA-FAM-3' as substrate measured after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 4.55E+4nMAssay Description:Inhibition of ALKBH5 (unknown origin) using 5'-ATTGTCA(m6A)CAGCAGA-FAM-3' as substrate measured after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 4.78E+4nMAssay Description:Inhibition of ALKBH5 (unknown origin) using 5'-ATTGTCA(m6A)CAGCAGA-FAM-3' as substrate measured after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 6.91E+4nMAssay Description:Inhibition of ALKBH5 (unknown origin) using 5'-ATTGTCA(m6A)CAGCAGA-FAM-3' as substrate measured after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of ALKBH5 (unknown origin) using 5'-TAGACATTGCCATTCTCGATAGG (m6A) TCCGGTCAAACCTAGAC GAATTCCA-3' as substrate measured after 2 hrs in prese...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 2.00E+5nMAssay Description:Inhibition of ALKBH5 (unknown origin) using 5'-ATTGTCA(m6A)CAGCAGA-FAM-3' as substrate measured after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 2.00E+5nMAssay Description:Inhibition of ALKBH5 (unknown origin) using 5'-ATTGTCA(m6A)CAGCAGA-FAM-3' as substrate measured after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 2.00E+5nMAssay Description:Inhibition of ALKBH5 (unknown origin) using 5'-ATTGTCA(m6A)CAGCAGA-FAM-3' as substrate measured after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 2.00E+5nMAssay Description:Inhibition of ALKBH5 (unknown origin) using 5'-ATTGTCA(m6A)CAGCAGA-FAM-3' as substrate measured after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 2.00E+5nMAssay Description:Inhibition of ALKBH5 (unknown origin) using 5'-ATTGTCA(m6A)CAGCAGA-FAM-3' as substrate measured after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 2.00E+5nMAssay Description:Inhibition of ALKBH5 (unknown origin) using 5'-ATTGTCA(m6A)CAGCAGA-FAM-3' as substrate measured after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 2.00E+5nMAssay Description:Inhibition of ALKBH5 (unknown origin) using 5'-ATTGTCA(m6A)CAGCAGA-FAM-3' as substrate measured after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 2.00E+5nMAssay Description:Inhibition of ALKBH5 (unknown origin) using 5'-ATTGTCA(m6A)CAGCAGA-FAM-3' as substrate measured after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 2.00E+5nMAssay Description:Inhibition of ALKBH5 (unknown origin) using 5'-ATTGTCA(m6A)CAGCAGA-FAM-3' as substrate measured after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 2.00E+5nMAssay Description:Inhibition of ALKBH5 (unknown origin) using 5'-ATTGTCA(m6A)CAGCAGA-FAM-3' as substrate measured after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 2.00E+5nMAssay Description:Inhibition of ALKBH5 (unknown origin) using 5'-ATTGTCA(m6A)CAGCAGA-FAM-3' as substrate measured after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 2.00E+5nMAssay Description:Inhibition of ALKBH5 (unknown origin) using 5'-ATTGTCA(m6A)CAGCAGA-FAM-3' as substrate measured after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand Info
TargetAlpha-ketoglutarate-dependent dioxygenase FTO(Human)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 2.50E+5nMAssay Description:Inhibition of FTO (unknown origin) using 5'-TAGACATTGCCATTCTCGATAGG (m6A) TCCGGTCAAACCTAGAC GAATTCCA-3' as substrate measured after 2 hrs in presence...More data for this Ligand-Target Pair
Ligand Info



























