Report error Found 34 Enz. Inhib. hit(s) with all data for entry = 50023667
Affinity DataKd: 3.70nMAssay Description:Binding affinity to Androgen receptor LBD (unknown origin) assessed as dissociation constant by biolayer interferometry assayMore data for this Ligand-Target Pair
Affinity DataKd: 4nMAssay Description:Binding affinity to Androgen receptor LBD (unknown origin) assessed as dissociation constant by biolayer interferometry assayMore data for this Ligand-Target Pair
Affinity DataIC50: 40nMAssay Description:Antagonist activity at Androgen receptor in human LNCaP cells expressing ARR2PB-eGFP incubated for 3 days by fluorescence based assayMore data for this Ligand-Target Pair
Affinity DataIC50: 40nMAssay Description:Antagonist activity at Androgen receptor in human LNCaP cells expressing ARR2PB-eGFP incubated for 3 days by fluorescence based assayMore data for this Ligand-Target Pair
Affinity DataIC50: 40nMAssay Description:Antagonist activity at Androgen receptor in human LNCaP cells expressing ARR2PB-eGFP incubated for 3 days by fluorescence based assayMore data for this Ligand-Target Pair
Affinity DataIC50: 50nMAssay Description:Antagonist activity at Androgen receptor in human LNCaP cells expressing ARR2PB-eGFP incubated for 3 days by fluorescence based assayMore data for this Ligand-Target Pair
Affinity DataIC50: 70nMAssay Description:Antagonist activity at Androgen receptor in human LNCaP cells expressing ARR2PB-eGFP incubated for 3 days by fluorescence based assayMore data for this Ligand-Target Pair
Affinity DataIC50: 90nMAssay Description:Antagonist activity at Androgen receptor in human LNCaP cells expressing ARR2PB-eGFP incubated for 3 days by fluorescence based assayMore data for this Ligand-Target Pair
Affinity DataIC50: 140nMAssay Description:Antagonist activity at Androgen receptor in human LNCaP cells expressing ARR2PB-eGFP incubated for 3 days by fluorescence based assayMore data for this Ligand-Target Pair
Affinity DataIC50: 140nMAssay Description:Antagonist activity at Androgen receptor in human LNCaP cells expressing ARR2PB-eGFP incubated for 3 days by fluorescence based assayMore data for this Ligand-Target Pair
Affinity DataIC50: 170nMAssay Description:Antagonist activity at Androgen receptor in human LNCaP cells expressing ARR2PB-eGFP incubated for 3 days by fluorescence based assayMore data for this Ligand-Target Pair
Affinity DataIC50: 170nMAssay Description:Antagonist activity at Androgen receptor in human LNCaP cells expressing ARR2PB-eGFP incubated for 3 days by fluorescence based assayMore data for this Ligand-Target Pair
Affinity DataIC50: 270nMAssay Description:Antagonist activity at Androgen receptor in human LNCaP cells expressing ARR2PB-eGFP incubated for 3 days by fluorescence based assayMore data for this Ligand-Target Pair
Affinity DataIC50: 320nMAssay Description:Antagonist activity at Androgen receptor in human LNCaP cells expressing ARR2PB-eGFP assessed as inhibition of secreted PSA level by Western blot ana...More data for this Ligand-Target Pair
Affinity DataIC50: 340nMAssay Description:Antagonist activity at Androgen receptor in human LNCaP cells expressing ARR2PB-eGFP incubated for 3 days by fluorescence based assayMore data for this Ligand-Target Pair
Affinity DataIC50: 360nMAssay Description:Antagonist activity at wild type Androgen receptor in human PC-3 cells expressing ARR2PB-eGFP incubated for 3 days by fluorescence based assayMore data for this Ligand-Target Pair
Affinity DataIC50: 370nMAssay Description:Antagonist activity at Androgen receptor in human LNCaP cells expressing ARR2PB-eGFP assessed as inhibition of secreted PSA level by Western blot ana...More data for this Ligand-Target Pair
Affinity DataIC50: 370nMAssay Description:Antagonist activity at Androgen receptor in human LNCaP cells expressing ARR2PB-eGFP incubated for 3 days by fluorescence based assayMore data for this Ligand-Target Pair
Affinity DataIC50: 470nMAssay Description:Antagonist activity at DHT-induced Androgen receptor W741C mutant in human PC-3 cells transfected with ARR2PB-Luc by dual-luciferase reporter assayMore data for this Ligand-Target Pair
Affinity DataIC50: 520nMAssay Description:Antagonist activity at Androgen receptor in human LNCaP cells expressing ARR2PB-eGFP incubated for 3 days by fluorescence based assayMore data for this Ligand-Target Pair
Affinity DataIC50: 580nMAssay Description:Antagonist activity at wild type Androgen receptor in human PC-3 cells expressing ARR2PB-eGFP incubated for 3 days by fluorescence based assayMore data for this Ligand-Target Pair
Affinity DataIC50: 620nMAssay Description:Antagonist activity at DHT-induced Androgen receptor W741C mutant in human PC-3 cells transfected with ARR2PB-Luc by dual-luciferase reporter assayMore data for this Ligand-Target Pair
Affinity DataIC50: 660nMAssay Description:Antagonist activity at DHT-induced Androgen receptor F876L/Y877A mutant in human PC-3 cells transfected with ARR2PB-Luc by dual-luciferase reporter a...More data for this Ligand-Target Pair
Affinity DataIC50: 680nMAssay Description:Antagonist activity at Androgen receptor in human LNCaP cells expressing ARR2PB-eGFP incubated for 3 days by fluorescence based assayMore data for this Ligand-Target Pair
Affinity DataIC50: 880nMAssay Description:Antagonist activity at DHT-induced Androgen receptor F876L/Y877A mutant in human PC-3 cells transfected with ARR2PB-Luc by dual-luciferase reporter a...More data for this Ligand-Target Pair
Affinity DataIC50: 910nMAssay Description:Antagonist activity at Androgen receptor in human LNCaP cells expressing ARR2PB-eGFP incubated for 3 days by fluorescence based assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.58E+3nMAssay Description:Antagonist activity at Androgen receptor in human LNCaP cells expressing ARR2PB-eGFP incubated for 3 days by fluorescence based assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.65E+3nMAssay Description:Antagonist activity at Androgen receptor in human LNCaP cells expressing ARR2PB-eGFP incubated for 3 days by fluorescence based assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.97E+3nMAssay Description:Antagonist activity at DHT-induced Androgen receptor W741C mutant in human PC-3 cells transfected with ARR2PB-Luc by dual-luciferase reporter assayMore data for this Ligand-Target Pair
Affinity DataIC50: 4.46E+3nMAssay Description:Antagonist activity at Androgen receptor (unknown origin) by PolarScreen competitive assayMore data for this Ligand-Target Pair
Affinity DataIC50: 6.70E+3nMAssay Description:Antagonist activity at Androgen receptor in human LNCaP cells expressing ARR2PB-eGFP incubated for 3 days by fluorescence based assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.60E+4nMAssay Description:Antagonist activity at Androgen receptor in human LNCaP cells expressing ARR2PB-eGFP incubated for 3 days by fluorescence based assayMore data for this Ligand-Target Pair
Affinity DataIC50: 3.06E+4nMAssay Description:Antagonist activity at Androgen receptor in human LNCaP cells expressing ARR2PB-eGFP incubated for 3 days by fluorescence based assayMore data for this Ligand-Target Pair
Affinity DataIC50: 6.75E+4nMAssay Description:Antagonist activity at Androgen receptor (unknown origin) by PolarScreen competitive assayMore data for this Ligand-Target Pair
