Report error Found 73 Enz. Inhib. hit(s) with all data for entry = 50023420
Affinity DataEC50: 1nMAssay Description:Agonist activity at recombinant rat GluN1/GluN2C NMDA receptor expressed in xenopus laevis oocytes in presence of glutamate by two-electrode voltage-...More data for this Ligand-Target Pair
Ligand Info
Affinity DataEC50: 3nMAssay Description:Agonist activity at recombinant rat GluN1/GluN2C NMDA receptor expressed in xenopus laevis oocytes in presence of L-glutamate by two-electrode voltag...More data for this Ligand-Target Pair
Ligand Info
Affinity DataEC50: 14nMAssay Description:Agonist activity at recombinant rat GluN1/GluN2B NMDA receptor expressed in xenopus laevis oocytes in presence of glutamate by two-electrode voltage-...More data for this Ligand-Target Pair
Ligand Info
Affinity DataEC50: 16nMAssay Description:Partial agonist activity at recombinant rat GluN1/GluN2D NMDA receptor expressed in xenopus laevis oocytes in presence of L-glutamate by two-electrod...More data for this Ligand-Target Pair
Ligand Info
Affinity DataEC50: 18nMAssay Description:Partial agonist activity at recombinant rat GluN1/GluN2A NMDA receptor expressed in xenopus laevis oocytes in presence of L-glutamate by two-electrod...More data for this Ligand-Target Pair
Ligand Info
Affinity DataEC50: 25nMAssay Description:Agonist activity at recombinant rat GluN1/GluN2C NMDA receptor expressed in xenopus laevis oocytes in presence of L-glutamate by two-electrode voltag...More data for this Ligand-Target Pair
Ligand Info
Affinity DataEC50: 31nMAssay Description:Agonist activity at recombinant rat GluN1/GluN2D NMDA receptor expressed in xenopus laevis oocytes in presence of glutamate by two-electrode voltage-...More data for this Ligand-Target Pair
Ligand Info
Affinity DataEC50: 34nMAssay Description:Agonist activity at recombinant rat GluN1/GluN2C NMDA receptor expressed in xenopus laevis oocytes in presence of L-glutamate by two-electrode voltag...More data for this Ligand-Target Pair
Ligand Info
Affinity DataEC50: 36nMAssay Description:Agonist activity at recombinant rat GluN1/GluN2A NMDA receptor expressed in xenopus laevis oocytes in presence of glutamate by two-electrode voltage-...More data for this Ligand-Target Pair
Ligand Info
Affinity DataEC50: 38nMAssay Description:Agonist activity at recombinant rat GluN1/GluN2C NMDA receptor expressed in xenopus laevis oocytes in presence of L-glutamate by two-electrode voltag...More data for this Ligand-Target Pair
Ligand Info
Affinity DataEC50: 41nMAssay Description:Agonist activity at recombinant rat GluN1/GluN2C NMDA receptor expressed in xenopus laevis oocytes in presence of L-glutamate by two-electrode voltag...More data for this Ligand-Target Pair
Ligand Info
Affinity DataEC50: 51nMAssay Description:Partial agonist activity at recombinant rat GluN1/GluN2A NMDA receptor expressed in xenopus laevis oocytes in presence of L-glutamate by two-electrod...More data for this Ligand-Target Pair
Ligand Info
Affinity DataEC50: 57nMAssay Description:Partial agonist activity at recombinant rat GluN1/GluN2A NMDA receptor expressed in xenopus laevis oocytes in presence of L-glutamate by two-electrod...More data for this Ligand-Target Pair
Ligand Info
Affinity DataEC50: 72nMAssay Description:Partial agonist activity at recombinant rat GluN1/GluN2D NMDA receptor expressed in xenopus laevis oocytes in presence of L-glutamate by two-electrod...More data for this Ligand-Target Pair
Ligand Info
Affinity DataEC50: 74nMAssay Description:Partial agonist activity at recombinant rat GluN1/GluN2A NMDA receptor expressed in xenopus laevis oocytes in presence of L-glutamate by two-electrod...More data for this Ligand-Target Pair
Ligand Info
Affinity DataEC50: 81nMAssay Description:Partial agonist activity at recombinant rat GluN1/GluN2D NMDA receptor expressed in xenopus laevis oocytes in presence of L-glutamate by two-electrod...More data for this Ligand-Target Pair
Ligand Info
Affinity DataEC50: 88nMAssay Description:Agonist activity at recombinant rat GluN1/GluN2C NMDA receptor expressed in xenopus laevis oocytes in presence of L-glutamate by two-electrode voltag...More data for this Ligand-Target Pair
Ligand Info
Affinity DataEC50: 102nMAssay Description:Partial agonist activity at recombinant rat GluN1/GluN2A NMDA receptor expressed in xenopus laevis oocytes in presence of L-glutamate by two-electrod...More data for this Ligand-Target Pair
Ligand Info
Affinity DataEC50: 110nMAssay Description:Agonist activity at recombinant rat GluN1/GluN2C NMDA receptor expressed in xenopus laevis oocytes in presence of L-glutamate by two-electrode voltag...More data for this Ligand-Target Pair
Ligand Info
Affinity DataEC50: 120nMAssay Description:Partial agonist activity at recombinant rat GluN1/GluN2D NMDA receptor expressed in xenopus laevis oocytes in presence of L-glutamate by two-electrod...More data for this Ligand-Target Pair
Ligand Info
Affinity DataEC50: 130nMAssay Description:Partial agonist activity at recombinant rat GluN1/GluN2D NMDA receptor expressed in xenopus laevis oocytes in presence of L-glutamate by two-electrod...More data for this Ligand-Target Pair
Affinity DataEC50: 133nMAssay Description:Agonist activity at recombinant rat GluN1/GluN2C NMDA receptor expressed in xenopus laevis oocytes in presence of L-glutamate by two-electrode voltag...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 150nMAssay Description:Inhibition of recombinant rat GluN1/GluN2B NMDA receptor expressed in xenopus laevis oocytes in presence of glycine and L-glutamate by two-electrode ...More data for this Ligand-Target Pair
Affinity DataEC50: 150nMAssay Description:Partial agonist activity at recombinant rat GluN1/GluN2A NMDA receptor expressed in xenopus laevis oocytes in presence of L-glutamate by two-electrod...More data for this Ligand-Target Pair
Ligand Info
Affinity DataEC50: 170nMAssay Description:Partial agonist activity at recombinant rat GluN1/GluN2D NMDA receptor expressed in xenopus laevis oocytes in presence of L-glutamate by two-electrod...More data for this Ligand-Target Pair
Affinity DataEC50: 180nMAssay Description:Partial agonist activity at recombinant rat GluN1/GluN2D NMDA receptor expressed in xenopus laevis oocytes in presence of L-glutamate by two-electrod...More data for this Ligand-Target Pair
Ligand Info
Affinity DataEC50: 200nMAssay Description:Partial agonist activity at recombinant rat GluN1/GluN2D NMDA receptor expressed in xenopus laevis oocytes in presence of L-glutamate by two-electrod...More data for this Ligand-Target Pair
Ligand Info
Affinity DataEC50: 210nMAssay Description:Agonist activity at recombinant rat GluN1/GluN2C NMDA receptor expressed in xenopus laevis oocytes in presence of L-glutamate by two-electrode voltag...More data for this Ligand-Target Pair
Affinity DataEC50: 210nMAssay Description:Partial agonist activity at recombinant rat GluN1/GluN2A NMDA receptor expressed in xenopus laevis oocytes in presence of L-glutamate by two-electrod...More data for this Ligand-Target Pair
Ligand Info
Affinity DataEC50: 230nMAssay Description:Agonist activity at recombinant rat GluN1/GluN2C NMDA receptor expressed in xenopus laevis oocytes in presence of L-glutamate by two-electrode voltag...More data for this Ligand-Target Pair
Ligand Info
Affinity DataEC50: 240nMAssay Description:Partial agonist activity at recombinant rat GluN1/GluN2D NMDA receptor expressed in xenopus laevis oocytes in presence of L-glutamate by two-electrod...More data for this Ligand-Target Pair
Ligand Info
Affinity DataEC50: 290nMAssay Description:Partial agonist activity at recombinant rat GluN1/GluN2A NMDA receptor expressed in xenopus laevis oocytes in presence of L-glutamate by two-electrod...More data for this Ligand-Target Pair
Ligand Info
Affinity DataEC50: 300nMAssay Description:Agonist activity at recombinant rat GluN1/GluN2C NMDA receptor expressed in xenopus laevis oocytes in presence of L-glutamate by two-electrode voltag...More data for this Ligand-Target Pair
Affinity DataEC50: 300nMAssay Description:Agonist activity at GluN1/GluN2D (unknown origin) expressed in xenopus laevis oocytes by two-electrode voltage-clamp methodMore data for this Ligand-Target Pair
Ligand Info
Affinity DataEC50: 303nMAssay Description:Partial agonist activity at recombinant rat GluN1/GluN2D NMDA receptor expressed in xenopus laevis oocytes in presence of L-glutamate by two-electrod...More data for this Ligand-Target Pair
Ligand Info
Affinity DataEC50: 320nMAssay Description:Agonist activity at GluN1/GluN2C (unknown origin) expressed in xenopus laevis oocytes by two-electrode voltage-clamp methodMore data for this Ligand-Target Pair
Ligand Info
Affinity DataEC50: 360nMAssay Description:Agonist activity at recombinant rat GluN1/GluN2B NMDA receptor expressed in xenopus laevis oocytes in presence of L-glutamate by two-electrode voltag...More data for this Ligand-Target Pair
Affinity DataEC50: 400nMAssay Description:Agonist activity at GluN1/GluN2B (unknown origin) expressed in xenopus laevis oocytes by two-electrode voltage-clamp methodMore data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 540nMAssay Description:Inhibition of recombinant rat GluN1/GluN2A NMDA receptor expressed in xenopus laevis oocytes in presence of glycine and L-glutamate by two-electrode ...More data for this Ligand-Target Pair
Affinity DataEC50: 640nMAssay Description:Agonist activity at recombinant rat GluN1/GluN2C NMDA receptor expressed in xenopus laevis oocytes in presence of L-glutamate by two-electrode voltag...More data for this Ligand-Target Pair
Ligand Info
Affinity DataEC50: 660nMAssay Description:Agonist activity at recombinant rat GluN1/GluN2C NMDA receptor expressed in xenopus laevis oocytes in presence of L-glutamate by two-electrode voltag...More data for this Ligand-Target Pair
Ligand Info
Affinity DataEC50: 670nMAssay Description:Agonist activity at recombinant rat GluN1/GluN2B NMDA receptor expressed in xenopus laevis oocytes in presence of L-glutamate by two-electrode voltag...More data for this Ligand-Target Pair
Affinity DataEC50: 740nMAssay Description:Agonist activity at recombinant rat GluN1/GluN2C NMDA receptor expressed in xenopus laevis oocytes in presence of L-glutamate by two-electrode voltag...More data for this Ligand-Target Pair
Ligand Info
Affinity DataEC50: 880nMAssay Description:Partial agonist activity at recombinant rat GluN1/GluN2A NMDA receptor expressed in xenopus laevis oocytes in presence of L-glutamate by two-electrod...More data for this Ligand-Target Pair
Ligand Info
Affinity DataEC50: 930nMAssay Description:Agonist activity at recombinant rat GluN1/GluN2C NMDA receptor expressed in xenopus laevis oocytes in presence of L-glutamate by two-electrode voltag...More data for this Ligand-Target Pair
Ligand Info
Affinity DataEC50: 980nMAssay Description:Partial agonist activity at recombinant rat GluN1/GluN2D NMDA receptor expressed in xenopus laevis oocytes in presence of L-glutamate by two-electrod...More data for this Ligand-Target Pair
Ligand Info
Affinity DataEC50: 1.00E+3nMAssay Description:Partial agonist activity at recombinant rat GluN1/GluN2A NMDA receptor expressed in xenopus laevis oocytes in presence of L-glutamate by two-electrod...More data for this Ligand-Target Pair
Affinity DataEC50: 1.07E+3nMAssay Description:Partial agonist activity at recombinant rat GluN1/GluN2A NMDA receptor expressed in xenopus laevis oocytes in presence of L-glutamate by two-electrod...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of recombinant rat GluN1/GluN2C NMDA receptor expressed in xenopus laevis oocytes in presence of glycine and L-glutamate by two-electrode ...More data for this Ligand-Target Pair
Affinity DataEC50: 1.13E+3nMAssay Description:Partial agonist activity at recombinant rat GluN1/GluN2A NMDA receptor expressed in xenopus laevis oocytes in presence of L-glutamate by two-electrod...More data for this Ligand-Target Pair










3D Structure (crystal)






