Report error Found 73 Enz. Inhib. hit(s) with all data for entry = 50023078
Affinity DataIC50: 4nMAssay Description:Inhibition of AURKA (unknown origin) using caliper substrate CTD3 by mobility shift assayMore data for this Ligand-Target Pair
Affinity DataIC50: 4.20nMAssay Description:Inhibition of CDK9 (unknown origin) using caliper substrate CTD3 by mobility shift assayMore data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Human)
University of Chinese Academy of Sciences
Curated by ChEMBL
University of Chinese Academy of Sciences
Curated by ChEMBL
Affinity DataIC50: 9.40nMAssay Description:Inhibition of BRD4 BD1 (unknown origin) incubated for 2 to 4 hrs under dark condition by FP assayMore data for this Ligand-Target Pair
Ligand Info
TargetBromodomain-containing protein 4(Human)
University of Chinese Academy of Sciences
Curated by ChEMBL
University of Chinese Academy of Sciences
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Inhibition of BRD4 BD1 (unknown origin) incubated for 2 to 4 hrs under dark condition by FP assayMore data for this Ligand-Target Pair
Ligand Info
TargetBromodomain-containing protein 4(Human)
University of Chinese Academy of Sciences
Curated by ChEMBL
University of Chinese Academy of Sciences
Curated by ChEMBL
Affinity DataIC50: 11nMAssay Description:Inhibition of BRD4 BD1 (unknown origin) incubated for 2 to 4 hrs under dark condition by FP assayMore data for this Ligand-Target Pair
Ligand Info
TargetBromodomain-containing protein 4(Human)
University of Chinese Academy of Sciences
Curated by ChEMBL
University of Chinese Academy of Sciences
Curated by ChEMBL
Affinity DataIC50: 11nMAssay Description:Inhibition of BRD4 BD1 (unknown origin) incubated for 2 to 4 hrs under dark condition by FP assayMore data for this Ligand-Target Pair
Ligand Info
TargetBromodomain-containing protein 4(Human)
University of Chinese Academy of Sciences
Curated by ChEMBL
University of Chinese Academy of Sciences
Curated by ChEMBL
Affinity DataIC50: 12nMAssay Description:Inhibition of BRD4 BD1 (unknown origin) incubated for 2 to 4 hrs under dark condition by FP assayMore data for this Ligand-Target Pair
Ligand Info
TargetBromodomain-containing protein 4(Human)
University of Chinese Academy of Sciences
Curated by ChEMBL
University of Chinese Academy of Sciences
Curated by ChEMBL
Affinity DataIC50: 14nMAssay Description:Inhibition of BRD4 BD1 (unknown origin) incubated for 2 to 4 hrs under dark condition by FP assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 15nMAssay Description:Inhibition of AURKA (unknown origin) using caliper substrate CTD3 by mobility shift assayMore data for this Ligand-Target Pair
Ligand Info
TargetBromodomain-containing protein 4(Human)
University of Chinese Academy of Sciences
Curated by ChEMBL
University of Chinese Academy of Sciences
Curated by ChEMBL
Affinity DataIC50: 16nMAssay Description:Inhibition of BRD4 BD1 (unknown origin) incubated for 2 to 4 hrs under dark condition by FP assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 16nMAssay Description:Inhibition of AURKA (unknown origin) using caliper substrate CTD3 by mobility shift assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 16nMAssay Description:Inhibition of AURKA (unknown origin) using caliper substrate CTD3 by mobility shift assayMore data for this Ligand-Target Pair
Ligand Info
TargetBromodomain-containing protein 4(Human)
University of Chinese Academy of Sciences
Curated by ChEMBL
University of Chinese Academy of Sciences
Curated by ChEMBL
Affinity DataIC50: 17nMAssay Description:Inhibition of BRD4 BD1 (unknown origin) incubated for 2 to 4 hrs under dark condition by FP assayMore data for this Ligand-Target Pair
Ligand Info
TargetBromodomain-containing protein 4(Human)
University of Chinese Academy of Sciences
Curated by ChEMBL
University of Chinese Academy of Sciences
Curated by ChEMBL
Affinity DataIC50: 20nMAssay Description:Inhibition of BRD4 BD1 (unknown origin) incubated for 2 to 4 hrs under dark condition by FP assayMore data for this Ligand-Target Pair
Ligand Info
TargetBromodomain-containing protein 4(Human)
University of Chinese Academy of Sciences
Curated by ChEMBL
University of Chinese Academy of Sciences
Curated by ChEMBL
Affinity DataIC50: 21nMAssay Description:Inhibition of BRD4 BD1 (unknown origin) incubated for 2 to 4 hrs under dark condition by FP assayMore data for this Ligand-Target Pair
Ligand Info
TargetBromodomain-containing protein 4(Human)
University of Chinese Academy of Sciences
Curated by ChEMBL
University of Chinese Academy of Sciences
Curated by ChEMBL
Affinity DataIC50: 26nMAssay Description:Inhibition of BRD4 BD1 (unknown origin) incubated for 2 to 4 hrs under dark condition by FP assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 28nMAssay Description:Inhibition of AURKA (unknown origin) using caliper substrate CTD3 by mobility shift assayMore data for this Ligand-Target Pair
Ligand Info
TargetBromodomain-containing protein 4(Human)
University of Chinese Academy of Sciences
Curated by ChEMBL
University of Chinese Academy of Sciences
Curated by ChEMBL
Affinity DataIC50: 29nMAssay Description:Inhibition of BRD4 BD1 (unknown origin) incubated for 2 to 4 hrs under dark condition by FP assayMore data for this Ligand-Target Pair
Ligand Info
TargetBromodomain-containing protein 4(Human)
University of Chinese Academy of Sciences
Curated by ChEMBL
University of Chinese Academy of Sciences
Curated by ChEMBL
Affinity DataIC50: 31nMAssay Description:Inhibition of BRD4 BD1 (unknown origin) incubated for 2 to 4 hrs under dark condition by FP assayMore data for this Ligand-Target Pair
Ligand Info
TargetBromodomain-containing protein 2(Human)
University of Chinese Academy of Sciences
Curated by ChEMBL
University of Chinese Academy of Sciences
Curated by ChEMBL
Affinity DataIC50: 35nMAssay Description:Inhibition of BRD2 BD1 (unknown origin) incubated for 2 to 4 hrs under dark condition by FP assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 35nMAssay Description:Inhibition of AURKA (unknown origin) using caliper substrate CTD3 by mobility shift assayMore data for this Ligand-Target Pair
Ligand Info
TargetBromodomain-containing protein 4(Human)
University of Chinese Academy of Sciences
Curated by ChEMBL
University of Chinese Academy of Sciences
Curated by ChEMBL
Affinity DataIC50: 36nMAssay Description:Inhibition of BRD4 BD1 (unknown origin) incubated for 2 to 4 hrs under dark condition by FP assayMore data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Human)
University of Chinese Academy of Sciences
Curated by ChEMBL
University of Chinese Academy of Sciences
Curated by ChEMBL
Affinity DataIC50: 39nMAssay Description:Inhibition of BRD4 BD1 (unknown origin) incubated for 2 to 4 hrs under dark condition by FP assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 39nMAssay Description:Inhibition of AURKA (unknown origin) using caliper substrate CTD3 by mobility shift assayMore data for this Ligand-Target Pair
Ligand Info
TargetBromodomain-containing protein 4(Human)
University of Chinese Academy of Sciences
Curated by ChEMBL
University of Chinese Academy of Sciences
Curated by ChEMBL
Affinity DataIC50: 41nMAssay Description:Inhibition of BRD4 BD1 (unknown origin) incubated for 2 to 4 hrs under dark condition by FP assayMore data for this Ligand-Target Pair
Ligand Info
TargetBromodomain-containing protein 4(Human)
University of Chinese Academy of Sciences
Curated by ChEMBL
University of Chinese Academy of Sciences
Curated by ChEMBL
Affinity DataIC50: 42nMAssay Description:Inhibition of BRD4 BD1 (unknown origin) incubated for 2 to 4 hrs under dark condition by FP assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 44nMAssay Description:Inhibition of AURKA (unknown origin) using caliper substrate CTD3 by mobility shift assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 45nMAssay Description:Inhibition of AURKA (unknown origin) using caliper substrate CTD3 by mobility shift assayMore data for this Ligand-Target Pair
Ligand Info
TargetBromodomain-containing protein 4(Human)
University of Chinese Academy of Sciences
Curated by ChEMBL
University of Chinese Academy of Sciences
Curated by ChEMBL
Affinity DataIC50: 45nMAssay Description:Inhibition of BRD4 BD1 (unknown origin) incubated for 2 to 4 hrs under dark condition by FP assayMore data for this Ligand-Target Pair
Ligand Info
TargetBromodomain-containing protein 4(Human)
University of Chinese Academy of Sciences
Curated by ChEMBL
University of Chinese Academy of Sciences
Curated by ChEMBL
Affinity DataIC50: 46nMAssay Description:Inhibition of BRD4 BD1 (unknown origin) incubated for 2 to 4 hrs under dark condition by FP assayMore data for this Ligand-Target Pair
Ligand Info
TargetBromodomain-containing protein 4(Human)
University of Chinese Academy of Sciences
Curated by ChEMBL
University of Chinese Academy of Sciences
Curated by ChEMBL
Affinity DataIC50: 47nMAssay Description:Inhibition of BRD4 BD1 (unknown origin) incubated for 2 to 4 hrs under dark condition by FP assayMore data for this Ligand-Target Pair
Ligand Info
TargetBromodomain-containing protein 2(Human)
University of Chinese Academy of Sciences
Curated by ChEMBL
University of Chinese Academy of Sciences
Curated by ChEMBL
Affinity DataIC50: 48nMAssay Description:Inhibition of BRD2 BD2 (unknown origin) incubated for 2 to 4 hrs under dark condition by FP assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 48nMAssay Description:Inhibition of AURKA (unknown origin) using caliper substrate CTD3 by mobility shift assayMore data for this Ligand-Target Pair
Ligand Info
TargetBromodomain-containing protein 4(Human)
University of Chinese Academy of Sciences
Curated by ChEMBL
University of Chinese Academy of Sciences
Curated by ChEMBL
Affinity DataIC50: 51nMAssay Description:Inhibition of BRD4 BD1 (unknown origin) incubated for 2 to 4 hrs under dark condition by FP assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 51nMAssay Description:Inhibition of AURKA (unknown origin) using caliper substrate CTD3 by mobility shift assayMore data for this Ligand-Target Pair
Ligand Info
TargetBromodomain-containing protein 4(Human)
University of Chinese Academy of Sciences
Curated by ChEMBL
University of Chinese Academy of Sciences
Curated by ChEMBL
Affinity DataIC50: 52nMAssay Description:Inhibition of BRD4 BD1 (unknown origin) incubated for 2 to 4 hrs under dark condition by FP assayMore data for this Ligand-Target Pair
Ligand Info
TargetBromodomain-containing protein 4(Human)
University of Chinese Academy of Sciences
Curated by ChEMBL
University of Chinese Academy of Sciences
Curated by ChEMBL
Affinity DataIC50: 54nMAssay Description:Inhibition of BRD4 BD1 (unknown origin) incubated for 2 to 4 hrs under dark condition by FP assayMore data for this Ligand-Target Pair
Ligand Info
TargetBromodomain-containing protein 4(Human)
University of Chinese Academy of Sciences
Curated by ChEMBL
University of Chinese Academy of Sciences
Curated by ChEMBL
Affinity DataIC50: 54nMAssay Description:Inhibition of BRD4 BD1 (unknown origin) incubated for 2 to 4 hrs under dark condition by FP assayMore data for this Ligand-Target Pair
Ligand Info
TargetBromodomain-containing protein 4(Human)
University of Chinese Academy of Sciences
Curated by ChEMBL
University of Chinese Academy of Sciences
Curated by ChEMBL
Affinity DataIC50: 55nMAssay Description:Inhibition of BRD4 BD1 (unknown origin) incubated for 2 to 4 hrs under dark condition by FP assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 56nMAssay Description:Inhibition of AURKA (unknown origin) using caliper substrate CTD3 by mobility shift assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 58nMAssay Description:Inhibition of AURKA (unknown origin) using caliper substrate CTD3 by mobility shift assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 62nMAssay Description:Inhibition of AURKA (unknown origin) using caliper substrate CTD3 by mobility shift assayMore data for this Ligand-Target Pair
Ligand Info
TargetBromodomain-containing protein 4(Human)
University of Chinese Academy of Sciences
Curated by ChEMBL
University of Chinese Academy of Sciences
Curated by ChEMBL
Affinity DataIC50: 63nMAssay Description:Inhibition of BRD4 BD1 (unknown origin) incubated for 2 to 4 hrs under dark condition by FP assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 65nMAssay Description:Inhibition of AURKA (unknown origin) using caliper substrate CTD3 by mobility shift assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 68nMAssay Description:Inhibition of AURKA (unknown origin) using caliper substrate CTD3 by mobility shift assayMore data for this Ligand-Target Pair
Ligand Info
TargetBromodomain-containing protein 4(Human)
University of Chinese Academy of Sciences
Curated by ChEMBL
University of Chinese Academy of Sciences
Curated by ChEMBL
Affinity DataIC50: 70nMAssay Description:Inhibition of BRD4 BD2 (unknown origin) incubated for 2 to 4 hrs under dark condition by FP assayMore data for this Ligand-Target Pair
Ligand Info
TargetBromodomain-containing protein 4(Human)
University of Chinese Academy of Sciences
Curated by ChEMBL
University of Chinese Academy of Sciences
Curated by ChEMBL
Affinity DataIC50: 72nMAssay Description:Inhibition of BRD4 BD1 (unknown origin) incubated for 2 to 4 hrs under dark condition by FP assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 72nMAssay Description:Inhibition of AURKA (unknown origin) using caliper substrate CTD3 by mobility shift assayMore data for this Ligand-Target Pair
Ligand Info
TargetBromodomain-containing protein 4(Human)
University of Chinese Academy of Sciences
Curated by ChEMBL
University of Chinese Academy of Sciences
Curated by ChEMBL
Affinity DataIC50: 74nMAssay Description:Inhibition of BRD4 BD1 (unknown origin) incubated for 2 to 4 hrs under dark condition by FP assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 78nMAssay Description:Inhibition of AURKA (unknown origin) using caliper substrate CTD3 by mobility shift assayMore data for this Ligand-Target Pair
Ligand Info

3D Structure (crystal)

































