Report error Found 16 Enz. Inhib. hit(s) with all data for entry = 50023415
Affinity DataIC50: 1.80nMAssay Description:Displacement of [125I] NDP-MSH from mouse MC4R expressed in HEK293 cells incubated for 60 mins by competitive radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:Displacement of [125I] NDP-MSH from mouse MC3R expressed in HEK293 cells incubated for 60 mins by competitive radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 2.10nMAssay Description:Agonist activity at human MC4R expressed in CHO-K1 cells assessed as inhibition constant by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
Affinity DataKi: 3.90nMAssay Description:Agonist activity at human MC1R expressed in CHO-K1 cells assessed as inhibition constant by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 5.80nMAssay Description:Agonist activity at human MC1R expressed in CHO-K1 cells incubated for 40 mins by electro-chemiluminescence assayMore data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Agonist activity at human MC3R expressed in CHO-K1 cells assessed as inhibition constant by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 335nMAssay Description:Displacement of [125I] NDP-MSH from mouse MC4R expressed in HEK293 cells incubated for 60 mins by competitive radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 360nMAssay Description:Displacement of [125I] NDP-MSH from mouse MC4R expressed in HEK293 cells incubated for 60 mins by competitive radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 365nMAssay Description:Displacement of [125I] NDP-MSH from mouse MC4R expressed in HEK293 cells incubated for 60 mins by competitive radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 406nMAssay Description:Displacement of [125I] NDP-MSH from mouse MC4R expressed in HEK293 cells incubated for 60 mins by competitive radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 548nMAssay Description:Displacement of [125I] NDP-MSH from mouse MC4R expressed in HEK293 cells incubated for 60 mins by competitive radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.50E+3nMAssay Description:Displacement of [125I] NDP-MSH from mouse MC3R expressed in HEK293 cells incubated for 60 mins by competitive radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.63E+3nMAssay Description:Displacement of [125I] NDP-MSH from mouse MC3R expressed in HEK293 cells incubated for 60 mins by competitive radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 2.76E+3nMAssay Description:Displacement of [125I] NDP-MSH from mouse MC3R expressed in HEK293 cells incubated for 60 mins by competitive radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 5.18E+3nMAssay Description:Displacement of [125I] NDP-MSH from mouse MC3R expressed in HEK293 cells incubated for 60 mins by competitive radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 7.15E+3nMAssay Description:Displacement of [125I] NDP-MSH from mouse MC3R expressed in HEK293 cells incubated for 60 mins by competitive radioligand binding assayMore data for this Ligand-Target Pair
