Compile Data Set for Download or QSAR
Report error Found 26 Enz. Inhib. hit(s) with all data for entry = 50023642
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-3/gamma-2(Mouse)
University of Copenhagen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50503144BDBM50503144(CHEBI:35420 | CHEMBL1179605)
Affinity DataIC50: 3.20E+3nMAssay Description:Negative allosteric modulation of recombinant mouse alpha1beta3gamma2 GABAA receptor expressed in GFP tagged HEK293 cells at steady state current by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-3/gamma-2(Mouse)
University of Copenhagen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50666250BDBM50666250(CHEMBL6175718)
Affinity DataIC50: 1.00E+4nMAssay Description:Negative allosteric modulation of recombinant mouse alpha1beta3gamma2 GABAA receptor expressed in GFP tagged HEK293 cells at steady state current by ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-3/gamma-2(Mouse)
University of Copenhagen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50666250BDBM50666250(CHEMBL6175718)
Affinity DataIC50: 1.00E+4nMAssay Description:Negative allosteric modulation of recombinant mouse alpha1beta3gamma2 GABAA receptor expressed in GFP tagged HEK293 cells at peak current by whole-ce...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-3/gamma-2(Mouse)
University of Copenhagen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50666241BDBM50666241(CHEMBL6170563)
Affinity DataIC50: 1.20E+4nMAssay Description:Negative allosteric modulation of recombinant mouse alpha1beta3gamma2 GABAA receptor expressed in GFP tagged HEK293 cells at steady state current by ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-3/gamma-2(Mouse)
University of Copenhagen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50666243BDBM50666243(CHEMBL6175627)
Affinity DataIC50: 1.40E+4nMAssay Description:Negative allosteric modulation of recombinant mouse alpha1beta3gamma2 GABAA receptor expressed in GFP tagged HEK293 cells at steady state current by ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-3/gamma-2(Mouse)
University of Copenhagen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50666240BDBM50666240(CHEMBL6177038)
Affinity DataIC50: 1.40E+4nMAssay Description:Negative allosteric modulation of recombinant mouse alpha1beta3gamma2 GABAA receptor expressed in GFP tagged HEK293 cells at steady state current by ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-3/gamma-2(Mouse)
University of Copenhagen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50666241BDBM50666241(CHEMBL6170563)
Affinity DataIC50: 1.50E+4nMAssay Description:Negative allosteric modulation of recombinant mouse alpha1beta3gamma2 GABAA receptor expressed in GFP tagged HEK293 cells at peak current by whole-ce...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-3/gamma-2(Mouse)
University of Copenhagen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50666242BDBM50666242(CHEMBL6162255)
Affinity DataIC50: 1.80E+4nMAssay Description:Negative allosteric modulation of recombinant mouse alpha1beta3gamma2 GABAA receptor expressed in GFP tagged HEK293 cells at steady state current by ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-3/gamma-2(Mouse)
University of Copenhagen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50666247BDBM50666247(CHEMBL6175784)
Affinity DataIC50: 2.00E+4nMAssay Description:Negative allosteric modulation of recombinant mouse alpha1beta3gamma2 GABAA receptor expressed in GFP tagged HEK293 cells at steady state current by ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-3/gamma-2(Mouse)
University of Copenhagen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50666246BDBM50666246(CHEMBL6163254)
Affinity DataIC50: 2.10E+4nMAssay Description:Negative allosteric modulation of recombinant mouse alpha1beta3gamma2 GABAA receptor expressed in GFP tagged HEK293 cells at steady state current by ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-3/gamma-2(Mouse)
University of Copenhagen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50666239BDBM50666239(CHEMBL6176277)
Affinity DataIC50: 2.30E+4nMAssay Description:Negative allosteric modulation of recombinant mouse alpha1beta3gamma2 GABAA receptor expressed in GFP tagged HEK293 cells at steady state current by ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-3/gamma-2(Mouse)
University of Copenhagen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50666246BDBM50666246(CHEMBL6163254)
Affinity DataIC50: 2.70E+4nMAssay Description:Negative allosteric modulation of recombinant mouse alpha1beta3gamma2 GABAA receptor expressed in GFP tagged HEK293 cells at peak current by whole-ce...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-3/gamma-2(Mouse)
University of Copenhagen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50666240BDBM50666240(CHEMBL6177038)
Affinity DataIC50: 2.90E+4nMAssay Description:Negative allosteric modulation of recombinant mouse alpha1beta3gamma2 GABAA receptor expressed in GFP tagged HEK293 cells at peak current by whole-ce...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-3/gamma-2(Mouse)
University of Copenhagen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50666247BDBM50666247(CHEMBL6175784)
Affinity DataIC50: 3.70E+4nMAssay Description:Negative allosteric modulation of recombinant mouse alpha1beta3gamma2 GABAA receptor expressed in GFP tagged HEK293 cells at peak current by whole-ce...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-3/gamma-2(Mouse)
University of Copenhagen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50666248BDBM50666248(CHEMBL6177873)
Affinity DataIC50: 4.20E+4nMAssay Description:Negative allosteric modulation of recombinant mouse alpha1beta3gamma2 GABAA receptor expressed in GFP tagged HEK293 cells at steady state current by ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-3/gamma-2(Mouse)
University of Copenhagen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50666244BDBM50666244(CHEMBL6176804)
Affinity DataIC50: 5.30E+4nMAssay Description:Negative allosteric modulation of recombinant mouse alpha1beta3gamma2 GABAA receptor expressed in GFP tagged HEK293 cells at steady state current by ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-3/gamma-2(Mouse)
University of Copenhagen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50666249BDBM50666249(CHEMBL6168656)
Affinity DataIC50: 5.40E+4nMAssay Description:Negative allosteric modulation of recombinant mouse alpha1beta3gamma2 GABAA receptor expressed in GFP tagged HEK293 cells at steady state current by ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-3/gamma-2(Mouse)
University of Copenhagen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50666242BDBM50666242(CHEMBL6162255)
Affinity DataIC50: 5.50E+4nMAssay Description:Negative allosteric modulation of recombinant mouse alpha1beta3gamma2 GABAA receptor expressed in GFP tagged HEK293 cells at peak current by whole-ce...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-3/gamma-2(Mouse)
University of Copenhagen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50666243BDBM50666243(CHEMBL6175627)
Affinity DataIC50: 5.90E+4nMAssay Description:Negative allosteric modulation of recombinant mouse alpha1beta3gamma2 GABAA receptor expressed in GFP tagged HEK293 cells at peak current by whole-ce...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-3/gamma-2(Mouse)
University of Copenhagen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50666245BDBM50666245(CHEMBL6177060)
Affinity DataIC50: 7.30E+4nMAssay Description:Negative allosteric modulation of recombinant mouse alpha1beta3gamma2 GABAA receptor expressed in GFP tagged HEK293 cells at steady state current by ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-3/gamma-2(Mouse)
University of Copenhagen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50666248BDBM50666248(CHEMBL6177873)
Affinity DataIC50: 7.60E+4nMAssay Description:Negative allosteric modulation of recombinant mouse alpha1beta3gamma2 GABAA receptor expressed in GFP tagged HEK293 cells at peak current by whole-ce...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-3/gamma-2(Mouse)
University of Copenhagen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50666239BDBM50666239(CHEMBL6176277)
Affinity DataIC50: 1.14E+5nMAssay Description:Negative allosteric modulation of recombinant mouse alpha1beta3gamma2 GABAA receptor expressed in GFP tagged HEK293 cells at peak current by whole-ce...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-3/gamma-2(Mouse)
University of Copenhagen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50666249BDBM50666249(CHEMBL6168656)
Affinity DataIC50: 1.28E+5nMAssay Description:Negative allosteric modulation of recombinant mouse alpha1beta3gamma2 GABAA receptor expressed in GFP tagged HEK293 cells at peak current by whole-ce...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-3/gamma-2(Mouse)
University of Copenhagen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50666245BDBM50666245(CHEMBL6177060)
Affinity DataIC50: 1.48E+5nMAssay Description:Negative allosteric modulation of recombinant mouse alpha1beta3gamma2 GABAA receptor expressed in GFP tagged HEK293 cells at peak current by whole-ce...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-3/gamma-2(Mouse)
University of Copenhagen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50666244BDBM50666244(CHEMBL6176804)
Affinity DataIC50: 1.90E+5nMAssay Description:Negative allosteric modulation of recombinant mouse alpha1beta3gamma2 GABAA receptor expressed in GFP tagged HEK293 cells at peak current by whole-ce...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-3/gamma-2(Mouse)
University of Copenhagen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50503144BDBM50503144(CHEBI:35420 | CHEMBL1179605)
Affinity DataIC50: 2.92E+5nMAssay Description:Negative allosteric modulation of recombinant mouse alpha1beta3gamma2 GABAA receptor expressed in GFP tagged HEK293 cells at peak current by whole-ce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMedPDB3D3D Structure (crystal)