Report error Found 24 Enz. Inhib. hit(s) with all data for entry = 50023056
Affinity DataKi: 0.270nMAssay Description:Binding affinity to KAT6A (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Affinity DataKi: 1.60nMAssay Description:Binding affinity to KAT6A (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 7.80nMAssay Description:Binding affinity to KAT6B (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 30nMAssay Description:Inhibition of KAT6A (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 71nMAssay Description:Inhibition of KAT6A (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 83nMAssay Description:Inhibition of KAT6B (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 99nMAssay Description:Inhibition of KAT6A (unknown origin)More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 168nMAssay Description:Inhibition of KAT6A in human MVLN cells assessed as decrease in estrogen receptor level incubated for 24 hrs by gene reporter assayMore data for this Ligand-Target Pair
Affinity DataIC50: 173nMAssay Description:Inhibition of KAT6A (unknown origin)More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 242nMAssay Description:Inhibition of KAT6B (unknown origin)More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 290nMAssay Description:Inhibition of KAT6A (unknown origin)More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 490nMAssay Description:Inhibition of KAT6A (unknown origin) extracted from baculovirus infected Sf9 cells using [3H]-acetyl-coA as substrate measured for 2 hrs by liquid sc...More data for this Ligand-Target Pair
Affinity DataIC50: 500nMAssay Description:Inhibition of KAT7 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 500nMAssay Description:Inhibition of KAT7 (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 500nMAssay Description:Binding affinity to KAT6A (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Affinity DataIC50: 900nMAssay Description:Inhibition of KAT5 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of KAT6A (unknown origin) extracted from baculovirus infected Sf9 cells using [3H]-acetyl-coA as substrate measured for 2 hrs by liquid sc...More data for this Ligand-Target Pair
Affinity DataIC50: 2.20E+3nMAssay Description:Inhibition of KAT5 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibition of KAT6A (unknown origin)More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 3.90E+3nMAssay Description:Inhibition of KAT6A in human MVLN cells assessed as decrease in estrogen receptor level incubated for 24 hrs by gene reporter assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of KAT6A (unknown origin) extracted from baculovirus infected Sf9 cells using [3H]-acetyl-coA as substrate measured for 2 hrs by liquid sc...More data for this Ligand-Target Pair
Affinity DataIC50: 5.40E+3nMAssay Description:Inhibition of KAT6A (unknown origin)More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 8.30E+3nMAssay Description:Inhibition of KAT6B (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of KAT6A in human MVLN cells assessed as decrease in estrogen receptor level incubated for 24 hrs by gene reporter assayMore data for this Ligand-Target Pair
Ligand Info

3D Structure (crystal)










