Compile Data Set for Download or QSAR
Report error Found 11 Enz. Inhib. hit(s) with all data for entry = 50022925
TargetProto-oncogene tyrosine-protein kinase receptor Ret(Human)
University of South Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50656284BDBM50656284(CHEMBL6149497)
Affinity DataIC50: 0.800nMAssay Description:Inhibition of RET auto-kinase activity in human TPC1 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/4/2026
Entry Details
PubMed
TargetProto-oncogene tyrosine-protein kinase receptor Ret(Human)
University of South Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50656285BDBM50656285(CHEMBL6146359)
Affinity DataIC50: 2.40nMAssay Description:Inhibition of RET auto-kinase activity in human TPC1 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/4/2026
Entry Details
PubMed
TargetProto-oncogene tyrosine-protein kinase receptor Ret(Human)
University of South Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50656286BDBM50656286(CHEMBL6103486)
Affinity DataIC50: 6.70nMAssay Description:Inhibition of RET auto-kinase activity in human TPC1 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/4/2026
Entry Details
PubMed
TargetProto-oncogene tyrosine-protein kinase receptor Ret(Human)
University of South Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50656287BDBM50656287(CHEMBL6145448)
Affinity DataIC50: 8.40nMAssay Description:Inhibition of RET auto-kinase activity in human TPC1 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/4/2026
Entry Details
PubMed
TargetProto-oncogene tyrosine-protein kinase receptor Ret(Human)
University of South Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50656288BDBM50656288(CHEMBL6102760)
Affinity DataIC50: 13nMAssay Description:Inhibition of RET auto-kinase activity in human TPC1 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/4/2026
Entry Details
PubMed
TargetProto-oncogene tyrosine-protein kinase receptor Ret(Human)
University of South Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50656280BDBM50656280(CHEMBL6133951)
Affinity DataIC50: 15nMAssay Description:Inhibition of RET auto-kinase activity in human TPC1 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/4/2026
Entry Details
PubMed
TargetProto-oncogene tyrosine-protein kinase receptor Ret(Human)
University of South Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50656279BDBM50656279(CHEMBL6146565)
Affinity DataIC50: 28nMAssay Description:Inhibition of RET auto-kinase activity in human TPC1 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/4/2026
Entry Details
PubMed
TargetProto-oncogene tyrosine-protein kinase receptor Ret(Human)
University of South Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50656278BDBM50656278(CHEMBL6147457)
Affinity DataIC50: 31nMAssay Description:Inhibition of RET auto-kinase activity in human TPC1 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/4/2026
Entry Details
PubMed
TargetProto-oncogene tyrosine-protein kinase receptor Ret(Human)
University of South Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50656281BDBM50656281(CHEMBL6164382)
Affinity DataIC50: 44nMAssay Description:Inhibition of RET auto-kinase activity in human TPC1 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/4/2026
Entry Details
PubMed
TargetProto-oncogene tyrosine-protein kinase receptor Ret(Human)
University of South Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50656283BDBM50656283(CHEMBL6166396)
Affinity DataIC50: 61nMAssay Description:Inhibition of RET auto-kinase activity in human TPC1 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/4/2026
Entry Details
PubMed
TargetProto-oncogene tyrosine-protein kinase receptor Ret(Human)
University of South Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50656282BDBM50656282(CHEMBL6143216)
Affinity DataIC50: 184nMAssay Description:Inhibition of RET auto-kinase activity in human TPC1 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/4/2026
Entry Details
PubMed