Report error Found 90 Enz. Inhib. hit(s) with all data for entry = 50023106
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Human)
Nanjing University of Chinese Medicine
Curated by ChEMBL
Nanjing University of Chinese Medicine
Curated by ChEMBL
Affinity DataKi: 0.0100nMAssay Description:Binding affinity to MCL-1 (unknown origin) assessed as inhibition constant by TR-FRET assayMore data for this Ligand-Target Pair
Ligand Info
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Human)
Nanjing University of Chinese Medicine
Curated by ChEMBL
Nanjing University of Chinese Medicine
Curated by ChEMBL
Affinity DataIC50: 0.0150nMAssay Description:Binding affinity to MCL-1 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Affinity DataKi: 0.0150nMAssay Description:Binding affinity to BCL-XL (unknown origin) assessed as inhibition constant incubated for 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
Ligand Info
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Human)
Nanjing University of Chinese Medicine
Curated by ChEMBL
Nanjing University of Chinese Medicine
Curated by ChEMBL
Affinity DataKi: 0.0150nMAssay Description:Binding affinity to MCL-1 (unknown origin) assessed as inhibition constant by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataKi: 0.0180nMAssay Description:Binding affinity to BCL-XL (unknown origin) assessed as inhibition constant incubated for 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 0.0200nMAssay Description:Binding affinity to BCL-XL (unknown origin) assessed as inhibition constant incubated for 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
Ligand Info
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Human)
Nanjing University of Chinese Medicine
Curated by ChEMBL
Nanjing University of Chinese Medicine
Curated by ChEMBL
Affinity DataKi: 0.0260nMAssay Description:Binding affinity to MCL-1 (unknown origin) assessed as inhibition constant by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Human)
Nanjing University of Chinese Medicine
Curated by ChEMBL
Nanjing University of Chinese Medicine
Curated by ChEMBL
Affinity DataIC50: 0.0500nMAssay Description:Binding affinity to MCL-1 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand Info
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Human)
Nanjing University of Chinese Medicine
Curated by ChEMBL
Nanjing University of Chinese Medicine
Curated by ChEMBL
Affinity DataIC50: 0.0600nMAssay Description:Binding affinity to MCL-1 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Human)
Nanjing University of Chinese Medicine
Curated by ChEMBL
Nanjing University of Chinese Medicine
Curated by ChEMBL
Affinity DataKi: 0.0600nMAssay Description:Binding affinity to MCL-1 (unknown origin) assessed as inhibition constant by TR-FRET assayMore data for this Ligand-Target Pair
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Human)
Nanjing University of Chinese Medicine
Curated by ChEMBL
Nanjing University of Chinese Medicine
Curated by ChEMBL
Affinity DataKi: 0.0970nMAssay Description:Binding affinity to MCL-1 (unknown origin) assessed as inhibition constant by TR-FRET assayMore data for this Ligand-Target Pair
Ligand Info
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Human)
Nanjing University of Chinese Medicine
Curated by ChEMBL
Nanjing University of Chinese Medicine
Curated by ChEMBL
Affinity DataKi: <0.100nMAssay Description:Binding affinity to MCL-1 (unknown origin) assessed as inhibition constant by TR-FRET assayMore data for this Ligand-Target Pair
Ligand Info
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Human)
Nanjing University of Chinese Medicine
Curated by ChEMBL
Nanjing University of Chinese Medicine
Curated by ChEMBL
Affinity DataKi: 0.190nMAssay Description:Binding affinity to MCL-1 (unknown origin) assessed as inhibition constant by SPR assayMore data for this Ligand-Target Pair
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Human)
Nanjing University of Chinese Medicine
Curated by ChEMBL
Nanjing University of Chinese Medicine
Curated by ChEMBL
Affinity DataKi: 0.200nMAssay Description:Binding affinity to MCL-1 (unknown origin) assessed as inhibition constant by TR-FRET assayMore data for this Ligand-Target Pair
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Human)
Nanjing University of Chinese Medicine
Curated by ChEMBL
Nanjing University of Chinese Medicine
Curated by ChEMBL
Affinity DataKi: 0.450nMAssay Description:Binding affinity to MCL-1 (unknown origin) assessed as inhibition constant by TR-FRET assayMore data for this Ligand-Target Pair
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Human)
Nanjing University of Chinese Medicine
Curated by ChEMBL
Nanjing University of Chinese Medicine
Curated by ChEMBL
Affinity DataIC50: 0.700nMAssay Description:Inhibition of N-terminal GST-tagged MCL-1 (unknown origin) extracted form Escherichia coli by TR-FRET assayMore data for this Ligand-Target Pair
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Human)
Nanjing University of Chinese Medicine
Curated by ChEMBL
Nanjing University of Chinese Medicine
Curated by ChEMBL
Affinity DataKi: 1nMAssay Description:Binding affinity to MCL-1 (unknown origin) assessed as inhibition constant by TR-FRET assayMore data for this Ligand-Target Pair
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Human)
Nanjing University of Chinese Medicine
Curated by ChEMBL
Nanjing University of Chinese Medicine
Curated by ChEMBL
Affinity DataKi: 1nMAssay Description:Binding affinity to MCL-1 (unknown origin) assessed as inhibition constant by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:Inhibition of Bcl-XL (unknown origin) by FRET assayMore data for this Ligand-Target Pair
Ligand Info
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Human)
Nanjing University of Chinese Medicine
Curated by ChEMBL
Nanjing University of Chinese Medicine
Curated by ChEMBL
Affinity DataKi: 5.5nMAssay Description:Binding affinity to MCL-1 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand Info
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Human)
Nanjing University of Chinese Medicine
Curated by ChEMBL
Nanjing University of Chinese Medicine
Curated by ChEMBL
Affinity DataIC50: 8nMAssay Description:Inhibition of MCL-1 (unknown origin)More data for this Ligand-Target Pair
Ligand Info
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Human)
Nanjing University of Chinese Medicine
Curated by ChEMBL
Nanjing University of Chinese Medicine
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Inhibition of MCL-1 (unknown origin) by FP assayMore data for this Ligand-Target Pair
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Human)
Nanjing University of Chinese Medicine
Curated by ChEMBL
Nanjing University of Chinese Medicine
Curated by ChEMBL
Affinity DataIC50: 14nMAssay Description:Inhibition of MCL-1 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Ligand Info
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Human)
Nanjing University of Chinese Medicine
Curated by ChEMBL
Nanjing University of Chinese Medicine
Curated by ChEMBL
Affinity DataIC50: 40nMAssay Description:Inhibition of MCL-1 (unknown origin) by FP assayMore data for this Ligand-Target Pair
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Human)
Nanjing University of Chinese Medicine
Curated by ChEMBL
Nanjing University of Chinese Medicine
Curated by ChEMBL
Affinity DataIC50: 42nMAssay Description:Inhibition of N-terminal GST-tagged MCL-1 (unknown origin) extracted form Escherichia coli by TR-FRET assayMore data for this Ligand-Target Pair
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Human)
Nanjing University of Chinese Medicine
Curated by ChEMBL
Nanjing University of Chinese Medicine
Curated by ChEMBL
Affinity DataKi: 51nMAssay Description:Binding affinity to MCL-1 (unknown origin) extracted from Escherichia coli BL21 (DE3) assessed as inhibition constantMore data for this Ligand-Target Pair
Affinity DataKi: 132nMAssay Description:Binding affinity to BCL-2 (unknown origin) assessed as inhibition constant incubated for 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Human)
Nanjing University of Chinese Medicine
Curated by ChEMBL
Nanjing University of Chinese Medicine
Curated by ChEMBL
Affinity DataKi: 180nMAssay Description:Binding affinity to MCL-1 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Affinity DataKi: 200nMAssay Description:Binding affinity to BCL-2 (unknown origin) as assessed as inhibition constantMore data for this Ligand-Target Pair
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Human)
Nanjing University of Chinese Medicine
Curated by ChEMBL
Nanjing University of Chinese Medicine
Curated by ChEMBL
Affinity DataIC50: 200nMAssay Description:Inhibition of MCL-1 (unknown origin)More data for this Ligand-Target Pair
Ligand Info
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Human)
Nanjing University of Chinese Medicine
Curated by ChEMBL
Nanjing University of Chinese Medicine
Curated by ChEMBL
Affinity DataKi: 260nMAssay Description:Binding affinity to MCL-1 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Affinity DataKi: 290nMAssay Description:Binding affinity to Bcl-XL (unknown origin) assessed as inhibition constant by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataKi: 290nMAssay Description:Binding affinity to BCL-2 (unknown origin) as assessed as inhibition constantMore data for this Ligand-Target Pair
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Human)
Nanjing University of Chinese Medicine
Curated by ChEMBL
Nanjing University of Chinese Medicine
Curated by ChEMBL
Affinity DataKi: 300nMAssay Description:Binding affinity to MCL-1 (unknown origin) assessed as inhibition constant by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand Info
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Human)
Nanjing University of Chinese Medicine
Curated by ChEMBL
Nanjing University of Chinese Medicine
Curated by ChEMBL
Affinity DataIC50: 300nMAssay Description:Inhibition of MCL-1 (unknown origin) by FP assayMore data for this Ligand-Target Pair
Affinity DataIC50: 310nMAssay Description:Inhibition of Bcl-XL (unknown origin) by FRET assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 320nMAssay Description:Inhibition of Bcl-2 (unknown origin) by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 320nMAssay Description:Binding affinity to BCL-2 (unknown origin) as assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 320nMAssay Description:Binding affinity to BCL-2 (unknown origin) as assessed as inhibition constantMore data for this Ligand-Target Pair
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Human)
Nanjing University of Chinese Medicine
Curated by ChEMBL
Nanjing University of Chinese Medicine
Curated by ChEMBL
Affinity DataKi: 370nMAssay Description:Binding affinity to MCL-1 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand Info
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Human)
Nanjing University of Chinese Medicine
Curated by ChEMBL
Nanjing University of Chinese Medicine
Curated by ChEMBL
Affinity DataKi: 400nMAssay Description:Binding affinity to MCL-1 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand Info
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Human)
Nanjing University of Chinese Medicine
Curated by ChEMBL
Nanjing University of Chinese Medicine
Curated by ChEMBL
Affinity DataKi: 410nMAssay Description:Binding affinity to MCL-1 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 420nMAssay Description:Binding affinity to BCL-2 (unknown origin) as assessed as inhibition constantMore data for this Ligand-Target Pair
Affinity DataKi: 480nMAssay Description:Binding affinity to Bcl-XL (unknown origin) assessed as inhibition constant by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Human)
Nanjing University of Chinese Medicine
Curated by ChEMBL
Nanjing University of Chinese Medicine
Curated by ChEMBL
Affinity DataKi: 490nMAssay Description:Binding affinity to N-terminal MCL-1 (unknown origin) using 5-FAM peptide as substrate by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 560nMAssay Description:Binding affinity to BCL-2 (unknown origin) as assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: >660nMAssay Description:Binding affinity to BCL-XL (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: >660nMAssay Description:Binding affinity to BCL-XL (unknown origin) assessed as inhibition constant incubated for 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataKi: 700nMAssay Description:Binding affinity to BCL-XL (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Human)
Nanjing University of Chinese Medicine
Curated by ChEMBL
Nanjing University of Chinese Medicine
Curated by ChEMBL
Affinity DataIC50: 770nMAssay Description:Inhibition of N-terminal GST-tagged MCL-1 (unknown origin) extracted form Escherichia coli by TR-FRET assayMore data for this Ligand-Target Pair
Ligand Info








3D Structure (crystal)
























