Compile Data Set for Download or QSAR
Report error Found 17 Enz. Inhib. hit(s) with all data for entry = 50022796
TargetDipeptidyl peptidase 4(Human)
ISF College of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50228403BDBM50228403(8-[(3R)-3-Aminopiperidin-1-yl]-7-but-2-yn-1-yl-3-m...)
Affinity DataIC50: 15nMAssay Description:Agonist activity at rat GPR40 assessed as increase in intracellular calcium flux by cell based FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetDipeptidyl peptidase 4(Human)
ISF College of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50654400BDBM50654400(CHEMBL6143955)
Affinity DataIC50: 16nMAssay Description:Agonist activity at human GPR40 assessed as increase in intracellular calcium flux by cell based FLIPR assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetDipeptidyl peptidase 4(Human)
ISF College of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50654391BDBM50654391(CHEMBL6133644)
Affinity DataIC50: 16nMAssay Description:Agonist activity at human GPR40 assessed as increase in intracellular calcium flux by cell based FLIPR assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetDipeptidyl peptidase 4(Human)
ISF College of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50654390BDBM50654390(CHEMBL1894963)
Affinity DataIC50: 16nMAssay Description:Agonist activity at human GPR40 assessed as increase in intracellular calcium flux by cell based FLIPR assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetDipeptidyl peptidase 4(Human)
ISF College of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50654402BDBM50654402(CHEMBL6150022)
Affinity DataIC50: 17nMAssay Description:Agonist activity at human GPR40 assessed as increase in intracellular calcium flux by cell based FLIPR assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetDipeptidyl peptidase 4(Human)
ISF College of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50654392BDBM50654392(CHEMBL6148404)
Affinity DataIC50: 17nMAssay Description:Agonist activity at human GPR40 assessed as increase in intracellular calcium flux by cell based FLIPR assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetDipeptidyl peptidase 4(Human)
ISF College of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50654396BDBM50654396(CHEMBL6146956)
Affinity DataIC50: 17nMAssay Description:Agonist activity at human GPR40 assessed as increase in intracellular calcium flux by cell based FLIPR assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetDipeptidyl peptidase 4(Human)
ISF College of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50654403BDBM50654403(CHEMBL6132632)
Affinity DataIC50: 19nMAssay Description:Agonist activity at human GPR40 assessed as increase in intracellular calcium flux by cell based FLIPR assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetDipeptidyl peptidase 4(Human)
ISF College of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50654395BDBM50654395(CHEMBL6091879)
Affinity DataIC50: 19nMAssay Description:Agonist activity at human GPR40 assessed as increase in intracellular calcium flux by cell based FLIPR assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetDipeptidyl peptidase 4(Human)
ISF College of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50654397BDBM50654397(CHEMBL6146627)
Affinity DataIC50: 20nMAssay Description:Agonist activity at human GPR40 assessed as increase in intracellular calcium flux by cell based FLIPR assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetDipeptidyl peptidase 4(Human)
ISF College of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50654394BDBM50654394(CHEMBL6160472)
Affinity DataIC50: 22nMAssay Description:Agonist activity at human GPR40 assessed as increase in intracellular calcium flux by cell based FLIPR assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetDipeptidyl peptidase 4(Human)
ISF College of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50654401BDBM50654401(CHEMBL6102689)
Affinity DataIC50: 23nMAssay Description:Agonist activity at human GPR40 assessed as increase in intracellular calcium flux by cell based FLIPR assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetDipeptidyl peptidase 4(Human)
ISF College of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50654405BDBM50654405(CHEMBL6133793)
Affinity DataIC50: 26nMAssay Description:Agonist activity at rat GPR40 assessed as increase in intracellular calcium flux by cell based FLIPR assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetDipeptidyl peptidase 4(Human)
ISF College of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50654404BDBM50654404(CHEMBL6091758)
Affinity DataIC50: 26nMAssay Description:Agonist activity at human GPR40 assessed as increase in intracellular calcium flux by cell based FLIPR assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetDipeptidyl peptidase 4(Human)
ISF College of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50654393BDBM50654393(CHEMBL6147781)
Affinity DataIC50: 28nMAssay Description:Agonist activity at human GPR40 assessed as increase in intracellular calcium flux by cell based FLIPR assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetDipeptidyl peptidase 4(Human)
ISF College of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50654399BDBM50654399(CHEMBL6133561)
Affinity DataIC50: 28nMAssay Description:Agonist activity at human GPR40 assessed as increase in intracellular calcium flux by cell based FLIPR assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetDipeptidyl peptidase 4(Human)
ISF College of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50654398BDBM50654398(CHEMBL5411258)
Affinity DataIC50: 28nMAssay Description:Agonist activity at human GPR40 assessed as increase in intracellular calcium flux by cell based FLIPR assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed