Report error Found 105 Enz. Inhib. hit(s) with all data for entry = 50022721
TargetDNA gyrase A/A/B/B tetramer(Escherichia coli (strain K12))
Ningxia Medical University
Curated by ChEMBL
Ningxia Medical University
Curated by ChEMBL
Affinity DataIC50: 11nMAssay Description:Antagonist activity at human cloned oxytocin receptor by cell based beta lactamase assayMore data for this Ligand-Target Pair
Ligand Info
TargetDNA gyrase A/A/B/B tetramer(Escherichia coli (strain K12))
Ningxia Medical University
Curated by ChEMBL
Ningxia Medical University
Curated by ChEMBL
Affinity DataIC50: 17nMAssay Description:Inhibition of Tie-2 phosphorylation by cell based assayMore data for this Ligand-Target Pair
Ligand Info
TargetDNA gyrase A/A/B/B tetramer(Escherichia coli (strain K12))
Ningxia Medical University
Curated by ChEMBL
Ningxia Medical University
Curated by ChEMBL
Affinity DataIC50: 20nMAssay Description:Antagonist activity at human cloned vasopressin V2 receptor by cell based beta lactamase assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 21nMAssay Description:Inhibition of EphB4 autophosphorylation by cell based assayMore data for this Ligand-Target Pair
Ligand Info
TargetDNA gyrase A/A/B/B tetramer(Escherichia coli (strain K12))
Ningxia Medical University
Curated by ChEMBL
Ningxia Medical University
Curated by ChEMBL
Affinity DataIC50: 21nMAssay Description:Antagonist activity at human cloned oxytocin receptor by cell based beta lactamase assayMore data for this Ligand-Target Pair
Ligand Info
TargetDNA gyrase A/A/B/B tetramer(Escherichia coli (strain K12))
Ningxia Medical University
Curated by ChEMBL
Ningxia Medical University
Curated by ChEMBL
Affinity DataIC50: 24nMAssay Description:Antagonist activity at human cloned oxytocin receptor by cell based beta lactamase assayMore data for this Ligand-Target Pair
Ligand Info
TargetDNA gyrase A/A/B/B tetramer(Escherichia coli (strain K12))
Ningxia Medical University
Curated by ChEMBL
Ningxia Medical University
Curated by ChEMBL
Affinity DataIC50: 32nMAssay Description:Antagonist activity at human cloned oxytocin receptor by cell based beta lactamase assayMore data for this Ligand-Target Pair
Ligand Info
TargetDNA gyrase A/A/B/B tetramer(Escherichia coli (strain K12))
Ningxia Medical University
Curated by ChEMBL
Ningxia Medical University
Curated by ChEMBL
Affinity DataIC50: 34nMAssay Description:Antagonist activity at human cloned oxytocin receptor by cell based beta lactamase assayMore data for this Ligand-Target Pair
Ligand Info
TargetDNA gyrase A/A/B/B tetramer(Escherichia coli (strain K12))
Ningxia Medical University
Curated by ChEMBL
Ningxia Medical University
Curated by ChEMBL
Affinity DataIC50: 42nMAssay Description:Inhibition of Tie-2 phosphorylation by cell based assayMore data for this Ligand-Target Pair
Ligand Info
TargetDNA gyrase A/A/B/B tetramer(Escherichia coli (strain K12))
Ningxia Medical University
Curated by ChEMBL
Ningxia Medical University
Curated by ChEMBL
Affinity DataIC50: 42nMAssay Description:Antagonist activity at human cloned oxytocin receptor by cell based beta lactamase assayMore data for this Ligand-Target Pair
Ligand Info
TargetDNA gyrase A/A/B/B tetramer(Escherichia coli (strain K12))
Ningxia Medical University
Curated by ChEMBL
Ningxia Medical University
Curated by ChEMBL
Affinity DataIC50: 42nMAssay Description:Antagonist activity at human cloned vasopressin V2 receptor by cell based beta lactamase assayMore data for this Ligand-Target Pair
Ligand Info
TargetDNA gyrase A/A/B/B tetramer(Escherichia coli (strain K12))
Ningxia Medical University
Curated by ChEMBL
Ningxia Medical University
Curated by ChEMBL
Affinity DataIC50: 44nMAssay Description:Inhibition of Tie-2 phosphorylation by cell based assayMore data for this Ligand-Target Pair
Ligand Info
TargetDNA gyrase A/A/B/B tetramer(Escherichia coli (strain K12))
Ningxia Medical University
Curated by ChEMBL
Ningxia Medical University
Curated by ChEMBL
Affinity DataIC50: 50nMAssay Description:Antagonist activity at human cloned oxytocin receptor by cell based beta lactamase assayMore data for this Ligand-Target Pair
Ligand Info
TargetDNA gyrase A/A/B/B tetramer(Escherichia coli (strain K12))
Ningxia Medical University
Curated by ChEMBL
Ningxia Medical University
Curated by ChEMBL
Affinity DataIC50: 51nMAssay Description:Antagonist activity at human cloned oxytocin receptor by cell based beta lactamase assayMore data for this Ligand-Target Pair
Ligand Info
TargetDNA gyrase A/A/B/B tetramer(Escherichia coli (strain K12))
Ningxia Medical University
Curated by ChEMBL
Ningxia Medical University
Curated by ChEMBL
Affinity DataIC50: 58nMAssay Description:Inhibition of Tie-2 phosphorylation by cell based assayMore data for this Ligand-Target Pair
Ligand Info
TargetDNA gyrase A/A/B/B tetramer(Escherichia coli (strain K12))
Ningxia Medical University
Curated by ChEMBL
Ningxia Medical University
Curated by ChEMBL
Affinity DataIC50: 59nMAssay Description:Antagonist activity at human cloned vasopressin V2 receptor by cell based beta lactamase assayMore data for this Ligand-Target Pair
Ligand Info
TargetDNA gyrase A/A/B/B tetramer(Escherichia coli (strain K12))
Ningxia Medical University
Curated by ChEMBL
Ningxia Medical University
Curated by ChEMBL
Affinity DataIC50: 67nMAssay Description:Antagonist activity at human cloned vasopressin V1a receptor by cell based beta lactamase assayMore data for this Ligand-Target Pair
Ligand Info
TargetDNA gyrase A/A/B/B tetramer(Escherichia coli (strain K12))
Ningxia Medical University
Curated by ChEMBL
Ningxia Medical University
Curated by ChEMBL
Affinity DataIC50: 70nMAssay Description:Antagonist activity at human cloned vasopressin V2 receptor by cell based beta lactamase assayMore data for this Ligand-Target Pair
Ligand Info
TargetDNA gyrase A/A/B/B tetramer(Escherichia coli (strain K12))
Ningxia Medical University
Curated by ChEMBL
Ningxia Medical University
Curated by ChEMBL
Affinity DataIC50: 70nMAssay Description:Inhibition of Tie-2 phosphorylation by cell based assayMore data for this Ligand-Target Pair
Ligand Info
TargetDNA gyrase A/A/B/B tetramer(Escherichia coli (strain K12))
Ningxia Medical University
Curated by ChEMBL
Ningxia Medical University
Curated by ChEMBL
Affinity DataIC50: 72nMAssay Description:Antagonist activity at human cloned vasopressin V1a receptor by cell based beta lactamase assayMore data for this Ligand-Target Pair
Ligand Info
TargetDNA gyrase A/A/B/B tetramer(Escherichia coli (strain K12))
Ningxia Medical University
Curated by ChEMBL
Ningxia Medical University
Curated by ChEMBL
Affinity DataIC50: 75nMAssay Description:Antagonist activity at human cloned vasopressin V2 receptor by cell based beta lactamase assayMore data for this Ligand-Target Pair
Ligand Info
TargetDNA gyrase A/A/B/B tetramer(Escherichia coli (strain K12))
Ningxia Medical University
Curated by ChEMBL
Ningxia Medical University
Curated by ChEMBL
Affinity DataIC50: 78nMAssay Description:Inhibition of Tie-2 phosphorylation by cell based assayMore data for this Ligand-Target Pair
Ligand Info
TargetDNA gyrase A/A/B/B tetramer(Escherichia coli (strain K12))
Ningxia Medical University
Curated by ChEMBL
Ningxia Medical University
Curated by ChEMBL
Affinity DataIC50: 79nMAssay Description:Antagonist activity at human cloned vasopressin V1a receptor by cell based beta lactamase assayMore data for this Ligand-Target Pair
Ligand Info
TargetDNA gyrase A/A/B/B tetramer(Escherichia coli (strain K12))
Ningxia Medical University
Curated by ChEMBL
Ningxia Medical University
Curated by ChEMBL
Affinity DataIC50: 83nMAssay Description:Inhibition of Tie-2 phosphorylation by cell based assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 85nMAssay Description:Inhibition of EphB4 autophosphorylation by cell based assayMore data for this Ligand-Target Pair
Ligand Info
TargetDNA gyrase A/A/B/B tetramer(Escherichia coli (strain K12))
Ningxia Medical University
Curated by ChEMBL
Ningxia Medical University
Curated by ChEMBL
Affinity DataIC50: 100nMAssay Description:Antagonist activity at human cloned vasopressin V1a receptor by cell based beta lactamase assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 110nMAssay Description:Inhibition of EphB4 autophosphorylation by cell based assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 120nMAssay Description:Inhibition of EphB4 autophosphorylation by cell based assayMore data for this Ligand-Target Pair
Ligand Info
TargetDNA gyrase A/A/B/B tetramer(Escherichia coli (strain K12))
Ningxia Medical University
Curated by ChEMBL
Ningxia Medical University
Curated by ChEMBL
Affinity DataIC50: 130nMAssay Description:Antagonist activity at human cloned vasopressin V1a receptor by cell based beta lactamase assayMore data for this Ligand-Target Pair
Ligand Info
TargetDNA gyrase A/A/B/B tetramer(Escherichia coli (strain K12))
Ningxia Medical University
Curated by ChEMBL
Ningxia Medical University
Curated by ChEMBL
Affinity DataIC50: 130nMAssay Description:Antagonist activity at human cloned vasopressin V1a receptor by cell based beta lactamase assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 130nMAssay Description:Inhibition of EphB4 autophosphorylation by cell based assayMore data for this Ligand-Target Pair
Ligand Info
TargetDNA gyrase A/A/B/B tetramer(Escherichia coli (strain K12))
Ningxia Medical University
Curated by ChEMBL
Ningxia Medical University
Curated by ChEMBL
Affinity DataIC50: 130nMAssay Description:Antagonist activity at human cloned vasopressin V1a receptor by cell based beta lactamase assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 150nMAssay Description:Inhibition of EphB4 autophosphorylation by cell based assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 160nMAssay Description:Inhibition of EphB4 autophosphorylation by cell based assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 170nMAssay Description:Inhibition of EphB4 autophosphorylation by cell based assayMore data for this Ligand-Target Pair
Ligand Info
TargetDNA gyrase A/A/B/B tetramer(Escherichia coli (strain K12))
Ningxia Medical University
Curated by ChEMBL
Ningxia Medical University
Curated by ChEMBL
Affinity DataIC50: 180nMAssay Description:Antagonist activity at human cloned oxytocin receptor by cell based beta lactamase assayMore data for this Ligand-Target Pair
Ligand Info
TargetDNA gyrase A/A/B/B tetramer(Escherichia coli (strain K12))
Ningxia Medical University
Curated by ChEMBL
Ningxia Medical University
Curated by ChEMBL
Affinity DataIC50: 190nMAssay Description:Antagonist activity at human cloned vasopressin V1a receptor by cell based beta lactamase assayMore data for this Ligand-Target Pair
Ligand Info
TargetDNA gyrase A/A/B/B tetramer(Escherichia coli (strain K12))
Ningxia Medical University
Curated by ChEMBL
Ningxia Medical University
Curated by ChEMBL
Affinity DataIC50: 190nMAssay Description:Antagonist activity at human cloned vasopressin V1a receptor by cell based beta lactamase assayMore data for this Ligand-Target Pair
Ligand Info
TargetDNA gyrase A/A/B/B tetramer(Escherichia coli (strain K12))
Ningxia Medical University
Curated by ChEMBL
Ningxia Medical University
Curated by ChEMBL
Affinity DataIC50: 230nMAssay Description:Antagonist activity at human cloned vasopressin V2 receptor by cell based beta lactamase assayMore data for this Ligand-Target Pair
Ligand Info
TargetDNA gyrase A/A/B/B tetramer(Escherichia coli (strain K12))
Ningxia Medical University
Curated by ChEMBL
Ningxia Medical University
Curated by ChEMBL
Affinity DataIC50: 240nMAssay Description:Antagonist activity at human cloned vasopressin V2 receptor by cell based beta lactamase assayMore data for this Ligand-Target Pair
Ligand Info
TargetDNA gyrase A/A/B/B tetramer(Escherichia coli (strain K12))
Ningxia Medical University
Curated by ChEMBL
Ningxia Medical University
Curated by ChEMBL
Affinity DataIC50: 250nMAssay Description:Antagonist activity at human cloned oxytocin receptor by cell based beta lactamase assayMore data for this Ligand-Target Pair
Ligand Info
TargetDNA gyrase A/A/B/B tetramer(Escherichia coli (strain K12))
Ningxia Medical University
Curated by ChEMBL
Ningxia Medical University
Curated by ChEMBL
Affinity DataIC50: 250nMAssay Description:Antagonist activity at human cloned vasopressin V1a receptor by cell based beta lactamase assayMore data for this Ligand-Target Pair
Ligand Info
TargetDNA gyrase A/A/B/B tetramer(Escherichia coli (strain K12))
Ningxia Medical University
Curated by ChEMBL
Ningxia Medical University
Curated by ChEMBL
Affinity DataIC50: 280nMAssay Description:Antagonist activity at human cloned oxytocin receptor by cell based beta lactamase assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 280nMAssay Description:Inhibition of EphB4 autophosphorylation by cell based assayMore data for this Ligand-Target Pair
Ligand Info
TargetDNA gyrase A/A/B/B tetramer(Escherichia coli (strain K12))
Ningxia Medical University
Curated by ChEMBL
Ningxia Medical University
Curated by ChEMBL
Affinity DataIC50: 280nMAssay Description:Inhibition of Tie-2 phosphorylation by cell based assayMore data for this Ligand-Target Pair
Ligand Info
TargetDNA gyrase A/A/B/B tetramer(Escherichia coli (strain K12))
Ningxia Medical University
Curated by ChEMBL
Ningxia Medical University
Curated by ChEMBL
Affinity DataIC50: 280nMAssay Description:Antagonist activity at human cloned vasopressin V1a receptor by cell based beta lactamase assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 280nMAssay Description:Inhibition of EphB4 autophosphorylation by cell based assayMore data for this Ligand-Target Pair
Ligand Info
TargetDNA gyrase A/A/B/B tetramer(Escherichia coli (strain K12))
Ningxia Medical University
Curated by ChEMBL
Ningxia Medical University
Curated by ChEMBL
Affinity DataIC50: 300nMAssay Description:Antagonist activity at human cloned oxytocin receptor by cell based beta lactamase assayMore data for this Ligand-Target Pair
Ligand Info
TargetDNA gyrase A/A/B/B tetramer(Escherichia coli (strain K12))
Ningxia Medical University
Curated by ChEMBL
Ningxia Medical University
Curated by ChEMBL
Affinity DataIC50: 330nMAssay Description:Antagonist activity at human cloned vasopressin V1a receptor by cell based beta lactamase assayMore data for this Ligand-Target Pair
Ligand Info
TargetDNA gyrase A/A/B/B tetramer(Escherichia coli (strain K12))
Ningxia Medical University
Curated by ChEMBL
Ningxia Medical University
Curated by ChEMBL
Affinity DataIC50: 340nMAssay Description:Inhibition of Tie-2 phosphorylation by cell based assayMore data for this Ligand-Target Pair
Ligand Info























