Compile Data Set for Download or QSAR
Report error Found 16 Enz. Inhib. hit(s) with all data for entry = 50022787
TargetEphrin type-A receptor 4(Human)
University of California Riverside

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50654300BDBM50654300(CHEMBL6133286)
Affinity DataKd:  137nMAssay Description:Activation of GIRK1/2 (unknown origin) by cell-based thallium flux assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetEphrin type-A receptor 4(Human)
University of California Riverside

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50654290BDBM50654290(CHEMBL6134295)
Affinity DataKd:  138nMAssay Description:Inhibition of JAK2 in human TF1 cells assessed as inhibition of Epo-induced STAT5 phosphorylation pretreated for 20 minutes prior to addition of cyto...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetEphrin type-A receptor 4(Human)
University of California Riverside

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50654299BDBM50654299(CHEMBL6083126)
Affinity DataKd:  168nMAssay Description:Activation of GIRK1/2 (unknown origin) by cell-based thallium flux assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetEphrin type-A receptor 4(Human)
University of California Riverside

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50654303BDBM50654303(CHEMBL6152488)
Affinity DataKd:  195nMAssay Description:Activation of GIRK1/4 (unknown origin) by cell-based thallium flux assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetEphrin type-A receptor 4(Human)
University of California Riverside

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50654293BDBM50654293(CHEMBL6159993)
Affinity DataKd:  196nMAssay Description:Activation of GIRK1/4 (unknown origin) by cell-based thallium flux assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetEphrin type-A receptor 4(Human)
University of California Riverside

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50654301BDBM50654301(CHEMBL6161313)
Affinity DataKd:  202nMAssay Description:Activation of GIRK1/2 (unknown origin) by cell-based thallium flux assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetEphrin type-A receptor 4(Human)
University of California Riverside

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50654292BDBM50654292(CHEMBL6102998)
Affinity DataKd:  203nMAssay Description:Activation of GIRK1/4 (unknown origin) by cell-based thallium flux assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetEphrin type-A receptor 4(Human)
University of California Riverside

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50654302BDBM50654302(CHEMBL6149801)
Affinity DataKd:  205nMAssay Description:Activation of GIRK1/4 (unknown origin) by cell-based thallium flux assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetEphrin type-A receptor 4(Human)
University of California Riverside

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50654289BDBM50654289(CHEMBL6161902)
Affinity DataKd:  208nMAssay Description:Inhibition of JAK1 in human TF1 cells assessed as inhibition of IL6-induced STAT3 phosphorylation pretreated for 20 minutes prior to addition of cyto...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetEphrin type-A receptor 4(Human)
University of California Riverside

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50654288BDBM50654288(CHEMBL6149414)
Affinity DataKd:  253nMAssay Description:Inhibition of TEL-fused TRKA (unknown origin) by cell-based assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetEphrin type-A receptor 4(Human)
University of California Riverside

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50654298BDBM50654298(CHEMBL6091958)
Affinity DataKd:  335nMAssay Description:Activation of GIRK1/2 (unknown origin) by cell-based thallium flux assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetEphrin type-A receptor 4(Human)
University of California Riverside

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50654295BDBM50654295(CHEMBL6120711)
Affinity DataKd:  346nMAssay Description:Activation of GIRK1/2 (unknown origin) by cell-based thallium flux assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetEphrin type-A receptor 4(Human)
University of California Riverside

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50654296BDBM50654296(CHEMBL6145036)
Affinity DataKd:  374nMAssay Description:Activation of GIRK1/2 (unknown origin) by cell-based thallium flux assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetEphrin type-A receptor 4(Human)
University of California Riverside

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50654297BDBM50654297(CHEMBL6120234)
Affinity DataKd:  381nMAssay Description:Activation of GIRK1/2 (unknown origin) by cell-based thallium flux assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetEphrin type-A receptor 4(Human)
University of California Riverside

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50654294BDBM50654294(CHEMBL6144489)
Affinity DataKd:  430nMAssay Description:Activation of GIRK1/4 (unknown origin) by cell-based thallium flux assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetEphrin type-A receptor 4(Human)
University of California Riverside

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50654291BDBM50654291(CHEMBL6133078)
Affinity DataKd:  436nMAssay Description:Activation of GIRK1/4 (unknown origin) by cell-based thallium flux assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed