Compile Data Set for Download or QSAR
Report error Found 22 Enz. Inhib. hit(s) with all data for entry = 50022775
TargetMelanocyte-stimulating hormone receptor(Human)
Mitsubishi Tanabe Pharma Corporation

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50654200BDBM50654200(Dersimelagon phosphoric acid | MT-7117 phosphate |...)
Affinity DataKi:  2.30nMAssay Description:Inhibition of Nav1.7 by cell based whole-cell voltage clamp electrophysiology assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetMelanocyte-stimulating hormone receptor(Human)
Mitsubishi Tanabe Pharma Corporation

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50654199BDBM50654199(CHEMBL6151605)
Affinity DataEC50:  5.90nMAssay Description:Inhibition of Nav1.5 by cell based whole-cell voltage clamp electrophysiology assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetMelanocyte-stimulating hormone receptor(Human)
Mitsubishi Tanabe Pharma Corporation

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50654200BDBM50654200(Dersimelagon phosphoric acid | MT-7117 phosphate |...)
Affinity DataEC50:  8.20nMAssay Description:Inhibition of Nav1.5 by cell based whole-cell voltage clamp electrophysiology assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetMelanocyte-stimulating hormone receptor(Human)
Mitsubishi Tanabe Pharma Corporation

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50654201BDBM50654201(CHEMBL6134400)
Affinity DataEC50:  10nMAssay Description:Inhibition of Nav1.5 by cell based whole-cell voltage clamp electrophysiology assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetMelanocyte-stimulating hormone receptor(Human)
Mitsubishi Tanabe Pharma Corporation

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50654191BDBM50654191(CHEMBL6151482)
Affinity DataEC50:  18nMAssay Description:Inhibition of Nav1.7 by cell based whole-cell voltage clamp electrophysiology assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetMelanocyte-stimulating hormone receptor(Human)
Mitsubishi Tanabe Pharma Corporation

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50654196BDBM50654196(CHEMBL6142685)
Affinity DataEC50:  23nMAssay Description:Inhibition of Nav1.5 by cell based whole-cell voltage clamp electrophysiology assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetMelanocyte-stimulating hormone receptor(Human)
Mitsubishi Tanabe Pharma Corporation

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50654186BDBM50654186(CHEMBL6151083)
Affinity DataEC50:  29nMAssay Description:Inhibition of Nav1.7 by cell based whole-cell voltage clamp electrophysiology assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetMelanocortin receptor 4(Human)
Mitsubishi Tanabe Pharma Corporation

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50654200BDBM50654200(Dersimelagon phosphoric acid | MT-7117 phosphate |...)
Affinity DataKi:  33nMAssay Description:Inhibition of Nav1.7 by cell based whole-cell voltage clamp electrophysiology assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetMelanocyte-stimulating hormone receptor(Human)
Mitsubishi Tanabe Pharma Corporation

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50654197BDBM50654197(CHEMBL6102073)
Affinity DataEC50:  51nMAssay Description:Inhibition of Nav1.7 by cell based whole-cell voltage clamp electrophysiology assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetMelanocyte-stimulating hormone receptor(Human)
Mitsubishi Tanabe Pharma Corporation

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50654198BDBM50654198(CHEMBL6133359)
Affinity DataEC50:  55nMAssay Description:Inhibition of Nav1.5 by cell based whole-cell voltage clamp electrophysiology assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetMelanocyte-stimulating hormone receptor(Human)
Mitsubishi Tanabe Pharma Corporation

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50654190BDBM50654190(CHEMBL6102507)
Affinity DataEC50:  55nMAssay Description:Inhibition of Nav1.7 by cell based whole-cell voltage clamp electrophysiology assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetMelanocyte-stimulating hormone receptor(Human)
Mitsubishi Tanabe Pharma Corporation

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50602084BDBM50602084(CHEMBL5177709)
Affinity DataEC50:  77nMAssay Description:Inhibition of Nav1.7 by cell based whole-cell voltage clamp electrophysiology assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetMelanocyte-stimulating hormone receptor(Human)
Mitsubishi Tanabe Pharma Corporation

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50654192BDBM50654192(CHEMBL6141822)
Affinity DataEC50:  125nMAssay Description:Inhibition of Nav1.7 by cell based whole-cell voltage clamp electrophysiology assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetMelanocyte-stimulating hormone receptor(Human)
Mitsubishi Tanabe Pharma Corporation

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50654193BDBM50654193(CHEMBL6147055)
Affinity DataEC50:  130nMAssay Description:Inhibition of Nav1.5 by cell based whole-cell voltage clamp electrophysiology assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetMelanocyte-stimulating hormone receptor(Human)
Mitsubishi Tanabe Pharma Corporation

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50654195BDBM50654195(CHEMBL6108925)
Affinity DataEC50:  158nMAssay Description:Inhibition of Nav1.5 by cell based whole-cell voltage clamp electrophysiology assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetMelanocyte-stimulating hormone receptor(Human)
Mitsubishi Tanabe Pharma Corporation

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50654188BDBM50654188(CHEMBL6133478)
Affinity DataEC50:  206nMAssay Description:Inhibition of Nav1.7 by cell based whole-cell voltage clamp electrophysiology assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetMelanocyte-stimulating hormone receptor(Human)
Mitsubishi Tanabe Pharma Corporation

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50654187BDBM50654187(CHEMBL6147466)
Affinity DataEC50:  261nMAssay Description:Inhibition of Nav1.7 by cell based whole-cell voltage clamp electrophysiology assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetMelanocyte-stimulating hormone receptor(Human)
Mitsubishi Tanabe Pharma Corporation

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50654189BDBM50654189(CHEMBL6147944)
Affinity DataEC50:  428nMAssay Description:Inhibition of Nav1.7 by cell based whole-cell voltage clamp electrophysiology assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetMelanocortin receptor 5(Human)
Mitsubishi Tanabe Pharma Corporation

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50654200BDBM50654200(Dersimelagon phosphoric acid | MT-7117 phosphate |...)
Affinity DataKi:  486nMAssay Description:Inhibition of Nav1.7 by cell based whole-cell voltage clamp electrophysiology assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetMelanocyte-stimulating hormone receptor(Human)
Mitsubishi Tanabe Pharma Corporation

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50654194BDBM50654194(CHEMBL6146325)
Affinity DataEC50:  599nMAssay Description:Inhibition of Nav1.5 by cell based whole-cell voltage clamp electrophysiology assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetMelanocyte-stimulating hormone receptor(Human)
Mitsubishi Tanabe Pharma Corporation

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50654185BDBM50654185(CHEMBL6133755)
Affinity DataEC50:  1.07E+3nMAssay Description:Inhibition of Nav1.7 by cell based whole-cell voltage clamp electrophysiology assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetMelanocortin receptor 3(Human)
Mitsubishi Tanabe Pharma Corporation

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50654200BDBM50654200(Dersimelagon phosphoric acid | MT-7117 phosphate |...)
Affinity DataKi:  1.42E+3nMAssay Description:Inhibition of Nav1.7 by cell based whole-cell voltage clamp electrophysiology assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed