Compile Data Set for Download or QSAR
Report error Found 20 Enz. Inhib. hit(s) with all data for entry = 50023277
TargetSolute carrier family 22 member 12(Human)
Peking Union Medical College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 290431BDBM290431(RDEA3170 | US10100016, Verinurad (RDEA3170) | CAS ...)
Affinity DataIC50: 25nMAssay Description:Inhibition of human URAT1 expressed in HEK293T cells using 14C-uric acid as substrate preincubated for 5 mins followed by substrate addition and meas...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2026
Entry Details
PubMed
TargetSolute carrier family 22 member 12(Human)
Peking Union Medical College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50661292BDBM50661292(CHEMBL6152505)
Affinity DataIC50: 180nMAssay Description:Inhibition of URAT1 (unknown origin) expressed in HEK293 cells using 14C-uric acid as substrateMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/5/2026
Entry Details
PubMed
TargetSolute carrier family 22 member 12(Human)
Peking Union Medical College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50661295BDBM50661295(CHEMBL6167127)
Affinity DataIC50: 290nMAssay Description:Inhibition of URAT1 (unknown origin) expressed in HEK293 cells using 14C-uric acid as substrateMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/5/2026
Entry Details
PubMed
TargetSolute carrier family 22 member 12(Human)
Peking Union Medical College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50158460BDBM50158460(cid_2333 | Benzbromarone | 3,5-dibromo-4-hydroxyph...)
Affinity DataIC50: 390nMAssay Description:Inhibition of URAT1 (unknown origin) expressed in HEK293 cells using 14C-uric acid as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2026
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetSolute carrier family 22 member 12(Human)
Peking Union Medical College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50661291BDBM50661291(CHEMBL6160672)
Affinity DataIC50: 490nMAssay Description:Inhibition of URAT1 (unknown origin) expressed in HEK293 cells using 14C-uric acid as substrateMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/5/2026
Entry Details
PubMed
TargetSolute carrier family 22 member 12(Human)
Peking Union Medical College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50661293BDBM50661293(CHEMBL6172772)
Affinity DataIC50: 650nMAssay Description:Inhibition of URAT1 (unknown origin) expressed in HEK293 cells using 14C-uric acid as substrateMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/5/2026
Entry Details
PubMed
TargetSolute carrier family 22 member 12(Human)
Peking Union Medical College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50661301BDBM50661301(CHEMBL6142674)
Affinity DataIC50: 700nMAssay Description:Inhibition of URAT1 (unknown origin) expressed in HEK293 cells using 14C-uric acid as substrateMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/5/2026
Entry Details
PubMed
TargetSolute carrier family 22 member 12(Human)
Peking Union Medical College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50661298BDBM50661298(CHEMBL6159847)
Affinity DataIC50: 750nMAssay Description:Inhibition of URAT1 (unknown origin) expressed in HEK293 cells using 14C-uric acid as substrateMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/5/2026
Entry Details
PubMed
TargetSolute carrier family 22 member 12(Human)
Peking Union Medical College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50661290BDBM50661290(CHEMBL6163421)
Affinity DataIC50: 780nMAssay Description:Inhibition of URAT1 (unknown origin) expressed in HEK293 cells using 14C-uric acid as substrateMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/5/2026
Entry Details
PubMed
TargetSolute carrier family 22 member 12(Human)
Peking Union Medical College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50661289BDBM50661289(CHEMBL6160542)
Affinity DataIC50: 940nMAssay Description:Inhibition of URAT1 (unknown origin) expressed in HEK293 cells using 14C-uric acid as substrateMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/5/2026
Entry Details
PubMed
TargetSolute carrier family 22 member 12(Human)
Peking Union Medical College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50661297BDBM50661297(CHEMBL6144160)
Affinity DataIC50: 990nMAssay Description:Inhibition of URAT1 (unknown origin) expressed in HEK293 cells using 14C-uric acid as substrateMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/5/2026
Entry Details
PubMed
TargetSolute carrier family 22 member 12(Human)
Peking Union Medical College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50661302BDBM50661302(CHEMBL6163087)
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of URAT1 (unknown origin) expressed in HEK293 cells using 14C-uric acid as substrateMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/5/2026
Entry Details
PubMed
TargetSolute carrier family 22 member 12(Human)
Peking Union Medical College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50661300BDBM50661300(CHEMBL6160181)
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of URAT1 (unknown origin) expressed in HEK293 cells using 14C-uric acid as substrateMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/5/2026
Entry Details
PubMed
TargetSolute carrier family 22 member 12(Human)
Peking Union Medical College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50661294BDBM50661294(CHEMBL6151370)
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of URAT1 (unknown origin) expressed in HEK293 cells using 14C-uric acid as substrateMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/5/2026
Entry Details
PubMed
TargetSolute carrier family 22 member 12(Human)
Peking Union Medical College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50661287BDBM50661287(CHEMBL6173784)
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of URAT1 (unknown origin) expressed in HEK293 cells using 14C-uric acid as substrateMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/5/2026
Entry Details
PubMed
TargetSolute carrier family 22 member 12(Human)
Peking Union Medical College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50661296BDBM50661296(CHEMBL6161793)
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of URAT1 (unknown origin) expressed in HEK293 cells using 14C-uric acid as substrateMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/5/2026
Entry Details
PubMed
TargetSolute carrier family 22 member 12(Human)
Peking Union Medical College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50661288BDBM50661288(CHEMBL6167300)
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of URAT1 (unknown origin) expressed in HEK293 cells using 14C-uric acid as substrateMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/5/2026
Entry Details
PubMed
TargetSolute carrier family 22 member 12(Human)
Peking Union Medical College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50661299BDBM50661299(CHEMBL6168363)
Affinity DataIC50: 2.20E+3nMAssay Description:Inhibition of URAT1 (unknown origin) expressed in HEK293 cells using 14C-uric acid as substrateMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/5/2026
Entry Details
PubMed
TargetSolute carrier family 22 member 12(Human)
Peking Union Medical College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50661303BDBM50661303(CHEMBL6159636)
Affinity DataIC50: 3.20E+3nMAssay Description:Inhibition of URAT1 (unknown origin) expressed in HEK293 cells using 14C-uric acid as substrateMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/5/2026
Entry Details
PubMed
TargetSolute carrier family 22 member 12(Human)
Peking Union Medical College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50661304BDBM50661304(CHEMBL6164271)
Affinity DataIC50: 5.10E+3nMAssay Description:Inhibition of URAT1 (unknown origin) expressed in HEK293 cells using 14C-uric acid as substrateMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/5/2026
Entry Details
PubMed