Report error Found 53 Enz. Inhib. hit(s) with all data for entry = 50023036
Affinity DataEC50: 48nMAssay Description:Agonist activity at FXR-LBD (unknown origin) incubated for 3 hrs using fluorescein coactivator peptide by FRET assayMore data for this Ligand-Target Pair
Affinity DataEC50: 51nMAssay Description:Agonist activity at FXR-LBD (unknown origin) incubated for 3 hrs using fluorescein coactivator peptide by FRET assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataEC50: 64nMAssay Description:Agonist activity at FXR-LBD (unknown origin) incubated for 3 hrs using fluorescein coactivator peptide by FRET assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataEC50: 72nMAssay Description:Agonist activity at FXR-LBD (unknown origin) incubated for 3 hrs using fluorescein coactivator peptide by FRET assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataEC50: 76nMAssay Description:Agonist activity at FXR-LBD (unknown origin) expressed in human HepG2 cells incubated for 24 hrs by cell based analysisMore data for this Ligand-Target Pair
Ligand Info
Affinity DataEC50: 76nMAssay Description:Agonist activity at FXR-LBD (unknown origin) incubated for 3 hrs using fluorescein coactivator peptide by FRET assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataEC50: 82nMAssay Description:Agonist activity at FXR-LBD (unknown origin) expressed in human HepG2 cells incubated for 24 hrs by cell based analysisMore data for this Ligand-Target Pair
Affinity DataEC50: 83nMAssay Description:Agonist activity at FXR-LBD (unknown origin) expressed in human HepG2 cells incubated for 24 hrs by cell based analysisMore data for this Ligand-Target Pair
Ligand Info
Affinity DataEC50: 85nMAssay Description:Agonist activity at FXR-LBD (unknown origin) incubated for 3 hrs using fluorescein coactivator peptide by FRET assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataEC50: 95nMAssay Description:Agonist activity at FXR-LBD (unknown origin) expressed in human HepG2 cells incubated for 24 hrs by cell based analysisMore data for this Ligand-Target Pair
Ligand Info
Affinity DataEC50: 98nMAssay Description:Agonist activity at FXR-LBD (unknown origin) incubated for 3 hrs using fluorescein coactivator peptide by FRET assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataEC50: 98nMAssay Description:Agonist activity at FXR-LBD (unknown origin) expressed in human HepG2 cells incubated for 24 hrs by cell based analysisMore data for this Ligand-Target Pair
Ligand Info
Affinity DataEC50: 125nMAssay Description:Agonist activity at FXR-LBD (unknown origin) expressed in human HepG2 cells incubated for 24 hrs by cell based analysisMore data for this Ligand-Target Pair
Ligand Info
Affinity DataEC50: 139nMAssay Description:Agonist activity at FXR-LBD (unknown origin) incubated for 3 hrs using fluorescein coactivator peptide by FRET assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataEC50: 163nMAssay Description:Agonist activity at FXR-LBD (unknown origin) expressed in human HepG2 cells incubated for 24 hrs by cell based analysisMore data for this Ligand-Target Pair
Ligand Info
Affinity DataEC50: 193nMAssay Description:Agonist activity at FXR-LBD (unknown origin) incubated for 3 hrs using fluorescein coactivator peptide by FRET assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataEC50: 206nMAssay Description:Agonist activity at FXR-LBD (unknown origin) incubated for 3 hrs using fluorescein coactivator peptide by FRET assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataEC50: 210nMAssay Description:Agonist activity at FXR-LBD (unknown origin) incubated for 3 hrs using fluorescein coactivator peptide by FRET assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataEC50: 253nMAssay Description:Agonist activity at FXR-LBD (unknown origin) incubated for 3 hrs using fluorescein coactivator peptide by FRET assayMore data for this Ligand-Target Pair
Affinity DataEC50: 254nMAssay Description:Agonist activity at FXR-LBD (unknown origin) incubated for 3 hrs using fluorescein coactivator peptide by FRET assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataEC50: 258nMAssay Description:Agonist activity at FXR-LBD (unknown origin) incubated for 3 hrs using fluorescein coactivator peptide by FRET assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataEC50: 268nMAssay Description:Agonist activity at FXR-LBD (unknown origin) incubated for 3 hrs using fluorescein coactivator peptide by FRET assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataEC50: 305nMAssay Description:Agonist activity at FXR-LBD (unknown origin) incubated for 3 hrs using fluorescein coactivator peptide by FRET assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataEC50: 320nMAssay Description:Agonist activity at FXR-LBD (unknown origin) incubated for 3 hrs using fluorescein coactivator peptide by FRET assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataEC50: 436nMAssay Description:Agonist activity at FXR-LBD (unknown origin) expressed in human HepG2 cells incubated for 24 hrs by cell based analysisMore data for this Ligand-Target Pair
Ligand Info
Affinity DataEC50: 447nMAssay Description:Agonist activity at FXR-LBD (unknown origin) expressed in human HepG2 cells incubated for 24 hrs by cell based analysisMore data for this Ligand-Target Pair
Ligand Info
Affinity DataEC50: 475nMAssay Description:Agonist activity at FXR-LBD (unknown origin) incubated for 3 hrs using fluorescein coactivator peptide by FRET assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataEC50: 497nMAssay Description:Agonist activity at FXR-LBD (unknown origin) incubated for 3 hrs using fluorescein coactivator peptide by FRET assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataEC50: 517nMAssay Description:Agonist activity at FXR-LBD (unknown origin) incubated for 3 hrs using fluorescein coactivator peptide by FRET assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataEC50: 558nMAssay Description:Agonist activity at FXR-LBD (unknown origin) expressed in human HepG2 cells incubated for 24 hrs by cell based analysisMore data for this Ligand-Target Pair
Ligand Info
Affinity DataEC50: 622nMAssay Description:Agonist activity at FXR-LBD (unknown origin) incubated for 3 hrs using fluorescein coactivator peptide by FRET assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataEC50: 629nMAssay Description:Agonist activity at FXR-LBD (unknown origin) expressed in human HepG2 cells incubated for 24 hrs by cell based analysisMore data for this Ligand-Target Pair
Ligand Info
Affinity DataEC50: 683nMAssay Description:Agonist activity at FXR-LBD (unknown origin) incubated for 3 hrs using fluorescein coactivator peptide by FRET assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataEC50: 762nMAssay Description:Agonist activity at FXR-LBD (unknown origin) incubated for 3 hrs using fluorescein coactivator peptide by FRET assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataEC50: 785nMAssay Description:Agonist activity at FXR-LBD (unknown origin) expressed in human HepG2 cells incubated for 24 hrs by cell based analysisMore data for this Ligand-Target Pair
Ligand Info
Affinity DataEC50: 835nMAssay Description:Agonist activity at FXR-LBD (unknown origin) incubated for 3 hrs using fluorescein coactivator peptide by FRET assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataEC50: 837nMAssay Description:Agonist activity at FXR-LBD (unknown origin) expressed in human HepG2 cells incubated for 24 hrs by cell based analysisMore data for this Ligand-Target Pair
Ligand Info
Affinity DataEC50: 853nMAssay Description:Agonist activity at FXR-LBD (unknown origin) incubated for 3 hrs using fluorescein coactivator peptide by FRET assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataEC50: 862nMAssay Description:Agonist activity at FXR-LBD (unknown origin) incubated for 3 hrs using fluorescein coactivator peptide by FRET assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataEC50: 872nMAssay Description:Agonist activity at FXR-LBD (unknown origin) incubated for 3 hrs using fluorescein coactivator peptide by FRET assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataEC50: 915nMAssay Description:Agonist activity at FXR-LBD (unknown origin) expressed in human HepG2 cells incubated for 24 hrs by cell based analysisMore data for this Ligand-Target Pair
Ligand Info
Affinity DataEC50: 947nMAssay Description:Agonist activity at FXR-LBD (unknown origin) expressed in human HepG2 cells incubated for 24 hrs by cell based analysisMore data for this Ligand-Target Pair
Ligand Info
Affinity DataEC50: 950nMAssay Description:Agonist activity at FXR-LBD (unknown origin) incubated for 3 hrs using fluorescein coactivator peptide by FRET assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataEC50: 952nMAssay Description:Agonist activity at FXR-LBD (unknown origin) expressed in human HepG2 cells incubated for 24 hrs by cell based analysisMore data for this Ligand-Target Pair
Ligand Info
Affinity DataEC50: 1.04E+3nMAssay Description:Agonist activity at FXR-LBD (unknown origin) expressed in human HepG2 cells incubated for 24 hrs by cell based analysisMore data for this Ligand-Target Pair
Ligand Info
Affinity DataEC50: 1.42E+3nMAssay Description:Agonist activity at FXR-LBD (unknown origin) incubated for 3 hrs using fluorescein coactivator peptide by FRET assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataEC50: 1.57E+3nMAssay Description:Agonist activity at FXR-LBD (unknown origin) expressed in human HepG2 cells incubated for 24 hrs by cell based analysisMore data for this Ligand-Target Pair
Ligand Info
Affinity DataEC50: 1.64E+3nMAssay Description:Agonist activity at FXR-LBD (unknown origin) expressed in human HepG2 cells incubated for 24 hrs by cell based analysisMore data for this Ligand-Target Pair
Ligand Info
Affinity DataEC50: 1.73E+3nMAssay Description:Agonist activity at FXR-LBD (unknown origin) incubated for 3 hrs using fluorescein coactivator peptide by FRET assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataEC50: 2.51E+3nMAssay Description:Agonist activity at FXR-LBD (unknown origin) incubated for 3 hrs using fluorescein coactivator peptide by FRET assayMore data for this Ligand-Target Pair
Ligand Info






























