Compile Data Set for Download or QSAR
Report error Found 17 Enz. Inhib. hit(s) with all data for entry = 50022766
TargetRelaxin-3 receptor 2(Human)
The University of Melbourne

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50654061BDBM50654061(CHEMBL6148111)
Affinity DataKi:  1.30nMAssay Description:Antagonist activity at human CCR3 assessed as inhibition of CCL11-induced calcium influx by cell based assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/3/2026
Entry Details PubMed
TargetRelaxin-3 receptor 2(Human)
The University of Melbourne

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50654060BDBM50654060(CHEMBL6148631)
Affinity DataKi:  2.30nMAssay Description:Antagonist activity at CCR9 assessed as inhibition of CCL25-induced chemotaxis by cell based assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/3/2026
Entry Details PubMed
TargetRelaxin-3 receptor 2(Human)
The University of Melbourne

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50654064BDBM50654064(CHEMBL6103355)
Affinity DataKi:  3.10nMAssay Description:Antagonist activity at histamine H1 receptor expressed in human PC3 cells inhibition of histamine-induced calcium influx by cell based assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/3/2026
Entry Details PubMed
TargetRelaxin-3 receptor 2(Human)
The University of Melbourne

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50654063BDBM50654063(CHEMBL6148405)
Affinity DataKi:  3.5nMAssay Description:Antagonist activity at CCR1 assessed as inhibition of CCL3-induced chemotaxis by cell based assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/3/2026
Entry Details PubMed
TargetRelaxin-3 receptor 2(Human)
The University of Melbourne

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50654059BDBM50654059(CHEMBL6132956)
Affinity DataKi:  4.70nMAssay Description:Agonist activity at human mGLUR2 assessed as inhibition of forskolin-stimulated cAMP production by cell-based assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/3/2026
Entry Details PubMed
TargetRelaxin-3 receptor 2(Human)
The University of Melbourne

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50654055BDBM50654055(CHEMBL6103273)
Affinity DataKi:  7.80nMAssay Description:Inhibition of ALK Tyr1604 phosphorylation by cell based assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/3/2026
Entry Details PubMed
TargetRelaxin-3 receptor 2(Human)
The University of Melbourne

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50654056BDBM50654056(CHEMBL6149303)
Affinity DataKi:  8.70nMAssay Description:Inhibition of ALK Tyr1604 phosphorylation by cell based assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/3/2026
Entry Details PubMed
TargetRelaxin-3 receptor 2(Human)
The University of Melbourne

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50654057BDBM50654057(CHEMBL6146291)
Affinity DataKi:  11nMAssay Description:Inhibition of ALK Tyr1604 phosphorylation by cell based assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/3/2026
Entry Details PubMed
TargetRelaxin-3 receptor 2(Human)
The University of Melbourne

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50654062BDBM50654062(CHEMBL6145134)
Affinity DataKi:  14nMAssay Description:Antagonist activity at CCR3 assessed as inhibition of chemotaxis by cell based assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/3/2026
Entry Details PubMed
TargetRelaxin-3 receptor 2(Human)
The University of Melbourne

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50654058BDBM50654058(CHEMBL6148324)
Affinity DataKi:  18nMAssay Description:Agonist activity at human mGLUR3 assessed as inhibition of forskolin-stimulated cAMP production by cell-based assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/3/2026
Entry Details PubMed
TargetRelaxin-3 receptor 1(Human)
The University of Melbourne

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50654059BDBM50654059(CHEMBL6132956)
Affinity DataKi:  76nMAssay Description:Inhibition of ALK Tyr1604 phosphorylation by cell based assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/3/2026
Entry Details PubMed
TargetRelaxin-3 receptor 1(Human)
The University of Melbourne

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50654055BDBM50654055(CHEMBL6103273)
Affinity DataKi:  195nMAssay Description:Inhibition of ALK Tyr1604 phosphorylation by cell based assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/3/2026
Entry Details PubMed
TargetRelaxin-3 receptor 1(Human)
The University of Melbourne

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50654056BDBM50654056(CHEMBL6149303)
Affinity DataKi:  426nMAssay Description:Inhibition of ALK Tyr1604 phosphorylation by cell based assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/3/2026
Entry Details PubMed
TargetRelaxin-3 receptor 1(Human)
The University of Melbourne

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50654058BDBM50654058(CHEMBL6148324)
Affinity DataKi:  427nMAssay Description:Inhibition of ALK Tyr1604 phosphorylation by cell based assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/3/2026
Entry Details PubMed
TargetRelaxin-3 receptor 1(Human)
The University of Melbourne

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50654057BDBM50654057(CHEMBL6146291)
Affinity DataKi:  589nMAssay Description:Inhibition of ALK Tyr1604 phosphorylation by cell based assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/3/2026
Entry Details PubMed
TargetRelaxin-3 receptor 1(Human)
The University of Melbourne

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50654060BDBM50654060(CHEMBL6148631)
Affinity DataKi:  603nMAssay Description:Inhibition of ALK Tyr1604 phosphorylation by cell based assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/3/2026
Entry Details PubMed
TargetRelaxin-3 receptor 1(Human)
The University of Melbourne

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50654061BDBM50654061(CHEMBL6148111)
Affinity DataKi:  2.19E+3nMAssay Description:Inhibition of ALK Tyr1604 phosphorylation by cell based assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/3/2026
Entry Details PubMed