Report error Found 25 Enz. Inhib. hit(s) with all data for entry = 50023028
Affinity DataIC50: 4nMAssay Description:Inhibition of recombinant CLK2 (unknown origin) incubated for 40 mins in presence of ATP by fluorescence based analysisMore data for this Ligand-Target Pair
3D Structure (crystal)
Affinity DataIC50: 4.20nMAssay Description:Inhibition of recombinant human CK2alpha extracted from Escherichia coli C41 (DE3) cellsMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1B(Human)
German University in Cairo
Curated by ChEMBL
German University in Cairo
Curated by ChEMBL
Affinity DataIC50: 6.80nMAssay Description:Inhibition of human Dyrk1BMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
German University in Cairo
Curated by ChEMBL
German University in Cairo
Curated by ChEMBL
Affinity DataIC50: 6.80nMAssay Description:Inhibition of human Dyrk1AMore data for this Ligand-Target Pair
Affinity DataIC50: 7nMAssay Description:Inhibition of CK2 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 7.30nMAssay Description:Inhibition of recombinant N-terminal his-6 tagged human CK2alpha extracted from Escherichia coli C41 (DE3) cells using H-RRRDDDSDDD-NH2 as substrate ...More data for this Ligand-Target Pair
Affinity DataIC50: 7.5nMAssay Description:Inhibition of recombinant N-terminal his-6 tagged human CK2alpha extracted from Escherichia coli C41 (DE3) cells using H-RRRDDDSDDD-NH2 as substrate ...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 16nMAssay Description:Inhibition of recombinant N-terminal his-6 tagged human CK2alpha extracted from Escherichia coli C41 (DE3) cells using H-RRRDDDSDDD-NH2 as substrate ...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 17nMAssay Description:Inhibition of recombinant N-terminal his-6 tagged human CK2alpha extracted from Escherichia coli C41 (DE3) cells using H-RRRDDDSDDD-NH2 as substrate ...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 18nMAssay Description:Inhibition of recombinant N-terminal his-6 tagged human CK2alpha extracted from Escherichia coli C41 (DE3) cells using H-RRRDDDSDDD-NH2 as substrate ...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 18nMAssay Description:Inhibition of recombinant N-terminal his-6 tagged human CK2alpha extracted from Escherichia coli C41 (DE3) cells using H-RRRDDDSDDD-NH2 as substrate ...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 20nMAssay Description:Inhibition of recombinant N-terminal his-6 tagged human CK2alpha extracted from Escherichia coli C41 (DE3) cells using H-RRRDDDSDDD-NH2 as substrate ...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 22nMAssay Description:Inhibition of recombinant N-terminal his-6 tagged human CK2alpha extracted from Escherichia coli C41 (DE3) cells using H-RRRDDDSDDD-NH2 as substrate ...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 30nMAssay Description:Inhibition of recombinant N-terminal his-6 tagged human CK2alpha extracted from Escherichia coli C41 (DE3) cells using H-RRRDDDSDDD-NH2 as substrate ...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 37nMAssay Description:Inhibition of recombinant N-terminal his-6 tagged human CK2alpha extracted from Escherichia coli C41 (DE3) cells using H-RRRDDDSDDD-NH2 as substrate ...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 39nMAssay Description:Inhibition of recombinant N-terminal his-6 tagged human CK2alpha extracted from Escherichia coli C41 (DE3) cells using H-RRRDDDSDDD-NH2 as substrate ...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 40nMAssay Description:Inhibition of CK2 (unknown origin) by radiometric assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 43nMAssay Description:Inhibition of recombinant N-terminal his-6 tagged human CK2alpha extracted from Escherichia coli C41 (DE3) cells using H-RRRDDDSDDD-NH2 as substrate ...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 100nMAssay Description:Inhibition of AKT1 phosphorylation in human HCT-116 cellsMore data for this Ligand-Target Pair
Affinity DataKd: 130nMAssay Description:Binding affinity to recombinant N-terminal his-6 tagged human CK2alpha extracted from Escherichia coli C41 (DE3) cells assessed as dissociation const...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 143nMAssay Description:Inhibition of recombinant N-terminal his-6 tagged human CK2alpha extracted from Escherichia coli C41 (DE3) cells using H-RRRDDDSDDD-NH2 as substrate ...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 150nMAssay Description:Inhibition of CK2alpha (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 440nMAssay Description:Inhibition of DRAK1 (unknown origin)More data for this Ligand-Target Pair
TargetEukaryotic translation initiation factor 2 subunit 2(Homo sapiens)
German University in Cairo
Curated by ChEMBL
German University in Cairo
Curated by ChEMBL
Affinity DataIC50: 500nMAssay Description:Inhibition of eIF2beta phosphorylation in human HCT-116 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 7.00E+3nMAssay Description:Inhibition of CK2alpha (unknown origin)More data for this Ligand-Target Pair
