Report error Found 72 Enz. Inhib. hit(s) with all data for entry = 50022677
TargetMitogen-activated protein kinase kinase kinase kinase 1(Human)
Insilico Medicine Shanghai Ltd
Curated by ChEMBL
Insilico Medicine Shanghai Ltd
Curated by ChEMBL
Affinity DataIC50: 0.440nMAssay Description:Inhibition of hypoxia-induced HIF1 activation in human T47D cells after 16 hrs by cell based luciferase assayMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase kinase 1(Human)
Insilico Medicine Shanghai Ltd
Curated by ChEMBL
Insilico Medicine Shanghai Ltd
Curated by ChEMBL
Affinity DataIC50: 0.510nMAssay Description:Antagonist activity at human PPARgamma receptor in CHO-K1 cells assessed as rosiglitazone-induced receptor activation by cell based reporter assayMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase kinase 1(Human)
Insilico Medicine Shanghai Ltd
Curated by ChEMBL
Insilico Medicine Shanghai Ltd
Curated by ChEMBL
Affinity DataIC50: 0.510nMAssay Description:Agonist activity at human PPARdelta assessed as receptor activation by cell based assayMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase kinase 1(Human)
Insilico Medicine Shanghai Ltd
Curated by ChEMBL
Insilico Medicine Shanghai Ltd
Curated by ChEMBL
Affinity DataIC50: 0.550nMAssay Description:Agonist activity at human PPARgamma assessed as receptor activation by cell based assayMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase kinase 1(Human)
Insilico Medicine Shanghai Ltd
Curated by ChEMBL
Insilico Medicine Shanghai Ltd
Curated by ChEMBL
Affinity DataIC50: 0.810nMAssay Description:Agonist activity at human PPARdelta assessed as receptor activation by cell based assayMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase kinase 1(Human)
Insilico Medicine Shanghai Ltd
Curated by ChEMBL
Insilico Medicine Shanghai Ltd
Curated by ChEMBL
Affinity DataIC50: 0.930nMAssay Description:Agonist activity at mouse PPARalpha assessed as receptor activation by cell based assayMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase kinase 1(Human)
Insilico Medicine Shanghai Ltd
Curated by ChEMBL
Insilico Medicine Shanghai Ltd
Curated by ChEMBL
Affinity DataIC50: 1nMAssay Description:Antagonist activity at human PPARgamma receptor in CHO-K1 cells assessed as rosiglitazone-induced receptor activation by cell based reporter assayMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase kinase 1(Human)
Insilico Medicine Shanghai Ltd
Curated by ChEMBL
Insilico Medicine Shanghai Ltd
Curated by ChEMBL
Affinity DataIC50: 2.40nMAssay Description:Agonist activity at human PPARdelta assessed as receptor activation by cell based assayMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase kinase 1(Human)
Insilico Medicine Shanghai Ltd
Curated by ChEMBL
Insilico Medicine Shanghai Ltd
Curated by ChEMBL
Affinity DataIC50: 2.5nMAssay Description:Antagonist activity at human PPARgamma receptor in CHO-K1 cells assessed as rosiglitazone-induced receptor activation by cell based reporter assayMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase kinase 1(Human)
Insilico Medicine Shanghai Ltd
Curated by ChEMBL
Insilico Medicine Shanghai Ltd
Curated by ChEMBL
Affinity DataIC50: 2.70nMAssay Description:Agonist activity at mouse PPARgamma assessed as receptor activation by cell based assayMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase kinase 1(Human)
Insilico Medicine Shanghai Ltd
Curated by ChEMBL
Insilico Medicine Shanghai Ltd
Curated by ChEMBL
Affinity DataIC50: 2.90nMAssay Description:Activity at human PPARalpha receptor by cell based transactivation assayMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase kinase 1(Human)
Insilico Medicine Shanghai Ltd
Curated by ChEMBL
Insilico Medicine Shanghai Ltd
Curated by ChEMBL
Affinity DataIC50: 3nMAssay Description:Inhibition of hypoxia-induced HIF1 activation in human T47D cells after 16 hrs by cell based luciferase assayMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase kinase 1(Human)
Insilico Medicine Shanghai Ltd
Curated by ChEMBL
Insilico Medicine Shanghai Ltd
Curated by ChEMBL
Affinity DataIC50: 4.40nMAssay Description:Agonist activity at mouse PPARgamma assessed as receptor activation by cell based assayMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase kinase 1(Human)
Insilico Medicine Shanghai Ltd
Curated by ChEMBL
Insilico Medicine Shanghai Ltd
Curated by ChEMBL
Affinity DataIC50: 6.5nMAssay Description:Inhibition of human 11-beta-HSD1 in presence of 3% HSA by cell based assayMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase kinase 1(Human)
Insilico Medicine Shanghai Ltd
Curated by ChEMBL
Insilico Medicine Shanghai Ltd
Curated by ChEMBL
Affinity DataIC50: 7nMAssay Description:Agonist activity at mouse PPARalpha assessed as receptor activation by cell based assayMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase kinase 1(Human)
Insilico Medicine Shanghai Ltd
Curated by ChEMBL
Insilico Medicine Shanghai Ltd
Curated by ChEMBL
Affinity DataIC50: 7.5nMAssay Description:Antagonist activity at human alpha1B adrenoceptor assessed as inhibition of norepinephrine-induced increase of intracellular calcium level by cell ba...More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase kinase 1(Human)
Insilico Medicine Shanghai Ltd
Curated by ChEMBL
Insilico Medicine Shanghai Ltd
Curated by ChEMBL
Affinity DataIC50: 12nMAssay Description:Inhibition of hypoxia-induced HIF1 activation in human T47D cells after 16 hrs by cell based luciferase assayMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase kinase 1(Human)
Insilico Medicine Shanghai Ltd
Curated by ChEMBL
Insilico Medicine Shanghai Ltd
Curated by ChEMBL
Affinity DataIC50: 14nMAssay Description:Inhibition of human 11-beta-HSD1 in presence of 3% HSA by cell based assayMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase kinase 1(Human)
Insilico Medicine Shanghai Ltd
Curated by ChEMBL
Insilico Medicine Shanghai Ltd
Curated by ChEMBL
Affinity DataIC50: 32nMAssay Description:Antagonist activity against human P2X7 receptor assessed as inhibition of IL-1beta production by cell based assayMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase kinase 1(Human)
Insilico Medicine Shanghai Ltd
Curated by ChEMBL
Insilico Medicine Shanghai Ltd
Curated by ChEMBL
Affinity DataIC50: 33nMAssay Description:Antagonist activity at human PPARgamma receptor in CHO-K1 cells assessed as rosiglitazone-induced receptor activation by cell based reporter assayMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase kinase 1(Human)
Insilico Medicine Shanghai Ltd
Curated by ChEMBL
Insilico Medicine Shanghai Ltd
Curated by ChEMBL
Affinity DataIC50: 36nMAssay Description:Inhibition of human 11-beta-HSD1 in presence of 3% HSA by cell based assayMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase kinase 1(Human)
Insilico Medicine Shanghai Ltd
Curated by ChEMBL
Insilico Medicine Shanghai Ltd
Curated by ChEMBL
Affinity DataIC50: 75nMAssay Description:Agonist activity at human PPARalpha assessed as receptor activation by cell based assayMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase kinase 3(Human)
Insilico Medicine Shanghai Ltd
Curated by ChEMBL
Insilico Medicine Shanghai Ltd
Curated by ChEMBL
Affinity DataIC50: 126nMAssay Description:Agonist activity at mouse PPARalpha assessed as receptor activation by cell based assayMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase kinase 3(Human)
Insilico Medicine Shanghai Ltd
Curated by ChEMBL
Insilico Medicine Shanghai Ltd
Curated by ChEMBL
Affinity DataIC50: 134nMAssay Description:Agonist activity at human PPARalpha assessed as receptor activation by cell based assayMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase kinase 3(Human)
Insilico Medicine Shanghai Ltd
Curated by ChEMBL
Insilico Medicine Shanghai Ltd
Curated by ChEMBL
Affinity DataIC50: 141nMAssay Description:Agonist activity at mouse PPARalpha assessed as receptor activation by cell based assayMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase kinase 5(Homo sapiens)
Insilico Medicine Shanghai Ltd
Curated by ChEMBL
Insilico Medicine Shanghai Ltd
Curated by ChEMBL
Affinity DataIC50: 183nMAssay Description:Agonist activity at mouse PPARalpha assessed as receptor activation by cell based assayMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase kinase 3(Human)
Insilico Medicine Shanghai Ltd
Curated by ChEMBL
Insilico Medicine Shanghai Ltd
Curated by ChEMBL
Affinity DataIC50: 196nMAssay Description:Agonist activity at human PPARgamma assessed as receptor activation by cell based assayMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase kinase 3(Human)
Insilico Medicine Shanghai Ltd
Curated by ChEMBL
Insilico Medicine Shanghai Ltd
Curated by ChEMBL
Affinity DataIC50: 214nMAssay Description:Agonist activity at mouse PPARalpha assessed as receptor activation by cell based assayMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase kinase 3(Human)
Insilico Medicine Shanghai Ltd
Curated by ChEMBL
Insilico Medicine Shanghai Ltd
Curated by ChEMBL
Affinity DataIC50: 224nMAssay Description:Agonist activity at human PPARgamma assessed as receptor activation by cell based assayMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase kinase 3(Human)
Insilico Medicine Shanghai Ltd
Curated by ChEMBL
Insilico Medicine Shanghai Ltd
Curated by ChEMBL
Affinity DataIC50: 227nMAssay Description:Agonist activity at mouse PPARalpha assessed as receptor activation by cell based assayMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase kinase 3(Human)
Insilico Medicine Shanghai Ltd
Curated by ChEMBL
Insilico Medicine Shanghai Ltd
Curated by ChEMBL
Affinity DataIC50: 228nMAssay Description:Agonist activity at human PPARalpha assessed as receptor activation by cell based assayMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase kinase 3(Human)
Insilico Medicine Shanghai Ltd
Curated by ChEMBL
Insilico Medicine Shanghai Ltd
Curated by ChEMBL
Affinity DataIC50: 260nMAssay Description:Agonist activity at human PPARalpha assessed as receptor activation by cell based assayMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase kinase 3(Human)
Insilico Medicine Shanghai Ltd
Curated by ChEMBL
Insilico Medicine Shanghai Ltd
Curated by ChEMBL
Affinity DataIC50: 279nMAssay Description:Agonist activity at mouse PPARalpha assessed as receptor activation by cell based assayMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase kinase 3(Human)
Insilico Medicine Shanghai Ltd
Curated by ChEMBL
Insilico Medicine Shanghai Ltd
Curated by ChEMBL
Affinity DataIC50: 279nMAssay Description:Agonist activity at human PPARalpha assessed as receptor activation by cell based assayMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase kinase 5(Homo sapiens)
Insilico Medicine Shanghai Ltd
Curated by ChEMBL
Insilico Medicine Shanghai Ltd
Curated by ChEMBL
Affinity DataIC50: 304nMAssay Description:Agonist activity at human PPARalpha assessed as receptor activation by cell based assayMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase kinase 3(Human)
Insilico Medicine Shanghai Ltd
Curated by ChEMBL
Insilico Medicine Shanghai Ltd
Curated by ChEMBL
Affinity DataIC50: 331nMAssay Description:Agonist activity at mouse PPARgamma assessed as receptor activation by cell based assayMore data for this Ligand-Target Pair
Affinity DataIC50: 350nMAssay Description:Agonist activity at human PPARalpha assessed as receptor activation by cell based assayMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase kinase 3(Human)
Insilico Medicine Shanghai Ltd
Curated by ChEMBL
Insilico Medicine Shanghai Ltd
Curated by ChEMBL
Affinity DataIC50: 360nMAssay Description:Agonist activity at human PPARdelta assessed as receptor activation by cell based assayMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase kinase 3(Human)
Insilico Medicine Shanghai Ltd
Curated by ChEMBL
Insilico Medicine Shanghai Ltd
Curated by ChEMBL
Affinity DataIC50: 388nMAssay Description:Agonist activity at mouse PPARgamma assessed as receptor activation by cell based assayMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase kinase 3(Human)
Insilico Medicine Shanghai Ltd
Curated by ChEMBL
Insilico Medicine Shanghai Ltd
Curated by ChEMBL
Affinity DataIC50: 407nMAssay Description:Agonist activity at human PPARgamma assessed as receptor activation by cell based assayMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase kinase 3(Human)
Insilico Medicine Shanghai Ltd
Curated by ChEMBL
Insilico Medicine Shanghai Ltd
Curated by ChEMBL
Affinity DataIC50: 504nMAssay Description:Agonist activity at human PPARalpha assessed as receptor activation by cell based assayMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase kinase 3(Human)
Insilico Medicine Shanghai Ltd
Curated by ChEMBL
Insilico Medicine Shanghai Ltd
Curated by ChEMBL
Affinity DataIC50: 553nMAssay Description:Agonist activity at human PPARgamma assessed as receptor activation by cell based assayMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase kinase 3(Human)
Insilico Medicine Shanghai Ltd
Curated by ChEMBL
Insilico Medicine Shanghai Ltd
Curated by ChEMBL
Affinity DataIC50: 870nMAssay Description:Agonist activity at mouse PPARalpha assessed as receptor activation by cell based assayMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase kinase 2(Human)
Insilico Medicine Shanghai Ltd
Curated by ChEMBL
Insilico Medicine Shanghai Ltd
Curated by ChEMBL
Affinity DataIC50: 1.00E+3nMAssay Description:Agonist activity at mouse PPARalpha assessed as receptor activation by cell based assayMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase kinase 2(Human)
Insilico Medicine Shanghai Ltd
Curated by ChEMBL
Insilico Medicine Shanghai Ltd
Curated by ChEMBL
Affinity DataIC50: 1.00E+3nMAssay Description:Agonist activity at human PPARgamma assessed as receptor activation by cell based assayMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase kinase 4(Human)
Insilico Medicine Shanghai Ltd
Curated by ChEMBL
Insilico Medicine Shanghai Ltd
Curated by ChEMBL
Affinity DataIC50: 1.00E+3nMAssay Description:Agonist activity at mouse PPARdelta assessed as receptor activation by cell based assayMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase kinase 4(Human)
Insilico Medicine Shanghai Ltd
Curated by ChEMBL
Insilico Medicine Shanghai Ltd
Curated by ChEMBL
Affinity DataIC50: 1.00E+3nMAssay Description:Agonist activity at mouse PPARalpha assessed as receptor activation by cell based assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+3nMAssay Description:Agonist activity at human PPARdelta assessed as receptor activation by cell based assayMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 7(Human)
Insilico Medicine Shanghai Ltd
Curated by ChEMBL
Insilico Medicine Shanghai Ltd
Curated by ChEMBL
Affinity DataIC50: 1.00E+3nMAssay Description:Agonist activity at mouse PPARalpha assessed as receptor activation by cell based assayMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 7(Human)
Insilico Medicine Shanghai Ltd
Curated by ChEMBL
Insilico Medicine Shanghai Ltd
Curated by ChEMBL
Affinity DataIC50: 1.00E+3nMAssay Description:Agonist activity at mouse PPARalpha assessed as receptor activation by cell based assayMore data for this Ligand-Target Pair





















