Compile Data Set for Download or QSAR
Report error Found 36 Enz. Inhib. hit(s) with all data for entry = 50022860
TargetReplicase polyprotein 1ab(2019-nCoV)
Shandong University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50655233BDBM50655233(CHEMBL6091834)
Affinity DataIC50: 150nMAssay Description:Agonist activity at OX1R (unknown origin) expressed in CHO cells by cell-based calcium assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetReplicase polyprotein 1ab(2019-nCoV)
Shandong University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50655241BDBM50655241(CHEMBL6149659)
Affinity DataIC50: 200nMAssay Description:Agonist activity at OX2R (unknown origin) expressed in CHO cells by cell-based calcium assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetReplicase polyprotein 1ab(2019-nCoV)
Shandong University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50655242BDBM50655242(CHEMBL6134130)
Affinity DataIC50: 220nMAssay Description:Agonist activity at OX2R (unknown origin) expressed in CHO cells by cell-based calcium assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetReplicase polyprotein 1ab(2019-nCoV)
Shandong University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50655230BDBM50655230(CHEMBL6159892)
Affinity DataIC50: 250nMAssay Description:Agonist activity at OX1R (unknown origin) expressed in CHO cells by cell-based calcium assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetReplicase polyprotein 1ab(2019-nCoV)
Shandong University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50655221BDBM50655221(CHEMBL6102335)
Affinity DataIC50: 250nMAssay Description:Modulation of mouse Utrophin in mouse myoblast expressing LUmdx assessed as upregulation of utrophin mRNA expression incubated for 24 hrs by cell-bas...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetReplicase polyprotein 1ab(2019-nCoV)
Shandong University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50655225BDBM50655225(CHEMBL6146049)
Affinity DataIC50: 250nMAssay Description:Modulation of mouse Utrophin in mouse myoblast expressing LUmdx assessed as upregulation of utrophin mRNA expression incubated for 24 hrs by cell-bas...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetReplicase polyprotein 1ab(2019-nCoV)
Shandong University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50655222BDBM50655222(CHEMBL6152614)
Affinity DataIC50: 300nMAssay Description:Modulation of mouse Utrophin in mouse myoblast expressing LUmdx assessed as upregulation of utrophin mRNA expression incubated for 24 hrs by cell-bas...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetReplicase polyprotein 1ab(2019-nCoV)
Shandong University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50655226BDBM50655226(CHEMBL6143389)
Affinity DataIC50: 300nMAssay Description:Modulation of mouse Utrophin in mouse myoblast expressing LUmdx assessed as upregulation of utrophin mRNA expression incubated for 24 hrs by cell-bas...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetReplicase polyprotein 1ab(2019-nCoV)
Shandong University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50655231BDBM50655231(CHEMBL6160622)
Affinity DataIC50: 320nMAssay Description:Agonist activity at OX1R (unknown origin) expressed in CHO cells by cell-based calcium assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetReplicase polyprotein 1ab(2019-nCoV)
Shandong University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50655245BDBM50655245(CHEMBL6151899)
Affinity DataIC50: 370nMAssay Description:Agonist activity at OX2R (unknown origin) expressed in CHO cells by cell-based calcium assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetReplicase polyprotein 1ab(2019-nCoV)
Shandong University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50655243BDBM50655243(CHEMBL6149893)
Affinity DataIC50: 390nMAssay Description:Agonist activity at OX2R (unknown origin) expressed in CHO cells by cell-based calcium assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetReplicase polyprotein 1ab(2019-nCoV)
Shandong University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50655232BDBM50655232(CHEMBL6141704)
Affinity DataIC50: 440nMAssay Description:Agonist activity at OX1R (unknown origin) expressed in CHO cells by cell-based calcium assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetReplicase polyprotein 1ab(2019-nCoV)
Shandong University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50655224BDBM50655224(CHEMBL6120712)
Affinity DataIC50: 460nMAssay Description:Modulation of mouse Utrophin in mouse myoblast expressing LUmdx assessed as upregulation of utrophin mRNA expression incubated for 24 hrs by cell-bas...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetReplicase polyprotein 1ab(2019-nCoV)
Shandong University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50655220BDBM50655220(CHEMBL6142386)
Affinity DataIC50: 500nMAssay Description:Modulation of mouse Utrophin in mouse myoblast expressing LUmdx assessed as upregulation of utrophin mRNA expression incubated for 24 hrs by cell-bas...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetReplicase polyprotein 1ab(2019-nCoV)
Shandong University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50655240BDBM50655240(CHEMBL6149649)
Affinity DataIC50: 510nMAssay Description:Agonist activity at OX2R (unknown origin) expressed in CHO cells by cell-based calcium assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetReplicase polyprotein 1ab(2019-nCoV)
Shandong University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50655246BDBM50655246(CHEMBL6142616)
Affinity DataIC50: 610nMAssay Description:Agonist activity at OX2R (unknown origin) expressed in CHO cells by cell-based calcium assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetReplicase polyprotein 1ab(2019-nCoV)
Shandong University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50655220BDBM50655220(CHEMBL6142386)
Affinity DataKd:  1.12E+3nMAssay Description:Agonist activity at OX2R (unknown origin) expressed in CHO cells by cell-based calcium assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetReplicase polyprotein 1ab(2019-nCoV)
Shandong University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50655229BDBM50655229(CHEMBL6151475)
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of gamma-secretase (unknown origin) assessed as inhibition of Amyloid beta 40 production by cell-based assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetReplicase polyprotein 1ab(2019-nCoV)
Shandong University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50655228BDBM50655228(CHEMBL6148184)
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of SYK (unknown origin) assessed as reduction of IgM-stimulated ERK phosphorylation by Cell-based assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetReplicase polyprotein 1ab(2019-nCoV)
Shandong University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50655227BDBM50655227(CHEMBL6144326)
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of SYK (unknown origin) assessed as reduction of IgM-stimulated ERK phosphorylation by Cell-based assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetReplicase polyprotein 1ab(2019-nCoV)
Shandong University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50655223BDBM50655223(CHEMBL6120738)
Affinity DataIC50: 1.45E+3nMAssay Description:Modulation of mouse Utrophin in mouse myoblast expressing LUmdx assessed as upregulation of utrophin mRNA expression incubated for 24 hrs by cell-bas...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetReplicase polyprotein 1ab(2019-nCoV)
Shandong University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50655237BDBM50655237(CHEMBL6103523)
Affinity DataIC50: 1.65E+3nMAssay Description:Agonist activity at OX1R (unknown origin) expressed in CHO cells by cell-based calcium assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetReplicase polyprotein 1ab(2019-nCoV)
Shandong University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50655247BDBM50655247(CHEMBL6144059)
Affinity DataIC50: 1.93E+3nMAssay Description:Agonist activity at OX2R (unknown origin) expressed in CHO cells by cell-based calcium assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetReplicase polyprotein 1ab(2019-nCoV)
Shandong University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50655221BDBM50655221(CHEMBL6102335)
Affinity DataKd:  2.54E+3nMAssay Description:Agonist activity at OX2R (unknown origin) expressed in CHO cells by cell-based calcium assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetReplicase polyprotein 1ab(2019-nCoV)
Shandong University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50655226BDBM50655226(CHEMBL6143389)
Affinity DataKd:  2.75E+3nMAssay Description:Antagonist activity at OX1R (unknown origin) by cell-based calcium assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetReplicase polyprotein 1ab(2019-nCoV)
Shandong University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50655224BDBM50655224(CHEMBL6120712)
Affinity DataKd:  2.78E+3nMAssay Description:Antagonist activity at OX1R (unknown origin) by cell-based calcium assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetReplicase polyprotein 1ab(2019-nCoV)
Shandong University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50655223BDBM50655223(CHEMBL6120738)
Affinity DataKd:  4.00E+3nMAssay Description:Antagonist activity at OX1R (unknown origin) by cell-based calcium assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetReplicase polyprotein 1ab(2019-nCoV)
Shandong University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50655235BDBM50655235(CHEMBL6141894)
Affinity DataIC50: 4.51E+3nMAssay Description:Agonist activity at OX1R (unknown origin) expressed in CHO cells by cell-based calcium assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetReplicase polyprotein 1ab(2019-nCoV)
Shandong University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50655225BDBM50655225(CHEMBL6146049)
Affinity DataKd:  4.80E+3nMAssay Description:Antagonist activity at OX1R (unknown origin) by cell-based calcium assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetReplicase polyprotein 1ab(2019-nCoV)
Shandong University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50655244BDBM50655244(CHEMBL6120795)
Affinity DataIC50: 5.78E+3nMAssay Description:Agonist activity at OX2R (unknown origin) expressed in CHO cells by cell-based calcium assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetReplicase polyprotein 1ab(2019-nCoV)
Shandong University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50655222BDBM50655222(CHEMBL6152614)
Affinity DataKd:  6.73E+3nMAssay Description:Antagonist activity at OX1R (unknown origin) by cell-based calcium assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetReplicase polyprotein 1ab(2019-nCoV)
Shandong University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50655236BDBM50655236(CHEMBL6149207)
Affinity DataIC50: 1.00E+4nMAssay Description:Agonist activity at OX1R (unknown origin) expressed in CHO cells by cell-based calcium assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetReplicase polyprotein 1ab(2019-nCoV)
Shandong University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50655238BDBM50655238(CHEMBL6146599)
Affinity DataIC50: 1.00E+4nMAssay Description:Agonist activity at OX1R (unknown origin) expressed in CHO cells by cell-based calcium assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetReplicase polyprotein 1ab(2019-nCoV)
Shandong University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50655239BDBM50655239(CHEMBL6142315)
Affinity DataIC50: 1.00E+4nMAssay Description:Agonist activity at OX1R (unknown origin) expressed in CHO cells by cell-based calcium assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetReplicase polyprotein 1ab(2019-nCoV)
Shandong University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50655234BDBM50655234(CHEMBL6150906)
Affinity DataIC50: 1.66E+4nMAssay Description:Agonist activity at OX1R (unknown origin) expressed in CHO cells by cell-based calcium assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetReplicase polyprotein 1ab(2019-nCoV)
Shandong University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50655219BDBM50655219(CHEMBL6120582)
Affinity DataIC50: 1.00E+5nMAssay Description:Modulation of mouse Utrophin in mouse myoblast expressing LUmdx assessed as upregulation of utrophin mRNA expression incubated for 24 hrs by cell-bas...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed