Compile Data Set for Download or QSAR
Report error Found 12 Enz. Inhib. hit(s) with all data for entry = 50022856
TargetAP2-associated protein kinase 1(Human)
Humanwell Healthcare (Group) Co., Ltd.

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50655180BDBM50655180(CHEMBL6147194)
Affinity DataIC50: 3.90nMAssay Description:Inhibition of TRKC (unknown origin) incubated for 60 mins and measured after 3 hrs by cell-based functional kinase assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetAP2-associated protein kinase 1(Human)
Humanwell Healthcare (Group) Co., Ltd.

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50655181BDBM50655181(CHEMBL6133691)
Affinity DataIC50: 4.20nMAssay Description:Antagonist activity at human P2X3 receptor by cell based assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetAP2-associated protein kinase 1(Human)
Humanwell Healthcare (Group) Co., Ltd.

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 311267BDBM311267(US10155760, Example 123 | (S)-1-((2′,6-bis(d...)
Affinity DataIC50: 5nMAssay Description:Agonist activity at human wild type full length STING expressed in 293T cells incubated for 7 hrs by luciferase/cell based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetAP2-associated protein kinase 1(Human)
Humanwell Healthcare (Group) Co., Ltd.

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50655184BDBM50655184(CHEMBL6162022)
Affinity DataIC50: 5.40nMAssay Description:Antagonist activity at human P2X3 receptor by cell based assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetAP2-associated protein kinase 1(Human)
Humanwell Healthcare (Group) Co., Ltd.

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50655189BDBM50655189(CHEMBL6160425)
Affinity DataIC50: 8nMAssay Description:Antagonist activity at human P2X3 receptor by cell based assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetAP2-associated protein kinase 1(Human)
Humanwell Healthcare (Group) Co., Ltd.

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50655183BDBM50655183(CHEMBL6102731)
Affinity DataIC50: 20nMAssay Description:Antagonist activity at human P2X3 receptor by cell based assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetAP2-associated protein kinase 1(Human)
Humanwell Healthcare (Group) Co., Ltd.

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50655186BDBM50655186(CHEMBL6148814)
Affinity DataIC50: 20nMAssay Description:Antagonist activity at human P2X3 receptor by cell based assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetAP2-associated protein kinase 1(Human)
Humanwell Healthcare (Group) Co., Ltd.

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50655185BDBM50655185(CHEMBL6120771)
Affinity DataIC50: 20nMAssay Description:Antagonist activity at human P2X3 receptor by cell based assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetAP2-associated protein kinase 1(Human)
Humanwell Healthcare (Group) Co., Ltd.

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50655188BDBM50655188(CHEMBL6151499)
Affinity DataIC50: 20nMAssay Description:Antagonist activity at human P2X3 receptor by cell based assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetAP2-associated protein kinase 1(Human)
Humanwell Healthcare (Group) Co., Ltd.

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50655187BDBM50655187(CHEMBL6149927)
Affinity DataIC50: 20nMAssay Description:Antagonist activity at human P2X3 receptor by cell based assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetAP2-associated protein kinase 1(Human)
Humanwell Healthcare (Group) Co., Ltd.

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50655190BDBM50655190(CHEMBL6149025)
Affinity DataIC50: 20nMAssay Description:Antagonist activity at human P2X3 receptor by cell based assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetAP2-associated protein kinase 1(Human)
Humanwell Healthcare (Group) Co., Ltd.

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50655182BDBM50655182(CHEMBL6150625)
Affinity DataIC50: 50nMAssay Description:Antagonist activity at human P2X3 receptor by cell based assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed