Compile Data Set for Download or QSAR
Report error Found 50 Enz. Inhib. hit(s) with all data for entry = 50022758
TargetAryl hydrocarbon receptor(Human)
Palacky University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50434122BDBM50434122(CHEMBL1232568)
Affinity DataEC50:  140nMAssay Description:Inhibition of mouse SGLT2-mediated [14C]alpha-methylglucopyranoside uptake by cell based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2026
Entry Details PubMed
TargetAryl hydrocarbon receptor(Human)
Palacky University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50653960BDBM50653960(CHEMBL6147011)
Affinity DataEC50:  400nMAssay Description:Inhibition of VEGFR2 in human U251 cells by phosphotyrosine cell-based ELISAMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/3/2026
Entry Details PubMed
TargetAryl hydrocarbon receptor(Human)
Palacky University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50653963BDBM50653963(CHEMBL3414692)
Affinity DataEC50:  1.14E+3nMAssay Description:Inhibition of PDGFRbeta in human SF539 cells by phosphotyrosine cell-based ELISAMore data for this Ligand-Target Pair
Ligand InfoPDB
In Depth
Date in BDB:
6/3/2026
Entry Details PubMed
TargetAryl hydrocarbon receptor(Human)
Palacky University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50653964BDBM50653964(CHEMBL6109019)
Affinity DataEC50:  1.50E+3nMAssay Description:Inhibition of Flt3 activity in human MV 3:11 cells by phosphotyrosine cell-based ELISAMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/3/2026
Entry Details PubMed
TargetAryl hydrocarbon receptor(Human)
Palacky University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50434121BDBM50434121(CHEMBL2381492)
Affinity DataEC50:  2.50E+3nMAssay Description:Inhibition of mouse SGLT2-mediated [14C]alpha-methylglucopyranoside uptake by cell based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2026
Entry Details PubMed
TargetAryl hydrocarbon receptor(Human)
Palacky University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50653958BDBM50653958(CHEMBL6120838)
Affinity DataEC50:  2.80E+3nMAssay Description:Inhibition of mouse SGLT2-mediated [14C]alpha-methylglucopyranoside uptake by cell based assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/3/2026
Entry Details PubMed
TargetAryl hydrocarbon receptor(Human)
Palacky University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50653957BDBM50653957(CHEMBL6132645)
Affinity DataEC50:  3.40E+3nMAssay Description:Inhibition of mouse SGLT2-mediated [14C]alpha-methylglucopyranoside uptake by cell based assayMore data for this Ligand-Target Pair
Ligand InfoPDB
In Depth
Date in BDB:
6/3/2026
Entry Details PubMed
TargetAryl hydrocarbon receptor(Mouse)
Palacky University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50434122BDBM50434122(CHEMBL1232568)
Affinity DataKi:  3.70E+3nMAssay Description:Inhibition of HCV NS5A Y93H mutant in HCV genotype 1a assessed as reduction in viral replication by cell based replicon assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2026
Entry Details PubMed
TargetAryl hydrocarbon receptor(Human)
Palacky University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50434114BDBM50434114(CHEMBL511085)
Affinity DataEC50:  4.30E+3nMAssay Description:Inhibition of Flt3 activity in human MV 3:11 cells by phosphotyrosine cell-based ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2026
Entry Details PubMed
TargetAryl hydrocarbon receptor(Human)
Palacky University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50358748BDBM50358748(CHEMBL1922275)
Affinity DataEC50:  4.70E+3nMAssay Description:Inhibition of VEGFR2 in human U251 cells by phosphotyrosine cell-based ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2026
Entry Details PubMed
TargetAryl hydrocarbon receptor(Human)
Palacky University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50434120BDBM50434120(OXINDOLE)
Affinity DataEC50:  5.20E+3nMAssay Description:Inhibition of mouse SGLT2-mediated [14C]alpha-methylglucopyranoside uptake by cell based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2026
Entry Details PubMed
TargetAryl hydrocarbon receptor(Human)
Palacky University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50434117BDBM50434117(CHEMBL2381488)
Affinity DataEC50:  5.60E+3nMAssay Description:Inhibition of mouse SGLT2-mediated [14C]alpha-methylglucopyranoside uptake by cell based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2026
Entry Details PubMed
TargetAryl hydrocarbon receptor(Human)
Palacky University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50358747BDBM50358747(CHEMBL325917)
Affinity DataEC50:  6.70E+3nMAssay Description:Inhibition of VEGFR1 in human A498 cells by phosphotyrosine cell-based ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2026
Entry Details PubMed
TargetAryl hydrocarbon receptor(Mouse)
Palacky University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50434122BDBM50434122(CHEMBL1232568)
Affinity DataIC50: 7.40E+3nMAssay Description:Inhibition of HCV NS5A L31V mutant in HCV genotype 1a assessed as reduction in viral replication by cell based replicon assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2026
Entry Details PubMed
TargetAryl hydrocarbon receptor(Human)
Palacky University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50653961BDBM50653961(CHEMBL6150516)
Affinity DataEC50:  7.90E+3nMAssay Description:Inhibition of VEGFR1 in human A498 cells by phosphotyrosine cell-based ELISAMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/3/2026
Entry Details PubMed
TargetAryl hydrocarbon receptor(Mouse)
Palacky University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50653958BDBM50653958(CHEMBL6120838)
Affinity DataKi:  9.10E+3nMAssay Description:Inhibition of HCV NS5A Y93C mutant in HCV genotype 1a assessed as reduction in viral replication by cell based replicon assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/3/2026
Entry Details PubMed
TargetAryl hydrocarbon receptor(Mouse)
Palacky University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50653964BDBM50653964(CHEMBL6109019)
Affinity DataKi:  9.10E+3nMAssay Description:Inhibition of HCV NS5A L31V mutant in HCV genotype 1b assessed as reduction in viral replication by cell based replicon assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/3/2026
Entry Details PubMed
TargetAryl hydrocarbon receptor(Mouse)
Palacky University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50653960BDBM50653960(CHEMBL6147011)
Affinity DataKi:  1.10E+4nMAssay Description:Inhibition of HCV NS5A Y93H mutant in HCV genotype 1a assessed as reduction in viral replication by cell based replicon assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/3/2026
Entry Details PubMed
TargetAryl hydrocarbon receptor(Human)
Palacky University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50094702BDBM50094702(CHEMBL15844 | indole | Indole, 7 | Indol | 1H-indo...)
Affinity DataEC50:  1.11E+4nMAssay Description:Inhibition of mouse SGLT2-mediated [14C]alpha-methylglucopyranoside uptake by cell based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2026
Entry Details PubMed
TargetAryl hydrocarbon receptor(Human)
Palacky University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50653957BDBM50653957(CHEMBL6132645)
Affinity DataEC50:  1.24E+4nMAssay Description:Inhibition of human c-Met in human GTL16 cells by cell-based assayMore data for this Ligand-Target Pair
Ligand InfoPDB
In Depth
Date in BDB:
6/3/2026
Entry Details PubMed
TargetAryl hydrocarbon receptor(Human)
Palacky University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50653962BDBM50653962(CHEMBL111579)
Affinity DataEC50:  1.39E+4nMAssay Description:Inhibition of EGFR in human A431 cells by phosphotyrosine cell-based ELISAMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/3/2026
Entry Details PubMed
TargetAryl hydrocarbon receptor(Human)
Palacky University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50653956BDBM50653956(CHEMBL6148002)
Affinity DataEC50:  1.63E+4nMAssay Description:Inhibition of mouse SGLT2-mediated [14C]alpha-methylglucopyranoside uptake by cell based assayMore data for this Ligand-Target Pair
Ligand InfoPDB
In Depth
Date in BDB:
6/3/2026
Entry Details PubMed
TargetAryl hydrocarbon receptor(Human)
Palacky University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50653964BDBM50653964(CHEMBL6109019)
Affinity DataEC50:  1.81E+4nMAssay Description:Inhibition of human c-Met in human GTL16 cells by cell-based assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/3/2026
Entry Details PubMed
TargetAryl hydrocarbon receptor(Mouse)
Palacky University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50653958BDBM50653958(CHEMBL6120838)
Affinity DataIC50: 1.82E+4nMAssay Description:Inhibition of human c-Met in human GTL16 cells by cell-based assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/3/2026
Entry Details PubMed
TargetAryl hydrocarbon receptor(Mouse)
Palacky University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50653964BDBM50653964(CHEMBL6109019)
Affinity DataIC50: 1.83E+4nMAssay Description:Inhibition of HCV NS5A Y93C mutant in HCV genotype 1a assessed as reduction in viral replication by cell based replicon assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/3/2026
Entry Details PubMed
TargetAryl hydrocarbon receptor(Human)
Palacky University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50434118BDBM50434118(CHEMBL2381491)
Affinity DataEC50:  1.83E+4nMAssay Description:Inhibition of mouse SGLT2-mediated [14C]alpha-methylglucopyranoside uptake by cell based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2026
Entry Details PubMed
TargetAryl hydrocarbon receptor(Human)
Palacky University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50434121BDBM50434121(CHEMBL2381492)
Affinity DataEC50:  1.86E+4nMAssay Description:Inhibition of human c-Met in human GTL16 cells by cell-based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2026
Entry Details PubMed
TargetAryl hydrocarbon receptor(Human)
Palacky University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50294170BDBM50294170(5-fluoro-1H-indole | CHEMBL555457)
Affinity DataEC50:  1.87E+4nMAssay Description:Inhibition of mouse SGLT2-mediated [14C]alpha-methylglucopyranoside uptake by cell based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2026
Entry Details PubMed
TargetAryl hydrocarbon receptor(Human)
Palacky University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50434118BDBM50434118(CHEMBL2381491)
Affinity DataEC50:  1.96E+4nMAssay Description:Inhibition of PDGFRbeta in human SF539 cells by phosphotyrosine cell-based ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2026
Entry Details PubMed
TargetAryl hydrocarbon receptor(Mouse)
Palacky University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50653963BDBM50653963(CHEMBL3414692)
Affinity DataKi:  2.17E+4nMAssay Description:Inhibition of HCV NS5A Y93H mutant in HCV genotype 1a assessed as reduction in viral replication by cell based replicon assayMore data for this Ligand-Target Pair
Ligand InfoPDB
In Depth
Date in BDB:
6/3/2026
Entry Details PubMed
TargetAryl hydrocarbon receptor(Mouse)
Palacky University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50653960BDBM50653960(CHEMBL6147011)
Affinity DataIC50: 2.21E+4nMAssay Description:Inhibition of HCV NS5A Y93H mutant in HCV genotype 1b assessed as reduction in viral replication by cell based replicon assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/3/2026
Entry Details PubMed
TargetAryl hydrocarbon receptor(Human)
Palacky University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50294169BDBM50294169(5-chloro-1H-indole | CHEMBL555013)
Affinity DataEC50:  2.41E+4nMAssay Description:Inhibition of PDGFRbeta in human SF539 cells by phosphotyrosine cell-based ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2026
Entry Details PubMed
TargetAryl hydrocarbon receptor(Human)
Palacky University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50434122BDBM50434122(CHEMBL1232568)
Affinity DataEC50:  2.51E+4nMAssay Description:Inhibition of Flt3 activity in human MV 3:11 cells by phosphotyrosine cell-based ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2026
Entry Details PubMed
TargetAryl hydrocarbon receptor(Human)
Palacky University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50653963BDBM50653963(CHEMBL3414692)
Affinity DataEC50:  4.01E+4nMAssay Description:Inhibition of human c-Met in human GTL16 cells by cell-based assayMore data for this Ligand-Target Pair
Ligand InfoPDB
In Depth
Date in BDB:
6/3/2026
Entry Details PubMed
TargetAryl hydrocarbon receptor(Human)
Palacky University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50094702BDBM50094702(CHEMBL15844 | indole | Indole, 7 | Indol | 1H-indo...)
Affinity DataEC50:  4.31E+4nMAssay Description:Inhibition of human c-Met in human GTL16 cells by cell-based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2026
Entry Details PubMed
TargetAryl hydrocarbon receptor(Mouse)
Palacky University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50653963BDBM50653963(CHEMBL3414692)
Affinity DataIC50: 4.34E+4nMAssay Description:Inhibition of HCV NS5A Y93C mutant in HCV genotype 1a assessed as reduction in viral replication by cell based replicon assayMore data for this Ligand-Target Pair
Ligand InfoPDB
In Depth
Date in BDB:
6/3/2026
Entry Details PubMed
TargetAryl hydrocarbon receptor(Human)
Palacky University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50653958BDBM50653958(CHEMBL6120838)
Affinity DataEC50:  4.37E+4nMAssay Description:Inhibition of human c-Met in human GTL16 cells by cell-based assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/3/2026
Entry Details PubMed
TargetAryl hydrocarbon receptor(Human)
Palacky University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50434117BDBM50434117(CHEMBL2381488)
Affinity DataEC50:  5.29E+4nMAssay Description:Inhibition of EGFR in human A431 cells by phosphotyrosine cell-based ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2026
Entry Details PubMed
TargetAryl hydrocarbon receptor(Human)
Palacky University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50653962BDBM50653962(CHEMBL111579)
Affinity DataEC50:  5.62E+4nMAssay Description:Inhibition of human c-Met in human GTL16 cells by cell-based assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/3/2026
Entry Details PubMed
TargetAryl hydrocarbon receptor(Human)
Palacky University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50653960BDBM50653960(CHEMBL6147011)
Affinity DataEC50:  5.68E+4nMAssay Description:Inhibition of human c-Met in human GTL16 cells by cell-based assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/3/2026
Entry Details PubMed
TargetAryl hydrocarbon receptor(Human)
Palacky University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50358747BDBM50358747(CHEMBL325917)
Affinity DataEC50:  5.81E+4nMAssay Description:Inhibition of human c-Met in human GTL16 cells by cell-based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2026
Entry Details PubMed
TargetAryl hydrocarbon receptor(Human)
Palacky University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50653959BDBM50653959(CHEMBL107324)
Affinity DataEC50:  6.96E+4nMAssay Description:Inhibition of EGFR in human A431 cells by phosphotyrosine cell-based ELISAMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/3/2026
Entry Details PubMed
TargetAryl hydrocarbon receptor(Human)
Palacky University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50653956BDBM50653956(CHEMBL6148002)
Affinity DataEC50:  7.10E+4nMAssay Description:Inhibition of VEGFR1 in human A498 cells by phosphotyrosine cell-based ELISAMore data for this Ligand-Target Pair
Ligand InfoPDB
In Depth
Date in BDB:
6/3/2026
Entry Details PubMed
TargetAryl hydrocarbon receptor(Human)
Palacky University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50294170BDBM50294170(5-fluoro-1H-indole | CHEMBL555457)
Affinity DataEC50:  7.45E+4nMAssay Description:Inhibition of human c-Met in human GTL16 cells by cell-based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2026
Entry Details PubMed
TargetAryl hydrocarbon receptor(Human)
Palacky University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50294169BDBM50294169(5-chloro-1H-indole | CHEMBL555013)
Affinity DataEC50:  7.72E+4nMAssay Description:Inhibition of human c-Met in human GTL16 cells by cell-based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2026
Entry Details PubMed
TargetAryl hydrocarbon receptor(Human)
Palacky University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50434114BDBM50434114(CHEMBL511085)
Affinity DataEC50:  8.06E+4nMAssay Description:Inhibition of human c-Met in human GTL16 cells by cell-based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2026
Entry Details PubMed
TargetAryl hydrocarbon receptor(Human)
Palacky University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50434120BDBM50434120(OXINDOLE)
Affinity DataEC50:  8.09E+4nMAssay Description:Inhibition of VEGFR2 in human U251 cells by phosphotyrosine cell-based ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2026
Entry Details PubMed
TargetAryl hydrocarbon receptor(Mouse)
Palacky University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50653957BDBM50653957(CHEMBL6132645)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of HCV NS5A L31V mutant in HCV genotype 1a assessed as reduction in viral replication by cell based replicon assayMore data for this Ligand-Target Pair
Ligand InfoPDB
In Depth
Date in BDB:
6/3/2026
Entry Details PubMed
TargetAryl hydrocarbon receptor(Mouse)
Palacky University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50434121BDBM50434121(CHEMBL2381492)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of HCV NS5A L31V mutant in HCV genotype 1a assessed as reduction in viral replication by cell based replicon assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2026
Entry Details PubMed
TargetAryl hydrocarbon receptor(Human)
Palacky University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50653959BDBM50653959(CHEMBL107324)
Affinity DataEC50:  1.64E+5nMAssay Description:Inhibition of human c-Met in human GTL16 cells by cell-based assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/3/2026
Entry Details PubMed