Report error Found 118 Enz. Inhib. hit(s) with all data for entry = 50022851
Affinity DataKi: 6nMAssay Description:Agonist activity at human PPARgamma transfected in COS-7 cells assessed luciferase activity measured after 24 hrs by cell based luciferase transactiv...More data for this Ligand-Target Pair
Affinity DataKi: 6nMAssay Description:Agonist activity at human PPARdelta transfected in COS-7 cells assessed luciferase activity measured after 24 hrs by cell based luciferase transactiv...More data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 12nMAssay Description:Inhibition of human GluN1-1a/NR2A receptor expressed in transgenic mouse fibroblast cells assessed as inhibition of L-glutamate-induced excitotoxicit...More data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 12nMAssay Description:Inhibition of human GluN1-1a/NR2B receptor expressed in transgenic mouse fibroblast cells assessed as inhibition of L-glutamate-induced excitotoxicit...More data for this Ligand-Target Pair
Affinity DataKi: 17nMAssay Description:Antagonist activity at human EP3 receptor expressed in CHO cells by cell based cAMP functional assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 18nMAssay Description:Antagonist activity at human EP3 receptor expressed in CHO cells by cell based cAMP functional assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 26nMAssay Description:Agonist activity at human PPARalpha transfected in COS-7 cells assessed luciferase activity measured after 24 hrs by cell based luciferase transactiv...More data for this Ligand-Target Pair
Affinity DataKi: 26nMAssay Description:Antagonist activity at human EP3 receptor expressed in CHO cells by cell based cAMP functional assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 26nMAssay Description:Inhibition of human ARG1 in HEK293 cells by cell based assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 28nMAssay Description:Antagonist activity at human EP3 receptor expressed in CHO cells by cell based cAMP functional assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 34nMAssay Description:Antagonist activity at human EP3 receptor expressed in CHO cells by cell based cAMP functional assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 62nMAssay Description:Antagonist activity at human EP3 receptor expressed in CHO cells by cell based cAMP functional assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 71nMAssay Description:Antagonist activity at human EP3 receptor expressed in CHO cells by cell based cAMP functional assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 71nMAssay Description:Antagonist activity at human EP3 receptor expressed in CHO cells by cell based cAMP functional assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 74nMAssay Description:Antagonist activity at human EP3 receptor expressed in CHO cells by cell based cAMP functional assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 74nMAssay Description:Antagonist activity at human EP3 receptor expressed in CHO cells by cell based cAMP functional assayMore data for this Ligand-Target Pair
Affinity DataKi: 76nMAssay Description:Antagonist activity at human EP3 receptor expressed in CHO cells by cell based cAMP functional assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 93nMAssay Description:Antagonist activity at human EP3 receptor expressed in CHO cells by cell based cAMP functional assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 94nMAssay Description:Antagonist activity at human EP3 receptor expressed in CHO cells by cell based cAMP functional assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 95nMAssay Description:Antagonist activity at human EP3 receptor expressed in CHO cells by cell based cAMP functional assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 130nMAssay Description:Antagonist activity at human EP3 receptor expressed in CHO cells by cell based cAMP functional assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 250nMAssay Description:Antagonist activity at human EP3 receptor expressed in CHO cells by cell based cAMP functional assayMore data for this Ligand-Target Pair
Affinity DataKi: 250nMAssay Description:Antagonist activity at human EP3 receptor expressed in CHO cells by cell based cAMP functional assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 270nMAssay Description:Inhibition of human GluN1-1a/NR2B receptor expressed in transgenic mouse fibroblast cells assessed as inhibition of L-glutamate-induced excitotoxicit...More data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 330nMAssay Description:Agonist activity at human PPARdelta transfected in COS-7 cells assessed luciferase activity measured after 24 hrs by cell based luciferase transactiv...More data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 380nMAssay Description:Inhibition of NGF-activated full length TRKA (unknown origin) by Cell-based beta-galactosidase PathHunter assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 400nMAssay Description:Inhibition of JAK2 (unknown origin) by EPO-stimulated cell based assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 450nMAssay Description:Agonist activity at human PPARgamma transfected in COS-7 cells assessed luciferase activity measured after 24 hrs by cell based luciferase transactiv...More data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 640nMAssay Description:Agonist activity at human PPARdelta transfected in COS-7 cells assessed luciferase activity measured after 24 hrs by cell based luciferase transactiv...More data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 660nMAssay Description:Agonist activity at human PPARdelta transfected in COS-7 cells assessed luciferase activity measured after 24 hrs by cell based luciferase transactiv...More data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 680nMAssay Description:Agonist activity at human PPARalpha transfected in COS-7 cells assessed luciferase activity measured after 24 hrs by cell based luciferase transactiv...More data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 720nMAssay Description:Inhibition of human GluN1-1a/NR2A receptor expressed in transgenic mouse fibroblast cells assessed as inhibition of L-glutamate-induced excitotoxicit...More data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 790nMAssay Description:Inhibition of human GluN1-1a/NR2A receptor expressed in transgenic mouse fibroblast cells assessed as inhibition of L-glutamate-induced excitotoxicit...More data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 1.03E+3nMAssay Description:Inhibition of mouse STC1 in cell based assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 1.11E+3nMAssay Description:Inhibition of human STC1 in cell based assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 1.44E+3nMAssay Description:Inhibition of human ARG1 in HEK293 cells by cell based assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 2.20E+3nMAssay Description:Inhibition of PD-1/PD-L1 interaction in human Jurkat cells cocultured with CHO cells expressing PD-Ll/TCRAct assessed as activation of effector Jurka...More data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 2.40E+3nMAssay Description:Antagonist activity at human EP3 receptor expressed in CHO cells by cell based cAMP functional assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 2.70E+3nMAssay Description:Inhibition of BDNF-activated full length TRKB (unknown origin) by Cell-based beta-galactosidase PathHunter assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 2.95E+3nMAssay Description:Inhibition of mouse STC1 in cell based assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 3.02E+3nMAssay Description:Antagonist activity at human EP3 receptor expressed in CHO cells by cell based cAMP functional assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 3.08E+3nMAssay Description:Agonist activity at human PPARalpha transfected in COS-7 cells assessed luciferase activity measured after 24 hrs by cell based luciferase transactiv...More data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 3.65E+3nMAssay Description:Agonist activity at human PPARalpha transfected in COS-7 cells assessed luciferase activity measured after 24 hrs by cell based luciferase transactiv...More data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 4.20E+3nMAssay Description:Agonist activity at human PPARalpha transfected in COS-7 cells assessed luciferase activity measured after 24 hrs by cell based luciferase transactiv...More data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 4.26E+3nMAssay Description:Inhibition of human GluN1-1a/NR2A receptor expressed in transgenic mouse fibroblast cells assessed as inhibition of L-glutamate-induced excitotoxicit...More data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 4.50E+3nMAssay Description:Antagonist activity at human EP3 receptor expressed in CHO cells by cell based cAMP functional assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 4.80E+3nMAssay Description:Agonist activity at human PPARgamma transfected in COS-7 cells assessed luciferase activity measured after 24 hrs by cell based luciferase transactiv...More data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 5.20E+3nMAssay Description:Agonist activity at human PPARdelta transfected in COS-7 cells assessed luciferase activity measured after 24 hrs by cell based luciferase transactiv...More data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 7.00E+3nMAssay Description:Agonist activity at human PPARalpha transfected in COS-7 cells assessed luciferase activity measured after 24 hrs by cell based luciferase transactiv...More data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 8.90E+3nMAssay Description:Antagonist activity at human EP3 receptor expressed in CHO cells by cell based cAMP functional assayMore data for this Ligand-Target Pair
Ligand Info

3D Structure (crystal)



















