Compile Data Set for Download or QSAR
Report error Found 12 Enz. Inhib. hit(s) with all data for entry = 50022844
TargetStructural capsid protein(Human immunodeficiency virus type 1)
Shandong University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50654957BDBM50654957(CHEMBL6150629)
Affinity DataKd:  25nMAssay Description:Antagonist activity at Prolink-tagged human CXCR6 receptor assessed as inhibition of forskolin-induced cAMP accumulation by DiscoveRx cell based assa...More data for this Ligand-Target Pair
Ligand InfoPDB
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetStructural capsid protein(Human immunodeficiency virus type 1)
Shandong University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50654957BDBM50654957(CHEMBL6150629)
Affinity DataKd:  81nMAssay Description:Antagonist activity at Prolink-tagged human CXCR6 receptor assessed as inhibition of CXCL16-induced beta-arrestin recruitment by DiscoveRx cell based...More data for this Ligand-Target Pair
Ligand InfoPDB
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetStructural capsid protein(Human immunodeficiency virus type 1)
Shandong University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50654958BDBM50654958(CHEMBL6168037)
Affinity DataKd:  88nMAssay Description:Antagonist activity at Prolink-tagged human CXCR6 receptor assessed as inhibition of forskolin-induced cAMP accumulation by DiscoveRx cell based assa...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetStructural capsid protein(Human immunodeficiency virus type 1)
Shandong University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50654959BDBM50654959(CHEMBL6146335)
Affinity DataKd:  95nMAssay Description:Antagonist activity at Prolink-tagged human CXCR6 receptor assessed as inhibition of forskolin-induced cAMP accumulation by DiscoveRx cell based assa...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetStructural capsid protein(Human immunodeficiency virus type 1)
Shandong University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50654958BDBM50654958(CHEMBL6168037)
Affinity DataKd:  153nMAssay Description:Antagonist activity at Prolink-tagged human CXCR6 receptor assessed as inhibition of forskolin-induced cAMP accumulation by DiscoveRx cell based assa...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetStructural capsid protein(Human immunodeficiency virus type 1)
Shandong University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50654959BDBM50654959(CHEMBL6146335)
Affinity DataKd:  196nMAssay Description:Antagonist activity at Prolink-tagged human CXCR6 receptor assessed as inhibition of forskolin-induced cAMP accumulation by DiscoveRx cell based assa...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetStructural capsid protein(Human immunodeficiency virus type 1)
Shandong University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50511740BDBM50511740(CHEMBL4471665)
Affinity DataKd:  215nMAssay Description:Antagonist activity at mouse CXCR6 by DiscoveRx cell based beta-arrestin assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetStructural capsid protein(Human immunodeficiency virus type 1)
Shandong University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50654956BDBM50654956(CHEMBL6143742)
Affinity DataKd:  267nMAssay Description:Antagonist activity at Prolink-tagged human CXCR6 receptor assessed as inhibition of CXCL16-induced beta-arrestin recruitment by DiscoveRx cell based...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetStructural capsid protein(Human immunodeficiency virus type 1)
Shandong University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50654956BDBM50654956(CHEMBL6143742)
Affinity DataKd:  305nMAssay Description:Antagonist activity at Prolink-tagged human CXCR6 receptor assessed as inhibition of forskolin-induced cAMP accumulation by DiscoveRx cell based assa...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetStructural capsid protein(Human immunodeficiency virus type 1)
Shandong University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50467395BDBM50467395(CHEMBL1229713)
Affinity DataKd:  2.33E+3nMAssay Description:Antagonist activity at Prolink-tagged human CXCR6 receptor assessed as inhibition of forskolin-induced cAMP accumulation by DiscoveRx cell based assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetStructural capsid protein(Human immunodeficiency virus type 1)
Shandong University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50511740BDBM50511740(CHEMBL4471665)
Affinity DataKd:  2.45E+3nMAssay Description:Antagonist activity at Prolink-tagged human CXCR6 receptor assessed as inhibition of forskolin-induced cAMP accumulation by DiscoveRx cell based assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetStructural capsid protein(Human immunodeficiency virus type 1)
Shandong University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50467395BDBM50467395(CHEMBL1229713)
Affinity DataKd:  4.44E+3nMAssay Description:Antagonist activity at Prolink-tagged human CXCR6 receptor assessed as inhibition of forskolin-induced cAMP accumulation by DiscoveRx cell based assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed