Report error Found 55 Enz. Inhib. hit(s) with all data for entry = 50022982
Affinity DataKi: 3.60nMAssay Description:Inhibition of N-terminal human Keap1 Kelch (321 to 609 residues)-Nrf2 protein-protein interaction assessed as inhibition constant incubated for 1 hr ...More data for this Ligand-Target Pair
Ligand Info
Affinity DataKd: 4.20nMAssay Description:Binding affinity to Keap1 Kelch domain (unknown origin) assessed as dissociation constant by SPR analysisMore data for this Ligand-Target Pair
Ligand InfoPDB
Affinity DataKi: 13nMAssay Description:Binding affinity to his-tagged human Keap1 Kelch (321 to 609 residues) expressed in Escherichia coli BL21 (DE3)-Nrf2 protein-protein interaction asse...More data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 14nMAssay Description:Binding affinity to his-tagged human Keap1 Kelch (321 to 609 residues) expressed in Escherichia coli BL21 (DE3)-Nrf2 protein-protein interaction asse...More data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 14nMAssay Description:Binding affinity to his-tagged human Keap1 Kelch (321 to 609 residues) expressed in Escherichia coli BL21 (DE3)-Nrf2 protein-protein interaction asse...More data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 15nMAssay Description:Binding affinity to his-tagged human Keap1 Kelch (321 to 609 residues) expressed in Escherichia coli BL21 (DE3)-Nrf2 protein-protein interaction asse...More data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 15nMAssay Description:Binding affinity to his-tagged human Keap1 Kelch (321 to 609 residues) expressed in Escherichia coli BL21 (DE3)-Nrf2 protein-protein interaction asse...More data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 16nMAssay Description:Binding affinity to his-tagged human Keap1 Kelch (321 to 609 residues) expressed in Escherichia coli BL21 (DE3)-Nrf2 protein-protein interaction asse...More data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 17nMAssay Description:Binding affinity to his-tagged human Keap1 Kelch (321 to 609 residues) expressed in Escherichia coli BL21 (DE3)-Nrf2 protein-protein interaction asse...More data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 24nMAssay Description:Binding affinity to his-tagged human Keap1 Kelch (321 to 609 residues) expressed in Escherichia coli BL21 (DE3)-Nrf2 protein-protein interaction asse...More data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 27nMAssay Description:Binding affinity to his-tagged human Keap1 Kelch (321 to 609 residues) expressed in Escherichia coli BL21 (DE3)-Nrf2 protein-protein interaction asse...More data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 32nMAssay Description:Binding affinity to his-tagged human Keap1 Kelch (321 to 609 residues) expressed in Escherichia coli BL21 (DE3)-Nrf2 protein-protein interaction asse...More data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 35nMAssay Description:Binding affinity to his-tagged human Keap1 Kelch (321 to 609 residues) expressed in Escherichia coli BL21 (DE3)-Nrf2 protein-protein interaction asse...More data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 36nMAssay Description:Binding affinity to his-tagged human Keap1 Kelch (321 to 609 residues) expressed in Escherichia coli BL21 (DE3)-Nrf2 protein-protein interaction asse...More data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 41nMAssay Description:Binding affinity to his-tagged human Keap1 Kelch (321 to 609 residues) expressed in Escherichia coli BL21 (DE3)-Nrf2 protein-protein interaction asse...More data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 43nMAssay Description:Binding affinity to his-tagged human Keap1 Kelch (321 to 609 residues) expressed in Escherichia coli BL21 (DE3)-Nrf2 protein-protein interaction asse...More data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 56nMAssay Description:Binding affinity to his-tagged human Keap1 Kelch (321 to 609 residues) expressed in Escherichia coli BL21 (DE3)-Nrf2 protein-protein interaction asse...More data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 65nMAssay Description:Binding affinity to his-tagged human Keap1 Kelch (321 to 609 residues) expressed in Escherichia coli BL21 (DE3)-Nrf2 protein-protein interaction asse...More data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 69nMAssay Description:Binding affinity to his-tagged human Keap1 Kelch (321 to 609 residues) expressed in Escherichia coli BL21 (DE3)-Nrf2 protein-protein interaction asse...More data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 81nMAssay Description:Binding affinity to his-tagged human Keap1 Kelch (321 to 609 residues) expressed in Escherichia coli BL21 (DE3)-Nrf2 protein-protein interaction asse...More data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 91nMAssay Description:Binding affinity to his-tagged human Keap1 Kelch (321 to 609 residues) expressed in Escherichia coli BL21 (DE3)-Nrf2 protein-protein interaction asse...More data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 110nMAssay Description:Binding affinity to his-tagged human Keap1 Kelch (321 to 609 residues) expressed in Escherichia coli BL21 (DE3)-Nrf2 protein-protein interaction asse...More data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 120nMAssay Description:Binding affinity to his-tagged human Keap1 Kelch (321 to 609 residues) expressed in Escherichia coli BL21 (DE3)-Nrf2 protein-protein interaction asse...More data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 130nMAssay Description:Binding affinity to his-tagged human Keap1 Kelch (321 to 609 residues) expressed in Escherichia coli BL21 (DE3)-Nrf2 protein-protein interaction asse...More data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 130nMAssay Description:Binding affinity to his-tagged human Keap1 Kelch (321 to 609 residues) expressed in Escherichia coli BL21 (DE3)-Nrf2 protein-protein interaction asse...More data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 130nMAssay Description:Binding affinity to his-tagged human Keap1 Kelch (321 to 609 residues) expressed in Escherichia coli BL21 (DE3)-Nrf2 protein-protein interaction asse...More data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 130nMAssay Description:Binding affinity to his-tagged human Keap1 Kelch (321 to 609 residues) expressed in Escherichia coli BL21 (DE3)-Nrf2 protein-protein interaction asse...More data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 140nMAssay Description:Binding affinity to his-tagged human Keap1 Kelch (321 to 609 residues) expressed in Escherichia coli BL21 (DE3)-Nrf2 protein-protein interaction asse...More data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 150nMAssay Description:Binding affinity to his-tagged human Keap1 Kelch (321 to 609 residues) expressed in Escherichia coli BL21 (DE3)-Nrf2 protein-protein interaction asse...More data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 170nMAssay Description:Binding affinity to his-tagged human Keap1 Kelch (321 to 609 residues) expressed in Escherichia coli BL21 (DE3)-Nrf2 protein-protein interaction asse...More data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 180nMAssay Description:Binding affinity to his-tagged human Keap1 Kelch (321 to 609 residues) expressed in Escherichia coli BL21 (DE3)-Nrf2 protein-protein interaction asse...More data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 180nMAssay Description:Binding affinity to his-tagged human Keap1 Kelch (321 to 609 residues) expressed in Escherichia coli BL21 (DE3)-Nrf2 protein-protein interaction asse...More data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 180nMAssay Description:Binding affinity to his-tagged human Keap1 Kelch (321 to 609 residues) expressed in Escherichia coli BL21 (DE3)-Nrf2 protein-protein interaction asse...More data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 190nMAssay Description:Binding affinity to his-tagged human Keap1 Kelch (321 to 609 residues) expressed in Escherichia coli BL21 (DE3)-Nrf2 protein-protein interaction asse...More data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 190nMAssay Description:Binding affinity to his-tagged human Keap1 Kelch (321 to 609 residues) expressed in Escherichia coli BL21 (DE3)-Nrf2 protein-protein interaction asse...More data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 260nMAssay Description:Binding affinity to his-tagged human Keap1 Kelch (321 to 609 residues) expressed in Escherichia coli BL21 (DE3)-Nrf2 protein-protein interaction asse...More data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 270nMAssay Description:Binding affinity to his-tagged human Keap1 Kelch (321 to 609 residues) expressed in Escherichia coli BL21 (DE3)-Nrf2 protein-protein interaction asse...More data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 280nMAssay Description:Binding affinity to his-tagged human Keap1 Kelch (321 to 609 residues) expressed in Escherichia coli BL21 (DE3)-Nrf2 protein-protein interaction asse...More data for this Ligand-Target Pair
Affinity DataKi: 350nMAssay Description:Binding affinity to his-tagged human Keap1 Kelch (321 to 609 residues) expressed in Escherichia coli BL21 (DE3)-Nrf2 protein-protein interaction asse...More data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 360nMAssay Description:Binding affinity to his-tagged human Keap1 Kelch (321 to 609 residues) expressed in Escherichia coli BL21 (DE3)-Nrf2 protein-protein interaction asse...More data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 370nMAssay Description:Binding affinity to his-tagged human Keap1 Kelch (321 to 609 residues) expressed in Escherichia coli BL21 (DE3)-Nrf2 protein-protein interaction asse...More data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 370nMAssay Description:Binding affinity to his-tagged human Keap1 Kelch (321 to 609 residues) expressed in Escherichia coli BL21 (DE3)-Nrf2 protein-protein interaction asse...More data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 590nMAssay Description:Binding affinity to his-tagged human Keap1 Kelch (321 to 609 residues) expressed in Escherichia coli BL21 (DE3)-Nrf2 protein-protein interaction asse...More data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 930nMAssay Description:Binding affinity to his-tagged human Keap1 Kelch (321 to 609 residues) expressed in Escherichia coli BL21 (DE3)-Nrf2 protein-protein interaction asse...More data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 1.20E+3nMAssay Description:Binding affinity to his-tagged human Keap1 Kelch (321 to 609 residues) expressed in Escherichia coli BL21 (DE3)-Nrf2 protein-protein interaction asse...More data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 1.30E+3nMAssay Description:Binding affinity to his-tagged human Keap1 Kelch (321 to 609 residues) expressed in Escherichia coli BL21 (DE3)-Nrf2 protein-protein interaction asse...More data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 2.90E+3nMAssay Description:Binding affinity to his-tagged human Keap1 Kelch (321 to 609 residues) expressed in Escherichia coli BL21 (DE3)-Nrf2 protein-protein interaction asse...More data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 2.90E+3nMAssay Description:Binding affinity to his-tagged human Keap1 Kelch (321 to 609 residues) expressed in Escherichia coli BL21 (DE3)-Nrf2 protein-protein interaction asse...More data for this Ligand-Target Pair
Affinity DataKi: 3.60E+3nMAssay Description:Binding affinity to his-tagged human Keap1 Kelch (321 to 609 residues) expressed in Escherichia coli BL21 (DE3)-Nrf2 protein-protein interaction asse...More data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 4.00E+3nMAssay Description:Binding affinity to his-tagged human Keap1 Kelch (321 to 609 residues) expressed in Escherichia coli BL21 (DE3)-Nrf2 protein-protein interaction asse...More data for this Ligand-Target Pair
Ligand Info


3D Structure (crystal)














































