Report error Found 67 Enz. Inhib. hit(s) with all data for entry = 50022972
TargetNuclear factor erythroid 2-related factor 2(Human)
Peking Union Medical College and Chinese Academy of Medical Sciences
Curated by ChEMBL
Peking Union Medical College and Chinese Academy of Medical Sciences
Curated by ChEMBL
Affinity DataKd: 1.30nMAssay Description:Binding affinity to human Keap1-Nrf2 protein-protein interaction assessed as dissociation constant by ITC assayMore data for this Ligand-Target Pair
TargetNuclear factor erythroid 2-related factor 2(Mouse)
Peking Union Medical College and Chinese Academy of Medical Sciences
Curated by ChEMBL
Peking Union Medical College and Chinese Academy of Medical Sciences
Curated by ChEMBL
Affinity DataKd: 1.80nMAssay Description:Binding affinity to his-tagged recombinant mouse Keap1 KELCH domain (321 to 609 residues) expressed in Escherichia coli BL21 DE3/Nrf2 assessed as dis...More data for this Ligand-Target Pair
Ligand Info
TargetNuclear factor erythroid 2-related factor 2(Human)
Peking Union Medical College and Chinese Academy of Medical Sciences
Curated by ChEMBL
Peking Union Medical College and Chinese Academy of Medical Sciences
Curated by ChEMBL
Affinity DataKd: 2.5nMAssay Description:Binding affinity to human Keap1-Nrf2 protein-protein interaction assessed as dissociation constant by SPR assayMore data for this Ligand-Target Pair
Ligand Info
TargetNuclear factor erythroid 2-related factor 2(Mouse)
Peking Union Medical College and Chinese Academy of Medical Sciences
Curated by ChEMBL
Peking Union Medical College and Chinese Academy of Medical Sciences
Curated by ChEMBL
Affinity DataKd: 3.10nMAssay Description:Binding affinity to his-tagged recombinant mouse Keap1 KELCH domain (321 to 609 residues) expressed in Escherichia coli BL21 DE3/Nrf2 assessed as dis...More data for this Ligand-Target Pair
Ligand Info
TargetNuclear factor erythroid 2-related factor 2(Mouse)
Peking Union Medical College and Chinese Academy of Medical Sciences
Curated by ChEMBL
Peking Union Medical College and Chinese Academy of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 13nMAssay Description:Competitive inhibition of his-tagged recombinant mouse Keap1 KELCH domain (321 to 609 residues) expressed in Escherichia coli BL21 DE3/Nrf2 incubated...More data for this Ligand-Target Pair
Ligand Info
TargetNuclear factor erythroid 2-related factor 2(Human)
Peking Union Medical College and Chinese Academy of Medical Sciences
Curated by ChEMBL
Peking Union Medical College and Chinese Academy of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 14nMAssay Description:Inhibition of Keap1-Nrf2 protein-protein interaction (unknown origin) by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetNuclear factor erythroid 2-related factor 2(Mouse)
Peking Union Medical College and Chinese Academy of Medical Sciences
Curated by ChEMBL
Peking Union Medical College and Chinese Academy of Medical Sciences
Curated by ChEMBL
Affinity DataKd: 14nMAssay Description:Binding affinity to his-tagged recombinant mouse Keap1 KELCH domain (321 to 609 residues) expressed in Escherichia coli BL21 DE3/Nrf2 assessed as dis...More data for this Ligand-Target Pair
Ligand Info
TargetNuclear factor erythroid 2-related factor 2(Human)
Peking Union Medical College and Chinese Academy of Medical Sciences
Curated by ChEMBL
Peking Union Medical College and Chinese Academy of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 15nMAssay Description:Inhibition of Keap1-Nrf2 protein-protein interaction (unknown origin) by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetNuclear factor erythroid 2-related factor 2(Human)
Peking Union Medical College and Chinese Academy of Medical Sciences
Curated by ChEMBL
Peking Union Medical College and Chinese Academy of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 15nMAssay Description:Inhibition of Keap1-Nrf2 protein-protein interaction (unknown origin) by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand Info
TargetNuclear factor erythroid 2-related factor 2(Mouse)
Peking Union Medical College and Chinese Academy of Medical Sciences
Curated by ChEMBL
Peking Union Medical College and Chinese Academy of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 16nMAssay Description:Competitive inhibition of his-tagged recombinant mouse Keap1 KELCH domain (321 to 609 residues) expressed in Escherichia coli BL21 DE3/Nrf2 incubated...More data for this Ligand-Target Pair
Ligand Info
TargetNuclear factor erythroid 2-related factor 2(Mouse)
Peking Union Medical College and Chinese Academy of Medical Sciences
Curated by ChEMBL
Peking Union Medical College and Chinese Academy of Medical Sciences
Curated by ChEMBL
Affinity DataKd: 17nMAssay Description:Binding affinity to his-tagged recombinant mouse Keap1 KELCH domain (321 to 609 residues) expressed in Escherichia coli BL21 DE3/Nrf2 assessed as dis...More data for this Ligand-Target Pair
Ligand Info
TargetNuclear factor erythroid 2-related factor 2(Mouse)
Peking Union Medical College and Chinese Academy of Medical Sciences
Curated by ChEMBL
Peking Union Medical College and Chinese Academy of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 20nMAssay Description:Competitive inhibition of his-tagged recombinant mouse Keap1 KELCH domain (321 to 609 residues) expressed in Escherichia coli BL21 DE3/Nrf2 incubated...More data for this Ligand-Target Pair
Ligand Info
TargetNuclear factor erythroid 2-related factor 2(Mouse)
Peking Union Medical College and Chinese Academy of Medical Sciences
Curated by ChEMBL
Peking Union Medical College and Chinese Academy of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 20nMAssay Description:Competitive inhibition of his-tagged recombinant mouse Keap1 KELCH domain (321 to 609 residues) expressed in Escherichia coli BL21 DE3/Nrf2 incubated...More data for this Ligand-Target Pair
Ligand Info
TargetNuclear factor erythroid 2-related factor 2(Human)
Peking Union Medical College and Chinese Academy of Medical Sciences
Curated by ChEMBL
Peking Union Medical College and Chinese Academy of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 22nMAssay Description:Inhibition of Keap1-Nrf2 protein-protein interaction (unknown origin) by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetNuclear factor erythroid 2-related factor 2(Mouse)
Peking Union Medical College and Chinese Academy of Medical Sciences
Curated by ChEMBL
Peking Union Medical College and Chinese Academy of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 22nMAssay Description:Competitive inhibition of his-tagged recombinant mouse Keap1 KELCH domain (321 to 609 residues) expressed in Escherichia coli BL21 DE3/Nrf2 incubated...More data for this Ligand-Target Pair
Ligand Info
TargetNuclear factor erythroid 2-related factor 2(Mouse)
Peking Union Medical College and Chinese Academy of Medical Sciences
Curated by ChEMBL
Peking Union Medical College and Chinese Academy of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 25nMAssay Description:Competitive inhibition of his-tagged recombinant mouse Keap1 KELCH domain (321 to 609 residues) expressed in Escherichia coli BL21 DE3/Nrf2 incubated...More data for this Ligand-Target Pair
Ligand Info
TargetNuclear factor erythroid 2-related factor 2(Mouse)
Peking Union Medical College and Chinese Academy of Medical Sciences
Curated by ChEMBL
Peking Union Medical College and Chinese Academy of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 38nMAssay Description:Competitive inhibition of his-tagged recombinant mouse Keap1 KELCH domain (321 to 609 residues) expressed in Escherichia coli BL21 DE3/Nrf2 incubated...More data for this Ligand-Target Pair
Ligand Info
TargetNuclear factor erythroid 2-related factor 2(Mouse)
Peking Union Medical College and Chinese Academy of Medical Sciences
Curated by ChEMBL
Peking Union Medical College and Chinese Academy of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 50nMAssay Description:Competitive inhibition of his-tagged recombinant mouse Keap1 KELCH domain (321 to 609 residues) expressed in Escherichia coli BL21 DE3/Nrf2 incubated...More data for this Ligand-Target Pair
Ligand Info
TargetNuclear factor erythroid 2-related factor 2(Mouse)
Peking Union Medical College and Chinese Academy of Medical Sciences
Curated by ChEMBL
Peking Union Medical College and Chinese Academy of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 50nMAssay Description:Competitive inhibition of his-tagged recombinant mouse Keap1 KELCH domain (321 to 609 residues) expressed in Escherichia coli BL21 DE3/Nrf2 incubated...More data for this Ligand-Target Pair
Ligand Info
TargetNuclear factor erythroid 2-related factor 2(Mouse)
Peking Union Medical College and Chinese Academy of Medical Sciences
Curated by ChEMBL
Peking Union Medical College and Chinese Academy of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 53nMAssay Description:Competitive inhibition of his-tagged recombinant mouse Keap1 KELCH domain (321 to 609 residues) expressed in Escherichia coli BL21 DE3/Nrf2 incubated...More data for this Ligand-Target Pair
Ligand Info
TargetNuclear factor erythroid 2-related factor 2(Human)
Peking Union Medical College and Chinese Academy of Medical Sciences
Curated by ChEMBL
Peking Union Medical College and Chinese Academy of Medical Sciences
Curated by ChEMBL
Affinity DataKd: 58nMAssay Description:Binding affinity to human Keap1-Nrf2 protein-protein interaction assessed as dissociation constant by ITC assayMore data for this Ligand-Target Pair
TargetNuclear factor erythroid 2-related factor 2(Mouse)
Peking Union Medical College and Chinese Academy of Medical Sciences
Curated by ChEMBL
Peking Union Medical College and Chinese Academy of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 61nMAssay Description:Competitive inhibition of his-tagged recombinant mouse Keap1 KELCH domain (321 to 609 residues) expressed in Escherichia coli BL21 DE3/Nrf2 incubated...More data for this Ligand-Target Pair
Ligand Info
TargetNuclear factor erythroid 2-related factor 2(Mouse)
Peking Union Medical College and Chinese Academy of Medical Sciences
Curated by ChEMBL
Peking Union Medical College and Chinese Academy of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 82nMAssay Description:Competitive inhibition of his-tagged recombinant mouse Keap1 KELCH domain (321 to 609 residues) expressed in Escherichia coli BL21 DE3/Nrf2 incubated...More data for this Ligand-Target Pair
Ligand Info
TargetNuclear factor erythroid 2-related factor 2(Mouse)
Peking Union Medical College and Chinese Academy of Medical Sciences
Curated by ChEMBL
Peking Union Medical College and Chinese Academy of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 122nMAssay Description:Competitive inhibition of his-tagged recombinant mouse Keap1 KELCH domain (321 to 609 residues) expressed in Escherichia coli BL21 DE3/Nrf2 incubated...More data for this Ligand-Target Pair
Ligand Info
TargetNuclear factor erythroid 2-related factor 2(Mouse)
Peking Union Medical College and Chinese Academy of Medical Sciences
Curated by ChEMBL
Peking Union Medical College and Chinese Academy of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 132nMAssay Description:Competitive inhibition of his-tagged recombinant mouse Keap1 KELCH domain (321 to 609 residues) expressed in Escherichia coli BL21 DE3/Nrf2 incubated...More data for this Ligand-Target Pair
Ligand Info
TargetNuclear factor erythroid 2-related factor 2(Mouse)
Peking Union Medical College and Chinese Academy of Medical Sciences
Curated by ChEMBL
Peking Union Medical College and Chinese Academy of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 140nMAssay Description:Competitive inhibition of his-tagged recombinant mouse Keap1 KELCH domain (321 to 609 residues) expressed in Escherichia coli BL21 DE3/Nrf2 incubated...More data for this Ligand-Target Pair
Ligand Info
TargetNuclear factor erythroid 2-related factor 2(Mouse)
Peking Union Medical College and Chinese Academy of Medical Sciences
Curated by ChEMBL
Peking Union Medical College and Chinese Academy of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 170nMAssay Description:Competitive inhibition of his-tagged recombinant mouse Keap1 KELCH domain (321 to 609 residues) expressed in Escherichia coli BL21 DE3/Nrf2 incubated...More data for this Ligand-Target Pair
Ligand Info
TargetNuclear factor erythroid 2-related factor 2(Mouse)
Peking Union Medical College and Chinese Academy of Medical Sciences
Curated by ChEMBL
Peking Union Medical College and Chinese Academy of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 179nMAssay Description:Competitive inhibition of his-tagged recombinant mouse Keap1 KELCH domain (321 to 609 residues) expressed in Escherichia coli BL21 DE3/Nrf2 incubated...More data for this Ligand-Target Pair
Ligand Info
TargetNuclear factor erythroid 2-related factor 2(Mouse)
Peking Union Medical College and Chinese Academy of Medical Sciences
Curated by ChEMBL
Peking Union Medical College and Chinese Academy of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 280nMAssay Description:Competitive inhibition of his-tagged recombinant mouse Keap1 KELCH domain (321 to 609 residues) expressed in Escherichia coli BL21 DE3/Nrf2 incubated...More data for this Ligand-Target Pair
Ligand Info
TargetNuclear factor erythroid 2-related factor 2(Mouse)
Peking Union Medical College and Chinese Academy of Medical Sciences
Curated by ChEMBL
Peking Union Medical College and Chinese Academy of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 300nMAssay Description:Competitive inhibition of his-tagged recombinant mouse Keap1 KELCH domain (321 to 609 residues) expressed in Escherichia coli BL21 DE3/Nrf2 incubated...More data for this Ligand-Target Pair
Ligand Info
TargetNuclear factor erythroid 2-related factor 2(Mouse)
Peking Union Medical College and Chinese Academy of Medical Sciences
Curated by ChEMBL
Peking Union Medical College and Chinese Academy of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 300nMAssay Description:Competitive inhibition of his-tagged recombinant mouse Keap1 KELCH domain (321 to 609 residues) expressed in Escherichia coli BL21 DE3/Nrf2 incubated...More data for this Ligand-Target Pair
Ligand Info
TargetNuclear factor erythroid 2-related factor 2(Mouse)
Peking Union Medical College and Chinese Academy of Medical Sciences
Curated by ChEMBL
Peking Union Medical College and Chinese Academy of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 330nMAssay Description:Competitive inhibition of his-tagged recombinant mouse Keap1 KELCH domain (321 to 609 residues) expressed in Escherichia coli BL21 DE3/Nrf2 incubated...More data for this Ligand-Target Pair
Ligand Info
TargetNuclear factor erythroid 2-related factor 2(Mouse)
Peking Union Medical College and Chinese Academy of Medical Sciences
Curated by ChEMBL
Peking Union Medical College and Chinese Academy of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 510nMAssay Description:Competitive inhibition of his-tagged recombinant mouse Keap1 KELCH domain (321 to 609 residues) expressed in Escherichia coli BL21 DE3/Nrf2 incubated...More data for this Ligand-Target Pair
Ligand Info
TargetNuclear factor erythroid 2-related factor 2(Mouse)
Peking Union Medical College and Chinese Academy of Medical Sciences
Curated by ChEMBL
Peking Union Medical College and Chinese Academy of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 520nMAssay Description:Competitive inhibition of his-tagged recombinant mouse Keap1 KELCH domain (321 to 609 residues) expressed in Escherichia coli BL21 DE3/Nrf2 incubated...More data for this Ligand-Target Pair
Ligand Info
TargetNuclear factor erythroid 2-related factor 2(Mouse)
Peking Union Medical College and Chinese Academy of Medical Sciences
Curated by ChEMBL
Peking Union Medical College and Chinese Academy of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 620nMAssay Description:Competitive inhibition of his-tagged recombinant mouse Keap1 KELCH domain (321 to 609 residues) expressed in Escherichia coli BL21 DE3/Nrf2 incubated...More data for this Ligand-Target Pair
Ligand Info
TargetNuclear factor erythroid 2-related factor 2(Mouse)
Peking Union Medical College and Chinese Academy of Medical Sciences
Curated by ChEMBL
Peking Union Medical College and Chinese Academy of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 708nMAssay Description:Competitive inhibition of his-tagged recombinant mouse Keap1 KELCH domain (321 to 609 residues) expressed in Escherichia coli BL21 DE3/Nrf2 incubated...More data for this Ligand-Target Pair
Ligand Info
TargetNuclear factor erythroid 2-related factor 2(Mouse)
Peking Union Medical College and Chinese Academy of Medical Sciences
Curated by ChEMBL
Peking Union Medical College and Chinese Academy of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 750nMAssay Description:Competitive inhibition of his-tagged recombinant mouse Keap1 KELCH domain (321 to 609 residues) expressed in Escherichia coli BL21 DE3/Nrf2 incubated...More data for this Ligand-Target Pair
Ligand Info
TargetNuclear factor erythroid 2-related factor 2(Mouse)
Peking Union Medical College and Chinese Academy of Medical Sciences
Curated by ChEMBL
Peking Union Medical College and Chinese Academy of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 860nMAssay Description:Competitive inhibition of his-tagged recombinant mouse Keap1 KELCH domain (321 to 609 residues) expressed in Escherichia coli BL21 DE3/Nrf2 incubated...More data for this Ligand-Target Pair
Ligand Info
TargetNuclear factor erythroid 2-related factor 2(Mouse)
Peking Union Medical College and Chinese Academy of Medical Sciences
Curated by ChEMBL
Peking Union Medical College and Chinese Academy of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 1.11E+3nMAssay Description:Competitive inhibition of his-tagged recombinant mouse Keap1 KELCH domain (321 to 609 residues) expressed in Escherichia coli BL21 DE3/Nrf2 incubated...More data for this Ligand-Target Pair
Ligand Info
TargetNuclear factor erythroid 2-related factor 2(Mouse)
Peking Union Medical College and Chinese Academy of Medical Sciences
Curated by ChEMBL
Peking Union Medical College and Chinese Academy of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 1.11E+3nMAssay Description:Competitive inhibition of his-tagged recombinant mouse Keap1 KELCH domain (321 to 609 residues) expressed in Escherichia coli BL21 DE3/Nrf2 incubated...More data for this Ligand-Target Pair
Ligand Info
TargetNuclear factor erythroid 2-related factor 2(Mouse)
Peking Union Medical College and Chinese Academy of Medical Sciences
Curated by ChEMBL
Peking Union Medical College and Chinese Academy of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 1.58E+3nMAssay Description:Competitive inhibition of his-tagged recombinant mouse Keap1 KELCH domain (321 to 609 residues) expressed in Escherichia coli BL21 DE3/Nrf2 incubated...More data for this Ligand-Target Pair
Ligand Info
TargetNuclear factor erythroid 2-related factor 2(Mouse)
Peking Union Medical College and Chinese Academy of Medical Sciences
Curated by ChEMBL
Peking Union Medical College and Chinese Academy of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 2.33E+3nMAssay Description:Competitive inhibition of his-tagged recombinant mouse Keap1 KELCH domain (321 to 609 residues) expressed in Escherichia coli BL21 DE3/Nrf2 incubated...More data for this Ligand-Target Pair
Ligand Info
TargetNuclear factor erythroid 2-related factor 2(Mouse)
Peking Union Medical College and Chinese Academy of Medical Sciences
Curated by ChEMBL
Peking Union Medical College and Chinese Academy of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 2.35E+3nMAssay Description:Competitive inhibition of his-tagged recombinant mouse Keap1 KELCH domain (321 to 609 residues) expressed in Escherichia coli BL21 DE3/Nrf2 incubated...More data for this Ligand-Target Pair
Ligand Info
TargetNuclear factor erythroid 2-related factor 2(Mouse)
Peking Union Medical College and Chinese Academy of Medical Sciences
Curated by ChEMBL
Peking Union Medical College and Chinese Academy of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 3.63E+3nMAssay Description:Competitive inhibition of his-tagged recombinant mouse Keap1 KELCH domain (321 to 609 residues) expressed in Escherichia coli BL21 DE3/Nrf2 incubated...More data for this Ligand-Target Pair
Ligand Info
TargetNuclear factor erythroid 2-related factor 2(Mouse)
Peking Union Medical College and Chinese Academy of Medical Sciences
Curated by ChEMBL
Peking Union Medical College and Chinese Academy of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 3.63E+3nMAssay Description:Competitive inhibition of his-tagged recombinant mouse Keap1 KELCH domain (321 to 609 residues) expressed in Escherichia coli BL21 DE3/Nrf2 incubated...More data for this Ligand-Target Pair
Ligand Info
TargetNuclear factor erythroid 2-related factor 2(Mouse)
Peking Union Medical College and Chinese Academy of Medical Sciences
Curated by ChEMBL
Peking Union Medical College and Chinese Academy of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 8.18E+3nMAssay Description:Competitive inhibition of his-tagged recombinant mouse Keap1 KELCH domain (321 to 609 residues) expressed in Escherichia coli BL21 DE3/Nrf2 incubated...More data for this Ligand-Target Pair
Ligand Info
TargetNuclear factor erythroid 2-related factor 2(Mouse)
Peking Union Medical College and Chinese Academy of Medical Sciences
Curated by ChEMBL
Peking Union Medical College and Chinese Academy of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 8.34E+3nMAssay Description:Competitive inhibition of his-tagged recombinant mouse Keap1 KELCH domain (321 to 609 residues) expressed in Escherichia coli BL21 DE3/Nrf2 incubated...More data for this Ligand-Target Pair
Ligand Info
TargetNuclear factor erythroid 2-related factor 2(Mouse)
Peking Union Medical College and Chinese Academy of Medical Sciences
Curated by ChEMBL
Peking Union Medical College and Chinese Academy of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 1.29E+4nMAssay Description:Competitive inhibition of his-tagged recombinant mouse Keap1 KELCH domain (321 to 609 residues) expressed in Escherichia coli BL21 DE3/Nrf2 incubated...More data for this Ligand-Target Pair
Ligand Info
TargetNuclear factor erythroid 2-related factor 2(Mouse)
Peking Union Medical College and Chinese Academy of Medical Sciences
Curated by ChEMBL
Peking Union Medical College and Chinese Academy of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 1.42E+4nMAssay Description:Competitive inhibition of his-tagged recombinant mouse Keap1 KELCH domain (321 to 609 residues) expressed in Escherichia coli BL21 DE3/Nrf2 incubated...More data for this Ligand-Target Pair
TargetNuclear factor erythroid 2-related factor 2(Mouse)
Peking Union Medical College and Chinese Academy of Medical Sciences
Curated by ChEMBL
Peking Union Medical College and Chinese Academy of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 1.76E+4nMAssay Description:Competitive inhibition of his-tagged recombinant mouse Keap1 KELCH domain (321 to 609 residues) expressed in Escherichia coli BL21 DE3/Nrf2 incubated...More data for this Ligand-Target Pair
Ligand Info









































