Compile Data Set for Download or QSAR
Report error Found 14 Enz. Inhib. hit(s) with all data for entry = 50023500
LigandChemical structure of BindingDB Monomer ID 50336640BDBM50336640((nifedipine) 2,6-Dimethyl-4-(2-nitro-phenyl)-1,4-d...)
Affinity DataIC50: 40nMAssay Description:Antagonist activity at Cav1.2 (unknown origin) stably expressed in HEK293 cells assessed as inhibition of LTCC current by Whole cell patch clamp assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed
TargetVoltage-gated L-type calcium channel(Human)
KU Leuven

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50336640BDBM50336640((nifedipine) 2,6-Dimethyl-4-(2-nitro-phenyl)-1,4-d...)
Affinity DataIC50: 369nMAssay Description:Antagonist activity at L-type calcium channel in Ca1520-loade human SH-SY5Y cells assessed as inhibition of KCL-mediated depolarization of cytosolic ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed
LigandChemical structure of BindingDB Monomer ID 50664309BDBM50664309(CHEMBL6164841)
Affinity DataIC50: 650nMAssay Description:Antagonist activity at Cav1.2 (unknown origin) stably expressed in HEK293 cells assessed as inhibition of LTCC current by Whole cell patch clamp assa...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed
LigandChemical structure of BindingDB Monomer ID 50664314BDBM50664314(CHEMBL6174562)
Affinity DataIC50: 1.07E+3nMAssay Description:Antagonist activity at Cav1.2 (unknown origin) stably expressed in HEK293 cells assessed as inhibition of LTCC current by Whole cell patch clamp assa...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed
TargetVoltage-gated L-type calcium channel(Human)
KU Leuven

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50664309BDBM50664309(CHEMBL6164841)
Affinity DataIC50: 1.08E+3nMAssay Description:Antagonist activity at L-type calcium channel in Ca1520-loade human SH-SY5Y cells assessed as inhibition of KCL-mediated depolarization of cytosolic ...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed
LigandChemical structure of BindingDB Monomer ID 50664315BDBM50664315(CHEMBL6173085)
Affinity DataIC50: 1.51E+3nMAssay Description:Antagonist activity at Cav1.2 (unknown origin) stably expressed in HEK293 cells assessed as inhibition of LTCC current by Whole cell patch clamp assa...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed
LigandChemical structure of BindingDB Monomer ID 50664312BDBM50664312(CHEMBL6171808)
Affinity DataIC50: 1.90E+3nMAssay Description:Antagonist activity at Cav1.2 (unknown origin) stably expressed in HEK293 cells assessed as inhibition of LTCC current by Whole cell patch clamp assa...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed
LigandChemical structure of BindingDB Monomer ID 50664313BDBM50664313(CHEMBL6161363)
Affinity DataIC50: 2.20E+3nMAssay Description:Antagonist activity at Cav1.2 (unknown origin) stably expressed in HEK293 cells assessed as inhibition of LTCC current by Whole cell patch clamp assa...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed
LigandChemical structure of BindingDB Monomer ID 50664310BDBM50664310(CHEMBL6168209)
Affinity DataIC50: 3.50E+3nMAssay Description:Antagonist activity at Cav1.2 (unknown origin) stably expressed in HEK293 cells assessed as inhibition of LTCC current by Whole cell patch clamp assa...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed
LigandChemical structure of BindingDB Monomer ID 50664305BDBM50664305(CHEMBL6163410)
Affinity DataIC50: 4.25E+3nMAssay Description:Antagonist activity at Cav1.2 (unknown origin) stably expressed in HEK293 cells assessed as inhibition of LTCC current by Whole cell patch clamp assa...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed
LigandChemical structure of BindingDB Monomer ID 50664308BDBM50664308(CHEMBL6160836)
Affinity DataIC50: 6.53E+3nMAssay Description:Antagonist activity at Cav1.2 (unknown origin) stably expressed in HEK293 cells assessed as inhibition of LTCC current by Whole cell patch clamp assa...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed
LigandChemical structure of BindingDB Monomer ID 50664307BDBM50664307(CHEMBL6169116)
Affinity DataIC50: 7.48E+3nMAssay Description:Antagonist activity at Cav1.2 (unknown origin) stably expressed in HEK293 cells assessed as inhibition of LTCC current by Whole cell patch clamp assa...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed
LigandChemical structure of BindingDB Monomer ID 50664306BDBM50664306(CHEMBL6163708)
Affinity DataIC50: 1.25E+4nMAssay Description:Antagonist activity at Cav1.2 (unknown origin) stably expressed in HEK293 cells assessed as inhibition of LTCC current by Whole cell patch clamp assa...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed
LigandChemical structure of BindingDB Monomer ID 50664311BDBM50664311(CHEMBL6162404)
Affinity DataIC50: 1.27E+4nMAssay Description:Antagonist activity at Cav1.2 (unknown origin) stably expressed in HEK293 cells assessed as inhibition of LTCC current by Whole cell patch clamp assa...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed