Report error Found 56 Enz. Inhib. hit(s) with all data for entry = 50022828
TargetPlatelet-derived growth factor receptor alpha(Human)
Arromax Pharmatech Co. Ltd.
Curated by ChEMBL
Arromax Pharmatech Co. Ltd.
Curated by ChEMBL
Affinity DataIC50: 0.180nMAssay Description:Inhibition of 20S constitutive proteasome beta 2 trypsin-like activity (unknown origin) by cell based ABPP assayMore data for this Ligand-Target Pair
Ligand Info
TargetPlatelet-derived growth factor receptor alpha(Human)
Arromax Pharmatech Co. Ltd.
Curated by ChEMBL
Arromax Pharmatech Co. Ltd.
Curated by ChEMBL
Affinity DataIC50: 0.220nMAssay Description:Inhibition of 20S constitutive proteasome beta 2 trypsin-like activity (unknown origin) by cell based ABPP assayMore data for this Ligand-Target Pair
Ligand Info
TargetPlatelet-derived growth factor receptor alpha(Human)
Arromax Pharmatech Co. Ltd.
Curated by ChEMBL
Arromax Pharmatech Co. Ltd.
Curated by ChEMBL
Affinity DataIC50: 0.280nMAssay Description:Inhibition of 20S immunoproteasome beta 2 (unknown origin) by cell based ABPP assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 0.330nMAssay Description:Agonist activity at human A2B adenosine receptor by cell based assayMore data for this Ligand-Target Pair
Ligand Info
TargetVascular endothelial growth factor receptor 3(Human)
Arromax Pharmatech Co. Ltd.
Curated by ChEMBL
Arromax Pharmatech Co. Ltd.
Curated by ChEMBL
Affinity DataIC50: 0.560nMAssay Description:Agonist activity at FXR (unknown origin) by cell based assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 0.590nMAssay Description:Inhibition of IDO1 (unknown origin) by cell-based assayMore data for this Ligand-Target Pair
Ligand Info
TargetVascular endothelial growth factor receptor 2(Human)
Arromax Pharmatech Co. Ltd.
Curated by ChEMBL
Arromax Pharmatech Co. Ltd.
Curated by ChEMBL
Affinity DataIC50: 0.600nMAssay Description:Inhibition of BACE1 (unknown origin) assessed as reduction in amyloidbeta 40 level after 24 hrs by cell-based sandwich ELISAMore data for this Ligand-Target Pair
Ligand Info
TargetVascular endothelial growth factor receptor 3(Human)
Arromax Pharmatech Co. Ltd.
Curated by ChEMBL
Arromax Pharmatech Co. Ltd.
Curated by ChEMBL
Affinity DataIC50: 0.670nMAssay Description:Inhibition TRKA (unknown origin) by cell based assayMore data for this Ligand-Target Pair
Ligand Info
TargetVascular endothelial growth factor receptor 3(Human)
Arromax Pharmatech Co. Ltd.
Curated by ChEMBL
Arromax Pharmatech Co. Ltd.
Curated by ChEMBL
Affinity DataIC50: 0.680nMAssay Description:Agonist activity at FXR (unknown origin) by cell based assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 0.730nMAssay Description:Agonist activity at human A2B adenosine receptor by cell based assayMore data for this Ligand-Target Pair
Ligand Info
TargetPlatelet-derived growth factor receptor beta(Human)
Arromax Pharmatech Co. Ltd.
Curated by ChEMBL
Arromax Pharmatech Co. Ltd.
Curated by ChEMBL
Affinity DataIC50: 0.890nMAssay Description:Inhibition of 20S immunoproteasome beta 2 (unknown origin) by cell based ABPP assayMore data for this Ligand-Target Pair
Ligand Info
TargetVascular endothelial growth factor receptor 2(Human)
Arromax Pharmatech Co. Ltd.
Curated by ChEMBL
Arromax Pharmatech Co. Ltd.
Curated by ChEMBL
Affinity DataIC50: 1nMAssay Description:Inhibition of BACE1 (unknown origin) assessed as reduction in amyloidbeta 40 level after 24 hrs by cell-based sandwich ELISAMore data for this Ligand-Target Pair
Ligand Info
TargetVascular endothelial growth factor receptor 2(Human)
Arromax Pharmatech Co. Ltd.
Curated by ChEMBL
Arromax Pharmatech Co. Ltd.
Curated by ChEMBL
Affinity DataIC50: 1nMAssay Description:Inhibition of JAK1 (unknown origin) by cell based assayMore data for this Ligand-Target Pair
Ligand Info
TargetVascular endothelial growth factor receptor 3(Human)
Arromax Pharmatech Co. Ltd.
Curated by ChEMBL
Arromax Pharmatech Co. Ltd.
Curated by ChEMBL
Affinity DataIC50: 1.10nMAssay Description:Agonist activity at TAS2R14 (unknown origin) by stably expressed cell-based assayMore data for this Ligand-Target Pair
Ligand Info
TargetVascular endothelial growth factor receptor 3(Human)
Arromax Pharmatech Co. Ltd.
Curated by ChEMBL
Arromax Pharmatech Co. Ltd.
Curated by ChEMBL
Affinity DataIC50: 1.20nMAssay Description:Agonist activity at FXR (unknown origin) by cell based assayMore data for this Ligand-Target Pair
Ligand Info
TargetVascular endothelial growth factor receptor 2(Human)
Arromax Pharmatech Co. Ltd.
Curated by ChEMBL
Arromax Pharmatech Co. Ltd.
Curated by ChEMBL
Affinity DataIC50: 1.20nMAssay Description:Inhibition of BACE1 (unknown origin) by cell-based assayMore data for this Ligand-Target Pair
Ligand Info
TargetVascular endothelial growth factor receptor 2(Human)
Arromax Pharmatech Co. Ltd.
Curated by ChEMBL
Arromax Pharmatech Co. Ltd.
Curated by ChEMBL
Affinity DataIC50: 1.20nMAssay Description:Inhibition of BACE1 (unknown origin) assessed as reduction in amyloidbeta 40 level after 24 hrs by cell-based sandwich ELISAMore data for this Ligand-Target Pair
Ligand Info
TargetPlatelet-derived growth factor receptor beta(Human)
Arromax Pharmatech Co. Ltd.
Curated by ChEMBL
Arromax Pharmatech Co. Ltd.
Curated by ChEMBL
Affinity DataIC50: 1.20nMAssay Description:Inhibition of 20S constitutive proteasome beta 2 trypsin-like activity (unknown origin) by cell based ABPP assayMore data for this Ligand-Target Pair
Ligand Info
TargetPlatelet-derived growth factor receptor beta(Human)
Arromax Pharmatech Co. Ltd.
Curated by ChEMBL
Arromax Pharmatech Co. Ltd.
Curated by ChEMBL
Affinity DataIC50: 1.30nMAssay Description:Inhibition of 20S immunoproteasome beta 2 (unknown origin) by cell based ABPP assayMore data for this Ligand-Target Pair
Ligand Info
TargetVascular endothelial growth factor receptor 3(Human)
Arromax Pharmatech Co. Ltd.
Curated by ChEMBL
Arromax Pharmatech Co. Ltd.
Curated by ChEMBL
Affinity DataIC50: 1.40nMAssay Description:Agonist activity at FXR (unknown origin) by cell based assayMore data for this Ligand-Target Pair
Ligand Info
TargetVascular endothelial growth factor receptor 1(Human)
Arromax Pharmatech Co. Ltd.
Curated by ChEMBL
Arromax Pharmatech Co. Ltd.
Curated by ChEMBL
Affinity DataIC50: 1.60nMAssay Description:Inhibition of human Nav1.5 at -50 mV holding potential by cell-based IonWorks barracuda automated electrophysiology methodMore data for this Ligand-Target Pair
Ligand Info
TargetVascular endothelial growth factor receptor 1(Human)
Arromax Pharmatech Co. Ltd.
Curated by ChEMBL
Arromax Pharmatech Co. Ltd.
Curated by ChEMBL
Affinity DataIC50: 1.60nMAssay Description:Inhibition of human Nav1.5 at -50 mV holding potential by cell-based IonWorks barracuda automated electrophysiology methodMore data for this Ligand-Target Pair
Ligand Info
TargetVascular endothelial growth factor receptor 2(Human)
Arromax Pharmatech Co. Ltd.
Curated by ChEMBL
Arromax Pharmatech Co. Ltd.
Curated by ChEMBL
Affinity DataIC50: 1.70nMAssay Description:Inhibition of BACE1 (unknown origin) by cell-based assayMore data for this Ligand-Target Pair
Ligand Info
TargetVascular endothelial growth factor receptor 1(Human)
Arromax Pharmatech Co. Ltd.
Curated by ChEMBL
Arromax Pharmatech Co. Ltd.
Curated by ChEMBL
Affinity DataIC50: 2nMAssay Description:Inhibition of human Nav1.7 at -60 mV holding potential by cell-based IonWorks barracuda automated electrophysiology methodMore data for this Ligand-Target Pair
Ligand Info
TargetPlatelet-derived growth factor receptor alpha(Human)
Arromax Pharmatech Co. Ltd.
Curated by ChEMBL
Arromax Pharmatech Co. Ltd.
Curated by ChEMBL
Affinity DataIC50: 2nMAssay Description:Inhibition of 20S immunoproteasome beta 2 (unknown origin) by cell based ABPP assayMore data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 1(Human)
Arromax Pharmatech Co. Ltd.
Curated by ChEMBL
Arromax Pharmatech Co. Ltd.
Curated by ChEMBL
Affinity DataIC50: 2nMAssay Description:Inhibition of human Nav1.7 at -60 mV holding potential by cell-based IonWorks barracuda automated electrophysiology methodMore data for this Ligand-Target Pair
Ligand Info
TargetVascular endothelial growth factor receptor 3(Human)
Arromax Pharmatech Co. Ltd.
Curated by ChEMBL
Arromax Pharmatech Co. Ltd.
Curated by ChEMBL
Affinity DataIC50: 2.20nMAssay Description:Inhibition TRKA (unknown origin) by cell based assayMore data for this Ligand-Target Pair
Ligand Info
TargetVascular endothelial growth factor receptor 3(Human)
Arromax Pharmatech Co. Ltd.
Curated by ChEMBL
Arromax Pharmatech Co. Ltd.
Curated by ChEMBL
Affinity DataIC50: 2.60nMAssay Description:Agonist activity at TAS2R1 (unknown origin) by stably expressed cell-based assayMore data for this Ligand-Target Pair
Ligand Info
TargetVascular endothelial growth factor receptor 2(Human)
Arromax Pharmatech Co. Ltd.
Curated by ChEMBL
Arromax Pharmatech Co. Ltd.
Curated by ChEMBL
Affinity DataIC50: 3.20nMAssay Description:Inhibition of BACE1 (unknown origin) by cell-based assayMore data for this Ligand-Target Pair
Ligand Info
TargetVascular endothelial growth factor receptor 1(Human)
Arromax Pharmatech Co. Ltd.
Curated by ChEMBL
Arromax Pharmatech Co. Ltd.
Curated by ChEMBL
Affinity DataIC50: 3.80nMAssay Description:Inhibition of human Nav1.7 at -60 mV holding potential by cell-based manual patch clamp electrophysiology methodMore data for this Ligand-Target Pair
Ligand Info
TargetVascular endothelial growth factor receptor 1(Human)
Arromax Pharmatech Co. Ltd.
Curated by ChEMBL
Arromax Pharmatech Co. Ltd.
Curated by ChEMBL
Affinity DataIC50: 5.70nMAssay Description:Inhibition of human Nav1.5 at -50 mV holding potential by cell-based IonWorks barracuda automated electrophysiology methodMore data for this Ligand-Target Pair
Ligand Info
TargetVascular endothelial growth factor receptor 1(Human)
Arromax Pharmatech Co. Ltd.
Curated by ChEMBL
Arromax Pharmatech Co. Ltd.
Curated by ChEMBL
Affinity DataIC50: 5.80nMAssay Description:Inhibition of human Nav1.5 at -50 mV holding potential by cell-based IonWorks barracuda automated electrophysiology methodMore data for this Ligand-Target Pair
Ligand Info
TargetVascular endothelial growth factor receptor 2(Human)
Arromax Pharmatech Co. Ltd.
Curated by ChEMBL
Arromax Pharmatech Co. Ltd.
Curated by ChEMBL
Affinity DataIC50: 6.5nMAssay Description:Inhibition of BACE1 (unknown origin) assessed as reduction in amyloidbeta 40 level after 24 hrs by cell-based sandwich ELISAMore data for this Ligand-Target Pair
Ligand Info
TargetVascular endothelial growth factor receptor 1(Human)
Arromax Pharmatech Co. Ltd.
Curated by ChEMBL
Arromax Pharmatech Co. Ltd.
Curated by ChEMBL
Affinity DataIC50: 9.5nMAssay Description:Inhibition of human Nav1.7 at -60 mV holding potential by cell-based IonWorks barracuda automated electrophysiology methodMore data for this Ligand-Target Pair
Ligand Info
TargetVascular endothelial growth factor receptor 2(Human)
Arromax Pharmatech Co. Ltd.
Curated by ChEMBL
Arromax Pharmatech Co. Ltd.
Curated by ChEMBL
Affinity DataIC50: 11nMAssay Description:Inhibition of BACE1 (unknown origin) by cell-based assayMore data for this Ligand-Target Pair
TargetPlatelet-derived growth factor receptor alpha(Human)
Arromax Pharmatech Co. Ltd.
Curated by ChEMBL
Arromax Pharmatech Co. Ltd.
Curated by ChEMBL
Affinity DataIC50: 11nMAssay Description:Inhibition of 20S immunoproteasome beta 2 (unknown origin) by cell based ABPP assayMore data for this Ligand-Target Pair
Ligand Info
TargetVascular endothelial growth factor receptor 3(Human)
Arromax Pharmatech Co. Ltd.
Curated by ChEMBL
Arromax Pharmatech Co. Ltd.
Curated by ChEMBL
Affinity DataIC50: 11nMAssay Description:Inhibition of OGA (unknown origin) by cell based assayMore data for this Ligand-Target Pair
TargetPlatelet-derived growth factor receptor beta(Human)
Arromax Pharmatech Co. Ltd.
Curated by ChEMBL
Arromax Pharmatech Co. Ltd.
Curated by ChEMBL
Affinity DataIC50: 12nMAssay Description:Inhibition of 20S immunoproteasome beta 2 (unknown origin) by cell based ABPP assayMore data for this Ligand-Target Pair
Ligand Info
TargetVascular endothelial growth factor receptor 2(Human)
Arromax Pharmatech Co. Ltd.
Curated by ChEMBL
Arromax Pharmatech Co. Ltd.
Curated by ChEMBL
Affinity DataIC50: 14nMAssay Description:Inhibition of BACE1 (unknown origin) assessed as reduction in amyloidbeta 40 level after 24 hrs by cell-based sandwich ELISAMore data for this Ligand-Target Pair
Ligand Info
TargetPlatelet-derived growth factor receptor beta(Human)
Arromax Pharmatech Co. Ltd.
Curated by ChEMBL
Arromax Pharmatech Co. Ltd.
Curated by ChEMBL
Affinity DataIC50: 17nMAssay Description:Inhibition of 20S immunoproteasome beta 2 (unknown origin) by cell based ABPP assayMore data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 3(Human)
Arromax Pharmatech Co. Ltd.
Curated by ChEMBL
Arromax Pharmatech Co. Ltd.
Curated by ChEMBL
Affinity DataIC50: 18nMAssay Description:Agonist activity at FXR (unknown origin) by cell based assayMore data for this Ligand-Target Pair
Ligand Info
TargetVascular endothelial growth factor receptor 1(Human)
Arromax Pharmatech Co. Ltd.
Curated by ChEMBL
Arromax Pharmatech Co. Ltd.
Curated by ChEMBL
Affinity DataIC50: 19nMAssay Description:Inhibition of JAK2 (unknown origin) by cell based assayMore data for this Ligand-Target Pair
Affinity DataIC50: 22nMAssay Description:Inhibition of 20S constitutive proteasome beta 2 trypsin-like activity (unknown origin) by cell based ABPP assayMore data for this Ligand-Target Pair
Ligand Info
TargetVascular endothelial growth factor receptor 1(Human)
Arromax Pharmatech Co. Ltd.
Curated by ChEMBL
Arromax Pharmatech Co. Ltd.
Curated by ChEMBL
Affinity DataIC50: 42nMAssay Description:Inhibition of human Nav1.5 at -50 mV holding potential by cell-based IonWorks barracuda automated electrophysiology methodMore data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 56nMAssay Description:Inhibition of 20S immunoproteasome beta 2 (unknown origin) by cell based ABPP assayMore data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 2(Human)
Arromax Pharmatech Co. Ltd.
Curated by ChEMBL
Arromax Pharmatech Co. Ltd.
Curated by ChEMBL
Affinity DataIC50: 79nMAssay Description:Inhibition of BACE1 (unknown origin) by cell-based assayMore data for this Ligand-Target Pair
Ligand Info
TargetVascular endothelial growth factor receptor 3(Human)
Arromax Pharmatech Co. Ltd.
Curated by ChEMBL
Arromax Pharmatech Co. Ltd.
Curated by ChEMBL
Affinity DataIC50: 87nMAssay Description:Inhibition of MPS1 (unknown origin) by cell based assayMore data for this Ligand-Target Pair
Ligand Info
TargetVascular endothelial growth factor receptor 1(Human)
Arromax Pharmatech Co. Ltd.
Curated by ChEMBL
Arromax Pharmatech Co. Ltd.
Curated by ChEMBL
Affinity DataIC50: 96nMAssay Description:Inhibition of human Nav1.5 at -50 mV holding potential by cell-based IonWorks barracuda automated electrophysiology methodMore data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 109nMAssay Description:Inhibition of 20S immunoproteasome beta 2 (unknown origin) by cell based ABPP assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 129nMAssay Description:Inhibition of 20S constitutive proteasome beta 2 trypsin-like activity (unknown origin) by cell based ABPP assayMore data for this Ligand-Target Pair
Ligand Info









3D Structure (crystal)


