Report error Found 90 Enz. Inhib. hit(s) with all data for entry = 50022820
Affinity DataIC50: 8.5nMAssay Description:Inhibition of IRAK4 (unknown origin) by cell based assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 22nMAssay Description:Inhibition of IRAK4 (unknown origin) by cell based assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 23nMAssay Description:Inhibition of IRAK4 (unknown origin) by cell based assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 26nMAssay Description:Inhibition of IRAK4 (unknown origin) by cell based assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 31nMAssay Description:Inhibition of IRAK4 (unknown origin) by cell based assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 50nMAssay Description:Inhibition of IRAK4 (unknown origin) by cell based assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 60nMAssay Description:Inhibition of IRAK4 (unknown origin) by cell based assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 73nMAssay Description:Inhibition of IRAK4 (unknown origin) by cell based assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 87nMAssay Description:Inhibition of IRAK4 (unknown origin) by cell based assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 91nMAssay Description:Inhibition of IRAK4 (unknown origin) by cell based assayMore data for this Ligand-Target Pair
Affinity DataIC50: 95nMAssay Description:Antagonist activity at human thyroid stimulating hormone receptor expressed in rat HTC133 cells assessed as reduction in agonist-induced cAMP product...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 127nMAssay Description:Inhibition of MAP4K4 (unknown origin) by cell based assayMore data for this Ligand-Target Pair
Affinity DataIC50: 155nMAssay Description:Negative allosteric modulation of human luteinizing hormone receptor assessed as reduction in glycoprotein human luteinizing hormone-induced agonist ...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 238nMAssay Description:Negative allosteric modulation of human luteinizing hormone receptor assessed as reduction in Org 43553-induced agonist activity preincubated for 20 ...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 264nMAssay Description:Antagonist activity at human luteinizing hormone receptor assessed as reduction in agonist-induced cAMP production preincubated for 20 mins followed ...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 339nMAssay Description:Inhibition of NS5A in HCV genotype 2a JFH-1 by cell based luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 360nMAssay Description:Antagonist activity at luteinizing hormone receptor in mouse MLTC-1 cells assessed as reduction in agonist-induced cAMP production preincubated for 3...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 366nMAssay Description:Antagonist activity at human luteinizing hormone receptor assessed as reduction in agonist-induced cAMP production preincubated for 20 mins followed ...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 426nMAssay Description:Inhibition of NS5A in HCV genotype 3a by cell based luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 490nMAssay Description:Inhibition of IRAK4 (unknown origin) by cell based assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 501nMAssay Description:Antagonist activity at human luteinizing hormone receptor assessed as reduction in agonist-induced cAMP production preincubated for 20 mins followed ...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 517nMAssay Description:Antagonist activity at human luteinizing hormone receptor assessed as reduction in agonist-induced cAMP production preincubated for 20 mins followed ...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 593nMAssay Description:Antagonist activity at human luteinizing hormone receptor assessed as reduction in agonist-induced cAMP production preincubated for 20 mins followed ...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 650nMAssay Description:Antagonist activity at human luteinizing hormone receptor assessed as reduction in agonist-induced cAMP production preincubated for 20 mins followed ...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 662nMAssay Description:Antagonist activity at human luteinizing hormone receptor assessed as reduction in agonist-induced cAMP production preincubated for 20 mins followed ...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 662nMAssay Description:Antagonist activity at human luteinizing hormone receptor assessed as reduction in agonist-induced cAMP production preincubated for 20 mins followed ...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 684nMAssay Description:Inhibition of Gal4-tagged RORbeta LBD (unknown origin) by cell based luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 685nMAssay Description:Antagonist activity at human luteinizing hormone receptor assessed as reduction in agonist-induced cAMP production preincubated for 20 mins followed ...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 687nMAssay Description:Antagonist activity at human follicle stimulating hormone receptor assessed as reduction in agonist-induced cAMP production preincubated for 20 mins ...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 695nMAssay Description:Antagonist activity at human follicle stimulating hormone receptor assessed as reduction in agonist-induced cAMP production preincubated for 20 mins ...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 727nMAssay Description:Inhibition of IRAK4 (unknown origin) by cell based assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 743nMAssay Description:Antagonist activity at human luteinizing hormone receptor assessed as reduction in agonist-induced cAMP production preincubated for 20 mins followed ...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 752nMAssay Description:Inhibition of IRAK4 (unknown origin) by cell based assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 878nMAssay Description:Antagonist activity at human follicle stimulating hormone receptor assessed as reduction in agonist-induced cAMP production preincubated for 20 mins ...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 890nMAssay Description:Antagonist activity at human luteinizing hormone receptor assessed as reduction in agonist-induced cAMP production preincubated for 20 mins followed ...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 974nMAssay Description:Antagonist activity at human luteinizing hormone receptor assessed as reduction in agonist-induced cAMP production preincubated for 20 mins followed ...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of IRAK4 (unknown origin) by cell based assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 1.24E+3nMAssay Description:Antagonist activity at human luteinizing hormone receptor assessed as reduction in agonist-induced cAMP production preincubated for 20 mins followed ...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 1.24E+3nMAssay Description:Antagonist activity at human luteinizing hormone receptor assessed as reduction in agonist-induced cAMP production preincubated for 20 mins followed ...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 1.27E+3nMAssay Description:Antagonist activity at human luteinizing hormone receptor assessed as reduction in agonist-induced cAMP production preincubated for 20 mins followed ...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 1.27E+3nMAssay Description:Antagonist activity at human luteinizing hormone receptor assessed as reduction in agonist-induced cAMP production preincubated for 20 mins followed ...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 1.35E+3nMAssay Description:Antagonist activity at human luteinizing hormone receptor assessed as reduction in agonist-induced cAMP production preincubated for 20 mins followed ...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 1.38E+3nMAssay Description:Antagonist activity at human luteinizing hormone receptor assessed as reduction in agonist-induced cAMP production preincubated for 20 mins followed ...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 1.39E+3nMAssay Description:Antagonist activity at human luteinizing hormone receptor assessed as reduction in agonist-induced cAMP production preincubated for 20 mins followed ...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 1.40E+3nMAssay Description:Antagonist activity at rat luteinizing hormone receptor expressed in rat ovary granulosa GLHR15 cell suspension assessed as reduction in agonist-indu...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 1.51E+3nMAssay Description:Antagonist activity at human luteinizing hormone receptor assessed as reduction in agonist-induced cAMP production preincubated for 20 mins followed ...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 1.55E+3nMAssay Description:Antagonist activity at human luteinizing hormone receptor assessed as reduction in agonist-induced cAMP production preincubated for 20 mins followed ...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 1.67E+3nMAssay Description:Antagonist activity at human follicle stimulating hormone receptor assessed as reduction in agonist-induced cAMP production preincubated for 20 mins ...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 1.75E+3nMAssay Description:Negative allosteric modulation of human luteinizing hormone receptor assessed as reduction in glycoprotein human luteinizing hormone-induced agonist ...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 1.81E+3nMAssay Description:Antagonist activity at cynomolgus monkey luteinizing hormone receptor expressed in HEK293 cells assessed as reduction in agonist-induced cAMP product...More data for this Ligand-Target Pair
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