Compile Data Set for Download or QSAR
Report error Found 35 Enz. Inhib. hit(s) with all data for entry = 50022685
TargetGlutamyl aminopeptidase(Mus musculus)
Quantum Genomics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50633859BDBM50633859(CHEMBL6101922)
Affinity DataIC50: 1nMAssay Description:Modulation of rat mGlu5 receptor assessed as calcium mobilization by cell based fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2026
Entry Details
PubMed
TargetGlutamyl aminopeptidase(Mus musculus)
Quantum Genomics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50633836BDBM50633836(CHEMBL6091985)
Affinity DataIC50: 4nMAssay Description:Negative allosteric modulation of rat mGlu3 receptor assessed as calcium mobilization by cell based fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2026
Entry Details
PubMed
TargetGlutamyl aminopeptidase(Mus musculus)
Quantum Genomics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50633862BDBM50633862(CHEMBL6091920)
Affinity DataIC50: 7nMAssay Description:Negative allosteric modulation of rat mGlu3 receptor assessed as calcium mobilization by cell based fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2026
Entry Details
PubMed
TargetGlutamyl aminopeptidase(Mus musculus)
Quantum Genomics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50633852BDBM50633852(CHEMBL6132685)
Affinity DataIC50: 9nMAssay Description:Modulation of rat mGlu5 receptor assessed as calcium mobilization by cell based fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2026
Entry Details
PubMed
TargetGlutamyl aminopeptidase(Mus musculus)
Quantum Genomics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50633858BDBM50633858(CHEMBL6078602)
Affinity DataIC50: 9nMAssay Description:Modulation of rat mGlu5 receptor assessed as calcium mobilization by cell based fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2026
Entry Details
PubMed
TargetGlutamyl aminopeptidase(Mus musculus)
Quantum Genomics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50633844BDBM50633844(CHEMBL6134529)
Affinity DataIC50: 10nMAssay Description:Modulation of rat mGlu5 receptor assessed as calcium mobilization by cell based fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2026
Entry Details
PubMed
TargetGlutamyl aminopeptidase(Mus musculus)
Quantum Genomics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50633857BDBM50633857(CHEMBL6141870)
Affinity DataIC50: 10nMAssay Description:Modulation of rat mGlu5 receptor assessed as calcium mobilization by cell based fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2026
Entry Details
PubMed
TargetGlutamyl aminopeptidase(Mus musculus)
Quantum Genomics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50633846BDBM50633846(CHEMBL6144468)
Affinity DataIC50: 18nMAssay Description:Modulation of rat mGlu5 receptor assessed as calcium mobilization by cell based fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2026
Entry Details
PubMed
TargetGlutamyl aminopeptidase(Mus musculus)
Quantum Genomics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50633861BDBM50633861(CHEMBL6102273)
Affinity DataIC50: 21nMAssay Description:Modulation of rat mGlu5 receptor assessed as calcium mobilization by cell based fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2026
Entry Details
PubMed
TargetGlutamyl aminopeptidase(Mus musculus)
Quantum Genomics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50633849BDBM50633849(CHEMBL6083014)
Affinity DataIC50: 21nMAssay Description:Modulation of rat mGlu5 receptor assessed as calcium mobilization by cell based fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2026
Entry Details
PubMed
TargetGlutamyl aminopeptidase(Mus musculus)
Quantum Genomics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50633848BDBM50633848(CHEMBL6142075)
Affinity DataIC50: 23nMAssay Description:Modulation of rat mGlu5 receptor assessed as calcium mobilization by cell based fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2026
Entry Details
PubMed
TargetGlutamyl aminopeptidase(Mus musculus)
Quantum Genomics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50633854BDBM50633854(CHEMBL6096566)
Affinity DataIC50: 24nMAssay Description:Modulation of rat mGlu5 receptor assessed as calcium mobilization by cell based fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2026
Entry Details
PubMed
TargetGlutamyl aminopeptidase(Mus musculus)
Quantum Genomics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50633851BDBM50633851(CHEMBL6145942)
Affinity DataIC50: 26nMAssay Description:Modulation of rat mGlu5 receptor assessed as calcium mobilization by cell based fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2026
Entry Details
PubMed
TargetGlutamyl aminopeptidase(Mus musculus)
Quantum Genomics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50633856BDBM50633856(CHEMBL6149319)
Affinity DataIC50: 26nMAssay Description:Modulation of rat mGlu5 receptor assessed as calcium mobilization by cell based fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2026
Entry Details
PubMed
TargetGlutamyl aminopeptidase(Mus musculus)
Quantum Genomics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50633847BDBM50633847(CHEMBL6147420)
Affinity DataIC50: 27nMAssay Description:Modulation of rat mGlu5 receptor assessed as calcium mobilization by cell based fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2026
Entry Details
PubMed
TargetGlutamyl aminopeptidase(Mus musculus)
Quantum Genomics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50633853BDBM50633853(CHEMBL6078318)
Affinity DataIC50: 28nMAssay Description:Modulation of rat mGlu5 receptor assessed as calcium mobilization by cell based fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2026
Entry Details
PubMed
TargetGlutamyl aminopeptidase(Mus musculus)
Quantum Genomics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50633839BDBM50633839(CHEMBL6120447)
Affinity DataIC50: 29nMAssay Description:Modulation of rat mGlu5 receptor assessed as calcium mobilization by cell based fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2026
Entry Details
PubMed
TargetGlutamyl aminopeptidase(Mus musculus)
Quantum Genomics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50633863BDBM50633863(CHEMBL6114886)
Affinity DataIC50: 30nMAssay Description:Negative allosteric modulation of rat mGlu3 receptor assessed as calcium mobilization by cell based fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2026
Entry Details
PubMed
TargetGlutamyl aminopeptidase(Mus musculus)
Quantum Genomics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50633840BDBM50633840(CHEMBL6146273)
Affinity DataIC50: 39nMAssay Description:Modulation of rat mGlu5 receptor assessed as calcium mobilization by cell based fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2026
Entry Details
PubMed
TargetGlutamyl aminopeptidase(Mus musculus)
Quantum Genomics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50633845BDBM50633845(CHEMBL6120664)
Affinity DataIC50: 41nMAssay Description:Modulation of rat mGlu5 receptor assessed as calcium mobilization by cell based fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2026
Entry Details
PubMed
TargetGlutamyl aminopeptidase(Mus musculus)
Quantum Genomics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50633860BDBM50633860(CHEMBL6083078)
Affinity DataIC50: 42nMAssay Description:Modulation of rat mGlu5 receptor assessed as calcium mobilization by cell based fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2026
Entry Details
PubMed
TargetGlutamyl aminopeptidase(Mus musculus)
Quantum Genomics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50633841BDBM50633841(CHEMBL6144088)
Affinity DataIC50: 54nMAssay Description:Modulation of rat mGlu5 receptor assessed as calcium mobilization by cell based fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2026
Entry Details
PubMed
TargetGlutamyl aminopeptidase(Mus musculus)
Quantum Genomics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50633855BDBM50633855(CHEMBL6091792)
Affinity DataIC50: 54nMAssay Description:Modulation of rat mGlu5 receptor assessed as calcium mobilization by cell based fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2026
Entry Details
PubMed
TargetGlutamyl aminopeptidase(Mus musculus)
Quantum Genomics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50633850BDBM50633850(CHEMBL6134712)
Affinity DataIC50: 61nMAssay Description:Modulation of rat mGlu5 receptor assessed as calcium mobilization by cell based fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2026
Entry Details
PubMed
TargetAminopeptidase N(Pig)
Quantum Genomics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50036824BDBM50036824((S)-4-Amino-5-mercapto-pentanoic acid | (S)-3-Carb...)
Affinity DataKi:  120nMAssay Description:Modulation of rat mGlu5 receptor assessed as calcium mobilization by cell based fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2026
Entry Details
PubMed
TargetGlutamyl aminopeptidase(Mus musculus)
Quantum Genomics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50633837BDBM50633837(CHEMBL6145468)
Affinity DataIC50: 310nMAssay Description:Modulation of rat mGlu5 receptor assessed as calcium mobilization by cell based fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2026
Entry Details
PubMed
TargetGlutamyl aminopeptidase(Mus musculus)
Quantum Genomics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50633864BDBM50633864(CHEMBL6132894)
Affinity DataIC50: 420nMAssay Description:Negative allosteric modulation of rat mGlu3 receptor assessed as calcium mobilization by cell based fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2026
Entry Details
PubMed
TargetGlutamyl aminopeptidase(Mus musculus)
Quantum Genomics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50633843BDBM50633843(CHEMBL6083031)
Affinity DataIC50: 660nMAssay Description:Modulation of rat mGlu5 receptor assessed as calcium mobilization by cell based fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2026
Entry Details
PubMed
TargetGlutamyl aminopeptidase(Mus musculus)
Quantum Genomics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50633834BDBM50633834(Ec33)
Affinity DataIC50: 710nMAssay Description:Modulation of rat mGlu5 receptor assessed as calcium mobilization by cell based fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2026
Entry Details
PubMed
TargetGlutamyl aminopeptidase(Mus musculus)
Quantum Genomics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50633842BDBM50633842(CHEMBL6101975)
Affinity DataIC50: 930nMAssay Description:Modulation of rat mGlu5 receptor assessed as calcium mobilization by cell based fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2026
Entry Details
PubMed
TargetGlutamyl aminopeptidase(Mus musculus)
Quantum Genomics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50633838BDBM50633838(CHEMBL6102762)
Affinity DataIC50: 5.40E+3nMAssay Description:Modulation of rat mGlu5 receptor assessed as calcium mobilization by cell based fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2026
Entry Details
PubMed
TargetAminopeptidase N(Human)
Quantum Genomics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50633835BDBM50633835(CHEMBL6142196)
Affinity DataKi: >1.00E+4nMAssay Description:Modulation of rat mGlu5 receptor assessed as calcium mobilization by cell based fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2026
Entry Details
PubMed
TargetAminopeptidase N(Human)
Quantum Genomics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50633833BDBM50633833(CHEMBL6120409)
Affinity DataKi:  1.60E+4nMAssay Description:Modulation of rat mGlu5 receptor assessed as calcium mobilization by cell based fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2026
Entry Details
PubMed
TargetAminopeptidase N(Human)
Quantum Genomics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50633836BDBM50633836(CHEMBL6091985)
Affinity DataIC50: 2.00E+4nMAssay Description:Modulation of rat mGlu5 receptor assessed as calcium mobilization by cell based fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2026
Entry Details
PubMed
TargetAminopeptidase N(Pig)
Quantum Genomics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50633834BDBM50633834(Ec33)
Affinity DataKi:  2.50E+4nMAssay Description:Modulation of rat mGlu5 receptor assessed as calcium mobilization by cell based fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2026
Entry Details
PubMed