Report error Found 12 Enz. Inhib. hit(s) with all data for entry = 50022817
TargetAmyloid-beta precursor protein(Human)
East China University of Science and Technology
Curated by ChEMBL
East China University of Science and Technology
Curated by ChEMBL
Affinity DataKd: 1nMAssay Description:Inhibition of gamma secretase (unknown origin)-mediated notch processing by cell based assayMore data for this Ligand-Target Pair
Ligand Info
TargetAmyloid-beta precursor protein(Human)
East China University of Science and Technology
Curated by ChEMBL
East China University of Science and Technology
Curated by ChEMBL
Affinity DataKd: 13nMAssay Description:Agonist activity at human PPARalpha assessed as induction of transactivation activity by cell based assayMore data for this Ligand-Target Pair
Ligand Info
TargetAmyloid-beta precursor protein(Human)
East China University of Science and Technology
Curated by ChEMBL
East China University of Science and Technology
Curated by ChEMBL
Affinity DataKd: 27nMAssay Description:Agonist activity at human PPARgamma assessed as induction of transactivation activity by cell based assayMore data for this Ligand-Target Pair
Ligand Info
TargetAmyloid-beta precursor protein(Human)
East China University of Science and Technology
Curated by ChEMBL
East China University of Science and Technology
Curated by ChEMBL
Affinity DataKd: 28nMAssay Description:Agonist activity at human PPARgamma assessed as induction of transactivation activity by cell based assayMore data for this Ligand-Target Pair
Ligand Info
TargetAmyloid-beta precursor protein(Human)
East China University of Science and Technology
Curated by ChEMBL
East China University of Science and Technology
Curated by ChEMBL
Affinity DataKd: 45nMAssay Description:Agonist activity at human PPARalpha assessed as induction of transactivation activity by cell based assayMore data for this Ligand-Target Pair
Ligand Info
TargetAmyloid-beta precursor protein(Human)
East China University of Science and Technology
Curated by ChEMBL
East China University of Science and Technology
Curated by ChEMBL
Affinity DataKd: 59nMAssay Description:Inhibition of gamma secretase (unknown origin)-mediated notch processing by cell based assayMore data for this Ligand-Target Pair
Ligand Info
TargetAmyloid-beta precursor protein(Human)
East China University of Science and Technology
Curated by ChEMBL
East China University of Science and Technology
Curated by ChEMBL
Affinity DataKd: 86nMAssay Description:Agonist activity at human PPARgamma assessed as induction of transactivation activity by cell based assayMore data for this Ligand-Target Pair
Ligand Info
TargetAmyloid-beta precursor protein(Human)
East China University of Science and Technology
Curated by ChEMBL
East China University of Science and Technology
Curated by ChEMBL
Affinity DataKd: 117nMAssay Description:Agonist activity at human PPARalpha assessed as induction of transactivation activity by cell based assayMore data for this Ligand-Target Pair
Ligand Info
TargetAmyloid-beta precursor protein(Human)
East China University of Science and Technology
Curated by ChEMBL
East China University of Science and Technology
Curated by ChEMBL
Affinity DataKd: 170nMAssay Description:Agonist activity at human PPARgamma assessed as induction of transactivation activity by cell based assayMore data for this Ligand-Target Pair
Ligand Info
TargetAmyloid-beta precursor protein(Human)
East China University of Science and Technology
Curated by ChEMBL
East China University of Science and Technology
Curated by ChEMBL
Affinity DataKd: 374nMAssay Description:Inhibition of gamma secretase (unknown origin)-mediated amyloid beta (1 to 42) production by cell based assayMore data for this Ligand-Target Pair
Ligand Info
TargetAmyloid-beta precursor protein(Human)
East China University of Science and Technology
Curated by ChEMBL
East China University of Science and Technology
Curated by ChEMBL
Affinity DataKd: 506nMAssay Description:Inhibition of gamma secretase (unknown origin)-mediated amyloid beta (1 to 40) production by cell based assayMore data for this Ligand-Target Pair
Ligand Info
TargetAmyloid-beta precursor protein(Human)
East China University of Science and Technology
Curated by ChEMBL
East China University of Science and Technology
Curated by ChEMBL
Affinity DataKd: 548nMAssay Description:Agonist activity at human PPARalpha assessed as induction of transactivation activity by cell based assayMore data for this Ligand-Target Pair
Ligand Info










