Compile Data Set for Download or QSAR
Report error Found 13 Enz. Inhib. hit(s) with all data for entry = 50023452
TargetSerine-protein kinase ATM(Human)
Sichuan Academy of Medical Sciences & Sichuan Provincial People's Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 155083BDBM155083(US9000153, 36)
Affinity DataIC50: 0.25nMAssay Description:Inhibition of ATM (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed
TargetSerine-protein kinase ATM(Human)
Sichuan Academy of Medical Sciences & Sichuan Provincial People's Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50571459BDBM50571459(CHEMBL4872830)
Affinity DataKi:  1nMAssay Description:Binding affinity to ATM (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed
TargetSerine-protein kinase ATM(Human)
Sichuan Academy of Medical Sciences & Sichuan Provincial People's Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50550657BDBM50550657(CHEMBL4792737)
Affinity DataIC50: 5nMAssay Description:Inhibition of full length human recombinant Flag-tagged ATMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed
TargetSerine-protein kinase ATM(Human)
Sichuan Academy of Medical Sciences & Sichuan Provincial People's Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50059640BDBM50059640(CHEMBL2140173)
Affinity DataIC50: 6.30nMAssay Description:Inhibition of ATM (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed
TargetSerine-protein kinase ATM(Human)
Sichuan Academy of Medical Sciences & Sichuan Provincial People's Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50565800BDBM50565800(Azd-1390 | Azd1390 | US20240294545, Compound AZD13...)
Affinity DataIC50: 7.80nMAssay Description:Inhibition of ATM (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed
TargetSerine-protein kinase ATM(Human)
Sichuan Academy of Medical Sciences & Sichuan Provincial People's Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50208517BDBM50208517(KU-55933 | 2-morpholin-4-yl-6-thianthren-1-yl-pyra...)
Affinity DataIC50: 13nMAssay Description:Inhibition of ATM in human HeLa cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetSerine-protein kinase ATM(Human)
Sichuan Academy of Medical Sciences & Sichuan Provincial People's Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50378201BDBM50378201(CHEMBL4159350)
Affinity DataIC50: 13nMAssay Description:Inhibition of ATM in human HeLa cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed
TargetSerine-protein kinase ATM(Human)
Sichuan Academy of Medical Sciences & Sichuan Provincial People's Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50604005BDBM50604005(CHEMBL5178407)
Affinity DataIC50: 310nMAssay Description:Inhibition of ATM (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed
TargetSerine-protein kinase ATM(Human)
Sichuan Academy of Medical Sciences & Sichuan Provincial People's Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50145038BDBM50145038(CHEMBL2143829)
Affinity DataIC50: 400nMAssay Description:Inhibition of recombinant GST-tagged full length ATM (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed
TargetSerine/threonine-protein kinase ATR(Human)
Sichuan Academy of Medical Sciences & Sichuan Provincial People's Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 27461BDBM27461(2-amino-5-(4-fluorophenyl)-N-methyl-3-[4-(pyrrolid...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of ATR (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed
TargetSerine/threonine-protein kinase mTOR(Human)
Sichuan Academy of Medical Sciences & Sichuan Provincial People's Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50378201BDBM50378201(CHEMBL4159350)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of mTOR (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed
TargetSerine-protein kinase ATM(Human)
Sichuan Academy of Medical Sciences & Sichuan Provincial People's Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50604006BDBM50604006(CHEMBL2094953 | DNDI1417761)
Affinity DataIC50: 3.34E+4nMAssay Description:Inhibition of ATM (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed
TargetSerine/threonine-protein kinase ATR(Human)
Sichuan Academy of Medical Sciences & Sichuan Provincial People's Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50378201BDBM50378201(CHEMBL4159350)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of ATR (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed