Compile Data Set for Download or QSAR
Report error Found 17 Enz. Inhib. hit(s) with all data for entry = 50011115
TargetInterleukin-1 receptor-associated kinase 4(Human)
Kymera Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50253994BDBM50253994(CHEMBL6092071)
Affinity DataIC50: 0.5nMAssay Description:Inhibition of ROCK2 assessed as myosin light chain phosphorylation by cell-based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/2/2026
Entry Details ArticlePubMed
TargetInterleukin-1 receptor-associated kinase 4(Human)
Kymera Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50254000BDBM50254000(CHEMBL6102395)
Affinity DataIC50: 4nMAssay Description:Inhibition of Huntingtin protein aggregation by cell based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/2/2026
Entry Details ArticlePubMed
TargetInterleukin-1 receptor-associated kinase 4(Human)
Kymera Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50254011BDBM50254011(CHEMBL6078355)
Affinity DataIC50: 12nMAssay Description:Inhibition of Huntingtin protein aggregation by cell based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/2/2026
Entry Details ArticlePubMed
TargetInterleukin-1 receptor-associated kinase 4(Human)
Kymera Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50253995BDBM50253995(CHEMBL6078441)
Affinity DataIC50: 13nMAssay Description:Inhibition of ROCK2 assessed as myosin light chain phosphorylation by cell-based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/2/2026
Entry Details ArticlePubMed
TargetInterleukin-1 receptor-associated kinase 4(Human)
Kymera Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50254012BDBM50254012(CHEMBL6102976)
Affinity DataIC50: 20nMAssay Description:Inhibition of Huntingtin protein aggregation by cell based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/2/2026
Entry Details ArticlePubMed
TargetInterleukin-1 receptor-associated kinase 4(Human)
Kymera Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50254004BDBM50254004(CHEMBL6114897)
Affinity DataIC50: 30nMAssay Description:Inhibition of Huntingtin protein aggregation by cell based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/2/2026
Entry Details ArticlePubMed
TargetInterleukin-1 receptor-associated kinase 4(Human)
Kymera Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50254009BDBM50254009(CHEMBL6078173)
Affinity DataIC50: 35nMAssay Description:Inhibition of Huntingtin protein aggregation by cell based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/2/2026
Entry Details ArticlePubMed
TargetInterleukin-1 receptor-associated kinase 4(Human)
Kymera Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50254008BDBM50254008(Kt-474 | SAR-444656 | SAR444656)
Affinity DataIC50: 41nMAssay Description:Inhibition of Huntingtin protein aggregation by cell based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/2/2026
Entry Details ArticlePubMed
TargetInterleukin-1 receptor-associated kinase 4(Human)
Kymera Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50254007BDBM50254007(CHEMBL6134203)
Affinity DataIC50: 43nMAssay Description:Inhibition of Huntingtin protein aggregation by cell based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/2/2026
Entry Details ArticlePubMed
TargetInterleukin-1 receptor-associated kinase 4(Human)
Kymera Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50254003BDBM50254003(CHEMBL6082887)
Affinity DataIC50: 48nMAssay Description:Inhibition of Huntingtin protein aggregation by cell based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/2/2026
Entry Details ArticlePubMed
TargetInterleukin-1 receptor-associated kinase 4(Human)
Kymera Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50253993BDBM50253993(CHEMBL6120263)
Affinity DataIC50: 58nMAssay Description:Inhibition of ROCK2 assessed as myosin light chain phosphorylation by cell-based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/2/2026
Entry Details ArticlePubMed
TargetInterleukin-1 receptor-associated kinase 4(Human)
Kymera Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50254001BDBM50254001(CHEMBL6120670)
Affinity DataIC50: 61nMAssay Description:Inhibition of Huntingtin protein aggregation by cell based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/2/2026
Entry Details ArticlePubMed
TargetInterleukin-1 receptor-associated kinase 4(Human)
Kymera Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50254002BDBM50254002(CHEMBL6078548)
Affinity DataIC50: 70nMAssay Description:Inhibition of Huntingtin protein aggregation by cell based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/2/2026
Entry Details ArticlePubMed
TargetInterleukin-1 receptor-associated kinase 4(Human)
Kymera Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50254005BDBM50254005(CHEMBL6102392)
Affinity DataIC50: 71nMAssay Description:Inhibition of Huntingtin protein aggregation by cell based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/2/2026
Entry Details ArticlePubMed
TargetInterleukin-1 receptor-associated kinase 4(Human)
Kymera Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50254010BDBM50254010(CHEMBL6102351)
Affinity DataIC50: 170nMAssay Description:Inhibition of Huntingtin protein aggregation by cell based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/2/2026
Entry Details ArticlePubMed
TargetInterleukin-1 receptor-associated kinase 4(Human)
Kymera Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50253999BDBM50253999(CHEMBL6078489)
Affinity DataIC50: 200nMAssay Description:Inhibition of ROCK2 assessed as myosin light chain phosphorylation by cell-based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/2/2026
Entry Details ArticlePubMed
TargetInterleukin-1 receptor-associated kinase 4(Human)
Kymera Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50253998BDBM50253998(CHEMBL6120604)
Affinity DataIC50: 970nMAssay Description:Inhibition of ROCK2 assessed as myosin light chain phosphorylation by cell-based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/2/2026
Entry Details ArticlePubMed