Compile Data Set for Download or QSAR
Report error Found 10 Enz. Inhib. hit(s) with all data for entry = 50004509
TargetSerine/threonine-protein kinase LATS2(Human)
Zhengzhou University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50213704BDBM50213704(CHEMBL6082870)
Affinity DataIC50: 0.520nMAssay Description:Displacement of [3H]-diprenorphine from human mu opioid receptor after 120 mins by cell based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/2/2026
Entry Details ArticlePubMed
TargetSerine/threonine-protein kinase LATS1(Human)
Zhengzhou University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50213704BDBM50213704(CHEMBL6082870)
Affinity DataIC50: 0.760nMAssay Description:Inhibition of DGAT1 (unknown origin) by cell-based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/2/2026
Entry Details ArticlePubMed
TargetHepatocyte growth factor-like protein(Human)
Zhengzhou University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50059277BDBM50059277(CHEMBL3393348 | US9156845, 4)
Affinity DataIC50: 34nMAssay Description:Inhibition of DGAT1 (unknown origin) by cell-based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/2/2026
Entry Details ArticlePubMed
TargetSerine/threonine-protein kinase 3(Human)
Zhengzhou University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50059277BDBM50059277(CHEMBL3393348 | US9156845, 4)
Affinity DataIC50: 76nMAssay Description:Inhibition of DGAT1 (unknown origin) by cell-based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/2/2026
Entry Details ArticlePubMed
TargetTranscriptional enhancer factor TEF-3(Human)
Zhengzhou University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50626281BDBM50626281(CHEMBL5397201)
Affinity DataIC50: 672nMAssay Description:Displacement of [3H]-diprenorphine from human mu opioid receptor after 120 mins by cell based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/2/2026
Entry Details ArticlePubMed
TargetTranscriptional enhancer factor TEF-4(Human)
Zhengzhou University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50626281BDBM50626281(CHEMBL5397201)
Affinity DataIC50: 710nMAssay Description:Displacement of [3H]-diprenorphine from human mu opioid receptor after 120 mins by cell based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/2/2026
Entry Details ArticlePubMedPDB3D3D Structure (crystal)
TargetTranscriptional enhancer factor TEF-3(Human)
Zhengzhou University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50213705BDBM50213705(CHEMBL6077986)
Affinity DataIC50: 1.30E+3nMAssay Description:Displacement of [3H]-diprenorphine from human mu opioid receptor after 120 mins by cell based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/2/2026
Entry Details ArticlePubMed
TargetTranscriptional coactivator YAP1(Homo sapiens)
Zhengzhou University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50547126BDBM50547126(CHEMBL4763473)
Affinity DataEC50:  4.30E+3nMAssay Description:Displacement of [3H]-diprenorphine from human mu opioid receptor after 120 mins by cell based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/2/2026
Entry Details ArticlePubMed
LigandChemical structure of BindingDB Monomer ID 50547126BDBM50547126(CHEMBL4763473)
Affinity DataEC50:  5.90E+3nMAssay Description:Displacement of [3H]-diprenorphine from human mu opioid receptor after 120 mins by cell based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/2/2026
Entry Details ArticlePubMed
TargetTranscriptional enhancer factor TEF-4(Human)
Zhengzhou University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 17636BDBM17636(2-{[3-(trifluoromethyl)phenyl]amino}benzoic acid |...)
Affinity DataKd:  7.30E+4nMAssay Description:Displacement of [3H]-diprenorphine from human mu opioid receptor after 120 mins by cell based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/2/2026
Entry Details ArticlePubMedPDB3D3D Structure (crystal)