BindingDB Reactant_set_id	Ligand SMILES	Ligand InChI	Ligand InChI Key	BindingDB MonomerID	BindingDB Ligand Name	Target Name	Target Source Organism According to Curator or DataSource	Ki (nM)	IC50 (nM)	Kd (nM)	EC50 (nM)	kon (M-1-s-1)	koff (s-1)	pH	Temp (C)	Curation/DataSource	Article DOI	BindingDB Entry DOI	PMID	PubChem AID	Patent Number	Authors	Institution	Link to Ligand in BindingDB	Link to Target in BindingDB	Link to Ligand-Target Pair in BindingDB	Ligand HET ID in PDB	PDB ID(s) for Ligand-Target Complex	PubChem CID of Ligand	PubChem SID of Ligand	ChEBI ID of Ligand	ChEMBL ID of Ligand	DrugBank ID of Ligand	IUPHAR_GRAC ID of Ligand	KEGG ID of Ligand	ZINC ID of Ligand	Number of Protein Chains in Target (>1 implies a multichain complex)	BindingDB Target Chain Sequence	PDB ID(s) of Target Chain	UniProt (SwissProt) Recommended Name of Target Chain	UniProt (SwissProt) Entry Name of Target Chain	UniProt (SwissProt) Primary ID of Target Chain	UniProt (SwissProt) Secondary ID(s) of Target Chain	UniProt (SwissProt) Alternative ID(s) of Target Chain	UniProt (TrEMBL) Submitted Name of Target Chain	UniProt (TrEMBL) Entry Name of Target Chain	UniProt (TrEMBL) Primary ID of Target Chain	UniProt (TrEMBL) Secondary ID(s) of Target Chain	UniProt (TrEMBL) Alternative ID(s) of Target Chain
339377	N#C\C=C\c1ccc(cc1)-c1ccncc1	InChI=1S/C14H10N2/c15-9-1-2-12-3-5-13(6-4-12)14-7-10-16-11-8-14/h1-8,10-11H/b2-1+	PCFKTRCTTGIQLS-OWOJBTEDSA-N	259826	US9505766, 30	Ribosomal protein S6 kinase alpha-3 [399-740]			>300000					8	22.00 C	US Patent		10.7270/Q2639NPR		aid1803661	US9505766	Taunton, Jr., JW; Maglathlin, R; Serafimova, I; Cohen, MS; Miller, R; Paavilainen, V; McFarland, J; Krishnan, S	The Regents of the University of California	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=259826	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=11170&target=Ribosomal+protein+S6+kinase+alpha-3+%5B399-740%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=259826&enzyme=Ribosomal+protein+S6+kinase+alpha-3+%5B399-740%5D&column=ki&startPg=0&Increment=50&submit=Search			89403409	350084520							1	MQTVGVHSIVQQLHRNSIQFTDGYEVKEDIGVGSYSVCKRCIHKATNMEFAVKIIDKSKRDPTEEIEILLRYGQHPNIITLKDVYDDGKYVYVVTELMKGGELLDKILRQKFFSEREASAVLFTITKTVEYLHAQGVVHRDLKPSNILYVDESGNPESIRICDFGFAKQLRAENGLLMTPCYTANFVAPEVLKRQGYDAACDIWSLGVLLYTMLTGYTPFANGPDDTPEEILARIGSGKFSLSGGYWNSVSDTAKDLVSKMLHVDPHQRLTAALVLRHPWIVHWDQLPQYQLNRQDAPHLVKGAMAATYSALNRNQSPVLEPVGRSTLAQRRGIKKITSTAL		Ribosomal protein S6 kinase alpha-3	KS6A3_HUMAN	P51812	B2R9V4 Q4VAP3 Q59H26 Q5JPK8 Q7Z3Z7						
452873	CC(=O)\C=C\c1c(-c2ccc(C)cc2)c2c(N)ncnc2n1CCCO	InChI=1S/C20H22N4O2/c1-13-4-7-15(8-5-13)17-16(9-6-14(2)26)24(10-3-11-25)20-18(17)19(21)22-12-23-20/h4-9,12,25H,3,10-11H2,1-2H3,(H2,21,22,23)/b9-6+	JUIPXPYGIKPHFM-RMKNXTFCSA-N	259802	US9505766, Me enone (1)	Ribosomal protein S6 kinase alpha-3 [399-740]			 87					8	22.00 C	US Patent		10.7270/Q2639NPR		aid1803661	US9505766	Taunton, Jr., JW; Maglathlin, R; Serafimova, I; Cohen, MS; Miller, R; Paavilainen, V; McFarland, J; Krishnan, S	The Regents of the University of California	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=259802	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=11170&target=Ribosomal+protein+S6+kinase+alpha-3+%5B399-740%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=259802&enzyme=Ribosomal+protein+S6+kinase+alpha-3+%5B399-740%5D&column=ki&startPg=0&Increment=50&submit=Search			57856455	350084496							1	MQTVGVHSIVQQLHRNSIQFTDGYEVKEDIGVGSYSVCKRCIHKATNMEFAVKIIDKSKRDPTEEIEILLRYGQHPNIITLKDVYDDGKYVYVVTELMKGGELLDKILRQKFFSEREASAVLFTITKTVEYLHAQGVVHRDLKPSNILYVDESGNPESIRICDFGFAKQLRAENGLLMTPCYTANFVAPEVLKRQGYDAACDIWSLGVLLYTMLTGYTPFANGPDDTPEEILARIGSGKFSLSGGYWNSVSDTAKDLVSKMLHVDPHQRLTAALVLRHPWIVHWDQLPQYQLNRQDAPHLVKGAMAATYSALNRNQSPVLEPVGRSTLAQRRGIKKITSTAL		Ribosomal protein S6 kinase alpha-3	KS6A3_HUMAN	P51812	B2R9V4 Q4VAP3 Q59H26 Q5JPK8 Q7Z3Z7						
452874	COC(=O)\C=C\c1c(-c2ccc(C)cc2)c2c(N)ncnc2n1CCCO	InChI=1S/C20H22N4O3/c1-13-4-6-14(7-5-13)17-15(8-9-16(26)27-2)24(10-3-11-25)20-18(17)19(21)22-12-23-20/h4-9,12,25H,3,10-11H2,1-2H3,(H2,21,22,23)/b9-8+	SUWNTOBZXIAHKB-CMDGGOBGSA-N	259804	US9505766, Me acrylate (2)	Ribosomal protein S6 kinase alpha-3 [399-740]			 250					8	22.00 C	US Patent		10.7270/Q2639NPR		aid1803661	US9505766	Taunton, Jr., JW; Maglathlin, R; Serafimova, I; Cohen, MS; Miller, R; Paavilainen, V; McFarland, J; Krishnan, S	The Regents of the University of California	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=259804	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=11170&target=Ribosomal+protein+S6+kinase+alpha-3+%5B399-740%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=259804&enzyme=Ribosomal+protein+S6+kinase+alpha-3+%5B399-740%5D&column=ki&startPg=0&Increment=50&submit=Search			16662748	350084498							1	MQTVGVHSIVQQLHRNSIQFTDGYEVKEDIGVGSYSVCKRCIHKATNMEFAVKIIDKSKRDPTEEIEILLRYGQHPNIITLKDVYDDGKYVYVVTELMKGGELLDKILRQKFFSEREASAVLFTITKTVEYLHAQGVVHRDLKPSNILYVDESGNPESIRICDFGFAKQLRAENGLLMTPCYTANFVAPEVLKRQGYDAACDIWSLGVLLYTMLTGYTPFANGPDDTPEEILARIGSGKFSLSGGYWNSVSDTAKDLVSKMLHVDPHQRLTAALVLRHPWIVHWDQLPQYQLNRQDAPHLVKGAMAATYSALNRNQSPVLEPVGRSTLAQRRGIKKITSTAL		Ribosomal protein S6 kinase alpha-3	KS6A3_HUMAN	P51812	B2R9V4 Q4VAP3 Q59H26 Q5JPK8 Q7Z3Z7						
452875	Cc1ccc(cc1)-c1c(\C=C\C#N)n(CCCO)c2ncnc(N)c12	InChI=1S/C19H19N5O/c1-13-5-7-14(8-6-13)16-15(4-2-9-20)24(10-3-11-25)19-17(16)18(21)22-12-23-19/h2,4-8,12,25H,3,10-11H2,1H3,(H2,21,22,23)/b4-2+	LPADWFDQODOOMS-DUXPYHPUSA-N	259803	US9505766, acrylonitrile (3)	Ribosomal protein S6 kinase alpha-3 [399-740]			 750					8	22.00 C	US Patent		10.7270/Q2639NPR		aid1803661	US9505766	Taunton, Jr., JW; Maglathlin, R; Serafimova, I; Cohen, MS; Miller, R; Paavilainen, V; McFarland, J; Krishnan, S	The Regents of the University of California	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=259803	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=11170&target=Ribosomal+protein+S6+kinase+alpha-3+%5B399-740%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=259803&enzyme=Ribosomal+protein+S6+kinase+alpha-3+%5B399-740%5D&column=ki&startPg=0&Increment=50&submit=Search			56840684	350084497							1	MQTVGVHSIVQQLHRNSIQFTDGYEVKEDIGVGSYSVCKRCIHKATNMEFAVKIIDKSKRDPTEEIEILLRYGQHPNIITLKDVYDDGKYVYVVTELMKGGELLDKILRQKFFSEREASAVLFTITKTVEYLHAQGVVHRDLKPSNILYVDESGNPESIRICDFGFAKQLRAENGLLMTPCYTANFVAPEVLKRQGYDAACDIWSLGVLLYTMLTGYTPFANGPDDTPEEILARIGSGKFSLSGGYWNSVSDTAKDLVSKMLHVDPHQRLTAALVLRHPWIVHWDQLPQYQLNRQDAPHLVKGAMAATYSALNRNQSPVLEPVGRSTLAQRRGIKKITSTAL		Ribosomal protein S6 kinase alpha-3	KS6A3_HUMAN	P51812	B2R9V4 Q4VAP3 Q59H26 Q5JPK8 Q7Z3Z7						
452876	COC(=O)C(=C\c1c(-c2ccc(C)cc2)c2c(N)ncnc2n1CCCO)\C#N	InChI=1S/C21H21N5O3/c1-13-4-6-14(7-5-13)17-16(10-15(11-22)21(28)29-2)26(8-3-9-27)20-18(17)19(23)24-12-25-20/h4-7,10,12,27H,3,8-9H2,1-2H3,(H2,23,24,25)/b15-10+	GDXHZXJALWQIPQ-XNTDXEJSSA-N	259805	US9505766, CN-OMe (4)	Ribosomal protein S6 kinase alpha-3 [399-740]			 13					8	22.00 C	US Patent		10.7270/Q2639NPR		aid1803661	US9505766	Taunton, Jr., JW; Maglathlin, R; Serafimova, I; Cohen, MS; Miller, R; Paavilainen, V; McFarland, J; Krishnan, S	The Regents of the University of California	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=259805	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=11170&target=Ribosomal+protein+S6+kinase+alpha-3+%5B399-740%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=259805&enzyme=Ribosomal+protein+S6+kinase+alpha-3+%5B399-740%5D&column=ki&startPg=0&Increment=50&submit=Search			52938515	350084499							1	MQTVGVHSIVQQLHRNSIQFTDGYEVKEDIGVGSYSVCKRCIHKATNMEFAVKIIDKSKRDPTEEIEILLRYGQHPNIITLKDVYDDGKYVYVVTELMKGGELLDKILRQKFFSEREASAVLFTITKTVEYLHAQGVVHRDLKPSNILYVDESGNPESIRICDFGFAKQLRAENGLLMTPCYTANFVAPEVLKRQGYDAACDIWSLGVLLYTMLTGYTPFANGPDDTPEEILARIGSGKFSLSGGYWNSVSDTAKDLVSKMLHVDPHQRLTAALVLRHPWIVHWDQLPQYQLNRQDAPHLVKGAMAATYSALNRNQSPVLEPVGRSTLAQRRGIKKITSTAL		Ribosomal protein S6 kinase alpha-3	KS6A3_HUMAN	P51812	B2R9V4 Q4VAP3 Q59H26 Q5JPK8 Q7Z3Z7						
452877	Cc1ccc(cc1)-c1c(\C=C(/C#N)C(=O)OC(C)(C)C)n(CCCO)c2ncnc(N)c12	InChI=1S/C24H27N5O3/c1-15-6-8-16(9-7-15)19-18(12-17(13-25)23(31)32-24(2,3)4)29(10-5-11-30)22-20(19)21(26)27-14-28-22/h6-9,12,14,30H,5,10-11H2,1-4H3,(H2,26,27,28)/b17-12+	IEUOMYJAIZIKES-SFQUDFHCSA-N	259806	US9505766, CN-OtBu (5)	Ribosomal protein S6 kinase alpha-3 [399-740]			 7					8	22.00 C	US Patent		10.7270/Q2639NPR		aid1803661	US9505766	Taunton, Jr., JW; Maglathlin, R; Serafimova, I; Cohen, MS; Miller, R; Paavilainen, V; McFarland, J; Krishnan, S	The Regents of the University of California	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=259806	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=11170&target=Ribosomal+protein+S6+kinase+alpha-3+%5B399-740%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=259806&enzyme=Ribosomal+protein+S6+kinase+alpha-3+%5B399-740%5D&column=ki&startPg=0&Increment=50&submit=Search			52938516	350084500							1	MQTVGVHSIVQQLHRNSIQFTDGYEVKEDIGVGSYSVCKRCIHKATNMEFAVKIIDKSKRDPTEEIEILLRYGQHPNIITLKDVYDDGKYVYVVTELMKGGELLDKILRQKFFSEREASAVLFTITKTVEYLHAQGVVHRDLKPSNILYVDESGNPESIRICDFGFAKQLRAENGLLMTPCYTANFVAPEVLKRQGYDAACDIWSLGVLLYTMLTGYTPFANGPDDTPEEILARIGSGKFSLSGGYWNSVSDTAKDLVSKMLHVDPHQRLTAALVLRHPWIVHWDQLPQYQLNRQDAPHLVKGAMAATYSALNRNQSPVLEPVGRSTLAQRRGIKKITSTAL		Ribosomal protein S6 kinase alpha-3	KS6A3_HUMAN	P51812	B2R9V4 Q4VAP3 Q59H26 Q5JPK8 Q7Z3Z7						
452878	Cc1ccc(cc1)-c1c(\C=C(/C#N)C(N)=O)n(CCCO)c2ncnc(N)c12	InChI=1S/C20H20N6O2/c1-12-3-5-13(6-4-12)16-15(9-14(10-21)19(23)28)26(7-2-8-27)20-17(16)18(22)24-11-25-20/h3-6,9,11,27H,2,7-8H2,1H3,(H2,23,28)(H2,22,24,25)/b14-9+	SZAXHJXUPGRTIP-NTEUORMPSA-N	259807	US9505766, CN-NH2 (6)	Ribosomal protein S6 kinase alpha-3 [399-740]			 3					8	22.00 C	US Patent		10.7270/Q2639NPR		aid1803661	US9505766	Taunton, Jr., JW; Maglathlin, R; Serafimova, I; Cohen, MS; Miller, R; Paavilainen, V; McFarland, J; Krishnan, S	The Regents of the University of California	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=259807	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=11170&target=Ribosomal+protein+S6+kinase+alpha-3+%5B399-740%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=259807&enzyme=Ribosomal+protein+S6+kinase+alpha-3+%5B399-740%5D&column=ki&startPg=0&Increment=50&submit=Search			52938641	350084501							1	MQTVGVHSIVQQLHRNSIQFTDGYEVKEDIGVGSYSVCKRCIHKATNMEFAVKIIDKSKRDPTEEIEILLRYGQHPNIITLKDVYDDGKYVYVVTELMKGGELLDKILRQKFFSEREASAVLFTITKTVEYLHAQGVVHRDLKPSNILYVDESGNPESIRICDFGFAKQLRAENGLLMTPCYTANFVAPEVLKRQGYDAACDIWSLGVLLYTMLTGYTPFANGPDDTPEEILARIGSGKFSLSGGYWNSVSDTAKDLVSKMLHVDPHQRLTAALVLRHPWIVHWDQLPQYQLNRQDAPHLVKGAMAATYSALNRNQSPVLEPVGRSTLAQRRGIKKITSTAL		Ribosomal protein S6 kinase alpha-3	KS6A3_HUMAN	P51812	B2R9V4 Q4VAP3 Q59H26 Q5JPK8 Q7Z3Z7						
452879	CC(C)NC(=O)C(=C\c1c(-c2ccc(C)cc2)c2c(N)ncnc2n1CCCO)\C#N	InChI=1S/C23H26N6O2/c1-14(2)28-23(31)17(12-24)11-18-19(16-7-5-15(3)6-8-16)20-21(25)26-13-27-22(20)29(18)9-4-10-30/h5-8,11,13-14,30H,4,9-10H2,1-3H3,(H,28,31)(H2,25,26,27)/b17-11+	POTINGKLYOETSI-GZTJUZNOSA-N	259808	US9505766, 74::US9505766, CN-NHiPr (7)	Ribosomal protein S6 kinase alpha-3 [399-740]			 5					8	22.00 C	US Patent		10.7270/Q2639NPR		aid1803661	US9505766	Taunton, Jr., JW; Maglathlin, R; Serafimova, I; Cohen, MS; Miller, R; Paavilainen, V; McFarland, J; Krishnan, S	The Regents of the University of California	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=259808	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=11170&target=Ribosomal+protein+S6+kinase+alpha-3+%5B399-740%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=259808&enzyme=Ribosomal+protein+S6+kinase+alpha-3+%5B399-740%5D&column=ki&startPg=0&Increment=50&submit=Search			52938644	350084502							1	MQTVGVHSIVQQLHRNSIQFTDGYEVKEDIGVGSYSVCKRCIHKATNMEFAVKIIDKSKRDPTEEIEILLRYGQHPNIITLKDVYDDGKYVYVVTELMKGGELLDKILRQKFFSEREASAVLFTITKTVEYLHAQGVVHRDLKPSNILYVDESGNPESIRICDFGFAKQLRAENGLLMTPCYTANFVAPEVLKRQGYDAACDIWSLGVLLYTMLTGYTPFANGPDDTPEEILARIGSGKFSLSGGYWNSVSDTAKDLVSKMLHVDPHQRLTAALVLRHPWIVHWDQLPQYQLNRQDAPHLVKGAMAATYSALNRNQSPVLEPVGRSTLAQRRGIKKITSTAL		Ribosomal protein S6 kinase alpha-3	KS6A3_HUMAN	P51812	B2R9V4 Q4VAP3 Q59H26 Q5JPK8 Q7Z3Z7						
452880	Cc1ccc(cc1)-c1c(\C=C(/C#N)C(=O)NCc2ccccc2)n(CCCO)c2ncnc(N)c12	InChI=1S/C27H26N6O2/c1-18-8-10-20(11-9-18)23-22(33(12-5-13-34)26-24(23)25(29)31-17-32-26)14-21(15-28)27(35)30-16-19-6-3-2-4-7-19/h2-4,6-11,14,17,34H,5,12-13,16H2,1H3,(H,30,35)(H2,29,31,32)/b21-14+	VGLWJTYWGAMQMT-KGENOOAVSA-N	259809	US9505766, CN-NHBn (8)	Ribosomal protein S6 kinase alpha-3 [399-740]			 40					8	22.00 C	US Patent		10.7270/Q2639NPR		aid1803661	US9505766	Taunton, Jr., JW; Maglathlin, R; Serafimova, I; Cohen, MS; Miller, R; Paavilainen, V; McFarland, J; Krishnan, S	The Regents of the University of California	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=259809	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=11170&target=Ribosomal+protein+S6+kinase+alpha-3+%5B399-740%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=259809&enzyme=Ribosomal+protein+S6+kinase+alpha-3+%5B399-740%5D&column=ki&startPg=0&Increment=50&submit=Search			52938642	350084503							1	MQTVGVHSIVQQLHRNSIQFTDGYEVKEDIGVGSYSVCKRCIHKATNMEFAVKIIDKSKRDPTEEIEILLRYGQHPNIITLKDVYDDGKYVYVVTELMKGGELLDKILRQKFFSEREASAVLFTITKTVEYLHAQGVVHRDLKPSNILYVDESGNPESIRICDFGFAKQLRAENGLLMTPCYTANFVAPEVLKRQGYDAACDIWSLGVLLYTMLTGYTPFANGPDDTPEEILARIGSGKFSLSGGYWNSVSDTAKDLVSKMLHVDPHQRLTAALVLRHPWIVHWDQLPQYQLNRQDAPHLVKGAMAATYSALNRNQSPVLEPVGRSTLAQRRGIKKITSTAL		Ribosomal protein S6 kinase alpha-3	KS6A3_HUMAN	P51812	B2R9V4 Q4VAP3 Q59H26 Q5JPK8 Q7Z3Z7						
452888	NC(=O)C(=C\c1ccc(cc1)-c1ncnc2[nH]cnc12)\C#N	InChI=1S/C15H10N6O/c16-6-11(14(17)22)5-9-1-3-10(4-2-9)12-13-15(20-7-18-12)21-8-19-13/h1-5,7-8H,(H2,17,22)(H,18,19,20,21)/b11-5+	BRZWHXQQGAAXPX-VZUCSPMQSA-N	259810	US9505766, 10	Ribosomal protein S6 kinase alpha-3 [399-740]			 5000					8	22.00 C	US Patent		10.7270/Q2639NPR		aid1803661	US9505766	Taunton, Jr., JW; Maglathlin, R; Serafimova, I; Cohen, MS; Miller, R; Paavilainen, V; McFarland, J; Krishnan, S	The Regents of the University of California	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=259810	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=11170&target=Ribosomal+protein+S6+kinase+alpha-3+%5B399-740%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=259810&enzyme=Ribosomal+protein+S6+kinase+alpha-3+%5B399-740%5D&column=ki&startPg=0&Increment=50&submit=Search			52938775	350084504							1	MQTVGVHSIVQQLHRNSIQFTDGYEVKEDIGVGSYSVCKRCIHKATNMEFAVKIIDKSKRDPTEEIEILLRYGQHPNIITLKDVYDDGKYVYVVTELMKGGELLDKILRQKFFSEREASAVLFTITKTVEYLHAQGVVHRDLKPSNILYVDESGNPESIRICDFGFAKQLRAENGLLMTPCYTANFVAPEVLKRQGYDAACDIWSLGVLLYTMLTGYTPFANGPDDTPEEILARIGSGKFSLSGGYWNSVSDTAKDLVSKMLHVDPHQRLTAALVLRHPWIVHWDQLPQYQLNRQDAPHLVKGAMAATYSALNRNQSPVLEPVGRSTLAQRRGIKKITSTAL		Ribosomal protein S6 kinase alpha-3	KS6A3_HUMAN	P51812	B2R9V4 Q4VAP3 Q59H26 Q5JPK8 Q7Z3Z7						
452889	NC(=O)C(=C\c1ccc(cc1)-c1c[nH]c2ncccc12)\C#N	InChI=1S/C17H12N4O/c18-9-13(16(19)22)8-11-3-5-12(6-4-11)15-10-21-17-14(15)2-1-7-20-17/h1-8,10H,(H2,19,22)(H,20,21)/b13-8+	AENKGHPUTMOKKU-MDWZMJQESA-N	259811	US9505766, 11	Ribosomal protein S6 kinase alpha-3 [399-740]			<750					8	22.00 C	US Patent		10.7270/Q2639NPR		aid1803661	US9505766	Taunton, Jr., JW; Maglathlin, R; Serafimova, I; Cohen, MS; Miller, R; Paavilainen, V; McFarland, J; Krishnan, S	The Regents of the University of California	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=259811	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=11170&target=Ribosomal+protein+S6+kinase+alpha-3+%5B399-740%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=259811&enzyme=Ribosomal+protein+S6+kinase+alpha-3+%5B399-740%5D&column=ki&startPg=0&Increment=50&submit=Search			67206349	350084505							1	MQTVGVHSIVQQLHRNSIQFTDGYEVKEDIGVGSYSVCKRCIHKATNMEFAVKIIDKSKRDPTEEIEILLRYGQHPNIITLKDVYDDGKYVYVVTELMKGGELLDKILRQKFFSEREASAVLFTITKTVEYLHAQGVVHRDLKPSNILYVDESGNPESIRICDFGFAKQLRAENGLLMTPCYTANFVAPEVLKRQGYDAACDIWSLGVLLYTMLTGYTPFANGPDDTPEEILARIGSGKFSLSGGYWNSVSDTAKDLVSKMLHVDPHQRLTAALVLRHPWIVHWDQLPQYQLNRQDAPHLVKGAMAATYSALNRNQSPVLEPVGRSTLAQRRGIKKITSTAL		Ribosomal protein S6 kinase alpha-3	KS6A3_HUMAN	P51812	B2R9V4 Q4VAP3 Q59H26 Q5JPK8 Q7Z3Z7						
452890	NC(=O)C(=C\c1cccc(c1)C(=O)c1c[nH]c2ncccc12)\C#N	InChI=1S/C18H12N4O2/c19-9-13(17(20)24)8-11-3-1-4-12(7-11)16(23)15-10-22-18-14(15)5-2-6-21-18/h1-8,10H,(H2,20,24)(H,21,22)/b13-8+	CEPQIZUYOXYNFQ-MDWZMJQESA-N	259812	US9505766, 12	Ribosomal protein S6 kinase alpha-3 [399-740]			 124					8	22.00 C	US Patent		10.7270/Q2639NPR		aid1803661	US9505766	Taunton, Jr., JW; Maglathlin, R; Serafimova, I; Cohen, MS; Miller, R; Paavilainen, V; McFarland, J; Krishnan, S	The Regents of the University of California	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=259812	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=11170&target=Ribosomal+protein+S6+kinase+alpha-3+%5B399-740%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=259812&enzyme=Ribosomal+protein+S6+kinase+alpha-3+%5B399-740%5D&column=ki&startPg=0&Increment=50&submit=Search			52938387	350084506							1	MQTVGVHSIVQQLHRNSIQFTDGYEVKEDIGVGSYSVCKRCIHKATNMEFAVKIIDKSKRDPTEEIEILLRYGQHPNIITLKDVYDDGKYVYVVTELMKGGELLDKILRQKFFSEREASAVLFTITKTVEYLHAQGVVHRDLKPSNILYVDESGNPESIRICDFGFAKQLRAENGLLMTPCYTANFVAPEVLKRQGYDAACDIWSLGVLLYTMLTGYTPFANGPDDTPEEILARIGSGKFSLSGGYWNSVSDTAKDLVSKMLHVDPHQRLTAALVLRHPWIVHWDQLPQYQLNRQDAPHLVKGAMAATYSALNRNQSPVLEPVGRSTLAQRRGIKKITSTAL		Ribosomal protein S6 kinase alpha-3	KS6A3_HUMAN	P51812	B2R9V4 Q4VAP3 Q59H26 Q5JPK8 Q7Z3Z7						
452891	NC(=O)C(=C\c1ccc2[nH]ncc2c1)\C#N	InChI=1S/C11H8N4O/c12-5-8(11(13)16)3-7-1-2-10-9(4-7)6-14-15-10/h1-4,6H,(H2,13,16)(H,14,15)/b8-3+	JIMIDTDLZHFIJW-FPYGCLRLSA-N	259813	US9505766, 13	Ribosomal protein S6 kinase alpha-3 [399-740]			 250					8	22.00 C	US Patent		10.7270/Q2639NPR		aid1803661	US9505766	Taunton, Jr., JW; Maglathlin, R; Serafimova, I; Cohen, MS; Miller, R; Paavilainen, V; McFarland, J; Krishnan, S	The Regents of the University of California	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=259813	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=11170&target=Ribosomal+protein+S6+kinase+alpha-3+%5B399-740%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=259813&enzyme=Ribosomal+protein+S6+kinase+alpha-3+%5B399-740%5D&column=ki&startPg=0&Increment=50&submit=Search			52938511	350084507							1	MQTVGVHSIVQQLHRNSIQFTDGYEVKEDIGVGSYSVCKRCIHKATNMEFAVKIIDKSKRDPTEEIEILLRYGQHPNIITLKDVYDDGKYVYVVTELMKGGELLDKILRQKFFSEREASAVLFTITKTVEYLHAQGVVHRDLKPSNILYVDESGNPESIRICDFGFAKQLRAENGLLMTPCYTANFVAPEVLKRQGYDAACDIWSLGVLLYTMLTGYTPFANGPDDTPEEILARIGSGKFSLSGGYWNSVSDTAKDLVSKMLHVDPHQRLTAALVLRHPWIVHWDQLPQYQLNRQDAPHLVKGAMAATYSALNRNQSPVLEPVGRSTLAQRRGIKKITSTAL		Ribosomal protein S6 kinase alpha-3	KS6A3_HUMAN	P51812	B2R9V4 Q4VAP3 Q59H26 Q5JPK8 Q7Z3Z7						
452892	O=C(N1CCCC1)C(=C\c1ccc2[nH]ncc2c1)\C#N	InChI=1S/C15H14N4O/c16-9-12(15(20)19-5-1-2-6-19)7-11-3-4-14-13(8-11)10-17-18-14/h3-4,7-8,10H,1-2,5-6H2,(H,17,18)/b12-7+	FJJMDXPMAYEZEB-KPKJPENVSA-N	259814	US9505766, 14	Ribosomal protein S6 kinase alpha-3 [399-740]			 1000					8	22.00 C	US Patent		10.7270/Q2639NPR		aid1803661	US9505766	Taunton, Jr., JW; Maglathlin, R; Serafimova, I; Cohen, MS; Miller, R; Paavilainen, V; McFarland, J; Krishnan, S	The Regents of the University of California	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=259814	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=11170&target=Ribosomal+protein+S6+kinase+alpha-3+%5B399-740%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=259814&enzyme=Ribosomal+protein+S6+kinase+alpha-3+%5B399-740%5D&column=ki&startPg=0&Increment=50&submit=Search			68347770	350084508							1	MQTVGVHSIVQQLHRNSIQFTDGYEVKEDIGVGSYSVCKRCIHKATNMEFAVKIIDKSKRDPTEEIEILLRYGQHPNIITLKDVYDDGKYVYVVTELMKGGELLDKILRQKFFSEREASAVLFTITKTVEYLHAQGVVHRDLKPSNILYVDESGNPESIRICDFGFAKQLRAENGLLMTPCYTANFVAPEVLKRQGYDAACDIWSLGVLLYTMLTGYTPFANGPDDTPEEILARIGSGKFSLSGGYWNSVSDTAKDLVSKMLHVDPHQRLTAALVLRHPWIVHWDQLPQYQLNRQDAPHLVKGAMAATYSALNRNQSPVLEPVGRSTLAQRRGIKKITSTAL		Ribosomal protein S6 kinase alpha-3	KS6A3_HUMAN	P51812	B2R9V4 Q4VAP3 Q59H26 Q5JPK8 Q7Z3Z7						
452893	NC(=O)C(=C\c1ccc2cn[nH]c2c1)\C#N	InChI=1S/C11H8N4O/c12-5-9(11(13)16)3-7-1-2-8-6-14-15-10(8)4-7/h1-4,6H,(H2,13,16)(H,14,15)/b9-3+	XLGYCNBBWHAJDG-YCRREMRBSA-N	259815	US9505766, 15	Ribosomal protein S6 kinase alpha-3 [399-740]			 183					8	22.00 C	US Patent		10.7270/Q2639NPR		aid1803661	US9505766	Taunton, Jr., JW; Maglathlin, R; Serafimova, I; Cohen, MS; Miller, R; Paavilainen, V; McFarland, J; Krishnan, S	The Regents of the University of California	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=259815	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=11170&target=Ribosomal+protein+S6+kinase+alpha-3+%5B399-740%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=259815&enzyme=Ribosomal+protein+S6+kinase+alpha-3+%5B399-740%5D&column=ki&startPg=0&Increment=50&submit=Search			52938388	350084509							1	MQTVGVHSIVQQLHRNSIQFTDGYEVKEDIGVGSYSVCKRCIHKATNMEFAVKIIDKSKRDPTEEIEILLRYGQHPNIITLKDVYDDGKYVYVVTELMKGGELLDKILRQKFFSEREASAVLFTITKTVEYLHAQGVVHRDLKPSNILYVDESGNPESIRICDFGFAKQLRAENGLLMTPCYTANFVAPEVLKRQGYDAACDIWSLGVLLYTMLTGYTPFANGPDDTPEEILARIGSGKFSLSGGYWNSVSDTAKDLVSKMLHVDPHQRLTAALVLRHPWIVHWDQLPQYQLNRQDAPHLVKGAMAATYSALNRNQSPVLEPVGRSTLAQRRGIKKITSTAL		Ribosomal protein S6 kinase alpha-3	KS6A3_HUMAN	P51812	B2R9V4 Q4VAP3 Q59H26 Q5JPK8 Q7Z3Z7						
452894	CNC(=O)C(=C\c1ccc2cn[nH]c2c1)\C#N	InChI=1S/C12H10N4O/c1-14-12(17)10(6-13)4-8-2-3-9-7-15-16-11(9)5-8/h2-5,7H,1H3,(H,14,17)(H,15,16)/b10-4+	NUHIVHBQXFZPJM-ONNFQVAWSA-N	259816	US9505766, 16	Ribosomal protein S6 kinase alpha-3 [399-740]			 92					8	22.00 C	US Patent		10.7270/Q2639NPR		aid1803661	US9505766	Taunton, Jr., JW; Maglathlin, R; Serafimova, I; Cohen, MS; Miller, R; Paavilainen, V; McFarland, J; Krishnan, S	The Regents of the University of California	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=259816	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=11170&target=Ribosomal+protein+S6+kinase+alpha-3+%5B399-740%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=259816&enzyme=Ribosomal+protein+S6+kinase+alpha-3+%5B399-740%5D&column=ki&startPg=0&Increment=50&submit=Search			68347769	350084510							1	MQTVGVHSIVQQLHRNSIQFTDGYEVKEDIGVGSYSVCKRCIHKATNMEFAVKIIDKSKRDPTEEIEILLRYGQHPNIITLKDVYDDGKYVYVVTELMKGGELLDKILRQKFFSEREASAVLFTITKTVEYLHAQGVVHRDLKPSNILYVDESGNPESIRICDFGFAKQLRAENGLLMTPCYTANFVAPEVLKRQGYDAACDIWSLGVLLYTMLTGYTPFANGPDDTPEEILARIGSGKFSLSGGYWNSVSDTAKDLVSKMLHVDPHQRLTAALVLRHPWIVHWDQLPQYQLNRQDAPHLVKGAMAATYSALNRNQSPVLEPVGRSTLAQRRGIKKITSTAL		Ribosomal protein S6 kinase alpha-3	KS6A3_HUMAN	P51812	B2R9V4 Q4VAP3 Q59H26 Q5JPK8 Q7Z3Z7						
452895	CC(C)NC(=O)C(=C\c1ccc2cn[nH]c2c1)\C#N	InChI=1S/C14H14N4O/c1-9(2)17-14(19)12(7-15)5-10-3-4-11-8-16-18-13(11)6-10/h3-6,8-9H,1-2H3,(H,16,18)(H,17,19)/b12-5+	ZPHLHEVVHGCJDL-LFYBBSHMSA-N	259817	US9505766, 17	Ribosomal protein S6 kinase alpha-3 [399-740]			 630					8	22.00 C	US Patent		10.7270/Q2639NPR		aid1803661	US9505766	Taunton, Jr., JW; Maglathlin, R; Serafimova, I; Cohen, MS; Miller, R; Paavilainen, V; McFarland, J; Krishnan, S	The Regents of the University of California	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=259817	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=11170&target=Ribosomal+protein+S6+kinase+alpha-3+%5B399-740%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=259817&enzyme=Ribosomal+protein+S6+kinase+alpha-3+%5B399-740%5D&column=ki&startPg=0&Increment=50&submit=Search			68347771	350084511							1	MQTVGVHSIVQQLHRNSIQFTDGYEVKEDIGVGSYSVCKRCIHKATNMEFAVKIIDKSKRDPTEEIEILLRYGQHPNIITLKDVYDDGKYVYVVTELMKGGELLDKILRQKFFSEREASAVLFTITKTVEYLHAQGVVHRDLKPSNILYVDESGNPESIRICDFGFAKQLRAENGLLMTPCYTANFVAPEVLKRQGYDAACDIWSLGVLLYTMLTGYTPFANGPDDTPEEILARIGSGKFSLSGGYWNSVSDTAKDLVSKMLHVDPHQRLTAALVLRHPWIVHWDQLPQYQLNRQDAPHLVKGAMAATYSALNRNQSPVLEPVGRSTLAQRRGIKKITSTAL		Ribosomal protein S6 kinase alpha-3	KS6A3_HUMAN	P51812	B2R9V4 Q4VAP3 Q59H26 Q5JPK8 Q7Z3Z7						
452896	NC(=O)C(=C\C1CCN(CC1)c1ncnc2[nH]cnc12)\C#N	InChI=1S/C14H15N7O/c15-6-10(12(16)22)5-9-1-3-21(4-2-9)14-11-13(18-7-17-11)19-8-20-14/h5,7-9H,1-4H2,(H2,16,22)(H,17,18,19,20)/b10-5+	UQVVQLRAEQBLIK-BJMVGYQFSA-N	259818	US9505766, 18	Ribosomal protein S6 kinase alpha-3 [399-740]			 758					8	22.00 C	US Patent		10.7270/Q2639NPR		aid1803661	US9505766	Taunton, Jr., JW; Maglathlin, R; Serafimova, I; Cohen, MS; Miller, R; Paavilainen, V; McFarland, J; Krishnan, S	The Regents of the University of California	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=259818	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=11170&target=Ribosomal+protein+S6+kinase+alpha-3+%5B399-740%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=259818&enzyme=Ribosomal+protein+S6+kinase+alpha-3+%5B399-740%5D&column=ki&startPg=0&Increment=50&submit=Search			67205351	350084512							1	MQTVGVHSIVQQLHRNSIQFTDGYEVKEDIGVGSYSVCKRCIHKATNMEFAVKIIDKSKRDPTEEIEILLRYGQHPNIITLKDVYDDGKYVYVVTELMKGGELLDKILRQKFFSEREASAVLFTITKTVEYLHAQGVVHRDLKPSNILYVDESGNPESIRICDFGFAKQLRAENGLLMTPCYTANFVAPEVLKRQGYDAACDIWSLGVLLYTMLTGYTPFANGPDDTPEEILARIGSGKFSLSGGYWNSVSDTAKDLVSKMLHVDPHQRLTAALVLRHPWIVHWDQLPQYQLNRQDAPHLVKGAMAATYSALNRNQSPVLEPVGRSTLAQRRGIKKITSTAL		Ribosomal protein S6 kinase alpha-3	KS6A3_HUMAN	P51812	B2R9V4 Q4VAP3 Q59H26 Q5JPK8 Q7Z3Z7						
452897	CS(=O)(=O)C(=C\c1ccc(cc1)-c1ncnc2[nH]cnc12)\C#N	InChI=1S/C15H11N5O2S/c1-23(21,22)12(7-16)6-10-2-4-11(5-3-10)13-14-15(19-8-17-13)20-9-18-14/h2-6,8-9H,1H3,(H,17,18,19,20)/b12-6+	NUTCBXHBYDJNKL-WUXMJOGZSA-N	259819	US9505766, 20	Ribosomal protein S6 kinase alpha-3 [399-740]			 60000					8	22.00 C	US Patent		10.7270/Q2639NPR		aid1803661	US9505766	Taunton, Jr., JW; Maglathlin, R; Serafimova, I; Cohen, MS; Miller, R; Paavilainen, V; McFarland, J; Krishnan, S	The Regents of the University of California	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=259819	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=11170&target=Ribosomal+protein+S6+kinase+alpha-3+%5B399-740%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=259819&enzyme=Ribosomal+protein+S6+kinase+alpha-3+%5B399-740%5D&column=ki&startPg=0&Increment=50&submit=Search			52938773	350084513							1	MQTVGVHSIVQQLHRNSIQFTDGYEVKEDIGVGSYSVCKRCIHKATNMEFAVKIIDKSKRDPTEEIEILLRYGQHPNIITLKDVYDDGKYVYVVTELMKGGELLDKILRQKFFSEREASAVLFTITKTVEYLHAQGVVHRDLKPSNILYVDESGNPESIRICDFGFAKQLRAENGLLMTPCYTANFVAPEVLKRQGYDAACDIWSLGVLLYTMLTGYTPFANGPDDTPEEILARIGSGKFSLSGGYWNSVSDTAKDLVSKMLHVDPHQRLTAALVLRHPWIVHWDQLPQYQLNRQDAPHLVKGAMAATYSALNRNQSPVLEPVGRSTLAQRRGIKKITSTAL		Ribosomal protein S6 kinase alpha-3	KS6A3_HUMAN	P51812	B2R9V4 Q4VAP3 Q59H26 Q5JPK8 Q7Z3Z7						
452898	O=S(=O)(C(=C\c1ccc(cc1)-c1ncnc2[nH]cnc12)\C#N)c1ccccc1	InChI=1S/C20H13N5O2S/c21-11-17(28(26,27)16-4-2-1-3-5-16)10-14-6-8-15(9-7-14)18-19-20(24-12-22-18)25-13-23-19/h1-10,12-13H,(H,22,23,24,25)/b17-10+	DZMXVPYWGQHCRO-LICLKQGHSA-N	259820	US9505766, 21	Ribosomal protein S6 kinase alpha-3 [399-740]			 60000					8	22.00 C	US Patent		10.7270/Q2639NPR		aid1803661	US9505766	Taunton, Jr., JW; Maglathlin, R; Serafimova, I; Cohen, MS; Miller, R; Paavilainen, V; McFarland, J; Krishnan, S	The Regents of the University of California	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=259820	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=11170&target=Ribosomal+protein+S6+kinase+alpha-3+%5B399-740%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=259820&enzyme=Ribosomal+protein+S6+kinase+alpha-3+%5B399-740%5D&column=ki&startPg=0&Increment=50&submit=Search			52938774	350084514							1	MQTVGVHSIVQQLHRNSIQFTDGYEVKEDIGVGSYSVCKRCIHKATNMEFAVKIIDKSKRDPTEEIEILLRYGQHPNIITLKDVYDDGKYVYVVTELMKGGELLDKILRQKFFSEREASAVLFTITKTVEYLHAQGVVHRDLKPSNILYVDESGNPESIRICDFGFAKQLRAENGLLMTPCYTANFVAPEVLKRQGYDAACDIWSLGVLLYTMLTGYTPFANGPDDTPEEILARIGSGKFSLSGGYWNSVSDTAKDLVSKMLHVDPHQRLTAALVLRHPWIVHWDQLPQYQLNRQDAPHLVKGAMAATYSALNRNQSPVLEPVGRSTLAQRRGIKKITSTAL		Ribosomal protein S6 kinase alpha-3	KS6A3_HUMAN	P51812	B2R9V4 Q4VAP3 Q59H26 Q5JPK8 Q7Z3Z7						
452899	NC(=O)C(=C\c1ccc(cc1)-c1ccncc1)\C#N	InChI=1S/C15H11N3O/c16-10-14(15(17)19)9-11-1-3-12(4-2-11)13-5-7-18-8-6-13/h1-9H,(H2,17,19)/b14-9+	FYPQUUUPVSAJTG-NTEUORMPSA-N	259821	US9505766, 22	Ribosomal protein S6 kinase alpha-3 [399-740]			 10000					8	22.00 C	US Patent		10.7270/Q2639NPR		aid1803661	US9505766	Taunton, Jr., JW; Maglathlin, R; Serafimova, I; Cohen, MS; Miller, R; Paavilainen, V; McFarland, J; Krishnan, S	The Regents of the University of California	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=259821	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=11170&target=Ribosomal+protein+S6+kinase+alpha-3+%5B399-740%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=259821&enzyme=Ribosomal+protein+S6+kinase+alpha-3+%5B399-740%5D&column=ki&startPg=0&Increment=50&submit=Search			68347790	350084515							1	MQTVGVHSIVQQLHRNSIQFTDGYEVKEDIGVGSYSVCKRCIHKATNMEFAVKIIDKSKRDPTEEIEILLRYGQHPNIITLKDVYDDGKYVYVVTELMKGGELLDKILRQKFFSEREASAVLFTITKTVEYLHAQGVVHRDLKPSNILYVDESGNPESIRICDFGFAKQLRAENGLLMTPCYTANFVAPEVLKRQGYDAACDIWSLGVLLYTMLTGYTPFANGPDDTPEEILARIGSGKFSLSGGYWNSVSDTAKDLVSKMLHVDPHQRLTAALVLRHPWIVHWDQLPQYQLNRQDAPHLVKGAMAATYSALNRNQSPVLEPVGRSTLAQRRGIKKITSTAL		Ribosomal protein S6 kinase alpha-3	KS6A3_HUMAN	P51812	B2R9V4 Q4VAP3 Q59H26 Q5JPK8 Q7Z3Z7						
452900	NC(=O)C(=C\c1cccc(c1)-c1ncnc2[nH]cnc12)\C#N	InChI=1S/C15H10N6O/c16-6-11(14(17)22)5-9-2-1-3-10(4-9)12-13-15(20-7-18-12)21-8-19-13/h1-5,7-8H,(H2,17,22)(H,18,19,20,21)/b11-5+	IFFOEIRCDOBKFH-VZUCSPMQSA-N	259822	US9505766, 23	Ribosomal protein S6 kinase alpha-3 [399-740]			 3000					8	22.00 C	US Patent		10.7270/Q2639NPR		aid1803661	US9505766	Taunton, Jr., JW; Maglathlin, R; Serafimova, I; Cohen, MS; Miller, R; Paavilainen, V; McFarland, J; Krishnan, S	The Regents of the University of California	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=259822	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=11170&target=Ribosomal+protein+S6+kinase+alpha-3+%5B399-740%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=259822&enzyme=Ribosomal+protein+S6+kinase+alpha-3+%5B399-740%5D&column=ki&startPg=0&Increment=50&submit=Search			68347773	350084516							1	MQTVGVHSIVQQLHRNSIQFTDGYEVKEDIGVGSYSVCKRCIHKATNMEFAVKIIDKSKRDPTEEIEILLRYGQHPNIITLKDVYDDGKYVYVVTELMKGGELLDKILRQKFFSEREASAVLFTITKTVEYLHAQGVVHRDLKPSNILYVDESGNPESIRICDFGFAKQLRAENGLLMTPCYTANFVAPEVLKRQGYDAACDIWSLGVLLYTMLTGYTPFANGPDDTPEEILARIGSGKFSLSGGYWNSVSDTAKDLVSKMLHVDPHQRLTAALVLRHPWIVHWDQLPQYQLNRQDAPHLVKGAMAATYSALNRNQSPVLEPVGRSTLAQRRGIKKITSTAL		Ribosomal protein S6 kinase alpha-3	KS6A3_HUMAN	P51812	B2R9V4 Q4VAP3 Q59H26 Q5JPK8 Q7Z3Z7						
452901	NC(=O)C(=C\c1ccc(cc1)-c1cn[nH]c1)\C#N	InChI=1S/C13H10N4O/c14-6-11(13(15)18)5-9-1-3-10(4-2-9)12-7-16-17-8-12/h1-5,7-8H,(H2,15,18)(H,16,17)/b11-5+	BNRLLVUNYCBXNJ-VZUCSPMQSA-N	259823	US9505766, 24	Ribosomal protein S6 kinase alpha-3 [399-740]			 5000					8	22.00 C	US Patent		10.7270/Q2639NPR		aid1803661	US9505766	Taunton, Jr., JW; Maglathlin, R; Serafimova, I; Cohen, MS; Miller, R; Paavilainen, V; McFarland, J; Krishnan, S	The Regents of the University of California	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=259823	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=11170&target=Ribosomal+protein+S6+kinase+alpha-3+%5B399-740%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=259823&enzyme=Ribosomal+protein+S6+kinase+alpha-3+%5B399-740%5D&column=ki&startPg=0&Increment=50&submit=Search			52938890	350084517							1	MQTVGVHSIVQQLHRNSIQFTDGYEVKEDIGVGSYSVCKRCIHKATNMEFAVKIIDKSKRDPTEEIEILLRYGQHPNIITLKDVYDDGKYVYVVTELMKGGELLDKILRQKFFSEREASAVLFTITKTVEYLHAQGVVHRDLKPSNILYVDESGNPESIRICDFGFAKQLRAENGLLMTPCYTANFVAPEVLKRQGYDAACDIWSLGVLLYTMLTGYTPFANGPDDTPEEILARIGSGKFSLSGGYWNSVSDTAKDLVSKMLHVDPHQRLTAALVLRHPWIVHWDQLPQYQLNRQDAPHLVKGAMAATYSALNRNQSPVLEPVGRSTLAQRRGIKKITSTAL		Ribosomal protein S6 kinase alpha-3	KS6A3_HUMAN	P51812	B2R9V4 Q4VAP3 Q59H26 Q5JPK8 Q7Z3Z7						
452902	O=C(N1CCCC1)C(=C\c1ccc2cn[nH]c2c1)\C#N	InChI=1S/C15H14N4O/c16-9-13(15(20)19-5-1-2-6-19)7-11-3-4-12-10-17-18-14(12)8-11/h3-4,7-8,10H,1-2,5-6H2,(H,17,18)/b13-7+	YZHVOWFHVJPKPH-NTUHNPAUSA-N	259824	US9505766, 25	Ribosomal protein S6 kinase alpha-3 [399-740]			 2600					8	22.00 C	US Patent		10.7270/Q2639NPR		aid1803661	US9505766	Taunton, Jr., JW; Maglathlin, R; Serafimova, I; Cohen, MS; Miller, R; Paavilainen, V; McFarland, J; Krishnan, S	The Regents of the University of California	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=259824	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=11170&target=Ribosomal+protein+S6+kinase+alpha-3+%5B399-740%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=259824&enzyme=Ribosomal+protein+S6+kinase+alpha-3+%5B399-740%5D&column=ki&startPg=0&Increment=50&submit=Search			52938891	350084518							1	MQTVGVHSIVQQLHRNSIQFTDGYEVKEDIGVGSYSVCKRCIHKATNMEFAVKIIDKSKRDPTEEIEILLRYGQHPNIITLKDVYDDGKYVYVVTELMKGGELLDKILRQKFFSEREASAVLFTITKTVEYLHAQGVVHRDLKPSNILYVDESGNPESIRICDFGFAKQLRAENGLLMTPCYTANFVAPEVLKRQGYDAACDIWSLGVLLYTMLTGYTPFANGPDDTPEEILARIGSGKFSLSGGYWNSVSDTAKDLVSKMLHVDPHQRLTAALVLRHPWIVHWDQLPQYQLNRQDAPHLVKGAMAATYSALNRNQSPVLEPVGRSTLAQRRGIKKITSTAL		Ribosomal protein S6 kinase alpha-3	KS6A3_HUMAN	P51812	B2R9V4 Q4VAP3 Q59H26 Q5JPK8 Q7Z3Z7						
452903	CS(=O)(=O)C(=C\c1cccc(c1)C(=O)c1c[nH]c2ncccc12)\C#N	InChI=1S/C18H13N3O3S/c1-25(23,24)14(10-19)9-12-4-2-5-13(8-12)17(22)16-11-21-18-15(16)6-3-7-20-18/h2-9,11H,1H3,(H,20,21)/b14-9+	JVUYFKGAACUDSV-NTEUORMPSA-N	259825	US9505766, 29	Ribosomal protein S6 kinase alpha-3 [399-740]			 1000					8	22.00 C	US Patent		10.7270/Q2639NPR		aid1803661	US9505766	Taunton, Jr., JW; Maglathlin, R; Serafimova, I; Cohen, MS; Miller, R; Paavilainen, V; McFarland, J; Krishnan, S	The Regents of the University of California	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=259825	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=11170&target=Ribosomal+protein+S6+kinase+alpha-3+%5B399-740%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=259825&enzyme=Ribosomal+protein+S6+kinase+alpha-3+%5B399-740%5D&column=ki&startPg=0&Increment=50&submit=Search			71250196	350084519							1	MQTVGVHSIVQQLHRNSIQFTDGYEVKEDIGVGSYSVCKRCIHKATNMEFAVKIIDKSKRDPTEEIEILLRYGQHPNIITLKDVYDDGKYVYVVTELMKGGELLDKILRQKFFSEREASAVLFTITKTVEYLHAQGVVHRDLKPSNILYVDESGNPESIRICDFGFAKQLRAENGLLMTPCYTANFVAPEVLKRQGYDAACDIWSLGVLLYTMLTGYTPFANGPDDTPEEILARIGSGKFSLSGGYWNSVSDTAKDLVSKMLHVDPHQRLTAALVLRHPWIVHWDQLPQYQLNRQDAPHLVKGAMAATYSALNRNQSPVLEPVGRSTLAQRRGIKKITSTAL		Ribosomal protein S6 kinase alpha-3	KS6A3_HUMAN	P51812	B2R9V4 Q4VAP3 Q59H26 Q5JPK8 Q7Z3Z7						
452904	CCOP(=O)(OCC)C(=C\c1ccc(cc1)-c1ccncc1)\C#N	InChI=1S/C18H19N2O3P/c1-3-22-24(21,23-4-2)18(14-19)13-15-5-7-16(8-6-15)17-9-11-20-12-10-17/h5-13H,3-4H2,1-2H3/b18-13+	FJKJKXLQLWSSGR-QGOAFFKASA-N	259827	US9505766, 31	Ribosomal protein S6 kinase alpha-3 [399-740]			 20000					8	22.00 C	US Patent		10.7270/Q2639NPR		aid1803661	US9505766	Taunton, Jr., JW; Maglathlin, R; Serafimova, I; Cohen, MS; Miller, R; Paavilainen, V; McFarland, J; Krishnan, S	The Regents of the University of California	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=259827	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=11170&target=Ribosomal+protein+S6+kinase+alpha-3+%5B399-740%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=259827&enzyme=Ribosomal+protein+S6+kinase+alpha-3+%5B399-740%5D&column=ki&startPg=0&Increment=50&submit=Search			52938894	350084521							1	MQTVGVHSIVQQLHRNSIQFTDGYEVKEDIGVGSYSVCKRCIHKATNMEFAVKIIDKSKRDPTEEIEILLRYGQHPNIITLKDVYDDGKYVYVVTELMKGGELLDKILRQKFFSEREASAVLFTITKTVEYLHAQGVVHRDLKPSNILYVDESGNPESIRICDFGFAKQLRAENGLLMTPCYTANFVAPEVLKRQGYDAACDIWSLGVLLYTMLTGYTPFANGPDDTPEEILARIGSGKFSLSGGYWNSVSDTAKDLVSKMLHVDPHQRLTAALVLRHPWIVHWDQLPQYQLNRQDAPHLVKGAMAATYSALNRNQSPVLEPVGRSTLAQRRGIKKITSTAL		Ribosomal protein S6 kinase alpha-3	KS6A3_HUMAN	P51812	B2R9V4 Q4VAP3 Q59H26 Q5JPK8 Q7Z3Z7						
452905	Cc1ccc(cc1)-c1c(\C=C(/C#N)c2ccccn2)n(CCCO)c2ncnc(N)c12	InChI=1S/C24H22N6O/c1-16-6-8-17(9-7-16)21-20(13-18(14-25)19-5-2-3-10-27-19)30(11-4-12-31)24-22(21)23(26)28-15-29-24/h2-3,5-10,13,15,31H,4,11-12H2,1H3,(H2,26,28,29)/b18-13+	PTVACVSGZJWNRY-QGOAFFKASA-N	259828	US9505766, 32	Ribosomal protein S6 kinase alpha-3 [399-740]			 142					8	22.00 C	US Patent		10.7270/Q2639NPR		aid1803661	US9505766	Taunton, Jr., JW; Maglathlin, R; Serafimova, I; Cohen, MS; Miller, R; Paavilainen, V; McFarland, J; Krishnan, S	The Regents of the University of California	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=259828	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=11170&target=Ribosomal+protein+S6+kinase+alpha-3+%5B399-740%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=259828&enzyme=Ribosomal+protein+S6+kinase+alpha-3+%5B399-740%5D&column=ki&startPg=0&Increment=50&submit=Search			68347712	350084522							1	MQTVGVHSIVQQLHRNSIQFTDGYEVKEDIGVGSYSVCKRCIHKATNMEFAVKIIDKSKRDPTEEIEILLRYGQHPNIITLKDVYDDGKYVYVVTELMKGGELLDKILRQKFFSEREASAVLFTITKTVEYLHAQGVVHRDLKPSNILYVDESGNPESIRICDFGFAKQLRAENGLLMTPCYTANFVAPEVLKRQGYDAACDIWSLGVLLYTMLTGYTPFANGPDDTPEEILARIGSGKFSLSGGYWNSVSDTAKDLVSKMLHVDPHQRLTAALVLRHPWIVHWDQLPQYQLNRQDAPHLVKGAMAATYSALNRNQSPVLEPVGRSTLAQRRGIKKITSTAL		Ribosomal protein S6 kinase alpha-3	KS6A3_HUMAN	P51812	B2R9V4 Q4VAP3 Q59H26 Q5JPK8 Q7Z3Z7						
452906	NC(=O)C(=C\c1nc2c(N)ncnc2n1CCCO)\C#N	InChI=1S/C12H13N7O2/c13-5-7(11(15)21)4-8-18-9-10(14)16-6-17-12(9)19(8)2-1-3-20/h4,6,20H,1-3H2,(H2,15,21)(H2,14,16,17)/b7-4+	YADAJQRYASQJMB-QPJJXVBHSA-N	259829	US9505766, 33	Ribosomal protein S6 kinase alpha-3 [399-740]			 80000					8	22.00 C	US Patent		10.7270/Q2639NPR		aid1803661	US9505766	Taunton, Jr., JW; Maglathlin, R; Serafimova, I; Cohen, MS; Miller, R; Paavilainen, V; McFarland, J; Krishnan, S	The Regents of the University of California	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=259829	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=11170&target=Ribosomal+protein+S6+kinase+alpha-3+%5B399-740%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=259829&enzyme=Ribosomal+protein+S6+kinase+alpha-3+%5B399-740%5D&column=ki&startPg=0&Increment=50&submit=Search			52938896	350084523							1	MQTVGVHSIVQQLHRNSIQFTDGYEVKEDIGVGSYSVCKRCIHKATNMEFAVKIIDKSKRDPTEEIEILLRYGQHPNIITLKDVYDDGKYVYVVTELMKGGELLDKILRQKFFSEREASAVLFTITKTVEYLHAQGVVHRDLKPSNILYVDESGNPESIRICDFGFAKQLRAENGLLMTPCYTANFVAPEVLKRQGYDAACDIWSLGVLLYTMLTGYTPFANGPDDTPEEILARIGSGKFSLSGGYWNSVSDTAKDLVSKMLHVDPHQRLTAALVLRHPWIVHWDQLPQYQLNRQDAPHLVKGAMAATYSALNRNQSPVLEPVGRSTLAQRRGIKKITSTAL		Ribosomal protein S6 kinase alpha-3	KS6A3_HUMAN	P51812	B2R9V4 Q4VAP3 Q59H26 Q5JPK8 Q7Z3Z7						
452907	CNC(=O)C(=C\c1ccc2[nH]ncc2c1)\C#N	InChI=1S/C12H10N4O/c1-14-12(17)9(6-13)4-8-2-3-11-10(5-8)7-15-16-11/h2-5,7H,1H3,(H,14,17)(H,15,16)/b9-4+	RQRJOTZDZIGRHX-RUDMXATFSA-N	259830	US9505766, 34	Ribosomal protein S6 kinase alpha-3 [399-740]			 129					8	22.00 C	US Patent		10.7270/Q2639NPR		aid1803661	US9505766	Taunton, Jr., JW; Maglathlin, R; Serafimova, I; Cohen, MS; Miller, R; Paavilainen, V; McFarland, J; Krishnan, S	The Regents of the University of California	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=259830	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=11170&target=Ribosomal+protein+S6+kinase+alpha-3+%5B399-740%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=259830&enzyme=Ribosomal+protein+S6+kinase+alpha-3+%5B399-740%5D&column=ki&startPg=0&Increment=50&submit=Search			71250219	350084524							1	MQTVGVHSIVQQLHRNSIQFTDGYEVKEDIGVGSYSVCKRCIHKATNMEFAVKIIDKSKRDPTEEIEILLRYGQHPNIITLKDVYDDGKYVYVVTELMKGGELLDKILRQKFFSEREASAVLFTITKTVEYLHAQGVVHRDLKPSNILYVDESGNPESIRICDFGFAKQLRAENGLLMTPCYTANFVAPEVLKRQGYDAACDIWSLGVLLYTMLTGYTPFANGPDDTPEEILARIGSGKFSLSGGYWNSVSDTAKDLVSKMLHVDPHQRLTAALVLRHPWIVHWDQLPQYQLNRQDAPHLVKGAMAATYSALNRNQSPVLEPVGRSTLAQRRGIKKITSTAL		Ribosomal protein S6 kinase alpha-3	KS6A3_HUMAN	P51812	B2R9V4 Q4VAP3 Q59H26 Q5JPK8 Q7Z3Z7						
452908	CC(C)NC(=O)C(=C\c1ccc2[nH]ncc2c1)\C#N	InChI=1S/C14H14N4O/c1-9(2)17-14(19)11(7-15)5-10-3-4-13-12(6-10)8-16-18-13/h3-6,8-9H,1-2H3,(H,16,18)(H,17,19)/b11-5+	MXPOJBLWSIKGTF-VZUCSPMQSA-N	259831	US9505766, 35	Ribosomal protein S6 kinase alpha-3 [399-740]			 493					8	22.00 C	US Patent		10.7270/Q2639NPR		aid1803661	US9505766	Taunton, Jr., JW; Maglathlin, R; Serafimova, I; Cohen, MS; Miller, R; Paavilainen, V; McFarland, J; Krishnan, S	The Regents of the University of California	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=259831	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=11170&target=Ribosomal+protein+S6+kinase+alpha-3+%5B399-740%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=259831&enzyme=Ribosomal+protein+S6+kinase+alpha-3+%5B399-740%5D&column=ki&startPg=0&Increment=50&submit=Search			68347768	350084525							1	MQTVGVHSIVQQLHRNSIQFTDGYEVKEDIGVGSYSVCKRCIHKATNMEFAVKIIDKSKRDPTEEIEILLRYGQHPNIITLKDVYDDGKYVYVVTELMKGGELLDKILRQKFFSEREASAVLFTITKTVEYLHAQGVVHRDLKPSNILYVDESGNPESIRICDFGFAKQLRAENGLLMTPCYTANFVAPEVLKRQGYDAACDIWSLGVLLYTMLTGYTPFANGPDDTPEEILARIGSGKFSLSGGYWNSVSDTAKDLVSKMLHVDPHQRLTAALVLRHPWIVHWDQLPQYQLNRQDAPHLVKGAMAATYSALNRNQSPVLEPVGRSTLAQRRGIKKITSTAL		Ribosomal protein S6 kinase alpha-3	KS6A3_HUMAN	P51812	B2R9V4 Q4VAP3 Q59H26 Q5JPK8 Q7Z3Z7						
452909	CN(C)C(=O)C(=C\c1ccc2[nH]ncc2c1)\C#N	InChI=1S/C13H12N4O/c1-17(2)13(18)10(7-14)5-9-3-4-12-11(6-9)8-15-16-12/h3-6,8H,1-2H3,(H,15,16)/b10-5+	FRHBBZWOHGDFFT-BJMVGYQFSA-N	259833	US9505766, 37	Ribosomal protein S6 kinase alpha-3 [399-740]			 747					8	22.00 C	US Patent		10.7270/Q2639NPR		aid1803661	US9505766	Taunton, Jr., JW; Maglathlin, R; Serafimova, I; Cohen, MS; Miller, R; Paavilainen, V; McFarland, J; Krishnan, S	The Regents of the University of California	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=259833	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=11170&target=Ribosomal+protein+S6+kinase+alpha-3+%5B399-740%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=259833&enzyme=Ribosomal+protein+S6+kinase+alpha-3+%5B399-740%5D&column=ki&startPg=0&Increment=50&submit=Search			52939017	350084527							1	MQTVGVHSIVQQLHRNSIQFTDGYEVKEDIGVGSYSVCKRCIHKATNMEFAVKIIDKSKRDPTEEIEILLRYGQHPNIITLKDVYDDGKYVYVVTELMKGGELLDKILRQKFFSEREASAVLFTITKTVEYLHAQGVVHRDLKPSNILYVDESGNPESIRICDFGFAKQLRAENGLLMTPCYTANFVAPEVLKRQGYDAACDIWSLGVLLYTMLTGYTPFANGPDDTPEEILARIGSGKFSLSGGYWNSVSDTAKDLVSKMLHVDPHQRLTAALVLRHPWIVHWDQLPQYQLNRQDAPHLVKGAMAATYSALNRNQSPVLEPVGRSTLAQRRGIKKITSTAL		Ribosomal protein S6 kinase alpha-3	KS6A3_HUMAN	P51812	B2R9V4 Q4VAP3 Q59H26 Q5JPK8 Q7Z3Z7						
452910	CNC(=O)C(=C\c1cccc(c1)C(=O)c1c[nH]c2ncccc12)\C#N	InChI=1S/C19H14N4O2/c1-21-19(25)14(10-20)9-12-4-2-5-13(8-12)17(24)16-11-23-18-15(16)6-3-7-22-18/h2-9,11H,1H3,(H,21,25)(H,22,23)/b14-9+	KEDKBMWYWUXRQQ-NTEUORMPSA-N	259834	US9505766, 38	Ribosomal protein S6 kinase alpha-3 [399-740]			 386					8	22.00 C	US Patent		10.7270/Q2639NPR		aid1803661	US9505766	Taunton, Jr., JW; Maglathlin, R; Serafimova, I; Cohen, MS; Miller, R; Paavilainen, V; McFarland, J; Krishnan, S	The Regents of the University of California	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=259834	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=11170&target=Ribosomal+protein+S6+kinase+alpha-3+%5B399-740%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=259834&enzyme=Ribosomal+protein+S6+kinase+alpha-3+%5B399-740%5D&column=ki&startPg=0&Increment=50&submit=Search			52939018	350084528							1	MQTVGVHSIVQQLHRNSIQFTDGYEVKEDIGVGSYSVCKRCIHKATNMEFAVKIIDKSKRDPTEEIEILLRYGQHPNIITLKDVYDDGKYVYVVTELMKGGELLDKILRQKFFSEREASAVLFTITKTVEYLHAQGVVHRDLKPSNILYVDESGNPESIRICDFGFAKQLRAENGLLMTPCYTANFVAPEVLKRQGYDAACDIWSLGVLLYTMLTGYTPFANGPDDTPEEILARIGSGKFSLSGGYWNSVSDTAKDLVSKMLHVDPHQRLTAALVLRHPWIVHWDQLPQYQLNRQDAPHLVKGAMAATYSALNRNQSPVLEPVGRSTLAQRRGIKKITSTAL		Ribosomal protein S6 kinase alpha-3	KS6A3_HUMAN	P51812	B2R9V4 Q4VAP3 Q59H26 Q5JPK8 Q7Z3Z7						
452911	CN(C)C(=O)C(=C\c1cccc(c1)C(=O)c1c[nH]c2ncccc12)\C#N	InChI=1S/C20H16N4O2/c1-24(2)20(26)15(11-21)10-13-5-3-6-14(9-13)18(25)17-12-23-19-16(17)7-4-8-22-19/h3-10,12H,1-2H3,(H,22,23)/b15-10+	ONYKCRXFMUZZBQ-XNTDXEJSSA-N	259835	US9505766, 39	Ribosomal protein S6 kinase alpha-3 [399-740]			 2000					8	22.00 C	US Patent		10.7270/Q2639NPR		aid1803661	US9505766	Taunton, Jr., JW; Maglathlin, R; Serafimova, I; Cohen, MS; Miller, R; Paavilainen, V; McFarland, J; Krishnan, S	The Regents of the University of California	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=259835	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=11170&target=Ribosomal+protein+S6+kinase+alpha-3+%5B399-740%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=259835&enzyme=Ribosomal+protein+S6+kinase+alpha-3+%5B399-740%5D&column=ki&startPg=0&Increment=50&submit=Search			52939019	350084529							1	MQTVGVHSIVQQLHRNSIQFTDGYEVKEDIGVGSYSVCKRCIHKATNMEFAVKIIDKSKRDPTEEIEILLRYGQHPNIITLKDVYDDGKYVYVVTELMKGGELLDKILRQKFFSEREASAVLFTITKTVEYLHAQGVVHRDLKPSNILYVDESGNPESIRICDFGFAKQLRAENGLLMTPCYTANFVAPEVLKRQGYDAACDIWSLGVLLYTMLTGYTPFANGPDDTPEEILARIGSGKFSLSGGYWNSVSDTAKDLVSKMLHVDPHQRLTAALVLRHPWIVHWDQLPQYQLNRQDAPHLVKGAMAATYSALNRNQSPVLEPVGRSTLAQRRGIKKITSTAL		Ribosomal protein S6 kinase alpha-3	KS6A3_HUMAN	P51812	B2R9V4 Q4VAP3 Q59H26 Q5JPK8 Q7Z3Z7						
452912	COc1cc(cc(OC)c1OC)-c1n[nH]c2ccc(\C=C(/C#N)C(N)=O)cc12	InChI=1S/C20H18N4O4/c1-26-16-8-12(9-17(27-2)19(16)28-3)18-14-7-11(4-5-15(14)23-24-18)6-13(10-21)20(22)25/h4-9H,1-3H3,(H2,22,25)(H,23,24)/b13-6+	IBUMAHMUIWPTCV-AWNIVKPZSA-N	259836	US9505766, 40	Ribosomal protein S6 kinase alpha-3 [399-740]			 14					8	22.00 C	US Patent		10.7270/Q2639NPR		aid1803661	US9505766	Taunton, Jr., JW; Maglathlin, R; Serafimova, I; Cohen, MS; Miller, R; Paavilainen, V; McFarland, J; Krishnan, S	The Regents of the University of California	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=259836	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=11170&target=Ribosomal+protein+S6+kinase+alpha-3+%5B399-740%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=259836&enzyme=Ribosomal+protein+S6+kinase+alpha-3+%5B399-740%5D&column=ki&startPg=0&Increment=50&submit=Search			131954194	350084530							1	MQTVGVHSIVQQLHRNSIQFTDGYEVKEDIGVGSYSVCKRCIHKATNMEFAVKIIDKSKRDPTEEIEILLRYGQHPNIITLKDVYDDGKYVYVVTELMKGGELLDKILRQKFFSEREASAVLFTITKTVEYLHAQGVVHRDLKPSNILYVDESGNPESIRICDFGFAKQLRAENGLLMTPCYTANFVAPEVLKRQGYDAACDIWSLGVLLYTMLTGYTPFANGPDDTPEEILARIGSGKFSLSGGYWNSVSDTAKDLVSKMLHVDPHQRLTAALVLRHPWIVHWDQLPQYQLNRQDAPHLVKGAMAATYSALNRNQSPVLEPVGRSTLAQRRGIKKITSTAL		Ribosomal protein S6 kinase alpha-3	KS6A3_HUMAN	P51812	B2R9V4 Q4VAP3 Q59H26 Q5JPK8 Q7Z3Z7						
452913	CNC(=O)C(=C\c1ccc2[nH]nc(-c3cc(OC)c(OC)c(OC)c3)c2c1)\C#N	InChI=1S/C21H20N4O4/c1-23-21(26)14(11-22)7-12-5-6-16-15(8-12)19(25-24-16)13-9-17(27-2)20(29-4)18(10-13)28-3/h5-10H,1-4H3,(H,23,26)(H,24,25)/b14-7+	JGIBKTCCYJBOMS-VGOFMYFVSA-N	259837	US9505766, 41	Ribosomal protein S6 kinase alpha-3 [399-740]			 14					8	22.00 C	US Patent		10.7270/Q2639NPR		aid1803661	US9505766	Taunton, Jr., JW; Maglathlin, R; Serafimova, I; Cohen, MS; Miller, R; Paavilainen, V; McFarland, J; Krishnan, S	The Regents of the University of California	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=259837	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=11170&target=Ribosomal+protein+S6+kinase+alpha-3+%5B399-740%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=259837&enzyme=Ribosomal+protein+S6+kinase+alpha-3+%5B399-740%5D&column=ki&startPg=0&Increment=50&submit=Search			131954195	350084531							1	MQTVGVHSIVQQLHRNSIQFTDGYEVKEDIGVGSYSVCKRCIHKATNMEFAVKIIDKSKRDPTEEIEILLRYGQHPNIITLKDVYDDGKYVYVVTELMKGGELLDKILRQKFFSEREASAVLFTITKTVEYLHAQGVVHRDLKPSNILYVDESGNPESIRICDFGFAKQLRAENGLLMTPCYTANFVAPEVLKRQGYDAACDIWSLGVLLYTMLTGYTPFANGPDDTPEEILARIGSGKFSLSGGYWNSVSDTAKDLVSKMLHVDPHQRLTAALVLRHPWIVHWDQLPQYQLNRQDAPHLVKGAMAATYSALNRNQSPVLEPVGRSTLAQRRGIKKITSTAL		Ribosomal protein S6 kinase alpha-3	KS6A3_HUMAN	P51812	B2R9V4 Q4VAP3 Q59H26 Q5JPK8 Q7Z3Z7						
452914	COc1cc(cc(OC)c1OC)-c1n[nH]c2ccc(\C=C(/C#N)C(=O)N(C)C)cc12	InChI=1S/C22H22N4O4/c1-26(2)22(27)15(12-23)8-13-6-7-17-16(9-13)20(25-24-17)14-10-18(28-3)21(30-5)19(11-14)29-4/h6-11H,1-5H3,(H,24,25)/b15-8+	VLDMPVNRZYIDHU-OVCLIPMQSA-N	259838	US9505766, 42	Ribosomal protein S6 kinase alpha-3 [399-740]			 89					8	22.00 C	US Patent		10.7270/Q2639NPR		aid1803661	US9505766	Taunton, Jr., JW; Maglathlin, R; Serafimova, I; Cohen, MS; Miller, R; Paavilainen, V; McFarland, J; Krishnan, S	The Regents of the University of California	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=259838	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=11170&target=Ribosomal+protein+S6+kinase+alpha-3+%5B399-740%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=259838&enzyme=Ribosomal+protein+S6+kinase+alpha-3+%5B399-740%5D&column=ki&startPg=0&Increment=50&submit=Search			131954196	350084532							1	MQTVGVHSIVQQLHRNSIQFTDGYEVKEDIGVGSYSVCKRCIHKATNMEFAVKIIDKSKRDPTEEIEILLRYGQHPNIITLKDVYDDGKYVYVVTELMKGGELLDKILRQKFFSEREASAVLFTITKTVEYLHAQGVVHRDLKPSNILYVDESGNPESIRICDFGFAKQLRAENGLLMTPCYTANFVAPEVLKRQGYDAACDIWSLGVLLYTMLTGYTPFANGPDDTPEEILARIGSGKFSLSGGYWNSVSDTAKDLVSKMLHVDPHQRLTAALVLRHPWIVHWDQLPQYQLNRQDAPHLVKGAMAATYSALNRNQSPVLEPVGRSTLAQRRGIKKITSTAL		Ribosomal protein S6 kinase alpha-3	KS6A3_HUMAN	P51812	B2R9V4 Q4VAP3 Q59H26 Q5JPK8 Q7Z3Z7						
452915	Cc1ccc(cc1)-c1c(\C=C(/C#N)C(=O)NC(C)(C)CO)n(CCCO)c2ncnc(N)c12	InChI=1S/C24H28N6O3/c1-15-5-7-16(8-6-15)19-18(11-17(12-25)23(33)29-24(2,3)13-32)30(9-4-10-31)22-20(19)21(26)27-14-28-22/h5-8,11,14,31-32H,4,9-10,13H2,1-3H3,(H,29,33)(H2,26,27,28)/b17-11+	SBWUFNYSAAEWDF-GZTJUZNOSA-N	259839	US9505766, 43	Ribosomal protein S6 kinase alpha-3 [399-740]			 3.8					8	22.00 C	US Patent		10.7270/Q2639NPR		aid1803661	US9505766	Taunton, Jr., JW; Maglathlin, R; Serafimova, I; Cohen, MS; Miller, R; Paavilainen, V; McFarland, J; Krishnan, S	The Regents of the University of California	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=259839	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=11170&target=Ribosomal+protein+S6+kinase+alpha-3+%5B399-740%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=259839&enzyme=Ribosomal+protein+S6+kinase+alpha-3+%5B399-740%5D&column=ki&startPg=0&Increment=50&submit=Search			52939143	350084533							1	MQTVGVHSIVQQLHRNSIQFTDGYEVKEDIGVGSYSVCKRCIHKATNMEFAVKIIDKSKRDPTEEIEILLRYGQHPNIITLKDVYDDGKYVYVVTELMKGGELLDKILRQKFFSEREASAVLFTITKTVEYLHAQGVVHRDLKPSNILYVDESGNPESIRICDFGFAKQLRAENGLLMTPCYTANFVAPEVLKRQGYDAACDIWSLGVLLYTMLTGYTPFANGPDDTPEEILARIGSGKFSLSGGYWNSVSDTAKDLVSKMLHVDPHQRLTAALVLRHPWIVHWDQLPQYQLNRQDAPHLVKGAMAATYSALNRNQSPVLEPVGRSTLAQRRGIKKITSTAL		Ribosomal protein S6 kinase alpha-3	KS6A3_HUMAN	P51812	B2R9V4 Q4VAP3 Q59H26 Q5JPK8 Q7Z3Z7						
452916	Cc1ccc(cc1)-c1c(\C=C(/C#N)C(=O)NC2CC2)n(CCCO)c2ncnc(N)c12	InChI=1S/C23H24N6O2/c1-14-3-5-15(6-4-14)19-18(11-16(12-24)23(31)28-17-7-8-17)29(9-2-10-30)22-20(19)21(25)26-13-27-22/h3-6,11,13,17,30H,2,7-10H2,1H3,(H,28,31)(H2,25,26,27)/b16-11+	NUHQJXSTTZFNIC-LFIBNONCSA-N	259840	US9505766, 44	Ribosomal protein S6 kinase alpha-3 [399-740]			 2.4					8	22.00 C	US Patent		10.7270/Q2639NPR		aid1803661	US9505766	Taunton, Jr., JW; Maglathlin, R; Serafimova, I; Cohen, MS; Miller, R; Paavilainen, V; McFarland, J; Krishnan, S	The Regents of the University of California	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=259840	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=11170&target=Ribosomal+protein+S6+kinase+alpha-3+%5B399-740%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=259840&enzyme=Ribosomal+protein+S6+kinase+alpha-3+%5B399-740%5D&column=ki&startPg=0&Increment=50&submit=Search			52939022	350084534							1	MQTVGVHSIVQQLHRNSIQFTDGYEVKEDIGVGSYSVCKRCIHKATNMEFAVKIIDKSKRDPTEEIEILLRYGQHPNIITLKDVYDDGKYVYVVTELMKGGELLDKILRQKFFSEREASAVLFTITKTVEYLHAQGVVHRDLKPSNILYVDESGNPESIRICDFGFAKQLRAENGLLMTPCYTANFVAPEVLKRQGYDAACDIWSLGVLLYTMLTGYTPFANGPDDTPEEILARIGSGKFSLSGGYWNSVSDTAKDLVSKMLHVDPHQRLTAALVLRHPWIVHWDQLPQYQLNRQDAPHLVKGAMAATYSALNRNQSPVLEPVGRSTLAQRRGIKKITSTAL		Ribosomal protein S6 kinase alpha-3	KS6A3_HUMAN	P51812	B2R9V4 Q4VAP3 Q59H26 Q5JPK8 Q7Z3Z7						
452917	CCN(CC)C(=O)C(=C\c1c(-c2ccc(C)cc2)c2c(N)ncnc2n1CCCO)\C#N	InChI=1S/C24H28N6O2/c1-4-29(5-2)24(32)18(14-25)13-19-20(17-9-7-16(3)8-10-17)21-22(26)27-15-28-23(21)30(19)11-6-12-31/h7-10,13,15,31H,4-6,11-12H2,1-3H3,(H2,26,27,28)/b18-13+	YTTVLNBTJVEKRY-QGOAFFKASA-N	259841	US9505766, 45	Ribosomal protein S6 kinase alpha-3 [399-740]			 24.3					8	22.00 C	US Patent		10.7270/Q2639NPR		aid1803661	US9505766	Taunton, Jr., JW; Maglathlin, R; Serafimova, I; Cohen, MS; Miller, R; Paavilainen, V; McFarland, J; Krishnan, S	The Regents of the University of California	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=259841	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=11170&target=Ribosomal+protein+S6+kinase+alpha-3+%5B399-740%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=259841&enzyme=Ribosomal+protein+S6+kinase+alpha-3+%5B399-740%5D&column=ki&startPg=0&Increment=50&submit=Search			52938646	350084535							1	MQTVGVHSIVQQLHRNSIQFTDGYEVKEDIGVGSYSVCKRCIHKATNMEFAVKIIDKSKRDPTEEIEILLRYGQHPNIITLKDVYDDGKYVYVVTELMKGGELLDKILRQKFFSEREASAVLFTITKTVEYLHAQGVVHRDLKPSNILYVDESGNPESIRICDFGFAKQLRAENGLLMTPCYTANFVAPEVLKRQGYDAACDIWSLGVLLYTMLTGYTPFANGPDDTPEEILARIGSGKFSLSGGYWNSVSDTAKDLVSKMLHVDPHQRLTAALVLRHPWIVHWDQLPQYQLNRQDAPHLVKGAMAATYSALNRNQSPVLEPVGRSTLAQRRGIKKITSTAL		Ribosomal protein S6 kinase alpha-3	KS6A3_HUMAN	P51812	B2R9V4 Q4VAP3 Q59H26 Q5JPK8 Q7Z3Z7						
452918	Cc1ccc(cc1)-c1c(\C=C(/C#N)C(=O)N2CCCC2)n(CCCO)c2ncnc(N)c12	InChI=1S/C24H26N6O2/c1-16-5-7-17(8-6-16)20-19(13-18(14-25)24(32)29-9-2-3-10-29)30(11-4-12-31)23-21(20)22(26)27-15-28-23/h5-8,13,15,31H,2-4,9-12H2,1H3,(H2,26,27,28)/b18-13+	HUNVXONHJJSTOV-QGOAFFKASA-N	259842	US9505766, 46	Ribosomal protein S6 kinase alpha-3 [399-740]			 23.2					8	22.00 C	US Patent		10.7270/Q2639NPR		aid1803661	US9505766	Taunton, Jr., JW; Maglathlin, R; Serafimova, I; Cohen, MS; Miller, R; Paavilainen, V; McFarland, J; Krishnan, S	The Regents of the University of California	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=259842	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=11170&target=Ribosomal+protein+S6+kinase+alpha-3+%5B399-740%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=259842&enzyme=Ribosomal+protein+S6+kinase+alpha-3+%5B399-740%5D&column=ki&startPg=0&Increment=50&submit=Search			52938645	350084536							1	MQTVGVHSIVQQLHRNSIQFTDGYEVKEDIGVGSYSVCKRCIHKATNMEFAVKIIDKSKRDPTEEIEILLRYGQHPNIITLKDVYDDGKYVYVVTELMKGGELLDKILRQKFFSEREASAVLFTITKTVEYLHAQGVVHRDLKPSNILYVDESGNPESIRICDFGFAKQLRAENGLLMTPCYTANFVAPEVLKRQGYDAACDIWSLGVLLYTMLTGYTPFANGPDDTPEEILARIGSGKFSLSGGYWNSVSDTAKDLVSKMLHVDPHQRLTAALVLRHPWIVHWDQLPQYQLNRQDAPHLVKGAMAATYSALNRNQSPVLEPVGRSTLAQRRGIKKITSTAL		Ribosomal protein S6 kinase alpha-3	KS6A3_HUMAN	P51812	B2R9V4 Q4VAP3 Q59H26 Q5JPK8 Q7Z3Z7						
452919	CN1CCN(CC1)C(=O)C(=C\c1c(-c2ccc(C)cc2)c2c(N)ncnc2n1CCCO)\C#N	InChI=1S/C25H29N7O2/c1-17-4-6-18(7-5-17)21-20(14-19(15-26)25(34)31-11-9-30(2)10-12-31)32(8-3-13-33)24-22(21)23(27)28-16-29-24/h4-7,14,16,33H,3,8-13H2,1-2H3,(H2,27,28,29)/b19-14+	ABLOIHSPETWVRL-XMHGGMMESA-N	259843	US9505766, 47	Ribosomal protein S6 kinase alpha-3 [399-740]			 41.3					8	22.00 C	US Patent		10.7270/Q2639NPR		aid1803661	US9505766	Taunton, Jr., JW; Maglathlin, R; Serafimova, I; Cohen, MS; Miller, R; Paavilainen, V; McFarland, J; Krishnan, S	The Regents of the University of California	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=259843	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=11170&target=Ribosomal+protein+S6+kinase+alpha-3+%5B399-740%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=259843&enzyme=Ribosomal+protein+S6+kinase+alpha-3+%5B399-740%5D&column=ki&startPg=0&Increment=50&submit=Search			52939144	350084537							1	MQTVGVHSIVQQLHRNSIQFTDGYEVKEDIGVGSYSVCKRCIHKATNMEFAVKIIDKSKRDPTEEIEILLRYGQHPNIITLKDVYDDGKYVYVVTELMKGGELLDKILRQKFFSEREASAVLFTITKTVEYLHAQGVVHRDLKPSNILYVDESGNPESIRICDFGFAKQLRAENGLLMTPCYTANFVAPEVLKRQGYDAACDIWSLGVLLYTMLTGYTPFANGPDDTPEEILARIGSGKFSLSGGYWNSVSDTAKDLVSKMLHVDPHQRLTAALVLRHPWIVHWDQLPQYQLNRQDAPHLVKGAMAATYSALNRNQSPVLEPVGRSTLAQRRGIKKITSTAL		Ribosomal protein S6 kinase alpha-3	KS6A3_HUMAN	P51812	B2R9V4 Q4VAP3 Q59H26 Q5JPK8 Q7Z3Z7						
452920	Cc1ccc(cc1)-c1c(\C=C(/C#N)C(=O)N2CCC2)n(CCCO)c2ncnc(N)c12	InChI=1S/C23H24N6O2/c1-15-4-6-16(7-5-15)19-18(12-17(13-24)23(31)28-8-2-9-28)29(10-3-11-30)22-20(19)21(25)26-14-27-22/h4-7,12,14,30H,2-3,8-11H2,1H3,(H2,25,26,27)/b17-12+	GOVRWUJNVPKOJV-SFQUDFHCSA-N	259844	US9505766, 48	Ribosomal protein S6 kinase alpha-3 [399-740]			 4.7					8	22.00 C	US Patent		10.7270/Q2639NPR		aid1803661	US9505766	Taunton, Jr., JW; Maglathlin, R; Serafimova, I; Cohen, MS; Miller, R; Paavilainen, V; McFarland, J; Krishnan, S	The Regents of the University of California	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=259844	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=11170&target=Ribosomal+protein+S6+kinase+alpha-3+%5B399-740%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=259844&enzyme=Ribosomal+protein+S6+kinase+alpha-3+%5B399-740%5D&column=ki&startPg=0&Increment=50&submit=Search			52939145	350084538							1	MQTVGVHSIVQQLHRNSIQFTDGYEVKEDIGVGSYSVCKRCIHKATNMEFAVKIIDKSKRDPTEEIEILLRYGQHPNIITLKDVYDDGKYVYVVTELMKGGELLDKILRQKFFSEREASAVLFTITKTVEYLHAQGVVHRDLKPSNILYVDESGNPESIRICDFGFAKQLRAENGLLMTPCYTANFVAPEVLKRQGYDAACDIWSLGVLLYTMLTGYTPFANGPDDTPEEILARIGSGKFSLSGGYWNSVSDTAKDLVSKMLHVDPHQRLTAALVLRHPWIVHWDQLPQYQLNRQDAPHLVKGAMAATYSALNRNQSPVLEPVGRSTLAQRRGIKKITSTAL		Ribosomal protein S6 kinase alpha-3	KS6A3_HUMAN	P51812	B2R9V4 Q4VAP3 Q59H26 Q5JPK8 Q7Z3Z7						
452921	CN(C)C(=O)C(=C\c1c(-c2ccc(C)cc2)c2c(N)ncnc2n1CCCO)\C#N	InChI=1S/C22H24N6O2/c1-14-5-7-15(8-6-14)18-17(11-16(12-23)22(30)27(2)3)28(9-4-10-29)21-19(18)20(24)25-13-26-21/h5-8,11,13,29H,4,9-10H2,1-3H3,(H2,24,25,26)/b16-11+	JOMCSJCBXRQYAV-LFIBNONCSA-N	259845	US9505766, 49	Ribosomal protein S6 kinase alpha-3 [399-740]			 6.5					8	22.00 C	US Patent		10.7270/Q2639NPR		aid1803661	US9505766	Taunton, Jr., JW; Maglathlin, R; Serafimova, I; Cohen, MS; Miller, R; Paavilainen, V; McFarland, J; Krishnan, S	The Regents of the University of California	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=259845	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=11170&target=Ribosomal+protein+S6+kinase+alpha-3+%5B399-740%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=259845&enzyme=Ribosomal+protein+S6+kinase+alpha-3+%5B399-740%5D&column=ki&startPg=0&Increment=50&submit=Search			52938768	350084539							1	MQTVGVHSIVQQLHRNSIQFTDGYEVKEDIGVGSYSVCKRCIHKATNMEFAVKIIDKSKRDPTEEIEILLRYGQHPNIITLKDVYDDGKYVYVVTELMKGGELLDKILRQKFFSEREASAVLFTITKTVEYLHAQGVVHRDLKPSNILYVDESGNPESIRICDFGFAKQLRAENGLLMTPCYTANFVAPEVLKRQGYDAACDIWSLGVLLYTMLTGYTPFANGPDDTPEEILARIGSGKFSLSGGYWNSVSDTAKDLVSKMLHVDPHQRLTAALVLRHPWIVHWDQLPQYQLNRQDAPHLVKGAMAATYSALNRNQSPVLEPVGRSTLAQRRGIKKITSTAL		Ribosomal protein S6 kinase alpha-3	KS6A3_HUMAN	P51812	B2R9V4 Q4VAP3 Q59H26 Q5JPK8 Q7Z3Z7						
452922	Cc1ccc(cc1)-c1c(\C=C(/C#N)C(=O)N2CC(O)C2)n(CCCO)c2ncnc(N)c12	InChI=1S/C23H24N6O3/c1-14-3-5-15(6-4-14)19-18(9-16(10-24)23(32)28-11-17(31)12-28)29(7-2-8-30)22-20(19)21(25)26-13-27-22/h3-6,9,13,17,30-31H,2,7-8,11-12H2,1H3,(H2,25,26,27)/b16-9+	LHVAADCVTGAJMC-CXUHLZMHSA-N	259846	US9505766, 50	Ribosomal protein S6 kinase alpha-3 [399-740]			 13.2					8	22.00 C	US Patent		10.7270/Q2639NPR		aid1803661	US9505766	Taunton, Jr., JW; Maglathlin, R; Serafimova, I; Cohen, MS; Miller, R; Paavilainen, V; McFarland, J; Krishnan, S	The Regents of the University of California	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=259846	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=11170&target=Ribosomal+protein+S6+kinase+alpha-3+%5B399-740%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=259846&enzyme=Ribosomal+protein+S6+kinase+alpha-3+%5B399-740%5D&column=ki&startPg=0&Increment=50&submit=Search			52939146	350084540							1	MQTVGVHSIVQQLHRNSIQFTDGYEVKEDIGVGSYSVCKRCIHKATNMEFAVKIIDKSKRDPTEEIEILLRYGQHPNIITLKDVYDDGKYVYVVTELMKGGELLDKILRQKFFSEREASAVLFTITKTVEYLHAQGVVHRDLKPSNILYVDESGNPESIRICDFGFAKQLRAENGLLMTPCYTANFVAPEVLKRQGYDAACDIWSLGVLLYTMLTGYTPFANGPDDTPEEILARIGSGKFSLSGGYWNSVSDTAKDLVSKMLHVDPHQRLTAALVLRHPWIVHWDQLPQYQLNRQDAPHLVKGAMAATYSALNRNQSPVLEPVGRSTLAQRRGIKKITSTAL		Ribosomal protein S6 kinase alpha-3	KS6A3_HUMAN	P51812	B2R9V4 Q4VAP3 Q59H26 Q5JPK8 Q7Z3Z7						
453005	Cc1ccc(cc1)-c1c(\C=C(/C#N)C(=O)N2CCOCC2)n(CCCO)c2ncnc(N)c12	InChI=1S/C24H26N6O3/c1-16-3-5-17(6-4-16)20-19(13-18(14-25)24(32)29-8-11-33-12-9-29)30(7-2-10-31)23-21(20)22(26)27-15-28-23/h3-6,13,15,31H,2,7-12H2,1H3,(H2,26,27,28)/b18-13+	MPGXYPKCYDKHRF-QGOAFFKASA-N	259858	US9505766, 62	Ribosomal protein S6 kinase alpha-3 [399-740]			 10.5					8	22.00 C	US Patent		10.7270/Q2639NPR		aid1803661	US9505766	Taunton, Jr., JW; Maglathlin, R; Serafimova, I; Cohen, MS; Miller, R; Paavilainen, V; McFarland, J; Krishnan, S	The Regents of the University of California	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=259858	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=11170&target=Ribosomal+protein+S6+kinase+alpha-3+%5B399-740%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=259858&enzyme=Ribosomal+protein+S6+kinase+alpha-3+%5B399-740%5D&column=ki&startPg=0&Increment=50&submit=Search			52939383	350084552							1	MQTVGVHSIVQQLHRNSIQFTDGYEVKEDIGVGSYSVCKRCIHKATNMEFAVKIIDKSKRDPTEEIEILLRYGQHPNIITLKDVYDDGKYVYVVTELMKGGELLDKILRQKFFSEREASAVLFTITKTVEYLHAQGVVHRDLKPSNILYVDESGNPESIRICDFGFAKQLRAENGLLMTPCYTANFVAPEVLKRQGYDAACDIWSLGVLLYTMLTGYTPFANGPDDTPEEILARIGSGKFSLSGGYWNSVSDTAKDLVSKMLHVDPHQRLTAALVLRHPWIVHWDQLPQYQLNRQDAPHLVKGAMAATYSALNRNQSPVLEPVGRSTLAQRRGIKKITSTAL		Ribosomal protein S6 kinase alpha-3	KS6A3_HUMAN	P51812	B2R9V4 Q4VAP3 Q59H26 Q5JPK8 Q7Z3Z7						
453006	Cc1ccc(cc1)-c1c(\C=C(/C#N)c2ccncc2)n(CCCO)c2ncnc(N)c12	InChI=1S/C24H22N6O/c1-16-3-5-18(6-4-16)21-20(13-19(14-25)17-7-9-27-10-8-17)30(11-2-12-31)24-22(21)23(26)28-15-29-24/h3-10,13,15,31H,2,11-12H2,1H3,(H2,26,28,29)/b19-13+	IEAISLSNZXMDMG-CPNJWEJPSA-N	259859	US9505766, 63	Ribosomal protein S6 kinase alpha-3 [399-740]			 71					8	22.00 C	US Patent		10.7270/Q2639NPR		aid1803661	US9505766	Taunton, Jr., JW; Maglathlin, R; Serafimova, I; Cohen, MS; Miller, R; Paavilainen, V; McFarland, J; Krishnan, S	The Regents of the University of California	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=259859	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=11170&target=Ribosomal+protein+S6+kinase+alpha-3+%5B399-740%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=259859&enzyme=Ribosomal+protein+S6+kinase+alpha-3+%5B399-740%5D&column=ki&startPg=0&Increment=50&submit=Search			52939756	350084553							1	MQTVGVHSIVQQLHRNSIQFTDGYEVKEDIGVGSYSVCKRCIHKATNMEFAVKIIDKSKRDPTEEIEILLRYGQHPNIITLKDVYDDGKYVYVVTELMKGGELLDKILRQKFFSEREASAVLFTITKTVEYLHAQGVVHRDLKPSNILYVDESGNPESIRICDFGFAKQLRAENGLLMTPCYTANFVAPEVLKRQGYDAACDIWSLGVLLYTMLTGYTPFANGPDDTPEEILARIGSGKFSLSGGYWNSVSDTAKDLVSKMLHVDPHQRLTAALVLRHPWIVHWDQLPQYQLNRQDAPHLVKGAMAATYSALNRNQSPVLEPVGRSTLAQRRGIKKITSTAL		Ribosomal protein S6 kinase alpha-3	KS6A3_HUMAN	P51812	B2R9V4 Q4VAP3 Q59H26 Q5JPK8 Q7Z3Z7						
453007	Cc1ccc(cc1)-c1c(\C=C(/C#N)C(=O)NC(C)(C)C)n(CCCO)c2ncnc(N)c12	InChI=1S/C24H28N6O2/c1-15-6-8-16(9-7-15)19-18(12-17(13-25)23(32)29-24(2,3)4)30(10-5-11-31)22-20(19)21(26)27-14-28-22/h6-9,12,14,31H,5,10-11H2,1-4H3,(H,29,32)(H2,26,27,28)/b17-12+	SVXJIKFFHBDTNV-SFQUDFHCSA-N	50403059	CHEMBL2216829::US9505766, 64	Ribosomal protein S6 kinase alpha-3 [399-740]			 4.5					8	22.00 C	US Patent		10.7270/Q2639NPR		aid1803661	US9505766	Taunton, Jr., JW; Maglathlin, R; Serafimova, I; Cohen, MS; Miller, R; Paavilainen, V; McFarland, J; Krishnan, S	The Regents of the University of California	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50403059	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=11170&target=Ribosomal+protein+S6+kinase+alpha-3+%5B399-740%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50403059&enzyme=Ribosomal+protein+S6+kinase+alpha-3+%5B399-740%5D&column=ki&startPg=0&Increment=50&submit=Search			52939498	163352083		CHEMBL2216829				ZINC95564455	1	MQTVGVHSIVQQLHRNSIQFTDGYEVKEDIGVGSYSVCKRCIHKATNMEFAVKIIDKSKRDPTEEIEILLRYGQHPNIITLKDVYDDGKYVYVVTELMKGGELLDKILRQKFFSEREASAVLFTITKTVEYLHAQGVVHRDLKPSNILYVDESGNPESIRICDFGFAKQLRAENGLLMTPCYTANFVAPEVLKRQGYDAACDIWSLGVLLYTMLTGYTPFANGPDDTPEEILARIGSGKFSLSGGYWNSVSDTAKDLVSKMLHVDPHQRLTAALVLRHPWIVHWDQLPQYQLNRQDAPHLVKGAMAATYSALNRNQSPVLEPVGRSTLAQRRGIKKITSTAL		Ribosomal protein S6 kinase alpha-3	KS6A3_HUMAN	P51812	B2R9V4 Q4VAP3 Q59H26 Q5JPK8 Q7Z3Z7						
453008	CN(C)CCN(C)C(=O)C(=C\c1c(-c2ccc(C)cc2)c2c(N)ncnc2n1CCCO)\C#N	InChI=1S/C25H31N7O2/c1-17-6-8-18(9-7-17)21-20(14-19(15-26)25(34)31(4)12-11-30(2)3)32(10-5-13-33)24-22(21)23(27)28-16-29-24/h6-9,14,16,33H,5,10-13H2,1-4H3,(H2,27,28,29)/b19-14+	GSFCMBOUJXZLQO-XMHGGMMESA-N	259860	US9505766, 65	Ribosomal protein S6 kinase alpha-3 [399-740]			 41.3					8	22.00 C	US Patent		10.7270/Q2639NPR		aid1803661	US9505766	Taunton, Jr., JW; Maglathlin, R; Serafimova, I; Cohen, MS; Miller, R; Paavilainen, V; McFarland, J; Krishnan, S	The Regents of the University of California	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=259860	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=11170&target=Ribosomal+protein+S6+kinase+alpha-3+%5B399-740%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=259860&enzyme=Ribosomal+protein+S6+kinase+alpha-3+%5B399-740%5D&column=ki&startPg=0&Increment=50&submit=Search			52939500	350084554							1	MQTVGVHSIVQQLHRNSIQFTDGYEVKEDIGVGSYSVCKRCIHKATNMEFAVKIIDKSKRDPTEEIEILLRYGQHPNIITLKDVYDDGKYVYVVTELMKGGELLDKILRQKFFSEREASAVLFTITKTVEYLHAQGVVHRDLKPSNILYVDESGNPESIRICDFGFAKQLRAENGLLMTPCYTANFVAPEVLKRQGYDAACDIWSLGVLLYTMLTGYTPFANGPDDTPEEILARIGSGKFSLSGGYWNSVSDTAKDLVSKMLHVDPHQRLTAALVLRHPWIVHWDQLPQYQLNRQDAPHLVKGAMAATYSALNRNQSPVLEPVGRSTLAQRRGIKKITSTAL		Ribosomal protein S6 kinase alpha-3	KS6A3_HUMAN	P51812	B2R9V4 Q4VAP3 Q59H26 Q5JPK8 Q7Z3Z7						
453009	Cc1ccc(cc1)-c1c(\C=C(/C#N)C(=O)NC(C)(CO)CO)n(CCCO)c2ncnc(N)c12	InChI=1S/C24H28N6O4/c1-15-4-6-16(7-5-15)19-18(10-17(11-25)23(34)29-24(2,12-32)13-33)30(8-3-9-31)22-20(19)21(26)27-14-28-22/h4-7,10,14,31-33H,3,8-9,12-13H2,1-2H3,(H,29,34)(H2,26,27,28)/b17-10+	WSGWSTKGKSCAAH-LICLKQGHSA-N	259861	US9505766, 66	Ribosomal protein S6 kinase alpha-3 [399-740]			 3.6					8	22.00 C	US Patent		10.7270/Q2639NPR		aid1803661	US9505766	Taunton, Jr., JW; Maglathlin, R; Serafimova, I; Cohen, MS; Miller, R; Paavilainen, V; McFarland, J; Krishnan, S	The Regents of the University of California	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=259861	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=11170&target=Ribosomal+protein+S6+kinase+alpha-3+%5B399-740%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=259861&enzyme=Ribosomal+protein+S6+kinase+alpha-3+%5B399-740%5D&column=ki&startPg=0&Increment=50&submit=Search			52939499	350084555							1	MQTVGVHSIVQQLHRNSIQFTDGYEVKEDIGVGSYSVCKRCIHKATNMEFAVKIIDKSKRDPTEEIEILLRYGQHPNIITLKDVYDDGKYVYVVTELMKGGELLDKILRQKFFSEREASAVLFTITKTVEYLHAQGVVHRDLKPSNILYVDESGNPESIRICDFGFAKQLRAENGLLMTPCYTANFVAPEVLKRQGYDAACDIWSLGVLLYTMLTGYTPFANGPDDTPEEILARIGSGKFSLSGGYWNSVSDTAKDLVSKMLHVDPHQRLTAALVLRHPWIVHWDQLPQYQLNRQDAPHLVKGAMAATYSALNRNQSPVLEPVGRSTLAQRRGIKKITSTAL		Ribosomal protein S6 kinase alpha-3	KS6A3_HUMAN	P51812	B2R9V4 Q4VAP3 Q59H26 Q5JPK8 Q7Z3Z7						
453010	Cc1ccc(cc1)-c1c(\C=C(/C#N)n2cncn2)n(CCCO)c2ncnc(N)c12	InChI=1S/C21H20N8O/c1-14-3-5-15(6-4-14)18-17(9-16(10-22)29-13-24-11-27-29)28(7-2-8-30)21-19(18)20(23)25-12-26-21/h3-6,9,11-13,30H,2,7-8H2,1H3,(H2,23,25,26)/b16-9+	MOWZNSSQRKLSGF-CXUHLZMHSA-N	259862	US9505766, 67	Ribosomal protein S6 kinase alpha-3 [399-740]			 14.8					8	22.00 C	US Patent		10.7270/Q2639NPR		aid1803661	US9505766	Taunton, Jr., JW; Maglathlin, R; Serafimova, I; Cohen, MS; Miller, R; Paavilainen, V; McFarland, J; Krishnan, S	The Regents of the University of California	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=259862	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=11170&target=Ribosomal+protein+S6+kinase+alpha-3+%5B399-740%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=259862&enzyme=Ribosomal+protein+S6+kinase+alpha-3+%5B399-740%5D&column=ki&startPg=0&Increment=50&submit=Search			52939758	350084556							1	MQTVGVHSIVQQLHRNSIQFTDGYEVKEDIGVGSYSVCKRCIHKATNMEFAVKIIDKSKRDPTEEIEILLRYGQHPNIITLKDVYDDGKYVYVVTELMKGGELLDKILRQKFFSEREASAVLFTITKTVEYLHAQGVVHRDLKPSNILYVDESGNPESIRICDFGFAKQLRAENGLLMTPCYTANFVAPEVLKRQGYDAACDIWSLGVLLYTMLTGYTPFANGPDDTPEEILARIGSGKFSLSGGYWNSVSDTAKDLVSKMLHVDPHQRLTAALVLRHPWIVHWDQLPQYQLNRQDAPHLVKGAMAATYSALNRNQSPVLEPVGRSTLAQRRGIKKITSTAL		Ribosomal protein S6 kinase alpha-3	KS6A3_HUMAN	P51812	B2R9V4 Q4VAP3 Q59H26 Q5JPK8 Q7Z3Z7						
453011	CC(C)NS(=O)(=O)C(=C\c1c(-c2ccc(C)cc2)c2c(N)ncnc2n1CCCO)\C#N	InChI=1S/C22H26N6O3S/c1-14(2)27-32(30,31)17(12-23)11-18-19(16-7-5-15(3)6-8-16)20-21(24)25-13-26-22(20)28(18)9-4-10-29/h5-8,11,13-14,27,29H,4,9-10H2,1-3H3,(H2,24,25,26)/b17-11+	MNFUNEVYKKTQFN-GZTJUZNOSA-N	259863	US9505766, 68	Ribosomal protein S6 kinase alpha-3 [399-740]			 2					8	22.00 C	US Patent		10.7270/Q2639NPR		aid1803661	US9505766	Taunton, Jr., JW; Maglathlin, R; Serafimova, I; Cohen, MS; Miller, R; Paavilainen, V; McFarland, J; Krishnan, S	The Regents of the University of California	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=259863	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=11170&target=Ribosomal+protein+S6+kinase+alpha-3+%5B399-740%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=259863&enzyme=Ribosomal+protein+S6+kinase+alpha-3+%5B399-740%5D&column=ki&startPg=0&Increment=50&submit=Search			68347890	350084557							1	MQTVGVHSIVQQLHRNSIQFTDGYEVKEDIGVGSYSVCKRCIHKATNMEFAVKIIDKSKRDPTEEIEILLRYGQHPNIITLKDVYDDGKYVYVVTELMKGGELLDKILRQKFFSEREASAVLFTITKTVEYLHAQGVVHRDLKPSNILYVDESGNPESIRICDFGFAKQLRAENGLLMTPCYTANFVAPEVLKRQGYDAACDIWSLGVLLYTMLTGYTPFANGPDDTPEEILARIGSGKFSLSGGYWNSVSDTAKDLVSKMLHVDPHQRLTAALVLRHPWIVHWDQLPQYQLNRQDAPHLVKGAMAATYSALNRNQSPVLEPVGRSTLAQRRGIKKITSTAL		Ribosomal protein S6 kinase alpha-3	KS6A3_HUMAN	P51812	B2R9V4 Q4VAP3 Q59H26 Q5JPK8 Q7Z3Z7						
453012	Cc1ccc(cc1)-c1c(C(=O)C(F)F)n(CCCO)c2ncnc(N)c12	InChI=1S/C18H18F2N4O2/c1-10-3-5-11(6-4-10)12-13-17(21)22-9-23-18(13)24(7-2-8-25)14(12)15(26)16(19)20/h3-6,9,16,25H,2,7-8H2,1H3,(H2,21,22,23)	ZIDZYKPYAIEZBO-UHFFFAOYSA-N	259864	US9505766, 69	Ribosomal protein S6 kinase alpha-3 [399-740]			>500					8	22.00 C	US Patent		10.7270/Q2639NPR		aid1803661	US9505766	Taunton, Jr., JW; Maglathlin, R; Serafimova, I; Cohen, MS; Miller, R; Paavilainen, V; McFarland, J; Krishnan, S	The Regents of the University of California	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=259864	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=11170&target=Ribosomal+protein+S6+kinase+alpha-3+%5B399-740%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=259864&enzyme=Ribosomal+protein+S6+kinase+alpha-3+%5B399-740%5D&column=ki&startPg=0&Increment=50&submit=Search			88947371	350084558							1	MQTVGVHSIVQQLHRNSIQFTDGYEVKEDIGVGSYSVCKRCIHKATNMEFAVKIIDKSKRDPTEEIEILLRYGQHPNIITLKDVYDDGKYVYVVTELMKGGELLDKILRQKFFSEREASAVLFTITKTVEYLHAQGVVHRDLKPSNILYVDESGNPESIRICDFGFAKQLRAENGLLMTPCYTANFVAPEVLKRQGYDAACDIWSLGVLLYTMLTGYTPFANGPDDTPEEILARIGSGKFSLSGGYWNSVSDTAKDLVSKMLHVDPHQRLTAALVLRHPWIVHWDQLPQYQLNRQDAPHLVKGAMAATYSALNRNQSPVLEPVGRSTLAQRRGIKKITSTAL		Ribosomal protein S6 kinase alpha-3	KS6A3_HUMAN	P51812	B2R9V4 Q4VAP3 Q59H26 Q5JPK8 Q7Z3Z7						
453013	Cc1ccc(cc1)-c1c(\C=C(/C#N)C(=O)NC23CC4CC(CC(C4)C2)C3)n(CCCO)c2ncnc(N)c12	InChI=1S/C30H34N6O2/c1-18-3-5-22(6-4-18)25-24(36(7-2-8-37)28-26(25)27(32)33-17-34-28)12-23(16-31)29(38)35-30-13-19-9-20(14-30)11-21(10-19)15-30/h3-6,12,17,19-21,37H,2,7-11,13-15H2,1H3,(H,35,38)(H2,32,33,34)/b23-12+	FRIZIFUZPGRSEX-FSJBWODESA-N	259865	US9505766, 70	Ribosomal protein S6 kinase alpha-3 [399-740]			>500					8	22.00 C	US Patent		10.7270/Q2639NPR		aid1803661	US9505766	Taunton, Jr., JW; Maglathlin, R; Serafimova, I; Cohen, MS; Miller, R; Paavilainen, V; McFarland, J; Krishnan, S	The Regents of the University of California	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=259865	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=11170&target=Ribosomal+protein+S6+kinase+alpha-3+%5B399-740%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=259865&enzyme=Ribosomal+protein+S6+kinase+alpha-3+%5B399-740%5D&column=ki&startPg=0&Increment=50&submit=Search			71245854	350084559							1	MQTVGVHSIVQQLHRNSIQFTDGYEVKEDIGVGSYSVCKRCIHKATNMEFAVKIIDKSKRDPTEEIEILLRYGQHPNIITLKDVYDDGKYVYVVTELMKGGELLDKILRQKFFSEREASAVLFTITKTVEYLHAQGVVHRDLKPSNILYVDESGNPESIRICDFGFAKQLRAENGLLMTPCYTANFVAPEVLKRQGYDAACDIWSLGVLLYTMLTGYTPFANGPDDTPEEILARIGSGKFSLSGGYWNSVSDTAKDLVSKMLHVDPHQRLTAALVLRHPWIVHWDQLPQYQLNRQDAPHLVKGAMAATYSALNRNQSPVLEPVGRSTLAQRRGIKKITSTAL		Ribosomal protein S6 kinase alpha-3	KS6A3_HUMAN	P51812	B2R9V4 Q4VAP3 Q59H26 Q5JPK8 Q7Z3Z7						
453014	Cc1ccc(cc1)-c1c(\C=C(/C#N)c2cc[n+]([O-])cc2)n(CCCO)c2ncnc(N)c12	InChI=1S/C24H22N6O2/c1-16-3-5-18(6-4-16)21-20(13-19(14-25)17-7-10-29(32)11-8-17)30(9-2-12-31)24-22(21)23(26)27-15-28-24/h3-8,10-11,13,15,31H,2,9,12H2,1H3,(H2,26,27,28)/b19-13+	HLVIJJBGDOMGGW-CPNJWEJPSA-N	259866	US9505766, 71	Ribosomal protein S6 kinase alpha-3 [399-740]			>500					8	22.00 C	US Patent		10.7270/Q2639NPR		aid1803661	US9505766	Taunton, Jr., JW; Maglathlin, R; Serafimova, I; Cohen, MS; Miller, R; Paavilainen, V; McFarland, J; Krishnan, S	The Regents of the University of California	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=259866	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=11170&target=Ribosomal+protein+S6+kinase+alpha-3+%5B399-740%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=259866&enzyme=Ribosomal+protein+S6+kinase+alpha-3+%5B399-740%5D&column=ki&startPg=0&Increment=50&submit=Search			52939760	350084560							1	MQTVGVHSIVQQLHRNSIQFTDGYEVKEDIGVGSYSVCKRCIHKATNMEFAVKIIDKSKRDPTEEIEILLRYGQHPNIITLKDVYDDGKYVYVVTELMKGGELLDKILRQKFFSEREASAVLFTITKTVEYLHAQGVVHRDLKPSNILYVDESGNPESIRICDFGFAKQLRAENGLLMTPCYTANFVAPEVLKRQGYDAACDIWSLGVLLYTMLTGYTPFANGPDDTPEEILARIGSGKFSLSGGYWNSVSDTAKDLVSKMLHVDPHQRLTAALVLRHPWIVHWDQLPQYQLNRQDAPHLVKGAMAATYSALNRNQSPVLEPVGRSTLAQRRGIKKITSTAL		Ribosomal protein S6 kinase alpha-3	KS6A3_HUMAN	P51812	B2R9V4 Q4VAP3 Q59H26 Q5JPK8 Q7Z3Z7						
453015	CN(CCO)C(=O)C(=C\c1c(-c2ccc(C)cc2)c2c(N)ncnc2n1CCCO)\C#N	InChI=1S/C23H26N6O3/c1-15-4-6-16(7-5-15)19-18(12-17(13-24)23(32)28(2)9-11-31)29(8-3-10-30)22-20(19)21(25)26-14-27-22/h4-7,12,14,30-31H,3,8-11H2,1-2H3,(H2,25,26,27)/b17-12+	YKHGZHUCBLLAOL-SFQUDFHCSA-N	259867	US9505766, 72	Ribosomal protein S6 kinase alpha-3 [399-740]			 17					8	22.00 C	US Patent		10.7270/Q2639NPR		aid1803661	US9505766	Taunton, Jr., JW; Maglathlin, R; Serafimova, I; Cohen, MS; Miller, R; Paavilainen, V; McFarland, J; Krishnan, S	The Regents of the University of California	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=259867	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=11170&target=Ribosomal+protein+S6+kinase+alpha-3+%5B399-740%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=259867&enzyme=Ribosomal+protein+S6+kinase+alpha-3+%5B399-740%5D&column=ki&startPg=0&Increment=50&submit=Search			52939502	350084561							1	MQTVGVHSIVQQLHRNSIQFTDGYEVKEDIGVGSYSVCKRCIHKATNMEFAVKIIDKSKRDPTEEIEILLRYGQHPNIITLKDVYDDGKYVYVVTELMKGGELLDKILRQKFFSEREASAVLFTITKTVEYLHAQGVVHRDLKPSNILYVDESGNPESIRICDFGFAKQLRAENGLLMTPCYTANFVAPEVLKRQGYDAACDIWSLGVLLYTMLTGYTPFANGPDDTPEEILARIGSGKFSLSGGYWNSVSDTAKDLVSKMLHVDPHQRLTAALVLRHPWIVHWDQLPQYQLNRQDAPHLVKGAMAATYSALNRNQSPVLEPVGRSTLAQRRGIKKITSTAL		Ribosomal protein S6 kinase alpha-3	KS6A3_HUMAN	P51812	B2R9V4 Q4VAP3 Q59H26 Q5JPK8 Q7Z3Z7						
453016	Cc1ccc(cc1)-c1c(\C=C(/C#N)C(=O)NC(C)(C)C(=O)OCC=C)n(CCCO)c2ncnc(N)c12	InChI=1S/C27H30N6O4/c1-5-13-37-26(36)27(3,4)32-25(35)19(15-28)14-20-21(18-9-7-17(2)8-10-18)22-23(29)30-16-31-24(22)33(20)11-6-12-34/h5,7-10,14,16,34H,1,6,11-13H2,2-4H3,(H,32,35)(H2,29,30,31)/b19-14+	XKPXPDVHQUUJTM-XMHGGMMESA-N	259868	US9505766, 73	Ribosomal protein S6 kinase alpha-3 [399-740]			 26.1					8	22.00 C	US Patent		10.7270/Q2639NPR		aid1803661	US9505766	Taunton, Jr., JW; Maglathlin, R; Serafimova, I; Cohen, MS; Miller, R; Paavilainen, V; McFarland, J; Krishnan, S	The Regents of the University of California	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=259868	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=11170&target=Ribosomal+protein+S6+kinase+alpha-3+%5B399-740%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=259868&enzyme=Ribosomal+protein+S6+kinase+alpha-3+%5B399-740%5D&column=ki&startPg=0&Increment=50&submit=Search			52939625	350084562							1	MQTVGVHSIVQQLHRNSIQFTDGYEVKEDIGVGSYSVCKRCIHKATNMEFAVKIIDKSKRDPTEEIEILLRYGQHPNIITLKDVYDDGKYVYVVTELMKGGELLDKILRQKFFSEREASAVLFTITKTVEYLHAQGVVHRDLKPSNILYVDESGNPESIRICDFGFAKQLRAENGLLMTPCYTANFVAPEVLKRQGYDAACDIWSLGVLLYTMLTGYTPFANGPDDTPEEILARIGSGKFSLSGGYWNSVSDTAKDLVSKMLHVDPHQRLTAALVLRHPWIVHWDQLPQYQLNRQDAPHLVKGAMAATYSALNRNQSPVLEPVGRSTLAQRRGIKKITSTAL		Ribosomal protein S6 kinase alpha-3	KS6A3_HUMAN	P51812	B2R9V4 Q4VAP3 Q59H26 Q5JPK8 Q7Z3Z7						
453017	CC(C)NC(=O)C(=C\c1c(-c2ccc(C)cc2)c2c(N)ncnc2n1CCCO)\C#N	InChI=1S/C23H26N6O2/c1-14(2)28-23(31)17(12-24)11-18-19(16-7-5-15(3)6-8-16)20-21(25)26-13-27-22(20)29(18)9-4-10-30/h5-8,11,13-14,30H,4,9-10H2,1-3H3,(H,28,31)(H2,25,26,27)/b17-11+	POTINGKLYOETSI-GZTJUZNOSA-N	259808	US9505766, 74::US9505766, CN-NHiPr (7)	Ribosomal protein S6 kinase alpha-3 [399-740]			>500					8	22.00 C	US Patent		10.7270/Q2639NPR		aid1803661	US9505766	Taunton, Jr., JW; Maglathlin, R; Serafimova, I; Cohen, MS; Miller, R; Paavilainen, V; McFarland, J; Krishnan, S	The Regents of the University of California	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=259808	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=11170&target=Ribosomal+protein+S6+kinase+alpha-3+%5B399-740%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=259808&enzyme=Ribosomal+protein+S6+kinase+alpha-3+%5B399-740%5D&column=ki&startPg=0&Increment=50&submit=Search			52938644	350084502							1	MQTVGVHSIVQQLHRNSIQFTDGYEVKEDIGVGSYSVCKRCIHKATNMEFAVKIIDKSKRDPTEEIEILLRYGQHPNIITLKDVYDDGKYVYVVTELMKGGELLDKILRQKFFSEREASAVLFTITKTVEYLHAQGVVHRDLKPSNILYVDESGNPESIRICDFGFAKQLRAENGLLMTPCYTANFVAPEVLKRQGYDAACDIWSLGVLLYTMLTGYTPFANGPDDTPEEILARIGSGKFSLSGGYWNSVSDTAKDLVSKMLHVDPHQRLTAALVLRHPWIVHWDQLPQYQLNRQDAPHLVKGAMAATYSALNRNQSPVLEPVGRSTLAQRRGIKKITSTAL		Ribosomal protein S6 kinase alpha-3	KS6A3_HUMAN	P51812	B2R9V4 Q4VAP3 Q59H26 Q5JPK8 Q7Z3Z7						
453018	CN(C)NC(=O)C(=C\c1c(-c2ccc(C)cc2)c2c(N)ncnc2n1CCCO)\C#N	InChI=1S/C22H25N7O2/c1-14-5-7-15(8-6-14)18-17(11-16(12-23)22(31)27-28(2)3)29(9-4-10-30)21-19(18)20(24)25-13-26-21/h5-8,11,13,30H,4,9-10H2,1-3H3,(H,27,31)(H2,24,25,26)/b16-11+	KEGOOQMDHSMWCY-LFIBNONCSA-N	259870	US9505766, 75	Ribosomal protein S6 kinase alpha-3 [399-740]			 4.8					8	22.00 C	US Patent		10.7270/Q2639NPR		aid1803661	US9505766	Taunton, Jr., JW; Maglathlin, R; Serafimova, I; Cohen, MS; Miller, R; Paavilainen, V; McFarland, J; Krishnan, S	The Regents of the University of California	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=259870	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=11170&target=Ribosomal+protein+S6+kinase+alpha-3+%5B399-740%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=259870&enzyme=Ribosomal+protein+S6+kinase+alpha-3+%5B399-740%5D&column=ki&startPg=0&Increment=50&submit=Search			52939628	350084563							1	MQTVGVHSIVQQLHRNSIQFTDGYEVKEDIGVGSYSVCKRCIHKATNMEFAVKIIDKSKRDPTEEIEILLRYGQHPNIITLKDVYDDGKYVYVVTELMKGGELLDKILRQKFFSEREASAVLFTITKTVEYLHAQGVVHRDLKPSNILYVDESGNPESIRICDFGFAKQLRAENGLLMTPCYTANFVAPEVLKRQGYDAACDIWSLGVLLYTMLTGYTPFANGPDDTPEEILARIGSGKFSLSGGYWNSVSDTAKDLVSKMLHVDPHQRLTAALVLRHPWIVHWDQLPQYQLNRQDAPHLVKGAMAATYSALNRNQSPVLEPVGRSTLAQRRGIKKITSTAL		Ribosomal protein S6 kinase alpha-3	KS6A3_HUMAN	P51812	B2R9V4 Q4VAP3 Q59H26 Q5JPK8 Q7Z3Z7						
453019	Cc1ccc(cc1)-c1c(\C=C(/C#N)c2cccnc2)n(CCCO)c2ncnc(N)c12	InChI=1S/C24H22N6O/c1-16-5-7-17(8-6-16)21-20(12-19(13-25)18-4-2-9-27-14-18)30(10-3-11-31)24-22(21)23(26)28-15-29-24/h2,4-9,12,14-15,31H,3,10-11H2,1H3,(H2,26,28,29)/b19-12+	NAJWGDOGTBBCJT-XDHOZWIPSA-N	259871	US9505766, 76	Ribosomal protein S6 kinase alpha-3 [399-740]			 224					8	22.00 C	US Patent		10.7270/Q2639NPR		aid1803661	US9505766	Taunton, Jr., JW; Maglathlin, R; Serafimova, I; Cohen, MS; Miller, R; Paavilainen, V; McFarland, J; Krishnan, S	The Regents of the University of California	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=259871	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=11170&target=Ribosomal+protein+S6+kinase+alpha-3+%5B399-740%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=259871&enzyme=Ribosomal+protein+S6+kinase+alpha-3+%5B399-740%5D&column=ki&startPg=0&Increment=50&submit=Search			68347837	350084564							1	MQTVGVHSIVQQLHRNSIQFTDGYEVKEDIGVGSYSVCKRCIHKATNMEFAVKIIDKSKRDPTEEIEILLRYGQHPNIITLKDVYDDGKYVYVVTELMKGGELLDKILRQKFFSEREASAVLFTITKTVEYLHAQGVVHRDLKPSNILYVDESGNPESIRICDFGFAKQLRAENGLLMTPCYTANFVAPEVLKRQGYDAACDIWSLGVLLYTMLTGYTPFANGPDDTPEEILARIGSGKFSLSGGYWNSVSDTAKDLVSKMLHVDPHQRLTAALVLRHPWIVHWDQLPQYQLNRQDAPHLVKGAMAATYSALNRNQSPVLEPVGRSTLAQRRGIKKITSTAL		Ribosomal protein S6 kinase alpha-3	KS6A3_HUMAN	P51812	B2R9V4 Q4VAP3 Q59H26 Q5JPK8 Q7Z3Z7						
453020	CONC(=O)C(=C\c1c(-c2ccc(C)cc2)c2c(N)ncnc2n1CCCO)\C#N	InChI=1S/C21H22N6O3/c1-13-4-6-14(7-5-13)17-16(10-15(11-22)21(29)26-30-2)27(8-3-9-28)20-18(17)19(23)24-12-25-20/h4-7,10,12,28H,3,8-9H2,1-2H3,(H,26,29)(H2,23,24,25)/b15-10+	OWNIBZDEHRWONY-XNTDXEJSSA-N	259872	US9505766, 77	Ribosomal protein S6 kinase alpha-3 [399-740]			 12.6					8	22.00 C	US Patent		10.7270/Q2639NPR		aid1803661	US9505766	Taunton, Jr., JW; Maglathlin, R; Serafimova, I; Cohen, MS; Miller, R; Paavilainen, V; McFarland, J; Krishnan, S	The Regents of the University of California	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=259872	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=11170&target=Ribosomal+protein+S6+kinase+alpha-3+%5B399-740%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=259872&enzyme=Ribosomal+protein+S6+kinase+alpha-3+%5B399-740%5D&column=ki&startPg=0&Increment=50&submit=Search			52939626	350084565							1	MQTVGVHSIVQQLHRNSIQFTDGYEVKEDIGVGSYSVCKRCIHKATNMEFAVKIIDKSKRDPTEEIEILLRYGQHPNIITLKDVYDDGKYVYVVTELMKGGELLDKILRQKFFSEREASAVLFTITKTVEYLHAQGVVHRDLKPSNILYVDESGNPESIRICDFGFAKQLRAENGLLMTPCYTANFVAPEVLKRQGYDAACDIWSLGVLLYTMLTGYTPFANGPDDTPEEILARIGSGKFSLSGGYWNSVSDTAKDLVSKMLHVDPHQRLTAALVLRHPWIVHWDQLPQYQLNRQDAPHLVKGAMAATYSALNRNQSPVLEPVGRSTLAQRRGIKKITSTAL		Ribosomal protein S6 kinase alpha-3	KS6A3_HUMAN	P51812	B2R9V4 Q4VAP3 Q59H26 Q5JPK8 Q7Z3Z7						
453021	Cc1csc(n1)C(=C\c1c(-c2ccc(C)cc2)c2c(N)ncnc2n1CCCO)\C#N	InChI=1S/C23H22N6OS/c1-14-4-6-16(7-5-14)19-18(10-17(11-24)23-28-15(2)12-31-23)29(8-3-9-30)22-20(19)21(25)26-13-27-22/h4-7,10,12-13,30H,3,8-9H2,1-2H3,(H2,25,26,27)/b17-10+	JINCFVYKIKUKAU-LICLKQGHSA-N	259873	US9505766, 78	Ribosomal protein S6 kinase alpha-3 [399-740]			 30.4					8	22.00 C	US Patent		10.7270/Q2639NPR		aid1803661	US9505766	Taunton, Jr., JW; Maglathlin, R; Serafimova, I; Cohen, MS; Miller, R; Paavilainen, V; McFarland, J; Krishnan, S	The Regents of the University of California	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=259873	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=11170&target=Ribosomal+protein+S6+kinase+alpha-3+%5B399-740%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=259873&enzyme=Ribosomal+protein+S6+kinase+alpha-3+%5B399-740%5D&column=ki&startPg=0&Increment=50&submit=Search			52939757	350084566							1	MQTVGVHSIVQQLHRNSIQFTDGYEVKEDIGVGSYSVCKRCIHKATNMEFAVKIIDKSKRDPTEEIEILLRYGQHPNIITLKDVYDDGKYVYVVTELMKGGELLDKILRQKFFSEREASAVLFTITKTVEYLHAQGVVHRDLKPSNILYVDESGNPESIRICDFGFAKQLRAENGLLMTPCYTANFVAPEVLKRQGYDAACDIWSLGVLLYTMLTGYTPFANGPDDTPEEILARIGSGKFSLSGGYWNSVSDTAKDLVSKMLHVDPHQRLTAALVLRHPWIVHWDQLPQYQLNRQDAPHLVKGAMAATYSALNRNQSPVLEPVGRSTLAQRRGIKKITSTAL		Ribosomal protein S6 kinase alpha-3	KS6A3_HUMAN	P51812	B2R9V4 Q4VAP3 Q59H26 Q5JPK8 Q7Z3Z7						
453022	Cc1ccc(cc1)-c1c(\C=C(/C#N)n2cccn2)n(CCCO)c2ncnc(N)c12	InChI=1S/C22H21N7O/c1-15-4-6-16(7-5-15)19-18(12-17(13-23)29-10-2-8-27-29)28(9-3-11-30)22-20(19)21(24)25-14-26-22/h2,4-8,10,12,14,30H,3,9,11H2,1H3,(H2,24,25,26)/b17-12+	XZPOPAZWILYPAH-SFQUDFHCSA-N	259874	US9505766, 79	Ribosomal protein S6 kinase alpha-3 [399-740]			 274					8	22.00 C	US Patent		10.7270/Q2639NPR		aid1803661	US9505766	Taunton, Jr., JW; Maglathlin, R; Serafimova, I; Cohen, MS; Miller, R; Paavilainen, V; McFarland, J; Krishnan, S	The Regents of the University of California	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=259874	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=11170&target=Ribosomal+protein+S6+kinase+alpha-3+%5B399-740%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=259874&enzyme=Ribosomal+protein+S6+kinase+alpha-3+%5B399-740%5D&column=ki&startPg=0&Increment=50&submit=Search			68347596	350084567							1	MQTVGVHSIVQQLHRNSIQFTDGYEVKEDIGVGSYSVCKRCIHKATNMEFAVKIIDKSKRDPTEEIEILLRYGQHPNIITLKDVYDDGKYVYVVTELMKGGELLDKILRQKFFSEREASAVLFTITKTVEYLHAQGVVHRDLKPSNILYVDESGNPESIRICDFGFAKQLRAENGLLMTPCYTANFVAPEVLKRQGYDAACDIWSLGVLLYTMLTGYTPFANGPDDTPEEILARIGSGKFSLSGGYWNSVSDTAKDLVSKMLHVDPHQRLTAALVLRHPWIVHWDQLPQYQLNRQDAPHLVKGAMAATYSALNRNQSPVLEPVGRSTLAQRRGIKKITSTAL		Ribosomal protein S6 kinase alpha-3	KS6A3_HUMAN	P51812	B2R9V4 Q4VAP3 Q59H26 Q5JPK8 Q7Z3Z7						
453023	Cc1ccc(cc1)-c1c(\C=C(/C#N)n2ccnn2)n(CCCO)c2ncnc(N)c12	InChI=1S/C21H20N8O/c1-14-3-5-15(6-4-14)18-17(11-16(12-22)29-9-7-26-27-29)28(8-2-10-30)21-19(18)20(23)24-13-25-21/h3-7,9,11,13,30H,2,8,10H2,1H3,(H2,23,24,25)/b16-11+	SSSVFBLQTNYBIU-LFIBNONCSA-N	259875	US9505766, 80	Ribosomal protein S6 kinase alpha-3 [399-740]			 20.9					8	22.00 C	US Patent		10.7270/Q2639NPR		aid1803661	US9505766	Taunton, Jr., JW; Maglathlin, R; Serafimova, I; Cohen, MS; Miller, R; Paavilainen, V; McFarland, J; Krishnan, S	The Regents of the University of California	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=259875	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=11170&target=Ribosomal+protein+S6+kinase+alpha-3+%5B399-740%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=259875&enzyme=Ribosomal+protein+S6+kinase+alpha-3+%5B399-740%5D&column=ki&startPg=0&Increment=50&submit=Search			52939759	350084568							1	MQTVGVHSIVQQLHRNSIQFTDGYEVKEDIGVGSYSVCKRCIHKATNMEFAVKIIDKSKRDPTEEIEILLRYGQHPNIITLKDVYDDGKYVYVVTELMKGGELLDKILRQKFFSEREASAVLFTITKTVEYLHAQGVVHRDLKPSNILYVDESGNPESIRICDFGFAKQLRAENGLLMTPCYTANFVAPEVLKRQGYDAACDIWSLGVLLYTMLTGYTPFANGPDDTPEEILARIGSGKFSLSGGYWNSVSDTAKDLVSKMLHVDPHQRLTAALVLRHPWIVHWDQLPQYQLNRQDAPHLVKGAMAATYSALNRNQSPVLEPVGRSTLAQRRGIKKITSTAL		Ribosomal protein S6 kinase alpha-3	KS6A3_HUMAN	P51812	B2R9V4 Q4VAP3 Q59H26 Q5JPK8 Q7Z3Z7						
453024	COc1cc(cc(OC)c1OC)-c1n[nH]c2ccc(\C=C(/C#N)C(=O)NC(C)(C)CO)cc12	InChI=1S/C24H26N4O5/c1-24(2,13-29)26-23(30)16(12-25)8-14-6-7-18-17(9-14)21(28-27-18)15-10-19(31-3)22(33-5)20(11-15)32-4/h6-11,29H,13H2,1-5H3,(H,26,30)(H,27,28)/b16-8+	FCCMYBKAZCDQGX-LZYBPNLTSA-N	259876	US9505766, 81	Ribosomal protein S6 kinase alpha-3 [399-740]			 3					8	22.00 C	US Patent		10.7270/Q2639NPR		aid1803661	US9505766	Taunton, Jr., JW; Maglathlin, R; Serafimova, I; Cohen, MS; Miller, R; Paavilainen, V; McFarland, J; Krishnan, S	The Regents of the University of California	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=259876	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=11170&target=Ribosomal+protein+S6+kinase+alpha-3+%5B399-740%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=259876&enzyme=Ribosomal+protein+S6+kinase+alpha-3+%5B399-740%5D&column=ki&startPg=0&Increment=50&submit=Search			131954197	350084569							1	MQTVGVHSIVQQLHRNSIQFTDGYEVKEDIGVGSYSVCKRCIHKATNMEFAVKIIDKSKRDPTEEIEILLRYGQHPNIITLKDVYDDGKYVYVVTELMKGGELLDKILRQKFFSEREASAVLFTITKTVEYLHAQGVVHRDLKPSNILYVDESGNPESIRICDFGFAKQLRAENGLLMTPCYTANFVAPEVLKRQGYDAACDIWSLGVLLYTMLTGYTPFANGPDDTPEEILARIGSGKFSLSGGYWNSVSDTAKDLVSKMLHVDPHQRLTAALVLRHPWIVHWDQLPQYQLNRQDAPHLVKGAMAATYSALNRNQSPVLEPVGRSTLAQRRGIKKITSTAL		Ribosomal protein S6 kinase alpha-3	KS6A3_HUMAN	P51812	B2R9V4 Q4VAP3 Q59H26 Q5JPK8 Q7Z3Z7						
453025	NC(=O)C(=C\c1ccc2[nH]nc(-c3cccnc3)c2c1)\C#N	InChI=1S/C16H11N5O/c17-8-12(16(18)22)6-10-3-4-14-13(7-10)15(21-20-14)11-2-1-5-19-9-11/h1-7,9H,(H2,18,22)(H,20,21)/b12-6+	FVHAHVQBXNWVHO-WUXMJOGZSA-N	259877	US9505766, 82	Ribosomal protein S6 kinase alpha-3 [399-740]			 41					8	22.00 C	US Patent		10.7270/Q2639NPR		aid1803661	US9505766	Taunton, Jr., JW; Maglathlin, R; Serafimova, I; Cohen, MS; Miller, R; Paavilainen, V; McFarland, J; Krishnan, S	The Regents of the University of California	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=259877	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=11170&target=Ribosomal+protein+S6+kinase+alpha-3+%5B399-740%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=259877&enzyme=Ribosomal+protein+S6+kinase+alpha-3+%5B399-740%5D&column=ki&startPg=0&Increment=50&submit=Search			131954198	350084570							1	MQTVGVHSIVQQLHRNSIQFTDGYEVKEDIGVGSYSVCKRCIHKATNMEFAVKIIDKSKRDPTEEIEILLRYGQHPNIITLKDVYDDGKYVYVVTELMKGGELLDKILRQKFFSEREASAVLFTITKTVEYLHAQGVVHRDLKPSNILYVDESGNPESIRICDFGFAKQLRAENGLLMTPCYTANFVAPEVLKRQGYDAACDIWSLGVLLYTMLTGYTPFANGPDDTPEEILARIGSGKFSLSGGYWNSVSDTAKDLVSKMLHVDPHQRLTAALVLRHPWIVHWDQLPQYQLNRQDAPHLVKGAMAATYSALNRNQSPVLEPVGRSTLAQRRGIKKITSTAL		Ribosomal protein S6 kinase alpha-3	KS6A3_HUMAN	P51812	B2R9V4 Q4VAP3 Q59H26 Q5JPK8 Q7Z3Z7						
