BindingDB Reactant_set_id	Ligand SMILES	Ligand InChI	Ligand InChI Key	BindingDB MonomerID	BindingDB Ligand Name	Target Name	Target Source Organism According to Curator or DataSource	Ki (nM)	IC50 (nM)	Kd (nM)	EC50 (nM)	kon (M-1-s-1)	koff (s-1)	pH	Temp (C)	Curation/DataSource	Article DOI	BindingDB Entry DOI	PMID	PubChem AID	Patent Number	Authors	Institution	Link to Ligand in BindingDB	Link to Target in BindingDB	Link to Ligand-Target Pair in BindingDB	Ligand HET ID in PDB	PDB ID(s) for Ligand-Target Complex	PubChem CID of Ligand	PubChem SID of Ligand	ChEBI ID of Ligand	ChEMBL ID of Ligand	DrugBank ID of Ligand	IUPHAR_GRAC ID of Ligand	KEGG ID of Ligand	ZINC ID of Ligand	Number of Protein Chains in Target (>1 implies a multichain complex)	BindingDB Target Chain Sequence	PDB ID(s) of Target Chain	UniProt (SwissProt) Recommended Name of Target Chain	UniProt (SwissProt) Entry Name of Target Chain	UniProt (SwissProt) Primary ID of Target Chain	UniProt (SwissProt) Secondary ID(s) of Target Chain	UniProt (SwissProt) Alternative ID(s) of Target Chain	UniProt (TrEMBL) Submitted Name of Target Chain	UniProt (TrEMBL) Entry Name of Target Chain	UniProt (TrEMBL) Primary ID of Target Chain	UniProt (TrEMBL) Secondary ID(s) of Target Chain	UniProt (TrEMBL) Alternative ID(s) of Target Chain
50492072	CN1CCN(CC1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(N)cc1	InChI=1S/C24H24F3N5O2/c1-31-8-10-32(11-9-31)21-7-4-16(15-2-5-17(28)6-3-15)12-20(21)30-23(34)18-14-29-22(33)13-19(18)24(25,26)27/h2-7,12-14H,8-11,28H2,1H3,(H,29,33)(H,30,34)	SSJVLCZVKGGJJO-UHFFFAOYSA-N	50164773	CHEMBL3799127	WD repeat-containing protein 5				 40						ChEMBL	10.1021/acs.jmedchem.5b01630	10.7270/Q2VT1V0C	26958703			Getlik, M; Smil, D; Zepeda-Velázquez, C; Bolshan, Y; Poda, G; Wu, H; Dong, A; Kuznetsova, E; Marcellus, R; Senisterra, G; Dombrovski, L; Hajian, T; Kiyota, T; Schapira, M; Arrowsmith, CH; Brown, PJ; Vedadi, M; Al-Awar, R	Ontario Institute for Cancer Research	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50164773	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50164773&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			127047790	104050452		CHEMBL3799127				ZINC28522130	1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50492073	CN1CCN(CC1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cnn(CCN2CCOCC2)c1	InChI=1S/C27H32F3N7O3/c1-34-4-7-36(8-5-34)24-3-2-19(20-16-32-37(18-20)9-6-35-10-12-40-13-11-35)14-23(24)33-26(39)21-17-31-25(38)15-22(21)27(28,29)30/h2-3,14-18H,4-13H2,1H3,(H,31,38)(H,33,39)	YKVQAEICJDUVNC-UHFFFAOYSA-N	50164785	CHEMBL3797967	WD repeat-containing protein 5				 210						ChEMBL	10.1021/acs.jmedchem.5b01630	10.7270/Q2VT1V0C	26958703			Getlik, M; Smil, D; Zepeda-Velázquez, C; Bolshan, Y; Poda, G; Wu, H; Dong, A; Kuznetsova, E; Marcellus, R; Senisterra, G; Dombrovski, L; Hajian, T; Kiyota, T; Schapira, M; Arrowsmith, CH; Brown, PJ; Vedadi, M; Al-Awar, R	Ontario Institute for Cancer Research	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50164785	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50164785&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			127047791	341097530		CHEMBL3797967					1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50492074	CN1CCN(CC1)c1ccc(cc1NC(=O)c1ccc(F)c(C)c1Cl)[N+]([O-])=O	InChI=1S/C19H20ClFN4O3/c1-12-15(21)5-4-14(18(12)20)19(26)22-16-11-13(25(27)28)3-6-17(16)24-9-7-23(2)8-10-24/h3-6,11H,7-10H2,1-2H3,(H,22,26)	QHWMIGPLLWYRIR-UHFFFAOYSA-N	50428271	CHEMBL2337032	WD repeat-containing protein 5				 380						ChEMBL	10.1021/acs.jmedchem.5b01630	10.7270/Q2VT1V0C	26958703			Getlik, M; Smil, D; Zepeda-Velázquez, C; Bolshan, Y; Poda, G; Wu, H; Dong, A; Kuznetsova, E; Marcellus, R; Senisterra, G; Dombrovski, L; Hajian, T; Kiyota, T; Schapira, M; Arrowsmith, CH; Brown, PJ; Vedadi, M; Al-Awar, R	Ontario Institute for Cancer Research	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50428271	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50428271&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	IA9	4IA9	70679466	164157146		CHEMBL2337032				ZINC95589389	1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50492075	CN1CCN(CC1)c1ccc(cc1NC(=O)c1cccc(C)c1)-c1cnc2ccccc2c1	InChI=1S/C28H28N4O/c1-20-6-5-8-23(16-20)28(33)30-26-18-21(10-11-27(26)32-14-12-31(2)13-15-32)24-17-22-7-3-4-9-25(22)29-19-24/h3-11,16-19H,12-15H2,1-2H3,(H,30,33)	SGTMEYAZQRHDJV-UHFFFAOYSA-N	50164786	CHEMBL3798573	WD repeat-containing protein 5				 720						ChEMBL	10.1021/acs.jmedchem.5b01630	10.7270/Q2VT1V0C	26958703			Getlik, M; Smil, D; Zepeda-Velázquez, C; Bolshan, Y; Poda, G; Wu, H; Dong, A; Kuznetsova, E; Marcellus, R; Senisterra, G; Dombrovski, L; Hajian, T; Kiyota, T; Schapira, M; Arrowsmith, CH; Brown, PJ; Vedadi, M; Al-Awar, R	Ontario Institute for Cancer Research	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50164786	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50164786&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	5ML	5EAL	91995965	341097531		CHEMBL3798573					1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50492076	CCC(CC)(NC(=O)C(C)C)C(=O)N[C@@H](CCCNC(N)=N)C(=O)NC1(CCCC1)C(=O)NC(c1ccccc1)c1ccccc1	InChI=1S/C35H51N7O4/c1-5-34(6-2,41-29(43)24(3)4)31(45)39-27(20-15-23-38-33(36)37)30(44)42-35(21-13-14-22-35)32(46)40-28(25-16-9-7-10-17-25)26-18-11-8-12-19-26/h7-12,16-19,24,27-28H,5-6,13-15,20-23H2,1-4H3,(H,39,45)(H,40,46)(H,41,43)(H,42,44)(H4,36,37,38)/t27-/m0/s1	BCIPILGGOSCOMC-MHZLTWQESA-N	200712	US9233086, 10A	WD repeat-containing protein 5			 2.9							ChEMBL	10.1021/acs.jmedchem.5b01630	10.7270/Q2VT1V0C	26958703			Getlik, M; Smil, D; Zepeda-Velázquez, C; Bolshan, Y; Poda, G; Wu, H; Dong, A; Kuznetsova, E; Marcellus, R; Senisterra, G; Dombrovski, L; Hajian, T; Kiyota, T; Schapira, M; Arrowsmith, CH; Brown, PJ; Vedadi, M; Al-Awar, R	Ontario Institute for Cancer Research	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=200712	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=200712&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			53356803	318834325							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50492078	CC[C@@H]1NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@@](C)(CCCCNC(=O)[C@H](NC1=O)c1ccccc1)NC(=O)C(C)C	InChI=1S/C29H46N8O5/c1-5-20-24(39)36-22(19-12-7-6-8-13-19)26(41)32-16-10-9-15-29(4,37-23(38)18(2)3)27(42)35-21(25(40)34-20)14-11-17-33-28(30)31/h6-8,12-13,18,20-22H,5,9-11,14-17H2,1-4H3,(H,32,41)(H,34,40)(H,35,42)(H,36,39)(H,37,38)(H4,30,31,33)/t20-,21-,22+,29+/m0/s1	SILRGLDFBXVGOQ-ZMROOPMESA-N	50164787	CHEMBL3798088	WD repeat-containing protein 5			 0.900000							ChEMBL	10.1021/acs.jmedchem.5b01630	10.7270/Q2VT1V0C	26958703			Getlik, M; Smil, D; Zepeda-Velázquez, C; Bolshan, Y; Poda, G; Wu, H; Dong, A; Kuznetsova, E; Marcellus, R; Senisterra, G; Dombrovski, L; Hajian, T; Kiyota, T; Schapira, M; Arrowsmith, CH; Brown, PJ; Vedadi, M; Al-Awar, R	Ontario Institute for Cancer Research	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50164787	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50164787&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			71586081	341097532		CHEMBL3798088					1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50492079	CN1CCN(CC1)c1ccc(cc1NC(=O)c1cc(C)cc(C)c1)[N+]([O-])=O	InChI=1S/C20H24N4O3/c1-14-10-15(2)12-16(11-14)20(25)21-18-13-17(24(26)27)4-5-19(18)23-8-6-22(3)7-9-23/h4-5,10-13H,6-9H2,1-3H3,(H,21,25)	GJFKROIMAOLXMH-UHFFFAOYSA-N	50164788	CHEMBL3800271	WD repeat-containing protein 5				 390						ChEMBL	10.1021/acs.jmedchem.5b01630	10.7270/Q2VT1V0C	26958703			Getlik, M; Smil, D; Zepeda-Velázquez, C; Bolshan, Y; Poda, G; Wu, H; Dong, A; Kuznetsova, E; Marcellus, R; Senisterra, G; Dombrovski, L; Hajian, T; Kiyota, T; Schapira, M; Arrowsmith, CH; Brown, PJ; Vedadi, M; Al-Awar, R	Ontario Institute for Cancer Research	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50164788	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50164788&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			127045996	341097533		CHEMBL3800271					1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50492080	CN1CCN(CC1)c1ccc(cc1NC(=O)c1cc(C)c(F)c(C)c1)[N+]([O-])=O	InChI=1S/C20H23FN4O3/c1-13-10-15(11-14(2)19(13)21)20(26)22-17-12-16(25(27)28)4-5-18(17)24-8-6-23(3)7-9-24/h4-5,10-12H,6-9H2,1-3H3,(H,22,26)	WNRFCVFYUVINJG-UHFFFAOYSA-N	50164789	CHEMBL3798578	WD repeat-containing protein 5				 330						ChEMBL	10.1021/acs.jmedchem.5b01630	10.7270/Q2VT1V0C	26958703			Getlik, M; Smil, D; Zepeda-Velázquez, C; Bolshan, Y; Poda, G; Wu, H; Dong, A; Kuznetsova, E; Marcellus, R; Senisterra, G; Dombrovski, L; Hajian, T; Kiyota, T; Schapira, M; Arrowsmith, CH; Brown, PJ; Vedadi, M; Al-Awar, R	Ontario Institute for Cancer Research	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50164789	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50164789&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			127046421	341097534		CHEMBL3798578					1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50492081	CN1CCN(CC1)c1ccc(cc1NC(=O)c1c(F)c(C)c(F)c(C)c1F)[N+]([O-])=O	InChI=1S/C20H21F3N4O3/c1-11-17(21)12(2)19(23)16(18(11)22)20(28)24-14-10-13(27(29)30)4-5-15(14)26-8-6-25(3)7-9-26/h4-5,10H,6-9H2,1-3H3,(H,24,28)	YVCXIHVVYPEYGI-UHFFFAOYSA-N	50164790	CHEMBL3797611	WD repeat-containing protein 5				 340						ChEMBL	10.1021/acs.jmedchem.5b01630	10.7270/Q2VT1V0C	26958703			Getlik, M; Smil, D; Zepeda-Velázquez, C; Bolshan, Y; Poda, G; Wu, H; Dong, A; Kuznetsova, E; Marcellus, R; Senisterra, G; Dombrovski, L; Hajian, T; Kiyota, T; Schapira, M; Arrowsmith, CH; Brown, PJ; Vedadi, M; Al-Awar, R	Ontario Institute for Cancer Research	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50164790	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50164790&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			127048151	341097535		CHEMBL3797611					1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50492082	CN1CCN(CC1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)[N+]([O-])=O	InChI=1S/C18H18F3N5O4/c1-24-4-6-25(7-5-24)15-3-2-11(26(29)30)8-14(15)23-17(28)12-10-22-16(27)9-13(12)18(19,20)21/h2-3,8-10H,4-7H2,1H3,(H,22,27)(H,23,28)	LXARWAORRXUDTM-UHFFFAOYSA-N	50164791	CHEMBL3799704	WD repeat-containing protein 5				 40						ChEMBL	10.1021/acs.jmedchem.5b01630	10.7270/Q2VT1V0C	26958703			Getlik, M; Smil, D; Zepeda-Velázquez, C; Bolshan, Y; Poda, G; Wu, H; Dong, A; Kuznetsova, E; Marcellus, R; Senisterra, G; Dombrovski, L; Hajian, T; Kiyota, T; Schapira, M; Arrowsmith, CH; Brown, PJ; Vedadi, M; Al-Awar, R	Ontario Institute for Cancer Research	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50164791	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50164791&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			127048152	341097536		CHEMBL3799704					1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50492083	CN1CCN(CC1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc2OCCc2c1	InChI=1S/C26H25F3N4O3/c1-32-7-9-33(10-8-32)22-4-2-17(16-3-5-23-18(12-16)6-11-36-23)13-21(22)31-25(35)19-15-30-24(34)14-20(19)26(27,28)29/h2-5,12-15H,6-11H2,1H3,(H,30,34)(H,31,35)	UAMABNCJOIOIEH-UHFFFAOYSA-N	50164792	CHEMBL3798198	WD repeat-containing protein 5				 40						ChEMBL	10.1021/acs.jmedchem.5b01630	10.7270/Q2VT1V0C	26958703			Getlik, M; Smil, D; Zepeda-Velázquez, C; Bolshan, Y; Poda, G; Wu, H; Dong, A; Kuznetsova, E; Marcellus, R; Senisterra, G; Dombrovski, L; Hajian, T; Kiyota, T; Schapira, M; Arrowsmith, CH; Brown, PJ; Vedadi, M; Al-Awar, R	Ontario Institute for Cancer Research	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50164792	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50164792&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			127046290	341097537		CHEMBL3798198					1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50492084	CN1CCN(CC1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cnc2ccccc2c1	InChI=1S/C27H24F3N5O2/c1-34-8-10-35(11-9-34)24-7-6-17(19-12-18-4-2-3-5-22(18)31-15-19)13-23(24)33-26(37)20-16-32-25(36)14-21(20)27(28,29)30/h2-7,12-16H,8-11H2,1H3,(H,32,36)(H,33,37)	BHSUCGLRVZHATB-UHFFFAOYSA-N	50164770	CHEMBL3799275	WD repeat-containing protein 5				 50						ChEMBL	10.1021/acs.jmedchem.5b01630	10.7270/Q2VT1V0C	26958703			Getlik, M; Smil, D; Zepeda-Velázquez, C; Bolshan, Y; Poda, G; Wu, H; Dong, A; Kuznetsova, E; Marcellus, R; Senisterra, G; Dombrovski, L; Hajian, T; Kiyota, T; Schapira, M; Arrowsmith, CH; Brown, PJ; Vedadi, M; Al-Awar, R	Ontario Institute for Cancer Research	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50164770	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50164770&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	37F	4QQE	76871930	104050449		CHEMBL3799275				ZINC28520610	1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50492085	CN1CCN(CC1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc2[nH]ccc2c1	InChI=1S/C26H24F3N5O2/c1-33-8-10-34(11-9-33)23-5-3-17(16-2-4-21-18(12-16)6-7-30-21)13-22(23)32-25(36)19-15-31-24(35)14-20(19)26(27,28)29/h2-7,12-15,30H,8-11H2,1H3,(H,31,35)(H,32,36)	YQJXVMGEVOIIMV-UHFFFAOYSA-N	50164793	CHEMBL3799840	WD repeat-containing protein 5				 50						ChEMBL	10.1021/acs.jmedchem.5b01630	10.7270/Q2VT1V0C	26958703			Getlik, M; Smil, D; Zepeda-Velázquez, C; Bolshan, Y; Poda, G; Wu, H; Dong, A; Kuznetsova, E; Marcellus, R; Senisterra, G; Dombrovski, L; Hajian, T; Kiyota, T; Schapira, M; Arrowsmith, CH; Brown, PJ; Vedadi, M; Al-Awar, R	Ontario Institute for Cancer Research	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50164793	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50164793&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			127046291	341097538		CHEMBL3799840					1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50492086	CN1CCN(CC1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cccc(CN2CCOCC2)c1	InChI=1S/C29H32F3N5O3/c1-35-7-9-37(10-8-35)26-6-5-22(21-4-2-3-20(15-21)19-36-11-13-40-14-12-36)16-25(26)34-28(39)23-18-33-27(38)17-24(23)29(30,31)32/h2-6,15-18H,7-14,19H2,1H3,(H,33,38)(H,34,39)	DJOVLOYCGXNVPI-UHFFFAOYSA-N	50164794	CHEMBL3798846::US11174250, Example Table4.1.1::US11319299, Comp. No. 57	WD repeat-containing protein 5				 30						ChEMBL	10.1021/acs.jmedchem.5b01630	10.7270/Q2VT1V0C	26958703			Getlik, M; Smil, D; Zepeda-Velázquez, C; Bolshan, Y; Poda, G; Wu, H; Dong, A; Kuznetsova, E; Marcellus, R; Senisterra, G; Dombrovski, L; Hajian, T; Kiyota, T; Schapira, M; Arrowsmith, CH; Brown, PJ; Vedadi, M; Al-Awar, R	Ontario Institute for Cancer Research	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50164794	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50164794&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	35Q	4QL1	91623360	341097539		CHEMBL3798846					1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50492087	CN1CCN(CC1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(NC(C)=O)nc1	InChI=1S/C25H25F3N6O3/c1-15(35)31-22-6-4-17(13-29-22)16-3-5-21(34-9-7-33(2)8-10-34)20(11-16)32-24(37)18-14-30-23(36)12-19(18)25(26,27)28/h3-6,11-14H,7-10H2,1-2H3,(H,30,36)(H,32,37)(H,29,31,35)	OJAXIKLEQGASLZ-UHFFFAOYSA-N	50164795	CHEMBL3799608	WD repeat-containing protein 5				 30						ChEMBL	10.1021/acs.jmedchem.5b01630	10.7270/Q2VT1V0C	26958703			Getlik, M; Smil, D; Zepeda-Velázquez, C; Bolshan, Y; Poda, G; Wu, H; Dong, A; Kuznetsova, E; Marcellus, R; Senisterra, G; Dombrovski, L; Hajian, T; Kiyota, T; Schapira, M; Arrowsmith, CH; Brown, PJ; Vedadi, M; Al-Awar, R	Ontario Institute for Cancer Research	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50164795	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50164795&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			127046292	341097540		CHEMBL3799608					1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50492088	CN1CCN(CC1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(N)nc1	InChI=1S/C23H23F3N6O2/c1-31-6-8-32(9-7-31)19-4-2-14(15-3-5-20(27)28-12-15)10-18(19)30-22(34)16-13-29-21(33)11-17(16)23(24,25)26/h2-5,10-13H,6-9H2,1H3,(H2,27,28)(H,29,33)(H,30,34)	QAFVKRAWTPAXFL-UHFFFAOYSA-N	50164796	CHEMBL3800054	WD repeat-containing protein 5				 50						ChEMBL	10.1021/acs.jmedchem.5b01630	10.7270/Q2VT1V0C	26958703			Getlik, M; Smil, D; Zepeda-Velázquez, C; Bolshan, Y; Poda, G; Wu, H; Dong, A; Kuznetsova, E; Marcellus, R; Senisterra, G; Dombrovski, L; Hajian, T; Kiyota, T; Schapira, M; Arrowsmith, CH; Brown, PJ; Vedadi, M; Al-Awar, R	Ontario Institute for Cancer Research	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50164796	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50164796&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			127047789	341097541		CHEMBL3800054					1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50505455	CN1CCN(CC1)c1ccc(cc1NC(=O)c1ccc(F)c(C)c1Cl)-c1ccncc1	InChI=1S/C24H24ClFN4O/c1-16-20(26)5-4-19(23(16)25)24(31)28-21-15-18(17-7-9-27-10-8-17)3-6-22(21)30-13-11-29(2)12-14-30/h3-10,15H,11-14H2,1-2H3,(H,28,31)	AICVIWJSFCXEOX-UHFFFAOYSA-N	50184787	CHEMBL3823308	WD repeat-containing protein 5				 133						ChEMBL	10.1016/j.ejmech.2016.04.032	10.7270/Q26H4KBP	27116709			Li, DD; Chen, WL; Xu, XL; Jiang, F; Wang, L; Xie, YY; Zhang, XJ; Guo, XK; You, QD; Sun, HP	China Pharmaceutical University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50184787	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50184787&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			127052837	104069106		CHEMBL3823308				ZINC40566038	1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50505456	CN1CCN(CC1)c1ccc(cc1NC(=O)c1cc(c(F)c(C)c1Cl)[N+]([O-])=O)[N+]([O-])=O	InChI=1S/C19H19ClFN5O5/c1-11-17(20)13(10-16(18(11)21)26(30)31)19(27)22-14-9-12(25(28)29)3-4-15(14)24-7-5-23(2)6-8-24/h3-4,9-10H,5-8H2,1-2H3,(H,22,27)	ZVZKRCIQYYCPMS-UHFFFAOYSA-N	50184789	CHEMBL3822691	WD repeat-containing protein 5				 343						ChEMBL	10.1016/j.ejmech.2016.04.032	10.7270/Q26H4KBP	27116709			Li, DD; Chen, WL; Xu, XL; Jiang, F; Wang, L; Xie, YY; Zhang, XJ; Guo, XK; You, QD; Sun, HP	China Pharmaceutical University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50184789	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50184789&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			127049253	104069108		CHEMBL3822691				ZINC01650372	1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50505621	CN1CCN(CC1)c1ccc(N)cc1NC(=O)c1ccc(F)c(C)c1Cl	InChI=1S/C19H22ClFN4O/c1-12-15(21)5-4-14(18(12)20)19(26)23-16-11-13(22)3-6-17(16)25-9-7-24(2)8-10-25/h3-6,11H,7-10,22H2,1-2H3,(H,23,26)	GRCZQAJZPPEKIZ-UHFFFAOYSA-N	50184790	CHEMBL3822666	WD repeat-containing protein 5			>20000							ChEMBL	10.1016/j.ejmech.2016.04.032	10.7270/Q26H4KBP	27116709			Li, DD; Chen, WL; Xu, XL; Jiang, F; Wang, L; Xie, YY; Zhang, XJ; Guo, XK; You, QD; Sun, HP	China Pharmaceutical University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50184790	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50184790&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			127050095	346550432		CHEMBL3822666					1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50505622	CN1CCN(CC1)c1ccc(cc1NC(=O)c1ccc(F)c(C)c1Cl)-c1cccc(c1)C(O)=O	InChI=1S/C26H25ClFN3O3/c1-16-21(28)8-7-20(24(16)27)25(32)29-22-15-18(17-4-3-5-19(14-17)26(33)34)6-9-23(22)31-12-10-30(2)11-13-31/h3-9,14-15H,10-13H2,1-2H3,(H,29,32)(H,33,34)	HWZFZBAVHVXKDN-UHFFFAOYSA-N	50184791	CHEMBL3823562	WD repeat-containing protein 5			 1604							ChEMBL	10.1016/j.ejmech.2016.04.032	10.7270/Q26H4KBP	27116709			Li, DD; Chen, WL; Xu, XL; Jiang, F; Wang, L; Xie, YY; Zhang, XJ; Guo, XK; You, QD; Sun, HP	China Pharmaceutical University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50184791	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50184791&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			127050385	346550433		CHEMBL3823562					1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50505623	CN1CCN(CC1)c1ccc(cc1NC(=O)c1ccc(F)c(C)c1Cl)-c1ccc(cc1)C(O)=O	InChI=1S/C26H25ClFN3O3/c1-16-21(28)9-8-20(24(16)27)25(32)29-22-15-19(17-3-5-18(6-4-17)26(33)34)7-10-23(22)31-13-11-30(2)12-14-31/h3-10,15H,11-14H2,1-2H3,(H,29,32)(H,33,34)	LCAMBAGLMBTSDA-UHFFFAOYSA-N	50184950	CHEMBL3823415	WD repeat-containing protein 5			 661							ChEMBL	10.1016/j.ejmech.2016.04.032	10.7270/Q26H4KBP	27116709			Li, DD; Chen, WL; Xu, XL; Jiang, F; Wang, L; Xie, YY; Zhang, XJ; Guo, XK; You, QD; Sun, HP	China Pharmaceutical University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50184950	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50184950&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			127048565	346550434		CHEMBL3823415					1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50505624	CN1CCN(CC1)c1ccc(cc1NC(=O)c1ccc(F)c(C)c1Cl)-c1ccc(cc1)C#N	InChI=1S/C26H24ClFN4O/c1-17-22(28)9-8-21(25(17)27)26(33)30-23-15-20(19-5-3-18(16-29)4-6-19)7-10-24(23)32-13-11-31(2)12-14-32/h3-10,15H,11-14H2,1-2H3,(H,30,33)	NKFXPDGOKFTCNC-UHFFFAOYSA-N	50184951	CHEMBL3823328	WD repeat-containing protein 5			 199							ChEMBL	10.1016/j.ejmech.2016.04.032	10.7270/Q26H4KBP	27116709			Li, DD; Chen, WL; Xu, XL; Jiang, F; Wang, L; Xie, YY; Zhang, XJ; Guo, XK; You, QD; Sun, HP	China Pharmaceutical University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50184951	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50184951&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			127050386	346550435		CHEMBL3823328					1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50505625	CN1CCN(CC1)c1ccc(cc1NC(=O)c1ccc(F)c(C)c1Cl)-c1ccccc1	InChI=1S/C25H25ClFN3O/c1-17-21(27)10-9-20(24(17)26)25(31)28-22-16-19(18-6-4-3-5-7-18)8-11-23(22)30-14-12-29(2)13-15-30/h3-11,16H,12-15H2,1-2H3,(H,28,31)	IJGXSYJCQSUICM-UHFFFAOYSA-N	50184952	CHEMBL3823476	WD repeat-containing protein 5			 466							ChEMBL	10.1016/j.ejmech.2016.04.032	10.7270/Q26H4KBP	27116709			Li, DD; Chen, WL; Xu, XL; Jiang, F; Wang, L; Xie, YY; Zhang, XJ; Guo, XK; You, QD; Sun, HP	China Pharmaceutical University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50184952	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50184952&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			127050387	346550436		CHEMBL3823476					1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50505626	CN1CCN(CC1)c1ccc(cc1NC(=O)c1ccc(F)c(C)c1Cl)-c1ccc(F)cc1	InChI=1S/C25H24ClF2N3O/c1-16-21(28)9-8-20(24(16)26)25(32)29-22-15-18(17-3-6-19(27)7-4-17)5-10-23(22)31-13-11-30(2)12-14-31/h3-10,15H,11-14H2,1-2H3,(H,29,32)	BAJACDAZJADWDF-UHFFFAOYSA-N	50184954	CHEMBL3822660	WD repeat-containing protein 5			 393							ChEMBL	10.1016/j.ejmech.2016.04.032	10.7270/Q26H4KBP	27116709			Li, DD; Chen, WL; Xu, XL; Jiang, F; Wang, L; Xie, YY; Zhang, XJ; Guo, XK; You, QD; Sun, HP	China Pharmaceutical University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50184954	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50184954&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			127052836	346550437		CHEMBL3822660					1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50505627	CN1CCN(CC1)c1ccc(cc1NC(=O)c1ccc(F)c(C)c1Cl)-c1ccncc1	InChI=1S/C24H24ClFN4O/c1-16-20(26)5-4-19(23(16)25)24(31)28-21-15-18(17-7-9-27-10-8-17)3-6-22(21)30-13-11-29(2)12-14-30/h3-10,15H,11-14H2,1-2H3,(H,28,31)	AICVIWJSFCXEOX-UHFFFAOYSA-N	50184787	CHEMBL3823308	WD repeat-containing protein 5			 104							ChEMBL	10.1016/j.ejmech.2016.04.032	10.7270/Q26H4KBP	27116709			Li, DD; Chen, WL; Xu, XL; Jiang, F; Wang, L; Xie, YY; Zhang, XJ; Guo, XK; You, QD; Sun, HP	China Pharmaceutical University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50184787	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50184787&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			127052837	104069106		CHEMBL3823308				ZINC40566038	1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50505628	CN1CCN(CC1)c1ccc(cc1NC(=O)c1ccc(F)c(C)c1Cl)-c1cncnc1	InChI=1S/C23H23ClFN5O/c1-15-19(25)5-4-18(22(15)24)23(31)28-20-11-16(17-12-26-14-27-13-17)3-6-21(20)30-9-7-29(2)8-10-30/h3-6,11-14H,7-10H2,1-2H3,(H,28,31)	YAWMNDGQFSPKNM-UHFFFAOYSA-N	50184955	CHEMBL3824206	WD repeat-containing protein 5			 733							ChEMBL	10.1016/j.ejmech.2016.04.032	10.7270/Q26H4KBP	27116709			Li, DD; Chen, WL; Xu, XL; Jiang, F; Wang, L; Xie, YY; Zhang, XJ; Guo, XK; You, QD; Sun, HP	China Pharmaceutical University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50184955	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50184955&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			127048926	346550438		CHEMBL3824206					1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50505629	CN1CCN(CC1)c1ccc(cc1NC(=O)c1ccc(F)c(C)c1Cl)-c1ccc(cc1)[N+]([O-])=O	InChI=1S/C25H24ClFN4O3/c1-16-21(27)9-8-20(24(16)26)25(32)28-22-15-18(17-3-6-19(7-4-17)31(33)34)5-10-23(22)30-13-11-29(2)12-14-30/h3-10,15H,11-14H2,1-2H3,(H,28,32)	OVQVBHOFYHZKAE-UHFFFAOYSA-N	50184956	CHEMBL3822521	WD repeat-containing protein 5			 127							ChEMBL	10.1016/j.ejmech.2016.04.032	10.7270/Q26H4KBP	27116709			Li, DD; Chen, WL; Xu, XL; Jiang, F; Wang, L; Xie, YY; Zhang, XJ; Guo, XK; You, QD; Sun, HP	China Pharmaceutical University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50184956	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50184956&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			127048927	346550439		CHEMBL3822521					1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50505630	CN1CCN(CC1)c1ccc(cc1NC(=O)c1ccc(F)c(C)c1Cl)-c1ccc(N)cc1	InChI=1S/C25H26ClFN4O/c1-16-21(27)9-8-20(24(16)26)25(32)29-22-15-18(17-3-6-19(28)7-4-17)5-10-23(22)31-13-11-30(2)12-14-31/h3-10,15H,11-14,28H2,1-2H3,(H,29,32)	BTGNRDWCEWBDNG-UHFFFAOYSA-N	50184957	CHEMBL3822596	WD repeat-containing protein 5			 206							ChEMBL	10.1016/j.ejmech.2016.04.032	10.7270/Q26H4KBP	27116709			Li, DD; Chen, WL; Xu, XL; Jiang, F; Wang, L; Xie, YY; Zhang, XJ; Guo, XK; You, QD; Sun, HP	China Pharmaceutical University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50184957	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50184957&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			127049251	346550440		CHEMBL3822596					1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50505631	CN1CCN(CC1)c1ccc(cc1NC(=O)c1cc(c(F)c(C)c1Cl)[N+]([O-])=O)-c1ccccc1	InChI=1S/C25H24ClFN4O3/c1-16-23(26)19(15-22(24(16)27)31(33)34)25(32)28-20-14-18(17-6-4-3-5-7-17)8-9-21(20)30-12-10-29(2)11-13-30/h3-9,14-15H,10-13H2,1-2H3,(H,28,32)	WOMZPTLUOWHXDN-UHFFFAOYSA-N	50184958	CHEMBL3823310	WD repeat-containing protein 5			 207							ChEMBL	10.1016/j.ejmech.2016.04.032	10.7270/Q26H4KBP	27116709			Li, DD; Chen, WL; Xu, XL; Jiang, F; Wang, L; Xie, YY; Zhang, XJ; Guo, XK; You, QD; Sun, HP	China Pharmaceutical University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50184958	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50184958&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			127049252	346550441		CHEMBL3823310					1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50505632	CN1CCN(CC1)c1ccc(cc1NC(=O)c1cc(c(F)c(C)c1Cl)[N+]([O-])=O)[N+]([O-])=O	InChI=1S/C19H19ClFN5O5/c1-11-17(20)13(10-16(18(11)21)26(30)31)19(27)22-14-9-12(25(28)29)3-4-15(14)24-7-5-23(2)6-8-24/h3-4,9-10H,5-8H2,1-2H3,(H,22,27)	ZVZKRCIQYYCPMS-UHFFFAOYSA-N	50184789	CHEMBL3822691	WD repeat-containing protein 5			 130							ChEMBL	10.1016/j.ejmech.2016.04.032	10.7270/Q26H4KBP	27116709			Li, DD; Chen, WL; Xu, XL; Jiang, F; Wang, L; Xie, YY; Zhang, XJ; Guo, XK; You, QD; Sun, HP	China Pharmaceutical University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50184789	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50184789&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			127049253	104069108		CHEMBL3822691				ZINC01650372	1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50505633	CN1CCN(CC1)c1cc(ccc1NC(=O)c1ccc(F)c(C)c1Cl)-c1ccc(cc1)C(O)=O	InChI=1S/C26H25ClFN3O3/c1-16-21(28)9-8-20(24(16)27)25(32)29-22-10-7-19(17-3-5-18(6-4-17)26(33)34)15-23(22)31-13-11-30(2)12-14-31/h3-10,15H,11-14H2,1-2H3,(H,29,32)(H,33,34)	ISYLXJINPZPCBF-UHFFFAOYSA-N	50184959	CHEMBL3822736	WD repeat-containing protein 5			>20000							ChEMBL	10.1016/j.ejmech.2016.04.032	10.7270/Q26H4KBP	27116709			Li, DD; Chen, WL; Xu, XL; Jiang, F; Wang, L; Xie, YY; Zhang, XJ; Guo, XK; You, QD; Sun, HP	China Pharmaceutical University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50184959	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50184959&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			127049254	346550442		CHEMBL3822736					1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50505634	CN1CCN(CC1)c1cc(ccc1NC(=O)c1ccc(F)c(C)c1Cl)-c1ccncc1	InChI=1S/C24H24ClFN4O/c1-16-20(26)5-4-19(23(16)25)24(31)28-21-6-3-18(17-7-9-27-10-8-17)15-22(21)30-13-11-29(2)12-14-30/h3-10,15H,11-14H2,1-2H3,(H,28,31)	RFRZTJPNSKENRI-UHFFFAOYSA-N	50184960	CHEMBL3823068	WD repeat-containing protein 5			>20000							ChEMBL	10.1016/j.ejmech.2016.04.032	10.7270/Q26H4KBP	27116709			Li, DD; Chen, WL; Xu, XL; Jiang, F; Wang, L; Xie, YY; Zhang, XJ; Guo, XK; You, QD; Sun, HP	China Pharmaceutical University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50184960	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50184960&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			127052955	346550443		CHEMBL3823068					1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50505635	CN1CCN(CC1)c1cc(ccc1NC(=O)c1ccc(F)c(C)c1Cl)-c1ccc(cc1)[N+]([O-])=O	InChI=1S/C25H24ClFN4O3/c1-16-21(27)9-8-20(24(16)26)25(32)28-22-10-5-18(17-3-6-19(7-4-17)31(33)34)15-23(22)30-13-11-29(2)12-14-30/h3-10,15H,11-14H2,1-2H3,(H,28,32)	LGNBAVDYDKZVKP-UHFFFAOYSA-N	50184961	CHEMBL3823125	WD repeat-containing protein 5			>20000							ChEMBL	10.1016/j.ejmech.2016.04.032	10.7270/Q26H4KBP	27116709			Li, DD; Chen, WL; Xu, XL; Jiang, F; Wang, L; Xie, YY; Zhang, XJ; Guo, XK; You, QD; Sun, HP	China Pharmaceutical University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50184961	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50184961&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			127052956	346550444		CHEMBL3823125					1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50505636	CN1CCN(CC1)c1cc(ccc1NC(=O)c1ccc(F)c(C)c1Cl)-c1ccc(N)cc1	InChI=1S/C25H26ClFN4O/c1-16-21(27)9-8-20(24(16)26)25(32)29-22-10-5-18(17-3-6-19(28)7-4-17)15-23(22)31-13-11-30(2)12-14-31/h3-10,15H,11-14,28H2,1-2H3,(H,29,32)	JKNBMDPRWBUIRK-UHFFFAOYSA-N	50184962	CHEMBL3823364	WD repeat-containing protein 5			>20000							ChEMBL	10.1016/j.ejmech.2016.04.032	10.7270/Q26H4KBP	27116709			Li, DD; Chen, WL; Xu, XL; Jiang, F; Wang, L; Xie, YY; Zhang, XJ; Guo, XK; You, QD; Sun, HP	China Pharmaceutical University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50184962	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50184962&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			127052957	346550445		CHEMBL3823364					1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50505637	CN1CCN(CC1)c1ccc(cc1NC(=O)c1ccc(F)c(C)c1Cl)[N+]([O-])=O	InChI=1S/C19H20ClFN4O3/c1-12-15(21)5-4-14(18(12)20)19(26)22-16-11-13(25(27)28)3-6-17(16)24-9-7-23(2)8-10-24/h3-6,11H,7-10H2,1-2H3,(H,22,26)	QHWMIGPLLWYRIR-UHFFFAOYSA-N	50428271	CHEMBL2337032	WD repeat-containing protein 5			 339							ChEMBL	10.1016/j.ejmech.2016.04.032	10.7270/Q26H4KBP	27116709			Li, DD; Chen, WL; Xu, XL; Jiang, F; Wang, L; Xie, YY; Zhang, XJ; Guo, XK; You, QD; Sun, HP	China Pharmaceutical University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50428271	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50428271&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	IA9	4IA9	70679466	164157146		CHEMBL2337032				ZINC95589389	1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50505638	CN1CCN(CC1)c1ccc(cc1NS(=O)(=O)c1ccc(F)cc1)[N+]([O-])=O	InChI=1S/C17H19FN4O4S/c1-20-8-10-21(11-9-20)17-7-4-14(22(23)24)12-16(17)19-27(25,26)15-5-2-13(18)3-6-15/h2-7,12,19H,8-11H2,1H3	PFLZCYDMTGTKRJ-UHFFFAOYSA-N	50184963	CHEMBL3822750	WD repeat-containing protein 5			>20000							ChEMBL	10.1016/j.ejmech.2016.04.032	10.7270/Q26H4KBP	27116709			Li, DD; Chen, WL; Xu, XL; Jiang, F; Wang, L; Xie, YY; Zhang, XJ; Guo, XK; You, QD; Sun, HP	China Pharmaceutical University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50184963	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50184963&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			127052958	346550446		CHEMBL3822750					1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50505639	COc1ccc(cc1)S(=O)(=O)Nc1cc(ccc1N1CCN(C)CC1)[N+]([O-])=O	InChI=1S/C18H22N4O5S/c1-20-9-11-21(12-10-20)18-8-3-14(22(23)24)13-17(18)19-28(25,26)16-6-4-15(27-2)5-7-16/h3-8,13,19H,9-12H2,1-2H3	KYEGUVDVMYZDDR-UHFFFAOYSA-N	50184964	CHEMBL3824152	WD repeat-containing protein 5			>20000							ChEMBL	10.1016/j.ejmech.2016.04.032	10.7270/Q26H4KBP	27116709			Li, DD; Chen, WL; Xu, XL; Jiang, F; Wang, L; Xie, YY; Zhang, XJ; Guo, XK; You, QD; Sun, HP	China Pharmaceutical University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50184964	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50184964&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			127052959	346550447		CHEMBL3824152					1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50505640	COc1ccc(cc1OC)S(=O)(=O)Nc1cc(ccc1N1CCN(C)CC1)[N+]([O-])=O	InChI=1S/C19H24N4O6S/c1-21-8-10-22(11-9-21)17-6-4-14(23(24)25)12-16(17)20-30(26,27)15-5-7-18(28-2)19(13-15)29-3/h4-7,12-13,20H,8-11H2,1-3H3	SPVBEEBVLVDAMB-UHFFFAOYSA-N	50184965	CHEMBL3822568	WD repeat-containing protein 5			>20000							ChEMBL	10.1016/j.ejmech.2016.04.032	10.7270/Q26H4KBP	27116709			Li, DD; Chen, WL; Xu, XL; Jiang, F; Wang, L; Xie, YY; Zhang, XJ; Guo, XK; You, QD; Sun, HP	China Pharmaceutical University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50184965	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50184965&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			127052960	346550448		CHEMBL3822568					1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50505641	COc1cc(OC)c(c(OC)c1)S(=O)(=O)Nc1cc(ccc1N1CCN(C)CC1)[N+]([O-])=O	InChI=1S/C20H26N4O7S/c1-22-7-9-23(10-8-22)17-6-5-14(24(25)26)11-16(17)21-32(27,28)20-18(30-3)12-15(29-2)13-19(20)31-4/h5-6,11-13,21H,7-10H2,1-4H3	OLEFCHDGMJFFIW-UHFFFAOYSA-N	50184966	CHEMBL3823731	WD repeat-containing protein 5			>20000							ChEMBL	10.1016/j.ejmech.2016.04.032	10.7270/Q26H4KBP	27116709			Li, DD; Chen, WL; Xu, XL; Jiang, F; Wang, L; Xie, YY; Zhang, XJ; Guo, XK; You, QD; Sun, HP	China Pharmaceutical University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50184966	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50184966&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			127048933	346550449		CHEMBL3823731					1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50505642	CN1CCN(CC1)c1ccc(cc1C(=O)Nc1ccc(F)c(C)c1Cl)[N+]([O-])=O	InChI=1S/C19H20ClFN4O3/c1-12-15(21)4-5-16(18(12)20)22-19(26)14-11-13(25(27)28)3-6-17(14)24-9-7-23(2)8-10-24/h3-6,11H,7-10H2,1-2H3,(H,22,26)	BHAFKZYJOYGKLL-UHFFFAOYSA-N	50184967	CHEMBL3823359	WD repeat-containing protein 5			 11400							ChEMBL	10.1016/j.ejmech.2016.04.032	10.7270/Q26H4KBP	27116709			Li, DD; Chen, WL; Xu, XL; Jiang, F; Wang, L; Xie, YY; Zhang, XJ; Guo, XK; You, QD; Sun, HP	China Pharmaceutical University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50184967	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50184967&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			127048934	346550450		CHEMBL3823359					1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50505643	COc1cccc(NC(=O)c2cc(ccc2N2CCN(C)CC2)[N+]([O-])=O)c1	InChI=1S/C19H22N4O4/c1-21-8-10-22(11-9-21)18-7-6-15(23(25)26)13-17(18)19(24)20-14-4-3-5-16(12-14)27-2/h3-7,12-13H,8-11H2,1-2H3,(H,20,24)	CUWVPDCPBIMKTB-UHFFFAOYSA-N	50184968	CHEMBL1607525	WD repeat-containing protein 5			>20000							ChEMBL	10.1016/j.ejmech.2016.04.032	10.7270/Q26H4KBP	27116709			Li, DD; Chen, WL; Xu, XL; Jiang, F; Wang, L; Xie, YY; Zhang, XJ; Guo, XK; You, QD; Sun, HP	China Pharmaceutical University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50184968	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50184968&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			2943337	346550451		CHEMBL1607525					1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50505644	CN1CCN(CC1)c1ccc(cc1C(=O)Nc1ccc(F)cc1F)[N+]([O-])=O	InChI=1S/C18H18F2N4O3/c1-22-6-8-23(9-7-22)17-5-3-13(24(26)27)11-14(17)18(25)21-16-4-2-12(19)10-15(16)20/h2-5,10-11H,6-9H2,1H3,(H,21,25)	KSNPYGMZTIUGFM-UHFFFAOYSA-N	50184969	CHEMBL3824177	WD repeat-containing protein 5			>20000							ChEMBL	10.1016/j.ejmech.2016.04.032	10.7270/Q26H4KBP	27116709			Li, DD; Chen, WL; Xu, XL; Jiang, F; Wang, L; Xie, YY; Zhang, XJ; Guo, XK; You, QD; Sun, HP	China Pharmaceutical University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50184969	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50184969&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			85721372	346550452		CHEMBL3824177					1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50505645	CN1CCN(CC1)c1ccc(cc1C(=O)Nc1ccccc1Cl)[N+]([O-])=O	InChI=1S/C18H19ClN4O3/c1-21-8-10-22(11-9-21)17-7-6-13(23(25)26)12-14(17)18(24)20-16-5-3-2-4-15(16)19/h2-7,12H,8-11H2,1H3,(H,20,24)	SNMZUFWTWXCSCR-UHFFFAOYSA-N	50184970	CHEMBL3823113	WD repeat-containing protein 5			>20000							ChEMBL	10.1016/j.ejmech.2016.04.032	10.7270/Q26H4KBP	27116709			Li, DD; Chen, WL; Xu, XL; Jiang, F; Wang, L; Xie, YY; Zhang, XJ; Guo, XK; You, QD; Sun, HP	China Pharmaceutical University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50184970	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50184970&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			127048935	346550453		CHEMBL3823113					1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50505646	CN1CCN(CC1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cccc(CN2CCOCC2)c1	InChI=1S/C29H32F3N5O3/c1-35-7-9-37(10-8-35)26-6-5-22(21-4-2-3-20(15-21)19-36-11-13-40-14-12-36)16-25(26)34-28(39)23-18-33-27(38)17-24(23)29(30,31)32/h2-6,15-18H,7-14,19H2,1H3,(H,33,38)(H,34,39)	DJOVLOYCGXNVPI-UHFFFAOYSA-N	50164794	CHEMBL3798846::US11174250, Example Table4.1.1::US11319299, Comp. No. 57	WD repeat-containing protein 5				 93						ChEMBL	10.1016/j.ejmech.2016.04.032	10.7270/Q26H4KBP	27116709			Li, DD; Chen, WL; Xu, XL; Jiang, F; Wang, L; Xie, YY; Zhang, XJ; Guo, XK; You, QD; Sun, HP	China Pharmaceutical University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50164794	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50164794&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	35Q	4QL1	91623360	341097539		CHEMBL3798846					1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50912995	CC(C)C[C@H](NC(=O)[C@H](Cc1cnc[nH]1)NC(=O)[C@@H](NC(=O)[C@H](CCC(O)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCN=C(N)N)NC(=O)[C@H](C)NC(=O)[C@H](CO)NC(=O)CNC(C)=O)C(C)C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CO)C(N)=O	InChI=1S/C56H98N22O17/c1-27(2)20-37(51(92)74-35(14-11-19-65-56(61)62)48(89)73-33(12-8-9-17-57)49(90)77-39(24-79)44(58)85)75-52(93)38(21-32-22-63-26-67-32)76-54(95)43(28(3)4)78-50(91)36(15-16-42(83)84)72-46(87)29(5)68-47(88)34(13-10-18-64-55(59)60)71-45(86)30(6)69-53(94)40(25-80)70-41(82)23-66-31(7)81/h22,26-30,33-40,43,79-80H,8-21,23-25,57H2,1-7H3,(H2,58,85)(H,63,67)(H,66,81)(H,68,88)(H,69,94)(H,70,82)(H,71,86)(H,72,87)(H,73,89)(H,74,92)(H,75,93)(H,76,95)(H,77,90)(H,78,91)(H,83,84)(H4,59,60,64)(H4,61,62,65)/t29-,30-,33-,34-,35-,36-,37-,38-,39-,40-,43-/m0/s1	PCONEFYGCDFYOM-UFBWGLHSSA-N	50318539	Ac-GSARAEVHLRKS-NH2::CHEMBL1086448	WD repeat-containing protein 5			 750							ChEMBL	10.1021/jm100139b	10.7270/Q2086678	20575550			Karatas, H; Townsend, EC; Bernard, D; Dou, Y; Wang, S	University of Michigan	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50318539	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50318539&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			46889977	104152900		CHEMBL1086448					1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50912996	CC(C)C[C@H](NC(=O)[C@H](Cc1cnc[nH]1)NC(=O)[C@@H](NC(=O)[C@H](CCC(O)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCN=C(N)N)NC(=O)[C@H](C)NC(=O)[C@H](CO)NC(C)=O)C(C)C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CO)C(N)=O	InChI=1S/C54H95N21O16/c1-26(2)20-36(49(88)71-34(14-11-19-63-54(59)60)46(85)70-32(12-8-9-17-55)47(86)74-38(23-76)42(56)81)72-50(89)37(21-31-22-61-25-64-31)73-52(91)41(27(3)4)75-48(87)35(15-16-40(79)80)69-44(83)28(5)65-45(84)33(13-10-18-62-53(57)58)68-43(82)29(6)66-51(90)39(24-77)67-30(7)78/h22,25-29,32-39,41,76-77H,8-21,23-24,55H2,1-7H3,(H2,56,81)(H,61,64)(H,65,84)(H,66,90)(H,67,78)(H,68,82)(H,69,83)(H,70,85)(H,71,88)(H,72,89)(H,73,91)(H,74,86)(H,75,87)(H,79,80)(H4,57,58,62)(H4,59,60,63)/t28-,29-,32-,33-,34-,35-,36-,37-,38-,39-,41-/m0/s1	QZWXANNPNSXHMO-RYYDISJRSA-N	50318540	Ac-SARAEVHLRKS-NH2::CHEMBL1086449	WD repeat-containing protein 5			 1040							ChEMBL	10.1021/jm100139b	10.7270/Q2086678	20575550			Karatas, H; Townsend, EC; Bernard, D; Dou, Y; Wang, S	University of Michigan	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50318540	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50318540&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			46866889	104152901		CHEMBL1086449					1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50912997	CC(C)C[C@H](NC(=O)[C@H](Cc1cnc[nH]1)NC(=O)[C@@H](NC(=O)[C@H](CCC(O)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCN=C(N)N)NC(=O)[C@H](C)NC(C)=O)C(C)C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CO)C(N)=O	InChI=1S/C51H90N20O14/c1-25(2)20-35(47(83)67-33(14-11-19-60-51(56)57)44(80)66-31(12-8-9-17-52)45(81)70-37(23-72)40(53)76)68-48(84)36(21-30-22-58-24-61-30)69-49(85)39(26(3)4)71-46(82)34(15-16-38(74)75)65-42(78)28(6)63-43(79)32(13-10-18-59-50(54)55)64-41(77)27(5)62-29(7)73/h22,24-28,31-37,39,72H,8-21,23,52H2,1-7H3,(H2,53,76)(H,58,61)(H,62,73)(H,63,79)(H,64,77)(H,65,78)(H,66,80)(H,67,83)(H,68,84)(H,69,85)(H,70,81)(H,71,82)(H,74,75)(H4,54,55,59)(H4,56,57,60)/t27-,28-,31-,32-,33-,34-,35-,36-,37-,39-/m0/s1	JDETYDIWHLTWSR-BJMIAJMISA-N	50318541	Ac-ARAEVHLRKS-NH2::CHEMBL1086450	WD repeat-containing protein 5			 20							ChEMBL	10.1021/jm100139b	10.7270/Q2086678	20575550			Karatas, H; Townsend, EC; Bernard, D; Dou, Y; Wang, S	University of Michigan	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50318541	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50318541&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			46867009	104152902		CHEMBL1086450			C04341		1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50912998	CC(C)C[C@H](NC(=O)[C@H](Cc1cnc[nH]1)NC(=O)[C@@H](NC(=O)[C@H](CCC(O)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCN=C(N)N)NC(=O)[C@H](C)NC(=O)[C@@H](N)CO)C(C)C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CO)C(N)=O	InChI=1S/C52H93N21O15/c1-25(2)19-35(48(86)69-33(13-10-18-62-52(58)59)45(83)68-31(11-7-8-16-53)46(84)72-37(23-75)40(55)78)70-49(87)36(20-29-21-60-24-63-29)71-50(88)39(26(3)4)73-47(85)34(14-15-38(76)77)67-42(80)28(6)65-44(82)32(12-9-17-61-51(56)57)66-41(79)27(5)64-43(81)30(54)22-74/h21,24-28,30-37,39,74-75H,7-20,22-23,53-54H2,1-6H3,(H2,55,78)(H,60,63)(H,64,81)(H,65,82)(H,66,79)(H,67,80)(H,68,83)(H,69,86)(H,70,87)(H,71,88)(H,72,84)(H,73,85)(H,76,77)(H4,56,57,61)(H4,58,59,62)/t27-,28-,30-,31-,32-,33-,34-,35-,36-,37-,39-/m0/s1	BKHVBKFFOKJNGM-PLNXYSOQSA-N	50318542	CHEMBL1086451::H2N-SARAEVHLRKS-NH2	WD repeat-containing protein 5			 80							ChEMBL	10.1021/jm100139b	10.7270/Q2086678	20575550			Karatas, H; Townsend, EC; Bernard, D; Dou, Y; Wang, S	University of Michigan	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50318542	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50318542&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			46867010	104152903		CHEMBL1086451					1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50912999	CC(C)C[C@H](NC(=O)[C@H](Cc1cnc[nH]1)NC(=O)[C@@H](NC(=O)[C@H](CCC(O)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCN=C(N)N)NC(C)=O)C(C)C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CO)C(N)=O	InChI=1S/C48H85N19O13/c1-24(2)19-33(44(78)63-31(13-10-18-57-48(53)54)41(75)62-30(11-7-8-16-49)42(76)66-35(22-68)38(50)72)64-45(79)34(20-28-21-55-23-58-28)65-46(80)37(25(3)4)67-43(77)32(14-15-36(70)71)61-39(73)26(5)59-40(74)29(60-27(6)69)12-9-17-56-47(51)52/h21,23-26,29-35,37,68H,7-20,22,49H2,1-6H3,(H2,50,72)(H,55,58)(H,59,74)(H,60,69)(H,61,73)(H,62,75)(H,63,78)(H,64,79)(H,65,80)(H,66,76)(H,67,77)(H,70,71)(H4,51,52,56)(H4,53,54,57)/t26-,29-,30-,31-,32-,33-,34-,35-,37-/m0/s1	DBRGJMAVCWIRNI-QXZHZWOVSA-N	50318543	Ac-RAEVHLRKS-NH2::CHEMBL1086452	WD repeat-containing protein 5			 29000							ChEMBL	10.1021/jm100139b	10.7270/Q2086678	20575550			Karatas, H; Townsend, EC; Bernard, D; Dou, Y; Wang, S	University of Michigan	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50318543	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50318543&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			46867121	104152904		CHEMBL1086452					1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50913000	CC(C)C[C@H](NC(=O)[C@H](Cc1cnc[nH]1)NC(=O)[C@@H](NC(=O)[C@H](CCC(O)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCN=C(N)N)NC(=O)[C@H](C)NC(C)=O)C(C)C)C(N)=O	InChI=1S/C36H61N13O10/c1-17(2)13-25(29(37)53)47-34(58)26(14-22-15-40-16-42-22)48-35(59)28(18(3)4)49-33(57)24(10-11-27(51)52)46-31(55)20(6)44-32(56)23(9-8-12-41-36(38)39)45-30(54)19(5)43-21(7)50/h15-20,23-26,28H,8-14H2,1-7H3,(H2,37,53)(H,40,42)(H,43,50)(H,44,56)(H,45,54)(H,46,55)(H,47,58)(H,48,59)(H,49,57)(H,51,52)(H4,38,39,41)/t19-,20-,23-,24-,25-,26-,28-/m0/s1	CEMFFHOCMZLMEO-IBQXPFEUSA-N	50318544	Ac-ARAEVHL-NH2::CHEMBL1086453	WD repeat-containing protein 5			 160							ChEMBL	10.1021/jm100139b	10.7270/Q2086678	20575550			Karatas, H; Townsend, EC; Bernard, D; Dou, Y; Wang, S	University of Michigan	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50318544	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50318544&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			46889978	104152905		CHEMBL1086453			C04341	ZINC95539298	1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50913001	CC(C)[C@H](NC(=O)[C@H](CCC(O)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCN=C(N)N)NC(=O)[C@H](C)NC(C)=O)C(=O)N[C@@H](Cc1cnc[nH]1)C(N)=O	InChI=1S/C30H50N12O9/c1-14(2)23(29(51)41-21(24(31)46)11-18-12-34-13-36-18)42-28(50)20(8-9-22(44)45)40-26(48)16(4)38-27(49)19(7-6-10-35-30(32)33)39-25(47)15(3)37-17(5)43/h12-16,19-21,23H,6-11H2,1-5H3,(H2,31,46)(H,34,36)(H,37,43)(H,38,49)(H,39,47)(H,40,48)(H,41,51)(H,42,50)(H,44,45)(H4,32,33,35)/t15-,16-,19-,20-,21-,23-/m0/s1	AFTMQAFHRKDEPI-CMQAMBHRSA-N	50318545	Ac-ARAEVH-NH2::CHEMBL1086454	WD repeat-containing protein 5			 400							ChEMBL	10.1021/jm100139b	10.7270/Q2086678	20575550			Karatas, H; Townsend, EC; Bernard, D; Dou, Y; Wang, S	University of Michigan	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50318545	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50318545&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			46889979	104152906		CHEMBL1086454			C04341	ZINC49777277	1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50913002	CC(C)[C@H](NC(=O)[C@H](CCC(O)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCN=C(N)N)NC(=O)[C@H](C)NC(C)=O)C(N)=O	InChI=1S/C24H43N9O8/c1-11(2)18(19(25)37)33-23(41)16(8-9-17(35)36)32-21(39)13(4)30-22(40)15(7-6-10-28-24(26)27)31-20(38)12(3)29-14(5)34/h11-13,15-16,18H,6-10H2,1-5H3,(H2,25,37)(H,29,34)(H,30,40)(H,31,38)(H,32,39)(H,33,41)(H,35,36)(H4,26,27,28)/t12-,13-,15-,16-,18-/m0/s1	CIWFPIIPIHNZNZ-XRDYDQJJSA-N	50318546	Ac-ARAEV-NH2::CHEMBL1086531	WD repeat-containing protein 5			 750							ChEMBL	10.1021/jm100139b	10.7270/Q2086678	20575550			Karatas, H; Townsend, EC; Bernard, D; Dou, Y; Wang, S	University of Michigan	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50318546	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50318546&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			46889980	104152907		CHEMBL1086531			C04341	ZINC49777659	1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50913003	C[C@H](NC(C)=O)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](C)C(=O)N[C@@H](CCC(O)=O)C(N)=O	InChI=1S/C19H34N8O7/c1-9(24-11(3)28)16(32)27-13(5-4-8-23-19(21)22)18(34)25-10(2)17(33)26-12(15(20)31)6-7-14(29)30/h9-10,12-13H,4-8H2,1-3H3,(H2,20,31)(H,24,28)(H,25,34)(H,26,33)(H,27,32)(H,29,30)(H4,21,22,23)/t9-,10-,12-,13-/m0/s1	ZFNWHWJOGHVTEW-UKJIMTQDSA-N	50318547	Ac-ARAE-NH2::CHEMBL1085604	WD repeat-containing protein 5			 400							ChEMBL	10.1021/jm100139b	10.7270/Q2086678	20575550			Karatas, H; Townsend, EC; Bernard, D; Dou, Y; Wang, S	University of Michigan	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50318547	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50318547&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			46889981	104152908		CHEMBL1085604			C04341	ZINC49047581	1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50913004	C[C@H](NC(=O)[C@H](CCCN=C(N)N)NC(=O)[C@H](C)NC(C)=O)C(N)=O	InChI=1S/C14H27N7O4/c1-7(11(15)23)20-13(25)10(5-4-6-18-14(16)17)21-12(24)8(2)19-9(3)22/h7-8,10H,4-6H2,1-3H3,(H2,15,23)(H,19,22)(H,20,25)(H,21,24)(H4,16,17,18)/t7-,8-,10-/m0/s1	ATPJZQHSTNYINS-NRPADANISA-N	50318548	Ac-ARA-NH2::CHEMBL1086455	WD repeat-containing protein 5			 540							ChEMBL	10.1021/jm100139b	10.7270/Q2086678	20575550			Karatas, H; Townsend, EC; Bernard, D; Dou, Y; Wang, S	University of Michigan	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50318548	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50318548&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			46864279	104152909		CHEMBL1086455			C04341	ZINC49049253	1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50913005	C[C@H](NC(C)=O)C(=O)N[C@@H](CCCN=C(N)N)C(N)=O	InChI=1S/C11H22N6O3/c1-6(16-7(2)18)10(20)17-8(9(12)19)4-3-5-15-11(13)14/h6,8H,3-5H2,1-2H3,(H2,12,19)(H,16,18)(H,17,20)(H4,13,14,15)/t6-,8-/m0/s1	WESUUTFORKSXRD-XPUUQOCRSA-N	50318549	Ac-AR-NH2::CHEMBL1085605	WD repeat-containing protein 5			 125000							ChEMBL	10.1021/jm100139b	10.7270/Q2086678	20575550			Karatas, H; Townsend, EC; Bernard, D; Dou, Y; Wang, S	University of Michigan	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50318549	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50318549&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			46889982	104152910		CHEMBL1085605			C04341	ZINC49047585	1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50913006	CC(C)C[C@H](NC(=O)[C@H](Cc1cnc[nH]1)NC(=O)[C@@H](NC(=O)[C@H](CCC(O)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCN=C(N)N)NC(=O)[C@H](C)NC(=O)[C@H](CO)NC(=O)CNC(C)=O)C(C)C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CO)C(N)=O	InChI=1S/C56H98N22O17/c1-27(2)20-37(51(92)74-35(14-11-19-65-56(61)62)48(89)73-33(12-8-9-17-57)49(90)77-39(24-79)44(58)85)75-52(93)38(21-32-22-63-26-67-32)76-54(95)43(28(3)4)78-50(91)36(15-16-42(83)84)72-46(87)29(5)68-47(88)34(13-10-18-64-55(59)60)71-45(86)30(6)69-53(94)40(25-80)70-41(82)23-66-31(7)81/h22,26-30,33-40,43,79-80H,8-21,23-25,57H2,1-7H3,(H2,58,85)(H,63,67)(H,66,81)(H,68,88)(H,69,94)(H,70,82)(H,71,86)(H,72,87)(H,73,89)(H,74,92)(H,75,93)(H,76,95)(H,77,90)(H,78,91)(H,83,84)(H4,59,60,64)(H4,61,62,65)/t29-,30-,33-,34-,35-,36-,37-,38-,39-,40-,43-/m0/s1	PCONEFYGCDFYOM-UFBWGLHSSA-N	50318539	Ac-GSARAEVHLRKS-NH2::CHEMBL1086448	WD repeat-containing protein 5		 160								ChEMBL	10.1021/jm100139b	10.7270/Q2086678	20575550			Karatas, H; Townsend, EC; Bernard, D; Dou, Y; Wang, S	University of Michigan	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50318539	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50318539&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			46889977	104152900		CHEMBL1086448					1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50913007	CC(C)C[C@H](NC(=O)[C@H](Cc1cnc[nH]1)NC(=O)[C@@H](NC(=O)[C@H](CCC(O)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCN=C(N)N)NC(=O)[C@H](C)NC(=O)[C@H](CO)NC(C)=O)C(C)C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CO)C(N)=O	InChI=1S/C54H95N21O16/c1-26(2)20-36(49(88)71-34(14-11-19-63-54(59)60)46(85)70-32(12-8-9-17-55)47(86)74-38(23-76)42(56)81)72-50(89)37(21-31-22-61-25-64-31)73-52(91)41(27(3)4)75-48(87)35(15-16-40(79)80)69-44(83)28(5)65-45(84)33(13-10-18-62-53(57)58)68-43(82)29(6)66-51(90)39(24-77)67-30(7)78/h22,25-29,32-39,41,76-77H,8-21,23-24,55H2,1-7H3,(H2,56,81)(H,61,64)(H,65,84)(H,66,90)(H,67,78)(H,68,82)(H,69,83)(H,70,85)(H,71,88)(H,72,89)(H,73,91)(H,74,86)(H,75,87)(H,79,80)(H4,57,58,62)(H4,59,60,63)/t28-,29-,32-,33-,34-,35-,36-,37-,38-,39-,41-/m0/s1	QZWXANNPNSXHMO-RYYDISJRSA-N	50318540	Ac-SARAEVHLRKS-NH2::CHEMBL1086449	WD repeat-containing protein 5		 200								ChEMBL	10.1021/jm100139b	10.7270/Q2086678	20575550			Karatas, H; Townsend, EC; Bernard, D; Dou, Y; Wang, S	University of Michigan	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50318540	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50318540&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			46866889	104152901		CHEMBL1086449					1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50913008	CC(C)C[C@H](NC(=O)[C@H](Cc1cnc[nH]1)NC(=O)[C@@H](NC(=O)[C@H](CCC(O)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCN=C(N)N)NC(=O)[C@H](C)NC(C)=O)C(C)C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CO)C(N)=O	InChI=1S/C51H90N20O14/c1-25(2)20-35(47(83)67-33(14-11-19-60-51(56)57)44(80)66-31(12-8-9-17-52)45(81)70-37(23-72)40(53)76)68-48(84)36(21-30-22-58-24-61-30)69-49(85)39(26(3)4)71-46(82)34(15-16-38(74)75)65-42(78)28(6)63-43(79)32(13-10-18-59-50(54)55)64-41(77)27(5)62-29(7)73/h22,24-28,31-37,39,72H,8-21,23,52H2,1-7H3,(H2,53,76)(H,58,61)(H,62,73)(H,63,79)(H,64,77)(H,65,78)(H,66,80)(H,67,83)(H,68,84)(H,69,85)(H,70,81)(H,71,82)(H,74,75)(H4,54,55,59)(H4,56,57,60)/t27-,28-,31-,32-,33-,34-,35-,36-,37-,39-/m0/s1	JDETYDIWHLTWSR-BJMIAJMISA-N	50318541	Ac-ARAEVHLRKS-NH2::CHEMBL1086450	WD repeat-containing protein 5		 3								ChEMBL	10.1021/jm100139b	10.7270/Q2086678	20575550			Karatas, H; Townsend, EC; Bernard, D; Dou, Y; Wang, S	University of Michigan	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50318541	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50318541&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			46867009	104152902		CHEMBL1086450			C04341		1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50913009	CC(C)C[C@H](NC(=O)[C@H](Cc1cnc[nH]1)NC(=O)[C@@H](NC(=O)[C@H](CCC(O)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCN=C(N)N)NC(=O)[C@H](C)NC(=O)[C@@H](N)CO)C(C)C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CO)C(N)=O	InChI=1S/C52H93N21O15/c1-25(2)19-35(48(86)69-33(13-10-18-62-52(58)59)45(83)68-31(11-7-8-16-53)46(84)72-37(23-75)40(55)78)70-49(87)36(20-29-21-60-24-63-29)71-50(88)39(26(3)4)73-47(85)34(14-15-38(76)77)67-42(80)28(6)65-44(82)32(12-9-17-61-51(56)57)66-41(79)27(5)64-43(81)30(54)22-74/h21,24-28,30-37,39,74-75H,7-20,22-23,53-54H2,1-6H3,(H2,55,78)(H,60,63)(H,64,81)(H,65,82)(H,66,79)(H,67,80)(H,68,83)(H,69,86)(H,70,87)(H,71,88)(H,72,84)(H,73,85)(H,76,77)(H4,56,57,61)(H4,58,59,62)/t27-,28-,30-,31-,32-,33-,34-,35-,36-,37-,39-/m0/s1	BKHVBKFFOKJNGM-PLNXYSOQSA-N	50318542	CHEMBL1086451::H2N-SARAEVHLRKS-NH2	WD repeat-containing protein 5		 20								ChEMBL	10.1021/jm100139b	10.7270/Q2086678	20575550			Karatas, H; Townsend, EC; Bernard, D; Dou, Y; Wang, S	University of Michigan	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50318542	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50318542&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			46867010	104152903		CHEMBL1086451					1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50913010	CC(C)C[C@H](NC(=O)[C@H](Cc1cnc[nH]1)NC(=O)[C@@H](NC(=O)[C@H](CCC(O)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCN=C(N)N)NC(C)=O)C(C)C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CO)C(N)=O	InChI=1S/C48H85N19O13/c1-24(2)19-33(44(78)63-31(13-10-18-57-48(53)54)41(75)62-30(11-7-8-16-49)42(76)66-35(22-68)38(50)72)64-45(79)34(20-28-21-55-23-58-28)65-46(80)37(25(3)4)67-43(77)32(14-15-36(70)71)61-39(73)26(5)59-40(74)29(60-27(6)69)12-9-17-56-47(51)52/h21,23-26,29-35,37,68H,7-20,22,49H2,1-6H3,(H2,50,72)(H,55,58)(H,59,74)(H,60,69)(H,61,73)(H,62,75)(H,63,78)(H,64,79)(H,65,80)(H,66,76)(H,67,77)(H,70,71)(H4,51,52,56)(H4,53,54,57)/t26-,29-,30-,31-,32-,33-,34-,35-,37-/m0/s1	DBRGJMAVCWIRNI-QXZHZWOVSA-N	50318543	Ac-RAEVHLRKS-NH2::CHEMBL1086452	WD repeat-containing protein 5		 6300								ChEMBL	10.1021/jm100139b	10.7270/Q2086678	20575550			Karatas, H; Townsend, EC; Bernard, D; Dou, Y; Wang, S	University of Michigan	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50318543	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50318543&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			46867121	104152904		CHEMBL1086452					1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50913011	CC(C)C[C@H](NC(=O)[C@H](Cc1cnc[nH]1)NC(=O)[C@@H](NC(=O)[C@H](CCC(O)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCN=C(N)N)NC(=O)[C@H](C)NC(C)=O)C(C)C)C(N)=O	InChI=1S/C36H61N13O10/c1-17(2)13-25(29(37)53)47-34(58)26(14-22-15-40-16-42-22)48-35(59)28(18(3)4)49-33(57)24(10-11-27(51)52)46-31(55)20(6)44-32(56)23(9-8-12-41-36(38)39)45-30(54)19(5)43-21(7)50/h15-20,23-26,28H,8-14H2,1-7H3,(H2,37,53)(H,40,42)(H,43,50)(H,44,56)(H,45,54)(H,46,55)(H,47,58)(H,48,59)(H,49,57)(H,51,52)(H4,38,39,41)/t19-,20-,23-,24-,25-,26-,28-/m0/s1	CEMFFHOCMZLMEO-IBQXPFEUSA-N	50318544	Ac-ARAEVHL-NH2::CHEMBL1086453	WD repeat-containing protein 5		 30								ChEMBL	10.1021/jm100139b	10.7270/Q2086678	20575550			Karatas, H; Townsend, EC; Bernard, D; Dou, Y; Wang, S	University of Michigan	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50318544	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50318544&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			46889978	104152905		CHEMBL1086453			C04341	ZINC95539298	1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50913012	CC(C)[C@H](NC(=O)[C@H](CCC(O)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCN=C(N)N)NC(=O)[C@H](C)NC(C)=O)C(=O)N[C@@H](Cc1cnc[nH]1)C(N)=O	InChI=1S/C30H50N12O9/c1-14(2)23(29(51)41-21(24(31)46)11-18-12-34-13-36-18)42-28(50)20(8-9-22(44)45)40-26(48)16(4)38-27(49)19(7-6-10-35-30(32)33)39-25(47)15(3)37-17(5)43/h12-16,19-21,23H,6-11H2,1-5H3,(H2,31,46)(H,34,36)(H,37,43)(H,38,49)(H,39,47)(H,40,48)(H,41,51)(H,42,50)(H,44,45)(H4,32,33,35)/t15-,16-,19-,20-,21-,23-/m0/s1	AFTMQAFHRKDEPI-CMQAMBHRSA-N	50318545	Ac-ARAEVH-NH2::CHEMBL1086454	WD repeat-containing protein 5		 90								ChEMBL	10.1021/jm100139b	10.7270/Q2086678	20575550			Karatas, H; Townsend, EC; Bernard, D; Dou, Y; Wang, S	University of Michigan	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50318545	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50318545&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			46889979	104152906		CHEMBL1086454			C04341	ZINC49777277	1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50913013	CC(C)[C@H](NC(=O)[C@H](CCC(O)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCN=C(N)N)NC(=O)[C@H](C)NC(C)=O)C(N)=O	InChI=1S/C24H43N9O8/c1-11(2)18(19(25)37)33-23(41)16(8-9-17(35)36)32-21(39)13(4)30-22(40)15(7-6-10-28-24(26)27)31-20(38)12(3)29-14(5)34/h11-13,15-16,18H,6-10H2,1-5H3,(H2,25,37)(H,29,34)(H,30,40)(H,31,38)(H,32,39)(H,33,41)(H,35,36)(H4,26,27,28)/t12-,13-,15-,16-,18-/m0/s1	CIWFPIIPIHNZNZ-XRDYDQJJSA-N	50318546	Ac-ARAEV-NH2::CHEMBL1086531	WD repeat-containing protein 5		 160								ChEMBL	10.1021/jm100139b	10.7270/Q2086678	20575550			Karatas, H; Townsend, EC; Bernard, D; Dou, Y; Wang, S	University of Michigan	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50318546	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50318546&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			46889980	104152907		CHEMBL1086531			C04341	ZINC49777659	1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50913014	CNC(=O)[C@H](C)NC(=O)[C@H](CCCN=C(N)N)NC(=O)[C@H](C)NC(C)=O	InChI=1S/C15H29N7O4/c1-8(12(24)18-4)21-14(26)11(6-5-7-19-15(16)17)22-13(25)9(2)20-10(3)23/h8-9,11H,5-7H2,1-4H3,(H,18,24)(H,20,23)(H,21,26)(H,22,25)(H4,16,17,19)/t8-,9-,11-/m0/s1	PYWIZEZTCCLSTR-QXEWZRGKSA-N	50318521	Ac-ARA-CONHMe::CHEMBL1084621	WD repeat-containing protein 5			 700							ChEMBL	10.1021/jm100139b	10.7270/Q2086678	20575550			Karatas, H; Townsend, EC; Bernard, D; Dou, Y; Wang, S	University of Michigan	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50318521	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50318521&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			46889986	104152882		CHEMBL1084621			C04341	ZINC49046214	1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50913015	C[C@H](NC(C)=O)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](C)C(=O)N(C)C	InChI=1S/C16H31N7O4/c1-9(20-11(3)24)13(25)22-12(7-6-8-19-16(17)18)14(26)21-10(2)15(27)23(4)5/h9-10,12H,6-8H2,1-5H3,(H,20,24)(H,21,26)(H,22,25)(H4,17,18,19)/t9-,10-,12-/m0/s1	XFBVAZQSPWDVFU-NHCYSSNCSA-N	50318522	Ac-ARA-CONMe2::CHEMBL1084622	WD repeat-containing protein 5			 30000							ChEMBL	10.1021/jm100139b	10.7270/Q2086678	20575550			Karatas, H; Townsend, EC; Bernard, D; Dou, Y; Wang, S	University of Michigan	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50318522	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50318522&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			46889987	104152883		CHEMBL1084622			C04341	ZINC49046218	1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50913016	COC(=O)[C@H](C)NC(=O)[C@H](CCCN=C(N)N)NC(=O)[C@H](C)NC(C)=O	InChI=1S/C15H28N6O5/c1-8(19-10(3)22)12(23)21-11(6-5-7-18-15(16)17)13(24)20-9(2)14(25)26-4/h8-9,11H,5-7H2,1-4H3,(H,19,22)(H,20,24)(H,21,23)(H4,16,17,18)/t8-,9-,11-/m0/s1	VXMGKWGBQTWNEN-QXEWZRGKSA-N	50318523	Ac-ARA-COOCH3::CHEMBL1084623	WD repeat-containing protein 5			 7300							ChEMBL	10.1021/jm100139b	10.7270/Q2086678	20575550			Karatas, H; Townsend, EC; Bernard, D; Dou, Y; Wang, S	University of Michigan	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50318523	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50318523&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			46889988	104152884		CHEMBL1084623			C04341	ZINC49802194	1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50913017	C[C@@H](O)[C@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@@H](NC(=O)[C@H](CCCN=C(N)N)NC(=O)[C@H](C)N)[C@@H](C)O)C(=O)N[C@@H](C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CO)C(N)=O	InChI=1S/C46H88N20O14/c1-22(49)36(72)59-29(14-10-20-57-46(54)55)41(77)66-34(25(4)69)44(80)63-27(12-6-8-18-48)38(74)62-30(15-16-32(50)70)42(78)65-33(24(3)68)43(79)58-23(2)37(73)60-28(13-9-19-56-45(52)53)39(75)61-26(11-5-7-17-47)40(76)64-31(21-67)35(51)71/h22-31,33-34,67-69H,5-21,47-49H2,1-4H3,(H2,50,70)(H2,51,71)(H,58,79)(H,59,72)(H,60,73)(H,61,75)(H,62,74)(H,63,80)(H,64,76)(H,65,78)(H,66,77)(H4,52,53,56)(H4,54,55,57)/t22-,23-,24+,25+,26-,27-,28-,29-,30-,31-,33-,34-/m0/s1	OZZZZNRCCWQVLU-ZKJUQCEXSA-N	50318524	CHEMBL1082281::H2N-ARTKQTARKS-NH2	WD repeat-containing protein 5			 70000							ChEMBL	10.1021/jm100139b	10.7270/Q2086678	20575550			Karatas, H; Townsend, EC; Bernard, D; Dou, Y; Wang, S	University of Michigan	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50318524	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50318524&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			46889989	104152885		CHEMBL1082281			C03803		1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50913018	C[C@@H](O)[C@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@@H](NC(=O)[C@H](CCCN=C(N)N)NC(=O)[C@H](C)NC(C)=O)[C@@H](C)O)C(=O)N[C@@H](C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CO)C(N)=O	InChI=1S/C48H90N20O15/c1-23(59-27(5)72)38(75)62-31(15-11-21-58-48(55)56)43(80)68-36(26(4)71)46(83)65-29(13-7-9-19-50)40(77)64-32(16-17-34(51)73)44(81)67-35(25(3)70)45(82)60-24(2)39(76)61-30(14-10-20-57-47(53)54)41(78)63-28(12-6-8-18-49)42(79)66-33(22-69)37(52)74/h23-26,28-33,35-36,69-71H,6-22,49-50H2,1-5H3,(H2,51,73)(H2,52,74)(H,59,72)(H,60,82)(H,61,76)(H,62,75)(H,63,78)(H,64,77)(H,65,83)(H,66,79)(H,67,81)(H,68,80)(H4,53,54,57)(H4,55,56,58)/t23-,24-,25+,26+,28-,29-,30-,31-,32-,33-,35-,36-/m0/s1	PTYYUNSMCQJTHL-JPPFDADPSA-N	50318525	Ac-ARTKQTARKS-NH2::CHEMBL1082282	WD repeat-containing protein 5			 6							ChEMBL	10.1021/jm100139b	10.7270/Q2086678	20575550			Karatas, H; Townsend, EC; Bernard, D; Dou, Y; Wang, S	University of Michigan	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50318525	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50318525&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			46867257	104152886		CHEMBL1082282			C04341		1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50913019	C[C@@H](O)[C@H](NC(=O)[C@H](CCCN=C(N)N)NC(=O)[C@H](C)N)C(N)=O	InChI=1S/C13H27N7O4/c1-6(14)11(23)19-8(4-3-5-18-13(16)17)12(24)20-9(7(2)21)10(15)22/h6-9,21H,3-5,14H2,1-2H3,(H2,15,22)(H,19,23)(H,20,24)(H4,16,17,18)/t6-,7+,8-,9-/m0/s1	TXVGTYORMOSCJR-KZVJFYERSA-N	50318526	CHEMBL1085864::H2N-ART-NH2	WD repeat-containing protein 5			 127000							ChEMBL	10.1021/jm100139b	10.7270/Q2086678	20575550			Karatas, H; Townsend, EC; Bernard, D; Dou, Y; Wang, S	University of Michigan	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50318526	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50318526&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			24757930	104152887		CHEMBL1085864			C03803	ZINC49049659	1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50913020	C[C@@H](O)[C@H](NC(=O)[C@H](CCCN=C(N)N)NC(=O)[C@H](C)NC(C)=O)C(N)=O	InChI=1S/C15H29N7O5/c1-7(20-9(3)24)13(26)21-10(5-4-6-19-15(17)18)14(27)22-11(8(2)23)12(16)25/h7-8,10-11,23H,4-6H2,1-3H3,(H2,16,25)(H,20,24)(H,21,26)(H,22,27)(H4,17,18,19)/t7-,8+,10-,11-/m0/s1	CYECJCHCQBPTIK-OEIWMXHLSA-N	50318527	Ac-ART-NH2::CHEMBL1085865	WD repeat-containing protein 5			 80							ChEMBL	10.1021/jm100139b	10.7270/Q2086678	20575550			Karatas, H; Townsend, EC; Bernard, D; Dou, Y; Wang, S	University of Michigan	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50318527	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50318527&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			46864280	104152888		CHEMBL1085865			C04341	ZINC49049663	1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50913021	C[C@@H](O)[C@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](CCCCN)N(C)C(=O)[C@@H](NC(=O)[C@H](CCCN=C(N)N)NC(=O)[C@H](C)N)[C@@H](C)O)C(=O)N[C@@H](C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CO)C(N)=O	InChI=1S/C47H90N20O14/c1-23(50)37(73)60-29(14-11-21-58-47(55)56)41(77)66-35(26(4)70)45(81)67(5)32(15-7-9-19-49)43(79)63-30(16-17-33(51)71)42(78)65-34(25(3)69)44(80)59-24(2)38(74)61-28(13-10-20-57-46(53)54)39(75)62-27(12-6-8-18-48)40(76)64-31(22-68)36(52)72/h23-32,34-35,68-70H,6-22,48-50H2,1-5H3,(H2,51,71)(H2,52,72)(H,59,80)(H,60,73)(H,61,74)(H,62,75)(H,63,79)(H,64,76)(H,65,78)(H,66,77)(H4,53,54,57)(H4,55,56,58)/t23-,24-,25+,26+,27-,28-,29-,30-,31-,32-,34-,35-/m0/s1	BMQKBMJJUNPVPV-NCKQPBNLSA-N	50318528	CHEMBL1082284::H2N-ARTK(Me)QTARKS-NH2	WD repeat-containing protein 5			 69000							ChEMBL	10.1021/jm100139b	10.7270/Q2086678	20575550			Karatas, H; Townsend, EC; Bernard, D; Dou, Y; Wang, S	University of Michigan	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50318528	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50318528&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			46889993	104152889		CHEMBL1082284			C03803		1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50913022	CNCCCC[C@H](N(C)C(=O)[C@@H](NC(=O)[C@H](CCCN=C(N)N)NC(=O)[C@H](C)N)[C@@H](C)O)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H]([C@@H](C)O)C(=O)N[C@@H](C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CO)C(N)=O	InChI=1S/C48H92N20O14/c1-24(50)38(74)61-30(15-12-22-59-48(55)56)42(78)67-36(27(4)71)46(82)68(6)33(16-8-10-20-57-5)44(80)64-31(17-18-34(51)72)43(79)66-35(26(3)70)45(81)60-25(2)39(75)62-29(14-11-21-58-47(53)54)40(76)63-28(13-7-9-19-49)41(77)65-32(23-69)37(52)73/h24-33,35-36,57,69-71H,7-23,49-50H2,1-6H3,(H2,51,72)(H2,52,73)(H,60,81)(H,61,74)(H,62,75)(H,63,76)(H,64,80)(H,65,77)(H,66,79)(H,67,78)(H4,53,54,58)(H4,55,56,59)/t24-,25-,26+,27+,28-,29-,30-,31-,32-,33-,35-,36-/m0/s1	YJQPFWYFQWTFRD-GTTQRSHYSA-N	50318529	CHEMBL1082285::H2N-ARTK(Me2)QTARKS-NH2	WD repeat-containing protein 5			 42000							ChEMBL	10.1021/jm100139b	10.7270/Q2086678	20575550			Karatas, H; Townsend, EC; Bernard, D; Dou, Y; Wang, S	University of Michigan	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50318529	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50318529&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			46889994	104152890		CHEMBL1082285			C03803		1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50913023	C[C@@H](O)[C@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](CCCCN(C)C)N(C)C(=O)[C@@H](NC(=O)[C@H](CCCN=C(N)N)NC(=O)[C@H](C)N)[C@@H](C)O)C(=O)N[C@@H](C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CO)C(N)=O	InChI=1S/C49H94N20O14/c1-25(51)39(75)61-31(16-13-22-59-49(56)57)43(79)67-37(28(4)72)47(83)69(7)34(17-9-11-23-68(5)6)45(81)64-32(18-19-35(52)73)44(80)66-36(27(3)71)46(82)60-26(2)40(76)62-30(15-12-21-58-48(54)55)41(77)63-29(14-8-10-20-50)42(78)65-33(24-70)38(53)74/h25-34,36-37,70-72H,8-24,50-51H2,1-7H3,(H2,52,73)(H2,53,74)(H,60,82)(H,61,75)(H,62,76)(H,63,77)(H,64,81)(H,65,78)(H,66,80)(H,67,79)(H4,54,55,58)(H4,56,57,59)/t25-,26-,27+,28+,29-,30-,31-,32-,33-,34-,36-,37-/m0/s1	PBPOVNDZNWBXLP-RETRBKMKSA-N	50318530	CHEMBL1082286::H2N-ARTK(Me3)QTARKS-NH2	WD repeat-containing protein 5			 73000							ChEMBL	10.1021/jm100139b	10.7270/Q2086678	20575550			Karatas, H; Townsend, EC; Bernard, D; Dou, Y; Wang, S	University of Michigan	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50318530	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50318530&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			46889995	104152891		CHEMBL1082286			C03803		1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50913024	CC(C)C[C@H](NC(=O)[C@H](Cc1cnc[nH]1)NC(=O)[C@@H](NC(=O)[C@H](CCC(O)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCN=C(N)N)NC(=O)[C@H](C)NC(=O)[C@H](CO)NC(=O)CNC(C)=O)C(C)C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CO)C(=O)NCC(=O)NCC(=O)NCC(=O)N[C@@H](CCCCNC(=O)c1c(cccc1-c1c2ccc(O)cc2oc2cc(=O)ccc12)C(O)=O)C(N)=O	InChI=1S/C89H129N27O27/c1-43(2)31-60(113-83(137)61(32-48-35-96-42-104-48)114-86(140)73(44(3)4)116-81(135)59(25-26-70(126)127)110-76(130)45(5)105-78(132)57(19-13-29-98-88(92)93)109-75(129)46(6)106-84(138)63(41-118)108-68(124)38-100-47(7)119)82(136)112-58(20-14-30-99-89(94)95)79(133)111-56(18-8-10-27-90)80(134)115-62(40-117)77(131)103-37-67(123)101-36-66(122)102-39-69(125)107-55(74(91)128)17-9-11-28-97-85(139)72-53(15-12-16-54(72)87(141)142)71-51-23-21-49(120)33-64(51)143-65-34-50(121)22-24-52(65)71/h12,15-16,21-24,33-35,42-46,55-63,73,117-118,120H,8-11,13-14,17-20,25-32,36-41,90H2,1-7H3,(H2,91,128)(H,96,104)(H,97,139)(H,100,119)(H,101,123)(H,102,122)(H,103,131)(H,105,132)(H,106,138)(H,107,125)(H,108,124)(H,109,129)(H,110,130)(H,111,133)(H,112,136)(H,113,137)(H,114,140)(H,115,134)(H,116,135)(H,126,127)(H,141,142)(H4,92,93,98)(H4,94,95,99)/t45-,46-,55-,56-,57-,58-,59-,60-,61-,62-,63-,73-/m0/s1	UHBFDUIAGURJOH-FFCVXIFFSA-N	50318531	(7S,19S,22S,25S,28S,31S,34S,37S)-31-((1H-imidazol-5-yl)methyl)-37-((2S,5S,8S,11S)-14-amino-5-(3-guanidinopropyl)-11-(hydroxymethyl)-2,8-dimethyl-4,7,10,13-tetraoxo-3,6,9,12-tetraazatetradecanamido)-22-(4-aminobutyl)-7-carbamoyl-1-(2-carboxy-6-(6-hydroxy-3-oxo-3H-xanthen-9-yl)phenyl)-25-(3-guanidinopropyl)-19-(hydroxymethyl)-28-isobutyl-34-isopropyl-1,9,12,15,18,21,24,27,30,33,36-undecaoxo-2,8,11,14,17,20,23,26,29,32,35-undecaazatetracontan-40-oic acid::CHEMBL1082287	WD repeat-containing protein 5			 860							ChEMBL	10.1021/jm100139b	10.7270/Q2086678	20575550			Karatas, H; Townsend, EC; Bernard, D; Dou, Y; Wang, S	University of Michigan	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50318531	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50318531&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			91933445	104152892		CHEMBL1082287					1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50913025	CC(C)C[C@H](NC(=O)[C@H](Cc1cnc[nH]1)NC(=O)[C@@H](NC(=O)[C@H](CCC(O)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCN=C(N)N)NC(=O)[C@H](C)NC(=O)[C@H](CO)NC(=O)CNC(C)=O)C(C)C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CO)C(=O)NCCCCCC(=O)NCCCCCC(=O)N[C@@H](CCCCNC(=O)c1c(cccc1-c1c2ccc(O)cc2oc2cc(=O)ccc12)C(O)=O)C(N)=O	InChI=1S/C95H142N26O26/c1-50(2)41-67(118-89(141)68(42-55-45-102-49-109-55)119-92(144)79(51(3)4)121-87(139)66(33-34-76(130)131)115-82(134)52(5)110-84(136)64(25-19-39-106-94(98)99)114-81(133)53(6)111-90(142)70(48-123)113-75(129)46-108-54(7)124)88(140)117-65(26-20-40-107-95(100)101)85(137)116-63(24-12-14-35-96)86(138)120-69(47-122)83(135)104-37-16-8-10-27-73(127)103-36-15-9-11-28-74(128)112-62(80(97)132)23-13-17-38-105-91(143)78-60(21-18-22-61(78)93(145)146)77-58-31-29-56(125)43-71(58)147-72-44-57(126)30-32-59(72)77/h18,21-22,29-32,43-45,49-53,62-70,79,122-123,125H,8-17,19-20,23-28,33-42,46-48,96H2,1-7H3,(H2,97,132)(H,102,109)(H,103,127)(H,104,135)(H,105,143)(H,108,124)(H,110,136)(H,111,142)(H,112,128)(H,113,129)(H,114,133)(H,115,134)(H,116,137)(H,117,140)(H,118,141)(H,119,144)(H,120,138)(H,121,139)(H,130,131)(H,145,146)(H4,98,99,106)(H4,100,101,107)/t52-,53-,62-,63-,64-,65-,66-,67-,68-,69-,70-,79-/m0/s1	UUCMVZMMEMCWDP-JTVDXHOOSA-N	50318532	(7S,24S,27S,30S,33S,36S,39S,42S)-36-((1H-imidazol-5-yl)methyl)-42-((2S,5S,8S,11S)-14-amino-5-(3-guanidinopropyl)-11-(hydroxymethyl)-2,8-dimethyl-4,7,10,13-tetraoxo-3,6,9,12-tetraazatetradecanamido)-27-(4-aminobutyl)-7-carbamoyl-1-(2-carboxy-6-(6-hydroxy-3-oxo-3H-xanthen-9-yl)phenyl)-30-(3-guanidinopropyl)-24-(hydroxymethyl)-33-isobutyl-39-isopropyl-1,9,16,23,26,29,32,35,38,41-decaoxo-2,8,15,22,25,28,31,34,37,40-decaazapentatetracontan-45-oic acid::CHEMBL1082288	WD repeat-containing protein 5			 940							ChEMBL	10.1021/jm100139b	10.7270/Q2086678	20575550			Karatas, H; Townsend, EC; Bernard, D; Dou, Y; Wang, S	University of Michigan	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50318532	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50318532&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			91933446	104152893		CHEMBL1082288					1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50913026	CC(C)C[C@H](NC(=O)[C@H](Cc1cnc[nH]1)NC(=O)[C@@H](NC(=O)[C@H](CCC(O)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCN=C(N)N)NC(=O)[C@H](C)NC(C)=O)C(C)C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CO)C(=O)NCCCCCC(=O)NCCCCCC(=O)N[C@@H](CCCCNC(=O)c1c(cccc1-c1c2ccc(O)cc2oc2cc(=O)ccc12)C(O)=O)C(N)=O	InChI=1S/C90H134N24O23/c1-48(2)41-65(111-85(132)66(42-53-45-97-47-103-53)112-87(134)75(49(3)4)114-83(130)64(33-34-72(121)122)108-78(125)51(6)105-80(127)62(25-19-39-101-89(93)94)107-77(124)50(5)104-52(7)116)84(131)110-63(26-20-40-102-90(95)96)81(128)109-61(24-12-14-35-91)82(129)113-67(46-115)79(126)99-37-16-8-10-27-70(119)98-36-15-9-11-28-71(120)106-60(76(92)123)23-13-17-38-100-86(133)74-58(21-18-22-59(74)88(135)136)73-56-31-29-54(117)43-68(56)137-69-44-55(118)30-32-57(69)73/h18,21-22,29-32,43-45,47-51,60-67,75,115,117H,8-17,19-20,23-28,33-42,46,91H2,1-7H3,(H2,92,123)(H,97,103)(H,98,119)(H,99,126)(H,100,133)(H,104,116)(H,105,127)(H,106,120)(H,107,124)(H,108,125)(H,109,128)(H,110,131)(H,111,132)(H,112,134)(H,113,129)(H,114,130)(H,121,122)(H,135,136)(H4,93,94,101)(H4,95,96,102)/t50-,51-,60-,61-,62-,63-,64-,65-,66-,67-,75-/m0/s1	DUUXVEDLVMAVQN-ATJHPVBWSA-N	50318533	(7S,24S,27S,30S,33S,36S,39S,42S)-36-((1H-imidazol-5-yl)methyl)-27-(4-aminobutyl)-42-((S)-2-((S)-2-((S)-2-aminopropanamido)-5-guanidinopentanamido)propanamido)-7-carbamoyl-1-(2-carboxy-6-(6-hydroxy-3-oxo-3H-xanthen-9-yl)phenyl)-30-(3-guanidinopropyl)-24-(hydroxymethyl)-33-isobutyl-39-isopropyl-1,9,16,23,26,29,32,35,38,41-decaoxo-2,8,15,22,25,28,31,34,37,40-decaazapentatetracontan-45-oic acid::CHEMBL1082289	WD repeat-containing protein 5			 14							ChEMBL	10.1021/jm100139b	10.7270/Q2086678	20575550			Karatas, H; Townsend, EC; Bernard, D; Dou, Y; Wang, S	University of Michigan	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50318533	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50318533&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			91933447	104152894		CHEMBL1082289			C04341		1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50913027	CC(C)C[C@H](NC(=O)[C@H](Cc1cnc[nH]1)NC(=O)[C@@H](NC(=O)[C@H](CCC(O)=O)NC(=O)[C@@H](NC(=O)[C@H](CCCN=C(N)N)NC(=O)[C@H](C)NC(C)=O)[C@@H](C)O)C(C)C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CO)C(=O)NCCCCCC(=O)NCCCCCC(=O)N[C@@H](CCCCNC(=O)c1c(cccc1-c1c2ccc(O)cc2oc2cc(=O)ccc12)C(O)=O)C(N)=O	InChI=1S/C91H136N24O24/c1-48(2)41-65(111-85(133)66(42-53-45-98-47-104-53)112-87(135)75(49(3)4)114-83(131)64(33-34-72(123)124)110-88(136)76(51(6)117)115-82(130)63(26-20-40-103-91(96)97)107-78(126)50(5)105-52(7)118)84(132)109-62(25-19-39-102-90(94)95)80(128)108-61(24-12-14-35-92)81(129)113-67(46-116)79(127)100-37-16-8-10-27-70(121)99-36-15-9-11-28-71(122)106-60(77(93)125)23-13-17-38-101-86(134)74-58(21-18-22-59(74)89(137)138)73-56-31-29-54(119)43-68(56)139-69-44-55(120)30-32-57(69)73/h18,21-22,29-32,43-45,47-51,60-67,75-76,116-117,119H,8-17,19-20,23-28,33-42,46,92H2,1-7H3,(H2,93,125)(H,98,104)(H,99,121)(H,100,127)(H,101,134)(H,105,118)(H,106,122)(H,107,126)(H,108,128)(H,109,132)(H,110,136)(H,111,133)(H,112,135)(H,113,129)(H,114,131)(H,115,130)(H,123,124)(H,137,138)(H4,94,95,102)(H4,96,97,103)/t50-,51+,60-,61-,62-,63-,64-,65-,66-,67-,75-,76-/m0/s1	XFKKUYQYPPAGIQ-PIHYDPKYSA-N	50318534	(7S,24S,27S,30S,33S,36S,39S,42S)-36-((1H-imidazol-5-yl)methyl)-27-(4-aminobutyl)-42-((2S,3R)-2-((S)-2-((S)-2-aminopropanamido)-5-guanidinopentanamido)-3-hydroxybutanamido)-7-carbamoyl-1-(2-carboxy-6-(6-hydroxy-3-oxo-3H-xanthen-9-yl)phenyl)-30-(3-guanidinopropyl)-24-(hydroxymethyl)-33-isobutyl-39-isopropyl-1,9,16,23,26,29,32,35,38,41-decaoxo-2,8,15,22,25,28,31,34,37,40-decaazapentatetracontan-45-oic acid::CHEMBL1082290	WD repeat-containing protein 5			 1							ChEMBL	10.1021/jm100139b	10.7270/Q2086678	20575550			Karatas, H; Townsend, EC; Bernard, D; Dou, Y; Wang, S	University of Michigan	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50318534	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50318534&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			91933448	104152895		CHEMBL1082290			C04341		1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50913028	CC(C)C[C@H](NC(=O)[C@H](Cc1cnc[nH]1)NC(=O)[C@@H](NC(=O)[C@H](CCC(O)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCN=C(N)N)NC(=O)[C@H](C)N)C(C)C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CO)C(N)=O	InChI=1S/C49H88N20O13/c1-24(2)19-33(45(80)65-31(13-10-18-59-49(55)56)42(77)64-29(11-7-8-16-50)43(78)68-35(22-70)38(52)73)66-46(81)34(20-28-21-57-23-60-28)67-47(82)37(25(3)4)69-44(79)32(14-15-36(71)72)63-40(75)27(6)61-41(76)30(62-39(74)26(5)51)12-9-17-58-48(53)54/h21,23-27,29-35,37,70H,7-20,22,50-51H2,1-6H3,(H2,52,73)(H,57,60)(H,61,76)(H,62,74)(H,63,75)(H,64,77)(H,65,80)(H,66,81)(H,67,82)(H,68,78)(H,69,79)(H,71,72)(H4,53,54,58)(H4,55,56,59)/t26-,27-,29-,30-,31-,32-,33-,34-,35-,37-/m0/s1	QSYBTXGBZPBRSE-CSNULDERSA-N	50318535	CHEMBL1086456::H2N-ARAEVHLRKS-NH2	WD repeat-containing protein 5		 7300								ChEMBL	10.1021/jm100139b	10.7270/Q2086678	20575550			Karatas, H; Townsend, EC; Bernard, D; Dou, Y; Wang, S	University of Michigan	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50318535	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50318535&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			46867122	104152896		CHEMBL1086456			C03803		1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50913029	C[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](C)C(N)=O	InChI=1S/C12H25N7O3/c1-6(13)10(21)19-8(4-3-5-17-12(15)16)11(22)18-7(2)9(14)20/h6-8H,3-5,13H2,1-2H3,(H2,14,20)(H,18,22)(H,19,21)(H4,15,16,17)/t6-,7-,8-/m0/s1	AQIJXACCRBWZOI-FXQIFTODSA-N	50318536	CHEMBL1085606::H2N-ARA-NH2	WD repeat-containing protein 5		>50000								ChEMBL	10.1021/jm100139b	10.7270/Q2086678	20575550			Karatas, H; Townsend, EC; Bernard, D; Dou, Y; Wang, S	University of Michigan	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50318536	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50318536&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			46889983	104152897		CHEMBL1085606			C03803	ZINC49111234	1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50913030	C[C@H](NC(=O)[C@H](CCCN=C(N)N)NC(=O)[C@H](C)NC=O)C(N)=O	InChI=1S/C13H25N7O4/c1-7(10(14)22)19-12(24)9(4-3-5-17-13(15)16)20-11(23)8(2)18-6-21/h6-9H,3-5H2,1-2H3,(H2,14,22)(H,18,21)(H,19,24)(H,20,23)(H4,15,16,17)/t7-,8-,9-/m0/s1	FEPXALARCRYGSN-CIUDSAMLSA-N	50318537	CHEMBL1086083::CHO-ARA-NH2	WD repeat-containing protein 5		 3200								ChEMBL	10.1021/jm100139b	10.7270/Q2086678	20575550			Karatas, H; Townsend, EC; Bernard, D; Dou, Y; Wang, S	University of Michigan	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50318537	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50318537&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			46889984	104152898		CHEMBL1086083			C06049	ZINC49053925	1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50913031	C[C@H](NC(C)=O)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N(C)[C@@H](C)C(N)=O	InChI=1S/C15H29N7O4/c1-8(20-10(3)23)13(25)21-11(6-5-7-19-15(17)18)14(26)22(4)9(2)12(16)24/h8-9,11H,5-7H2,1-4H3,(H2,16,24)(H,20,23)(H,21,25)(H4,17,18,19)/t8-,9-,11-/m0/s1	YQYYSSWBEIIDLB-QXEWZRGKSA-N	50318538	Ac-AR-(N-Me)A-NH2::CHEMBL1084620	WD repeat-containing protein 5		>50000								ChEMBL	10.1021/jm100139b	10.7270/Q2086678	20575550			Karatas, H; Townsend, EC; Bernard, D; Dou, Y; Wang, S	University of Michigan	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50318538	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50318538&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			46889985	104152899		CHEMBL1084620			C04341	ZINC49046210	1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50913032	CNC(=O)[C@H](C)NC(=O)[C@H](CCCN=C(N)N)NC(=O)[C@H](C)NC(C)=O	InChI=1S/C15H29N7O4/c1-8(12(24)18-4)21-14(26)11(6-5-7-19-15(16)17)22-13(25)9(2)20-10(3)23/h8-9,11H,5-7H2,1-4H3,(H,18,24)(H,20,23)(H,21,26)(H,22,25)(H4,16,17,19)/t8-,9-,11-/m0/s1	PYWIZEZTCCLSTR-QXEWZRGKSA-N	50318521	Ac-ARA-CONHMe::CHEMBL1084621	WD repeat-containing protein 5		 150								ChEMBL	10.1021/jm100139b	10.7270/Q2086678	20575550			Karatas, H; Townsend, EC; Bernard, D; Dou, Y; Wang, S	University of Michigan	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50318521	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50318521&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			46889986	104152882		CHEMBL1084621			C04341	ZINC49046214	1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50913033	C[C@H](NC(C)=O)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](C)C(=O)N(C)C	InChI=1S/C16H31N7O4/c1-9(20-11(3)24)13(25)22-12(7-6-8-19-16(17)18)14(26)21-10(2)15(27)23(4)5/h9-10,12H,6-8H2,1-5H3,(H,20,24)(H,21,26)(H,22,25)(H4,17,18,19)/t9-,10-,12-/m0/s1	XFBVAZQSPWDVFU-NHCYSSNCSA-N	50318522	Ac-ARA-CONMe2::CHEMBL1084622	WD repeat-containing protein 5		 6500								ChEMBL	10.1021/jm100139b	10.7270/Q2086678	20575550			Karatas, H; Townsend, EC; Bernard, D; Dou, Y; Wang, S	University of Michigan	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50318522	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50318522&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			46889987	104152883		CHEMBL1084622			C04341	ZINC49046218	1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50913034	COC(=O)[C@H](C)NC(=O)[C@H](CCCN=C(N)N)NC(=O)[C@H](C)NC(C)=O	InChI=1S/C15H28N6O5/c1-8(19-10(3)22)12(23)21-11(6-5-7-18-15(16)17)13(24)20-9(2)14(25)26-4/h8-9,11H,5-7H2,1-4H3,(H,19,22)(H,20,24)(H,21,23)(H4,16,17,18)/t8-,9-,11-/m0/s1	VXMGKWGBQTWNEN-QXEWZRGKSA-N	50318523	Ac-ARA-COOCH3::CHEMBL1084623	WD repeat-containing protein 5		 1600								ChEMBL	10.1021/jm100139b	10.7270/Q2086678	20575550			Karatas, H; Townsend, EC; Bernard, D; Dou, Y; Wang, S	University of Michigan	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50318523	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50318523&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			46889988	104152884		CHEMBL1084623			C04341	ZINC49802194	1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50913035	C[C@@H](O)[C@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@@H](NC(=O)[C@H](CCCN=C(N)N)NC(=O)[C@H](C)N)[C@@H](C)O)C(=O)N[C@@H](C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CO)C(N)=O	InChI=1S/C46H88N20O14/c1-22(49)36(72)59-29(14-10-20-57-46(54)55)41(77)66-34(25(4)69)44(80)63-27(12-6-8-18-48)38(74)62-30(15-16-32(50)70)42(78)65-33(24(3)68)43(79)58-23(2)37(73)60-28(13-9-19-56-45(52)53)39(75)61-26(11-5-7-17-47)40(76)64-31(21-67)35(51)71/h22-31,33-34,67-69H,5-21,47-49H2,1-4H3,(H2,50,70)(H2,51,71)(H,58,79)(H,59,72)(H,60,73)(H,61,75)(H,62,74)(H,63,80)(H,64,76)(H,65,78)(H,66,77)(H4,52,53,56)(H4,54,55,57)/t22-,23-,24+,25+,26-,27-,28-,29-,30-,31-,33-,34-/m0/s1	OZZZZNRCCWQVLU-ZKJUQCEXSA-N	50318524	CHEMBL1082281::H2N-ARTKQTARKS-NH2	WD repeat-containing protein 5		 15100								ChEMBL	10.1021/jm100139b	10.7270/Q2086678	20575550			Karatas, H; Townsend, EC; Bernard, D; Dou, Y; Wang, S	University of Michigan	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50318524	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50318524&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			46889989	104152885		CHEMBL1082281			C03803		1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50913036	C[C@@H](O)[C@H](NC(=O)[C@H](CCCN=C(N)N)NC(=O)[C@H](C)N)C(N)=O	InChI=1S/C13H27N7O4/c1-6(14)11(23)19-8(4-3-5-18-13(16)17)12(24)20-9(7(2)21)10(15)22/h6-9,21H,3-5,14H2,1-2H3,(H2,15,22)(H,19,23)(H,20,24)(H4,16,17,18)/t6-,7+,8-,9-/m0/s1	TXVGTYORMOSCJR-KZVJFYERSA-N	50318526	CHEMBL1085864::H2N-ART-NH2	WD repeat-containing protein 5		 27300								ChEMBL	10.1021/jm100139b	10.7270/Q2086678	20575550			Karatas, H; Townsend, EC; Bernard, D; Dou, Y; Wang, S	University of Michigan	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50318526	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50318526&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			24757930	104152887		CHEMBL1085864			C03803	ZINC49049659	1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50913037	C[C@@H](O)[C@H](NC(=O)[C@H](CCCN=C(N)N)NC(=O)[C@H](C)NC(C)=O)C(N)=O	InChI=1S/C15H29N7O5/c1-7(20-9(3)24)13(26)21-10(5-4-6-19-15(17)18)14(27)22-11(8(2)23)12(16)25/h7-8,10-11,23H,4-6H2,1-3H3,(H2,16,25)(H,20,24)(H,21,26)(H,22,27)(H4,17,18,19)/t7-,8+,10-,11-/m0/s1	CYECJCHCQBPTIK-OEIWMXHLSA-N	50318527	Ac-ART-NH2::CHEMBL1085865	WD repeat-containing protein 5		 20								ChEMBL	10.1021/jm100139b	10.7270/Q2086678	20575550			Karatas, H; Townsend, EC; Bernard, D; Dou, Y; Wang, S	University of Michigan	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50318527	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50318527&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			46864280	104152888		CHEMBL1085865			C04341	ZINC49049663	1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50913038	C[C@@H](O)[C@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](CCCCN)N(C)C(=O)[C@@H](NC(=O)[C@H](CCCN=C(N)N)NC(=O)[C@H](C)N)[C@@H](C)O)C(=O)N[C@@H](C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CO)C(N)=O	InChI=1S/C47H90N20O14/c1-23(50)37(73)60-29(14-11-21-58-47(55)56)41(77)66-35(26(4)70)45(81)67(5)32(15-7-9-19-49)43(79)63-30(16-17-33(51)71)42(78)65-34(25(3)69)44(80)59-24(2)38(74)61-28(13-10-20-57-46(53)54)39(75)62-27(12-6-8-18-48)40(76)64-31(22-68)36(52)72/h23-32,34-35,68-70H,6-22,48-50H2,1-5H3,(H2,51,71)(H2,52,72)(H,59,80)(H,60,73)(H,61,74)(H,62,75)(H,63,79)(H,64,76)(H,65,78)(H,66,77)(H4,53,54,57)(H4,55,56,58)/t23-,24-,25+,26+,27-,28-,29-,30-,31-,32-,34-,35-/m0/s1	BMQKBMJJUNPVPV-NCKQPBNLSA-N	50318528	CHEMBL1082284::H2N-ARTK(Me)QTARKS-NH2	WD repeat-containing protein 5		 15000								ChEMBL	10.1021/jm100139b	10.7270/Q2086678	20575550			Karatas, H; Townsend, EC; Bernard, D; Dou, Y; Wang, S	University of Michigan	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50318528	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50318528&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			46889993	104152889		CHEMBL1082284			C03803		1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50913039	CNCCCC[C@H](N(C)C(=O)[C@@H](NC(=O)[C@H](CCCN=C(N)N)NC(=O)[C@H](C)N)[C@@H](C)O)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H]([C@@H](C)O)C(=O)N[C@@H](C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CO)C(N)=O	InChI=1S/C48H92N20O14/c1-24(50)38(74)61-30(15-12-22-59-48(55)56)42(78)67-36(27(4)71)46(82)68(6)33(16-8-10-20-57-5)44(80)64-31(17-18-34(51)72)43(79)66-35(26(3)70)45(81)60-25(2)39(75)62-29(14-11-21-58-47(53)54)40(76)63-28(13-7-9-19-49)41(77)65-32(23-69)37(52)73/h24-33,35-36,57,69-71H,7-23,49-50H2,1-6H3,(H2,51,72)(H2,52,73)(H,60,81)(H,61,74)(H,62,75)(H,63,76)(H,64,80)(H,65,77)(H,66,79)(H,67,78)(H4,53,54,58)(H4,55,56,59)/t24-,25-,26+,27+,28-,29-,30-,31-,32-,33-,35-,36-/m0/s1	YJQPFWYFQWTFRD-GTTQRSHYSA-N	50318529	CHEMBL1082285::H2N-ARTK(Me2)QTARKS-NH2	WD repeat-containing protein 5		 9000								ChEMBL	10.1021/jm100139b	10.7270/Q2086678	20575550			Karatas, H; Townsend, EC; Bernard, D; Dou, Y; Wang, S	University of Michigan	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50318529	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50318529&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			46889994	104152890		CHEMBL1082285			C03803		1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50913040	C[C@@H](O)[C@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](CCCCN(C)C)N(C)C(=O)[C@@H](NC(=O)[C@H](CCCN=C(N)N)NC(=O)[C@H](C)N)[C@@H](C)O)C(=O)N[C@@H](C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CO)C(N)=O	InChI=1S/C49H94N20O14/c1-25(51)39(75)61-31(16-13-22-59-49(56)57)43(79)67-37(28(4)72)47(83)69(7)34(17-9-11-23-68(5)6)45(81)64-32(18-19-35(52)73)44(80)66-36(27(3)71)46(82)60-26(2)40(76)62-30(15-12-21-58-48(54)55)41(77)63-29(14-8-10-20-50)42(78)65-33(24-70)38(53)74/h25-34,36-37,70-72H,8-24,50-51H2,1-7H3,(H2,52,73)(H2,53,74)(H,60,82)(H,61,75)(H,62,76)(H,63,77)(H,64,81)(H,65,78)(H,66,80)(H,67,79)(H4,54,55,58)(H4,56,57,59)/t25-,26-,27+,28+,29-,30-,31-,32-,33-,34-,36-,37-/m0/s1	PBPOVNDZNWBXLP-RETRBKMKSA-N	50318530	CHEMBL1082286::H2N-ARTK(Me3)QTARKS-NH2	WD repeat-containing protein 5		 15600								ChEMBL	10.1021/jm100139b	10.7270/Q2086678	20575550			Karatas, H; Townsend, EC; Bernard, D; Dou, Y; Wang, S	University of Michigan	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50318530	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50318530&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			46889995	104152891		CHEMBL1082286			C03803		1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50913041	C[C@H](NC(C)=O)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](C)C(=O)N[C@@H](CCC(O)=O)C(N)=O	InChI=1S/C19H34N8O7/c1-9(24-11(3)28)16(32)27-13(5-4-8-23-19(21)22)18(34)25-10(2)17(33)26-12(15(20)31)6-7-14(29)30/h9-10,12-13H,4-8H2,1-3H3,(H2,20,31)(H,24,28)(H,25,34)(H,26,33)(H,27,32)(H,29,30)(H4,21,22,23)/t9-,10-,12-,13-/m0/s1	ZFNWHWJOGHVTEW-UKJIMTQDSA-N	50318547	Ac-ARAE-NH2::CHEMBL1085604	WD repeat-containing protein 5		 80								ChEMBL	10.1021/jm100139b	10.7270/Q2086678	20575550			Karatas, H; Townsend, EC; Bernard, D; Dou, Y; Wang, S	University of Michigan	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50318547	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50318547&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			46889981	104152908		CHEMBL1085604			C04341	ZINC49047581	1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50913042	C[C@H](NC(=O)[C@H](CCCN=C(N)N)NC(=O)[C@H](C)NC(C)=O)C(N)=O	InChI=1S/C14H27N7O4/c1-7(11(15)23)20-13(25)10(5-4-6-18-14(16)17)21-12(24)8(2)19-9(3)22/h7-8,10H,4-6H2,1-3H3,(H2,15,23)(H,19,22)(H,20,25)(H,21,24)(H4,16,17,18)/t7-,8-,10-/m0/s1	ATPJZQHSTNYINS-NRPADANISA-N	50318548	Ac-ARA-NH2::CHEMBL1086455	WD repeat-containing protein 5		 120								ChEMBL	10.1021/jm100139b	10.7270/Q2086678	20575550			Karatas, H; Townsend, EC; Bernard, D; Dou, Y; Wang, S	University of Michigan	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50318548	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50318548&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			46864279	104152909		CHEMBL1086455			C04341	ZINC49049253	1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50913043	C[C@H](NC(C)=O)C(=O)N[C@@H](CCCN=C(N)N)C(N)=O	InChI=1S/C11H22N6O3/c1-6(16-7(2)18)10(20)17-8(9(12)19)4-3-5-15-11(13)14/h6,8H,3-5H2,1-2H3,(H2,12,19)(H,16,18)(H,17,20)(H4,13,14,15)/t6-,8-/m0/s1	WESUUTFORKSXRD-XPUUQOCRSA-N	50318549	Ac-AR-NH2::CHEMBL1085605	WD repeat-containing protein 5		 27000								ChEMBL	10.1021/jm100139b	10.7270/Q2086678	20575550			Karatas, H; Townsend, EC; Bernard, D; Dou, Y; Wang, S	University of Michigan	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50318549	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50318549&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			46889982	104152910		CHEMBL1085605			C04341	ZINC49047585	1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50913044	CC(C)C[C@H](NC(=O)[C@H](Cc1cnc[nH]1)NC(=O)[C@@H](NC(=O)[C@H](CCC(O)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCN=C(N)N)NC(=O)[C@H](C)NC(=O)[C@H](CO)NC(=O)CNC(C)=O)C(C)C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CO)C(N)=O	InChI=1S/C56H98N22O17/c1-27(2)20-37(51(92)74-35(14-11-19-65-56(61)62)48(89)73-33(12-8-9-17-57)49(90)77-39(24-79)44(58)85)75-52(93)38(21-32-22-63-26-67-32)76-54(95)43(28(3)4)78-50(91)36(15-16-42(83)84)72-46(87)29(5)68-47(88)34(13-10-18-64-55(59)60)71-45(86)30(6)69-53(94)40(25-80)70-41(82)23-66-31(7)81/h22,26-30,33-40,43,79-80H,8-21,23-25,57H2,1-7H3,(H2,58,85)(H,63,67)(H,66,81)(H,68,88)(H,69,94)(H,70,82)(H,71,86)(H,72,87)(H,73,89)(H,74,92)(H,75,93)(H,76,95)(H,77,90)(H,78,91)(H,83,84)(H4,59,60,64)(H4,61,62,65)/t29-,30-,33-,34-,35-,36-,37-,38-,39-,40-,43-/m0/s1	PCONEFYGCDFYOM-UFBWGLHSSA-N	50318539	Ac-GSARAEVHLRKS-NH2::CHEMBL1086448	WD repeat-containing protein 5				 15100						ChEMBL	10.1021/jm100139b	10.7270/Q2086678	20575550			Karatas, H; Townsend, EC; Bernard, D; Dou, Y; Wang, S	University of Michigan	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50318539	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50318539&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			46889977	104152900		CHEMBL1086448					1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50913045	CC(C)C[C@H](NC(=O)[C@H](Cc1cnc[nH]1)NC(=O)[C@@H](NC(=O)[C@H](CCC(O)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCN=C(N)N)NC(=O)[C@H](C)N)C(C)C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CO)C(N)=O	InChI=1S/C49H88N20O13/c1-24(2)19-33(45(80)65-31(13-10-18-59-49(55)56)42(77)64-29(11-7-8-16-50)43(78)68-35(22-70)38(52)73)66-46(81)34(20-28-21-57-23-60-28)67-47(82)37(25(3)4)69-44(79)32(14-15-36(71)72)63-40(75)27(6)61-41(76)30(62-39(74)26(5)51)12-9-17-58-48(53)54/h21,23-27,29-35,37,70H,7-20,22,50-51H2,1-6H3,(H2,52,73)(H,57,60)(H,61,76)(H,62,74)(H,63,75)(H,64,77)(H,65,80)(H,66,81)(H,67,82)(H,68,78)(H,69,79)(H,71,72)(H4,53,54,58)(H4,55,56,59)/t26-,27-,29-,30-,31-,32-,33-,34-,35-,37-/m0/s1	QSYBTXGBZPBRSE-CSNULDERSA-N	50318535	CHEMBL1086456::H2N-ARAEVHLRKS-NH2	WD repeat-containing protein 5			 34000							ChEMBL	10.1021/jm100139b	10.7270/Q2086678	20575550			Karatas, H; Townsend, EC; Bernard, D; Dou, Y; Wang, S	University of Michigan	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50318535	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50318535&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			46867122	104152896		CHEMBL1086456			C03803		1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50913046	C[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](C)C(N)=O	InChI=1S/C12H25N7O3/c1-6(13)10(21)19-8(4-3-5-17-12(15)16)11(22)18-7(2)9(14)20/h6-8H,3-5,13H2,1-2H3,(H2,14,20)(H,18,22)(H,19,21)(H4,15,16,17)/t6-,7-,8-/m0/s1	AQIJXACCRBWZOI-FXQIFTODSA-N	50318536	CHEMBL1085606::H2N-ARA-NH2	WD repeat-containing protein 5			>300000							ChEMBL	10.1021/jm100139b	10.7270/Q2086678	20575550			Karatas, H; Townsend, EC; Bernard, D; Dou, Y; Wang, S	University of Michigan	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50318536	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50318536&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			46889983	104152897		CHEMBL1085606			C03803	ZINC49111234	1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50913047	C[C@H](NC(=O)[C@H](CCCN=C(N)N)NC(=O)[C@H](C)NC=O)C(N)=O	InChI=1S/C13H25N7O4/c1-7(10(14)22)19-12(24)9(4-3-5-17-13(15)16)20-11(23)8(2)18-6-21/h6-9H,3-5H2,1-2H3,(H2,14,22)(H,18,21)(H,19,24)(H,20,23)(H4,15,16,17)/t7-,8-,9-/m0/s1	FEPXALARCRYGSN-CIUDSAMLSA-N	50318537	CHEMBL1086083::CHO-ARA-NH2	WD repeat-containing protein 5			 14900							ChEMBL	10.1021/jm100139b	10.7270/Q2086678	20575550			Karatas, H; Townsend, EC; Bernard, D; Dou, Y; Wang, S	University of Michigan	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50318537	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50318537&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			46889984	104152898		CHEMBL1086083			C06049	ZINC49053925	1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50913048	C[C@H](NC(C)=O)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N(C)[C@@H](C)C(N)=O	InChI=1S/C15H29N7O4/c1-8(20-10(3)23)13(25)21-11(6-5-7-19-15(17)18)14(26)22(4)9(2)12(16)24/h8-9,11H,5-7H2,1-4H3,(H2,16,24)(H,20,23)(H,21,25)(H4,17,18,19)/t8-,9-,11-/m0/s1	YQYYSSWBEIIDLB-QXEWZRGKSA-N	50318538	Ac-AR-(N-Me)A-NH2::CHEMBL1084620	WD repeat-containing protein 5			>300000							ChEMBL	10.1021/jm100139b	10.7270/Q2086678	20575550			Karatas, H; Townsend, EC; Bernard, D; Dou, Y; Wang, S	University of Michigan	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50318538	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50318538&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			46889985	104152899		CHEMBL1084620			C04341	ZINC49046210	1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51049254	CN1CCN(CC1)c1ccc(cc1NC(=O)c1ccc(F)cc1)[N+]([O-])=O	InChI=1S/C18H19FN4O3/c1-21-8-10-22(11-9-21)17-7-6-15(23(25)26)12-16(17)20-18(24)13-2-4-14(19)5-3-13/h2-7,12H,8-11H2,1H3,(H,20,24)	BKPPOLBWVUWRTJ-UHFFFAOYSA-N	50428235	CHEMBL2337028	WD repeat-containing protein 5				 3100						ChEMBL	10.1021/ml300467n	10.7270/Q2C53N6F	24900672			Bolshan, Y; Getlik, M; Kuznetsova, E; Wasney, GA; Hajian, T; Poda, G; Nguyen, KT; Wu, H; Dombrovski, L; Dong, A; Senisterra, G; Schapira, M; Arrowsmith, CH; Brown, PJ; Al-Awar, R; Vedadi, M; Smil, D	EntreMed Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50428235	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50428235&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			71718900	164157110		CHEMBL2337028				ZINC95592807	1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51049255	COc1cccc(c1)C(=O)Nc1cc(ccc1N1CCN(C)CC1)[N+]([O-])=O	InChI=1S/C19H22N4O4/c1-21-8-10-22(11-9-21)18-7-6-15(23(25)26)13-17(18)20-19(24)14-4-3-5-16(12-14)27-2/h3-7,12-13H,8-11H2,1-2H3,(H,20,24)	XUPWXLOPCYFDQV-UHFFFAOYSA-N	50428236	CHEMBL1457864	WD repeat-containing protein 5				 1400						ChEMBL	10.1021/ml300467n	10.7270/Q2C53N6F	24900672			Bolshan, Y; Getlik, M; Kuznetsova, E; Wasney, GA; Hajian, T; Poda, G; Nguyen, KT; Wu, H; Dombrovski, L; Dong, A; Senisterra, G; Schapira, M; Arrowsmith, CH; Brown, PJ; Al-Awar, R; Vedadi, M; Smil, D	EntreMed Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50428236	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50428236&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			2966069	164157111		CHEMBL1457864				ZINC05049440	1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51049256	CN1CCN(CC1)c1ccc(cc1NC(=O)c1cccc(O)c1)[N+]([O-])=O	InChI=1S/C18H20N4O4/c1-20-7-9-21(10-8-20)17-6-5-14(22(25)26)12-16(17)19-18(24)13-3-2-4-15(23)11-13/h2-6,11-12,23H,7-10H2,1H3,(H,19,24)	YJZGLINFUJXTHC-UHFFFAOYSA-N	50428237	CHEMBL2337450	WD repeat-containing protein 5				>10000						ChEMBL	10.1021/ml300467n	10.7270/Q2C53N6F	24900672			Bolshan, Y; Getlik, M; Kuznetsova, E; Wasney, GA; Hajian, T; Poda, G; Nguyen, KT; Wu, H; Dombrovski, L; Dong, A; Senisterra, G; Schapira, M; Arrowsmith, CH; Brown, PJ; Al-Awar, R; Vedadi, M; Smil, D	EntreMed Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50428237	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50428237&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			71718311	164157112		CHEMBL2337450				ZINC95590772	1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51049257	CN1CCN(CC1)c1ccc(cc1NC(=O)c1cccc(C)c1Cl)[N+]([O-])=O	InChI=1S/C19H21ClN4O3/c1-13-4-3-5-15(18(13)20)19(25)21-16-12-14(24(26)27)6-7-17(16)23-10-8-22(2)9-11-23/h3-7,12H,8-11H2,1-2H3,(H,21,25)	CAKDOAZUWFITOS-UHFFFAOYSA-N	50428238	CHEMBL2337449	WD repeat-containing protein 5				 1100						ChEMBL	10.1021/ml300467n	10.7270/Q2C53N6F	24900672			Bolshan, Y; Getlik, M; Kuznetsova, E; Wasney, GA; Hajian, T; Poda, G; Nguyen, KT; Wu, H; Dombrovski, L; Dong, A; Senisterra, G; Schapira, M; Arrowsmith, CH; Brown, PJ; Al-Awar, R; Vedadi, M; Smil, D	EntreMed Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50428238	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50428238&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			71720108	164157113		CHEMBL2337449				ZINC95589405	1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51049258	CN1CCN(CC1)c1ccc(cc1NC(=O)c1cccc(C)c1)[N+]([O-])=O	InChI=1S/C19H22N4O3/c1-14-4-3-5-15(12-14)19(24)20-17-13-16(23(25)26)6-7-18(17)22-10-8-21(2)9-11-22/h3-7,12-13H,8-11H2,1-2H3,(H,20,24)	MYLOZIMRILOZFD-UHFFFAOYSA-N	50428239	CHEMBL2337448	WD repeat-containing protein 5				 1100						ChEMBL	10.1021/ml300467n	10.7270/Q2C53N6F	24900672			Bolshan, Y; Getlik, M; Kuznetsova, E; Wasney, GA; Hajian, T; Poda, G; Nguyen, KT; Wu, H; Dombrovski, L; Dong, A; Senisterra, G; Schapira, M; Arrowsmith, CH; Brown, PJ; Al-Awar, R; Vedadi, M; Smil, D	EntreMed Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50428239	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50428239&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			71719517	164157114		CHEMBL2337448				ZINC95588321	1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51049259	CN1CCN(CC1)c1ccc(cc1NC(=O)c1cccc(Cl)c1)[N+]([O-])=O	InChI=1S/C18H19ClN4O3/c1-21-7-9-22(10-8-21)17-6-5-15(23(25)26)12-16(17)20-18(24)13-3-2-4-14(19)11-13/h2-6,11-12H,7-10H2,1H3,(H,20,24)	QQMREAFPDZRCQL-UHFFFAOYSA-N	50428240	CHEMBL2337447	WD repeat-containing protein 5				 1800						ChEMBL	10.1021/ml300467n	10.7270/Q2C53N6F	24900672			Bolshan, Y; Getlik, M; Kuznetsova, E; Wasney, GA; Hajian, T; Poda, G; Nguyen, KT; Wu, H; Dombrovski, L; Dong, A; Senisterra, G; Schapira, M; Arrowsmith, CH; Brown, PJ; Al-Awar, R; Vedadi, M; Smil, D	EntreMed Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50428240	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50428240&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			71720107	164157115		CHEMBL2337447				ZINC95588890	1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51049260	CN1CCN(CC1)c1ccc(cc1NC(C)=O)[N+]([O-])=O	InChI=1S/C13H18N4O3/c1-10(18)14-12-9-11(17(19)20)3-4-13(12)16-7-5-15(2)6-8-16/h3-4,9H,5-8H2,1-2H3,(H,14,18)	FSQBTKZGKQMDMQ-UHFFFAOYSA-N	50428241	CHEMBL2337446	WD repeat-containing protein 5				>10000						ChEMBL	10.1021/ml300467n	10.7270/Q2C53N6F	24900672			Bolshan, Y; Getlik, M; Kuznetsova, E; Wasney, GA; Hajian, T; Poda, G; Nguyen, KT; Wu, H; Dombrovski, L; Dong, A; Senisterra, G; Schapira, M; Arrowsmith, CH; Brown, PJ; Al-Awar, R; Vedadi, M; Smil, D	EntreMed Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50428241	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50428241&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			2966356	164157116		CHEMBL2337446				ZINC05049873	1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51049261	CN(C)CCN(C)c1ccc(cc1NC(=O)c1ccccc1Cl)[N+]([O-])=O	InChI=1S/C18H21ClN4O3/c1-21(2)10-11-22(3)17-9-8-13(23(25)26)12-16(17)20-18(24)14-6-4-5-7-15(14)19/h4-9,12H,10-11H2,1-3H3,(H,20,24)	BUELYUFPHSYCND-UHFFFAOYSA-N	50428242	CHEMBL2337445	WD repeat-containing protein 5				>20000						ChEMBL	10.1021/ml300467n	10.7270/Q2C53N6F	24900672			Bolshan, Y; Getlik, M; Kuznetsova, E; Wasney, GA; Hajian, T; Poda, G; Nguyen, KT; Wu, H; Dombrovski, L; Dong, A; Senisterra, G; Schapira, M; Arrowsmith, CH; Brown, PJ; Al-Awar, R; Vedadi, M; Smil, D	EntreMed Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50428242	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50428242&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			71717691	164157117		CHEMBL2337445				ZINC95589690	1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51049262	NC1CCN(CC1)c1ccc(cc1NC(=O)c1ccccc1Cl)[N+]([O-])=O	InChI=1S/C18H19ClN4O3/c19-15-4-2-1-3-14(15)18(24)21-16-11-13(23(25)26)5-6-17(16)22-9-7-12(20)8-10-22/h1-6,11-12H,7-10,20H2,(H,21,24)	HEIWDGOGAQQRED-UHFFFAOYSA-N	50428243	CHEMBL2337444	WD repeat-containing protein 5				>20000						ChEMBL	10.1021/ml300467n	10.7270/Q2C53N6F	24900672			Bolshan, Y; Getlik, M; Kuznetsova, E; Wasney, GA; Hajian, T; Poda, G; Nguyen, KT; Wu, H; Dombrovski, L; Dong, A; Senisterra, G; Schapira, M; Arrowsmith, CH; Brown, PJ; Al-Awar, R; Vedadi, M; Smil, D	EntreMed Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50428243	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50428243&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			71719516	164157118		CHEMBL2337444				ZINC95587314	1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51049263	NC1CCN(C1)c1ccc(cc1NC(=O)c1ccccc1Cl)[N+]([O-])=O	InChI=1S/C17H17ClN4O3/c18-14-4-2-1-3-13(14)17(23)20-15-9-12(22(24)25)5-6-16(15)21-8-7-11(19)10-21/h1-6,9,11H,7-8,10,19H2,(H,20,23)	PJYBDMFDAJSLOC-UHFFFAOYSA-N	50428244	CHEMBL2337443	WD repeat-containing protein 5				>20000						ChEMBL	10.1021/ml300467n	10.7270/Q2C53N6F	24900672			Bolshan, Y; Getlik, M; Kuznetsova, E; Wasney, GA; Hajian, T; Poda, G; Nguyen, KT; Wu, H; Dombrovski, L; Dong, A; Senisterra, G; Schapira, M; Arrowsmith, CH; Brown, PJ; Al-Awar, R; Vedadi, M; Smil, D	EntreMed Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50428244	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50428244&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			71718310	164157119		CHEMBL2337443				ZINC95587984	1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51049264	[O-][N+](=O)c1ccc(N2CCNCC2)c(NC(=O)c2ccccc2Cl)c1	InChI=1S/C17H17ClN4O3/c18-14-4-2-1-3-13(14)17(23)20-15-11-12(22(24)25)5-6-16(15)21-9-7-19-8-10-21/h1-6,11,19H,7-10H2,(H,20,23)	UDAPACXOKFFESJ-UHFFFAOYSA-N	50428245	CHEMBL2337442	WD repeat-containing protein 5				>20000						ChEMBL	10.1021/ml300467n	10.7270/Q2C53N6F	24900672			Bolshan, Y; Getlik, M; Kuznetsova, E; Wasney, GA; Hajian, T; Poda, G; Nguyen, KT; Wu, H; Dombrovski, L; Dong, A; Senisterra, G; Schapira, M; Arrowsmith, CH; Brown, PJ; Al-Awar, R; Vedadi, M; Smil, D	EntreMed Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50428245	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50428245&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			71718908	164157120		CHEMBL2337442				ZINC95590206	1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51049265	CN(C)C1CCN(CC1)c1ccc(cc1NC(=O)c1ccccc1Cl)[N+]([O-])=O	InChI=1S/C20H23ClN4O3/c1-23(2)14-9-11-24(12-10-14)19-8-7-15(25(27)28)13-18(19)22-20(26)16-5-3-4-6-17(16)21/h3-8,13-14H,9-12H2,1-2H3,(H,22,26)	VKCPJTGJMTXVTH-UHFFFAOYSA-N	50428246	CHEMBL2337441	WD repeat-containing protein 5				>20000						ChEMBL	10.1021/ml300467n	10.7270/Q2C53N6F	24900672			Bolshan, Y; Getlik, M; Kuznetsova, E; Wasney, GA; Hajian, T; Poda, G; Nguyen, KT; Wu, H; Dombrovski, L; Dong, A; Senisterra, G; Schapira, M; Arrowsmith, CH; Brown, PJ; Al-Awar, R; Vedadi, M; Smil, D	EntreMed Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50428246	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50428246&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			71716466	164157121		CHEMBL2337441				ZINC95591129	1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51049266	CN(C)C1CCN(C1)c1ccc(cc1NC(=O)c1ccccc1Cl)[N+]([O-])=O	InChI=1S/C19H21ClN4O3/c1-22(2)14-9-10-23(12-14)18-8-7-13(24(26)27)11-17(18)21-19(25)15-5-3-4-6-16(15)20/h3-8,11,14H,9-10,12H2,1-2H3,(H,21,25)	WWEQETXLXQGPFH-UHFFFAOYSA-N	50428247	CHEMBL2337039	WD repeat-containing protein 5				 15800						ChEMBL	10.1021/ml300467n	10.7270/Q2C53N6F	24900672			Bolshan, Y; Getlik, M; Kuznetsova, E; Wasney, GA; Hajian, T; Poda, G; Nguyen, KT; Wu, H; Dombrovski, L; Dong, A; Senisterra, G; Schapira, M; Arrowsmith, CH; Brown, PJ; Al-Awar, R; Vedadi, M; Smil, D	EntreMed Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50428247	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50428247&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			71718297	164157122		CHEMBL2337039				ZINC95590299	1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51049267	CCN1CCN(CC1)c1ccc(cc1NC(=O)c1ccccc1Cl)[N+]([O-])=O	InChI=1S/C19H21ClN4O3/c1-2-22-9-11-23(12-10-22)18-8-7-14(24(26)27)13-17(18)21-19(25)15-5-3-4-6-16(15)20/h3-8,13H,2,9-12H2,1H3,(H,21,25)	OTWKATJZXRXYER-UHFFFAOYSA-N	50428248	CHEMBL2337038	WD repeat-containing protein 5				>20000						ChEMBL	10.1021/ml300467n	10.7270/Q2C53N6F	24900672			Bolshan, Y; Getlik, M; Kuznetsova, E; Wasney, GA; Hajian, T; Poda, G; Nguyen, KT; Wu, H; Dombrovski, L; Dong, A; Senisterra, G; Schapira, M; Arrowsmith, CH; Brown, PJ; Al-Awar, R; Vedadi, M; Smil, D	EntreMed Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50428248	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50428248&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			71720102	164157123		CHEMBL2337038				ZINC95592834	1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51049268	[O-][N+](=O)c1ccc(N2CCCCC2)c(NC(=O)c2ccccc2Cl)c1	InChI=1S/C18H18ClN3O3/c19-15-7-3-2-6-14(15)18(23)20-16-12-13(22(24)25)8-9-17(16)21-10-4-1-5-11-21/h2-3,6-9,12H,1,4-5,10-11H2,(H,20,23)	NUZBTILHBGOJEY-UHFFFAOYSA-N	50428249	CHEMBL2337037	WD repeat-containing protein 5				>20000						ChEMBL	10.1021/ml300467n	10.7270/Q2C53N6F	24900672			Bolshan, Y; Getlik, M; Kuznetsova, E; Wasney, GA; Hajian, T; Poda, G; Nguyen, KT; Wu, H; Dombrovski, L; Dong, A; Senisterra, G; Schapira, M; Arrowsmith, CH; Brown, PJ; Al-Awar, R; Vedadi, M; Smil, D	EntreMed Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50428249	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50428249&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			2966177	164157124		CHEMBL2337037				ZINC05049648	1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51049269	[O-][N+](=O)c1ccc(N2CCOCC2)c(NC(=O)c2ccccc2Cl)c1	InChI=1S/C17H16ClN3O4/c18-14-4-2-1-3-13(14)17(22)19-15-11-12(21(23)24)5-6-16(15)20-7-9-25-10-8-20/h1-6,11H,7-10H2,(H,19,22)	UXHRSRFKFFQNBQ-UHFFFAOYSA-N	50428250	CHEMBL2337036	WD repeat-containing protein 5				>20000						ChEMBL	10.1021/ml300467n	10.7270/Q2C53N6F	24900672			Bolshan, Y; Getlik, M; Kuznetsova, E; Wasney, GA; Hajian, T; Poda, G; Nguyen, KT; Wu, H; Dombrovski, L; Dong, A; Senisterra, G; Schapira, M; Arrowsmith, CH; Brown, PJ; Al-Awar, R; Vedadi, M; Smil, D	EntreMed Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50428250	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50428250&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			71717683	164157125		CHEMBL2337036				ZINC95590207	1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51049270	CN1CCCN(CC1)c1ccc(cc1NC(=O)c1ccccc1Cl)[N+]([O-])=O	InChI=1S/C19H21ClN4O3/c1-22-9-4-10-23(12-11-22)18-8-7-14(24(26)27)13-17(18)21-19(25)15-5-2-3-6-16(15)20/h2-3,5-8,13H,4,9-12H2,1H3,(H,21,25)	KGNCUTSDWNMVFL-UHFFFAOYSA-N	50428251	CHEMBL2337035	WD repeat-containing protein 5				 7000						ChEMBL	10.1021/ml300467n	10.7270/Q2C53N6F	24900672			Bolshan, Y; Getlik, M; Kuznetsova, E; Wasney, GA; Hajian, T; Poda, G; Nguyen, KT; Wu, H; Dombrovski, L; Dong, A; Senisterra, G; Schapira, M; Arrowsmith, CH; Brown, PJ; Al-Awar, R; Vedadi, M; Smil, D	EntreMed Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50428251	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50428251&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			71719508	164157126		CHEMBL2337035				ZINC95586369	1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51049271	CC1CN(CCN1C)c1ccc(cc1NC(=O)c1ccccc1Cl)[N+]([O-])=O	InChI=1S/C19H21ClN4O3/c1-13-12-23(10-9-22(13)2)18-8-7-14(24(26)27)11-17(18)21-19(25)15-5-3-4-6-16(15)20/h3-8,11,13H,9-10,12H2,1-2H3,(H,21,25)	FPXFGQWJDCLQGG-UHFFFAOYSA-N	50428252	CHEMBL2337034	WD repeat-containing protein 5				 4700						ChEMBL	10.1021/ml300467n	10.7270/Q2C53N6F	24900672			Bolshan, Y; Getlik, M; Kuznetsova, E; Wasney, GA; Hajian, T; Poda, G; Nguyen, KT; Wu, H; Dombrovski, L; Dong, A; Senisterra, G; Schapira, M; Arrowsmith, CH; Brown, PJ; Al-Awar, R; Vedadi, M; Smil, D	EntreMed Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50428252	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50428252&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			71719507	164157127		CHEMBL2337034				ZINC95589849	1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51049272	[O-][N+](=O)c1ccc(F)c(NC(=O)c2ccccc2Cl)c1	InChI=1S/C13H8ClFN2O3/c14-10-4-2-1-3-9(10)13(18)16-12-7-8(17(19)20)5-6-11(12)15/h1-7H,(H,16,18)	RNKVTOGYKGPJLB-UHFFFAOYSA-N	50428253	CHEMBL2337033	WD repeat-containing protein 5				>20000						ChEMBL	10.1021/ml300467n	10.7270/Q2C53N6F	24900672			Bolshan, Y; Getlik, M; Kuznetsova, E; Wasney, GA; Hajian, T; Poda, G; Nguyen, KT; Wu, H; Dombrovski, L; Dong, A; Senisterra, G; Schapira, M; Arrowsmith, CH; Brown, PJ; Al-Awar, R; Vedadi, M; Smil, D	EntreMed Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50428253	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50428253&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			871463	164157128		CHEMBL2337033				ZINC00437824	1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51049273	CN1CCN(CC1)c1ccc(cc1NC(=O)c1ccccc1Cl)[N+]([O-])=O	InChI=1S/C18H19ClN4O3/c1-21-8-10-22(11-9-21)17-7-6-13(23(25)26)12-16(17)20-18(24)14-4-2-3-5-15(14)19/h2-7,12H,8-11H2,1H3,(H,20,24)	WOGZFCMBPXJNFI-UHFFFAOYSA-N	50428254	CHEMBL1609857	WD repeat-containing protein 5				 6900						ChEMBL	10.1021/ml300467n	10.7270/Q2C53N6F	24900672			Bolshan, Y; Getlik, M; Kuznetsova, E; Wasney, GA; Hajian, T; Poda, G; Nguyen, KT; Wu, H; Dombrovski, L; Dong, A; Senisterra, G; Schapira, M; Arrowsmith, CH; Brown, PJ; Al-Awar, R; Vedadi, M; Smil, D	EntreMed Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50428254	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50428254&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	NP7	3SMR	2965974	164157129		CHEMBL1609857				ZINC05049228	1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51049274	CN1CCN(CC1)c1ccc(cc1NC(=O)c1ccccc1Cl)[N+]([O-])=O	InChI=1S/C18H19ClN4O3/c1-21-8-10-22(11-9-21)17-7-6-13(23(25)26)12-16(17)20-18(24)14-4-2-3-5-15(14)19/h2-7,12H,8-11H2,1H3,(H,20,24)	WOGZFCMBPXJNFI-UHFFFAOYSA-N	50428254	CHEMBL1609857	WD repeat-containing protein 5				 7000						ChEMBL	10.1021/ml300467n	10.7270/Q2C53N6F	24900672			Bolshan, Y; Getlik, M; Kuznetsova, E; Wasney, GA; Hajian, T; Poda, G; Nguyen, KT; Wu, H; Dombrovski, L; Dong, A; Senisterra, G; Schapira, M; Arrowsmith, CH; Brown, PJ; Al-Awar, R; Vedadi, M; Smil, D	EntreMed Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50428254	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50428254&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	NP7	3SMR	2965974	164157129		CHEMBL1609857				ZINC05049228	1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51049275	OC(=O)c1ccc2ccccc2c1-c1c(ccc2ccccc12)C(O)=O	InChI=1S/C22H14O4/c23-21(24)17-11-9-13-5-1-3-7-15(13)19(17)20-16-8-4-2-6-14(16)10-12-18(20)22(25)26/h1-12H,(H,23,24)(H,25,26)	YDZNRNHKJQTGCG-UHFFFAOYSA-N	50428255	CHEMBL1231559	WD repeat-containing protein 5			 6000							ChEMBL	10.1021/ml300467n	10.7270/Q2C53N6F	24900672			Bolshan, Y; Getlik, M; Kuznetsova, E; Wasney, GA; Hajian, T; Poda, G; Nguyen, KT; Wu, H; Dombrovski, L; Dong, A; Senisterra, G; Schapira, M; Arrowsmith, CH; Brown, PJ; Al-Awar, R; Vedadi, M; Smil, D	EntreMed Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50428255	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50428255&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	C1C	3MKS	2810167	164157130		CHEMBL1231559				ZINC00119674	1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51049276	CN1CCN(CC1)c1ccc(cc1NC(=O)c1ccccc1Cl)-c1ccncc1	InChI=1S/C23H23ClN4O/c1-27-12-14-28(15-13-27)22-7-6-18(17-8-10-25-11-9-17)16-21(22)26-23(29)19-4-2-3-5-20(19)24/h2-11,16H,12-15H2,1H3,(H,26,29)	UPWKAPBSVLJPOJ-UHFFFAOYSA-N	50428256	CHEMBL2337027	WD repeat-containing protein 5				 2200						ChEMBL	10.1021/ml300467n	10.7270/Q2C53N6F	24900672			Bolshan, Y; Getlik, M; Kuznetsova, E; Wasney, GA; Hajian, T; Poda, G; Nguyen, KT; Wu, H; Dombrovski, L; Dong, A; Senisterra, G; Schapira, M; Arrowsmith, CH; Brown, PJ; Al-Awar, R; Vedadi, M; Smil, D	EntreMed Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50428256	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50428256&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			71720101	164157131		CHEMBL2337027				ZINC95590072	1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51049277	CN1CCN(CC1)c1ccc(cc1NC(=O)c1ccccc1Cl)-c1ccco1	InChI=1S/C22H22ClN3O2/c1-25-10-12-26(13-11-25)20-9-8-16(21-7-4-14-28-21)15-19(20)24-22(27)17-5-2-3-6-18(17)23/h2-9,14-15H,10-13H2,1H3,(H,24,27)	NXHDMDGEYLWCRN-UHFFFAOYSA-N	50428257	CHEMBL2337026	WD repeat-containing protein 5				 3500						ChEMBL	10.1021/ml300467n	10.7270/Q2C53N6F	24900672			Bolshan, Y; Getlik, M; Kuznetsova, E; Wasney, GA; Hajian, T; Poda, G; Nguyen, KT; Wu, H; Dombrovski, L; Dong, A; Senisterra, G; Schapira, M; Arrowsmith, CH; Brown, PJ; Al-Awar, R; Vedadi, M; Smil, D	EntreMed Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50428257	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50428257&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			71718899	164157132		CHEMBL2337026				ZINC95587353	1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51049278	CN1CCN(CC1)c1ccc(cc1NC(=O)c1ccccc1Cl)C1CC1	InChI=1S/C21H24ClN3O/c1-24-10-12-25(13-11-24)20-9-8-16(15-6-7-15)14-19(20)23-21(26)17-4-2-3-5-18(17)22/h2-5,8-9,14-15H,6-7,10-13H2,1H3,(H,23,26)	VBVCNJXTZLDSHA-UHFFFAOYSA-N	50428258	CHEMBL2337025	WD repeat-containing protein 5				>10000						ChEMBL	10.1021/ml300467n	10.7270/Q2C53N6F	24900672			Bolshan, Y; Getlik, M; Kuznetsova, E; Wasney, GA; Hajian, T; Poda, G; Nguyen, KT; Wu, H; Dombrovski, L; Dong, A; Senisterra, G; Schapira, M; Arrowsmith, CH; Brown, PJ; Al-Awar, R; Vedadi, M; Smil, D	EntreMed Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50428258	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50428258&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			71717061	164157133		CHEMBL2337025				ZINC95588153	1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51049279	CN1CCN(CC1)c1ccc(cc1NC(=O)c1ccccc1Cl)C(O)=O	InChI=1S/C19H20ClN3O3/c1-22-8-10-23(11-9-22)17-7-6-13(19(25)26)12-16(17)21-18(24)14-4-2-3-5-15(14)20/h2-7,12H,8-11H2,1H3,(H,21,24)(H,25,26)	KEPFMIZOMNTDGG-UHFFFAOYSA-N	50428259	CHEMBL2331612	WD repeat-containing protein 5				>10000						ChEMBL	10.1021/ml300467n	10.7270/Q2C53N6F	24900672			Bolshan, Y; Getlik, M; Kuznetsova, E; Wasney, GA; Hajian, T; Poda, G; Nguyen, KT; Wu, H; Dombrovski, L; Dong, A; Senisterra, G; Schapira, M; Arrowsmith, CH; Brown, PJ; Al-Awar, R; Vedadi, M; Smil, D	EntreMed Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50428259	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50428259&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			46285198	164157134		CHEMBL2331612				ZINC21882283	1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51049280	CN1CCN(CC1)c1ccc(N)cc1NC(=O)c1ccccc1Cl	InChI=1S/C18H21ClN4O/c1-22-8-10-23(11-9-22)17-7-6-13(20)12-16(17)21-18(24)14-4-2-3-5-15(14)19/h2-7,12H,8-11,20H2,1H3,(H,21,24)	SDUBCOUFFIWCSZ-UHFFFAOYSA-N	50428260	CHEMBL2337024	WD repeat-containing protein 5				>10000						ChEMBL	10.1021/ml300467n	10.7270/Q2C53N6F	24900672			Bolshan, Y; Getlik, M; Kuznetsova, E; Wasney, GA; Hajian, T; Poda, G; Nguyen, KT; Wu, H; Dombrovski, L; Dong, A; Senisterra, G; Schapira, M; Arrowsmith, CH; Brown, PJ; Al-Awar, R; Vedadi, M; Smil, D	EntreMed Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50428260	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50428260&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			71719506	164157135		CHEMBL2337024				ZINC95592126	1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51049281	CN1CCN(CC1)c1ccc(Br)cc1NC(=O)c1ccccc1Cl	InChI=1S/C18H19BrClN3O/c1-22-8-10-23(11-9-22)17-7-6-13(19)12-16(17)21-18(24)14-4-2-3-5-15(14)20/h2-7,12H,8-11H2,1H3,(H,21,24)	NKADDVCLXKIBGB-UHFFFAOYSA-N	50428261	CHEMBL2337023	WD repeat-containing protein 5				>10000						ChEMBL	10.1021/ml300467n	10.7270/Q2C53N6F	24900672			Bolshan, Y; Getlik, M; Kuznetsova, E; Wasney, GA; Hajian, T; Poda, G; Nguyen, KT; Wu, H; Dombrovski, L; Dong, A; Senisterra, G; Schapira, M; Arrowsmith, CH; Brown, PJ; Al-Awar, R; Vedadi, M; Smil, D	EntreMed Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50428261	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50428261&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			71718898	164157136		CHEMBL2337023				ZINC57468778	1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51049282	CN1CCN(CC1)c1ccc(cc1NC(=O)c1ccccc1Cl)C(F)(F)F	InChI=1S/C19H19ClF3N3O/c1-25-8-10-26(11-9-25)17-7-6-13(19(21,22)23)12-16(17)24-18(27)14-4-2-3-5-15(14)20/h2-7,12H,8-11H2,1H3,(H,24,27)	YTLAEOWNJMXXPD-UHFFFAOYSA-N	50428262	CHEMBL2337022	WD repeat-containing protein 5				>10000						ChEMBL	10.1021/ml300467n	10.7270/Q2C53N6F	24900672			Bolshan, Y; Getlik, M; Kuznetsova, E; Wasney, GA; Hajian, T; Poda, G; Nguyen, KT; Wu, H; Dombrovski, L; Dong, A; Senisterra, G; Schapira, M; Arrowsmith, CH; Brown, PJ; Al-Awar, R; Vedadi, M; Smil, D	EntreMed Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50428262	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50428262&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			37442281	164157137		CHEMBL2337022				ZINC30254641	1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51049283	COC(=O)c1ccc(N2CCN(C)CC2)c(NC(=O)c2ccccc2Cl)c1	InChI=1S/C20H22ClN3O3/c1-23-9-11-24(12-10-23)18-8-7-14(20(26)27-2)13-17(18)22-19(25)15-5-3-4-6-16(15)21/h3-8,13H,9-12H2,1-2H3,(H,22,25)	ZWRKGBYBETUEKJ-UHFFFAOYSA-N	50428263	CHEMBL2337021	WD repeat-containing protein 5				 6600						ChEMBL	10.1021/ml300467n	10.7270/Q2C53N6F	24900672			Bolshan, Y; Getlik, M; Kuznetsova, E; Wasney, GA; Hajian, T; Poda, G; Nguyen, KT; Wu, H; Dombrovski, L; Dong, A; Senisterra, G; Schapira, M; Arrowsmith, CH; Brown, PJ; Al-Awar, R; Vedadi, M; Smil, D	EntreMed Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50428263	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50428263&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			6456876	164157138		CHEMBL2337021				ZINC04412473	1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51049284	CN1CCN(CC1)c1ccc(cc1NC(=O)c1ccco1)[N+]([O-])=O	InChI=1S/C16H18N4O4/c1-18-6-8-19(9-7-18)14-5-4-12(20(22)23)11-13(14)17-16(21)15-3-2-10-24-15/h2-5,10-11H,6-9H2,1H3,(H,17,21)	PKNMGNVMKCLCTL-UHFFFAOYSA-N	50428264	CHEMBL1559278	WD repeat-containing protein 5				>10000						ChEMBL	10.1021/ml300467n	10.7270/Q2C53N6F	24900672			Bolshan, Y; Getlik, M; Kuznetsova, E; Wasney, GA; Hajian, T; Poda, G; Nguyen, KT; Wu, H; Dombrovski, L; Dong, A; Senisterra, G; Schapira, M; Arrowsmith, CH; Brown, PJ; Al-Awar, R; Vedadi, M; Smil, D	EntreMed Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50428264	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50428264&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			2965795	164157139		CHEMBL1559278				ZINC05048926	1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51049285	CN1CCN(CC1)c1ccc(cc1NC(=O)c1cccnc1)[N+]([O-])=O	InChI=1S/C17H19N5O3/c1-20-7-9-21(10-8-20)16-5-4-14(22(24)25)11-15(16)19-17(23)13-3-2-6-18-12-13/h2-6,11-12H,7-10H2,1H3,(H,19,23)	CZFAQVHGTJZPJI-UHFFFAOYSA-N	50428265	CHEMBL2337020	WD repeat-containing protein 5				>10000						ChEMBL	10.1021/ml300467n	10.7270/Q2C53N6F	24900672			Bolshan, Y; Getlik, M; Kuznetsova, E; Wasney, GA; Hajian, T; Poda, G; Nguyen, KT; Wu, H; Dombrovski, L; Dong, A; Senisterra, G; Schapira, M; Arrowsmith, CH; Brown, PJ; Al-Awar, R; Vedadi, M; Smil, D	EntreMed Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50428265	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50428265&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			71718296	164157140		CHEMBL2337020				ZINC95591300	1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51049286	CN1CCN(CC1)c1ccc(cc1NC(=O)Cc1ccccc1)[N+]([O-])=O	InChI=1S/C19H22N4O3/c1-21-9-11-22(12-10-21)18-8-7-16(23(25)26)14-17(18)20-19(24)13-15-5-3-2-4-6-15/h2-8,14H,9-13H2,1H3,(H,20,24)	AXUPWEWVMWMSJE-UHFFFAOYSA-N	50428266	CHEMBL2337019	WD repeat-containing protein 5				>10000						ChEMBL	10.1021/ml300467n	10.7270/Q2C53N6F	24900672			Bolshan, Y; Getlik, M; Kuznetsova, E; Wasney, GA; Hajian, T; Poda, G; Nguyen, KT; Wu, H; Dombrovski, L; Dong, A; Senisterra, G; Schapira, M; Arrowsmith, CH; Brown, PJ; Al-Awar, R; Vedadi, M; Smil, D	EntreMed Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50428266	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50428266&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			2965831	164157141		CHEMBL2337019				ZINC05048970	1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51049287	CN1CCN(CC1)c1ccc(cc1NC(=O)c1cccc2ncccc12)[N+]([O-])=O	InChI=1S/C21H21N5O3/c1-24-10-12-25(13-11-24)20-8-7-15(26(28)29)14-19(20)23-21(27)17-4-2-6-18-16(17)5-3-9-22-18/h2-9,14H,10-13H2,1H3,(H,23,27)	APGXJSWMXYPTEA-UHFFFAOYSA-N	50428267	CHEMBL2337018	WD repeat-containing protein 5				 1500						ChEMBL	10.1021/ml300467n	10.7270/Q2C53N6F	24900672			Bolshan, Y; Getlik, M; Kuznetsova, E; Wasney, GA; Hajian, T; Poda, G; Nguyen, KT; Wu, H; Dombrovski, L; Dong, A; Senisterra, G; Schapira, M; Arrowsmith, CH; Brown, PJ; Al-Awar, R; Vedadi, M; Smil, D	EntreMed Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50428267	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50428267&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			71717060	164157142		CHEMBL2337018				ZINC95589948	1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51049288	CN1CCN(CC1)c1ccc(cc1NC(=O)c1cccc2ccccc12)[N+]([O-])=O	InChI=1S/C22H22N4O3/c1-24-11-13-25(14-12-24)21-10-9-17(26(28)29)15-20(21)23-22(27)19-8-4-6-16-5-2-3-7-18(16)19/h2-10,15H,11-14H2,1H3,(H,23,27)	COUROXWHMHIUCJ-UHFFFAOYSA-N	50428268	CHEMBL2337017	WD repeat-containing protein 5				 710						ChEMBL	10.1021/ml300467n	10.7270/Q2C53N6F	24900672			Bolshan, Y; Getlik, M; Kuznetsova, E; Wasney, GA; Hajian, T; Poda, G; Nguyen, KT; Wu, H; Dombrovski, L; Dong, A; Senisterra, G; Schapira, M; Arrowsmith, CH; Brown, PJ; Al-Awar, R; Vedadi, M; Smil, D	EntreMed Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50428268	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50428268&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			71718295	164157143		CHEMBL2337017				ZINC95589189	1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51049289	CN1CCN(CC1)c1ccc(cc1NC(=O)C1CCCCC1)[N+]([O-])=O	InChI=1S/C18H26N4O3/c1-20-9-11-21(12-10-20)17-8-7-15(22(24)25)13-16(17)19-18(23)14-5-3-2-4-6-14/h7-8,13-14H,2-6,9-12H2,1H3,(H,19,23)	UVXDPFXNDMLVCT-UHFFFAOYSA-N	50428269	CHEMBL2337016	WD repeat-containing protein 5				>10000						ChEMBL	10.1021/ml300467n	10.7270/Q2C53N6F	24900672			Bolshan, Y; Getlik, M; Kuznetsova, E; Wasney, GA; Hajian, T; Poda, G; Nguyen, KT; Wu, H; Dombrovski, L; Dong, A; Senisterra, G; Schapira, M; Arrowsmith, CH; Brown, PJ; Al-Awar, R; Vedadi, M; Smil, D	EntreMed Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50428269	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50428269&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			71716461	164157144		CHEMBL2337016				ZINC95591616	1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51049290	CN1CCN(CC1)c1ccc(cc1NC(=O)c1ccccc1)[N+]([O-])=O	InChI=1S/C18H20N4O3/c1-20-9-11-21(12-10-20)17-8-7-15(22(24)25)13-16(17)19-18(23)14-5-3-2-4-6-14/h2-8,13H,9-12H2,1H3,(H,19,23)	YAJPGTFQZOVDPT-UHFFFAOYSA-N	50428270	CHEMBL1407785	WD repeat-containing protein 5				 5800						ChEMBL	10.1021/ml300467n	10.7270/Q2C53N6F	24900672			Bolshan, Y; Getlik, M; Kuznetsova, E; Wasney, GA; Hajian, T; Poda, G; Nguyen, KT; Wu, H; Dombrovski, L; Dong, A; Senisterra, G; Schapira, M; Arrowsmith, CH; Brown, PJ; Al-Awar, R; Vedadi, M; Smil, D	EntreMed Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50428270	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50428270&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			2966170	164157145		CHEMBL1407785				ZINC05049644	1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51049291	CN1CCN(CC1)c1ccc(cc1NC(=O)c1ccc(F)c(C)c1Cl)[N+]([O-])=O	InChI=1S/C19H20ClFN4O3/c1-12-15(21)5-4-14(18(12)20)19(26)22-16-11-13(25(27)28)3-6-17(16)24-9-7-23(2)8-10-24/h3-6,11H,7-10H2,1-2H3,(H,22,26)	QHWMIGPLLWYRIR-UHFFFAOYSA-N	50428271	CHEMBL2337032	WD repeat-containing protein 5				 270						ChEMBL	10.1021/ml300467n	10.7270/Q2C53N6F	24900672			Bolshan, Y; Getlik, M; Kuznetsova, E; Wasney, GA; Hajian, T; Poda, G; Nguyen, KT; Wu, H; Dombrovski, L; Dong, A; Senisterra, G; Schapira, M; Arrowsmith, CH; Brown, PJ; Al-Awar, R; Vedadi, M; Smil, D	EntreMed Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50428271	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50428271&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	IA9	4IA9	70679466	164157146		CHEMBL2337032				ZINC95589389	1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51049292	COc1cc(ccc1F)C(=O)Nc1cc(ccc1N1CCN(C)CC1)[N+]([O-])=O	InChI=1S/C19H21FN4O4/c1-22-7-9-23(10-8-22)17-6-4-14(24(26)27)12-16(17)21-19(25)13-3-5-15(20)18(11-13)28-2/h3-6,11-12H,7-10H2,1-2H3,(H,21,25)	AHYWBDAIZHOANP-UHFFFAOYSA-N	50428272	CHEMBL2337031	WD repeat-containing protein 5				 680						ChEMBL	10.1021/ml300467n	10.7270/Q2C53N6F	24900672			Bolshan, Y; Getlik, M; Kuznetsova, E; Wasney, GA; Hajian, T; Poda, G; Nguyen, KT; Wu, H; Dombrovski, L; Dong, A; Senisterra, G; Schapira, M; Arrowsmith, CH; Brown, PJ; Al-Awar, R; Vedadi, M; Smil, D	EntreMed Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50428272	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50428272&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			71720755	164157147		CHEMBL2337031				ZINC95590674	1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51049293	CN1CCN(CC1)c1ccc(cc1NC(=O)c1ccc(F)c(C)c1)[N+]([O-])=O	InChI=1S/C19H21FN4O3/c1-13-11-14(3-5-16(13)20)19(25)21-17-12-15(24(26)27)4-6-18(17)23-9-7-22(2)8-10-23/h3-6,11-12H,7-10H2,1-2H3,(H,21,25)	QHEDRWKYLRDRMG-UHFFFAOYSA-N	50428273	CHEMBL2337030	WD repeat-containing protein 5				 590						ChEMBL	10.1021/ml300467n	10.7270/Q2C53N6F	24900672			Bolshan, Y; Getlik, M; Kuznetsova, E; Wasney, GA; Hajian, T; Poda, G; Nguyen, KT; Wu, H; Dombrovski, L; Dong, A; Senisterra, G; Schapira, M; Arrowsmith, CH; Brown, PJ; Al-Awar, R; Vedadi, M; Smil, D	EntreMed Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50428273	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50428273&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			71717063	164157148		CHEMBL2337030				ZINC95590501	1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51049294	CN1CCN(CC1)c1ccc(cc1NC(=O)c1ccc(F)cc1Cl)[N+]([O-])=O	InChI=1S/C18H18ClFN4O3/c1-22-6-8-23(9-7-22)17-5-3-13(24(26)27)11-16(17)21-18(25)14-4-2-12(20)10-15(14)19/h2-5,10-11H,6-9H2,1H3,(H,21,25)	WYHSEIRNBDYXNL-UHFFFAOYSA-N	50428274	CHEMBL2337029	WD repeat-containing protein 5				 630						ChEMBL	10.1021/ml300467n	10.7270/Q2C53N6F	24900672			Bolshan, Y; Getlik, M; Kuznetsova, E; Wasney, GA; Hajian, T; Poda, G; Nguyen, KT; Wu, H; Dombrovski, L; Dong, A; Senisterra, G; Schapira, M; Arrowsmith, CH; Brown, PJ; Al-Awar, R; Vedadi, M; Smil, D	EntreMed Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50428274	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50428274&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			71717062	164157149		CHEMBL2337029				ZINC95588565	1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50521628	CCOC(=O)c1ccc(N2CCN(C)CC2)c(NC(=O)c2ccc(F)c(c2)[N+]([O-])=O)c1	InChI=1S/C21H23FN4O5/c1-3-31-21(28)15-5-7-18(25-10-8-24(2)9-11-25)17(12-15)23-20(27)14-4-6-16(22)19(13-14)26(29)30/h4-7,12-13H,3,8-11H2,1-2H3,(H,23,27)	PNNOENQRMKNOMV-UHFFFAOYSA-N	50195326	CHEMBL3935228	WD repeat-containing protein 5			>20							ChEMBL	10.1016/j.bmc.2016.09.073	10.7270/Q2F47R4K	27720555			Li, DD; Wang, ZH; Chen, WL; Xie, YY; You, QD; Guo, XK	China Pharmaceutical University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50195326	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50195326&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			134148875	375977162		CHEMBL3935228					1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50521629	CN1CCN(CC1)c1ccc(cc1NC(=O)c1ccc(F)c(c1)[N+]([O-])=O)C(=O)Oc1ccccc1	InChI=1S/C25H23FN4O5/c1-28-11-13-29(14-12-28)22-10-8-18(25(32)35-19-5-3-2-4-6-19)15-21(22)27-24(31)17-7-9-20(26)23(16-17)30(33)34/h2-10,15-16H,11-14H2,1H3,(H,27,31)	UBBBAGFZVYRTEM-UHFFFAOYSA-N	50195327	CHEMBL3904098	WD repeat-containing protein 5			 484							ChEMBL	10.1016/j.bmc.2016.09.073	10.7270/Q2F47R4K	27720555			Li, DD; Wang, ZH; Chen, WL; Xie, YY; You, QD; Guo, XK	China Pharmaceutical University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50195327	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50195327&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			134135619	375977163		CHEMBL3904098					1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50521630	COC(=O)c1ccc(N2CCN(C)CC2)c(NC(=O)c2cc(c(F)c(C)c2Cl)[N+]([O-])=O)c1	InChI=1S/C21H22ClFN4O5/c1-12-18(22)14(11-17(19(12)23)27(30)31)20(28)24-15-10-13(21(29)32-3)4-5-16(15)26-8-6-25(2)7-9-26/h4-5,10-11H,6-9H2,1-3H3,(H,24,28)	WFIKFJIEAAJWSY-UHFFFAOYSA-N	50195361	CHEMBL3971604	WD repeat-containing protein 5			 245							ChEMBL	10.1016/j.bmc.2016.09.073	10.7270/Q2F47R4K	27720555			Li, DD; Wang, ZH; Chen, WL; Xie, YY; You, QD; Guo, XK	China Pharmaceutical University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50195361	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50195361&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			134153992	375977164		CHEMBL3971604					1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50521631	COC(=O)c1ccc(N2CCN(C)CC2)c(NC(=O)c2cc(N)c(F)c(C)c2Cl)c1	InChI=1S/C21H24ClFN4O3/c1-12-18(22)14(11-15(24)19(12)23)20(28)25-16-10-13(21(29)30-3)4-5-17(16)27-8-6-26(2)7-9-27/h4-5,10-11H,6-9,24H2,1-3H3,(H,25,28)	PLRPRYDOPJNKDZ-UHFFFAOYSA-N	50195362	CHEMBL3907289	WD repeat-containing protein 5			 47							ChEMBL	10.1016/j.bmc.2016.09.073	10.7270/Q2F47R4K	27720555			Li, DD; Wang, ZH; Chen, WL; Xie, YY; You, QD; Guo, XK	China Pharmaceutical University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50195362	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50195362&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			132580838	375977165		CHEMBL3907289					1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50521632	CCOC(=O)c1ccc(N2CCN(C)CC2)c(NC(=O)c2ccc(F)c(C)c2Cl)c1	InChI=1S/C22H25ClFN3O3/c1-4-30-22(29)15-5-8-19(27-11-9-26(3)10-12-27)18(13-15)25-21(28)16-6-7-17(24)14(2)20(16)23/h5-8,13H,4,9-12H2,1-3H3,(H,25,28)	SVLKQOVNUKFHLT-UHFFFAOYSA-N	50195363	CHEMBL3922104	WD repeat-containing protein 5			 284							ChEMBL	10.1016/j.bmc.2016.09.073	10.7270/Q2F47R4K	27720555			Li, DD; Wang, ZH; Chen, WL; Xie, YY; You, QD; Guo, XK	China Pharmaceutical University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50195363	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50195363&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			134140087	375977166		CHEMBL3922104					1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50521633	CC(C)OC(=O)c1ccc(N2CCN(C)CC2)c(NC(=O)c2ccc(F)c(c2)[N+]([O-])=O)c1	InChI=1S/C22H25FN4O5/c1-14(2)32-22(29)16-5-7-19(26-10-8-25(3)9-11-26)18(12-16)24-21(28)15-4-6-17(23)20(13-15)27(30)31/h4-7,12-14H,8-11H2,1-3H3,(H,24,28)	DNLIZFPSNXONRN-UHFFFAOYSA-N	50195364	CHEMBL3894097	WD repeat-containing protein 5			 1171							ChEMBL	10.1016/j.bmc.2016.09.073	10.7270/Q2F47R4K	27720555			Li, DD; Wang, ZH; Chen, WL; Xie, YY; You, QD; Guo, XK	China Pharmaceutical University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50195364	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50195364&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			134136312	375977167		CHEMBL3894097					1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50521634	CC(C)OC(=O)c1ccc(N2CCN(C)CC2)c(NC(=O)c2ccc(F)c(N)c2)c1	InChI=1S/C22H27FN4O3/c1-14(2)30-22(29)16-5-7-20(27-10-8-26(3)9-11-27)19(13-16)25-21(28)15-4-6-17(23)18(24)12-15/h4-7,12-14H,8-11,24H2,1-3H3,(H,25,28)	PJLBFBFTPCCHAI-UHFFFAOYSA-N	50195365	CHEMBL3943757	WD repeat-containing protein 5			>20							ChEMBL	10.1016/j.bmc.2016.09.073	10.7270/Q2F47R4K	27720555			Li, DD; Wang, ZH; Chen, WL; Xie, YY; You, QD; Guo, XK	China Pharmaceutical University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50195365	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50195365&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			134145666	375977168		CHEMBL3943757					1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50521635	CN1CCN(CC1)c1ccc(cc1NC(=O)c1ccc(F)c(N)c1)C(=O)Oc1ccccc1	InChI=1S/C25H25FN4O3/c1-29-11-13-30(14-12-29)23-10-8-18(25(32)33-19-5-3-2-4-6-19)16-22(23)28-24(31)17-7-9-20(26)21(27)15-17/h2-10,15-16H,11-14,27H2,1H3,(H,28,31)	BLIPFJSFYMJJHD-UHFFFAOYSA-N	50195366	CHEMBL3906985	WD repeat-containing protein 5			>20							ChEMBL	10.1016/j.bmc.2016.09.073	10.7270/Q2F47R4K	27720555			Li, DD; Wang, ZH; Chen, WL; Xie, YY; You, QD; Guo, XK	China Pharmaceutical University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50195366	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50195366&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			134135674	375977169		CHEMBL3906985					1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50521636	CN1CCN(CC1)c1ccc(cc1NC(=O)c1cc(c(F)c(C)c1Cl)[N+]([O-])=O)C(=O)Oc1ccccc1	InChI=1S/C26H24ClFN4O5/c1-16-23(27)19(15-22(24(16)28)32(35)36)25(33)29-20-14-17(26(34)37-18-6-4-3-5-7-18)8-9-21(20)31-12-10-30(2)11-13-31/h3-9,14-15H,10-13H2,1-2H3,(H,29,33)	PWJBUQPIXZCODS-UHFFFAOYSA-N	50195367	CHEMBL3982971	WD repeat-containing protein 5			 812							ChEMBL	10.1016/j.bmc.2016.09.073	10.7270/Q2F47R4K	27720555			Li, DD; Wang, ZH; Chen, WL; Xie, YY; You, QD; Guo, XK	China Pharmaceutical University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50195367	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50195367&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			134157644	375977170		CHEMBL3982971					1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50521637	CN1CCN(CC1)c1ccc(cc1NC(=O)c1ccc(F)c(C)c1Cl)C(=O)OC1CCCCC1	InChI=1S/C26H31ClFN3O3/c1-17-21(28)10-9-20(24(17)27)25(32)29-22-16-18(26(33)34-19-6-4-3-5-7-19)8-11-23(22)31-14-12-30(2)13-15-31/h8-11,16,19H,3-7,12-15H2,1-2H3,(H,29,32)	ATXIWJPPCIZTFI-UHFFFAOYSA-N	50195368	CHEMBL3953704	WD repeat-containing protein 5			>20							ChEMBL	10.1016/j.bmc.2016.09.073	10.7270/Q2F47R4K	27720555			Li, DD; Wang, ZH; Chen, WL; Xie, YY; You, QD; Guo, XK	China Pharmaceutical University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50195368	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50195368&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			134143930	375977171		CHEMBL3953704					1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50521638	CN1CCN(CC1)c1ccc(cc1NC(=O)c1cc(N)c(F)c(C)c1Cl)C(=O)OC1CCCCC1	InChI=1S/C26H32ClFN4O3/c1-16-23(27)19(15-20(29)24(16)28)25(33)30-21-14-17(26(34)35-18-6-4-3-5-7-18)8-9-22(21)32-12-10-31(2)11-13-32/h8-9,14-15,18H,3-7,10-13,29H2,1-2H3,(H,30,33)	SNWJZGNROVHLJC-UHFFFAOYSA-N	50195369	CHEMBL3962459	WD repeat-containing protein 5			 59							ChEMBL	10.1016/j.bmc.2016.09.073	10.7270/Q2F47R4K	27720555			Li, DD; Wang, ZH; Chen, WL; Xie, YY; You, QD; Guo, XK	China Pharmaceutical University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50195369	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50195369&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			134155604	375977172		CHEMBL3962459					1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50521639	CN1CCN(CC1)c1ccc(cc1NC(=O)c1ccc(F)c(C)c1Cl)C(O)=O	InChI=1S/C20H21ClFN3O3/c1-12-15(22)5-4-14(18(12)21)19(26)23-16-11-13(20(27)28)3-6-17(16)25-9-7-24(2)8-10-25/h3-6,11H,7-10H2,1-2H3,(H,23,26)(H,27,28)	AYROZPQFRORZAA-UHFFFAOYSA-N	50195370	CHEMBL3936042	WD repeat-containing protein 5			>20							ChEMBL	10.1016/j.bmc.2016.09.073	10.7270/Q2F47R4K	27720555			Li, DD; Wang, ZH; Chen, WL; Xie, YY; You, QD; Guo, XK	China Pharmaceutical University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50195370	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50195370&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			134149266	375977173		CHEMBL3936042					1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50521640	COC(=O)c1ccc(N2CCN(C)CC2)c(NC(=O)c2cccc(OC)c2)c1	InChI=1S/C21H25N3O4/c1-23-9-11-24(12-10-23)19-8-7-16(21(26)28-3)14-18(19)22-20(25)15-5-4-6-17(13-15)27-2/h4-8,13-14H,9-12H2,1-3H3,(H,22,25)	ZPLBXOVTSNRBFB-UHFFFAOYSA-N	50195371	CHEMBL3906778	WD repeat-containing protein 5				 3000						ChEMBL	10.1016/j.bmc.2016.09.073	10.7270/Q2F47R4K	27720555			Li, DD; Wang, ZH; Chen, WL; Xie, YY; You, QD; Guo, XK	China Pharmaceutical University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50195371	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50195371&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	0BW	3UR4	6457069	375977174		CHEMBL3906778					1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50521641	CCC(CC)(NC(=O)C(C)C)C(=O)N[C@@H](CCCNC(N)=N)C(=O)NC1(CCCC1)C(=O)NC(c1ccc(F)cc1)c1ccc(F)cc1	InChI=1S/C35H49F2N7O4/c1-5-34(6-2,43-29(45)22(3)4)31(47)41-27(10-9-21-40-33(38)39)30(46)44-35(19-7-8-20-35)32(48)42-28(23-11-15-25(36)16-12-23)24-13-17-26(37)18-14-24/h11-18,22,27-28H,5-10,19-21H2,1-4H3,(H,41,47)(H,42,48)(H,43,45)(H,44,46)(H4,38,39,40)/t27-/m0/s1	RZKSQRIPRKWVBU-MHZLTWQESA-N	200723	US9233086, 10L	WD repeat-containing protein 5			 2.4							ChEMBL	10.1016/j.bmc.2016.09.073	10.7270/Q2F47R4K	27720555			Li, DD; Wang, ZH; Chen, WL; Xie, YY; You, QD; Guo, XK	China Pharmaceutical University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=200723	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=200723&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			54766613	318834336							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50521642	COC(=O)c1ccc(N2CCN(C)CC2)c(NC(=O)c2ccc(F)c(N)c2)c1	InChI=1S/C20H23FN4O3/c1-24-7-9-25(10-8-24)18-6-4-14(20(27)28-2)12-17(18)23-19(26)13-3-5-15(21)16(22)11-13/h3-6,11-12H,7-10,22H2,1-2H3,(H,23,26)	YCXCGHRJLIOJRZ-UHFFFAOYSA-N	50195428	CHEMBL3938878	WD repeat-containing protein 5			>20							ChEMBL	10.1016/j.bmc.2016.09.073	10.7270/Q2F47R4K	27720555			Li, DD; Wang, ZH; Chen, WL; Xie, YY; You, QD; Guo, XK	China Pharmaceutical University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50195428	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50195428&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			134149023	375977175		CHEMBL3938878					1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50521643	CN1CCN(CC1)c1ccc(cc1NC(=O)c1ccc(F)c(N)c1)C(=O)OC1CCCCC1	InChI=1S/C25H31FN4O3/c1-29-11-13-30(14-12-29)23-10-8-18(25(32)33-19-5-3-2-4-6-19)16-22(23)28-24(31)17-7-9-20(26)21(27)15-17/h7-10,15-16,19H,2-6,11-14,27H2,1H3,(H,28,31)	AVKUOEOZJRYWPN-UHFFFAOYSA-N	50195429	CHEMBL3956505	WD repeat-containing protein 5			>20							ChEMBL	10.1016/j.bmc.2016.09.073	10.7270/Q2F47R4K	27720555			Li, DD; Wang, ZH; Chen, WL; Xie, YY; You, QD; Guo, XK	China Pharmaceutical University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50195429	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50195429&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			134144485	375977176		CHEMBL3956505					1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50521644	COC(=O)c1ccc(N2CCN(C)CC2)c(NC(=O)c2ccc(F)c(c2)[N+]([O-])=O)c1	InChI=1S/C20H21FN4O5/c1-23-7-9-24(10-8-23)17-6-4-14(20(27)30-2)11-16(17)22-19(26)13-3-5-15(21)18(12-13)25(28)29/h3-6,11-12H,7-10H2,1-2H3,(H,22,26)	KWVCATVDUJCDJM-UHFFFAOYSA-N	50195430	CHEMBL3950744	WD repeat-containing protein 5			 454							ChEMBL	10.1016/j.bmc.2016.09.073	10.7270/Q2F47R4K	27720555			Li, DD; Wang, ZH; Chen, WL; Xie, YY; You, QD; Guo, XK	China Pharmaceutical University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50195430	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50195430&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			134148078	375977177		CHEMBL3950744					1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50521645	CN1CCN(CC1)c1ccc(cc1NC(=O)c1ccc(F)c(c1)[N+]([O-])=O)C(O)=O	InChI=1S/C19H19FN4O5/c1-22-6-8-23(9-7-22)16-5-3-13(19(26)27)10-15(16)21-18(25)12-2-4-14(20)17(11-12)24(28)29/h2-5,10-11H,6-9H2,1H3,(H,21,25)(H,26,27)	CUGSOCSAMZMPMR-UHFFFAOYSA-N	50195431	CHEMBL3965924	WD repeat-containing protein 5			>20							ChEMBL	10.1016/j.bmc.2016.09.073	10.7270/Q2F47R4K	27720555			Li, DD; Wang, ZH; Chen, WL; Xie, YY; You, QD; Guo, XK	China Pharmaceutical University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50195431	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50195431&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			134149901	375977178		CHEMBL3965924					1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50521648	COC(=O)c1ccc(N2CCN(C)CC2)c(NC(=O)c2ccc(F)c(C)c2Cl)c1	InChI=1S/C21H23ClFN3O3/c1-13-16(23)6-5-15(19(13)22)20(27)24-17-12-14(21(28)29-3)4-7-18(17)26-10-8-25(2)9-11-26/h4-7,12H,8-11H2,1-3H3,(H,24,27)	JFXRDCZYPFPWDU-UHFFFAOYSA-N	50195449	CHEMBL3942025	WD repeat-containing protein 5			 433							ChEMBL	10.1016/j.bmc.2016.09.073	10.7270/Q2F47R4K	27720555			Li, DD; Wang, ZH; Chen, WL; Xie, YY; You, QD; Guo, XK	China Pharmaceutical University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50195449	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50195449&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			134145642	375977180		CHEMBL3942025					1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50521649	CC(C)OC(=O)c1ccc(N2CCN(C)CC2)c(NC(=O)c2ccc(F)c(C)c2Cl)c1	InChI=1S/C23H27ClFN3O3/c1-14(2)31-23(30)16-5-8-20(28-11-9-27(4)10-12-28)19(13-16)26-22(29)17-6-7-18(25)15(3)21(17)24/h5-8,13-14H,9-12H2,1-4H3,(H,26,29)	JUFBKCRECNYVRA-UHFFFAOYSA-N	50195451	CHEMBL3903051	WD repeat-containing protein 5			 264							ChEMBL	10.1016/j.bmc.2016.09.073	10.7270/Q2F47R4K	27720555			Li, DD; Wang, ZH; Chen, WL; Xie, YY; You, QD; Guo, XK	China Pharmaceutical University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50195451	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50195451&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			134135702	375977181		CHEMBL3903051					1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50521650	CN1CCN(CC1)c1ccc(cc1NC(=O)c1ccc(F)c(c1)[N+]([O-])=O)C(=O)OC1CCCCC1	InChI=1S/C25H29FN4O5/c1-28-11-13-29(14-12-28)22-10-8-18(25(32)35-19-5-3-2-4-6-19)15-21(22)27-24(31)17-7-9-20(26)23(16-17)30(33)34/h7-10,15-16,19H,2-6,11-14H2,1H3,(H,27,31)	NMVMUWSPFJBBIL-UHFFFAOYSA-N	50195452	CHEMBL3929919	WD repeat-containing protein 5			>20							ChEMBL	10.1016/j.bmc.2016.09.073	10.7270/Q2F47R4K	27720555			Li, DD; Wang, ZH; Chen, WL; Xie, YY; You, QD; Guo, XK	China Pharmaceutical University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50195452	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50195452&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			134137967	375977182		CHEMBL3929919					1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50521651	CN1CCN(CC1)c1ccc(cc1NC(=O)c1cc(c(F)c(C)c1Cl)[N+]([O-])=O)C(=O)OC1CCCCC1	InChI=1S/C26H30ClFN4O5/c1-16-23(27)19(15-22(24(16)28)32(35)36)25(33)29-20-14-17(26(34)37-18-6-4-3-5-7-18)8-9-21(20)31-12-10-30(2)11-13-31/h8-9,14-15,18H,3-7,10-13H2,1-2H3,(H,29,33)	NTIQYFYUMZEOGI-UHFFFAOYSA-N	50195454	CHEMBL3893446	WD repeat-containing protein 5			>20							ChEMBL	10.1016/j.bmc.2016.09.073	10.7270/Q2F47R4K	27720555			Li, DD; Wang, ZH; Chen, WL; Xie, YY; You, QD; Guo, XK	China Pharmaceutical University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50195454	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50195454&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			134137047	375977183		CHEMBL3893446					1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50521653	CN1CCN(CC1)c1ccc(cc1NC(=O)c1ccc(F)c(C)c1Cl)C(=O)Oc1ccccc1	InChI=1S/C26H25ClFN3O3/c1-17-21(28)10-9-20(24(17)27)25(32)29-22-16-18(26(33)34-19-6-4-3-5-7-19)8-11-23(22)31-14-12-30(2)13-15-31/h3-11,16H,12-15H2,1-2H3,(H,29,32)	FNEAREWNQVQFAL-UHFFFAOYSA-N	50195455	CHEMBL3913104	WD repeat-containing protein 5			 162							ChEMBL	10.1016/j.bmc.2016.09.073	10.7270/Q2F47R4K	27720555			Li, DD; Wang, ZH; Chen, WL; Xie, YY; You, QD; Guo, XK	China Pharmaceutical University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50195455	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50195455&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			134143014	375977184		CHEMBL3913104					1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50521654	CN1CCN(CC1)c1ccc(cc1NC(=O)c1cc(N)c(F)c(C)c1Cl)C(=O)Oc1ccccc1	InChI=1S/C26H26ClFN4O3/c1-16-23(27)19(15-20(29)24(16)28)25(33)30-21-14-17(26(34)35-18-6-4-3-5-7-18)8-9-22(21)32-12-10-31(2)11-13-32/h3-9,14-15H,10-13,29H2,1-2H3,(H,30,33)	VKUIARDCYFJGLG-UHFFFAOYSA-N	50195432	CHEMBL3957478	WD repeat-containing protein 5			 26							ChEMBL	10.1016/j.bmc.2016.09.073	10.7270/Q2F47R4K	27720555			Li, DD; Wang, ZH; Chen, WL; Xie, YY; You, QD; Guo, XK	China Pharmaceutical University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50195432	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50195432&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			132580839	375977179		CHEMBL3957478					1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50544302	CN1CCN(CC1)c1ccc(cc1NC(=O)c1cc(N)c(F)c(C)c1Cl)-c1ccc(NC(=O)C2CCNCC2)cc1	InChI=1S/C31H36ClFN6O2/c1-19-28(32)24(18-25(34)29(19)33)31(41)37-26-17-22(5-8-27(26)39-15-13-38(2)14-16-39)20-3-6-23(7-4-20)36-30(40)21-9-11-35-12-10-21/h3-8,17-18,21,35H,9-16,34H2,1-2H3,(H,36,40)(H,37,41)	CZWZZEUKNASAHM-UHFFFAOYSA-N	50208353	CHEMBL3884726	WD repeat-containing protein 5				 7.5						ChEMBL	10.1016/j.ejmech.2016.08.036	10.7270/Q2251M6G	27598236			Li, DD; Chen, WL; Wang, ZH; Xie, YY; Xu, XL; Jiang, ZY; Zhang, XJ; You, QD; Guo, XK	China Pharmaceutical University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50208353	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50208353&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			134130592	375982007		CHEMBL3884726					1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50544303	CN1CCN(CC1)c1ccc(cc1NC(=O)c1cc(N)c(F)c(C)c1Cl)-c1ccc(NC(=O)CCCN)cc1	InChI=1S/C29H34ClFN6O2/c1-18-27(30)22(17-23(33)28(18)31)29(39)35-24-16-20(7-10-25(24)37-14-12-36(2)13-15-37)19-5-8-21(9-6-19)34-26(38)4-3-11-32/h5-10,16-17H,3-4,11-15,32-33H2,1-2H3,(H,34,38)(H,35,39)	PVXYYWORFYROCX-UHFFFAOYSA-N	50208354	CHEMBL3884329	WD repeat-containing protein 5			 7.6							ChEMBL	10.1016/j.ejmech.2016.08.036	10.7270/Q2251M6G	27598236			Li, DD; Chen, WL; Wang, ZH; Xie, YY; Xu, XL; Jiang, ZY; Zhang, XJ; You, QD; Guo, XK	China Pharmaceutical University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50208354	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50208354&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			134130757	375982008		CHEMBL3884329					1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50544304	CC(N)C(=O)Nc1ccc(cc1)-c1ccc(N2CCN(C)CC2)c(NC(=O)c2cc(N)c(F)c(C)c2Cl)c1	InChI=1S/C28H32ClFN6O2/c1-16-25(29)21(15-22(32)26(16)30)28(38)34-23-14-19(6-9-24(23)36-12-10-35(3)11-13-36)18-4-7-20(8-5-18)33-27(37)17(2)31/h4-9,14-15,17H,10-13,31-32H2,1-3H3,(H,33,37)(H,34,38)	NKBTWLQKWYNUFU-UHFFFAOYSA-N	50208355	CHEMBL3885099	WD repeat-containing protein 5			 15							ChEMBL	10.1016/j.ejmech.2016.08.036	10.7270/Q2251M6G	27598236			Li, DD; Chen, WL; Wang, ZH; Xie, YY; Xu, XL; Jiang, ZY; Zhang, XJ; You, QD; Guo, XK	China Pharmaceutical University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50208355	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50208355&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			134131045	375982009		CHEMBL3885099					1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50544305	CN1CCN(CC1)c1ccc(cc1NC(=O)c1cc(N)c(F)c(C)c1Cl)-c1ccc(NC(=O)c2ccccc2)cc1	InChI=1S/C32H31ClFN5O2/c1-20-29(33)25(19-26(35)30(20)34)32(41)37-27-18-23(10-13-28(27)39-16-14-38(2)15-17-39)21-8-11-24(12-9-21)36-31(40)22-6-4-3-5-7-22/h3-13,18-19H,14-17,35H2,1-2H3,(H,36,40)(H,37,41)	GPVQJDJXUWECIP-UHFFFAOYSA-N	50208356	CHEMBL3884738	WD repeat-containing protein 5			 422							ChEMBL	10.1016/j.ejmech.2016.08.036	10.7270/Q2251M6G	27598236			Li, DD; Chen, WL; Wang, ZH; Xie, YY; Xu, XL; Jiang, ZY; Zhang, XJ; You, QD; Guo, XK	China Pharmaceutical University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50208356	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50208356&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			134130958	375982010		CHEMBL3884738					1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50544306	CN1CCN(CC1)c1ccc(cc1NC(=O)c1cccc(c1)[N+]([O-])=O)-c1ccc(cc1)[N+]([O-])=O	InChI=1S/C24H23N5O5/c1-26-11-13-27(14-12-26)23-10-7-18(17-5-8-20(9-6-17)28(31)32)16-22(23)25-24(30)19-3-2-4-21(15-19)29(33)34/h2-10,15-16H,11-14H2,1H3,(H,25,30)	XJIVMMRBTQMQRL-UHFFFAOYSA-N	50208357	CHEMBL3884315	WD repeat-containing protein 5			 285							ChEMBL	10.1016/j.ejmech.2016.08.036	10.7270/Q2251M6G	27598236			Li, DD; Chen, WL; Wang, ZH; Xie, YY; Xu, XL; Jiang, ZY; Zhang, XJ; You, QD; Guo, XK	China Pharmaceutical University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50208357	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50208357&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			134130199	375982011		CHEMBL3884315					1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50544307	COC(=O)c1ccc(cc1)-c1ccc(N2CCN(C)CC2)c(NC(=O)c2cc(c(F)c(C)c2Cl)[N+]([O-])=O)c1	InChI=1S/C27H26ClFN4O5/c1-16-24(28)20(15-23(25(16)29)33(36)37)26(34)30-21-14-19(17-4-6-18(7-5-17)27(35)38-3)8-9-22(21)32-12-10-31(2)11-13-32/h4-9,14-15H,10-13H2,1-3H3,(H,30,34)	FUNIBWOVENEVSY-UHFFFAOYSA-N	50208358	CHEMBL3885409	WD repeat-containing protein 5			 93							ChEMBL	10.1016/j.ejmech.2016.08.036	10.7270/Q2251M6G	27598236			Li, DD; Chen, WL; Wang, ZH; Xie, YY; Xu, XL; Jiang, ZY; Zhang, XJ; You, QD; Guo, XK	China Pharmaceutical University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50208358	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50208358&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			134130465	375982012		CHEMBL3885409					1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50544308	CN1CCN(CC1)c1ccc(cc1NC(=O)c1ccc(F)c(C)c1Cl)-c1ccccc1	InChI=1S/C25H25ClFN3O/c1-17-21(27)10-9-20(24(17)26)25(31)28-22-16-19(18-6-4-3-5-7-18)8-11-23(22)30-14-12-29(2)13-15-30/h3-11,16H,12-15H2,1-2H3,(H,28,31)	IJGXSYJCQSUICM-UHFFFAOYSA-N	50184952	CHEMBL3823476	WD repeat-containing protein 5			 466							ChEMBL	10.1016/j.ejmech.2016.08.036	10.7270/Q2251M6G	27598236			Li, DD; Chen, WL; Wang, ZH; Xie, YY; Xu, XL; Jiang, ZY; Zhang, XJ; You, QD; Guo, XK	China Pharmaceutical University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50184952	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50184952&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			127050387	346550436		CHEMBL3823476					1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50544309	Cc1c(F)ccc(C(=O)Nc2cc(ccc2NCCN)[N+]([O-])=O)c1Cl	InChI=1S/C16H16ClFN4O3/c1-9-12(18)4-3-11(15(9)17)16(23)21-14-8-10(22(24)25)2-5-13(14)20-7-6-19/h2-5,8,20H,6-7,19H2,1H3,(H,21,23)	QIETXXKZXFWBCA-UHFFFAOYSA-N	50208361	CHEMBL3883659	WD repeat-containing protein 5			>20000							ChEMBL	10.1016/j.ejmech.2016.08.036	10.7270/Q2251M6G	27598236			Li, DD; Chen, WL; Wang, ZH; Xie, YY; Xu, XL; Jiang, ZY; Zhang, XJ; You, QD; Guo, XK	China Pharmaceutical University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50208361	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50208361&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			134131302	104085519		CHEMBL3883659				ZINC11679922	1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50544310	CN1CCN(CC1)c1ccc(cc1NC(=O)c1cc(N)c(F)c(C)c1Cl)-c1ccc(NC(=O)CCCN)cc1	InChI=1S/C29H34ClFN6O2/c1-18-27(30)22(17-23(33)28(18)31)29(39)35-24-16-20(7-10-25(24)37-14-12-36(2)13-15-37)19-5-8-21(9-6-19)34-26(38)4-3-11-32/h5-10,16-17H,3-4,11-15,32-33H2,1-2H3,(H,34,38)(H,35,39)	PVXYYWORFYROCX-UHFFFAOYSA-N	50208354	CHEMBL3884329	WD repeat-containing protein 5				 14						ChEMBL	10.1016/j.ejmech.2016.08.036	10.7270/Q2251M6G	27598236			Li, DD; Chen, WL; Wang, ZH; Xie, YY; Xu, XL; Jiang, ZY; Zhang, XJ; You, QD; Guo, XK	China Pharmaceutical University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50208354	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50208354&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			134130757	375982008		CHEMBL3884329					1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50544311	CCCC(=O)Nc1ccc(cc1)-c1ccc(N2CCN(C)CC2)c(NC(=O)c2cc(N)c(F)c(C)c2Cl)c1	InChI=1S/C29H33ClFN5O2/c1-4-5-26(37)33-21-9-6-19(7-10-21)20-8-11-25(36-14-12-35(3)13-15-36)24(16-20)34-29(38)22-17-23(32)28(31)18(2)27(22)30/h6-11,16-17H,4-5,12-15,32H2,1-3H3,(H,33,37)(H,34,38)	HKSCDRGODSGHMJ-UHFFFAOYSA-N	50208365	CHEMBL3885462	WD repeat-containing protein 5			 76							ChEMBL	10.1016/j.ejmech.2016.08.036	10.7270/Q2251M6G	27598236			Li, DD; Chen, WL; Wang, ZH; Xie, YY; Xu, XL; Jiang, ZY; Zhang, XJ; You, QD; Guo, XK	China Pharmaceutical University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50208365	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50208365&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			134131410	375982013		CHEMBL3885462					1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50544312	CN1CCN(CC1)c1ccc(cc1NC(=O)c1cc(c(F)c(C)c1Cl)[N+]([O-])=O)-c1ccncc1	InChI=1S/C24H23ClFN5O3/c1-15-22(25)18(14-21(23(15)26)31(33)34)24(32)28-19-13-17(16-5-7-27-8-6-16)3-4-20(19)30-11-9-29(2)10-12-30/h3-8,13-14H,9-12H2,1-2H3,(H,28,32)	ACUIMZWGYBOVKD-UHFFFAOYSA-N	50208366	CHEMBL3885279	WD repeat-containing protein 5			 77							ChEMBL	10.1016/j.ejmech.2016.08.036	10.7270/Q2251M6G	27598236			Li, DD; Chen, WL; Wang, ZH; Xie, YY; Xu, XL; Jiang, ZY; Zhang, XJ; You, QD; Guo, XK	China Pharmaceutical University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50208366	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50208366&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			134130278	375982014		CHEMBL3885279					1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50544313	Cc1c(F)ccc(C(=O)Nc2cc(ccc2N2CCN(CC2)c2ccc(F)cc2)[N+]([O-])=O)c1Cl	InChI=1S/C24H21ClF2N4O3/c1-15-20(27)8-7-19(23(15)25)24(32)28-21-14-18(31(33)34)6-9-22(21)30-12-10-29(11-13-30)17-4-2-16(26)3-5-17/h2-9,14H,10-13H2,1H3,(H,28,32)	TWDNCVYJWJBLGG-UHFFFAOYSA-N	50208367	CHEMBL3883759	WD repeat-containing protein 5			>20000							ChEMBL	10.1016/j.ejmech.2016.08.036	10.7270/Q2251M6G	27598236			Li, DD; Chen, WL; Wang, ZH; Xie, YY; Xu, XL; Jiang, ZY; Zhang, XJ; You, QD; Guo, XK	China Pharmaceutical University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50208367	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50208367&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			134130359	375982015		CHEMBL3883759					1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50544314	CN1CCN(CC1)c1ccc(cc1NC(=O)c1ccc(F)c(c1)[N+]([O-])=O)-c1ccncc1	InChI=1S/C23H22FN5O3/c1-27-10-12-28(13-11-27)21-5-3-17(16-6-8-25-9-7-16)14-20(21)26-23(30)18-2-4-19(24)22(15-18)29(31)32/h2-9,14-15H,10-13H2,1H3,(H,26,30)	GHGXZZPYSYWLSZ-UHFFFAOYSA-N	50208368	CHEMBL3885231	WD repeat-containing protein 5			 198							ChEMBL	10.1016/j.ejmech.2016.08.036	10.7270/Q2251M6G	27598236			Li, DD; Chen, WL; Wang, ZH; Xie, YY; Xu, XL; Jiang, ZY; Zhang, XJ; You, QD; Guo, XK	China Pharmaceutical University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50208368	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50208368&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			134130102	375982016		CHEMBL3885231					1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50544315	CN1CCN(CC1)c1ccc(cc1NC(=O)c1cc(N)c(F)c(C)c1Cl)-c1ccncc1	InChI=1S/C24H25ClFN5O/c1-15-22(25)18(14-19(27)23(15)26)24(32)29-20-13-17(16-5-7-28-8-6-16)3-4-21(20)31-11-9-30(2)10-12-31/h3-8,13-14H,9-12,27H2,1-2H3,(H,29,32)	OLHOQKZOYHDOQK-UHFFFAOYSA-N	50208369	CHEMBL3884291	WD repeat-containing protein 5			 18							ChEMBL	10.1016/j.ejmech.2016.08.036	10.7270/Q2251M6G	27598236			Li, DD; Chen, WL; Wang, ZH; Xie, YY; Xu, XL; Jiang, ZY; Zhang, XJ; You, QD; Guo, XK	China Pharmaceutical University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50208369	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50208369&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			134130570	375982017		CHEMBL3884291					1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50544316	CN1CCN(CC1)c1ccc(cc1NC(=O)c1ccc(F)c(C)c1Cl)[N+]([O-])=O	InChI=1S/C19H20ClFN4O3/c1-12-15(21)5-4-14(18(12)20)19(26)22-16-11-13(25(27)28)3-6-17(16)24-9-7-23(2)8-10-24/h3-6,11H,7-10H2,1-2H3,(H,22,26)	QHWMIGPLLWYRIR-UHFFFAOYSA-N	50428271	CHEMBL2337032	WD repeat-containing protein 5			 338							ChEMBL	10.1016/j.ejmech.2016.08.036	10.7270/Q2251M6G	27598236			Li, DD; Chen, WL; Wang, ZH; Xie, YY; Xu, XL; Jiang, ZY; Zhang, XJ; You, QD; Guo, XK	China Pharmaceutical University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50428271	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50428271&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	IA9	4IA9	70679466	164157146		CHEMBL2337032				ZINC95589389	1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50544318	CC(C)C(=O)Nc1ccc(cc1)-c1ccc(N2CCN(C)CC2)c(NC(=O)c2cc(N)c(F)c(C)c2Cl)c1	InChI=1S/C29H33ClFN5O2/c1-17(2)28(37)33-21-8-5-19(6-9-21)20-7-10-25(36-13-11-35(4)12-14-36)24(15-20)34-29(38)22-16-23(32)27(31)18(3)26(22)30/h5-10,15-17H,11-14,32H2,1-4H3,(H,33,37)(H,34,38)	JARBRNCXRXGKGG-UHFFFAOYSA-N	50208370	CHEMBL3884538	WD repeat-containing protein 5			 96							ChEMBL	10.1016/j.ejmech.2016.08.036	10.7270/Q2251M6G	27598236			Li, DD; Chen, WL; Wang, ZH; Xie, YY; Xu, XL; Jiang, ZY; Zhang, XJ; You, QD; Guo, XK	China Pharmaceutical University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50208370	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50208370&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			134130945	375982018		CHEMBL3884538					1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50544319	CN1CCN(CC1)c1ccc(cc1NC(=O)c1cc(NC(C)=O)c(F)c(C)c1Cl)-c1ccc(cc1)[N+]([O-])=O	InChI=1S/C27H27ClFN5O4/c1-16-25(28)21(15-23(26(16)29)30-17(2)35)27(36)31-22-14-19(18-4-7-20(8-5-18)34(37)38)6-9-24(22)33-12-10-32(3)11-13-33/h4-9,14-15H,10-13H2,1-3H3,(H,30,35)(H,31,36)	BABRCHGZJZETCK-UHFFFAOYSA-N	50208371	CHEMBL3884067	WD repeat-containing protein 5			>20000							ChEMBL	10.1016/j.ejmech.2016.08.036	10.7270/Q2251M6G	27598236			Li, DD; Chen, WL; Wang, ZH; Xie, YY; Xu, XL; Jiang, ZY; Zhang, XJ; You, QD; Guo, XK	China Pharmaceutical University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50208371	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50208371&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			134130903	375982019		CHEMBL3884067					1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50544321	CN1CCN(CC1)c1ccc(cc1NC(=O)c1cc(N)c(F)c(C)c1Cl)-c1ccc(N)cc1	InChI=1S/C25H27ClFN5O/c1-15-23(26)19(14-20(29)24(15)27)25(33)30-21-13-17(16-3-6-18(28)7-4-16)5-8-22(21)32-11-9-31(2)10-12-32/h3-8,13-14H,9-12,28-29H2,1-2H3,(H,30,33)	HVMNEZGNJGWWQS-UHFFFAOYSA-N	50208372	CHEMBL3885241	WD repeat-containing protein 5				 202						ChEMBL	10.1016/j.ejmech.2016.08.036	10.7270/Q2251M6G	27598236			Li, DD; Chen, WL; Wang, ZH; Xie, YY; Xu, XL; Jiang, ZY; Zhang, XJ; You, QD; Guo, XK	China Pharmaceutical University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50208372	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50208372&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			134131003	375982020		CHEMBL3885241					1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50544322	CN1CCN(CC1)c1ccc(cc1NC(=O)c1cc(N)c(F)c(C)c1Cl)-c1ccc(NC(=O)CCCNC(=O)OC(C)(C)C)cc1	InChI=1S/C34H42ClFN6O4/c1-21-30(35)25(20-26(37)31(21)36)32(44)40-27-19-23(10-13-28(27)42-17-15-41(5)16-18-42)22-8-11-24(12-9-22)39-29(43)7-6-14-38-33(45)46-34(2,3)4/h8-13,19-20H,6-7,14-18,37H2,1-5H3,(H,38,45)(H,39,43)(H,40,44)	QLCFRZUEAHBEEG-UHFFFAOYSA-N	50208373	CHEMBL3884933	WD repeat-containing protein 5			 80							ChEMBL	10.1016/j.ejmech.2016.08.036	10.7270/Q2251M6G	27598236			Li, DD; Chen, WL; Wang, ZH; Xie, YY; Xu, XL; Jiang, ZY; Zhang, XJ; You, QD; Guo, XK	China Pharmaceutical University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50208373	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50208373&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			134131594	375982021		CHEMBL3884933					1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50544323	CN1CCN(CC1)c1ccc(cc1NC(=O)c1cc(N)c(F)c(C)c1Cl)-c1ccc(NC(=O)C(C)(C)NC(=O)OC(C)(C)C)cc1	InChI=1S/C34H42ClFN6O4/c1-20-28(35)24(19-25(37)29(20)36)30(43)39-26-18-22(10-13-27(26)42-16-14-41(7)15-17-42)21-8-11-23(12-9-21)38-31(44)34(5,6)40-32(45)46-33(2,3)4/h8-13,18-19H,14-17,37H2,1-7H3,(H,38,44)(H,39,43)(H,40,45)	YDKLHYJHKCPSJM-UHFFFAOYSA-N	50208374	CHEMBL3884185	WD repeat-containing protein 5			 113							ChEMBL	10.1016/j.ejmech.2016.08.036	10.7270/Q2251M6G	27598236			Li, DD; Chen, WL; Wang, ZH; Xie, YY; Xu, XL; Jiang, ZY; Zhang, XJ; You, QD; Guo, XK	China Pharmaceutical University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50208374	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50208374&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			134130560	375982022		CHEMBL3884185					1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50544324	CN1CCN(CC1)c1ccc(cc1NC(=O)c1cc(N)c(F)c(C)c1Cl)-c1ccc(NC(=O)CCNC(=O)OC(C)(C)C)cc1	InChI=1S/C33H40ClFN6O4/c1-20-29(34)24(19-25(36)30(20)35)31(43)39-26-18-22(8-11-27(26)41-16-14-40(5)15-17-41)21-6-9-23(10-7-21)38-28(42)12-13-37-32(44)45-33(2,3)4/h6-11,18-19H,12-17,36H2,1-5H3,(H,37,44)(H,38,42)(H,39,43)	MWPXTZNYBKJJLY-UHFFFAOYSA-N	50208375	CHEMBL3884091	WD repeat-containing protein 5			 102							ChEMBL	10.1016/j.ejmech.2016.08.036	10.7270/Q2251M6G	27598236			Li, DD; Chen, WL; Wang, ZH; Xie, YY; Xu, XL; Jiang, ZY; Zhang, XJ; You, QD; Guo, XK	China Pharmaceutical University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50208375	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50208375&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			134130017	375982023		CHEMBL3884091					1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50544325	CC(NC(=O)OC(C)(C)C)C(=O)Nc1ccc(cc1)-c1ccc(N2CCN(C)CC2)c(NC(=O)c2cc(N)c(F)c(C)c2Cl)c1	InChI=1S/C33H40ClFN6O4/c1-19-28(34)24(18-25(36)29(19)35)31(43)39-26-17-22(9-12-27(26)41-15-13-40(6)14-16-41)21-7-10-23(11-8-21)38-30(42)20(2)37-32(44)45-33(3,4)5/h7-12,17-18,20H,13-16,36H2,1-6H3,(H,37,44)(H,38,42)(H,39,43)	HXCUOKXDZNRSGW-UHFFFAOYSA-N	50208376	CHEMBL3883988	WD repeat-containing protein 5			 78							ChEMBL	10.1016/j.ejmech.2016.08.036	10.7270/Q2251M6G	27598236			Li, DD; Chen, WL; Wang, ZH; Xie, YY; Xu, XL; Jiang, ZY; Zhang, XJ; You, QD; Guo, XK	China Pharmaceutical University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50208376	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50208376&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			134131065	375982024		CHEMBL3883988					1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50544326	CN1CCN(CC1)c1ccc(cc1NC(=O)c1cc(N)c(F)c(C)c1Cl)-c1ccc(NC(=O)CNC(=O)OC(C)(C)C)cc1	InChI=1S/C32H38ClFN6O4/c1-19-28(33)23(17-24(35)29(19)34)30(42)38-25-16-21(8-11-26(25)40-14-12-39(5)13-15-40)20-6-9-22(10-7-20)37-27(41)18-36-31(43)44-32(2,3)4/h6-11,16-17H,12-15,18,35H2,1-5H3,(H,36,43)(H,37,41)(H,38,42)	KJMBWXSFSFEDPP-UHFFFAOYSA-N	50208377	CHEMBL3884567	WD repeat-containing protein 5			 1553							ChEMBL	10.1016/j.ejmech.2016.08.036	10.7270/Q2251M6G	27598236			Li, DD; Chen, WL; Wang, ZH; Xie, YY; Xu, XL; Jiang, ZY; Zhang, XJ; You, QD; Guo, XK	China Pharmaceutical University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50208377	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50208377&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			134130408	375982025		CHEMBL3884567					1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50544327	CCC(=O)Nc1ccc(cc1)-c1ccc(N2CCN(C)CC2)c(NC(=O)c2cc(N)c(F)c(C)c2Cl)c1	InChI=1S/C28H31ClFN5O2/c1-4-25(36)32-20-8-5-18(6-9-20)19-7-10-24(35-13-11-34(3)12-14-35)23(15-19)33-28(37)21-16-22(31)27(30)17(2)26(21)29/h5-10,15-16H,4,11-14,31H2,1-3H3,(H,32,36)(H,33,37)	AVJROSXSSUHEEH-UHFFFAOYSA-N	50208378	CHEMBL3884501	WD repeat-containing protein 5			 82							ChEMBL	10.1016/j.ejmech.2016.08.036	10.7270/Q2251M6G	27598236			Li, DD; Chen, WL; Wang, ZH; Xie, YY; Xu, XL; Jiang, ZY; Zhang, XJ; You, QD; Guo, XK	China Pharmaceutical University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50208378	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50208378&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			134129880	375982026		CHEMBL3884501					1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50544328	CN1CCN(CC1)c1ccc(cc1NC(=O)c1cc(N)c(F)c(C)c1Cl)-c1ccc(NC(C)=O)cc1	InChI=1S/C27H29ClFN5O2/c1-16-25(28)21(15-22(30)26(16)29)27(36)32-23-14-19(18-4-7-20(8-5-18)31-17(2)35)6-9-24(23)34-12-10-33(3)11-13-34/h4-9,14-15H,10-13,30H2,1-3H3,(H,31,35)(H,32,36)	LEEAQXLPUJRMOE-UHFFFAOYSA-N	50208379	CHEMBL3885048	WD repeat-containing protein 5			 70							ChEMBL	10.1016/j.ejmech.2016.08.036	10.7270/Q2251M6G	27598236			Li, DD; Chen, WL; Wang, ZH; Xie, YY; Xu, XL; Jiang, ZY; Zhang, XJ; You, QD; Guo, XK	China Pharmaceutical University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50208379	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50208379&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			134129955	375982027		CHEMBL3885048					1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50544329	CN1CCN(CC1)c1ccc(cc1NC(=O)c1ccc(F)c(N)c1)-c1ccncc1	InChI=1S/C23H24FN5O/c1-28-10-12-29(13-11-28)22-5-3-17(16-6-8-26-9-7-16)15-21(22)27-23(30)18-2-4-19(24)20(25)14-18/h2-9,14-15H,10-13,25H2,1H3,(H,27,30)	JDEUAGGKXMSXFO-UHFFFAOYSA-N	50208380	CHEMBL3884903	WD repeat-containing protein 5			 5800							ChEMBL	10.1016/j.ejmech.2016.08.036	10.7270/Q2251M6G	27598236			Li, DD; Chen, WL; Wang, ZH; Xie, YY; Xu, XL; Jiang, ZY; Zhang, XJ; You, QD; Guo, XK	China Pharmaceutical University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50208380	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50208380&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			134130074	375982028		CHEMBL3884903					1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50544330	CN1CCN(CC1)c1ccc(cc1NC(=O)c1ccc(F)c(N)c1)-c1ccc(N)cc1	InChI=1S/C24H26FN5O/c1-29-10-12-30(13-11-29)23-9-5-17(16-2-6-19(26)7-3-16)15-22(23)28-24(31)18-4-8-20(25)21(27)14-18/h2-9,14-15H,10-13,26-27H2,1H3,(H,28,31)	GZMWCHPEWVDBSX-UHFFFAOYSA-N	50208381	CHEMBL3884757	WD repeat-containing protein 5			 13600							ChEMBL	10.1016/j.ejmech.2016.08.036	10.7270/Q2251M6G	27598236			Li, DD; Chen, WL; Wang, ZH; Xie, YY; Xu, XL; Jiang, ZY; Zhang, XJ; You, QD; Guo, XK	China Pharmaceutical University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50208381	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50208381&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			134129903	375982029		CHEMBL3884757					1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50544331	CN1CCN(CC1)c1ccc(cc1NC(=O)c1cc(NC(C)=O)c(F)c(C)c1Cl)-c1ccncc1	InChI=1S/C26H27ClFN5O2/c1-16-24(27)20(15-22(25(16)28)30-17(2)34)26(35)31-21-14-19(18-6-8-29-9-7-18)4-5-23(21)33-12-10-32(3)11-13-33/h4-9,14-15H,10-13H2,1-3H3,(H,30,34)(H,31,35)	LIHRXRADZIXZEX-UHFFFAOYSA-N	50208382	CHEMBL3885262	WD repeat-containing protein 5			 1363							ChEMBL	10.1016/j.ejmech.2016.08.036	10.7270/Q2251M6G	27598236			Li, DD; Chen, WL; Wang, ZH; Xie, YY; Xu, XL; Jiang, ZY; Zhang, XJ; You, QD; Guo, XK	China Pharmaceutical University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50208382	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50208382&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			134130275	375982030		CHEMBL3885262					1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50544332	CN1CCN(CC1)c1ccc(cc1NC(=O)c1cc(NC(C)=O)c(F)c(C)c1Cl)-c1ccc(N)cc1	InChI=1S/C27H29ClFN5O2/c1-16-25(28)21(15-23(26(16)29)31-17(2)35)27(36)32-22-14-19(18-4-7-20(30)8-5-18)6-9-24(22)34-12-10-33(3)11-13-34/h4-9,14-15H,10-13,30H2,1-3H3,(H,31,35)(H,32,36)	FWPLARWSUMKWOX-UHFFFAOYSA-N	50208383	CHEMBL3884156	WD repeat-containing protein 5			 3186							ChEMBL	10.1016/j.ejmech.2016.08.036	10.7270/Q2251M6G	27598236			Li, DD; Chen, WL; Wang, ZH; Xie, YY; Xu, XL; Jiang, ZY; Zhang, XJ; You, QD; Guo, XK	China Pharmaceutical University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50208383	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50208383&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			134131117	375982031		CHEMBL3884156					1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50544333	COC(=O)c1ccc(cc1)-c1ccc(N2CCN(C)CC2)c(NC(=O)c2cc(N)c(F)c(C)c2Cl)c1	InChI=1S/C27H28ClFN4O3/c1-16-24(28)20(15-21(30)25(16)29)26(34)31-22-14-19(17-4-6-18(7-5-17)27(35)36-3)8-9-23(22)33-12-10-32(2)11-13-33/h4-9,14-15H,10-13,30H2,1-3H3,(H,31,34)	ADXWUOCLGQOCFF-UHFFFAOYSA-N	50208384	CHEMBL3884212	WD repeat-containing protein 5			 70							ChEMBL	10.1016/j.ejmech.2016.08.036	10.7270/Q2251M6G	27598236			Li, DD; Chen, WL; Wang, ZH; Xie, YY; Xu, XL; Jiang, ZY; Zhang, XJ; You, QD; Guo, XK	China Pharmaceutical University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50208384	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50208384&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			134131548	375982032		CHEMBL3884212					1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50544334	CN1CCN(CC1)c1ccc(cc1NC(=O)c1ccc(F)c(C)c1Cl)-c1ccc(N)cc1	InChI=1S/C25H26ClFN4O/c1-16-21(27)9-8-20(24(16)26)25(32)29-22-15-18(17-3-6-19(28)7-4-17)5-10-23(22)31-13-11-30(2)12-14-31/h3-10,15H,11-14,28H2,1-2H3,(H,29,32)	BTGNRDWCEWBDNG-UHFFFAOYSA-N	50184957	CHEMBL3822596	WD repeat-containing protein 5			 206							ChEMBL	10.1016/j.ejmech.2016.08.036	10.7270/Q2251M6G	27598236			Li, DD; Chen, WL; Wang, ZH; Xie, YY; Xu, XL; Jiang, ZY; Zhang, XJ; You, QD; Guo, XK	China Pharmaceutical University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50184957	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50184957&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			127049251	346550440		CHEMBL3822596					1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50544335	CN1CCN(CC1)c1ccc(cc1NC(=O)c1ccc(F)c(C)c1Cl)-c1ccncc1	InChI=1S/C24H24ClFN4O/c1-16-20(26)5-4-19(23(16)25)24(31)28-21-15-18(17-7-9-27-10-8-17)3-6-22(21)30-13-11-29(2)12-14-30/h3-10,15H,11-14H2,1-2H3,(H,28,31)	AICVIWJSFCXEOX-UHFFFAOYSA-N	50184787	CHEMBL3823308	WD repeat-containing protein 5			 104							ChEMBL	10.1016/j.ejmech.2016.08.036	10.7270/Q2251M6G	27598236			Li, DD; Chen, WL; Wang, ZH; Xie, YY; Xu, XL; Jiang, ZY; Zhang, XJ; You, QD; Guo, XK	China Pharmaceutical University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50184787	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50184787&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			127052837	104069106		CHEMBL3823308				ZINC40566038	1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50544336	COc1ccc(cc1)N1CCN(CC1)c1ccc(cc1NC(=O)c1ccc(F)c(C)c1Cl)[N+]([O-])=O	InChI=1S/C25H24ClFN4O4/c1-16-21(27)9-8-20(24(16)26)25(32)28-22-15-18(31(33)34)5-10-23(22)30-13-11-29(12-14-30)17-3-6-19(35-2)7-4-17/h3-10,15H,11-14H2,1-2H3,(H,28,32)	MWTFJVURBZQCAG-UHFFFAOYSA-N	50208385	CHEMBL3883800	WD repeat-containing protein 5			>20000							ChEMBL	10.1016/j.ejmech.2016.08.036	10.7270/Q2251M6G	27598236			Li, DD; Chen, WL; Wang, ZH; Xie, YY; Xu, XL; Jiang, ZY; Zhang, XJ; You, QD; Guo, XK	China Pharmaceutical University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50208385	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50208385&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			134130001	375982033		CHEMBL3883800					1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50544337	Cc1c(F)ccc(C(=O)Nc2cc(ccc2N2CCN(Cc3ccccc3)CC2)[N+]([O-])=O)c1Cl	InChI=1S/C25H24ClFN4O3/c1-17-21(27)9-8-20(24(17)26)25(32)28-22-15-19(31(33)34)7-10-23(22)30-13-11-29(12-14-30)16-18-5-3-2-4-6-18/h2-10,15H,11-14,16H2,1H3,(H,28,32)	MMLDLXUWPKPKHD-UHFFFAOYSA-N	50208386	CHEMBL3884930	WD repeat-containing protein 5			>20000							ChEMBL	10.1016/j.ejmech.2016.08.036	10.7270/Q2251M6G	27598236			Li, DD; Chen, WL; Wang, ZH; Xie, YY; Xu, XL; Jiang, ZY; Zhang, XJ; You, QD; Guo, XK	China Pharmaceutical University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50208386	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50208386&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			134131374	375982034		CHEMBL3884930					1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50544338	Cc1c(F)ccc(C(=O)Nc2cc(ccc2NCCN2CCCC2)[N+]([O-])=O)c1Cl	InChI=1S/C20H22ClFN4O3/c1-13-16(22)6-5-15(19(13)21)20(27)24-18-12-14(26(28)29)4-7-17(18)23-8-11-25-9-2-3-10-25/h4-7,12,23H,2-3,8-11H2,1H3,(H,24,27)	FEYNTWWQARYCSA-UHFFFAOYSA-N	50208387	CHEMBL3884724	WD repeat-containing protein 5			>20000							ChEMBL	10.1016/j.ejmech.2016.08.036	10.7270/Q2251M6G	27598236			Li, DD; Chen, WL; Wang, ZH; Xie, YY; Xu, XL; Jiang, ZY; Zhang, XJ; You, QD; Guo, XK	China Pharmaceutical University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50208387	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50208387&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			134130589	375982035		CHEMBL3884724					1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50544340	CN1CCN(CC1)c1ccc(cc1NC(=O)c1ccc(F)c(c1)[N+]([O-])=O)-c1ccc(cc1)[N+]([O-])=O	InChI=1S/C24H22FN5O5/c1-27-10-12-28(13-11-27)22-9-5-17(16-2-6-19(7-3-16)29(32)33)14-21(22)26-24(31)18-4-8-20(25)23(15-18)30(34)35/h2-9,14-15H,10-13H2,1H3,(H,26,31)	YEDLGSGWZKSCHJ-UHFFFAOYSA-N	50208388	CHEMBL3883948	WD repeat-containing protein 5			 1093							ChEMBL	10.1016/j.ejmech.2016.08.036	10.7270/Q2251M6G	27598236			Li, DD; Chen, WL; Wang, ZH; Xie, YY; Xu, XL; Jiang, ZY; Zhang, XJ; You, QD; Guo, XK	China Pharmaceutical University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50208388	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50208388&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			134131257	375982036		CHEMBL3883948					1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50544341	CN1CCN(CC1)c1ccc(cc1NC(=O)c1cc(N)c(F)c(C)c1Cl)-c1ccc(NC(=O)C(C)(C)N)cc1	InChI=1S/C29H34ClFN6O2/c1-17-25(30)21(16-22(32)26(17)31)27(38)35-23-15-19(7-10-24(23)37-13-11-36(4)12-14-37)18-5-8-20(9-6-18)34-28(39)29(2,3)33/h5-10,15-16H,11-14,32-33H2,1-4H3,(H,34,39)(H,35,38)	BILJOXOVCXLIKP-UHFFFAOYSA-N	50208389	CHEMBL3884527	WD repeat-containing protein 5			 30							ChEMBL	10.1016/j.ejmech.2016.08.036	10.7270/Q2251M6G	27598236			Li, DD; Chen, WL; Wang, ZH; Xie, YY; Xu, XL; Jiang, ZY; Zhang, XJ; You, QD; Guo, XK	China Pharmaceutical University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50208389	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50208389&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			134130407	375982037		CHEMBL3884527					1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50544342	CN1CCN(CC1)c1ccc(cc1NC(=O)c1cc(c(F)c(C)c1Cl)[N+]([O-])=O)-c1ccc(cc1)[N+]([O-])=O	InChI=1S/C25H23ClFN5O5/c1-15-23(26)19(14-22(24(15)27)32(36)37)25(33)28-20-13-17(16-3-6-18(7-4-16)31(34)35)5-8-21(20)30-11-9-29(2)10-12-30/h3-8,13-14H,9-12H2,1-2H3,(H,28,33)	RVHIQZXLOPWHQA-UHFFFAOYSA-N	50208390	CHEMBL3884058	WD repeat-containing protein 5			 285							ChEMBL	10.1016/j.ejmech.2016.08.036	10.7270/Q2251M6G	27598236			Li, DD; Chen, WL; Wang, ZH; Xie, YY; Xu, XL; Jiang, ZY; Zhang, XJ; You, QD; Guo, XK	China Pharmaceutical University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50208390	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50208390&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			134130734	375982038		CHEMBL3884058					1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50544343	CCC(CC)(NC(=O)C(C)C)C(=O)N[C@@H](CCCNC(N)=N)C(=O)NC1(CCCC1)C(=O)NC(c1ccc(F)cc1)c1ccc(F)cc1	InChI=1S/C35H49F2N7O4/c1-5-34(6-2,43-29(45)22(3)4)31(47)41-27(10-9-21-40-33(38)39)30(46)44-35(19-7-8-20-35)32(48)42-28(23-11-15-25(36)16-12-23)24-13-17-26(37)18-14-24/h11-18,22,27-28H,5-10,19-21H2,1-4H3,(H,41,47)(H,42,48)(H,43,45)(H,44,46)(H4,38,39,40)/t27-/m0/s1	RZKSQRIPRKWVBU-MHZLTWQESA-N	200723	US9233086, 10L	WD repeat-containing protein 5			 2.4							ChEMBL	10.1016/j.ejmech.2016.08.036	10.7270/Q2251M6G	27598236			Li, DD; Chen, WL; Wang, ZH; Xie, YY; Xu, XL; Jiang, ZY; Zhang, XJ; You, QD; Guo, XK	China Pharmaceutical University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=200723	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=200723&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			54766613	318834336							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50544345	CN1CCN(CC1)c1ccc(cc1NC(=O)c1cc(N)c(F)c(C)c1Cl)-c1ccc(NC(=O)C2CC2)cc1	InChI=1S/C29H31ClFN5O2/c1-17-26(30)22(16-23(32)27(17)31)29(38)34-24-15-20(7-10-25(24)36-13-11-35(2)12-14-36)18-5-8-21(9-6-18)33-28(37)19-3-4-19/h5-10,15-16,19H,3-4,11-14,32H2,1-2H3,(H,33,37)(H,34,38)	QLWDARVGOYOKOB-UHFFFAOYSA-N	50208391	CHEMBL3884230	WD repeat-containing protein 5			 76							ChEMBL	10.1016/j.ejmech.2016.08.036	10.7270/Q2251M6G	27598236			Li, DD; Chen, WL; Wang, ZH; Xie, YY; Xu, XL; Jiang, ZY; Zhang, XJ; You, QD; Guo, XK	China Pharmaceutical University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50208391	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50208391&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			134130925	375982039		CHEMBL3884230					1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50544346	CN1CCN(CC1)c1ccc(cc1NC(=O)c1cc(N)c(F)c(C)c1Cl)-c1ccc(NC(=O)C2CCNCC2)cc1	InChI=1S/C31H36ClFN6O2/c1-19-28(32)24(18-25(34)29(19)33)31(41)37-26-17-22(5-8-27(26)39-15-13-38(2)14-16-39)20-3-6-23(7-4-20)36-30(40)21-9-11-35-12-10-21/h3-8,17-18,21,35H,9-16,34H2,1-2H3,(H,36,40)(H,37,41)	CZWZZEUKNASAHM-UHFFFAOYSA-N	50208353	CHEMBL3884726	WD repeat-containing protein 5			 8.5							ChEMBL	10.1016/j.ejmech.2016.08.036	10.7270/Q2251M6G	27598236			Li, DD; Chen, WL; Wang, ZH; Xie, YY; Xu, XL; Jiang, ZY; Zhang, XJ; You, QD; Guo, XK	China Pharmaceutical University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50208353	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50208353&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			134130592	375982007		CHEMBL3884726					1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50544347	CN1CCN(CC1)c1ccc(cc1NC(=O)c1cc(N)c(F)c(C)c1Cl)-c1ccc(NC(=O)CCN)cc1	InChI=1S/C28H32ClFN6O2/c1-17-26(29)21(16-22(32)27(17)30)28(38)34-23-15-19(5-8-24(23)36-13-11-35(2)12-14-36)18-3-6-20(7-4-18)33-25(37)9-10-31/h3-8,15-16H,9-14,31-32H2,1-2H3,(H,33,37)(H,34,38)	ICSAHQQKONDURX-UHFFFAOYSA-N	50208392	CHEMBL3885308	WD repeat-containing protein 5			 50							ChEMBL	10.1016/j.ejmech.2016.08.036	10.7270/Q2251M6G	27598236			Li, DD; Chen, WL; Wang, ZH; Xie, YY; Xu, XL; Jiang, ZY; Zhang, XJ; You, QD; Guo, XK	China Pharmaceutical University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50208392	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50208392&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			134131026	375982040		CHEMBL3885308					1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50544348	CN1CCN(CC1)c1ccc(cc1NC(=O)c1cc(N)c(F)c(C)c1Cl)-c1ccc(NC(=O)CN)cc1	InChI=1S/C27H30ClFN6O2/c1-16-25(28)20(14-21(31)26(16)29)27(37)33-22-13-18(5-8-23(22)35-11-9-34(2)10-12-35)17-3-6-19(7-4-17)32-24(36)15-30/h3-8,13-14H,9-12,15,30-31H2,1-2H3,(H,32,36)(H,33,37)	ITXTXDPYKWZOMT-UHFFFAOYSA-N	50208393	CHEMBL3885025	WD repeat-containing protein 5			 63							ChEMBL	10.1016/j.ejmech.2016.08.036	10.7270/Q2251M6G	27598236			Li, DD; Chen, WL; Wang, ZH; Xie, YY; Xu, XL; Jiang, ZY; Zhang, XJ; You, QD; Guo, XK	China Pharmaceutical University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50208393	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50208393&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			134130500	375982041		CHEMBL3885025					1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50544349	CN1CCN(CC1)c1ccc(cc1NC(=O)c1cc(N)c(F)c(C)c1Cl)-c1ccc(NC(=O)C2CCCCC2)cc1	InChI=1S/C32H37ClFN5O2/c1-20-29(33)25(19-26(35)30(20)34)32(41)37-27-18-23(10-13-28(27)39-16-14-38(2)15-17-39)21-8-11-24(12-9-21)36-31(40)22-6-4-3-5-7-22/h8-13,18-19,22H,3-7,14-17,35H2,1-2H3,(H,36,40)(H,37,41)	WEIRPNVMAAQNJT-UHFFFAOYSA-N	50208394	CHEMBL3884705	WD repeat-containing protein 5			 341							ChEMBL	10.1016/j.ejmech.2016.08.036	10.7270/Q2251M6G	27598236			Li, DD; Chen, WL; Wang, ZH; Xie, YY; Xu, XL; Jiang, ZY; Zhang, XJ; You, QD; Guo, XK	China Pharmaceutical University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50208394	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50208394&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			134129898	375982042		CHEMBL3884705					1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50544350	CN1CCN(CC1)c1ccc(cc1NC(=O)c1cc(N)c(F)c(C)c1Cl)-c1ccc(N)cc1	InChI=1S/C25H27ClFN5O/c1-15-23(26)19(14-20(29)24(15)27)25(33)30-21-13-17(16-3-6-18(28)7-4-16)5-8-22(21)32-11-9-31(2)10-12-32/h3-8,13-14H,9-12,28-29H2,1-2H3,(H,30,33)	HVMNEZGNJGWWQS-UHFFFAOYSA-N	50208372	CHEMBL3885241	WD repeat-containing protein 5			 89							ChEMBL	10.1016/j.ejmech.2016.08.036	10.7270/Q2251M6G	27598236			Li, DD; Chen, WL; Wang, ZH; Xie, YY; Xu, XL; Jiang, ZY; Zhang, XJ; You, QD; Guo, XK	China Pharmaceutical University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50208372	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50208372&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			134131003	375982020		CHEMBL3885241					1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50544351	CN1CCN(CC1)c1ccc(cc1NC(=O)c1cc(N)c(F)c(C)c1Cl)-c1ccccc1	InChI=1S/C25H26ClFN4O/c1-16-23(26)19(15-20(28)24(16)27)25(32)29-21-14-18(17-6-4-3-5-7-17)8-9-22(21)31-12-10-30(2)11-13-31/h3-9,14-15H,10-13,28H2,1-2H3,(H,29,32)	DTVSOQNFDJEARZ-UHFFFAOYSA-N	50208395	CHEMBL3884136	WD repeat-containing protein 5			 48							ChEMBL	10.1016/j.ejmech.2016.08.036	10.7270/Q2251M6G	27598236			Li, DD; Chen, WL; Wang, ZH; Xie, YY; Xu, XL; Jiang, ZY; Zhang, XJ; You, QD; Guo, XK	China Pharmaceutical University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50208395	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50208395&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			134130195	375982043		CHEMBL3884136					1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50544352	CN1CCN(CC1)c1ccc(cc1NC(=O)c1cc(c(F)c(C)c1Cl)[N+]([O-])=O)-c1ccccc1	InChI=1S/C25H24ClFN4O3/c1-16-23(26)19(15-22(24(16)27)31(33)34)25(32)28-20-14-18(17-6-4-3-5-7-17)8-9-21(20)30-12-10-29(2)11-13-30/h3-9,14-15H,10-13H2,1-2H3,(H,28,32)	WOMZPTLUOWHXDN-UHFFFAOYSA-N	50184958	CHEMBL3823310	WD repeat-containing protein 5			 207							ChEMBL	10.1016/j.ejmech.2016.08.036	10.7270/Q2251M6G	27598236			Li, DD; Chen, WL; Wang, ZH; Xie, YY; Xu, XL; Jiang, ZY; Zhang, XJ; You, QD; Guo, XK	China Pharmaceutical University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50184958	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50184958&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			127049252	346550441		CHEMBL3823310					1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50544353	CCC(CC)(NC(=O)C(C)C)C(=O)N[C@@H](CCCNC(N)=N)C(=O)NC1(CCCC1)C(=O)NC(c1ccc(F)cc1)c1ccc(F)cc1	InChI=1S/C35H49F2N7O4/c1-5-34(6-2,43-29(45)22(3)4)31(47)41-27(10-9-21-40-33(38)39)30(46)44-35(19-7-8-20-35)32(48)42-28(23-11-15-25(36)16-12-23)24-13-17-26(37)18-14-24/h11-18,22,27-28H,5-10,19-21H2,1-4H3,(H,41,47)(H,42,48)(H,43,45)(H,44,46)(H4,38,39,40)/t27-/m0/s1	RZKSQRIPRKWVBU-MHZLTWQESA-N	200723	US9233086, 10L	WD repeat-containing protein 5			 1.7							ChEMBL	10.1016/j.ejmech.2016.08.036	10.7270/Q2251M6G	27598236			Li, DD; Chen, WL; Wang, ZH; Xie, YY; Xu, XL; Jiang, ZY; Zhang, XJ; You, QD; Guo, XK	China Pharmaceutical University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=200723	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=200723&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			54766613	318834336							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50544354	Cc1c(F)ccc(C(=O)Nc2cc(ccc2NCCCn2ccnc2)[N+]([O-])=O)c1Cl	InChI=1S/C20H19ClFN5O3/c1-13-16(22)5-4-15(19(13)21)20(28)25-18-11-14(27(29)30)3-6-17(18)24-7-2-9-26-10-8-23-12-26/h3-6,8,10-12,24H,2,7,9H2,1H3,(H,25,28)	XUDVUSWLCSLWNU-UHFFFAOYSA-N	50208396	CHEMBL3885484	WD repeat-containing protein 5			>20000							ChEMBL	10.1016/j.ejmech.2016.08.036	10.7270/Q2251M6G	27598236			Li, DD; Chen, WL; Wang, ZH; Xie, YY; Xu, XL; Jiang, ZY; Zhang, XJ; You, QD; Guo, XK	China Pharmaceutical University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50208396	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50208396&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			134131411	375982044		CHEMBL3885484					1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50544356	CC[C@@H]1NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@@](C)(CCCCNC(=O)[C@H](NC1=O)c1ccccc1)NC(=O)C(C)C	InChI=1S/C29H46N8O5/c1-5-20-24(39)36-22(19-12-7-6-8-13-19)26(41)32-16-10-9-15-29(4,37-23(38)18(2)3)27(42)35-21(25(40)34-20)14-11-17-33-28(30)31/h6-8,12-13,18,20-22H,5,9-11,14-17H2,1-4H3,(H,32,41)(H,34,40)(H,35,42)(H,36,39)(H,37,38)(H4,30,31,33)/t20-,21-,22+,29+/m0/s1	SILRGLDFBXVGOQ-ZMROOPMESA-N	50164787	CHEMBL3798088	WD repeat-containing protein 5			 0.900000							ChEMBL	10.1016/j.ejmech.2016.08.036	10.7270/Q2251M6G	27598236			Li, DD; Chen, WL; Wang, ZH; Xie, YY; Xu, XL; Jiang, ZY; Zhang, XJ; You, QD; Guo, XK	China Pharmaceutical University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50164787	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50164787&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			71586081	341097532		CHEMBL3798088					1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50544357	CC(C)CC(=O)Nc1ccc(cc1)-c1ccc(N2CCN(C)CC2)c(NC(=O)c2cc(N)c(F)c(C)c2Cl)c1	InChI=1S/C30H35ClFN5O2/c1-18(2)15-27(38)34-22-8-5-20(6-9-22)21-7-10-26(37-13-11-36(4)12-14-37)25(16-21)35-30(39)23-17-24(33)29(32)19(3)28(23)31/h5-10,16-18H,11-15,33H2,1-4H3,(H,34,38)(H,35,39)	QOLSGBASXRXNIO-UHFFFAOYSA-N	50208417	CHEMBL3885261	WD repeat-containing protein 5			 105							ChEMBL	10.1016/j.ejmech.2016.08.036	10.7270/Q2251M6G	27598236			Li, DD; Chen, WL; Wang, ZH; Xie, YY; Xu, XL; Jiang, ZY; Zhang, XJ; You, QD; Guo, XK	China Pharmaceutical University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50208417	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50208417&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			134130274	375982045		CHEMBL3885261					1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50544358	CN1CCN(CC1)c1ccc(cc1NC(=O)c1cccc(N)c1)-c1ccc(N)cc1	InChI=1S/C24H27N5O/c1-28-11-13-29(14-12-28)23-10-7-18(17-5-8-20(25)9-6-17)16-22(23)27-24(30)19-3-2-4-21(26)15-19/h2-10,15-16H,11-14,25-26H2,1H3,(H,27,30)	VPXJJUSYXGVJQW-UHFFFAOYSA-N	50208421	CHEMBL3884990	WD repeat-containing protein 5			>20000							ChEMBL	10.1016/j.ejmech.2016.08.036	10.7270/Q2251M6G	27598236			Li, DD; Chen, WL; Wang, ZH; Xie, YY; Xu, XL; Jiang, ZY; Zhang, XJ; You, QD; Guo, XK	China Pharmaceutical University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50208421	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50208421&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			134130118	375982046		CHEMBL3884990					1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
50544359	Cc1c(F)ccc(C(=O)Nc2cc(ccc2N2CCN(CC2)c2ccccn2)[N+]([O-])=O)c1Cl	InChI=1S/C23H21ClFN5O3/c1-15-18(25)7-6-17(22(15)24)23(31)27-19-14-16(30(32)33)5-8-20(19)28-10-12-29(13-11-28)21-4-2-3-9-26-21/h2-9,14H,10-13H2,1H3,(H,27,31)	UIGUIQVPCKAJLZ-UHFFFAOYSA-N	50208422	CHEMBL3884249	WD repeat-containing protein 5			>20000							ChEMBL	10.1016/j.ejmech.2016.08.036	10.7270/Q2251M6G	27598236			Li, DD; Chen, WL; Wang, ZH; Xie, YY; Xu, XL; Jiang, ZY; Zhang, XJ; You, QD; Guo, XK	China Pharmaceutical University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50208422	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50208422&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			134129874	375982047		CHEMBL3884249					1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51111909	CN1CCN(CC1)c1ccc(cc1NC(=O)c1ccccc1Cl)[N+]([O-])=O	InChI=1S/C18H19ClN4O3/c1-21-8-10-22(11-9-21)17-7-6-13(23(25)26)12-16(17)20-18(24)14-4-2-3-5-15(14)19/h2-7,12H,8-11H2,1H3,(H,20,24)	WOGZFCMBPXJNFI-UHFFFAOYSA-N	50428254	CHEMBL1609857	WD repeat-containing protein 5				 7000						ChEMBL	10.1016/j.bmc.2017.11.045	10.7270/Q2SQ92ZS	29254892			Wang, ZH; Li, DD; Chen, WL; You, QD; Guo, XK	China Pharmaceutical University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50428254	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50428254&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	NP7	3SMR	2965974	164157129		CHEMBL1609857				ZINC05049228	1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51135312	COc1cc(cc(OC)c1C)C(=O)N[C@@H]1CCc2ccc(cc12)-c1cn2CCCc2n1	InChI=1S/C25H27N3O3/c1-15-22(30-2)12-18(13-23(15)31-3)25(29)27-20-9-8-16-6-7-17(11-19(16)20)21-14-28-10-4-5-24(28)26-21/h6-7,11-14,20H,4-5,8-10H2,1-3H3,(H,27,29)/t20-/m1/s1	GRFBFSARRYJWSN-HXUWFJFHSA-N	50465552	CHEMBL4291641::US10501466, Example B29	WD repeat-containing protein 5		 0.902000								ChEMBL	10.1021/acs.jmedchem.8b00375	10.7270/Q2KD21KT	29889518			Wang, F; Jeon, KO; Salovich, JM; Macdonald, JD; Alvarado, J; Gogliotti, RD; Phan, J; Olejniczak, ET; Sun, Q; Wang, S; Camper, D; Yuh, JP; Shaw, JG; Sai, J; Rossanese, OW; Tansey, WP; Stauffer, SR; Fesik, SW	TBA	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50465552	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50465552&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138470423	433932817							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51135313	CC(=O)Nc1ccc(cc1)-c1cn2CCCc2n1	InChI=1S/C14H15N3O/c1-10(18)15-12-6-4-11(5-7-12)13-9-17-8-2-3-14(17)16-13/h4-7,9H,2-3,8H2,1H3,(H,15,18)	MQCINXVRFIDBMO-UHFFFAOYSA-N	50465553	CHEMBL4284833	WD repeat-containing protein 5		 118000								ChEMBL	10.1021/acs.jmedchem.8b00375	10.7270/Q2KD21KT	29889518			Wang, F; Jeon, KO; Salovich, JM; Macdonald, JD; Alvarado, J; Gogliotti, RD; Phan, J; Olejniczak, ET; Sun, Q; Wang, S; Camper, D; Yuh, JP; Shaw, JG; Sai, J; Rossanese, OW; Tansey, WP; Stauffer, SR; Fesik, SW	TBA	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50465553	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50465553&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			145992826	433932818							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51135314	COc1cccc(c1)C(=O)N(CC1CC1)Cc1cc(ccc1OC(C)C)-c1cn2CCCc2n1	InChI=1S/C28H33N3O3/c1-19(2)34-26-12-11-21(25-18-30-13-5-8-27(30)29-25)14-23(26)17-31(16-20-9-10-20)28(32)22-6-4-7-24(15-22)33-3/h4,6-7,11-12,14-15,18-20H,5,8-10,13,16-17H2,1-3H3	STTMASRUYCPJKT-UHFFFAOYSA-N	50465554	CHEMBL4286527	WD repeat-containing protein 5		 28								ChEMBL	10.1021/acs.jmedchem.8b00375	10.7270/Q2KD21KT	29889518			Wang, F; Jeon, KO; Salovich, JM; Macdonald, JD; Alvarado, J; Gogliotti, RD; Phan, J; Olejniczak, ET; Sun, Q; Wang, S; Camper, D; Yuh, JP; Shaw, JG; Sai, J; Rossanese, OW; Tansey, WP; Stauffer, SR; Fesik, SW	TBA	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50465554	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50465554&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			134369637	433932819							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51135315	COc1cc(CC(=O)N[C@@H]2CCc3ccc(cc23)-c2cn3CCCc3n2)ccc1C	InChI=1S/C25H27N3O2/c1-16-5-6-17(12-23(16)30-2)13-25(29)27-21-10-9-18-7-8-19(14-20(18)21)22-15-28-11-3-4-24(28)26-22/h5-8,12,14-15,21H,3-4,9-11,13H2,1-2H3,(H,27,29)/t21-/m1/s1	WHKWYCMXCHKNSQ-OAQYLSRUSA-N	50465555	CHEMBL4287817	WD repeat-containing protein 5		 4.9								ChEMBL	10.1021/acs.jmedchem.8b00375	10.7270/Q2KD21KT	29889518			Wang, F; Jeon, KO; Salovich, JM; Macdonald, JD; Alvarado, J; Gogliotti, RD; Phan, J; Olejniczak, ET; Sun, Q; Wang, S; Camper, D; Yuh, JP; Shaw, JG; Sai, J; Rossanese, OW; Tansey, WP; Stauffer, SR; Fesik, SW	TBA	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50465555	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50465555&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			145993387	433932820							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51135316	Cc1cncc(c1)C(=O)NCc1cccc(c1)-c1cn2CCCc2n1	InChI=1S/C20H20N4O/c1-14-8-17(12-21-10-14)20(25)22-11-15-4-2-5-16(9-15)18-13-24-7-3-6-19(24)23-18/h2,4-5,8-10,12-13H,3,6-7,11H2,1H3,(H,22,25)	VDHLGRKJCUPRLS-UHFFFAOYSA-N	50465556	CHEMBL4283572	WD repeat-containing protein 5		 924								ChEMBL	10.1021/acs.jmedchem.8b00375	10.7270/Q2KD21KT	29889518			Wang, F; Jeon, KO; Salovich, JM; Macdonald, JD; Alvarado, J; Gogliotti, RD; Phan, J; Olejniczak, ET; Sun, Q; Wang, S; Camper, D; Yuh, JP; Shaw, JG; Sai, J; Rossanese, OW; Tansey, WP; Stauffer, SR; Fesik, SW	TBA	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50465556	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50465556&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			134369681	433932821							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51135317	Cc1cccc(c1)C(=O)NCc1cccc(c1)-c1cn2CCCc2n1	InChI=1S/C21H21N3O/c1-15-5-2-8-18(11-15)21(25)22-13-16-6-3-7-17(12-16)19-14-24-10-4-9-20(24)23-19/h2-3,5-8,11-12,14H,4,9-10,13H2,1H3,(H,22,25)	XDICNJLKVAZJMN-UHFFFAOYSA-N	50465557	CHEMBL4281521	WD repeat-containing protein 5		 2600								ChEMBL	10.1021/acs.jmedchem.8b00375	10.7270/Q2KD21KT	29889518			Wang, F; Jeon, KO; Salovich, JM; Macdonald, JD; Alvarado, J; Gogliotti, RD; Phan, J; Olejniczak, ET; Sun, Q; Wang, S; Camper, D; Yuh, JP; Shaw, JG; Sai, J; Rossanese, OW; Tansey, WP; Stauffer, SR; Fesik, SW	TBA	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50465557	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50465557&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			134369557	433932822							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51135318	O=C(NCc1cccc(c1)-c1cn2CCCc2n1)c1ccncc1	InChI=1S/C19H18N4O/c24-19(15-6-8-20-9-7-15)21-12-14-3-1-4-16(11-14)17-13-23-10-2-5-18(23)22-17/h1,3-4,6-9,11,13H,2,5,10,12H2,(H,21,24)	JTCBCDHSPFWEGS-UHFFFAOYSA-N	50465558	CHEMBL4287245	WD repeat-containing protein 5		 1380								ChEMBL	10.1021/acs.jmedchem.8b00375	10.7270/Q2KD21KT	29889518			Wang, F; Jeon, KO; Salovich, JM; Macdonald, JD; Alvarado, J; Gogliotti, RD; Phan, J; Olejniczak, ET; Sun, Q; Wang, S; Camper, D; Yuh, JP; Shaw, JG; Sai, J; Rossanese, OW; Tansey, WP; Stauffer, SR; Fesik, SW	TBA	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50465558	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50465558&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			134369576	433932823							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51135319	COc1cccc(c1)C(=O)NCc1cc(ccc1OC(C)C)-c1cn2CCCc2n1	InChI=1S/C24H27N3O3/c1-16(2)30-22-10-9-17(21-15-27-11-5-8-23(27)26-21)12-19(22)14-25-24(28)18-6-4-7-20(13-18)29-3/h4,6-7,9-10,12-13,15-16H,5,8,11,14H2,1-3H3,(H,25,28)	DXZYVORRTZPJAD-UHFFFAOYSA-N	50465559	CHEMBL4285902	WD repeat-containing protein 5		 76								ChEMBL	10.1021/acs.jmedchem.8b00375	10.7270/Q2KD21KT	29889518			Wang, F; Jeon, KO; Salovich, JM; Macdonald, JD; Alvarado, J; Gogliotti, RD; Phan, J; Olejniczak, ET; Sun, Q; Wang, S; Camper, D; Yuh, JP; Shaw, JG; Sai, J; Rossanese, OW; Tansey, WP; Stauffer, SR; Fesik, SW	TBA	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50465559	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50465559&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			134369653	433932824							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51135320	C1Cc2nc(cn2C1)-c1ccccc1	InChI=1S/C12H12N2/c1-2-5-10(6-3-1)11-9-14-8-4-7-12(14)13-11/h1-3,5-6,9H,4,7-8H2	PPYLPCSLYXBQRM-UHFFFAOYSA-N	50465560	CHEMBL1380070	WD repeat-containing protein 5		 323000								ChEMBL	10.1021/acs.jmedchem.8b00375	10.7270/Q2KD21KT	29889518			Wang, F; Jeon, KO; Salovich, JM; Macdonald, JD; Alvarado, J; Gogliotti, RD; Phan, J; Olejniczak, ET; Sun, Q; Wang, S; Camper, D; Yuh, JP; Shaw, JG; Sai, J; Rossanese, OW; Tansey, WP; Stauffer, SR; Fesik, SW	TBA	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50465560	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50465560&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	FZM	6D9X	765511	433932825							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51135321	Cc1ccc(OCC(N)=N)cc1	InChI=1S/C9H12N2O/c1-7-2-4-8(5-3-7)12-6-9(10)11/h2-5H,6H2,1H3,(H3,10,11)	GNNCNKKBHNXZED-UHFFFAOYSA-N	50465561	CHEMBL4282498	WD repeat-containing protein 5		 589000								ChEMBL	10.1021/acs.jmedchem.8b00375	10.7270/Q2KD21KT	29889518			Wang, F; Jeon, KO; Salovich, JM; Macdonald, JD; Alvarado, J; Gogliotti, RD; Phan, J; Olejniczak, ET; Sun, Q; Wang, S; Camper, D; Yuh, JP; Shaw, JG; Sai, J; Rossanese, OW; Tansey, WP; Stauffer, SR; Fesik, SW	TBA	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50465561	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50465561&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			13430822	433932826							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51135322	Oc1ccc(cc1)-c1cn2CCSc2n1	InChI=1S/C11H10N2OS/c14-9-3-1-8(2-4-9)10-7-13-5-6-15-11(13)12-10/h1-4,7,14H,5-6H2	ZAKNXVYBQHMJDW-UHFFFAOYSA-N	50465562	CHEMBL1502560	WD repeat-containing protein 5		>1000000								ChEMBL	10.1021/acs.jmedchem.8b00375	10.7270/Q2KD21KT	29889518			Wang, F; Jeon, KO; Salovich, JM; Macdonald, JD; Alvarado, J; Gogliotti, RD; Phan, J; Olejniczak, ET; Sun, Q; Wang, S; Camper, D; Yuh, JP; Shaw, JG; Sai, J; Rossanese, OW; Tansey, WP; Stauffer, SR; Fesik, SW	TBA	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50465562	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50465562&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			700755	433932827							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51135323	CCOc1ccc(cc1)-c1cn2ccccc2n1	InChI=1S/C15H14N2O/c1-2-18-13-8-6-12(7-9-13)14-11-17-10-4-3-5-15(17)16-14/h3-11H,2H2,1H3	BWAXYFPYNGSSKF-UHFFFAOYSA-N	50465563	CHEMBL1602085	WD repeat-containing protein 5		>1000000								ChEMBL	10.1021/acs.jmedchem.8b00375	10.7270/Q2KD21KT	29889518			Wang, F; Jeon, KO; Salovich, JM; Macdonald, JD; Alvarado, J; Gogliotti, RD; Phan, J; Olejniczak, ET; Sun, Q; Wang, S; Camper, D; Yuh, JP; Shaw, JG; Sai, J; Rossanese, OW; Tansey, WP; Stauffer, SR; Fesik, SW	TBA	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50465563	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50465563&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			720519	433932828							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51135324	C1Cc2nc(cn2C1)-c1ccc(cc1)-c1ccccc1	InChI=1S/C18H16N2/c1-2-5-14(6-3-1)15-8-10-16(11-9-15)17-13-20-12-4-7-18(20)19-17/h1-3,5-6,8-11,13H,4,7,12H2	IMYNUXAXHXLXJE-UHFFFAOYSA-N	49419	2-(4-phenylphenyl)-6,7-dihydro-5H-pyrrol[1,2-a]imidazole;hydrobromide::2-(4-phenylphenyl)-6,7-dihydro-5H-pyrrolo[1,2-a]imidazole;hydrobromide::2-Biphenyl-4-yl-6,7-dihydro-5H-pyrrolo[1,2-a]imidazole::MLS000552669::SMR000146184::cid_9550136	WD repeat-containing protein 5		 8440								ChEMBL	10.1021/acs.jmedchem.8b00375	10.7270/Q2KD21KT	29889518			Wang, F; Jeon, KO; Salovich, JM; Macdonald, JD; Alvarado, J; Gogliotti, RD; Phan, J; Olejniczak, ET; Sun, Q; Wang, S; Camper, D; Yuh, JP; Shaw, JG; Sai, J; Rossanese, OW; Tansey, WP; Stauffer, SR; Fesik, SW	TBA	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=49419	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=49419&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			3697667	252629698						ZINC06110614	1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51135325	C(Oc1ccc(cc1)-c1cn2CCCc2n1)c1ccccc1	InChI=1S/C19H18N2O/c1-2-5-15(6-3-1)14-22-17-10-8-16(9-11-17)18-13-21-12-4-7-19(21)20-18/h1-3,5-6,8-11,13H,4,7,12,14H2	HRBBIEXCIXPOSD-UHFFFAOYSA-N	50465564	CHEMBL4284526	WD repeat-containing protein 5		 64300								ChEMBL	10.1021/acs.jmedchem.8b00375	10.7270/Q2KD21KT	29889518			Wang, F; Jeon, KO; Salovich, JM; Macdonald, JD; Alvarado, J; Gogliotti, RD; Phan, J; Olejniczak, ET; Sun, Q; Wang, S; Camper, D; Yuh, JP; Shaw, JG; Sai, J; Rossanese, OW; Tansey, WP; Stauffer, SR; Fesik, SW	TBA	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50465564	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50465564&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			145991249	433932829							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51135326	Fc1cccc(c1F)-c1ccc(cc1)-c1cn2CCCc2n1	InChI=1S/C18H14F2N2/c19-15-4-1-3-14(18(15)20)12-6-8-13(9-7-12)16-11-22-10-2-5-17(22)21-16/h1,3-4,6-9,11H,2,5,10H2	QZUPTAQWXCJUMM-UHFFFAOYSA-N	50465565	CHEMBL4292418	WD repeat-containing protein 5		 1120								ChEMBL	10.1021/acs.jmedchem.8b00375	10.7270/Q2KD21KT	29889518			Wang, F; Jeon, KO; Salovich, JM; Macdonald, JD; Alvarado, J; Gogliotti, RD; Phan, J; Olejniczak, ET; Sun, Q; Wang, S; Camper, D; Yuh, JP; Shaw, JG; Sai, J; Rossanese, OW; Tansey, WP; Stauffer, SR; Fesik, SW	TBA	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50465565	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50465565&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			145988536	433932830							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51135327	C1Cc2nc(cn2C1)-c1ccc2OCOc2c1	InChI=1S/C13H12N2O2/c1-2-13-14-10(7-15(13)5-1)9-3-4-11-12(6-9)17-8-16-11/h3-4,6-7H,1-2,5,8H2	DVDJUGXQHFTHNO-UHFFFAOYSA-N	50465566	CHEMBL4289013	WD repeat-containing protein 5		 64000								ChEMBL	10.1021/acs.jmedchem.8b00375	10.7270/Q2KD21KT	29889518			Wang, F; Jeon, KO; Salovich, JM; Macdonald, JD; Alvarado, J; Gogliotti, RD; Phan, J; Olejniczak, ET; Sun, Q; Wang, S; Camper, D; Yuh, JP; Shaw, JG; Sai, J; Rossanese, OW; Tansey, WP; Stauffer, SR; Fesik, SW	TBA	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50465566	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50465566&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			145989019	433932831							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51135328	COc1cccc(c1)-c1cn2CCCc2n1	InChI=1S/C13H14N2O/c1-16-11-5-2-4-10(8-11)12-9-15-7-3-6-13(15)14-12/h2,4-5,8-9H,3,6-7H2,1H3	PQMZLEHESQYFPF-UHFFFAOYSA-N	50465567	CHEMBL4291321	WD repeat-containing protein 5		 117000								ChEMBL	10.1021/acs.jmedchem.8b00375	10.7270/Q2KD21KT	29889518			Wang, F; Jeon, KO; Salovich, JM; Macdonald, JD; Alvarado, J; Gogliotti, RD; Phan, J; Olejniczak, ET; Sun, Q; Wang, S; Camper, D; Yuh, JP; Shaw, JG; Sai, J; Rossanese, OW; Tansey, WP; Stauffer, SR; Fesik, SW	TBA	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50465567	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50465567&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			145989142	433932832							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51135329	CC(=O)Nc1cccc(c1)-c1cn2CCCc2n1	InChI=1S/C14H15N3O/c1-10(18)15-12-5-2-4-11(8-12)13-9-17-7-3-6-14(17)16-13/h2,4-5,8-9H,3,6-7H2,1H3,(H,15,18)	ARTHFRPUYUQHNY-UHFFFAOYSA-N	50465568	CHEMBL4287916	WD repeat-containing protein 5		>125000								ChEMBL	10.1021/acs.jmedchem.8b00375	10.7270/Q2KD21KT	29889518			Wang, F; Jeon, KO; Salovich, JM; Macdonald, JD; Alvarado, J; Gogliotti, RD; Phan, J; Olejniczak, ET; Sun, Q; Wang, S; Camper, D; Yuh, JP; Shaw, JG; Sai, J; Rossanese, OW; Tansey, WP; Stauffer, SR; Fesik, SW	TBA	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50465568	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50465568&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			145990286	433932833							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51135330	COc1cccc(c1)C(=O)NCc1cccc(c1)-c1cn2CCCc2n1	InChI=1S/C21H21N3O2/c1-26-18-8-3-7-17(12-18)21(25)22-13-15-5-2-6-16(11-15)19-14-24-10-4-9-20(24)23-19/h2-3,5-8,11-12,14H,4,9-10,13H2,1H3,(H,22,25)	KWPMSLGCMXLIRE-UHFFFAOYSA-N	50465569	CHEMBL4278737	WD repeat-containing protein 5		 665								ChEMBL	10.1021/acs.jmedchem.8b00375	10.7270/Q2KD21KT	29889518			Wang, F; Jeon, KO; Salovich, JM; Macdonald, JD; Alvarado, J; Gogliotti, RD; Phan, J; Olejniczak, ET; Sun, Q; Wang, S; Camper, D; Yuh, JP; Shaw, JG; Sai, J; Rossanese, OW; Tansey, WP; Stauffer, SR; Fesik, SW	TBA	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50465569	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50465569&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			134369556	433932834							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51135331	COc1ccc(cc1)C(=O)NCc1cccc(c1)-c1cn2CCCc2n1	InChI=1S/C21H21N3O2/c1-26-18-9-7-16(8-10-18)21(25)22-13-15-4-2-5-17(12-15)19-14-24-11-3-6-20(24)23-19/h2,4-5,7-10,12,14H,3,6,11,13H2,1H3,(H,22,25)	WOHXAOWQRBNCMD-UHFFFAOYSA-N	50465570	CHEMBL4292147	WD repeat-containing protein 5		 3130								ChEMBL	10.1021/acs.jmedchem.8b00375	10.7270/Q2KD21KT	29889518			Wang, F; Jeon, KO; Salovich, JM; Macdonald, JD; Alvarado, J; Gogliotti, RD; Phan, J; Olejniczak, ET; Sun, Q; Wang, S; Camper, D; Yuh, JP; Shaw, JG; Sai, J; Rossanese, OW; Tansey, WP; Stauffer, SR; Fesik, SW	TBA	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50465570	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50465570&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			134369561	433932835							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51135332	O=C(Cc1ccccc1)NCc1cccc(c1)-c1cn2CCCc2n1	InChI=1S/C21H21N3O/c25-21(13-16-6-2-1-3-7-16)22-14-17-8-4-9-18(12-17)19-15-24-11-5-10-20(24)23-19/h1-4,6-9,12,15H,5,10-11,13-14H2,(H,22,25)	GKIAAVNOBCFHHP-UHFFFAOYSA-N	50465571	CHEMBL4278066	WD repeat-containing protein 5		 17600								ChEMBL	10.1021/acs.jmedchem.8b00375	10.7270/Q2KD21KT	29889518			Wang, F; Jeon, KO; Salovich, JM; Macdonald, JD; Alvarado, J; Gogliotti, RD; Phan, J; Olejniczak, ET; Sun, Q; Wang, S; Camper, D; Yuh, JP; Shaw, JG; Sai, J; Rossanese, OW; Tansey, WP; Stauffer, SR; Fesik, SW	TBA	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50465571	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50465571&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			134369558	433932836							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51135333	COc1cc(C)cc(c1)C(=O)NCc1cccc(c1)-c1cn2CCCc2n1	InChI=1S/C22H23N3O2/c1-15-9-18(12-19(10-15)27-2)22(26)23-13-16-5-3-6-17(11-16)20-14-25-8-4-7-21(25)24-20/h3,5-6,9-12,14H,4,7-8,13H2,1-2H3,(H,23,26)	BOBQZWKOBBWGCV-UHFFFAOYSA-N	50465572	CHEMBL4284948	WD repeat-containing protein 5		 184								ChEMBL	10.1021/acs.jmedchem.8b00375	10.7270/Q2KD21KT	29889518			Wang, F; Jeon, KO; Salovich, JM; Macdonald, JD; Alvarado, J; Gogliotti, RD; Phan, J; Olejniczak, ET; Sun, Q; Wang, S; Camper, D; Yuh, JP; Shaw, JG; Sai, J; Rossanese, OW; Tansey, WP; Stauffer, SR; Fesik, SW	TBA	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50465572	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50465572&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			134369668	433932837							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51135334	O=C(NCc1cccc(c1)-c1cn2CCCc2n1)c1ccccn1	InChI=1S/C19H18N4O/c24-19(16-7-1-2-9-20-16)21-12-14-5-3-6-15(11-14)17-13-23-10-4-8-18(23)22-17/h1-3,5-7,9,11,13H,4,8,10,12H2,(H,21,24)	QBKBBNQVYLLISY-UHFFFAOYSA-N	50465573	CHEMBL4276998	WD repeat-containing protein 5		 3910								ChEMBL	10.1021/acs.jmedchem.8b00375	10.7270/Q2KD21KT	29889518			Wang, F; Jeon, KO; Salovich, JM; Macdonald, JD; Alvarado, J; Gogliotti, RD; Phan, J; Olejniczak, ET; Sun, Q; Wang, S; Camper, D; Yuh, JP; Shaw, JG; Sai, J; Rossanese, OW; Tansey, WP; Stauffer, SR; Fesik, SW	TBA	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50465573	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50465573&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			134369563	433932838							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51135335	COc1cccc(c1)C(=O)N(C)Cc1cccc(c1)-c1cn2CCCc2n1	InChI=1S/C22H23N3O2/c1-24(22(26)18-8-4-9-19(13-18)27-2)14-16-6-3-7-17(12-16)20-15-25-11-5-10-21(25)23-20/h3-4,6-9,12-13,15H,5,10-11,14H2,1-2H3	HDBYUCSDPPUAQR-UHFFFAOYSA-N	50465574	CHEMBL4291414	WD repeat-containing protein 5		 473								ChEMBL	10.1021/acs.jmedchem.8b00375	10.7270/Q2KD21KT	29889518			Wang, F; Jeon, KO; Salovich, JM; Macdonald, JD; Alvarado, J; Gogliotti, RD; Phan, J; Olejniczak, ET; Sun, Q; Wang, S; Camper, D; Yuh, JP; Shaw, JG; Sai, J; Rossanese, OW; Tansey, WP; Stauffer, SR; Fesik, SW	TBA	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50465574	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50465574&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			134369647	433932839							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51135336	COc1cccc(c1)C(=O)N(Cc1cccc(c1)-c1cn2CCCc2n1)C(C)C	InChI=1S/C24H27N3O2/c1-17(2)27(24(28)20-9-5-10-21(14-20)29-3)15-18-7-4-8-19(13-18)22-16-26-12-6-11-23(26)25-22/h4-5,7-10,13-14,16-17H,6,11-12,15H2,1-3H3	OBJNBTSQQVOQHS-UHFFFAOYSA-N	50465575	CHEMBL4286932	WD repeat-containing protein 5		 503								ChEMBL	10.1021/acs.jmedchem.8b00375	10.7270/Q2KD21KT	29889518			Wang, F; Jeon, KO; Salovich, JM; Macdonald, JD; Alvarado, J; Gogliotti, RD; Phan, J; Olejniczak, ET; Sun, Q; Wang, S; Camper, D; Yuh, JP; Shaw, JG; Sai, J; Rossanese, OW; Tansey, WP; Stauffer, SR; Fesik, SW	TBA	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50465575	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50465575&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			134369560	433932840							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51135337	COc1cccc(c1)C(=O)N(CC1CCC1)Cc1cccc(c1)-c1cn2CCCc2n1	InChI=1S/C26H29N3O2/c1-31-23-11-4-10-22(15-23)26(30)29(16-19-6-2-7-19)17-20-8-3-9-21(14-20)24-18-28-13-5-12-25(28)27-24/h3-4,8-11,14-15,18-19H,2,5-7,12-13,16-17H2,1H3	FAWBSWIPJHTAOZ-UHFFFAOYSA-N	50465576	CHEMBL4276691	WD repeat-containing protein 5		 1260								ChEMBL	10.1021/acs.jmedchem.8b00375	10.7270/Q2KD21KT	29889518			Wang, F; Jeon, KO; Salovich, JM; Macdonald, JD; Alvarado, J; Gogliotti, RD; Phan, J; Olejniczak, ET; Sun, Q; Wang, S; Camper, D; Yuh, JP; Shaw, JG; Sai, J; Rossanese, OW; Tansey, WP; Stauffer, SR; Fesik, SW	TBA	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50465576	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50465576&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			134369583	433932841							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51135338	COc1cccc(c1)C(=O)N(CC1CC1)Cc1cc(OC)cc(c1)-c1cn2CCCc2n1	InChI=1S/C26H29N3O3/c1-31-22-6-3-5-20(13-22)26(30)29(15-18-8-9-18)16-19-11-21(14-23(12-19)32-2)24-17-28-10-4-7-25(28)27-24/h3,5-6,11-14,17-18H,4,7-10,15-16H2,1-2H3	AJNBKDGZXWYQNH-UHFFFAOYSA-N	50465577	CHEMBL4280115	WD repeat-containing protein 5		 1460								ChEMBL	10.1021/acs.jmedchem.8b00375	10.7270/Q2KD21KT	29889518			Wang, F; Jeon, KO; Salovich, JM; Macdonald, JD; Alvarado, J; Gogliotti, RD; Phan, J; Olejniczak, ET; Sun, Q; Wang, S; Camper, D; Yuh, JP; Shaw, JG; Sai, J; Rossanese, OW; Tansey, WP; Stauffer, SR; Fesik, SW	TBA	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50465577	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50465577&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			134369619	433932842							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51135339	COc1cccc(c1)C(=O)N(CC1CC1)Cc1cc(ccc1OC)-c1cn2CCCc2n1	InChI=1S/C26H29N3O3/c1-31-22-6-3-5-20(14-22)26(30)29(15-18-8-9-18)16-21-13-19(10-11-24(21)32-2)23-17-28-12-4-7-25(28)27-23/h3,5-6,10-11,13-14,17-18H,4,7-9,12,15-16H2,1-2H3	YLEJBBJFQLXMGW-UHFFFAOYSA-N	50465578	CHEMBL4288010	WD repeat-containing protein 5		 148								ChEMBL	10.1021/acs.jmedchem.8b00375	10.7270/Q2KD21KT	29889518			Wang, F; Jeon, KO; Salovich, JM; Macdonald, JD; Alvarado, J; Gogliotti, RD; Phan, J; Olejniczak, ET; Sun, Q; Wang, S; Camper, D; Yuh, JP; Shaw, JG; Sai, J; Rossanese, OW; Tansey, WP; Stauffer, SR; Fesik, SW	TBA	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50465578	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50465578&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			134369620	433932843							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51135340	COc1cccc(c1)C(=O)N(CC1CC1)Cc1cc(ccc1OC1CCC1)-c1cn2CCCc2n1	InChI=1S/C29H33N3O3/c1-34-25-8-2-5-22(16-25)29(33)32(17-20-10-11-20)18-23-15-21(12-13-27(23)35-24-6-3-7-24)26-19-31-14-4-9-28(31)30-26/h2,5,8,12-13,15-16,19-20,24H,3-4,6-7,9-11,14,17-18H2,1H3	IDRQLZRSEYEXMR-UHFFFAOYSA-N	50465579	CHEMBL4294133	WD repeat-containing protein 5		 23								ChEMBL	10.1021/acs.jmedchem.8b00375	10.7270/Q2KD21KT	29889518			Wang, F; Jeon, KO; Salovich, JM; Macdonald, JD; Alvarado, J; Gogliotti, RD; Phan, J; Olejniczak, ET; Sun, Q; Wang, S; Camper, D; Yuh, JP; Shaw, JG; Sai, J; Rossanese, OW; Tansey, WP; Stauffer, SR; Fesik, SW	TBA	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50465579	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50465579&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			134369650	433932844							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51135341	COc1cccc(c1)C(=O)NCc1cc(ccc1N(C)C)-c1cn2CCCc2n1	InChI=1S/C23H26N4O2/c1-26(2)21-10-9-16(20-15-27-11-5-8-22(27)25-20)12-18(21)14-24-23(28)17-6-4-7-19(13-17)29-3/h4,6-7,9-10,12-13,15H,5,8,11,14H2,1-3H3,(H,24,28)	NYCQMHOKYBUOQV-UHFFFAOYSA-N	50465580	CHEMBL4276791	WD repeat-containing protein 5		 185								ChEMBL	10.1021/acs.jmedchem.8b00375	10.7270/Q2KD21KT	29889518			Wang, F; Jeon, KO; Salovich, JM; Macdonald, JD; Alvarado, J; Gogliotti, RD; Phan, J; Olejniczak, ET; Sun, Q; Wang, S; Camper, D; Yuh, JP; Shaw, JG; Sai, J; Rossanese, OW; Tansey, WP; Stauffer, SR; Fesik, SW	TBA	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50465580	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50465580&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			134369666	433932845							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51135342	CN(C)c1ccc(cc1CNC(=O)Cc1ccc(Cl)c(Cl)c1)-c1cn2CCCc2n1	InChI=1S/C23H24Cl2N4O/c1-28(2)21-8-6-16(20-14-29-9-3-4-22(29)27-20)12-17(21)13-26-23(30)11-15-5-7-18(24)19(25)10-15/h5-8,10,12,14H,3-4,9,11,13H2,1-2H3,(H,26,30)	KMARVDJMQLSDNW-UHFFFAOYSA-N	50465581	CHEMBL4292999	WD repeat-containing protein 5		 52								ChEMBL	10.1021/acs.jmedchem.8b00375	10.7270/Q2KD21KT	29889518			Wang, F; Jeon, KO; Salovich, JM; Macdonald, JD; Alvarado, J; Gogliotti, RD; Phan, J; Olejniczak, ET; Sun, Q; Wang, S; Camper, D; Yuh, JP; Shaw, JG; Sai, J; Rossanese, OW; Tansey, WP; Stauffer, SR; Fesik, SW	TBA	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50465581	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50465581&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			134369670	433932846							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51135343	CC(C)Oc1ccc(cc1CNC(=O)Cc1ccc(Cl)c(Cl)c1)-c1cn2CCCc2n1	InChI=1S/C24H25Cl2N3O2/c1-15(2)31-22-8-6-17(21-14-29-9-3-4-23(29)28-21)12-18(22)13-27-24(30)11-16-5-7-19(25)20(26)10-16/h5-8,10,12,14-15H,3-4,9,11,13H2,1-2H3,(H,27,30)	WLIGSGXPGRTAPA-UHFFFAOYSA-N	50465582	CHEMBL4277864	WD repeat-containing protein 5		 9.9								ChEMBL	10.1021/acs.jmedchem.8b00375	10.7270/Q2KD21KT	29889518			Wang, F; Jeon, KO; Salovich, JM; Macdonald, JD; Alvarado, J; Gogliotti, RD; Phan, J; Olejniczak, ET; Sun, Q; Wang, S; Camper, D; Yuh, JP; Shaw, JG; Sai, J; Rossanese, OW; Tansey, WP; Stauffer, SR; Fesik, SW	TBA	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50465582	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50465582&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			134369648	433932847							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51135344	CC(C)Oc1ccc(cc1CN(CC1CC1)C(=O)Cc1ccc(Cl)c(Cl)c1)-c1cn2CCCc2n1	InChI=1S/C28H31Cl2N3O2/c1-18(2)35-26-10-8-21(25-17-32-11-3-4-27(32)31-25)14-22(26)16-33(15-19-5-6-19)28(34)13-20-7-9-23(29)24(30)12-20/h7-10,12,14,17-19H,3-6,11,13,15-16H2,1-2H3	WDTUWBJQTSAVHL-UHFFFAOYSA-N	50465583	CHEMBL4288521	WD repeat-containing protein 5		 13								ChEMBL	10.1021/acs.jmedchem.8b00375	10.7270/Q2KD21KT	29889518			Wang, F; Jeon, KO; Salovich, JM; Macdonald, JD; Alvarado, J; Gogliotti, RD; Phan, J; Olejniczak, ET; Sun, Q; Wang, S; Camper, D; Yuh, JP; Shaw, JG; Sai, J; Rossanese, OW; Tansey, WP; Stauffer, SR; Fesik, SW	TBA	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50465583	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50465583&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			134369665	433932848							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51135345	Clc1ccc(CC(=O)NCc2cc(ccc2OC2CCC2)-c2cn3CCCc3n2)cc1Cl	InChI=1S/C25H25Cl2N3O2/c26-20-8-6-16(11-21(20)27)12-25(31)28-14-18-13-17(7-9-23(18)32-19-3-1-4-19)22-15-30-10-2-5-24(30)29-22/h6-9,11,13,15,19H,1-5,10,12,14H2,(H,28,31)	UVVAQRKKDXENDO-UHFFFAOYSA-N	50465584	CHEMBL4293572	WD repeat-containing protein 5		 2.8								ChEMBL	10.1021/acs.jmedchem.8b00375	10.7270/Q2KD21KT	29889518			Wang, F; Jeon, KO; Salovich, JM; Macdonald, JD; Alvarado, J; Gogliotti, RD; Phan, J; Olejniczak, ET; Sun, Q; Wang, S; Camper, D; Yuh, JP; Shaw, JG; Sai, J; Rossanese, OW; Tansey, WP; Stauffer, SR; Fesik, SW	TBA	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50465584	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50465584&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			134369676	433932849							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51135346	Clc1ccc(CC(=O)N[C@@H]2CCc3ccc(cc23)-c2cn3CCCc3n2)cc1Cl	InChI=1S/C23H21Cl2N3O/c24-18-7-3-14(10-19(18)25)11-23(29)27-20-8-6-15-4-5-16(12-17(15)20)21-13-28-9-1-2-22(28)26-21/h3-5,7,10,12-13,20H,1-2,6,8-9,11H2,(H,27,29)/t20-/m1/s1	HLGZWOPKLXYBFI-HXUWFJFHSA-N	50465585	CHEMBL4279907::US10501466, Example B11	WD repeat-containing protein 5		 2.5								ChEMBL	10.1021/acs.jmedchem.8b00375	10.7270/Q2KD21KT	29889518			Wang, F; Jeon, KO; Salovich, JM; Macdonald, JD; Alvarado, J; Gogliotti, RD; Phan, J; Olejniczak, ET; Sun, Q; Wang, S; Camper, D; Yuh, JP; Shaw, JG; Sai, J; Rossanese, OW; Tansey, WP; Stauffer, SR; Fesik, SW	TBA	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50465585	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50465585&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138470418	433932850							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51135347	COc1cc(ccc1C)C(=O)N[C@@H]1CCCc2ccc(cc12)-c1cn2CCCc2n1	InChI=1S/C25H27N3O2/c1-16-8-9-19(14-23(16)30-2)25(29)27-21-6-3-5-17-10-11-18(13-20(17)21)22-15-28-12-4-7-24(28)26-22/h8-11,13-15,21H,3-7,12H2,1-2H3,(H,27,29)/t21-/m1/s1	HMOMQPHKMPWUKJ-OAQYLSRUSA-N	50465586	CHEMBL4294174::US10501466, Example B14	WD repeat-containing protein 5		 9.4								ChEMBL	10.1021/acs.jmedchem.8b00375	10.7270/Q2KD21KT	29889518			Wang, F; Jeon, KO; Salovich, JM; Macdonald, JD; Alvarado, J; Gogliotti, RD; Phan, J; Olejniczak, ET; Sun, Q; Wang, S; Camper, D; Yuh, JP; Shaw, JG; Sai, J; Rossanese, OW; Tansey, WP; Stauffer, SR; Fesik, SW	TBA	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50465586	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50465586&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138470399	433932851							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51135348	NC(=N)COc1cccc(Cl)c1	InChI=1S/C8H9ClN2O/c9-6-2-1-3-7(4-6)12-5-8(10)11/h1-4H,5H2,(H3,10,11)	GQIZPSYLKHRSNS-UHFFFAOYSA-N	50465587	CHEMBL4293101	WD repeat-containing protein 5		 651000								ChEMBL	10.1021/acs.jmedchem.8b00375	10.7270/Q2KD21KT	29889518			Wang, F; Jeon, KO; Salovich, JM; Macdonald, JD; Alvarado, J; Gogliotti, RD; Phan, J; Olejniczak, ET; Sun, Q; Wang, S; Camper, D; Yuh, JP; Shaw, JG; Sai, J; Rossanese, OW; Tansey, WP; Stauffer, SR; Fesik, SW	TBA	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50465587	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50465587&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			15561337	433932852							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51135349	CC(C)Oc1cccc(c1)-c1cn2CCCc2n1	InChI=1S/C15H18N2O/c1-11(2)18-13-6-3-5-12(9-13)14-10-17-8-4-7-15(17)16-14/h3,5-6,9-11H,4,7-8H2,1-2H3	VYEYXWPFGSQWDX-UHFFFAOYSA-N	50465588	CHEMBL4280671	WD repeat-containing protein 5		 109000								ChEMBL	10.1021/acs.jmedchem.8b00375	10.7270/Q2KD21KT	29889518			Wang, F; Jeon, KO; Salovich, JM; Macdonald, JD; Alvarado, J; Gogliotti, RD; Phan, J; Olejniczak, ET; Sun, Q; Wang, S; Camper, D; Yuh, JP; Shaw, JG; Sai, J; Rossanese, OW; Tansey, WP; Stauffer, SR; Fesik, SW	TBA	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50465588	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50465588&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			145981722	433932853							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51135350	CCC(C)Oc1ccc(cc1)-c1cn2CCCc2n1	InChI=1S/C16H20N2O/c1-3-12(2)19-14-8-6-13(7-9-14)15-11-18-10-4-5-16(18)17-15/h6-9,11-12H,3-5,10H2,1-2H3	BDPHPPKMHJHHFF-UHFFFAOYSA-N	50465589	CHEMBL4279456	WD repeat-containing protein 5		>125000								ChEMBL	10.1021/acs.jmedchem.8b00375	10.7270/Q2KD21KT	29889518			Wang, F; Jeon, KO; Salovich, JM; Macdonald, JD; Alvarado, J; Gogliotti, RD; Phan, J; Olejniczak, ET; Sun, Q; Wang, S; Camper, D; Yuh, JP; Shaw, JG; Sai, J; Rossanese, OW; Tansey, WP; Stauffer, SR; Fesik, SW	TBA	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50465589	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50465589&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			145982119	433932854							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51135351	O=C(NCc1cccc(c1)-c1cn2CCCc2n1)c1ccccc1	InChI=1S/C20H19N3O/c24-20(16-7-2-1-3-8-16)21-13-15-6-4-9-17(12-15)18-14-23-11-5-10-19(23)22-18/h1-4,6-9,12,14H,5,10-11,13H2,(H,21,24)	OHOWMSISBAWFED-UHFFFAOYSA-N	50465590	CHEMBL4277278	WD repeat-containing protein 5		 7210								ChEMBL	10.1021/acs.jmedchem.8b00375	10.7270/Q2KD21KT	29889518			Wang, F; Jeon, KO; Salovich, JM; Macdonald, JD; Alvarado, J; Gogliotti, RD; Phan, J; Olejniczak, ET; Sun, Q; Wang, S; Camper, D; Yuh, JP; Shaw, JG; Sai, J; Rossanese, OW; Tansey, WP; Stauffer, SR; Fesik, SW	TBA	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50465590	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50465590&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	G1Y	6DAK	134369552	433932855							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51135352	COc1cccc(c1)C(=O)N(CC1CC1)Cc1cccc(c1)-c1cn2CCCc2n1	InChI=1S/C25H27N3O2/c1-30-22-8-3-7-21(14-22)25(29)28(15-18-10-11-18)16-19-5-2-6-20(13-19)23-17-27-12-4-9-24(27)26-23/h2-3,5-8,13-14,17-18H,4,9-12,15-16H2,1H3	UVWAIBUOXKRXQY-UHFFFAOYSA-N	50465591	CHEMBL4294825	WD repeat-containing protein 5		 219								ChEMBL	10.1021/acs.jmedchem.8b00375	10.7270/Q2KD21KT	29889518			Wang, F; Jeon, KO; Salovich, JM; Macdonald, JD; Alvarado, J; Gogliotti, RD; Phan, J; Olejniczak, ET; Sun, Q; Wang, S; Camper, D; Yuh, JP; Shaw, JG; Sai, J; Rossanese, OW; Tansey, WP; Stauffer, SR; Fesik, SW	TBA	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50465591	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50465591&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	G2J	6DAR	134369559	433932856							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51135353	COc1cccc(c1)C(=O)NCc1cc(ccc1OC1CCC1)-c1cn2CCCc2n1	InChI=1S/C25H27N3O3/c1-30-21-8-2-5-18(14-21)25(29)26-15-19-13-17(10-11-23(19)31-20-6-3-7-20)22-16-28-12-4-9-24(28)27-22/h2,5,8,10-11,13-14,16,20H,3-4,6-7,9,12,15H2,1H3,(H,26,29)	VDRHHZQQKHUNMM-UHFFFAOYSA-N	50465592	CHEMBL4284733	WD repeat-containing protein 5		 105								ChEMBL	10.1021/acs.jmedchem.8b00375	10.7270/Q2KD21KT	29889518			Wang, F; Jeon, KO; Salovich, JM; Macdonald, JD; Alvarado, J; Gogliotti, RD; Phan, J; Olejniczak, ET; Sun, Q; Wang, S; Camper, D; Yuh, JP; Shaw, JG; Sai, J; Rossanese, OW; Tansey, WP; Stauffer, SR; Fesik, SW	TBA	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50465592	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50465592&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			134364178	433932857							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51135354	COc1cc(ccc1C)C(=O)N(CC1CC1)Cc1cc(ccc1OC1CCC1)-c1cn2CCCc2n1	InChI=1S/C30H35N3O3/c1-20-8-11-23(16-28(20)35-2)30(34)33(17-21-9-10-21)18-24-15-22(12-13-27(24)36-25-5-3-6-25)26-19-32-14-4-7-29(32)31-26/h8,11-13,15-16,19,21,25H,3-7,9-10,14,17-18H2,1-2H3	OSPGDFKBCFSGOZ-UHFFFAOYSA-N	50465593	CHEMBL4283374	WD repeat-containing protein 5		 3.5								ChEMBL	10.1021/acs.jmedchem.8b00375	10.7270/Q2KD21KT	29889518			Wang, F; Jeon, KO; Salovich, JM; Macdonald, JD; Alvarado, J; Gogliotti, RD; Phan, J; Olejniczak, ET; Sun, Q; Wang, S; Camper, D; Yuh, JP; Shaw, JG; Sai, J; Rossanese, OW; Tansey, WP; Stauffer, SR; Fesik, SW	TBA	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50465593	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50465593&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			134364156	433932858							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51135355	COc1cc(cc(OC)c1C)C(=O)N[C@@H]1CCc2ccc(cc12)-c1cn2CCCc2n1	InChI=1S/C25H27N3O3/c1-15-22(30-2)12-18(13-23(15)31-3)25(29)27-20-9-8-16-6-7-17(11-19(16)20)21-14-28-10-4-5-24(28)26-21/h6-7,11-14,20H,4-5,8-10H2,1-3H3,(H,27,29)/t20-/m1/s1	GRFBFSARRYJWSN-HXUWFJFHSA-N	50465552	CHEMBL4291641::US10501466, Example B29	WD repeat-containing protein 5		<1.000000								ChEMBL	10.1021/acs.jmedchem.8b00375	10.7270/Q2KD21KT	29889518			Wang, F; Jeon, KO; Salovich, JM; Macdonald, JD; Alvarado, J; Gogliotti, RD; Phan, J; Olejniczak, ET; Sun, Q; Wang, S; Camper, D; Yuh, JP; Shaw, JG; Sai, J; Rossanese, OW; Tansey, WP; Stauffer, SR; Fesik, SW	TBA	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50465552	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50465552&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138470423	433932817							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51135356	COc1cc(CC(=O)N[C@@H]2CCc3ccc(cc23)-c2cn3CCCc3n2)ccc1C	InChI=1S/C25H27N3O2/c1-16-5-6-17(12-23(16)30-2)13-25(29)27-21-10-9-18-7-8-19(14-20(18)21)22-15-28-11-3-4-24(28)26-22/h5-8,12,14-15,21H,3-4,9-11,13H2,1-2H3,(H,27,29)/t21-/m1/s1	WHKWYCMXCHKNSQ-OAQYLSRUSA-N	50465555	CHEMBL4287817	WD repeat-containing protein 5		 8.4								ChEMBL	10.1021/acs.jmedchem.8b00375	10.7270/Q2KD21KT	29889518			Wang, F; Jeon, KO; Salovich, JM; Macdonald, JD; Alvarado, J; Gogliotti, RD; Phan, J; Olejniczak, ET; Sun, Q; Wang, S; Camper, D; Yuh, JP; Shaw, JG; Sai, J; Rossanese, OW; Tansey, WP; Stauffer, SR; Fesik, SW	TBA	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50465555	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50465555&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			145993387	433932820							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51135357	Cc1cc(ccn1)C(=O)N[C@@H]1CCc2ccc(cc12)-c1cn2CCCc2n1	InChI=1S/C22H22N4O/c1-14-11-17(8-9-23-14)22(27)25-19-7-6-15-4-5-16(12-18(15)19)20-13-26-10-2-3-21(26)24-20/h4-5,8-9,11-13,19H,2-3,6-7,10H2,1H3,(H,25,27)/t19-/m1/s1	YKUGUWMZBHIDFR-LJQANCHMSA-N	50465594	CHEMBL4284408::US10501466, Example B24	WD repeat-containing protein 5		 182								ChEMBL	10.1021/acs.jmedchem.8b00375	10.7270/Q2KD21KT	29889518			Wang, F; Jeon, KO; Salovich, JM; Macdonald, JD; Alvarado, J; Gogliotti, RD; Phan, J; Olejniczak, ET; Sun, Q; Wang, S; Camper, D; Yuh, JP; Shaw, JG; Sai, J; Rossanese, OW; Tansey, WP; Stauffer, SR; Fesik, SW	TBA	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50465594	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50465594&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138470404	433932859							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51135358	Clc1ccc(CC(=O)N[C@@H]2CCc3ccc(cc23)-c2cn3CCCc3n2)cc1Cl	InChI=1S/C23H21Cl2N3O/c24-18-7-3-14(10-19(18)25)11-23(29)27-20-8-6-15-4-5-16(12-17(15)20)21-13-28-9-1-2-22(28)26-21/h3-5,7,10,12-13,20H,1-2,6,8-9,11H2,(H,27,29)/t20-/m1/s1	HLGZWOPKLXYBFI-HXUWFJFHSA-N	50465585	CHEMBL4279907::US10501466, Example B11	WD repeat-containing protein 5			 9270							ChEMBL	10.1021/acs.jmedchem.8b00375	10.7270/Q2KD21KT	29889518			Wang, F; Jeon, KO; Salovich, JM; Macdonald, JD; Alvarado, J; Gogliotti, RD; Phan, J; Olejniczak, ET; Sun, Q; Wang, S; Camper, D; Yuh, JP; Shaw, JG; Sai, J; Rossanese, OW; Tansey, WP; Stauffer, SR; Fesik, SW	TBA	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50465585	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50465585&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138470418	433932850							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51135359	COc1cc(ccc1C)C(=O)N[C@@H]1CCCc2ccc(cc12)-c1cn2CCCc2n1	InChI=1S/C25H27N3O2/c1-16-8-9-19(14-23(16)30-2)25(29)27-21-6-3-5-17-10-11-18(13-20(17)21)22-15-28-12-4-7-24(28)26-22/h8-11,13-15,21H,3-7,12H2,1-2H3,(H,27,29)/t21-/m1/s1	HMOMQPHKMPWUKJ-OAQYLSRUSA-N	50465586	CHEMBL4294174::US10501466, Example B14	WD repeat-containing protein 5			>20000							ChEMBL	10.1021/acs.jmedchem.8b00375	10.7270/Q2KD21KT	29889518			Wang, F; Jeon, KO; Salovich, JM; Macdonald, JD; Alvarado, J; Gogliotti, RD; Phan, J; Olejniczak, ET; Sun, Q; Wang, S; Camper, D; Yuh, JP; Shaw, JG; Sai, J; Rossanese, OW; Tansey, WP; Stauffer, SR; Fesik, SW	TBA	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50465586	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50465586&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138470399	433932851							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51135360	Cc1cc(ccn1)C(=O)N[C@@H]1CCc2ccc(cc12)-c1cn2CCCc2n1	InChI=1S/C22H22N4O/c1-14-11-17(8-9-23-14)22(27)25-19-7-6-15-4-5-16(12-18(15)19)20-13-26-10-2-3-21(26)24-20/h4-5,8-9,11-13,19H,2-3,6-7,10H2,1H3,(H,25,27)/t19-/m1/s1	YKUGUWMZBHIDFR-LJQANCHMSA-N	50465594	CHEMBL4284408::US10501466, Example B24	WD repeat-containing protein 5			>20000							ChEMBL	10.1021/acs.jmedchem.8b00375	10.7270/Q2KD21KT	29889518			Wang, F; Jeon, KO; Salovich, JM; Macdonald, JD; Alvarado, J; Gogliotti, RD; Phan, J; Olejniczak, ET; Sun, Q; Wang, S; Camper, D; Yuh, JP; Shaw, JG; Sai, J; Rossanese, OW; Tansey, WP; Stauffer, SR; Fesik, SW	TBA	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50465594	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50465594&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138470404	433932859							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51135361	COc1cc(ccc1C)C(=O)N[C@@H]1CCCc2ccc(cc12)-c1cn2CCCc2n1	InChI=1S/C25H27N3O2/c1-16-8-9-19(14-23(16)30-2)25(29)27-21-6-3-5-17-10-11-18(13-20(17)21)22-15-28-12-4-7-24(28)26-22/h8-11,13-15,21H,3-7,12H2,1-2H3,(H,27,29)/t21-/m1/s1	HMOMQPHKMPWUKJ-OAQYLSRUSA-N	50465586	CHEMBL4294174::US10501466, Example B14	WD repeat-containing protein 5		 27								ChEMBL	10.1021/acs.jmedchem.8b00375	10.7270/Q2KD21KT	29889518			Wang, F; Jeon, KO; Salovich, JM; Macdonald, JD; Alvarado, J; Gogliotti, RD; Phan, J; Olejniczak, ET; Sun, Q; Wang, S; Camper, D; Yuh, JP; Shaw, JG; Sai, J; Rossanese, OW; Tansey, WP; Stauffer, SR; Fesik, SW	TBA	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50465586	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50465586&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138470399	433932851							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51135362	NC(=N)c1ccc(cc1)-c1ccccc1	InChI=1S/C13H12N2/c14-13(15)12-8-6-11(7-9-12)10-4-2-1-3-5-10/h1-9H,(H3,14,15)	VHEYCTCATJSAAI-UHFFFAOYSA-N	50465595	CHEMBL4285882	WD repeat-containing protein 5		 843000								ChEMBL	10.1021/acs.jmedchem.8b00375	10.7270/Q2KD21KT	29889518			Wang, F; Jeon, KO; Salovich, JM; Macdonald, JD; Alvarado, J; Gogliotti, RD; Phan, J; Olejniczak, ET; Sun, Q; Wang, S; Camper, D; Yuh, JP; Shaw, JG; Sai, J; Rossanese, OW; Tansey, WP; Stauffer, SR; Fesik, SW	TBA	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50465595	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50465595&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			3308644	433932860							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51135363	COc1ccc(cc1)-c1cn2CCCc2n1	InChI=1S/C13H14N2O/c1-16-11-6-4-10(5-7-11)12-9-15-8-2-3-13(15)14-12/h4-7,9H,2-3,8H2,1H3	WOYRQBRHXBCHHZ-UHFFFAOYSA-N	50465596	CHEMBL1625120	WD repeat-containing protein 5		 61000								ChEMBL	10.1021/acs.jmedchem.8b00375	10.7270/Q2KD21KT	29889518			Wang, F; Jeon, KO; Salovich, JM; Macdonald, JD; Alvarado, J; Gogliotti, RD; Phan, J; Olejniczak, ET; Sun, Q; Wang, S; Camper, D; Yuh, JP; Shaw, JG; Sai, J; Rossanese, OW; Tansey, WP; Stauffer, SR; Fesik, SW	TBA	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50465596	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50465596&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			910123	433932861							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51135364	CN1CCc2cc(ccc12)-c1cn2CCCc2n1	InChI=1S/C15H17N3/c1-17-8-6-12-9-11(4-5-14(12)17)13-10-18-7-2-3-15(18)16-13/h4-5,9-10H,2-3,6-8H2,1H3	GANOSYHSDIPGSR-UHFFFAOYSA-N	50465597	CHEMBL4281112	WD repeat-containing protein 5		 85200								ChEMBL	10.1021/acs.jmedchem.8b00375	10.7270/Q2KD21KT	29889518			Wang, F; Jeon, KO; Salovich, JM; Macdonald, JD; Alvarado, J; Gogliotti, RD; Phan, J; Olejniczak, ET; Sun, Q; Wang, S; Camper, D; Yuh, JP; Shaw, JG; Sai, J; Rossanese, OW; Tansey, WP; Stauffer, SR; Fesik, SW	TBA	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50465597	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50465597&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	G2V	6DAI	137349384	433932862							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51135365	O=C(NCc1cccc(c1)-c1cn2CCCc2n1)C1CCCCC1	InChI=1S/C20H25N3O/c24-20(16-7-2-1-3-8-16)21-13-15-6-4-9-17(12-15)18-14-23-11-5-10-19(23)22-18/h4,6,9,12,14,16H,1-3,5,7-8,10-11,13H2,(H,21,24)	GZZSSYVKMPAQRS-UHFFFAOYSA-N	50465598	CHEMBL4289405	WD repeat-containing protein 5		 7540								ChEMBL	10.1021/acs.jmedchem.8b00375	10.7270/Q2KD21KT	29889518			Wang, F; Jeon, KO; Salovich, JM; Macdonald, JD; Alvarado, J; Gogliotti, RD; Phan, J; Olejniczak, ET; Sun, Q; Wang, S; Camper, D; Yuh, JP; Shaw, JG; Sai, J; Rossanese, OW; Tansey, WP; Stauffer, SR; Fesik, SW	TBA	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50465598	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50465598&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			134369551	433932863							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51135366	Clc1ccc(CC(=O)NCc2cccc(c2)-c2cn3CCCc3n2)cc1Cl	InChI=1S/C21H19Cl2N3O/c22-17-7-6-14(10-18(17)23)11-21(27)24-12-15-3-1-4-16(9-15)19-13-26-8-2-5-20(26)25-19/h1,3-4,6-7,9-10,13H,2,5,8,11-12H2,(H,24,27)	QOIRVBBMKNKETR-UHFFFAOYSA-N	50465599	CHEMBL4288724	WD repeat-containing protein 5		 118								ChEMBL	10.1021/acs.jmedchem.8b00375	10.7270/Q2KD21KT	29889518			Wang, F; Jeon, KO; Salovich, JM; Macdonald, JD; Alvarado, J; Gogliotti, RD; Phan, J; Olejniczak, ET; Sun, Q; Wang, S; Camper, D; Yuh, JP; Shaw, JG; Sai, J; Rossanese, OW; Tansey, WP; Stauffer, SR; Fesik, SW	TBA	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50465599	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50465599&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			134369623	433932864							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51135367	O=C(NCc1cccc(c1)-c1cn2CCCc2n1)c1cccnc1	InChI=1S/C19H18N4O/c24-19(16-6-2-8-20-12-16)21-11-14-4-1-5-15(10-14)17-13-23-9-3-7-18(23)22-17/h1-2,4-6,8,10,12-13H,3,7,9,11H2,(H,21,24)	MCEVWKLGFYQYRT-UHFFFAOYSA-N	50465600	CHEMBL4295183	WD repeat-containing protein 5		 4130								ChEMBL	10.1021/acs.jmedchem.8b00375	10.7270/Q2KD21KT	29889518			Wang, F; Jeon, KO; Salovich, JM; Macdonald, JD; Alvarado, J; Gogliotti, RD; Phan, J; Olejniczak, ET; Sun, Q; Wang, S; Camper, D; Yuh, JP; Shaw, JG; Sai, J; Rossanese, OW; Tansey, WP; Stauffer, SR; Fesik, SW	TBA	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50465600	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50465600&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			134369579	433932865							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51135368	COc1cc(ccn1)C(=O)N(CC1CC1)Cc1cccc(c1)-c1cn2CCCc2n1	InChI=1S/C24H26N4O2/c1-30-23-13-20(9-10-25-23)24(29)28(14-17-7-8-17)15-18-4-2-5-19(12-18)21-16-27-11-3-6-22(27)26-21/h2,4-5,9-10,12-13,16-17H,3,6-8,11,14-15H2,1H3	OTONOFNXSMNLHM-UHFFFAOYSA-N	50465601	CHEMBL4284629	WD repeat-containing protein 5		 480								ChEMBL	10.1021/acs.jmedchem.8b00375	10.7270/Q2KD21KT	29889518			Wang, F; Jeon, KO; Salovich, JM; Macdonald, JD; Alvarado, J; Gogliotti, RD; Phan, J; Olejniczak, ET; Sun, Q; Wang, S; Camper, D; Yuh, JP; Shaw, JG; Sai, J; Rossanese, OW; Tansey, WP; Stauffer, SR; Fesik, SW	TBA	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50465601	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50465601&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			134369594	433932866							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51135369	CCOc1ccc(cc1CN(CC1CC1)C(=O)c1cccc(OC)c1)-c1cn2CCCc2n1	InChI=1S/C27H31N3O3/c1-3-33-25-12-11-20(24-18-29-13-5-8-26(29)28-24)14-22(25)17-30(16-19-9-10-19)27(31)21-6-4-7-23(15-21)32-2/h4,6-7,11-12,14-15,18-19H,3,5,8-10,13,16-17H2,1-2H3	LZJTUJUGRLHZQK-UHFFFAOYSA-N	50465602	CHEMBL4278618	WD repeat-containing protein 5		 43								ChEMBL	10.1021/acs.jmedchem.8b00375	10.7270/Q2KD21KT	29889518			Wang, F; Jeon, KO; Salovich, JM; Macdonald, JD; Alvarado, J; Gogliotti, RD; Phan, J; Olejniczak, ET; Sun, Q; Wang, S; Camper, D; Yuh, JP; Shaw, JG; Sai, J; Rossanese, OW; Tansey, WP; Stauffer, SR; Fesik, SW	TBA	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50465602	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50465602&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			134369629	433932867							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51135370	Clc1ccc(CC(=O)NCc2cc(ccc2N2CCOCC2)-c2cn3CCCc3n2)cc1Cl	InChI=1S/C25H26Cl2N4O2/c26-20-5-3-17(12-21(20)27)13-25(32)28-15-19-14-18(22-16-31-7-1-2-24(31)29-22)4-6-23(19)30-8-10-33-11-9-30/h3-6,12,14,16H,1-2,7-11,13,15H2,(H,28,32)	OIGLFJGNJOWHFL-UHFFFAOYSA-N	50465603	CHEMBL4285163	WD repeat-containing protein 5		 21								ChEMBL	10.1021/acs.jmedchem.8b00375	10.7270/Q2KD21KT	29889518			Wang, F; Jeon, KO; Salovich, JM; Macdonald, JD; Alvarado, J; Gogliotti, RD; Phan, J; Olejniczak, ET; Sun, Q; Wang, S; Camper, D; Yuh, JP; Shaw, JG; Sai, J; Rossanese, OW; Tansey, WP; Stauffer, SR; Fesik, SW	TBA	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50465603	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50465603&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			134369672	433932868							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51135371	Clc1ccc(CC(=O)N(CC2CC2)Cc2cc(ccc2OC2CCC2)-c2cn3CCCc3n2)cc1Cl	InChI=1S/C29H31Cl2N3O2/c30-24-10-8-20(13-25(24)31)14-29(35)34(16-19-6-7-19)17-22-15-21(9-11-27(22)36-23-3-1-4-23)26-18-33-12-2-5-28(33)32-26/h8-11,13,15,18-19,23H,1-7,12,14,16-17H2	PSFBUFWKSANDIK-UHFFFAOYSA-N	50465604	CHEMBL4283339	WD repeat-containing protein 5		 29								ChEMBL	10.1021/acs.jmedchem.8b00375	10.7270/Q2KD21KT	29889518			Wang, F; Jeon, KO; Salovich, JM; Macdonald, JD; Alvarado, J; Gogliotti, RD; Phan, J; Olejniczak, ET; Sun, Q; Wang, S; Camper, D; Yuh, JP; Shaw, JG; Sai, J; Rossanese, OW; Tansey, WP; Stauffer, SR; Fesik, SW	TBA	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50465604	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50465604&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			134369652	433932869							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51135372	Cc1cc(ccn1)C(=O)N[C@@H]1CCc2ccc(cc12)-c1cn2CCCc2n1	InChI=1S/C22H22N4O/c1-14-11-17(8-9-23-14)22(27)25-19-7-6-15-4-5-16(12-18(15)19)20-13-26-10-2-3-21(26)24-20/h4-5,8-9,11-13,19H,2-3,6-7,10H2,1H3,(H,25,27)/t19-/m1/s1	YKUGUWMZBHIDFR-LJQANCHMSA-N	50465594	CHEMBL4284408::US10501466, Example B24	WD repeat-containing protein 5		 65								ChEMBL	10.1021/acs.jmedchem.8b00375	10.7270/Q2KD21KT	29889518			Wang, F; Jeon, KO; Salovich, JM; Macdonald, JD; Alvarado, J; Gogliotti, RD; Phan, J; Olejniczak, ET; Sun, Q; Wang, S; Camper, D; Yuh, JP; Shaw, JG; Sai, J; Rossanese, OW; Tansey, WP; Stauffer, SR; Fesik, SW	TBA	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50465594	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50465594&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138470404	433932859							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51135373	Clc1ccc(CC(=O)N[C@@H]2CCc3ccc(cc23)-c2cn3CCCc3n2)cc1Cl	InChI=1S/C23H21Cl2N3O/c24-18-7-3-14(10-19(18)25)11-23(29)27-20-8-6-15-4-5-16(12-17(15)20)21-13-28-9-1-2-22(28)26-21/h3-5,7,10,12-13,20H,1-2,6,8-9,11H2,(H,27,29)/t20-/m1/s1	HLGZWOPKLXYBFI-HXUWFJFHSA-N	50465585	CHEMBL4279907::US10501466, Example B11	WD repeat-containing protein 5		 2.7								ChEMBL	10.1021/acs.jmedchem.8b00375	10.7270/Q2KD21KT	29889518			Wang, F; Jeon, KO; Salovich, JM; Macdonald, JD; Alvarado, J; Gogliotti, RD; Phan, J; Olejniczak, ET; Sun, Q; Wang, S; Camper, D; Yuh, JP; Shaw, JG; Sai, J; Rossanese, OW; Tansey, WP; Stauffer, SR; Fesik, SW	TBA	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50465585	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50465585&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138470418	433932850							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51135374	COc1cc(CC(=O)N[C@@H]2CCc3ccc(cc23)-c2cn3CCCc3n2)ccc1C	InChI=1S/C25H27N3O2/c1-16-5-6-17(12-23(16)30-2)13-25(29)27-21-10-9-18-7-8-19(14-20(18)21)22-15-28-11-3-4-24(28)26-22/h5-8,12,14-15,21H,3-4,9-11,13H2,1-2H3,(H,27,29)/t21-/m1/s1	WHKWYCMXCHKNSQ-OAQYLSRUSA-N	50465555	CHEMBL4287817	WD repeat-containing protein 5			 12000							ChEMBL	10.1021/acs.jmedchem.8b00375	10.7270/Q2KD21KT	29889518			Wang, F; Jeon, KO; Salovich, JM; Macdonald, JD; Alvarado, J; Gogliotti, RD; Phan, J; Olejniczak, ET; Sun, Q; Wang, S; Camper, D; Yuh, JP; Shaw, JG; Sai, J; Rossanese, OW; Tansey, WP; Stauffer, SR; Fesik, SW	TBA	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50465555	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50465555&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			145993387	433932820							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51135375	COc1cc(cc(OC)c1C)C(=O)N[C@@H]1CCc2ccc(cc12)-c1cn2CCCc2n1	InChI=1S/C25H27N3O3/c1-15-22(30-2)12-18(13-23(15)31-3)25(29)27-20-9-8-16-6-7-17(11-19(16)20)21-14-28-10-4-5-24(28)26-21/h6-7,11-14,20H,4-5,8-10H2,1-3H3,(H,27,29)/t20-/m1/s1	GRFBFSARRYJWSN-HXUWFJFHSA-N	50465552	CHEMBL4291641::US10501466, Example B29	WD repeat-containing protein 5			 3200							ChEMBL	10.1021/acs.jmedchem.8b00375	10.7270/Q2KD21KT	29889518			Wang, F; Jeon, KO; Salovich, JM; Macdonald, JD; Alvarado, J; Gogliotti, RD; Phan, J; Olejniczak, ET; Sun, Q; Wang, S; Camper, D; Yuh, JP; Shaw, JG; Sai, J; Rossanese, OW; Tansey, WP; Stauffer, SR; Fesik, SW	TBA	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50465552	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50465552&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138470423	433932817							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51135376	CC(C)Oc1ccc(cc1)-c1cn2CCCc2n1	InChI=1S/C15H18N2O/c1-11(2)18-13-7-5-12(6-8-13)14-10-17-9-3-4-15(17)16-14/h5-8,10-11H,3-4,9H2,1-2H3	CUBMKZQQTMBJBK-UHFFFAOYSA-N	50465605	CHEMBL4287371	WD repeat-containing protein 5		 29700								ChEMBL	10.1021/acs.jmedchem.8b00375	10.7270/Q2KD21KT	29889518			Wang, F; Jeon, KO; Salovich, JM; Macdonald, JD; Alvarado, J; Gogliotti, RD; Phan, J; Olejniczak, ET; Sun, Q; Wang, S; Camper, D; Yuh, JP; Shaw, JG; Sai, J; Rossanese, OW; Tansey, WP; Stauffer, SR; Fesik, SW	TBA	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50465605	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50465605&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			145992918	433932870							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51135377	COc1cc(ccc1C)C(=O)NCc1cc(ccc1OC1CCC1)-c1cn2CCCc2n1	InChI=1S/C26H29N3O3/c1-17-8-9-19(14-24(17)31-2)26(30)27-15-20-13-18(10-11-23(20)32-21-5-3-6-21)22-16-29-12-4-7-25(29)28-22/h8-11,13-14,16,21H,3-7,12,15H2,1-2H3,(H,27,30)	ASFCKFRAVIIYOS-UHFFFAOYSA-N	50465606	CHEMBL4291223	WD repeat-containing protein 5		 16								ChEMBL	10.1021/acs.jmedchem.8b00375	10.7270/Q2KD21KT	29889518			Wang, F; Jeon, KO; Salovich, JM; Macdonald, JD; Alvarado, J; Gogliotti, RD; Phan, J; Olejniczak, ET; Sun, Q; Wang, S; Camper, D; Yuh, JP; Shaw, JG; Sai, J; Rossanese, OW; Tansey, WP; Stauffer, SR; Fesik, SW	TBA	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50465606	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50465606&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			134369708	433932871							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51135378	COc1cc(ccc1C)C(=O)NCc1cccc(c1)-c1cn2CCCc2n1	InChI=1S/C22H23N3O2/c1-15-8-9-18(12-20(15)27-2)22(26)23-13-16-5-3-6-17(11-16)19-14-25-10-4-7-21(25)24-19/h3,5-6,8-9,11-12,14H,4,7,10,13H2,1-2H3,(H,23,26)	NBPITMNATCCMHH-UHFFFAOYSA-N	50465607	CHEMBL4280428	WD repeat-containing protein 5		 95								ChEMBL	10.1021/acs.jmedchem.8b00375	10.7270/Q2KD21KT	29889518			Wang, F; Jeon, KO; Salovich, JM; Macdonald, JD; Alvarado, J; Gogliotti, RD; Phan, J; Olejniczak, ET; Sun, Q; Wang, S; Camper, D; Yuh, JP; Shaw, JG; Sai, J; Rossanese, OW; Tansey, WP; Stauffer, SR; Fesik, SW	TBA	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50465607	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50465607&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			134369669	433932872							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51135379	COc1ccc(cc1OC)C(=O)NCc1cccc(c1)-c1cn2CCCc2n1	InChI=1S/C22H23N3O3/c1-27-19-9-8-17(12-20(19)28-2)22(26)23-13-15-5-3-6-16(11-15)18-14-25-10-4-7-21(25)24-18/h3,5-6,8-9,11-12,14H,4,7,10,13H2,1-2H3,(H,23,26)	LMHMRAKBMDJZRC-UHFFFAOYSA-N	50465608	CHEMBL4288332	WD repeat-containing protein 5		 690								ChEMBL	10.1021/acs.jmedchem.8b00375	10.7270/Q2KD21KT	29889518			Wang, F; Jeon, KO; Salovich, JM; Macdonald, JD; Alvarado, J; Gogliotti, RD; Phan, J; Olejniczak, ET; Sun, Q; Wang, S; Camper, D; Yuh, JP; Shaw, JG; Sai, J; Rossanese, OW; Tansey, WP; Stauffer, SR; Fesik, SW	TBA	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50465608	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50465608&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			134369568	433932873							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
854168	COc1cccc(c1)C(=O)N(CC1CC1)C1CCc2ccc(cc12)-c1cn2CCCc2n1	InChI=1S/C27H29N3O2/c1-32-22-5-2-4-21(14-22)27(31)30(16-18-7-8-18)25-12-11-19-9-10-20(15-23(19)25)24-17-29-13-3-6-26(29)28-24/h2,4-5,9-10,14-15,17-18,25H,3,6-8,11-13,16H2,1H3	CPIAIQHDZOTIHD-UHFFFAOYSA-N	423366	US10501466, Example B1	WD repeat-containing protein 5		 693								US Patent		10.7270/Q2319Z71		aid1804048	US10501466	Fesik, SW; Stauffer, SR; Salovich, JM; Tansey, WP; Wang, F; Phan, J; Olejniczak, ET	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=423366	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=423366&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138470383	434149159							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
854169	Cc1ccc(cc1C(F)(F)F)C(=O)NC1CCc2ccc(cc12)-c1cn2CCCc2n1	InChI=1S/C24H22F3N3O/c1-14-4-5-17(12-19(14)24(25,26)27)23(31)29-20-9-8-15-6-7-16(11-18(15)20)21-13-30-10-2-3-22(30)28-21/h4-7,11-13,20H,2-3,8-10H2,1H3,(H,29,31)	VCRJNMVHRSWNIS-UHFFFAOYSA-N	423367	US10501466, Example B2	WD repeat-containing protein 5		 1380								US Patent		10.7270/Q2319Z71		aid1804048	US10501466	Fesik, SW; Stauffer, SR; Salovich, JM; Tansey, WP; Wang, F; Phan, J; Olejniczak, ET	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=423367	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=423367&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138470406	434149160							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
854170	COc1cc(ccc1C)C(=O)NC1CCc2ccc(cc12)-c1cn2CCCc2n1	InChI=1S/C24H25N3O2/c1-15-5-6-18(13-22(15)29-2)24(28)26-20-10-9-16-7-8-17(12-19(16)20)21-14-27-11-3-4-23(27)25-21/h5-8,12-14,20H,3-4,9-11H2,1-2H3,(H,26,28)	PHINNLAJTUGZSZ-UHFFFAOYSA-N	423368	US10501466, Example B3	WD repeat-containing protein 5		 30.2								US Patent		10.7270/Q2319Z71		aid1804048	US10501466	Fesik, SW; Stauffer, SR; Salovich, JM; Tansey, WP; Wang, F; Phan, J; Olejniczak, ET	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=423368	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=423368&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	G2D	6DAS	138470393	434149161							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
854171	CCOc1cccc(c1)C(=O)NC1CCc2ccc(cc12)-c1cn2CCCc2n1	InChI=1S/C24H25N3O2/c1-2-29-19-6-3-5-18(13-19)24(28)26-21-11-10-16-8-9-17(14-20(16)21)22-15-27-12-4-7-23(27)25-22/h3,5-6,8-9,13-15,21H,2,4,7,10-12H2,1H3,(H,26,28)	UFFWQQMDJDHECY-UHFFFAOYSA-N	423369	US10501466, Example B4	WD repeat-containing protein 5		 19.1								US Patent		10.7270/Q2319Z71		aid1804048	US10501466	Fesik, SW; Stauffer, SR; Salovich, JM; Tansey, WP; Wang, F; Phan, J; Olejniczak, ET	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=423369	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=423369&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138470445	434149162							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
854172	COc1cc(C)cc(c1)C(=O)NC1CCc2ccc(cc12)-c1cn2CCCc2n1	InChI=1S/C24H25N3O2/c1-15-10-18(12-19(11-15)29-2)24(28)26-21-8-7-16-5-6-17(13-20(16)21)22-14-27-9-3-4-23(27)25-22/h5-6,10-14,21H,3-4,7-9H2,1-2H3,(H,26,28)	JGLPLQYDHABILB-UHFFFAOYSA-N	423370	US10501466, Example B5	WD repeat-containing protein 5		 27.0								US Patent		10.7270/Q2319Z71		aid1804048	US10501466	Fesik, SW; Stauffer, SR; Salovich, JM; Tansey, WP; Wang, F; Phan, J; Olejniczak, ET	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=423370	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=423370&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138470382	434149163							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
854173	Clc1ccc(CC(=O)NC2CCc3ccc(cc23)-c2cn3CCCc3n2)cc1Cl	InChI=1S/C23H21Cl2N3O/c24-18-7-3-14(10-19(18)25)11-23(29)27-20-8-6-15-4-5-16(12-17(15)20)21-13-28-9-1-2-22(28)26-21/h3-5,7,10,12-13,20H,1-2,6,8-9,11H2,(H,27,29)	HLGZWOPKLXYBFI-UHFFFAOYSA-N	423371	US10501466, Example B6	WD repeat-containing protein 5		 3.35								US Patent		10.7270/Q2319Z71		aid1804048	US10501466	Fesik, SW; Stauffer, SR; Salovich, JM; Tansey, WP; Wang, F; Phan, J; Olejniczak, ET	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=423371	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=423371&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138470407	434149164							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
854174	CC(=O)N1CCCC(C1)C(=O)NC1CCc2ccc(cc12)-c1cn2CCCc2n1	InChI=1S/C23H28N4O2/c1-15(28)26-10-2-4-18(13-26)23(29)25-20-9-8-16-6-7-17(12-19(16)20)21-14-27-11-3-5-22(27)24-21/h6-7,12,14,18,20H,2-5,8-11,13H2,1H3,(H,25,29)	BKBBJFFASFNPGD-UHFFFAOYSA-N	423372	US10501466, Example B7	WD repeat-containing protein 5		 33.0								US Patent		10.7270/Q2319Z71		aid1804048	US10501466	Fesik, SW; Stauffer, SR; Salovich, JM; Tansey, WP; Wang, F; Phan, J; Olejniczak, ET	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=423372	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=423372&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138470440	434149165							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
854175	CCC(=O)N1CCCC(C1)C(=O)NC1CCc2ccc(cc12)-c1cn2CCCc2n1	InChI=1S/C24H30N4O2/c1-2-23(29)28-12-3-5-18(14-28)24(30)26-20-10-9-16-7-8-17(13-19(16)20)21-15-27-11-4-6-22(27)25-21/h7-8,13,15,18,20H,2-6,9-12,14H2,1H3,(H,26,30)	NLYDZVTWTSGDDI-UHFFFAOYSA-N	423373	US10501466, Example B8	WD repeat-containing protein 5		 21.0								US Patent		10.7270/Q2319Z71		aid1804048	US10501466	Fesik, SW; Stauffer, SR; Salovich, JM; Tansey, WP; Wang, F; Phan, J; Olejniczak, ET	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=423373	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=423373&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138470417	434149166							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
854176	FC(F)(F)CC(=O)N1CCCC(C1)C(=O)NC1CCc2ccc(cc12)-c1cn2CCCc2n1	InChI=1S/C24H27F3N4O2/c25-24(26,27)12-22(32)31-10-1-3-17(13-31)23(33)29-19-8-7-15-5-6-16(11-18(15)19)20-14-30-9-2-4-21(30)28-20/h5-6,11,14,17,19H,1-4,7-10,12-13H2,(H,29,33)	ZBFBWTCDWNQFHE-UHFFFAOYSA-N	423374	US10501466, Example B9	WD repeat-containing protein 5		 90.0								US Patent		10.7270/Q2319Z71		aid1804048	US10501466	Fesik, SW; Stauffer, SR; Salovich, JM; Tansey, WP; Wang, F; Phan, J; Olejniczak, ET	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=423374	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=423374&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138470434	434149167							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
854177	CC(C)C(=O)N1CCCC(C1)C(=O)NC1CCc2ccc(cc12)-c1cn2CCCc2n1	InChI=1S/C25H32N4O2/c1-16(2)25(31)29-12-3-5-19(14-29)24(30)27-21-10-9-17-7-8-18(13-20(17)21)22-15-28-11-4-6-23(28)26-22/h7-8,13,15-16,19,21H,3-6,9-12,14H2,1-2H3,(H,27,30)	BSXACVXBICDKEQ-UHFFFAOYSA-N	423375	US10501466, Example B10	WD repeat-containing protein 5		 70.9								US Patent		10.7270/Q2319Z71		aid1804048	US10501466	Fesik, SW; Stauffer, SR; Salovich, JM; Tansey, WP; Wang, F; Phan, J; Olejniczak, ET	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=423375	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=423375&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138470447	434149168							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
854178	Clc1ccc(CC(=O)N[C@@H]2CCc3ccc(cc23)-c2cn3CCCc3n2)cc1Cl	InChI=1S/C23H21Cl2N3O/c24-18-7-3-14(10-19(18)25)11-23(29)27-20-8-6-15-4-5-16(12-17(15)20)21-13-28-9-1-2-22(28)26-21/h3-5,7,10,12-13,20H,1-2,6,8-9,11H2,(H,27,29)/t20-/m1/s1	HLGZWOPKLXYBFI-HXUWFJFHSA-N	50465585	CHEMBL4279907::US10501466, Example B11	WD repeat-containing protein 5		 2.66								US Patent		10.7270/Q2319Z71		aid1804048	US10501466	Fesik, SW; Stauffer, SR; Salovich, JM; Tansey, WP; Wang, F; Phan, J; Olejniczak, ET	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50465585	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50465585&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138470418	433932850							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
854179	COc1cc(ccc1C)C(=O)N[C@@H]1CCc2ccc(cc12)-c1cn2CCCc2n1	InChI=1S/C24H25N3O2/c1-15-5-6-18(13-22(15)29-2)24(28)26-20-10-9-16-7-8-17(12-19(16)20)21-14-27-11-3-4-23(27)25-21/h5-8,12-14,20H,3-4,9-11H2,1-2H3,(H,26,28)/t20-/m1/s1	PHINNLAJTUGZSZ-HXUWFJFHSA-N	423377	US10501466, Example B12	WD repeat-containing protein 5		 8.38								US Patent		10.7270/Q2319Z71		aid1804048	US10501466	Fesik, SW; Stauffer, SR; Salovich, JM; Tansey, WP; Wang, F; Phan, J; Olejniczak, ET	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=423377	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=423377&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	G2D	6DAS	137349382	434149170							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
854180	CC(=O)N1CCCC(C1)C(=O)N[C@@H]1CCc2ccc(cc12)-c1cn2CCCc2n1	InChI=1S/C23H28N4O2/c1-15(28)26-10-2-4-18(13-26)23(29)25-20-9-8-16-6-7-17(12-19(16)20)21-14-27-11-3-5-22(27)24-21/h6-7,12,14,18,20H,2-5,8-11,13H2,1H3,(H,25,29)/t18?,20-/m1/s1	BKBBJFFASFNPGD-ROPPNANJSA-N	423378	US10501466, Example B13	WD repeat-containing protein 5		 17.4								US Patent		10.7270/Q2319Z71		aid1804048	US10501466	Fesik, SW; Stauffer, SR; Salovich, JM; Tansey, WP; Wang, F; Phan, J; Olejniczak, ET	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=423378	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=423378&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138470398	434149171							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
854181	COc1cc(ccc1C)C(=O)N[C@@H]1CCCc2ccc(cc12)-c1cn2CCCc2n1	InChI=1S/C25H27N3O2/c1-16-8-9-19(14-23(16)30-2)25(29)27-21-6-3-5-17-10-11-18(13-20(17)21)22-15-28-12-4-7-24(28)26-22/h8-11,13-15,21H,3-7,12H2,1-2H3,(H,27,29)/t21-/m1/s1	HMOMQPHKMPWUKJ-OAQYLSRUSA-N	50465586	CHEMBL4294174::US10501466, Example B14	WD repeat-containing protein 5		 26.8								US Patent		10.7270/Q2319Z71		aid1804048	US10501466	Fesik, SW; Stauffer, SR; Salovich, JM; Tansey, WP; Wang, F; Phan, J; Olejniczak, ET	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50465586	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50465586&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138470399	433932851							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
854182	Fc1cc(CC(=O)N[C@@H]2CCc3ccc(cc23)-c2cn3CCCc3n2)ccc1Cl	InChI=1S/C23H21ClFN3O/c24-18-7-3-14(10-19(18)25)11-23(29)27-20-8-6-15-4-5-16(12-17(15)20)21-13-28-9-1-2-22(28)26-21/h3-5,7,10,12-13,20H,1-2,6,8-9,11H2,(H,27,29)/t20-/m1/s1	GGGPWQGUARQJME-HXUWFJFHSA-N	423380	US10501466, Example B15	WD repeat-containing protein 5		 2.37								US Patent		10.7270/Q2319Z71		aid1804048	US10501466	Fesik, SW; Stauffer, SR; Salovich, JM; Tansey, WP; Wang, F; Phan, J; Olejniczak, ET	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=423380	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=423380&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138470442	434149173							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
854183	CCC(=O)N1CCCC(C1)C(=O)N[C@@H]1CCc2ccc(cc12)-c1cn2CCCc2n1	InChI=1S/C24H30N4O2/c1-2-23(29)28-12-3-5-18(14-28)24(30)26-20-10-9-16-7-8-17(13-19(16)20)21-15-27-11-4-6-22(27)25-21/h7-8,13,15,18,20H,2-6,9-12,14H2,1H3,(H,26,30)/t18?,20-/m1/s1	NLYDZVTWTSGDDI-ROPPNANJSA-N	423381	US10501466, Example B16	WD repeat-containing protein 5		 7.16								US Patent		10.7270/Q2319Z71		aid1804048	US10501466	Fesik, SW; Stauffer, SR; Salovich, JM; Tansey, WP; Wang, F; Phan, J; Olejniczak, ET	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=423381	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=423381&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138470390	434149174							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
854184	CC(=O)N1CCCC(C1)C(=O)N[C@@H]1CCCc2ccc(cc12)-c1cn2CCCc2n1	InChI=1S/C24H30N4O2/c1-16(29)27-11-3-6-19(14-27)24(30)26-21-7-2-5-17-9-10-18(13-20(17)21)22-15-28-12-4-8-23(28)25-22/h9-10,13,15,19,21H,2-8,11-12,14H2,1H3,(H,26,30)/t19?,21-/m1/s1	YJLBZFIPBLITQN-VGAJERRHSA-N	423382	US10501466, Example B17	WD repeat-containing protein 5		 36.2								US Patent		10.7270/Q2319Z71		aid1804048	US10501466	Fesik, SW; Stauffer, SR; Salovich, JM; Tansey, WP; Wang, F; Phan, J; Olejniczak, ET	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=423382	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=423382&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138470403	434149175							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
854185	CCC(=O)N1CCCC(C1)C(=O)N[C@@H]1CCCc2ccc(cc12)-c1cn2CCCc2n1	InChI=1S/C25H32N4O2/c1-2-24(30)29-13-4-7-19(15-29)25(31)27-21-8-3-6-17-10-11-18(14-20(17)21)22-16-28-12-5-9-23(28)26-22/h10-11,14,16,19,21H,2-9,12-13,15H2,1H3,(H,27,31)/t19?,21-/m1/s1	KKYMBAIJDZSLOJ-VGAJERRHSA-N	423383	US10501466, Example B18	WD repeat-containing protein 5		 14.3								US Patent		10.7270/Q2319Z71		aid1804048	US10501466	Fesik, SW; Stauffer, SR; Salovich, JM; Tansey, WP; Wang, F; Phan, J; Olejniczak, ET	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=423383	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=423383&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138470412	434149176							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
854186	COc1ccc(cn1)C(=O)N[C@@H]1CCc2ccc(cc12)-c1cn2CCCc2n1	InChI=1S/C22H22N4O2/c1-28-21-9-7-16(12-23-21)22(27)25-18-8-6-14-4-5-15(11-17(14)18)19-13-26-10-2-3-20(26)24-19/h4-5,7,9,11-13,18H,2-3,6,8,10H2,1H3,(H,25,27)/t18-/m1/s1	JHBFXUUQTVMGDD-GOSISDBHSA-N	423384	US10501466, Example B19	WD repeat-containing protein 5		 172								US Patent		10.7270/Q2319Z71		aid1804048	US10501466	Fesik, SW; Stauffer, SR; Salovich, JM; Tansey, WP; Wang, F; Phan, J; Olejniczak, ET	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=423384	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=423384&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138470419	434149177							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
854187	Clc1cc(ccn1)C(=O)N[C@@H]1CCc2ccc(cc12)-c1cn2CCCc2n1	InChI=1S/C21H19ClN4O/c22-19-11-15(7-8-23-19)21(27)25-17-6-5-13-3-4-14(10-16(13)17)18-12-26-9-1-2-20(26)24-18/h3-4,7-8,10-12,17H,1-2,5-6,9H2,(H,25,27)/t17-/m1/s1	JNYVXUXMJYRFJD-QGZVFWFLSA-N	423385	US10501466, Example B20	WD repeat-containing protein 5		 95.6								US Patent		10.7270/Q2319Z71		aid1804048	US10501466	Fesik, SW; Stauffer, SR; Salovich, JM; Tansey, WP; Wang, F; Phan, J; Olejniczak, ET	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=423385	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=423385&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138470413	434149178							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
854188	Cc1cnc(Cl)c(c1)C(=O)N[C@@H]1CCc2ccc(cc12)-c1cn2CCCc2n1	InChI=1S/C22H21ClN4O/c1-13-9-17(21(23)24-11-13)22(28)26-18-7-6-14-4-5-15(10-16(14)18)19-12-27-8-2-3-20(27)25-19/h4-5,9-12,18H,2-3,6-8H2,1H3,(H,26,28)/t18-/m1/s1	KOKZZJAMDJWEFM-GOSISDBHSA-N	423386	US10501466, Example B21	WD repeat-containing protein 5		 22.9								US Patent		10.7270/Q2319Z71		aid1804048	US10501466	Fesik, SW; Stauffer, SR; Salovich, JM; Tansey, WP; Wang, F; Phan, J; Olejniczak, ET	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=423386	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=423386&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138470430	434149179							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
854189	Cc1cc(cc(=O)[nH]1)C(=O)N[C@@H]1CCc2ccc(cc12)-c1cn2CCCc2n1			423387	US10501466, Example B22	WD repeat-containing protein 5		 426								US Patent		10.7270/Q2319Z71		aid1804048	US10501466	Fesik, SW; Stauffer, SR; Salovich, JM; Tansey, WP; Wang, F; Phan, J; Olejniczak, ET	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=423387	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=423387&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			154702358	434149180							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
854190	Cc1cc(Cl)nc(c1)C(=O)N[C@@H]1CCc2ccc(cc12)-c1cn2CCCc2n1	InChI=1S/C22H21ClN4O/c1-13-9-18(24-20(23)10-13)22(28)26-17-7-6-14-4-5-15(11-16(14)17)19-12-27-8-2-3-21(27)25-19/h4-5,9-12,17H,2-3,6-8H2,1H3,(H,26,28)/t17-/m1/s1	JLEPAWFWJUFHPA-QGZVFWFLSA-N	423388	US10501466, Example B23	WD repeat-containing protein 5		 769								US Patent		10.7270/Q2319Z71		aid1804048	US10501466	Fesik, SW; Stauffer, SR; Salovich, JM; Tansey, WP; Wang, F; Phan, J; Olejniczak, ET	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=423388	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=423388&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138470421	434149181							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
854191	Cc1cc(ccn1)C(=O)N[C@@H]1CCc2ccc(cc12)-c1cn2CCCc2n1	InChI=1S/C22H22N4O/c1-14-11-17(8-9-23-14)22(27)25-19-7-6-15-4-5-16(12-18(15)19)20-13-26-10-2-3-21(26)24-20/h4-5,8-9,11-13,19H,2-3,6-7,10H2,1H3,(H,25,27)/t19-/m1/s1	YKUGUWMZBHIDFR-LJQANCHMSA-N	50465594	CHEMBL4284408::US10501466, Example B24	WD repeat-containing protein 5		 33.0								US Patent		10.7270/Q2319Z71		aid1804048	US10501466	Fesik, SW; Stauffer, SR; Salovich, JM; Tansey, WP; Wang, F; Phan, J; Olejniczak, ET	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50465594	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50465594&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138470404	433932859							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
854192	Cc1ccc(cc1O)C(=O)N[C@@H]1CCc2ccc(cc12)-c1cn2CCCc2n1	InChI=1S/C23H23N3O2/c1-14-4-5-17(12-21(14)27)23(28)25-19-9-8-15-6-7-16(11-18(15)19)20-13-26-10-2-3-22(26)24-20/h4-7,11-13,19,27H,2-3,8-10H2,1H3,(H,25,28)/t19-/m1/s1	YEQJXZRAEIPGPE-LJQANCHMSA-N	423390	US10501466, Example B25	WD repeat-containing protein 5		 710								US Patent		10.7270/Q2319Z71		aid1804048	US10501466	Fesik, SW; Stauffer, SR; Salovich, JM; Tansey, WP; Wang, F; Phan, J; Olejniczak, ET	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=423390	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=423390&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138470443	434149183							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
854193	COc1cncc(c1)C(=O)N[C@@H]1CCc2ccc(cc12)-c1cn2CCCc2n1	InChI=1S/C22H22N4O2/c1-28-17-9-16(11-23-12-17)22(27)25-19-7-6-14-4-5-15(10-18(14)19)20-13-26-8-2-3-21(26)24-20/h4-5,9-13,19H,2-3,6-8H2,1H3,(H,25,27)/t19-/m1/s1	FFQMCFOEUABQDI-LJQANCHMSA-N	423391	US10501466, Example B26	WD repeat-containing protein 5		 18.5								US Patent		10.7270/Q2319Z71		aid1804048	US10501466	Fesik, SW; Stauffer, SR; Salovich, JM; Tansey, WP; Wang, F; Phan, J; Olejniczak, ET	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=423391	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=423391&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138470438	434149184							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
854194	CC(=O)Nc1cc(ccc1C)C(=O)N[C@@H]1CCc2ccc(cc12)-c1cn2CCCc2n1	InChI=1S/C25H26N4O2/c1-15-5-6-19(13-22(15)26-16(2)30)25(31)28-21-10-9-17-7-8-18(12-20(17)21)23-14-29-11-3-4-24(29)27-23/h5-8,12-14,21H,3-4,9-11H2,1-2H3,(H,26,30)(H,28,31)/t21-/m1/s1	CGNCXJAPEYAQOP-OAQYLSRUSA-N	423392	US10501466, Example B27	WD repeat-containing protein 5		 730								US Patent		10.7270/Q2319Z71		aid1804048	US10501466	Fesik, SW; Stauffer, SR; Salovich, JM; Tansey, WP; Wang, F; Phan, J; Olejniczak, ET	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=423392	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=423392&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138470384	434149185							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
854195	Cc1ccc(C(=O)N[C@@H]2CCc3ccc(cc23)-c2cn3CCCc3n2)c(Cl)n1	InChI=1S/C22H21ClN4O/c1-13-4-8-16(21(23)24-13)22(28)26-18-9-7-14-5-6-15(11-17(14)18)19-12-27-10-2-3-20(27)25-19/h4-6,8,11-12,18H,2-3,7,9-10H2,1H3,(H,26,28)/t18-/m1/s1	ATDHZYGGNBFPOC-GOSISDBHSA-N	423393	US10501466, Example B28	WD repeat-containing protein 5		 169								US Patent		10.7270/Q2319Z71		aid1804048	US10501466	Fesik, SW; Stauffer, SR; Salovich, JM; Tansey, WP; Wang, F; Phan, J; Olejniczak, ET	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=423393	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=423393&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138470401	434149186							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
854196	COc1cc(cc(OC)c1C)C(=O)N[C@@H]1CCc2ccc(cc12)-c1cn2CCCc2n1	InChI=1S/C25H27N3O3/c1-15-22(30-2)12-18(13-23(15)31-3)25(29)27-20-9-8-16-6-7-17(11-19(16)20)21-14-28-10-4-5-24(28)26-21/h6-7,11-14,20H,4-5,8-10H2,1-3H3,(H,27,29)/t20-/m1/s1	GRFBFSARRYJWSN-HXUWFJFHSA-N	50465552	CHEMBL4291641::US10501466, Example B29	WD repeat-containing protein 5		 0.902								US Patent		10.7270/Q2319Z71		aid1804048	US10501466	Fesik, SW; Stauffer, SR; Salovich, JM; Tansey, WP; Wang, F; Phan, J; Olejniczak, ET	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50465552	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50465552&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138470423	433932817							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
854197	Fc1cnccc1C(=O)N[C@@H]1CCc2ccc(cc12)-c1cn2CCCc2n1	InChI=1S/C21H19FN4O/c22-17-11-23-8-7-15(17)21(27)25-18-6-5-13-3-4-14(10-16(13)18)19-12-26-9-1-2-20(26)24-19/h3-4,7-8,10-12,18H,1-2,5-6,9H2,(H,25,27)/t18-/m1/s1	OSBWPKZUGXXQDV-GOSISDBHSA-N	423395	US10501466, Example B30	WD repeat-containing protein 5		 3750								US Patent		10.7270/Q2319Z71		aid1804048	US10501466	Fesik, SW; Stauffer, SR; Salovich, JM; Tansey, WP; Wang, F; Phan, J; Olejniczak, ET	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=423395	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=423395&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138470396	434149188							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
854198	O=C(N[C@@H]1CCc2ccc(cc12)-c1cn2CCCc2n1)c1ccc(=O)[nH]c1			423396	US10501466, Example B31	WD repeat-containing protein 5		 835								US Patent		10.7270/Q2319Z71		aid1804048	US10501466	Fesik, SW; Stauffer, SR; Salovich, JM; Tansey, WP; Wang, F; Phan, J; Olejniczak, ET	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=423396	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=423396&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			154702359	434149189							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
854199	Fc1cncc(c1)C(=O)N[C@@H]1CCc2ccc(cc12)-c1cn2CCCc2n1	InChI=1S/C21H19FN4O/c22-16-8-15(10-23-11-16)21(27)25-18-6-5-13-3-4-14(9-17(13)18)19-12-26-7-1-2-20(26)24-19/h3-4,8-12,18H,1-2,5-7H2,(H,25,27)/t18-/m1/s1	RRZCKOOFKYVOEI-GOSISDBHSA-N	423397	US10501466, Example B32	WD repeat-containing protein 5		 568								US Patent		10.7270/Q2319Z71		aid1804048	US10501466	Fesik, SW; Stauffer, SR; Salovich, JM; Tansey, WP; Wang, F; Phan, J; Olejniczak, ET	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=423397	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=423397&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138470415	434149190							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
854200	COc1cc(ccc1C)C(=O)N[C@@H]1CCN(C(C)=O)c2ccc(cc12)-c1cn2CCCc2n1	InChI=1S/C26H28N4O3/c1-16-6-7-19(14-24(16)33-3)26(32)28-21-10-12-30(17(2)31)23-9-8-18(13-20(21)23)22-15-29-11-4-5-25(29)27-22/h6-9,13-15,21H,4-5,10-12H2,1-3H3,(H,28,32)/t21-/m1/s1	SVURARXEASTTAN-OAQYLSRUSA-N	423398	US10501466, Example B33	WD repeat-containing protein 5		 22.2								US Patent		10.7270/Q2319Z71		aid1804048	US10501466	Fesik, SW; Stauffer, SR; Salovich, JM; Tansey, WP; Wang, F; Phan, J; Olejniczak, ET	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=423398	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=423398&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138470435	434149191							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51242559	Cn1c(c(C2N(CC(O)=O)C(=O)c3ccccc23)c2ccccc12)-c1ccc(F)cc1	InChI=1S/C25H19FN2O3/c1-27-20-9-5-4-8-19(20)22(23(27)15-10-12-16(26)13-11-15)24-17-6-2-3-7-18(17)25(31)28(24)14-21(29)30/h2-13,24H,14H2,1H3,(H,29,30)	OCOHWMKYWBSCIV-UHFFFAOYSA-N	50508566	CHEMBL4435755	WD repeat-containing protein 5			 24000							ChEMBL	10.1016/j.bmcl.2018.12.035	10.7270/Q26W9FC5	30626558			Ye, X; Zhang, R; Lian, F; Zhang, W; Lu, W; Han, J; Zhang, N; Jin, J; Luo, C; Chen, K; Ye, F; Ding, H	Zhejiang Sci-Tech University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50508566	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50508566&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			16483718	440717151							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51242560	OC(=O)c1cc(NS(=O)(=O)c2ccc(Cl)cc2)cc(c1)C(O)=O	InChI=1S/C14H10ClNO6S/c15-10-1-3-12(4-2-10)23(21,22)16-11-6-8(13(17)18)5-9(7-11)14(19)20/h1-7,16H,(H,17,18)(H,19,20)	XNUMMVFWNYQDKB-UHFFFAOYSA-N	50508567	CHEMBL4578737	WD repeat-containing protein 5			 22000							ChEMBL	10.1016/j.bmcl.2018.12.035	10.7270/Q26W9FC5	30626558			Ye, X; Zhang, R; Lian, F; Zhang, W; Lu, W; Han, J; Zhang, N; Jin, J; Luo, C; Chen, K; Ye, F; Ding, H	Zhejiang Sci-Tech University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50508567	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50508567&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			1025961	440717152							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51242561	OC(=O)COc1ccc(Br)cc1C1C2=C(CCCC2=O)NC2=C1C(=O)CCC2	InChI=1S/C21H20BrNO5/c22-11-7-8-17(28-10-18(26)27)12(9-11)19-20-13(3-1-5-15(20)24)23-14-4-2-6-16(25)21(14)19/h7-9,19,23H,1-6,10H2,(H,26,27)	PDRDJMMDVAHCEE-UHFFFAOYSA-N	50508568	CHEMBL4474886	WD repeat-containing protein 5				 13800						ChEMBL	10.1016/j.bmcl.2018.12.035	10.7270/Q26W9FC5	30626558			Ye, X; Zhang, R; Lian, F; Zhang, W; Lu, W; Han, J; Zhang, N; Jin, J; Luo, C; Chen, K; Ye, F; Ding, H	Zhejiang Sci-Tech University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50508568	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50508568&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			1006833	440717153							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51242562	CCC(CC)(NC(=O)C(C)C)C(=O)N[C@@H](CCCNC(N)=N)C(=O)NC1(CCCC1)C(=O)NC(c1ccc(Cl)cc1)c1ccc(Cl)cc1	InChI=1S/C35H49Cl2N7O4/c1-5-34(6-2,43-29(45)22(3)4)31(47)41-27(10-9-21-40-33(38)39)30(46)44-35(19-7-8-20-35)32(48)42-28(23-11-15-25(36)16-12-23)24-13-17-26(37)18-14-24/h11-18,22,27-28H,5-10,19-21H2,1-4H3,(H,41,47)(H,42,48)(H,43,45)(H,44,46)(H4,38,39,40)/t27-/m0/s1	PTJOIPPVAWDZSV-MHZLTWQESA-N	200722	US9233086, 10K	WD repeat-containing protein 5		<1.000000								ChEMBL	10.1016/j.bmcl.2018.12.035	10.7270/Q26W9FC5	30626558			Ye, X; Zhang, R; Lian, F; Zhang, W; Lu, W; Han, J; Zhang, N; Jin, J; Luo, C; Chen, K; Ye, F; Ding, H	Zhejiang Sci-Tech University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=200722	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=200722&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			54766612	318834335							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51242563	CCC(CC)(NC(=O)C(C)C)C(=O)N[C@@H](CCCNC(N)=N)C(=O)NC1(CCCC1)C(=O)NC(c1ccc(F)cc1)c1ccc(F)cc1	InChI=1S/C35H49F2N7O4/c1-5-34(6-2,43-29(45)22(3)4)31(47)41-27(10-9-21-40-33(38)39)30(46)44-35(19-7-8-20-35)32(48)42-28(23-11-15-25(36)16-12-23)24-13-17-26(37)18-14-24/h11-18,22,27-28H,5-10,19-21H2,1-4H3,(H,41,47)(H,42,48)(H,43,45)(H,44,46)(H4,38,39,40)/t27-/m0/s1	RZKSQRIPRKWVBU-MHZLTWQESA-N	200723	US9233086, 10L	WD repeat-containing protein 5		<1.000000								ChEMBL	10.1016/j.bmcl.2018.12.035	10.7270/Q26W9FC5	30626558			Ye, X; Zhang, R; Lian, F; Zhang, W; Lu, W; Han, J; Zhang, N; Jin, J; Luo, C; Chen, K; Ye, F; Ding, H	Zhejiang Sci-Tech University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=200723	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=200723&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			54766613	318834336							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51242564	CCC(CC)(NC(=O)C(C)C)C(=O)N[C@@H](CCCNC(N)=N)C(=O)NC1(CCCC1)C(=O)NC(c1ccc(Cl)cc1)c1ccc(Cl)cc1	InChI=1S/C35H49Cl2N7O4/c1-5-34(6-2,43-29(45)22(3)4)31(47)41-27(10-9-21-40-33(38)39)30(46)44-35(19-7-8-20-35)32(48)42-28(23-11-15-25(36)16-12-23)24-13-17-26(37)18-14-24/h11-18,22,27-28H,5-10,19-21H2,1-4H3,(H,41,47)(H,42,48)(H,43,45)(H,44,46)(H4,38,39,40)/t27-/m0/s1	PTJOIPPVAWDZSV-MHZLTWQESA-N	200722	US9233086, 10K	WD repeat-containing protein 5			 4.5							ChEMBL	10.1016/j.bmcl.2018.12.035	10.7270/Q26W9FC5	30626558			Ye, X; Zhang, R; Lian, F; Zhang, W; Lu, W; Han, J; Zhang, N; Jin, J; Luo, C; Chen, K; Ye, F; Ding, H	Zhejiang Sci-Tech University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=200722	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=200722&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			54766612	318834335							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51242565	CCC(CC)(NC(=O)C(C)C)C(=O)N[C@@H](CCCNC(N)=N)C(=O)NC1(CCCC1)C(=O)NC(c1ccccc1)c1ccccc1	InChI=1S/C35H51N7O4/c1-5-34(6-2,41-29(43)24(3)4)31(45)39-27(20-15-23-38-33(36)37)30(44)42-35(21-13-14-22-35)32(46)40-28(25-16-9-7-10-17-25)26-18-11-8-12-19-26/h7-12,16-19,24,27-28H,5-6,13-15,20-23H2,1-4H3,(H,39,45)(H,40,46)(H,41,43)(H,42,44)(H4,36,37,38)/t27-/m0/s1	BCIPILGGOSCOMC-MHZLTWQESA-N	200712	US9233086, 10A	WD repeat-containing protein 5			 2.9							ChEMBL	10.1016/j.bmcl.2018.12.035	10.7270/Q26W9FC5	30626558			Ye, X; Zhang, R; Lian, F; Zhang, W; Lu, W; Han, J; Zhang, N; Jin, J; Luo, C; Chen, K; Ye, F; Ding, H	Zhejiang Sci-Tech University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=200712	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=200712&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			53356803	318834325							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51242569	CN1C2=C(C(C3=C1CCCC3=O)c1cc(Br)cc(Br)c1OCC(O)=O)C(=O)CCC2	InChI=1S/C22H21Br2NO5/c1-25-14-4-2-6-16(26)20(14)19(21-15(25)5-3-7-17(21)27)12-8-11(23)9-13(24)22(12)30-10-18(28)29/h8-9,19H,2-7,10H2,1H3,(H,28,29)	FTNCWZXKFRDDIM-UHFFFAOYSA-N	50508570	CHEMBL4534707	WD repeat-containing protein 5			 25000							ChEMBL	10.1016/j.bmcl.2018.12.035	10.7270/Q26W9FC5	30626558			Ye, X; Zhang, R; Lian, F; Zhang, W; Lu, W; Han, J; Zhang, N; Jin, J; Luo, C; Chen, K; Ye, F; Ding, H	Zhejiang Sci-Tech University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50508570	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50508570&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			1006789	440717155							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51242570	OC(=O)COc1ccc(Br)cc1C1C2=C(CCCC2=O)NC2=C1C(=O)CCC2	InChI=1S/C21H20BrNO5/c22-11-7-8-17(28-10-18(26)27)12(9-11)19-20-13(3-1-5-15(20)24)23-14-4-2-6-16(25)21(14)19/h7-9,19,23H,1-6,10H2,(H,26,27)	PDRDJMMDVAHCEE-UHFFFAOYSA-N	50508568	CHEMBL4474886	WD repeat-containing protein 5			 9630							ChEMBL	10.1016/j.bmcl.2018.12.035	10.7270/Q26W9FC5	30626558			Ye, X; Zhang, R; Lian, F; Zhang, W; Lu, W; Han, J; Zhang, N; Jin, J; Luo, C; Chen, K; Ye, F; Ding, H	Zhejiang Sci-Tech University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50508568	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50508568&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			1006833	440717153							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51242571	CN1C2=C(C(C3=C1CCCC3=O)c1cc(Cl)ccc1OCC(O)=O)C(=O)CCC2	InChI=1S/C22H22ClNO5/c1-24-14-4-2-6-16(25)21(14)20(22-15(24)5-3-7-17(22)26)13-10-12(23)8-9-18(13)29-11-19(27)28/h8-10,20H,2-7,11H2,1H3,(H,27,28)	OJWNDLQTNXZWHJ-UHFFFAOYSA-N	50508571	CHEMBL4469769	WD repeat-containing protein 5			 24000							ChEMBL	10.1016/j.bmcl.2018.12.035	10.7270/Q26W9FC5	30626558			Ye, X; Zhang, R; Lian, F; Zhang, W; Lu, W; Han, J; Zhang, N; Jin, J; Luo, C; Chen, K; Ye, F; Ding, H	Zhejiang Sci-Tech University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50508571	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50508571&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			1006808	440717156							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51242572	OC(=O)c1cccc(NS(=O)(=O)c2ccc(Cl)c3ccccc23)c1	InChI=1S/C17H12ClNO4S/c18-15-8-9-16(14-7-2-1-6-13(14)15)24(22,23)19-12-5-3-4-11(10-12)17(20)21/h1-10,19H,(H,20,21)	KULMRMPKELUUKN-UHFFFAOYSA-N	50508572	CHEMBL4514062	WD repeat-containing protein 5			 23000							ChEMBL	10.1016/j.bmcl.2018.12.035	10.7270/Q26W9FC5	30626558			Ye, X; Zhang, R; Lian, F; Zhang, W; Lu, W; Han, J; Zhang, N; Jin, J; Luo, C; Chen, K; Ye, F; Ding, H	Zhejiang Sci-Tech University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50508572	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50508572&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			39845125	440717157							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51242573	CCCCOc1ccc(cc1C)S(=O)(=O)Nc1cccc(c1)C(O)=O	InChI=1S/C18H21NO5S/c1-3-4-10-24-17-9-8-16(11-13(17)2)25(22,23)19-15-7-5-6-14(12-15)18(20)21/h5-9,11-12,19H,3-4,10H2,1-2H3,(H,20,21)	GWCWFDSPSQQCSU-UHFFFAOYSA-N	50508573	CHEMBL4455781	WD repeat-containing protein 5			 30000							ChEMBL	10.1016/j.bmcl.2018.12.035	10.7270/Q26W9FC5	30626558			Ye, X; Zhang, R; Lian, F; Zhang, W; Lu, W; Han, J; Zhang, N; Jin, J; Luo, C; Chen, K; Ye, F; Ding, H	Zhejiang Sci-Tech University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50508573	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50508573&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			16645215	440717158							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51242574	CCCCOc1ccc(cc1C)S(=O)(=O)Nc1ccc(cc1)C(O)=O	InChI=1S/C18H21NO5S/c1-3-4-11-24-17-10-9-16(12-13(17)2)25(22,23)19-15-7-5-14(6-8-15)18(20)21/h5-10,12,19H,3-4,11H2,1-2H3,(H,20,21)	PYEVWZHTBYTQQI-UHFFFAOYSA-N	50508569	CHEMBL4557353	WD repeat-containing protein 5			 12970							ChEMBL	10.1016/j.bmcl.2018.12.035	10.7270/Q26W9FC5	30626558			Ye, X; Zhang, R; Lian, F; Zhang, W; Lu, W; Han, J; Zhang, N; Jin, J; Luo, C; Chen, K; Ye, F; Ding, H	Zhejiang Sci-Tech University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50508569	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50508569&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			16645216	440717154							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51242575	CN1C2=C(C(C3=C1CCCC3=O)c1cc(Br)ccc1OCC(O)=O)C(=O)CCC2	InChI=1S/C22H22BrNO5/c1-24-14-4-2-6-16(25)21(14)20(22-15(24)5-3-7-17(22)26)13-10-12(23)8-9-18(13)29-11-19(27)28/h8-10,20H,2-7,11H2,1H3,(H,27,28)	FILGLJILLSAIJW-UHFFFAOYSA-N	50508574	CHEMBL4435564	WD repeat-containing protein 5			 13620							ChEMBL	10.1016/j.bmcl.2018.12.035	10.7270/Q26W9FC5	30626558			Ye, X; Zhang, R; Lian, F; Zhang, W; Lu, W; Han, J; Zhang, N; Jin, J; Luo, C; Chen, K; Ye, F; Ding, H	Zhejiang Sci-Tech University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50508574	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50508574&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			1006800	440717159							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51242576	CCC(CC)(NC(=O)C(C)C)C(=O)N[C@@H](CCCNC(N)=N)C(=O)NC1(CCCC1)C(=O)NC(c1ccccc1)c1ccccc1	InChI=1S/C35H51N7O4/c1-5-34(6-2,41-29(43)24(3)4)31(45)39-27(20-15-23-38-33(36)37)30(44)42-35(21-13-14-22-35)32(46)40-28(25-16-9-7-10-17-25)26-18-11-8-12-19-26/h7-12,16-19,24,27-28H,5-6,13-15,20-23H2,1-4H3,(H,39,45)(H,40,46)(H,41,43)(H,42,44)(H4,36,37,38)/t27-/m0/s1	BCIPILGGOSCOMC-MHZLTWQESA-N	200712	US9233086, 10A	WD repeat-containing protein 5		<1.000000								ChEMBL	10.1016/j.bmcl.2018.12.035	10.7270/Q26W9FC5	30626558			Ye, X; Zhang, R; Lian, F; Zhang, W; Lu, W; Han, J; Zhang, N; Jin, J; Luo, C; Chen, K; Ye, F; Ding, H	Zhejiang Sci-Tech University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=200712	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=200712&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			53356803	318834325							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51242578	Cc1c(Cl)ccc(c1Cl)S(=O)(=O)Nc1cccc(c1)C(O)=O	InChI=1S/C14H11Cl2NO4S/c1-8-11(15)5-6-12(13(8)16)22(20,21)17-10-4-2-3-9(7-10)14(18)19/h2-7,17H,1H3,(H,18,19)	PZLKNWTZRUVXIL-UHFFFAOYSA-N	50508575	CHEMBL4464601	WD repeat-containing protein 5			 13000							ChEMBL	10.1016/j.bmcl.2018.12.035	10.7270/Q26W9FC5	30626558			Ye, X; Zhang, R; Lian, F; Zhang, W; Lu, W; Han, J; Zhang, N; Jin, J; Luo, C; Chen, K; Ye, F; Ding, H	Zhejiang Sci-Tech University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50508575	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50508575&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			39845172	440717160							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51242579	CC[C@@H]1NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@@](C)(CCCCNC(=O)[C@H](NC1=O)c1ccccc1)NC(=O)C(C)C	InChI=1S/C29H46N8O5/c1-5-20-24(39)36-22(19-12-7-6-8-13-19)26(41)32-16-10-9-15-29(4,37-23(38)18(2)3)27(42)35-21(25(40)34-20)14-11-17-33-28(30)31/h6-8,12-13,18,20-22H,5,9-11,14-17H2,1-4H3,(H,32,41)(H,34,40)(H,35,42)(H,36,39)(H,37,38)(H4,30,31,33)/t20-,21-,22+,29+/m0/s1	SILRGLDFBXVGOQ-ZMROOPMESA-N	50164787	CHEMBL3798088	WD repeat-containing protein 5			 0.900000							ChEMBL	10.1016/j.bmcl.2018.12.035	10.7270/Q26W9FC5	30626558			Ye, X; Zhang, R; Lian, F; Zhang, W; Lu, W; Han, J; Zhang, N; Jin, J; Luo, C; Chen, K; Ye, F; Ding, H	Zhejiang Sci-Tech University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50164787	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50164787&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			71586081	341097532		CHEMBL3798088					1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51242580	CCCCOc1ccc(cc1C)S(=O)(=O)Nc1ccc(cc1)C(O)=O	InChI=1S/C18H21NO5S/c1-3-4-11-24-17-10-9-16(12-13(17)2)25(22,23)19-15-7-5-14(6-8-15)18(20)21/h5-10,12,19H,3-4,11H2,1-2H3,(H,20,21)	PYEVWZHTBYTQQI-UHFFFAOYSA-N	50508569	CHEMBL4557353	WD repeat-containing protein 5				 15800						ChEMBL	10.1016/j.bmcl.2018.12.035	10.7270/Q26W9FC5	30626558			Ye, X; Zhang, R; Lian, F; Zhang, W; Lu, W; Han, J; Zhang, N; Jin, J; Luo, C; Chen, K; Ye, F; Ding, H	Zhejiang Sci-Tech University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50508569	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50508569&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			16645216	440717154							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51242581	COc1cccc(c1)-c1[nH]c2ccccc2c1C1N(CC(O)=O)C(=O)c2ccccc12	InChI=1S/C25H20N2O4/c1-31-16-8-6-7-15(13-16)23-22(19-11-4-5-12-20(19)26-23)24-17-9-2-3-10-18(17)25(30)27(24)14-21(28)29/h2-13,24,26H,14H2,1H3,(H,28,29)	CTNRDFOTOJCFMD-UHFFFAOYSA-N	50508576	CHEMBL4449119	WD repeat-containing protein 5			 22000							ChEMBL	10.1016/j.bmcl.2018.12.035	10.7270/Q26W9FC5	30626558			Ye, X; Zhang, R; Lian, F; Zhang, W; Lu, W; Han, J; Zhang, N; Jin, J; Luo, C; Chen, K; Ye, F; Ding, H	Zhejiang Sci-Tech University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50508576	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50508576&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			16487351	440717161							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51242582	COc1ccc(cc1C(C)(C)C)S(=O)(=O)Nc1ccc(cc1)C(O)=O	InChI=1S/C18H21NO5S/c1-18(2,3)15-11-14(9-10-16(15)24-4)25(22,23)19-13-7-5-12(6-8-13)17(20)21/h5-11,19H,1-4H3,(H,20,21)	MFQXNLCWGLUVFN-UHFFFAOYSA-N	50508577	CHEMBL4452985	WD repeat-containing protein 5			 48000							ChEMBL	10.1016/j.bmcl.2018.12.035	10.7270/Q26W9FC5	30626558			Ye, X; Zhang, R; Lian, F; Zhang, W; Lu, W; Han, J; Zhang, N; Jin, J; Luo, C; Chen, K; Ye, F; Ding, H	Zhejiang Sci-Tech University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50508577	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50508577&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			39845054	440717162							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51242583	CCCCOc1ccc(cc1C)S(=O)(=O)Nc1ccccc1C(O)=O	InChI=1S/C18H21NO5S/c1-3-4-11-24-17-10-9-14(12-13(17)2)25(22,23)19-16-8-6-5-7-15(16)18(20)21/h5-10,12,19H,3-4,11H2,1-2H3,(H,20,21)	KTAWOZGYMMJCRD-UHFFFAOYSA-N	50508578	CHEMBL4579304	WD repeat-containing protein 5			 22000							ChEMBL	10.1016/j.bmcl.2018.12.035	10.7270/Q26W9FC5	30626558			Ye, X; Zhang, R; Lian, F; Zhang, W; Lu, W; Han, J; Zhang, N; Jin, J; Luo, C; Chen, K; Ye, F; Ding, H	Zhejiang Sci-Tech University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50508578	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50508578&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			16645214	440717163							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51242584	CCC(CC)(NC(=O)C(C)C)C(=O)N[C@@H](CCCNC(N)=N)C(=O)NC1(CCCC1)C(=O)NC(c1ccc(F)cc1)c1ccc(F)cc1	InChI=1S/C35H49F2N7O4/c1-5-34(6-2,43-29(45)22(3)4)31(47)41-27(10-9-21-40-33(38)39)30(46)44-35(19-7-8-20-35)32(48)42-28(23-11-15-25(36)16-12-23)24-13-17-26(37)18-14-24/h11-18,22,27-28H,5-10,19-21H2,1-4H3,(H,41,47)(H,42,48)(H,43,45)(H,44,46)(H4,38,39,40)/t27-/m0/s1	RZKSQRIPRKWVBU-MHZLTWQESA-N	200723	US9233086, 10L	WD repeat-containing protein 5			 2.4							ChEMBL	10.1016/j.bmcl.2018.12.035	10.7270/Q26W9FC5	30626558			Ye, X; Zhang, R; Lian, F; Zhang, W; Lu, W; Han, J; Zhang, N; Jin, J; Luo, C; Chen, K; Ye, F; Ding, H	Zhejiang Sci-Tech University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=200723	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=200723&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			54766613	318834336							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51242585	OC(=O)c1ccc(NS(=O)(=O)c2cc(C(=O)Nc3ccccc3)c(Cl)cc2Cl)cc1	InChI=1S/C20H14Cl2N2O5S/c21-16-11-17(22)18(10-15(16)19(25)23-13-4-2-1-3-5-13)30(28,29)24-14-8-6-12(7-9-14)20(26)27/h1-11,24H,(H,23,25)(H,26,27)	ZRQJVMRJBGWMRM-UHFFFAOYSA-N	50508579	CHEMBL4453261	WD repeat-containing protein 5			 38000							ChEMBL	10.1016/j.bmcl.2018.12.035	10.7270/Q26W9FC5	30626558			Ye, X; Zhang, R; Lian, F; Zhang, W; Lu, W; Han, J; Zhang, N; Jin, J; Luo, C; Chen, K; Ye, F; Ding, H	Zhejiang Sci-Tech University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50508579	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50508579&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			1266319	440717164							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51242586	CCN1C2=C(C(C3=C1CCCC3=O)c1cc(Br)ccc1OCC(O)=O)C(=O)CCC2	InChI=1S/C23H24BrNO5/c1-2-25-15-5-3-7-17(26)22(15)21(23-16(25)6-4-8-18(23)27)14-11-13(24)9-10-19(14)30-12-20(28)29/h9-11,21H,2-8,12H2,1H3,(H,28,29)	ADAUAVVRTHYGGG-UHFFFAOYSA-N	50508580	CHEMBL4557413	WD repeat-containing protein 5			 22000							ChEMBL	10.1016/j.bmcl.2018.12.035	10.7270/Q26W9FC5	30626558			Ye, X; Zhang, R; Lian, F; Zhang, W; Lu, W; Han, J; Zhang, N; Jin, J; Luo, C; Chen, K; Ye, F; Ding, H	Zhejiang Sci-Tech University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50508580	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50508580&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			1006856	440717165							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51274353	Cc1cc(CN2CCc3c(cc(Cn4ccn(C)c4=N)cc3-c3ccc(F)cc3C)C2=O)ccc1Cl	InChI=1S/C29H28ClFN4O/c1-18-13-22(31)5-6-23(18)25-14-21(17-35-11-10-33(3)29(35)32)15-26-24(25)8-9-34(28(26)36)16-20-4-7-27(30)19(2)12-20/h4-7,10-15,32H,8-9,16-17H2,1-3H3	HNKHSIKLIGVXPW-UHFFFAOYSA-N	50520120	CHEMBL4476662	WD repeat-containing protein 5				 0.027000						ChEMBL	10.1021/acs.jmedchem.9b01608	10.7270/Q2HD801W	31858797			Tian, J; Teuscher, KB; Aho, ER; Alvarado, JR; Mills, JJ; Meyers, KM; Gogliotti, RD; Han, C; Macdonald, JD; Sai, J; Shaw, JG; Sensintaffar, JL; Zhao, B; Rietz, TA; Thomas, LR; Payne, WG; Moore, WJ; Stott, GM; Kondo, J; Inoue, M; Coffey, RJ; Tansey, WP; Stauffer, SR; Lee, T; Fesik, SW	Frederick National Laboratory for Cancer Research	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50520120	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50520120&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			153572631	440728702							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51274354	Cc1nc(F)ccc1-c1cc(Cn2ccn(C)c2=N)cc(c1)C(=O)NCc1ccc(Cl)c(Cl)c1	InChI=1S/C25H22Cl2FN5O/c1-15-20(4-6-23(28)31-15)18-9-17(14-33-8-7-32(2)25(33)29)10-19(12-18)24(34)30-13-16-3-5-21(26)22(27)11-16/h3-12,29H,13-14H2,1-2H3,(H,30,34)	ZPVQIJIWGMKMQN-UHFFFAOYSA-N	50520121	CHEMBL4441671::US10844044, Example 1	WD repeat-containing protein 5		 0.044000								ChEMBL	10.1021/acs.jmedchem.9b01608	10.7270/Q2HD801W	31858797			Tian, J; Teuscher, KB; Aho, ER; Alvarado, JR; Mills, JJ; Meyers, KM; Gogliotti, RD; Han, C; Macdonald, JD; Sai, J; Shaw, JG; Sensintaffar, JL; Zhao, B; Rietz, TA; Thomas, LR; Payne, WG; Moore, WJ; Stott, GM; Kondo, J; Inoue, M; Coffey, RJ; Tansey, WP; Stauffer, SR; Lee, T; Fesik, SW	Frederick National Laboratory for Cancer Research	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50520121	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50520121&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	HLJ	6E23	138319680	440728703							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51274355	Cc1cc(F)ccc1-c1cc(Cn2ccn(C)c2=N)cc(c1)C(=O)NCc1cccc(OC(F)(F)F)c1	InChI=1S/C27H24F4N4O2/c1-17-10-22(28)6-7-24(17)20-11-19(16-35-9-8-34(2)26(35)32)12-21(14-20)25(36)33-15-18-4-3-5-23(13-18)37-27(29,30)31/h3-14,32H,15-16H2,1-2H3,(H,33,36)	XAYYLIMJMPHLEU-UHFFFAOYSA-N	50520122	CHEMBL4528067	WD repeat-containing protein 5				 16						ChEMBL	10.1021/acs.jmedchem.9b01608	10.7270/Q2HD801W	31858797			Tian, J; Teuscher, KB; Aho, ER; Alvarado, JR; Mills, JJ; Meyers, KM; Gogliotti, RD; Han, C; Macdonald, JD; Sai, J; Shaw, JG; Sensintaffar, JL; Zhao, B; Rietz, TA; Thomas, LR; Payne, WG; Moore, WJ; Stott, GM; Kondo, J; Inoue, M; Coffey, RJ; Tansey, WP; Stauffer, SR; Lee, T; Fesik, SW	Frederick National Laboratory for Cancer Research	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50520122	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50520122&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			155544527	440728704							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51274356	Cc1cc(F)ccc1-c1cc(Cn2ccn(C)c2=N)cc(c1)C(=O)NCc1ccccc1	InChI=1S/C26H25FN4O/c1-18-12-23(27)8-9-24(18)21-13-20(17-31-11-10-30(2)26(31)28)14-22(15-21)25(32)29-16-19-6-4-3-5-7-19/h3-15,28H,16-17H2,1-2H3,(H,29,32)	QKCLNALYVLGWBJ-UHFFFAOYSA-N	50520123	CHEMBL4567878	WD repeat-containing protein 5				 1.5						ChEMBL	10.1021/acs.jmedchem.9b01608	10.7270/Q2HD801W	31858797			Tian, J; Teuscher, KB; Aho, ER; Alvarado, JR; Mills, JJ; Meyers, KM; Gogliotti, RD; Han, C; Macdonald, JD; Sai, J; Shaw, JG; Sensintaffar, JL; Zhao, B; Rietz, TA; Thomas, LR; Payne, WG; Moore, WJ; Stott, GM; Kondo, J; Inoue, M; Coffey, RJ; Tansey, WP; Stauffer, SR; Lee, T; Fesik, SW	Frederick National Laboratory for Cancer Research	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50520123	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50520123&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			155560512	440728705							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51274357	Cc1cccc(CNC(=O)c2cc(Cn3ccn(C)c3=N)cc(c2)-c2ccc(F)cc2C)c1	InChI=1S/C27H27FN4O/c1-18-5-4-6-20(11-18)16-30-26(33)23-14-21(17-32-10-9-31(3)27(32)29)13-22(15-23)25-8-7-24(28)12-19(25)2/h4-15,29H,16-17H2,1-3H3,(H,30,33)	MWCGNILUFFTCKB-UHFFFAOYSA-N	50520124	CHEMBL4570860	WD repeat-containing protein 5				 0.500000						ChEMBL	10.1021/acs.jmedchem.9b01608	10.7270/Q2HD801W	31858797			Tian, J; Teuscher, KB; Aho, ER; Alvarado, JR; Mills, JJ; Meyers, KM; Gogliotti, RD; Han, C; Macdonald, JD; Sai, J; Shaw, JG; Sensintaffar, JL; Zhao, B; Rietz, TA; Thomas, LR; Payne, WG; Moore, WJ; Stott, GM; Kondo, J; Inoue, M; Coffey, RJ; Tansey, WP; Stauffer, SR; Lee, T; Fesik, SW	Frederick National Laboratory for Cancer Research	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50520124	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50520124&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			155562726	440728706							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51274358	Cc1cc(F)ccc1-c1cc(Cn2ccn(C)c2=N)cc(c1)C(=O)NCc1cccc(Cl)c1	InChI=1S/C26H24ClFN4O/c1-17-10-23(28)6-7-24(17)20-11-19(16-32-9-8-31(2)26(32)29)12-21(14-20)25(33)30-15-18-4-3-5-22(27)13-18/h3-14,29H,15-16H2,1-2H3,(H,30,33)	TVZUKBJFTYWVNB-UHFFFAOYSA-N	50520125	CHEMBL4578661	WD repeat-containing protein 5				 0.140000						ChEMBL	10.1021/acs.jmedchem.9b01608	10.7270/Q2HD801W	31858797			Tian, J; Teuscher, KB; Aho, ER; Alvarado, JR; Mills, JJ; Meyers, KM; Gogliotti, RD; Han, C; Macdonald, JD; Sai, J; Shaw, JG; Sensintaffar, JL; Zhao, B; Rietz, TA; Thomas, LR; Payne, WG; Moore, WJ; Stott, GM; Kondo, J; Inoue, M; Coffey, RJ; Tansey, WP; Stauffer, SR; Lee, T; Fesik, SW	Frederick National Laboratory for Cancer Research	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50520125	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50520125&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			155564728	440728707							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51274359	Cc1cc(F)ccc1-c1cc(Cn2ccn(C)c2=N)cc(c1)C(=O)NCc1ccc(Cl)c(Cl)c1	InChI=1S/C26H23Cl2FN4O/c1-16-9-21(29)4-5-22(16)19-10-18(15-33-8-7-32(2)26(33)30)11-20(13-19)25(34)31-14-17-3-6-23(27)24(28)12-17/h3-13,30H,14-15H2,1-2H3,(H,31,34)	PLTUYQPTAZNZMJ-UHFFFAOYSA-N	50520126	CHEMBL4557848	WD repeat-containing protein 5				 0.030000						ChEMBL	10.1021/acs.jmedchem.9b01608	10.7270/Q2HD801W	31858797			Tian, J; Teuscher, KB; Aho, ER; Alvarado, JR; Mills, JJ; Meyers, KM; Gogliotti, RD; Han, C; Macdonald, JD; Sai, J; Shaw, JG; Sensintaffar, JL; Zhao, B; Rietz, TA; Thomas, LR; Payne, WG; Moore, WJ; Stott, GM; Kondo, J; Inoue, M; Coffey, RJ; Tansey, WP; Stauffer, SR; Lee, T; Fesik, SW	Frederick National Laboratory for Cancer Research	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50520126	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50520126&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			155554755	440728708							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51274360	Cc1cc(CNC(=O)c2cc(Cn3ccn(C)c3=N)cc(c2)-c2ccc(F)cc2C)ccc1F	InChI=1S/C27H26F2N4O/c1-17-11-23(28)5-6-24(17)21-12-20(16-33-9-8-32(3)27(33)30)13-22(14-21)26(34)31-15-19-4-7-25(29)18(2)10-19/h4-14,30H,15-16H2,1-3H3,(H,31,34)	LEOZOVLOEOWBAL-UHFFFAOYSA-N	50520127	CHEMBL4585441::US10844044, Example 87	WD repeat-containing protein 5				 0.032000						ChEMBL	10.1021/acs.jmedchem.9b01608	10.7270/Q2HD801W	31858797			Tian, J; Teuscher, KB; Aho, ER; Alvarado, JR; Mills, JJ; Meyers, KM; Gogliotti, RD; Han, C; Macdonald, JD; Sai, J; Shaw, JG; Sensintaffar, JL; Zhao, B; Rietz, TA; Thomas, LR; Payne, WG; Moore, WJ; Stott, GM; Kondo, J; Inoue, M; Coffey, RJ; Tansey, WP; Stauffer, SR; Lee, T; Fesik, SW	Frederick National Laboratory for Cancer Research	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50520127	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50520127&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456497	440728709							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51274361	Cc1cc(C)cc(CNC(=O)c2cc(Cn3ccn(C)c3=N)cc(c2)-c2ccc(F)cc2C)c1	InChI=1S/C28H29FN4O/c1-18-9-19(2)11-21(10-18)16-31-27(34)24-14-22(17-33-8-7-32(4)28(33)30)13-23(15-24)26-6-5-25(29)12-20(26)3/h5-15,30H,16-17H2,1-4H3,(H,31,34)	GOOQUIWHDCJDCE-UHFFFAOYSA-N	50520128	CHEMBL4555492	WD repeat-containing protein 5				 0.055000						ChEMBL	10.1021/acs.jmedchem.9b01608	10.7270/Q2HD801W	31858797			Tian, J; Teuscher, KB; Aho, ER; Alvarado, JR; Mills, JJ; Meyers, KM; Gogliotti, RD; Han, C; Macdonald, JD; Sai, J; Shaw, JG; Sensintaffar, JL; Zhao, B; Rietz, TA; Thomas, LR; Payne, WG; Moore, WJ; Stott, GM; Kondo, J; Inoue, M; Coffey, RJ; Tansey, WP; Stauffer, SR; Lee, T; Fesik, SW	Frederick National Laboratory for Cancer Research	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50520128	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50520128&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			155556853	440728710							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51274362	Cc1cc(F)ccc1-c1cc(Cn2ccn(C)c2=N)cc(c1)C(=O)NCc1cc(Cl)cc(Cl)c1	InChI=1S/C26H23Cl2FN4O/c1-16-7-23(29)3-4-24(16)19-8-18(15-33-6-5-32(2)26(33)30)9-20(12-19)25(34)31-14-17-10-21(27)13-22(28)11-17/h3-13,30H,14-15H2,1-2H3,(H,31,34)	MMZHNVVOIBRRPP-UHFFFAOYSA-N	50520129	CHEMBL4593719	WD repeat-containing protein 5				 0.061000						ChEMBL	10.1021/acs.jmedchem.9b01608	10.7270/Q2HD801W	31858797			Tian, J; Teuscher, KB; Aho, ER; Alvarado, JR; Mills, JJ; Meyers, KM; Gogliotti, RD; Han, C; Macdonald, JD; Sai, J; Shaw, JG; Sensintaffar, JL; Zhao, B; Rietz, TA; Thomas, LR; Payne, WG; Moore, WJ; Stott, GM; Kondo, J; Inoue, M; Coffey, RJ; Tansey, WP; Stauffer, SR; Lee, T; Fesik, SW	Frederick National Laboratory for Cancer Research	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50520129	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50520129&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			155569468	440728711							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51274363	COc1cc(CNC(=O)c2cc(Cn3ccn(C)c3=N)cc(c2)-c2ccc(F)cc2C)cc(OC)c1	InChI=1S/C28H29FN4O3/c1-18-9-23(29)5-6-26(18)21-10-20(17-33-8-7-32(2)28(33)30)11-22(14-21)27(34)31-16-19-12-24(35-3)15-25(13-19)36-4/h5-15,30H,16-17H2,1-4H3,(H,31,34)	PSABMKXBOJUOBD-UHFFFAOYSA-N	50520130	CHEMBL4435250	WD repeat-containing protein 5				 0.049000						ChEMBL	10.1021/acs.jmedchem.9b01608	10.7270/Q2HD801W	31858797			Tian, J; Teuscher, KB; Aho, ER; Alvarado, JR; Mills, JJ; Meyers, KM; Gogliotti, RD; Han, C; Macdonald, JD; Sai, J; Shaw, JG; Sensintaffar, JL; Zhao, B; Rietz, TA; Thomas, LR; Payne, WG; Moore, WJ; Stott, GM; Kondo, J; Inoue, M; Coffey, RJ; Tansey, WP; Stauffer, SR; Lee, T; Fesik, SW	Frederick National Laboratory for Cancer Research	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50520130	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50520130&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	Q6S	6UFX	145946119	440728712							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51274364	COc1cc(CN2CCc3c(cc(Cn4ccn(C)c4=N)cc3-c3ccc(F)cc3C)C2=O)cc(OC)c1	InChI=1S/C30H31FN4O3/c1-19-11-22(31)5-6-25(19)27-14-21(18-35-10-9-33(2)30(35)32)15-28-26(27)7-8-34(29(28)36)17-20-12-23(37-3)16-24(13-20)38-4/h5-6,9-16,32H,7-8,17-18H2,1-4H3	PKONCIPMLLIAIL-UHFFFAOYSA-N	50520131	CHEMBL4588661	WD repeat-containing protein 5				<0.020000						ChEMBL	10.1021/acs.jmedchem.9b01608	10.7270/Q2HD801W	31858797			Tian, J; Teuscher, KB; Aho, ER; Alvarado, JR; Mills, JJ; Meyers, KM; Gogliotti, RD; Han, C; Macdonald, JD; Sai, J; Shaw, JG; Sensintaffar, JL; Zhao, B; Rietz, TA; Thomas, LR; Payne, WG; Moore, WJ; Stott, GM; Kondo, J; Inoue, M; Coffey, RJ; Tansey, WP; Stauffer, SR; Lee, T; Fesik, SW	Frederick National Laboratory for Cancer Research	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50520131	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50520131&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146014479	440728713							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51274365	COc1cc(CN2CCc3c(cc(Cn4ccn(C5CC5)c4=N)cc3-c3ccc(F)cc3C)C2=O)cc(OC)c1	InChI=1S/C32H33FN4O3/c1-20-12-23(33)4-7-27(20)29-15-22(19-36-10-11-37(32(36)34)24-5-6-24)16-30-28(29)8-9-35(31(30)38)18-21-13-25(39-2)17-26(14-21)40-3/h4,7,10-17,24,34H,5-6,8-9,18-19H2,1-3H3	BJMSIHKKVXBQDK-UHFFFAOYSA-N	50520132	CHEMBL4453355	WD repeat-containing protein 5				 0.043000						ChEMBL	10.1021/acs.jmedchem.9b01608	10.7270/Q2HD801W	31858797			Tian, J; Teuscher, KB; Aho, ER; Alvarado, JR; Mills, JJ; Meyers, KM; Gogliotti, RD; Han, C; Macdonald, JD; Sai, J; Shaw, JG; Sensintaffar, JL; Zhao, B; Rietz, TA; Thomas, LR; Payne, WG; Moore, WJ; Stott, GM; Kondo, J; Inoue, M; Coffey, RJ; Tansey, WP; Stauffer, SR; Lee, T; Fesik, SW	Frederick National Laboratory for Cancer Research	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50520132	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50520132&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			153572603	440728714							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51274366	COc1cc(CN2CCc3c(cc(CN4CCSC4=N)cc3-c3ccc(F)cc3C)C2=O)cc(OC)c1	InChI=1S/C29H30FN3O3S/c1-18-10-21(30)4-5-24(18)26-13-20(17-33-8-9-37-29(33)31)14-27-25(26)6-7-32(28(27)34)16-19-11-22(35-2)15-23(12-19)36-3/h4-5,10-15,31H,6-9,16-17H2,1-3H3	HDYJKMSOEDNXNO-UHFFFAOYSA-N	50520133	CHEMBL4530969	WD repeat-containing protein 5				 0.033000						ChEMBL	10.1021/acs.jmedchem.9b01608	10.7270/Q2HD801W	31858797			Tian, J; Teuscher, KB; Aho, ER; Alvarado, JR; Mills, JJ; Meyers, KM; Gogliotti, RD; Han, C; Macdonald, JD; Sai, J; Shaw, JG; Sensintaffar, JL; Zhao, B; Rietz, TA; Thomas, LR; Payne, WG; Moore, WJ; Stott, GM; Kondo, J; Inoue, M; Coffey, RJ; Tansey, WP; Stauffer, SR; Lee, T; Fesik, SW	Frederick National Laboratory for Cancer Research	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50520133	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50520133&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			153572528	440728715							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51274367	COc1cc(CN2CCc3c(cc(CN4CCCC4=N)cc3-c3ccc(F)cc3C)C2=O)cc(OC)c1	InChI=1S/C30H32FN3O3/c1-19-11-22(31)6-7-25(19)27-14-21(17-33-9-4-5-29(33)32)15-28-26(27)8-10-34(30(28)35)18-20-12-23(36-2)16-24(13-20)37-3/h6-7,11-16,32H,4-5,8-10,17-18H2,1-3H3	OOPRWCNRGGKSBQ-UHFFFAOYSA-N	50520134	CHEMBL4556167	WD repeat-containing protein 5				 0.063000						ChEMBL	10.1021/acs.jmedchem.9b01608	10.7270/Q2HD801W	31858797			Tian, J; Teuscher, KB; Aho, ER; Alvarado, JR; Mills, JJ; Meyers, KM; Gogliotti, RD; Han, C; Macdonald, JD; Sai, J; Shaw, JG; Sensintaffar, JL; Zhao, B; Rietz, TA; Thomas, LR; Payne, WG; Moore, WJ; Stott, GM; Kondo, J; Inoue, M; Coffey, RJ; Tansey, WP; Stauffer, SR; Lee, T; Fesik, SW	Frederick National Laboratory for Cancer Research	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50520134	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50520134&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			153572445	440728716							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51274368	COc1cc(CN2CCc3c(cc(Cn4cnn(C)c4=N)cc3-c3ccc(F)cc3C)C2=O)cc(OC)c1	InChI=1S/C29H30FN5O3/c1-18-9-21(30)5-6-24(18)26-12-20(16-35-17-32-33(2)29(35)31)13-27-25(26)7-8-34(28(27)36)15-19-10-22(37-3)14-23(11-19)38-4/h5-6,9-14,17,31H,7-8,15-16H2,1-4H3	DPAOKXUQYUWDHZ-UHFFFAOYSA-N	50520135	CHEMBL4463486	WD repeat-containing protein 5				 0.023000						ChEMBL	10.1021/acs.jmedchem.9b01608	10.7270/Q2HD801W	31858797			Tian, J; Teuscher, KB; Aho, ER; Alvarado, JR; Mills, JJ; Meyers, KM; Gogliotti, RD; Han, C; Macdonald, JD; Sai, J; Shaw, JG; Sensintaffar, JL; Zhao, B; Rietz, TA; Thomas, LR; Payne, WG; Moore, WJ; Stott, GM; Kondo, J; Inoue, M; Coffey, RJ; Tansey, WP; Stauffer, SR; Lee, T; Fesik, SW	Frederick National Laboratory for Cancer Research	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50520135	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50520135&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			153572410	440728717							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51274369	COc1cccc(CNC(=O)c2cc(Cn3ccn(C)c3=N)cc(c2)-c2ccc(F)cc2C)c1	InChI=1S/C27H27FN4O2/c1-18-11-23(28)7-8-25(18)21-12-20(17-32-10-9-31(2)27(32)29)13-22(15-21)26(33)30-16-19-5-4-6-24(14-19)34-3/h4-15,29H,16-17H2,1-3H3,(H,30,33)	SEUVFFLCJSGGCV-UHFFFAOYSA-N	50520136	CHEMBL4436638	WD repeat-containing protein 5				 0.160000						ChEMBL	10.1021/acs.jmedchem.9b01608	10.7270/Q2HD801W	31858797			Tian, J; Teuscher, KB; Aho, ER; Alvarado, JR; Mills, JJ; Meyers, KM; Gogliotti, RD; Han, C; Macdonald, JD; Sai, J; Shaw, JG; Sensintaffar, JL; Zhao, B; Rietz, TA; Thomas, LR; Payne, WG; Moore, WJ; Stott, GM; Kondo, J; Inoue, M; Coffey, RJ; Tansey, WP; Stauffer, SR; Lee, T; Fesik, SW	Frederick National Laboratory for Cancer Research	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50520136	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50520136&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			155512057	440728718							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51274370	COc1cc(CNC(=O)c2cc(Cn3ccn(C)c3=N)cc(c2)-c2ccc(F)cc2C)ccc1F	InChI=1S/C27H26F2N4O2/c1-17-10-22(28)5-6-23(17)20-11-19(16-33-9-8-32(2)27(33)30)12-21(14-20)26(34)31-15-18-4-7-24(29)25(13-18)35-3/h4-14,30H,15-16H2,1-3H3,(H,31,34)	HJWNICYTTDSUAA-UHFFFAOYSA-N	50520137	CHEMBL4439051	WD repeat-containing protein 5				 0.035000						ChEMBL	10.1021/acs.jmedchem.9b01608	10.7270/Q2HD801W	31858797			Tian, J; Teuscher, KB; Aho, ER; Alvarado, JR; Mills, JJ; Meyers, KM; Gogliotti, RD; Han, C; Macdonald, JD; Sai, J; Shaw, JG; Sensintaffar, JL; Zhao, B; Rietz, TA; Thomas, LR; Payne, WG; Moore, WJ; Stott, GM; Kondo, J; Inoue, M; Coffey, RJ; Tansey, WP; Stauffer, SR; Lee, T; Fesik, SW	Frederick National Laboratory for Cancer Research	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50520137	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50520137&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			155513664	440728719							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51274371	Cc1cc(CN2CCc3c(cc(Cn4ccn(C)c4=N)cc3-c3ccc(F)cc3C)C2=O)ccc1F	InChI=1S/C29H28F2N4O/c1-18-13-22(30)5-6-23(18)25-14-21(17-35-11-10-33(3)29(35)32)15-26-24(25)8-9-34(28(26)36)16-20-4-7-27(31)19(2)12-20/h4-7,10-15,32H,8-9,16-17H2,1-3H3	QQLAXBUUMWUFLV-UHFFFAOYSA-N	50520138	CHEMBL4463776	WD repeat-containing protein 5				<0.020000						ChEMBL	10.1021/acs.jmedchem.9b01608	10.7270/Q2HD801W	31858797			Tian, J; Teuscher, KB; Aho, ER; Alvarado, JR; Mills, JJ; Meyers, KM; Gogliotti, RD; Han, C; Macdonald, JD; Sai, J; Shaw, JG; Sensintaffar, JL; Zhao, B; Rietz, TA; Thomas, LR; Payne, WG; Moore, WJ; Stott, GM; Kondo, J; Inoue, M; Coffey, RJ; Tansey, WP; Stauffer, SR; Lee, T; Fesik, SW	Frederick National Laboratory for Cancer Research	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50520138	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50520138&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			153572470	440728720							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51274372	COc1cc(CN2CCc3c(cc(CNC(=N)C4CC4)cc3-c3ccc(F)cc3C)C2=O)cc(OC)c1	InChI=1S/C30H32FN3O3/c1-18-10-22(31)6-7-25(18)27-13-19(16-33-29(32)21-4-5-21)14-28-26(27)8-9-34(30(28)35)17-20-11-23(36-2)15-24(12-20)37-3/h6-7,10-15,21H,4-5,8-9,16-17H2,1-3H3,(H2,32,33)	RYGKJPYPENITQS-UHFFFAOYSA-N	50520139	CHEMBL4534270	WD repeat-containing protein 5				 0.030000						ChEMBL	10.1021/acs.jmedchem.9b01608	10.7270/Q2HD801W	31858797			Tian, J; Teuscher, KB; Aho, ER; Alvarado, JR; Mills, JJ; Meyers, KM; Gogliotti, RD; Han, C; Macdonald, JD; Sai, J; Shaw, JG; Sensintaffar, JL; Zhao, B; Rietz, TA; Thomas, LR; Payne, WG; Moore, WJ; Stott, GM; Kondo, J; Inoue, M; Coffey, RJ; Tansey, WP; Stauffer, SR; Lee, T; Fesik, SW	Frederick National Laboratory for Cancer Research	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50520139	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50520139&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			153572609	440728721							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51274373	Cc1cc(CNC(=O)c2cc(Cn3ccn(C)c3=N)cc(c2)-c2ccc(F)cc2C)ccc1Cl	InChI=1S/C27H26ClFN4O/c1-17-11-23(29)5-6-24(17)21-12-20(16-33-9-8-32(3)27(33)30)13-22(14-21)26(34)31-15-19-4-7-25(28)18(2)10-19/h4-14,30H,15-16H2,1-3H3,(H,31,34)	IARSEIRVTAVNDY-UHFFFAOYSA-N	50520140	CHEMBL4474045	WD repeat-containing protein 5				 0.090000						ChEMBL	10.1021/acs.jmedchem.9b01608	10.7270/Q2HD801W	31858797			Tian, J; Teuscher, KB; Aho, ER; Alvarado, JR; Mills, JJ; Meyers, KM; Gogliotti, RD; Han, C; Macdonald, JD; Sai, J; Shaw, JG; Sensintaffar, JL; Zhao, B; Rietz, TA; Thomas, LR; Payne, WG; Moore, WJ; Stott, GM; Kondo, J; Inoue, M; Coffey, RJ; Tansey, WP; Stauffer, SR; Lee, T; Fesik, SW	Frederick National Laboratory for Cancer Research	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50520140	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50520140&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456000	440728722							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51274374	COc1cc(CN2CCc3c(cc(Cn4ccoc4=N)cc3-c3ccc(F)cc3C)C2=O)cc(OC)c1	InChI=1S/C29H28FN3O4/c1-18-10-21(30)4-5-24(18)26-13-20(17-33-8-9-37-29(33)31)14-27-25(26)6-7-32(28(27)34)16-19-11-22(35-2)15-23(12-19)36-3/h4-5,8-15,31H,6-7,16-17H2,1-3H3	UEMUOVAYMDAREG-UHFFFAOYSA-N	50520141	CHEMBL4462065	WD repeat-containing protein 5				<0.020000						ChEMBL	10.1021/acs.jmedchem.9b01608	10.7270/Q2HD801W	31858797			Tian, J; Teuscher, KB; Aho, ER; Alvarado, JR; Mills, JJ; Meyers, KM; Gogliotti, RD; Han, C; Macdonald, JD; Sai, J; Shaw, JG; Sensintaffar, JL; Zhao, B; Rietz, TA; Thomas, LR; Payne, WG; Moore, WJ; Stott, GM; Kondo, J; Inoue, M; Coffey, RJ; Tansey, WP; Stauffer, SR; Lee, T; Fesik, SW	Frederick National Laboratory for Cancer Research	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50520141	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50520141&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			153572353	440728723							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51308023	COc1ccc(Br)cc1S(=O)(=O)Nc1cc(Cl)ccc1O	InChI=1S/C13H11BrClNO4S/c1-20-12-5-2-8(14)6-13(12)21(18,19)16-10-7-9(15)3-4-11(10)17/h2-7,16-17H,1H3	UQWYDZCIYINORK-UHFFFAOYSA-N	50531083	CHEMBL4514537	WD repeat-containing protein 5				 4710						ChEMBL	10.1021/acs.jmedchem.9b01411	10.7270/Q2B85CM0	31724864			Macdonald, JD; Chacón Simon, S; Han, C; Wang, F; Shaw, JG; Howes, JE; Sai, J; Yuh, JP; Camper, D; Alicie, BM; Alvarado, J; Nikhar, S; Payne, W; Aho, ER; Bauer, JA; Zhao, B; Phan, J; Thomas, LR; Rossanese, OW; Tansey, WP; Waterson, AG; Stauffer, SR; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50531083	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50531083&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	Q0Y	6U6W	44117787	440739665							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51308024	Oc1ccc(cc1NS(=O)(=O)c1cc(Br)ccc1O)C1CC1	InChI=1S/C15H14BrNO4S/c16-11-4-6-14(19)15(8-11)22(20,21)17-12-7-10(9-1-2-9)3-5-13(12)18/h3-9,17-19H,1-2H2	PZPFYZKXLXAXNP-UHFFFAOYSA-N	50531084	CHEMBL4459698	WD repeat-containing protein 5				 818						ChEMBL	10.1021/acs.jmedchem.9b01411	10.7270/Q2B85CM0	31724864			Macdonald, JD; Chacón Simon, S; Han, C; Wang, F; Shaw, JG; Howes, JE; Sai, J; Yuh, JP; Camper, D; Alicie, BM; Alvarado, J; Nikhar, S; Payne, W; Aho, ER; Bauer, JA; Zhao, B; Phan, J; Thomas, LR; Rossanese, OW; Tansey, WP; Waterson, AG; Stauffer, SR; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50531084	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50531084&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			155527316	440739666							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51308025	COc1ccc(Br)cc1S(=O)(=O)Nc1cc(Cl)ccc1O	InChI=1S/C13H11BrClNO4S/c1-20-12-5-2-8(14)6-13(12)21(18,19)16-10-7-9(15)3-4-11(10)17/h2-7,16-17H,1H3	UQWYDZCIYINORK-UHFFFAOYSA-N	50531083	CHEMBL4514537	WD repeat-containing protein 5				 4710						ChEMBL	10.1021/acs.jmedchem.9b01411	10.7270/Q2B85CM0	31724864			Macdonald, JD; Chacón Simon, S; Han, C; Wang, F; Shaw, JG; Howes, JE; Sai, J; Yuh, JP; Camper, D; Alicie, BM; Alvarado, J; Nikhar, S; Payne, W; Aho, ER; Bauer, JA; Zhao, B; Phan, J; Thomas, LR; Rossanese, OW; Tansey, WP; Waterson, AG; Stauffer, SR; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50531083	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50531083&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	Q0Y	6U6W	44117787	440739665							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51308026	COc1ccc(Cl)cc1S(=O)(=O)Nc1cc(Cl)ccc1O	InChI=1S/C13H11Cl2NO4S/c1-20-12-5-3-9(15)7-13(12)21(18,19)16-10-6-8(14)2-4-11(10)17/h2-7,16-17H,1H3	GPRUVNBBDBNFJU-UHFFFAOYSA-N	50531085	CHEMBL4457898	WD repeat-containing protein 5				 8410						ChEMBL	10.1021/acs.jmedchem.9b01411	10.7270/Q2B85CM0	31724864			Macdonald, JD; Chacón Simon, S; Han, C; Wang, F; Shaw, JG; Howes, JE; Sai, J; Yuh, JP; Camper, D; Alicie, BM; Alvarado, J; Nikhar, S; Payne, W; Aho, ER; Bauer, JA; Zhao, B; Phan, J; Thomas, LR; Rossanese, OW; Tansey, WP; Waterson, AG; Stauffer, SR; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50531085	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50531085&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			44117786	440739667							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51308027	COc1ccc(Br)cc1S(=O)(=O)Nc1ccccc1O	InChI=1S/C13H12BrNO4S/c1-19-12-7-6-9(14)8-13(12)20(17,18)15-10-4-2-3-5-11(10)16/h2-8,15-16H,1H3	MDXFESLYXHRFDS-UHFFFAOYSA-N	50531086	CHEMBL4445624	WD repeat-containing protein 5				>40000						ChEMBL	10.1021/acs.jmedchem.9b01411	10.7270/Q2B85CM0	31724864			Macdonald, JD; Chacón Simon, S; Han, C; Wang, F; Shaw, JG; Howes, JE; Sai, J; Yuh, JP; Camper, D; Alicie, BM; Alvarado, J; Nikhar, S; Payne, W; Aho, ER; Bauer, JA; Zhao, B; Phan, J; Thomas, LR; Rossanese, OW; Tansey, WP; Waterson, AG; Stauffer, SR; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50531086	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50531086&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			2210942	440739668							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51308028	Oc1ccc(Cl)cc1NS(=O)(=O)c1cc(Br)ccc1O	InChI=1S/C12H9BrClNO4S/c13-7-1-3-11(17)12(5-7)20(18,19)15-9-6-8(14)2-4-10(9)16/h1-6,15-17H	NVBGVGWRMDACKA-UHFFFAOYSA-N	50531087	CHEMBL4470230	WD repeat-containing protein 5				 1250						ChEMBL	10.1021/acs.jmedchem.9b01411	10.7270/Q2B85CM0	31724864			Macdonald, JD; Chacón Simon, S; Han, C; Wang, F; Shaw, JG; Howes, JE; Sai, J; Yuh, JP; Camper, D; Alicie, BM; Alvarado, J; Nikhar, S; Payne, W; Aho, ER; Bauer, JA; Zhao, B; Phan, J; Thomas, LR; Rossanese, OW; Tansey, WP; Waterson, AG; Stauffer, SR; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50531087	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50531087&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			155534245	440739669							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51308029	Oc1ccc(OC(F)(F)F)cc1NS(=O)(=O)c1cc(Br)ccc1O	InChI=1S/C13H9BrF3NO5S/c14-7-1-3-11(20)12(5-7)24(21,22)18-9-6-8(2-4-10(9)19)23-13(15,16)17/h1-6,18-20H	HNNNOZOIFLCBOK-UHFFFAOYSA-N	50531088	CHEMBL4462398	WD repeat-containing protein 5				 549						ChEMBL	10.1021/acs.jmedchem.9b01411	10.7270/Q2B85CM0	31724864			Macdonald, JD; Chacón Simon, S; Han, C; Wang, F; Shaw, JG; Howes, JE; Sai, J; Yuh, JP; Camper, D; Alicie, BM; Alvarado, J; Nikhar, S; Payne, W; Aho, ER; Bauer, JA; Zhao, B; Phan, J; Thomas, LR; Rossanese, OW; Tansey, WP; Waterson, AG; Stauffer, SR; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50531088	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50531088&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			155529149	440739670							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51308030	Oc1ccc(cc1NS(=O)(=O)c1cc(Br)ccc1O)S(F)(F)(F)(F)F	InChI=1S/C12H9BrF5NO4S2/c13-7-1-3-11(21)12(5-7)24(22,23)19-9-6-8(2-4-10(9)20)25(14,15,16,17)18/h1-6,19-21H	ATCYNRMRQJYXTG-UHFFFAOYSA-N	50531089	CHEMBL4569742	WD repeat-containing protein 5				 110						ChEMBL	10.1021/acs.jmedchem.9b01411	10.7270/Q2B85CM0	31724864			Macdonald, JD; Chacón Simon, S; Han, C; Wang, F; Shaw, JG; Howes, JE; Sai, J; Yuh, JP; Camper, D; Alicie, BM; Alvarado, J; Nikhar, S; Payne, W; Aho, ER; Bauer, JA; Zhao, B; Phan, J; Thomas, LR; Rossanese, OW; Tansey, WP; Waterson, AG; Stauffer, SR; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50531089	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50531089&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			155552109	440739671							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51308031	Oc1ccc(cc1NS(=O)(=O)c1cc(Br)ccc1O)C1(CC1)C(F)(F)F	InChI=1S/C16H13BrF3NO4S/c17-10-2-4-13(23)14(8-10)26(24,25)21-11-7-9(1-3-12(11)22)15(5-6-15)16(18,19)20/h1-4,7-8,21-23H,5-6H2	UFMQRARCXUCJDI-UHFFFAOYSA-N	50531090	CHEMBL4583201	WD repeat-containing protein 5				 547						ChEMBL	10.1021/acs.jmedchem.9b01411	10.7270/Q2B85CM0	31724864			Macdonald, JD; Chacón Simon, S; Han, C; Wang, F; Shaw, JG; Howes, JE; Sai, J; Yuh, JP; Camper, D; Alicie, BM; Alvarado, J; Nikhar, S; Payne, W; Aho, ER; Bauer, JA; Zhao, B; Phan, J; Thomas, LR; Rossanese, OW; Tansey, WP; Waterson, AG; Stauffer, SR; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50531090	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50531090&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			155566133	440739672							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51308032	Oc1ccc(cc1NS(=O)(=O)c1cc(Br)ccc1O)C1(CCC1)C#N	InChI=1S/C17H15BrN2O4S/c18-12-3-5-15(22)16(9-12)25(23,24)20-13-8-11(2-4-14(13)21)17(10-19)6-1-7-17/h2-5,8-9,20-22H,1,6-7H2	DMCFTKWJTBOJFX-UHFFFAOYSA-N	50531091	CHEMBL4470498	WD repeat-containing protein 5				 289						ChEMBL	10.1021/acs.jmedchem.9b01411	10.7270/Q2B85CM0	31724864			Macdonald, JD; Chacón Simon, S; Han, C; Wang, F; Shaw, JG; Howes, JE; Sai, J; Yuh, JP; Camper, D; Alicie, BM; Alvarado, J; Nikhar, S; Payne, W; Aho, ER; Bauer, JA; Zhao, B; Phan, J; Thomas, LR; Rossanese, OW; Tansey, WP; Waterson, AG; Stauffer, SR; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50531091	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50531091&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	Q1G	6U8O	145704703	440739673							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51308033	Oc1ccc(cc1NS(=O)(=O)c1cc(Br)ccc1O)C1(CCCCC1)C#N	InChI=1S/C19H19BrN2O4S/c20-14-5-7-17(24)18(11-14)27(25,26)22-15-10-13(4-6-16(15)23)19(12-21)8-2-1-3-9-19/h4-7,10-11,22-24H,1-3,8-9H2	NJDVFBPUGNOISW-UHFFFAOYSA-N	50531092	CHEMBL4537674	WD repeat-containing protein 5				 229						ChEMBL	10.1021/acs.jmedchem.9b01411	10.7270/Q2B85CM0	31724864			Macdonald, JD; Chacón Simon, S; Han, C; Wang, F; Shaw, JG; Howes, JE; Sai, J; Yuh, JP; Camper, D; Alicie, BM; Alvarado, J; Nikhar, S; Payne, W; Aho, ER; Bauer, JA; Zhao, B; Phan, J; Thomas, LR; Rossanese, OW; Tansey, WP; Waterson, AG; Stauffer, SR; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50531092	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50531092&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			155548095	440739674							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51308034	OC(=O)c1cc(Cl)cc(NS(=O)(=O)c2cc(Br)cc(Cl)c2O)c1O	InChI=1S/C13H8BrCl2NO6S/c14-5-1-8(16)12(19)10(2-5)24(22,23)17-9-4-6(15)3-7(11(9)18)13(20)21/h1-4,17-19H,(H,20,21)	GTSWUTVZEJOAKU-UHFFFAOYSA-N	50531093	CHEMBL4518711	WD repeat-containing protein 5				 163						ChEMBL	10.1021/acs.jmedchem.9b01411	10.7270/Q2B85CM0	31724864			Macdonald, JD; Chacón Simon, S; Han, C; Wang, F; Shaw, JG; Howes, JE; Sai, J; Yuh, JP; Camper, D; Alicie, BM; Alvarado, J; Nikhar, S; Payne, W; Aho, ER; Bauer, JA; Zhao, B; Phan, J; Thomas, LR; Rossanese, OW; Tansey, WP; Waterson, AG; Stauffer, SR; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50531093	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50531093&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			155541573	440739675							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51308035	OC(=O)c1cc(cc(NS(=O)(=O)c2cc(Br)ccc2O)c1O)C1CC1	InChI=1S/C16H14BrNO6S/c17-10-3-4-13(19)14(7-10)25(23,24)18-12-6-9(8-1-2-8)5-11(15(12)20)16(21)22/h3-8,18-20H,1-2H2,(H,21,22)	LYWDFIFQOBDOLA-UHFFFAOYSA-N	50531094	CHEMBL4473507	WD repeat-containing protein 5				 184						ChEMBL	10.1021/acs.jmedchem.9b01411	10.7270/Q2B85CM0	31724864			Macdonald, JD; Chacón Simon, S; Han, C; Wang, F; Shaw, JG; Howes, JE; Sai, J; Yuh, JP; Camper, D; Alicie, BM; Alvarado, J; Nikhar, S; Payne, W; Aho, ER; Bauer, JA; Zhao, B; Phan, J; Thomas, LR; Rossanese, OW; Tansey, WP; Waterson, AG; Stauffer, SR; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50531094	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50531094&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			155536166	440739676							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51308036	OC(=O)c1cc(cc(NS(=O)(=O)c2cc(Br)cc(Cl)c2O)c1O)C1CC1	InChI=1S/C16H13BrClNO6S/c17-9-5-11(18)15(21)13(6-9)26(24,25)19-12-4-8(7-1-2-7)3-10(14(12)20)16(22)23/h3-7,19-21H,1-2H2,(H,22,23)	RWFJMOHRSSMXSO-UHFFFAOYSA-N	50531095	CHEMBL4586914	WD repeat-containing protein 5				 207						ChEMBL	10.1021/acs.jmedchem.9b01411	10.7270/Q2B85CM0	31724864			Macdonald, JD; Chacón Simon, S; Han, C; Wang, F; Shaw, JG; Howes, JE; Sai, J; Yuh, JP; Camper, D; Alicie, BM; Alvarado, J; Nikhar, S; Payne, W; Aho, ER; Bauer, JA; Zhao, B; Phan, J; Thomas, LR; Rossanese, OW; Tansey, WP; Waterson, AG; Stauffer, SR; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50531095	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50531095&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			155566622	440739677							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51308037	OC(=O)c1c(O)c(NS(=O)(=O)c2cc(Br)cc(Cl)c2O)cc(C2CC2)c1F	InChI=1S/C16H12BrClFNO6S/c17-7-3-9(18)14(21)11(4-7)27(25,26)20-10-5-8(6-1-2-6)13(19)12(15(10)22)16(23)24/h3-6,20-22H,1-2H2,(H,23,24)	YFKMWXIJANJZQK-UHFFFAOYSA-N	50531096	CHEMBL4518895	WD repeat-containing protein 5				 50						ChEMBL	10.1021/acs.jmedchem.9b01411	10.7270/Q2B85CM0	31724864			Macdonald, JD; Chacón Simon, S; Han, C; Wang, F; Shaw, JG; Howes, JE; Sai, J; Yuh, JP; Camper, D; Alicie, BM; Alvarado, J; Nikhar, S; Payne, W; Aho, ER; Bauer, JA; Zhao, B; Phan, J; Thomas, LR; Rossanese, OW; Tansey, WP; Waterson, AG; Stauffer, SR; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50531096	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50531096&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			155541613	440739678							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51308038	OC(=O)c1cc(OC(F)(F)F)cc(NS(=O)(=O)c2cc(Br)ccc2O)c1O	InChI=1S/C14H9BrF3NO7S/c15-6-1-2-10(20)11(3-6)27(24,25)19-9-5-7(26-14(16,17)18)4-8(12(9)21)13(22)23/h1-5,19-21H,(H,22,23)	HJSHYSJMDZOUAB-UHFFFAOYSA-N	50531078	CHEMBL4575067	WD repeat-containing protein 5				 137						ChEMBL	10.1021/acs.jmedchem.9b01411	10.7270/Q2B85CM0	31724864			Macdonald, JD; Chacón Simon, S; Han, C; Wang, F; Shaw, JG; Howes, JE; Sai, J; Yuh, JP; Camper, D; Alicie, BM; Alvarado, J; Nikhar, S; Payne, W; Aho, ER; Bauer, JA; Zhao, B; Phan, J; Thomas, LR; Rossanese, OW; Tansey, WP; Waterson, AG; Stauffer, SR; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50531078	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50531078&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			155561018	440739660							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51308039	OC(=O)c1cc(cc(NS(=O)(=O)c2cc(Br)ccc2O)c1O)S(F)(F)(F)(F)F	InChI=1S/C13H9BrF5NO6S2/c14-6-1-2-10(21)11(3-6)27(25,26)20-9-5-7(28(15,16,17,18)19)4-8(12(9)22)13(23)24/h1-5,20-22H,(H,23,24)	QJKRMFMEFICLPS-UHFFFAOYSA-N	50531097	CHEMBL4544635	WD repeat-containing protein 5				 47						ChEMBL	10.1021/acs.jmedchem.9b01411	10.7270/Q2B85CM0	31724864			Macdonald, JD; Chacón Simon, S; Han, C; Wang, F; Shaw, JG; Howes, JE; Sai, J; Yuh, JP; Camper, D; Alicie, BM; Alvarado, J; Nikhar, S; Payne, W; Aho, ER; Bauer, JA; Zhao, B; Phan, J; Thomas, LR; Rossanese, OW; Tansey, WP; Waterson, AG; Stauffer, SR; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50531097	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50531097&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			155552825	440739679							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51308040	OC(=O)c1cc(cc(NS(=O)(=O)c2cc(Br)cc(Cl)c2O)c1O)S(F)(F)(F)(F)F	InChI=1S/C13H8BrClF5NO6S2/c14-5-1-8(15)12(23)10(2-5)28(26,27)21-9-4-6(29(16,17,18,19)20)3-7(11(9)22)13(24)25/h1-4,21-23H,(H,24,25)	ALXZNAKOFKFAFI-UHFFFAOYSA-N	50531098	CHEMBL4437642	WD repeat-containing protein 5				 31						ChEMBL	10.1021/acs.jmedchem.9b01411	10.7270/Q2B85CM0	31724864			Macdonald, JD; Chacón Simon, S; Han, C; Wang, F; Shaw, JG; Howes, JE; Sai, J; Yuh, JP; Camper, D; Alicie, BM; Alvarado, J; Nikhar, S; Payne, W; Aho, ER; Bauer, JA; Zhao, B; Phan, J; Thomas, LR; Rossanese, OW; Tansey, WP; Waterson, AG; Stauffer, SR; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50531098	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50531098&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			155512493	440739680							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51308041	OC(=O)c1cc(NS(=O)(=O)c2cc(Br)ccc2O)cc(c1)C1(CCC1)C#N	InChI=1S/C18H15BrN2O5S/c19-13-2-3-15(22)16(9-13)27(25,26)21-14-7-11(17(23)24)6-12(8-14)18(10-20)4-1-5-18/h2-3,6-9,21-22H,1,4-5H2,(H,23,24)	QCBAZYFNAWSSQJ-UHFFFAOYSA-N	50531099	CHEMBL4473122	WD repeat-containing protein 5				 229						ChEMBL	10.1021/acs.jmedchem.9b01411	10.7270/Q2B85CM0	31724864			Macdonald, JD; Chacón Simon, S; Han, C; Wang, F; Shaw, JG; Howes, JE; Sai, J; Yuh, JP; Camper, D; Alicie, BM; Alvarado, J; Nikhar, S; Payne, W; Aho, ER; Bauer, JA; Zhao, B; Phan, J; Thomas, LR; Rossanese, OW; Tansey, WP; Waterson, AG; Stauffer, SR; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50531099	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50531099&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			155536348	440739681							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51308042	OC(=O)c1cc(cc(NS(=O)(=O)c2cc(Br)ccc2O)c1O)C1(CCCCC1)C#N	InChI=1S/C20H19BrN2O6S/c21-13-4-5-16(24)17(10-13)30(28,29)23-15-9-12(8-14(18(15)25)19(26)27)20(11-22)6-2-1-3-7-20/h4-5,8-10,23-25H,1-3,6-7H2,(H,26,27)	LHQJNKXEQDMDIL-UHFFFAOYSA-N	50531079	CHEMBL4471282	WD repeat-containing protein 5				 195						ChEMBL	10.1021/acs.jmedchem.9b01411	10.7270/Q2B85CM0	31724864			Macdonald, JD; Chacón Simon, S; Han, C; Wang, F; Shaw, JG; Howes, JE; Sai, J; Yuh, JP; Camper, D; Alicie, BM; Alvarado, J; Nikhar, S; Payne, W; Aho, ER; Bauer, JA; Zhao, B; Phan, J; Thomas, LR; Rossanese, OW; Tansey, WP; Waterson, AG; Stauffer, SR; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50531079	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50531079&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			155534803	440739661							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51308043	OC(=O)c1cc(cc(NS(=O)(=O)c2cc(Br)cc(Cl)c2O)c1O)C1(CCCCC1)C#N	InChI=1S/C20H18BrClN2O6S/c21-12-8-14(22)18(26)16(9-12)31(29,30)24-15-7-11(6-13(17(15)25)19(27)28)20(10-23)4-2-1-3-5-20/h6-9,24-26H,1-5H2,(H,27,28)	MYQBJFOHGUHFHE-UHFFFAOYSA-N	50531100	CHEMBL4483349	WD repeat-containing protein 5				 38						ChEMBL	10.1021/acs.jmedchem.9b01411	10.7270/Q2B85CM0	31724864			Macdonald, JD; Chacón Simon, S; Han, C; Wang, F; Shaw, JG; Howes, JE; Sai, J; Yuh, JP; Camper, D; Alicie, BM; Alvarado, J; Nikhar, S; Payne, W; Aho, ER; Bauer, JA; Zhao, B; Phan, J; Thomas, LR; Rossanese, OW; Tansey, WP; Waterson, AG; Stauffer, SR; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50531100	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50531100&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			155540337	440739682							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51308044	CNC(=O)c1c(O)c(NS(=O)(=O)c2cc(Br)ccc2O)cc(C2CC2)c1F	InChI=1S/C17H16BrFN2O5S/c1-20-17(24)14-15(19)10(8-2-3-8)7-11(16(14)23)21-27(25,26)13-6-9(18)4-5-12(13)22/h4-8,21-23H,2-3H2,1H3,(H,20,24)	ZGDLNIYADXDMAW-UHFFFAOYSA-N	50531101	CHEMBL4465545	WD repeat-containing protein 5				 1420						ChEMBL	10.1021/acs.jmedchem.9b01411	10.7270/Q2B85CM0	31724864			Macdonald, JD; Chacón Simon, S; Han, C; Wang, F; Shaw, JG; Howes, JE; Sai, J; Yuh, JP; Camper, D; Alicie, BM; Alvarado, J; Nikhar, S; Payne, W; Aho, ER; Bauer, JA; Zhao, B; Phan, J; Thomas, LR; Rossanese, OW; Tansey, WP; Waterson, AG; Stauffer, SR; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50531101	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50531101&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			155531049	440739683							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51308045	CNC(=O)c1c(O)c(NS(=O)(=O)c2cc(Br)cc(Cl)c2O)cc(C2CC2)c1F	InChI=1S/C17H15BrClFN2O5S/c1-21-17(25)13-14(20)9(7-2-3-7)6-11(16(13)24)22-28(26,27)12-5-8(18)4-10(19)15(12)23/h4-7,22-24H,2-3H2,1H3,(H,21,25)	YVPZGFQMOJVHEN-UHFFFAOYSA-N	50531102	CHEMBL4594023	WD repeat-containing protein 5				 238						ChEMBL	10.1021/acs.jmedchem.9b01411	10.7270/Q2B85CM0	31724864			Macdonald, JD; Chacón Simon, S; Han, C; Wang, F; Shaw, JG; Howes, JE; Sai, J; Yuh, JP; Camper, D; Alicie, BM; Alvarado, J; Nikhar, S; Payne, W; Aho, ER; Bauer, JA; Zhao, B; Phan, J; Thomas, LR; Rossanese, OW; Tansey, WP; Waterson, AG; Stauffer, SR; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50531102	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50531102&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			155569544	440739684							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51308046	CNC(=O)c1cc(cc(NS(=O)(=O)c2cc(Br)cc(Cl)c2O)c1O)S(F)(F)(F)(F)F	InChI=1S/C14H11BrClF5N2O5S2/c1-22-14(26)8-4-7(30(17,18,19,20)21)5-10(12(8)24)23-29(27,28)11-3-6(15)2-9(16)13(11)25/h2-5,23-25H,1H3,(H,22,26)	VAZWKKNFRGLKJW-UHFFFAOYSA-N	50531103	CHEMBL4455721	WD repeat-containing protein 5				 190						ChEMBL	10.1021/acs.jmedchem.9b01411	10.7270/Q2B85CM0	31724864			Macdonald, JD; Chacón Simon, S; Han, C; Wang, F; Shaw, JG; Howes, JE; Sai, J; Yuh, JP; Camper, D; Alicie, BM; Alvarado, J; Nikhar, S; Payne, W; Aho, ER; Bauer, JA; Zhao, B; Phan, J; Thomas, LR; Rossanese, OW; Tansey, WP; Waterson, AG; Stauffer, SR; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50531103	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50531103&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			155524406	440739685							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51308047	CNC(=O)c1cc(NS(=O)(=O)c2cc(Br)cc(Cl)c2O)cc(c1)C1(CCC1)C#N	InChI=1S/C19H17BrClN3O4S/c1-23-18(26)11-5-12(19(10-22)3-2-4-19)7-14(6-11)24-29(27,28)16-9-13(20)8-15(21)17(16)25/h5-9,24-25H,2-4H2,1H3,(H,23,26)	CTKIIQPJMPIAAG-UHFFFAOYSA-N	50531104	CHEMBL4549544	WD repeat-containing protein 5				 128						ChEMBL	10.1021/acs.jmedchem.9b01411	10.7270/Q2B85CM0	31724864			Macdonald, JD; Chacón Simon, S; Han, C; Wang, F; Shaw, JG; Howes, JE; Sai, J; Yuh, JP; Camper, D; Alicie, BM; Alvarado, J; Nikhar, S; Payne, W; Aho, ER; Bauer, JA; Zhao, B; Phan, J; Thomas, LR; Rossanese, OW; Tansey, WP; Waterson, AG; Stauffer, SR; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50531104	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50531104&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			155550324	440739686							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51308048	CNC(=O)c1cc(cc(NS(=O)(=O)c2cc(Br)ccc2O)c1O)C1(CCC1)C#N	InChI=1S/C19H18BrN3O5S/c1-22-18(26)13-7-11(19(10-21)5-2-6-19)8-14(17(13)25)23-29(27,28)16-9-12(20)3-4-15(16)24/h3-4,7-9,23-25H,2,5-6H2,1H3,(H,22,26)	QNUCCYVBZDQUMB-UHFFFAOYSA-N	50531105	CHEMBL4543629	WD repeat-containing protein 5				 566						ChEMBL	10.1021/acs.jmedchem.9b01411	10.7270/Q2B85CM0	31724864			Macdonald, JD; Chacón Simon, S; Han, C; Wang, F; Shaw, JG; Howes, JE; Sai, J; Yuh, JP; Camper, D; Alicie, BM; Alvarado, J; Nikhar, S; Payne, W; Aho, ER; Bauer, JA; Zhao, B; Phan, J; Thomas, LR; Rossanese, OW; Tansey, WP; Waterson, AG; Stauffer, SR; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50531105	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50531105&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			155552279	440739687							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51308049	CNC(=O)c1cc(cc(NS(=O)(=O)c2cc(Br)cc(Cl)c2O)c1O)C1(CCCCC1)C#N	InChI=1S/C21H21BrClN3O5S/c1-25-20(29)14-7-12(21(11-24)5-3-2-4-6-21)8-16(18(14)27)26-32(30,31)17-10-13(22)9-15(23)19(17)28/h7-10,26-28H,2-6H2,1H3,(H,25,29)	RFZNGPIYBXOUDK-UHFFFAOYSA-N	50531106	CHEMBL4441794	WD repeat-containing protein 5				 362						ChEMBL	10.1021/acs.jmedchem.9b01411	10.7270/Q2B85CM0	31724864			Macdonald, JD; Chacón Simon, S; Han, C; Wang, F; Shaw, JG; Howes, JE; Sai, J; Yuh, JP; Camper, D; Alicie, BM; Alvarado, J; Nikhar, S; Payne, W; Aho, ER; Bauer, JA; Zhao, B; Phan, J; Thomas, LR; Rossanese, OW; Tansey, WP; Waterson, AG; Stauffer, SR; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50531106	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50531106&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			155515725	440739688							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51308050	COCCNc1cc(cc(NS(=O)(=O)c2cc(Br)ccc2O)c1O)C1(CCC1)C#N	InChI=1S/C20H22BrN3O5S/c1-29-8-7-23-15-9-13(20(12-22)5-2-6-20)10-16(19(15)26)24-30(27,28)18-11-14(21)3-4-17(18)25/h3-4,9-11,23-26H,2,5-8H2,1H3	BEQYRUOOCAHDEO-UHFFFAOYSA-N	50531107	CHEMBL4551051	WD repeat-containing protein 5				 757						ChEMBL	10.1021/acs.jmedchem.9b01411	10.7270/Q2B85CM0	31724864			Macdonald, JD; Chacón Simon, S; Han, C; Wang, F; Shaw, JG; Howes, JE; Sai, J; Yuh, JP; Camper, D; Alicie, BM; Alvarado, J; Nikhar, S; Payne, W; Aho, ER; Bauer, JA; Zhao, B; Phan, J; Thomas, LR; Rossanese, OW; Tansey, WP; Waterson, AG; Stauffer, SR; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50531107	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50531107&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			155554897	440739689							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51308051	CS(=O)(=O)c1cc(Cl)cc(NS(=O)(=O)c2cc(Br)ccc2O)c1	InChI=1S/C13H11BrClNO5S2/c1-22(18,19)11-6-9(15)5-10(7-11)16-23(20,21)13-4-8(14)2-3-12(13)17/h2-7,16-17H,1H3	OSGUHHXXRHWXPS-UHFFFAOYSA-N	50531108	CHEMBL4456384	WD repeat-containing protein 5				 1880						ChEMBL	10.1021/acs.jmedchem.9b01411	10.7270/Q2B85CM0	31724864			Macdonald, JD; Chacón Simon, S; Han, C; Wang, F; Shaw, JG; Howes, JE; Sai, J; Yuh, JP; Camper, D; Alicie, BM; Alvarado, J; Nikhar, S; Payne, W; Aho, ER; Bauer, JA; Zhao, B; Phan, J; Thomas, LR; Rossanese, OW; Tansey, WP; Waterson, AG; Stauffer, SR; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50531108	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50531108&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			155524907	440739690							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51308052	CS(=O)(=O)c1cc(Cl)cc(NS(=O)(=O)c2cc(Br)cc(Cl)c2O)c1O	InChI=1S/C13H10BrCl2NO6S2/c1-24(20,21)10-5-7(15)4-9(13(10)19)17-25(22,23)11-3-6(14)2-8(16)12(11)18/h2-5,17-19H,1H3	DMNYWAGZZMQKRG-UHFFFAOYSA-N	50531082	CHEMBL4455527	WD repeat-containing protein 5				 123						ChEMBL	10.1021/acs.jmedchem.9b01411	10.7270/Q2B85CM0	31724864			Macdonald, JD; Chacón Simon, S; Han, C; Wang, F; Shaw, JG; Howes, JE; Sai, J; Yuh, JP; Camper, D; Alicie, BM; Alvarado, J; Nikhar, S; Payne, W; Aho, ER; Bauer, JA; Zhao, B; Phan, J; Thomas, LR; Rossanese, OW; Tansey, WP; Waterson, AG; Stauffer, SR; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50531082	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50531082&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			155524950	440739664							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51308053	CS(=O)(=O)c1cc(NS(=O)(=O)c2cc(Br)cc(Cl)c2O)cc(c1)S(F)(F)(F)(F)F	InChI=1S/C13H10BrClF5NO5S3/c1-27(23,24)9-4-8(5-10(6-9)29(16,17,18,19)20)21-28(25,26)12-3-7(14)2-11(15)13(12)22/h2-6,21-22H,1H3	JZTVYUDUOQSWCQ-UHFFFAOYSA-N	50531109	CHEMBL4589677	WD repeat-containing protein 5				 93						ChEMBL	10.1021/acs.jmedchem.9b01411	10.7270/Q2B85CM0	31724864			Macdonald, JD; Chacón Simon, S; Han, C; Wang, F; Shaw, JG; Howes, JE; Sai, J; Yuh, JP; Camper, D; Alicie, BM; Alvarado, J; Nikhar, S; Payne, W; Aho, ER; Bauer, JA; Zhao, B; Phan, J; Thomas, LR; Rossanese, OW; Tansey, WP; Waterson, AG; Stauffer, SR; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50531109	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50531109&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			155568525	440739691							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51308054	CS(=O)(=O)c1cc(NS(=O)(=O)c2cc(Br)cc(Cl)c2O)cc(c1)C1(CCC1)C#N	InChI=1S/C18H16BrClN2O5S2/c1-28(24,25)14-6-11(18(10-21)3-2-4-18)5-13(9-14)22-29(26,27)16-8-12(19)7-15(20)17(16)23/h5-9,22-23H,2-4H2,1H3	AVODLYHEBPIIPG-UHFFFAOYSA-N	50531110	CHEMBL4447845	WD repeat-containing protein 5				 215						ChEMBL	10.1021/acs.jmedchem.9b01411	10.7270/Q2B85CM0	31724864			Macdonald, JD; Chacón Simon, S; Han, C; Wang, F; Shaw, JG; Howes, JE; Sai, J; Yuh, JP; Camper, D; Alicie, BM; Alvarado, J; Nikhar, S; Payne, W; Aho, ER; Bauer, JA; Zhao, B; Phan, J; Thomas, LR; Rossanese, OW; Tansey, WP; Waterson, AG; Stauffer, SR; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50531110	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50531110&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			155519558	440739692							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51308055	CS(=O)(=O)c1cc(cc(NS(=O)(=O)c2cc(Br)ccc2O)c1O)C1(CCC1)C#N	InChI=1S/C18H17BrN2O6S2/c1-28(24,25)16-8-11(18(10-20)5-2-6-18)7-13(17(16)23)21-29(26,27)15-9-12(19)3-4-14(15)22/h3-4,7-9,21-23H,2,5-6H2,1H3	ZOQUNXATFSLGSS-UHFFFAOYSA-N	50531111	CHEMBL4465645	WD repeat-containing protein 5				 349						ChEMBL	10.1021/acs.jmedchem.9b01411	10.7270/Q2B85CM0	31724864			Macdonald, JD; Chacón Simon, S; Han, C; Wang, F; Shaw, JG; Howes, JE; Sai, J; Yuh, JP; Camper, D; Alicie, BM; Alvarado, J; Nikhar, S; Payne, W; Aho, ER; Bauer, JA; Zhao, B; Phan, J; Thomas, LR; Rossanese, OW; Tansey, WP; Waterson, AG; Stauffer, SR; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50531111	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50531111&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			155531053	440739693							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51308056	CS(=O)(=O)c1cc(cc(NS(=O)(=O)c2cc(Br)cc(Cl)c2O)c1O)C1(CCC1)C#N	InChI=1S/C18H16BrClN2O6S2/c1-29(25,26)14-6-10(18(9-21)3-2-4-18)5-13(17(14)24)22-30(27,28)15-8-11(19)7-12(20)16(15)23/h5-8,22-24H,2-4H2,1H3	SUJUXKUBROGCLA-UHFFFAOYSA-N	50531112	CHEMBL4573903	WD repeat-containing protein 5				 110						ChEMBL	10.1021/acs.jmedchem.9b01411	10.7270/Q2B85CM0	31724864			Macdonald, JD; Chacón Simon, S; Han, C; Wang, F; Shaw, JG; Howes, JE; Sai, J; Yuh, JP; Camper, D; Alicie, BM; Alvarado, J; Nikhar, S; Payne, W; Aho, ER; Bauer, JA; Zhao, B; Phan, J; Thomas, LR; Rossanese, OW; Tansey, WP; Waterson, AG; Stauffer, SR; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50531112	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50531112&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			155563363	440739694							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51308057	CCOc1cc(ccc1F)S(=O)(=O)Nc1ccccc1C(O)=O	InChI=1S/C15H14FNO5S/c1-2-22-14-9-10(7-8-12(14)16)23(20,21)17-13-6-4-3-5-11(13)15(18)19/h3-9,17H,2H2,1H3,(H,18,19)	DMIRFYYZRJSZPF-UHFFFAOYSA-N	50531080	CHEMBL4465263	WD repeat-containing protein 5				 71000						ChEMBL	10.1021/acs.jmedchem.9b01411	10.7270/Q2B85CM0	31724864			Macdonald, JD; Chacón Simon, S; Han, C; Wang, F; Shaw, JG; Howes, JE; Sai, J; Yuh, JP; Camper, D; Alicie, BM; Alvarado, J; Nikhar, S; Payne, W; Aho, ER; Bauer, JA; Zhao, B; Phan, J; Thomas, LR; Rossanese, OW; Tansey, WP; Waterson, AG; Stauffer, SR; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50531080	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50531080&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			15943973	440739662							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51308058	CS(=O)(=O)c1cc(Cl)cc(NS(=O)(=O)c2cc(Br)cc3cccnc23)c1O	InChI=1S/C16H12BrClN2O5S2/c1-26(22,23)14-8-11(18)7-12(16(14)21)20-27(24,25)13-6-10(17)5-9-3-2-4-19-15(9)13/h2-8,20-21H,1H3	HVHOOKABEVVVMP-UHFFFAOYSA-N	50531113	CHEMBL4458101	WD repeat-containing protein 5				 385						ChEMBL	10.1021/acs.jmedchem.9b01411	10.7270/Q2B85CM0	31724864			Macdonald, JD; Chacón Simon, S; Han, C; Wang, F; Shaw, JG; Howes, JE; Sai, J; Yuh, JP; Camper, D; Alicie, BM; Alvarado, J; Nikhar, S; Payne, W; Aho, ER; Bauer, JA; Zhao, B; Phan, J; Thomas, LR; Rossanese, OW; Tansey, WP; Waterson, AG; Stauffer, SR; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50531113	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50531113&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			155526979	440739695							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51308059	OC(=O)c1cc(cc(NS(=O)(=O)c2cc(Br)cc3cccnc23)c1O)S(F)(F)(F)(F)F	InChI=1S/C16H10BrF5N2O5S2/c17-9-4-8-2-1-3-23-14(8)13(5-9)30(28,29)24-12-7-10(31(18,19,20,21)22)6-11(15(12)25)16(26)27/h1-7,24-25H,(H,26,27)	HTNUDGDQTGKVCW-UHFFFAOYSA-N	50531114	CHEMBL4468085	WD repeat-containing protein 5				 47						ChEMBL	10.1021/acs.jmedchem.9b01411	10.7270/Q2B85CM0	31724864			Macdonald, JD; Chacón Simon, S; Han, C; Wang, F; Shaw, JG; Howes, JE; Sai, J; Yuh, JP; Camper, D; Alicie, BM; Alvarado, J; Nikhar, S; Payne, W; Aho, ER; Bauer, JA; Zhao, B; Phan, J; Thomas, LR; Rossanese, OW; Tansey, WP; Waterson, AG; Stauffer, SR; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50531114	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50531114&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			155533048	440739696							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51308060	CS(=O)(=O)c1cc(cc(NS(=O)(=O)c2cc(Br)cc3cccnc23)c1O)C1(CCC1)C#N	InChI=1S/C21H18BrN3O5S2/c1-31(27,28)18-10-14(21(12-23)5-3-6-21)9-16(20(18)26)25-32(29,30)17-11-15(22)8-13-4-2-7-24-19(13)17/h2,4,7-11,25-26H,3,5-6H2,1H3	ZMYXSAKLPAHVLY-UHFFFAOYSA-N	50531115	CHEMBL4476737	WD repeat-containing protein 5				 272						ChEMBL	10.1021/acs.jmedchem.9b01411	10.7270/Q2B85CM0	31724864			Macdonald, JD; Chacón Simon, S; Han, C; Wang, F; Shaw, JG; Howes, JE; Sai, J; Yuh, JP; Camper, D; Alicie, BM; Alvarado, J; Nikhar, S; Payne, W; Aho, ER; Bauer, JA; Zhao, B; Phan, J; Thomas, LR; Rossanese, OW; Tansey, WP; Waterson, AG; Stauffer, SR; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50531115	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50531115&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			155538685	440739697							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51308061	COc1ccccc1S(=O)(=O)Nc1cc(Cl)ccc1O	InChI=1S/C13H12ClNO4S/c1-19-12-4-2-3-5-13(12)20(17,18)15-10-8-9(14)6-7-11(10)16/h2-8,15-16H,1H3	UFEFPYMMZBYZCH-UHFFFAOYSA-N	50531116	CHEMBL4532993	WD repeat-containing protein 5				>40000						ChEMBL	10.1021/acs.jmedchem.9b01411	10.7270/Q2B85CM0	31724864			Macdonald, JD; Chacón Simon, S; Han, C; Wang, F; Shaw, JG; Howes, JE; Sai, J; Yuh, JP; Camper, D; Alicie, BM; Alvarado, J; Nikhar, S; Payne, W; Aho, ER; Bauer, JA; Zhao, B; Phan, J; Thomas, LR; Rossanese, OW; Tansey, WP; Waterson, AG; Stauffer, SR; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50531116	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50531116&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			53541930	440739698							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51308062	Oc1ccc(cc1NS(=O)(=O)c1cc(Br)ccc1O)C1CC1	InChI=1S/C15H14BrNO4S/c16-11-4-6-14(19)15(8-11)22(20,21)17-12-7-10(9-1-2-9)3-5-13(12)18/h3-9,17-19H,1-2H2	PZPFYZKXLXAXNP-UHFFFAOYSA-N	50531084	CHEMBL4459698	WD repeat-containing protein 5				 818						ChEMBL	10.1021/acs.jmedchem.9b01411	10.7270/Q2B85CM0	31724864			Macdonald, JD; Chacón Simon, S; Han, C; Wang, F; Shaw, JG; Howes, JE; Sai, J; Yuh, JP; Camper, D; Alicie, BM; Alvarado, J; Nikhar, S; Payne, W; Aho, ER; Bauer, JA; Zhao, B; Phan, J; Thomas, LR; Rossanese, OW; Tansey, WP; Waterson, AG; Stauffer, SR; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50531084	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50531084&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			155527316	440739666							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51308063	OC(=O)c1cc(NS(=O)(=O)c2cc(Br)ccc2O)cc(OC(F)(F)F)c1	InChI=1S/C14H9BrF3NO6S/c15-8-1-2-11(20)12(5-8)26(23,24)19-9-3-7(13(21)22)4-10(6-9)25-14(16,17)18/h1-6,19-20H,(H,21,22)	PAORABHCETVZBY-UHFFFAOYSA-N	50531117	CHEMBL4469816	WD repeat-containing protein 5				 194						ChEMBL	10.1021/acs.jmedchem.9b01411	10.7270/Q2B85CM0	31724864			Macdonald, JD; Chacón Simon, S; Han, C; Wang, F; Shaw, JG; Howes, JE; Sai, J; Yuh, JP; Camper, D; Alicie, BM; Alvarado, J; Nikhar, S; Payne, W; Aho, ER; Bauer, JA; Zhao, B; Phan, J; Thomas, LR; Rossanese, OW; Tansey, WP; Waterson, AG; Stauffer, SR; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50531117	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50531117&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			155534418	440739699							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51308064	OC(=O)c1cc(cc(NS(=O)(=O)c2cc(Br)cc(Cl)c2O)c1O)C1(CCC1)C#N	InChI=1S/C18H14BrClN2O6S/c19-10-6-12(20)16(24)14(7-10)29(27,28)22-13-5-9(18(8-21)2-1-3-18)4-11(15(13)23)17(25)26/h4-7,22-24H,1-3H2,(H,25,26)	CVNNFNZYVCGPJF-UHFFFAOYSA-N	50531118	CHEMBL4535695	WD repeat-containing protein 5				 30						ChEMBL	10.1021/acs.jmedchem.9b01411	10.7270/Q2B85CM0	31724864			Macdonald, JD; Chacón Simon, S; Han, C; Wang, F; Shaw, JG; Howes, JE; Sai, J; Yuh, JP; Camper, D; Alicie, BM; Alvarado, J; Nikhar, S; Payne, W; Aho, ER; Bauer, JA; Zhao, B; Phan, J; Thomas, LR; Rossanese, OW; Tansey, WP; Waterson, AG; Stauffer, SR; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50531118	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50531118&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			155547929	440739700							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51308065	CNC(=O)c1cc(cc(NS(=O)(=O)c2cc(Br)ccc2O)c1O)S(F)(F)(F)(F)F	InChI=1S/C14H12BrF5N2O5S2/c1-21-14(25)9-5-8(29(16,17,18,19)20)6-10(13(9)24)22-28(26,27)12-4-7(15)2-3-11(12)23/h2-6,22-24H,1H3,(H,21,25)	UYPDTLHHKDBIQU-UHFFFAOYSA-N	50531119	CHEMBL4523046	WD repeat-containing protein 5				 204						ChEMBL	10.1021/acs.jmedchem.9b01411	10.7270/Q2B85CM0	31724864			Macdonald, JD; Chacón Simon, S; Han, C; Wang, F; Shaw, JG; Howes, JE; Sai, J; Yuh, JP; Camper, D; Alicie, BM; Alvarado, J; Nikhar, S; Payne, W; Aho, ER; Bauer, JA; Zhao, B; Phan, J; Thomas, LR; Rossanese, OW; Tansey, WP; Waterson, AG; Stauffer, SR; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50531119	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50531119&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			155543818	440739701							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51308066	CS(=O)(=O)c1cc(cc(NS(=O)(=O)c2cc(Br)ccc2O)c1O)S(F)(F)(F)(F)F	InChI=1S/C13H11BrF5NO6S3/c1-27(23,24)12-6-8(29(15,16,17,18)19)5-9(13(12)22)20-28(25,26)11-4-7(14)2-3-10(11)21/h2-6,20-22H,1H3	PUYSPWVTNKPCJD-UHFFFAOYSA-N	50531120	CHEMBL4554506	WD repeat-containing protein 5				 167						ChEMBL	10.1021/acs.jmedchem.9b01411	10.7270/Q2B85CM0	31724864			Macdonald, JD; Chacón Simon, S; Han, C; Wang, F; Shaw, JG; Howes, JE; Sai, J; Yuh, JP; Camper, D; Alicie, BM; Alvarado, J; Nikhar, S; Payne, W; Aho, ER; Bauer, JA; Zhao, B; Phan, J; Thomas, LR; Rossanese, OW; Tansey, WP; Waterson, AG; Stauffer, SR; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50531120	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50531120&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			155556036	440739702							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51308067	CNC(=O)c1cc(cc(NS(=O)(=O)c2cc(Br)ccc2OC)c1O)C1(CCC1)C#N	InChI=1S/C20H20BrN3O5S/c1-23-19(26)14-8-12(20(11-22)6-3-7-20)9-15(18(14)25)24-30(27,28)17-10-13(21)4-5-16(17)29-2/h4-5,8-10,24-25H,3,6-7H2,1-2H3,(H,23,26)	OGIHPKRHJNELFY-UHFFFAOYSA-N	50531121	CHEMBL4464746	WD repeat-containing protein 5				 906						ChEMBL	10.1021/acs.jmedchem.9b01411	10.7270/Q2B85CM0	31724864			Macdonald, JD; Chacón Simon, S; Han, C; Wang, F; Shaw, JG; Howes, JE; Sai, J; Yuh, JP; Camper, D; Alicie, BM; Alvarado, J; Nikhar, S; Payne, W; Aho, ER; Bauer, JA; Zhao, B; Phan, J; Thomas, LR; Rossanese, OW; Tansey, WP; Waterson, AG; Stauffer, SR; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50531121	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50531121&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			155530388	440739703							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51308068	COc1ccccc1S(=O)(=O)Nc1cc(Cl)ccc1O	InChI=1S/C13H12ClNO4S/c1-19-12-4-2-3-5-13(12)20(17,18)15-10-8-9(14)6-7-11(10)16/h2-8,15-16H,1H3	UFEFPYMMZBYZCH-UHFFFAOYSA-N	50531116	CHEMBL4532993	WD repeat-containing protein 5				>40000						ChEMBL	10.1021/acs.jmedchem.9b01411	10.7270/Q2B85CM0	31724864			Macdonald, JD; Chacón Simon, S; Han, C; Wang, F; Shaw, JG; Howes, JE; Sai, J; Yuh, JP; Camper, D; Alicie, BM; Alvarado, J; Nikhar, S; Payne, W; Aho, ER; Bauer, JA; Zhao, B; Phan, J; Thomas, LR; Rossanese, OW; Tansey, WP; Waterson, AG; Stauffer, SR; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50531116	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50531116&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			53541930	440739698							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51308069	COc1ccc(I)cc1S(=O)(=O)Nc1cc(Cl)ccc1O	InChI=1S/C13H11ClINO4S/c1-20-12-5-3-9(15)7-13(12)21(18,19)16-10-6-8(14)2-4-11(10)17/h2-7,16-17H,1H3	LPFIQDGAKMDLDS-UHFFFAOYSA-N	50531122	CHEMBL4443470	WD repeat-containing protein 5				 8390						ChEMBL	10.1021/acs.jmedchem.9b01411	10.7270/Q2B85CM0	31724864			Macdonald, JD; Chacón Simon, S; Han, C; Wang, F; Shaw, JG; Howes, JE; Sai, J; Yuh, JP; Camper, D; Alicie, BM; Alvarado, J; Nikhar, S; Payne, W; Aho, ER; Bauer, JA; Zhao, B; Phan, J; Thomas, LR; Rossanese, OW; Tansey, WP; Waterson, AG; Stauffer, SR; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50531122	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50531122&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			155516611	440739704							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51308070	Oc1ccc(Cl)cc1NS(=O)(=O)c1cccc(Br)c1	InChI=1S/C12H9BrClNO3S/c13-8-2-1-3-10(6-8)19(17,18)15-11-7-9(14)4-5-12(11)16/h1-7,15-16H	BYEKHFXVAPCFIJ-UHFFFAOYSA-N	50531123	CHEMBL4574127	WD repeat-containing protein 5				 36100						ChEMBL	10.1021/acs.jmedchem.9b01411	10.7270/Q2B85CM0	31724864			Macdonald, JD; Chacón Simon, S; Han, C; Wang, F; Shaw, JG; Howes, JE; Sai, J; Yuh, JP; Camper, D; Alicie, BM; Alvarado, J; Nikhar, S; Payne, W; Aho, ER; Bauer, JA; Zhao, B; Phan, J; Thomas, LR; Rossanese, OW; Tansey, WP; Waterson, AG; Stauffer, SR; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50531123	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50531123&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			28973441	440739705							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51308071	COc1ccc(Br)cc1S(=O)(=O)Nc1cc(ccc1O)-c1ccccc1	InChI=1S/C19H16BrNO4S/c1-25-18-10-8-15(20)12-19(18)26(23,24)21-16-11-14(7-9-17(16)22)13-5-3-2-4-6-13/h2-12,21-22H,1H3	LSOYIZUYLCYRNG-UHFFFAOYSA-N	50531124	CHEMBL4443499	WD repeat-containing protein 5				 37000						ChEMBL	10.1021/acs.jmedchem.9b01411	10.7270/Q2B85CM0	31724864			Macdonald, JD; Chacón Simon, S; Han, C; Wang, F; Shaw, JG; Howes, JE; Sai, J; Yuh, JP; Camper, D; Alicie, BM; Alvarado, J; Nikhar, S; Payne, W; Aho, ER; Bauer, JA; Zhao, B; Phan, J; Thomas, LR; Rossanese, OW; Tansey, WP; Waterson, AG; Stauffer, SR; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50531124	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50531124&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	Q1J	6U80	145704699	440739706							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51308072	COc1ccc(Br)cc1S(=O)(=O)Nc1cc(ccc1O)C(C)(C)C	InChI=1S/C17H20BrNO4S/c1-17(2,3)11-5-7-14(20)13(9-11)19-24(21,22)16-10-12(18)6-8-15(16)23-4/h5-10,19-20H,1-4H3	NUCBFUKPFYXFNL-UHFFFAOYSA-N	50531076	CHEMBL4514703	WD repeat-containing protein 5				 3780						ChEMBL	10.1021/acs.jmedchem.9b01411	10.7270/Q2B85CM0	31724864			Macdonald, JD; Chacón Simon, S; Han, C; Wang, F; Shaw, JG; Howes, JE; Sai, J; Yuh, JP; Camper, D; Alicie, BM; Alvarado, J; Nikhar, S; Payne, W; Aho, ER; Bauer, JA; Zhao, B; Phan, J; Thomas, LR; Rossanese, OW; Tansey, WP; Waterson, AG; Stauffer, SR; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50531076	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50531076&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			155539506	440739658							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51308073	Oc1ccc(OC(F)(F)F)cc1NS(=O)(=O)c1cc(Br)ccc1O	InChI=1S/C13H9BrF3NO5S/c14-7-1-3-11(20)12(5-7)24(21,22)18-9-6-8(2-4-10(9)19)23-13(15,16)17/h1-6,18-20H	HNNNOZOIFLCBOK-UHFFFAOYSA-N	50531088	CHEMBL4462398	WD repeat-containing protein 5				 549						ChEMBL	10.1021/acs.jmedchem.9b01411	10.7270/Q2B85CM0	31724864			Macdonald, JD; Chacón Simon, S; Han, C; Wang, F; Shaw, JG; Howes, JE; Sai, J; Yuh, JP; Camper, D; Alicie, BM; Alvarado, J; Nikhar, S; Payne, W; Aho, ER; Bauer, JA; Zhao, B; Phan, J; Thomas, LR; Rossanese, OW; Tansey, WP; Waterson, AG; Stauffer, SR; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50531088	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50531088&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			155529149	440739670							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51308074	Oc1ccc(cc1NS(=O)(=O)c1cc(Br)ccc1O)C1(CC1)C(F)(F)F	InChI=1S/C16H13BrF3NO4S/c17-10-2-4-13(23)14(8-10)26(24,25)21-11-7-9(1-3-12(11)22)15(5-6-15)16(18,19)20/h1-4,7-8,21-23H,5-6H2	UFMQRARCXUCJDI-UHFFFAOYSA-N	50531090	CHEMBL4583201	WD repeat-containing protein 5				 547						ChEMBL	10.1021/acs.jmedchem.9b01411	10.7270/Q2B85CM0	31724864			Macdonald, JD; Chacón Simon, S; Han, C; Wang, F; Shaw, JG; Howes, JE; Sai, J; Yuh, JP; Camper, D; Alicie, BM; Alvarado, J; Nikhar, S; Payne, W; Aho, ER; Bauer, JA; Zhao, B; Phan, J; Thomas, LR; Rossanese, OW; Tansey, WP; Waterson, AG; Stauffer, SR; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50531090	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50531090&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			155566133	440739672							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51308075	Oc1ccc(cc1NS(=O)(=O)c1cc(Br)ccc1O)C1(CC1)C#N	InChI=1S/C16H13BrN2O4S/c17-11-2-4-14(21)15(8-11)24(22,23)19-12-7-10(1-3-13(12)20)16(9-18)5-6-16/h1-4,7-8,19-21H,5-6H2	BZJQKWLSPXGRHB-UHFFFAOYSA-N	50531125	CHEMBL4436954	WD repeat-containing protein 5				 852						ChEMBL	10.1021/acs.jmedchem.9b01411	10.7270/Q2B85CM0	31724864			Macdonald, JD; Chacón Simon, S; Han, C; Wang, F; Shaw, JG; Howes, JE; Sai, J; Yuh, JP; Camper, D; Alicie, BM; Alvarado, J; Nikhar, S; Payne, W; Aho, ER; Bauer, JA; Zhao, B; Phan, J; Thomas, LR; Rossanese, OW; Tansey, WP; Waterson, AG; Stauffer, SR; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50531125	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50531125&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			155512250	440739707							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51308076	Oc1ccc(cc1NS(=O)(=O)c1cc(Br)ccc1O)C1(CCCC1)C#N	InChI=1S/C18H17BrN2O4S/c19-13-4-6-16(23)17(10-13)26(24,25)21-14-9-12(3-5-15(14)22)18(11-20)7-1-2-8-18/h3-6,9-10,21-23H,1-2,7-8H2	IFBNCOFMJUTHRR-UHFFFAOYSA-N	50531126	CHEMBL4434999	WD repeat-containing protein 5				 614						ChEMBL	10.1021/acs.jmedchem.9b01411	10.7270/Q2B85CM0	31724864			Macdonald, JD; Chacón Simon, S; Han, C; Wang, F; Shaw, JG; Howes, JE; Sai, J; Yuh, JP; Camper, D; Alicie, BM; Alvarado, J; Nikhar, S; Payne, W; Aho, ER; Bauer, JA; Zhao, B; Phan, J; Thomas, LR; Rossanese, OW; Tansey, WP; Waterson, AG; Stauffer, SR; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50531126	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50531126&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			155511088	440739708							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51308077	Oc1ccc(cc1NS(=O)(=O)c1cc(Br)ccc1O)C1(CCCCC1)C#N	InChI=1S/C19H19BrN2O4S/c20-14-5-7-17(24)18(11-14)27(25,26)22-15-10-13(4-6-16(15)23)19(12-21)8-2-1-3-9-19/h4-7,10-11,22-24H,1-3,8-9H2	NJDVFBPUGNOISW-UHFFFAOYSA-N	50531092	CHEMBL4537674	WD repeat-containing protein 5				 229						ChEMBL	10.1021/acs.jmedchem.9b01411	10.7270/Q2B85CM0	31724864			Macdonald, JD; Chacón Simon, S; Han, C; Wang, F; Shaw, JG; Howes, JE; Sai, J; Yuh, JP; Camper, D; Alicie, BM; Alvarado, J; Nikhar, S; Payne, W; Aho, ER; Bauer, JA; Zhao, B; Phan, J; Thomas, LR; Rossanese, OW; Tansey, WP; Waterson, AG; Stauffer, SR; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50531092	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50531092&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			155548095	440739674							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51308078	OC(=O)c1cc(Cl)cc(NS(=O)(=O)c2cc(Br)ccc2O)c1O	InChI=1S/C13H9BrClNO6S/c14-6-1-2-10(17)11(3-6)23(21,22)16-9-5-7(15)4-8(12(9)18)13(19)20/h1-5,16-18H,(H,19,20)	YKNSJAKLAKAVKH-UHFFFAOYSA-N	50531071	CHEMBL4573789	WD repeat-containing protein 5				 223						ChEMBL	10.1021/acs.jmedchem.9b01411	10.7270/Q2B85CM0	31724864			Macdonald, JD; Chacón Simon, S; Han, C; Wang, F; Shaw, JG; Howes, JE; Sai, J; Yuh, JP; Camper, D; Alicie, BM; Alvarado, J; Nikhar, S; Payne, W; Aho, ER; Bauer, JA; Zhao, B; Phan, J; Thomas, LR; Rossanese, OW; Tansey, WP; Waterson, AG; Stauffer, SR; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50531071	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50531071&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			155563120	440739653							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51308079	OC(=O)c1cc(cc(NS(=O)(=O)c2cc(Br)ccc2O)c1O)C1CC1	InChI=1S/C16H14BrNO6S/c17-10-3-4-13(19)14(7-10)25(23,24)18-12-6-9(8-1-2-8)5-11(15(12)20)16(21)22/h3-8,18-20H,1-2H2,(H,21,22)	LYWDFIFQOBDOLA-UHFFFAOYSA-N	50531094	CHEMBL4473507	WD repeat-containing protein 5				 184						ChEMBL	10.1021/acs.jmedchem.9b01411	10.7270/Q2B85CM0	31724864			Macdonald, JD; Chacón Simon, S; Han, C; Wang, F; Shaw, JG; Howes, JE; Sai, J; Yuh, JP; Camper, D; Alicie, BM; Alvarado, J; Nikhar, S; Payne, W; Aho, ER; Bauer, JA; Zhao, B; Phan, J; Thomas, LR; Rossanese, OW; Tansey, WP; Waterson, AG; Stauffer, SR; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50531094	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50531094&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			155536166	440739676							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51308080	OC(=O)c1cc(cc(NS(=O)(=O)c2cc(Br)cc(Cl)c2O)c1O)C1CC1	InChI=1S/C16H13BrClNO6S/c17-9-5-11(18)15(21)13(6-9)26(24,25)19-12-4-8(7-1-2-7)3-10(14(12)20)16(22)23/h3-7,19-21H,1-2H2,(H,22,23)	RWFJMOHRSSMXSO-UHFFFAOYSA-N	50531095	CHEMBL4586914	WD repeat-containing protein 5				 207						ChEMBL	10.1021/acs.jmedchem.9b01411	10.7270/Q2B85CM0	31724864			Macdonald, JD; Chacón Simon, S; Han, C; Wang, F; Shaw, JG; Howes, JE; Sai, J; Yuh, JP; Camper, D; Alicie, BM; Alvarado, J; Nikhar, S; Payne, W; Aho, ER; Bauer, JA; Zhao, B; Phan, J; Thomas, LR; Rossanese, OW; Tansey, WP; Waterson, AG; Stauffer, SR; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50531095	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50531095&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			155566622	440739677							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51308081	OC(=O)c1c(O)c(NS(=O)(=O)c2cc(Br)cc(Cl)c2O)cc(C2CC2)c1F	InChI=1S/C16H12BrClFNO6S/c17-7-3-9(18)14(21)11(4-7)27(25,26)20-10-5-8(6-1-2-6)13(19)12(15(10)22)16(23)24/h3-6,20-22H,1-2H2,(H,23,24)	YFKMWXIJANJZQK-UHFFFAOYSA-N	50531096	CHEMBL4518895	WD repeat-containing protein 5				 50						ChEMBL	10.1021/acs.jmedchem.9b01411	10.7270/Q2B85CM0	31724864			Macdonald, JD; Chacón Simon, S; Han, C; Wang, F; Shaw, JG; Howes, JE; Sai, J; Yuh, JP; Camper, D; Alicie, BM; Alvarado, J; Nikhar, S; Payne, W; Aho, ER; Bauer, JA; Zhao, B; Phan, J; Thomas, LR; Rossanese, OW; Tansey, WP; Waterson, AG; Stauffer, SR; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50531096	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50531096&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			155541613	440739678							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51308082	OC(=O)c1cc(NS(=O)(=O)c2cc(Br)ccc2O)cc(OC(F)(F)F)c1	InChI=1S/C14H9BrF3NO6S/c15-8-1-2-11(20)12(5-8)26(23,24)19-9-3-7(13(21)22)4-10(6-9)25-14(16,17)18/h1-6,19-20H,(H,21,22)	PAORABHCETVZBY-UHFFFAOYSA-N	50531117	CHEMBL4469816	WD repeat-containing protein 5				 194						ChEMBL	10.1021/acs.jmedchem.9b01411	10.7270/Q2B85CM0	31724864			Macdonald, JD; Chacón Simon, S; Han, C; Wang, F; Shaw, JG; Howes, JE; Sai, J; Yuh, JP; Camper, D; Alicie, BM; Alvarado, J; Nikhar, S; Payne, W; Aho, ER; Bauer, JA; Zhao, B; Phan, J; Thomas, LR; Rossanese, OW; Tansey, WP; Waterson, AG; Stauffer, SR; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50531117	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50531117&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			155534418	440739699							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51308083	OC(=O)c1cc(OC(F)(F)F)cc(NS(=O)(=O)c2cc(Br)cc(Cl)c2O)c1O	InChI=1S/C14H8BrClF3NO7S/c15-5-1-8(16)12(22)10(2-5)28(25,26)20-9-4-6(27-14(17,18)19)3-7(11(9)21)13(23)24/h1-4,20-22H,(H,23,24)	NJAWBWFLAWGPAQ-UHFFFAOYSA-N	50531127	CHEMBL4529202	WD repeat-containing protein 5				 51						ChEMBL	10.1021/acs.jmedchem.9b01411	10.7270/Q2B85CM0	31724864			Macdonald, JD; Chacón Simon, S; Han, C; Wang, F; Shaw, JG; Howes, JE; Sai, J; Yuh, JP; Camper, D; Alicie, BM; Alvarado, J; Nikhar, S; Payne, W; Aho, ER; Bauer, JA; Zhao, B; Phan, J; Thomas, LR; Rossanese, OW; Tansey, WP; Waterson, AG; Stauffer, SR; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50531127	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50531127&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			155545363	440739709							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51308084	OC(=O)c1cc(cc(NS(=O)(=O)c2cc(Br)cc(Cl)c2O)c1O)S(F)(F)(F)(F)F	InChI=1S/C13H8BrClF5NO6S2/c14-5-1-8(15)12(23)10(2-5)28(26,27)21-9-4-6(29(16,17,18,19)20)3-7(11(9)22)13(24)25/h1-4,21-23H,(H,24,25)	ALXZNAKOFKFAFI-UHFFFAOYSA-N	50531098	CHEMBL4437642	WD repeat-containing protein 5				 31						ChEMBL	10.1021/acs.jmedchem.9b01411	10.7270/Q2B85CM0	31724864			Macdonald, JD; Chacón Simon, S; Han, C; Wang, F; Shaw, JG; Howes, JE; Sai, J; Yuh, JP; Camper, D; Alicie, BM; Alvarado, J; Nikhar, S; Payne, W; Aho, ER; Bauer, JA; Zhao, B; Phan, J; Thomas, LR; Rossanese, OW; Tansey, WP; Waterson, AG; Stauffer, SR; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50531098	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50531098&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			155512493	440739680							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51308085	OC(=O)c1cc(NS(=O)(=O)c2cc(Br)ccc2O)cc(c1)C1(CCC1)C#N	InChI=1S/C18H15BrN2O5S/c19-13-2-3-15(22)16(9-13)27(25,26)21-14-7-11(17(23)24)6-12(8-14)18(10-20)4-1-5-18/h2-3,6-9,21-22H,1,4-5H2,(H,23,24)	QCBAZYFNAWSSQJ-UHFFFAOYSA-N	50531099	CHEMBL4473122	WD repeat-containing protein 5				 229						ChEMBL	10.1021/acs.jmedchem.9b01411	10.7270/Q2B85CM0	31724864			Macdonald, JD; Chacón Simon, S; Han, C; Wang, F; Shaw, JG; Howes, JE; Sai, J; Yuh, JP; Camper, D; Alicie, BM; Alvarado, J; Nikhar, S; Payne, W; Aho, ER; Bauer, JA; Zhao, B; Phan, J; Thomas, LR; Rossanese, OW; Tansey, WP; Waterson, AG; Stauffer, SR; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50531099	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50531099&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			155536348	440739681							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51308086	OC(=O)c1cc(cc(NS(=O)(=O)c2cc(Br)cc(Cl)c2O)c1O)C1(CCC1)C#N	InChI=1S/C18H14BrClN2O6S/c19-10-6-12(20)16(24)14(7-10)29(27,28)22-13-5-9(18(8-21)2-1-3-18)4-11(15(13)23)17(25)26/h4-7,22-24H,1-3H2,(H,25,26)	CVNNFNZYVCGPJF-UHFFFAOYSA-N	50531118	CHEMBL4535695	WD repeat-containing protein 5				 30						ChEMBL	10.1021/acs.jmedchem.9b01411	10.7270/Q2B85CM0	31724864			Macdonald, JD; Chacón Simon, S; Han, C; Wang, F; Shaw, JG; Howes, JE; Sai, J; Yuh, JP; Camper, D; Alicie, BM; Alvarado, J; Nikhar, S; Payne, W; Aho, ER; Bauer, JA; Zhao, B; Phan, J; Thomas, LR; Rossanese, OW; Tansey, WP; Waterson, AG; Stauffer, SR; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50531118	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50531118&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			155547929	440739700							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51308087	OC(=O)c1cc(cc(NS(=O)(=O)c2cc(Br)cc(Cl)c2O)c1O)C1(CCCCC1)C#N	InChI=1S/C20H18BrClN2O6S/c21-12-8-14(22)18(26)16(9-12)31(29,30)24-15-7-11(6-13(17(15)25)19(27)28)20(10-23)4-2-1-3-5-20/h6-9,24-26H,1-5H2,(H,27,28)	MYQBJFOHGUHFHE-UHFFFAOYSA-N	50531100	CHEMBL4483349	WD repeat-containing protein 5				 38						ChEMBL	10.1021/acs.jmedchem.9b01411	10.7270/Q2B85CM0	31724864			Macdonald, JD; Chacón Simon, S; Han, C; Wang, F; Shaw, JG; Howes, JE; Sai, J; Yuh, JP; Camper, D; Alicie, BM; Alvarado, J; Nikhar, S; Payne, W; Aho, ER; Bauer, JA; Zhao, B; Phan, J; Thomas, LR; Rossanese, OW; Tansey, WP; Waterson, AG; Stauffer, SR; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50531100	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50531100&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			155540337	440739682							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51308088	CNC(=O)c1c(O)c(NS(=O)(=O)c2cc(Br)ccc2O)cc(C2CC2)c1F	InChI=1S/C17H16BrFN2O5S/c1-20-17(24)14-15(19)10(8-2-3-8)7-11(16(14)23)21-27(25,26)13-6-9(18)4-5-12(13)22/h4-8,21-23H,2-3H2,1H3,(H,20,24)	ZGDLNIYADXDMAW-UHFFFAOYSA-N	50531101	CHEMBL4465545	WD repeat-containing protein 5				 1420						ChEMBL	10.1021/acs.jmedchem.9b01411	10.7270/Q2B85CM0	31724864			Macdonald, JD; Chacón Simon, S; Han, C; Wang, F; Shaw, JG; Howes, JE; Sai, J; Yuh, JP; Camper, D; Alicie, BM; Alvarado, J; Nikhar, S; Payne, W; Aho, ER; Bauer, JA; Zhao, B; Phan, J; Thomas, LR; Rossanese, OW; Tansey, WP; Waterson, AG; Stauffer, SR; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50531101	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50531101&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			155531049	440739683							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51308089	CNC(=O)c1c(O)c(NS(=O)(=O)c2cc(Br)cc(Cl)c2O)cc(C2CC2)c1F	InChI=1S/C17H15BrClFN2O5S/c1-21-17(25)13-14(20)9(7-2-3-7)6-11(16(13)24)22-28(26,27)12-5-8(18)4-10(19)15(12)23/h4-7,22-24H,2-3H2,1H3,(H,21,25)	YVPZGFQMOJVHEN-UHFFFAOYSA-N	50531102	CHEMBL4594023	WD repeat-containing protein 5				 238						ChEMBL	10.1021/acs.jmedchem.9b01411	10.7270/Q2B85CM0	31724864			Macdonald, JD; Chacón Simon, S; Han, C; Wang, F; Shaw, JG; Howes, JE; Sai, J; Yuh, JP; Camper, D; Alicie, BM; Alvarado, J; Nikhar, S; Payne, W; Aho, ER; Bauer, JA; Zhao, B; Phan, J; Thomas, LR; Rossanese, OW; Tansey, WP; Waterson, AG; Stauffer, SR; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50531102	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50531102&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			155569544	440739684							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51308090	CNC(=O)c1cc(NS(=O)(=O)c2cc(Br)ccc2O)cc(c1)S(F)(F)(F)(F)F	InChI=1S/C14H12BrF5N2O4S2/c1-21-14(24)8-4-10(7-11(5-8)28(16,17,18,19)20)22-27(25,26)13-6-9(15)2-3-12(13)23/h2-7,22-23H,1H3,(H,21,24)	JJPIOPKOYIGQSD-UHFFFAOYSA-N	50531128	CHEMBL4471513	WD repeat-containing protein 5				 848						ChEMBL	10.1021/acs.jmedchem.9b01411	10.7270/Q2B85CM0	31724864			Macdonald, JD; Chacón Simon, S; Han, C; Wang, F; Shaw, JG; Howes, JE; Sai, J; Yuh, JP; Camper, D; Alicie, BM; Alvarado, J; Nikhar, S; Payne, W; Aho, ER; Bauer, JA; Zhao, B; Phan, J; Thomas, LR; Rossanese, OW; Tansey, WP; Waterson, AG; Stauffer, SR; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50531128	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50531128&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			155535349	440739710							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51308091	CNC(=O)c1cc(NS(=O)(=O)c2cc(Br)cc(Cl)c2O)cc(c1)C1(CCC1)C#N	InChI=1S/C19H17BrClN3O4S/c1-23-18(26)11-5-12(19(10-22)3-2-4-19)7-14(6-11)24-29(27,28)16-9-13(20)8-15(21)17(16)25/h5-9,24-25H,2-4H2,1H3,(H,23,26)	CTKIIQPJMPIAAG-UHFFFAOYSA-N	50531104	CHEMBL4549544	WD repeat-containing protein 5				 128						ChEMBL	10.1021/acs.jmedchem.9b01411	10.7270/Q2B85CM0	31724864			Macdonald, JD; Chacón Simon, S; Han, C; Wang, F; Shaw, JG; Howes, JE; Sai, J; Yuh, JP; Camper, D; Alicie, BM; Alvarado, J; Nikhar, S; Payne, W; Aho, ER; Bauer, JA; Zhao, B; Phan, J; Thomas, LR; Rossanese, OW; Tansey, WP; Waterson, AG; Stauffer, SR; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50531104	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50531104&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			155550324	440739686							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51308092	CNC(=O)c1cc(cc(NS(=O)(=O)c2cc(Br)cc(Cl)c2O)c1O)C1(CCC1)C#N	InChI=1S/C19H17BrClN3O5S/c1-23-18(27)12-5-10(19(9-22)3-2-4-19)6-14(16(12)25)24-30(28,29)15-8-11(20)7-13(21)17(15)26/h5-8,24-26H,2-4H2,1H3,(H,23,27)	COYGYHFILXAMSQ-UHFFFAOYSA-N	50531074	CHEMBL4472649	WD repeat-containing protein 5				 69						ChEMBL	10.1021/acs.jmedchem.9b01411	10.7270/Q2B85CM0	31724864			Macdonald, JD; Chacón Simon, S; Han, C; Wang, F; Shaw, JG; Howes, JE; Sai, J; Yuh, JP; Camper, D; Alicie, BM; Alvarado, J; Nikhar, S; Payne, W; Aho, ER; Bauer, JA; Zhao, B; Phan, J; Thomas, LR; Rossanese, OW; Tansey, WP; Waterson, AG; Stauffer, SR; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50531074	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50531074&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	Q0M	6U5Y	145704698	440739656							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51308093	Oc1ccc(Br)cc1S(=O)(=O)Nc1cc(cc(Nc2nc[nH]n2)c1O)C1(CCC1)C#N	InChI=1S/C19H17BrN6O4S/c20-12-2-3-15(27)16(8-12)31(29,30)26-14-7-11(19(9-21)4-1-5-19)6-13(17(14)28)24-18-22-10-23-25-18/h2-3,6-8,10,26-28H,1,4-5H2,(H2,22,23,24,25)	FOGZDMZPYDJTOI-UHFFFAOYSA-N	50531129	CHEMBL4450684	WD repeat-containing protein 5				 46						ChEMBL	10.1021/acs.jmedchem.9b01411	10.7270/Q2B85CM0	31724864			Macdonald, JD; Chacón Simon, S; Han, C; Wang, F; Shaw, JG; Howes, JE; Sai, J; Yuh, JP; Camper, D; Alicie, BM; Alvarado, J; Nikhar, S; Payne, W; Aho, ER; Bauer, JA; Zhao, B; Phan, J; Thomas, LR; Rossanese, OW; Tansey, WP; Waterson, AG; Stauffer, SR; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50531129	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50531129&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			155521779	440739711							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51308094	COCCNc1cc(cc(NS(=O)(=O)c2cc(Br)ccc2O)c1O)C1(CCC1)C#N	InChI=1S/C20H22BrN3O5S/c1-29-8-7-23-15-9-13(20(12-22)5-2-6-20)10-16(19(15)26)24-30(27,28)18-11-14(21)3-4-17(18)25/h3-4,9-11,23-26H,2,5-8H2,1H3	BEQYRUOOCAHDEO-UHFFFAOYSA-N	50531107	CHEMBL4551051	WD repeat-containing protein 5				 757						ChEMBL	10.1021/acs.jmedchem.9b01411	10.7270/Q2B85CM0	31724864			Macdonald, JD; Chacón Simon, S; Han, C; Wang, F; Shaw, JG; Howes, JE; Sai, J; Yuh, JP; Camper, D; Alicie, BM; Alvarado, J; Nikhar, S; Payne, W; Aho, ER; Bauer, JA; Zhao, B; Phan, J; Thomas, LR; Rossanese, OW; Tansey, WP; Waterson, AG; Stauffer, SR; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50531107	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50531107&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			155554897	440739689							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51308095	CS(=O)(=O)c1cc(Cl)cc(NS(=O)(=O)c2cc(Br)cc(Cl)c2O)c1	InChI=1S/C13H10BrCl2NO5S2/c1-23(19,20)10-5-8(15)4-9(6-10)17-24(21,22)12-3-7(14)2-11(16)13(12)18/h2-6,17-18H,1H3	WYGIOFXYDQDPBX-UHFFFAOYSA-N	50531130	CHEMBL4534549	WD repeat-containing protein 5				 220						ChEMBL	10.1021/acs.jmedchem.9b01411	10.7270/Q2B85CM0	31724864			Macdonald, JD; Chacón Simon, S; Han, C; Wang, F; Shaw, JG; Howes, JE; Sai, J; Yuh, JP; Camper, D; Alicie, BM; Alvarado, J; Nikhar, S; Payne, W; Aho, ER; Bauer, JA; Zhao, B; Phan, J; Thomas, LR; Rossanese, OW; Tansey, WP; Waterson, AG; Stauffer, SR; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50531130	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50531130&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			155547031	440739712							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51308096	CS(=O)(=O)c1cc(NS(=O)(=O)c2cc(Br)cc(Cl)c2O)cc(c1)S(F)(F)(F)(F)F	InChI=1S/C13H10BrClF5NO5S3/c1-27(23,24)9-4-8(5-10(6-9)29(16,17,18,19)20)21-28(25,26)12-3-7(14)2-11(15)13(12)22/h2-6,21-22H,1H3	JZTVYUDUOQSWCQ-UHFFFAOYSA-N	50531109	CHEMBL4589677	WD repeat-containing protein 5				 93						ChEMBL	10.1021/acs.jmedchem.9b01411	10.7270/Q2B85CM0	31724864			Macdonald, JD; Chacón Simon, S; Han, C; Wang, F; Shaw, JG; Howes, JE; Sai, J; Yuh, JP; Camper, D; Alicie, BM; Alvarado, J; Nikhar, S; Payne, W; Aho, ER; Bauer, JA; Zhao, B; Phan, J; Thomas, LR; Rossanese, OW; Tansey, WP; Waterson, AG; Stauffer, SR; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50531109	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50531109&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			155568525	440739691							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51308097	CS(=O)(=O)c1cc(cc(NS(=O)(=O)c2cc(Br)cc(Cl)c2O)c1O)S(F)(F)(F)(F)F	InChI=1S/C13H10BrClF5NO6S3/c1-28(24,25)10-5-7(30(16,17,18,19)20)4-9(13(10)23)21-29(26,27)11-3-6(14)2-8(15)12(11)22/h2-5,21-23H,1H3	VXOKTNHNKMORHH-UHFFFAOYSA-N	50531131	CHEMBL4552035	WD repeat-containing protein 5				 45						ChEMBL	10.1021/acs.jmedchem.9b01411	10.7270/Q2B85CM0	31724864			Macdonald, JD; Chacón Simon, S; Han, C; Wang, F; Shaw, JG; Howes, JE; Sai, J; Yuh, JP; Camper, D; Alicie, BM; Alvarado, J; Nikhar, S; Payne, W; Aho, ER; Bauer, JA; Zhao, B; Phan, J; Thomas, LR; Rossanese, OW; Tansey, WP; Waterson, AG; Stauffer, SR; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50531131	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50531131&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			155555468	440739713							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51308098	CS(=O)(=O)c1cc(NS(=O)(=O)c2cc(Br)cc(Cl)c2O)cc(c1)C1(CCC1)C#N	InChI=1S/C18H16BrClN2O5S2/c1-28(24,25)14-6-11(18(10-21)3-2-4-18)5-13(9-14)22-29(26,27)16-8-12(19)7-15(20)17(16)23/h5-9,22-23H,2-4H2,1H3	AVODLYHEBPIIPG-UHFFFAOYSA-N	50531110	CHEMBL4447845	WD repeat-containing protein 5				 215						ChEMBL	10.1021/acs.jmedchem.9b01411	10.7270/Q2B85CM0	31724864			Macdonald, JD; Chacón Simon, S; Han, C; Wang, F; Shaw, JG; Howes, JE; Sai, J; Yuh, JP; Camper, D; Alicie, BM; Alvarado, J; Nikhar, S; Payne, W; Aho, ER; Bauer, JA; Zhao, B; Phan, J; Thomas, LR; Rossanese, OW; Tansey, WP; Waterson, AG; Stauffer, SR; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50531110	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50531110&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			155519558	440739692							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51308099	CS(=O)(=O)c1cc(cc(NS(=O)(=O)c2cc(Br)ccc2O)c1O)C1(CCC1)C#N	InChI=1S/C18H17BrN2O6S2/c1-28(24,25)16-8-11(18(10-20)5-2-6-18)7-13(17(16)23)21-29(26,27)15-9-12(19)3-4-14(15)22/h3-4,7-9,21-23H,2,5-6H2,1H3	ZOQUNXATFSLGSS-UHFFFAOYSA-N	50531111	CHEMBL4465645	WD repeat-containing protein 5				 349						ChEMBL	10.1021/acs.jmedchem.9b01411	10.7270/Q2B85CM0	31724864			Macdonald, JD; Chacón Simon, S; Han, C; Wang, F; Shaw, JG; Howes, JE; Sai, J; Yuh, JP; Camper, D; Alicie, BM; Alvarado, J; Nikhar, S; Payne, W; Aho, ER; Bauer, JA; Zhao, B; Phan, J; Thomas, LR; Rossanese, OW; Tansey, WP; Waterson, AG; Stauffer, SR; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50531111	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50531111&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			155531053	440739693							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51308100	COc1ccc(Br)cc1S(=O)(=O)Nc1cc(Cl)cc(c1O)S(C)(=O)=O	InChI=1S/C14H13BrClNO6S2/c1-23-11-4-3-8(15)5-12(11)25(21,22)17-10-6-9(16)7-13(14(10)18)24(2,19)20/h3-7,17-18H,1-2H3	XSNDBCXTZMGFDN-UHFFFAOYSA-N	50531070	CHEMBL4532703	WD repeat-containing protein 5				 304						ChEMBL	10.1021/acs.jmedchem.9b01411	10.7270/Q2B85CM0	31724864			Macdonald, JD; Chacón Simon, S; Han, C; Wang, F; Shaw, JG; Howes, JE; Sai, J; Yuh, JP; Camper, D; Alicie, BM; Alvarado, J; Nikhar, S; Payne, W; Aho, ER; Bauer, JA; Zhao, B; Phan, J; Thomas, LR; Rossanese, OW; Tansey, WP; Waterson, AG; Stauffer, SR; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50531070	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50531070&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			155547690	440739652							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51308101	CNC(=O)c1cc(cc(NS(=O)(=O)c2cc(Br)ccc2OC)c1O)C1(CCC1)C#N	InChI=1S/C20H20BrN3O5S/c1-23-19(26)14-8-12(20(11-22)6-3-7-20)9-15(18(14)25)24-30(27,28)17-10-13(21)4-5-16(17)29-2/h4-5,8-10,24-25H,3,6-7H2,1-2H3,(H,23,26)	OGIHPKRHJNELFY-UHFFFAOYSA-N	50531121	CHEMBL4464746	WD repeat-containing protein 5				 906						ChEMBL	10.1021/acs.jmedchem.9b01411	10.7270/Q2B85CM0	31724864			Macdonald, JD; Chacón Simon, S; Han, C; Wang, F; Shaw, JG; Howes, JE; Sai, J; Yuh, JP; Camper, D; Alicie, BM; Alvarado, J; Nikhar, S; Payne, W; Aho, ER; Bauer, JA; Zhao, B; Phan, J; Thomas, LR; Rossanese, OW; Tansey, WP; Waterson, AG; Stauffer, SR; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50531121	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50531121&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			155530388	440739703							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51308102	OC(=O)c1cc(cc(NS(=O)(=O)c2cc(Br)cc3cccnc23)c1O)S(F)(F)(F)(F)F	InChI=1S/C16H10BrF5N2O5S2/c17-9-4-8-2-1-3-23-14(8)13(5-9)30(28,29)24-12-7-10(31(18,19,20,21)22)6-11(15(12)25)16(26)27/h1-7,24-25H,(H,26,27)	HTNUDGDQTGKVCW-UHFFFAOYSA-N	50531114	CHEMBL4468085	WD repeat-containing protein 5				 47						ChEMBL	10.1021/acs.jmedchem.9b01411	10.7270/Q2B85CM0	31724864			Macdonald, JD; Chacón Simon, S; Han, C; Wang, F; Shaw, JG; Howes, JE; Sai, J; Yuh, JP; Camper, D; Alicie, BM; Alvarado, J; Nikhar, S; Payne, W; Aho, ER; Bauer, JA; Zhao, B; Phan, J; Thomas, LR; Rossanese, OW; Tansey, WP; Waterson, AG; Stauffer, SR; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50531114	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50531114&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			155533048	440739696							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51308103	CNC(=O)c1cc(cc(NS(=O)(=O)c2cc(Br)cc3cccnc23)c1O)S(F)(F)(F)(F)F	InChI=1S/C17H13BrF5N3O4S2/c1-24-17(28)12-7-11(32(19,20,21,22)23)8-13(16(12)27)26-31(29,30)14-6-10(18)5-9-3-2-4-25-15(9)14/h2-8,26-27H,1H3,(H,24,28)	YJHTXYKBEWYLEI-UHFFFAOYSA-N	50531132	CHEMBL4578283	WD repeat-containing protein 5				 122						ChEMBL	10.1021/acs.jmedchem.9b01411	10.7270/Q2B85CM0	31724864			Macdonald, JD; Chacón Simon, S; Han, C; Wang, F; Shaw, JG; Howes, JE; Sai, J; Yuh, JP; Camper, D; Alicie, BM; Alvarado, J; Nikhar, S; Payne, W; Aho, ER; Bauer, JA; Zhao, B; Phan, J; Thomas, LR; Rossanese, OW; Tansey, WP; Waterson, AG; Stauffer, SR; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50531132	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50531132&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			155564871	440739714							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51308104	Oc1ccc(Cl)cc1NS(=O)(=O)c1cccc(Br)c1	InChI=1S/C12H9BrClNO3S/c13-8-2-1-3-10(6-8)19(17,18)15-11-7-9(14)4-5-12(11)16/h1-7,15-16H	BYEKHFXVAPCFIJ-UHFFFAOYSA-N	50531123	CHEMBL4574127	WD repeat-containing protein 5				 36100						ChEMBL	10.1021/acs.jmedchem.9b01411	10.7270/Q2B85CM0	31724864			Macdonald, JD; Chacón Simon, S; Han, C; Wang, F; Shaw, JG; Howes, JE; Sai, J; Yuh, JP; Camper, D; Alicie, BM; Alvarado, J; Nikhar, S; Payne, W; Aho, ER; Bauer, JA; Zhao, B; Phan, J; Thomas, LR; Rossanese, OW; Tansey, WP; Waterson, AG; Stauffer, SR; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50531123	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50531123&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			28973441	440739705							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51308105	COc1ccc(Br)cc1S(=O)(=O)Nc1cc(ccc1O)-c1ccccc1	InChI=1S/C19H16BrNO4S/c1-25-18-10-8-15(20)12-19(18)26(23,24)21-16-11-14(7-9-17(16)22)13-5-3-2-4-6-13/h2-12,21-22H,1H3	LSOYIZUYLCYRNG-UHFFFAOYSA-N	50531124	CHEMBL4443499	WD repeat-containing protein 5				 37000						ChEMBL	10.1021/acs.jmedchem.9b01411	10.7270/Q2B85CM0	31724864			Macdonald, JD; Chacón Simon, S; Han, C; Wang, F; Shaw, JG; Howes, JE; Sai, J; Yuh, JP; Camper, D; Alicie, BM; Alvarado, J; Nikhar, S; Payne, W; Aho, ER; Bauer, JA; Zhao, B; Phan, J; Thomas, LR; Rossanese, OW; Tansey, WP; Waterson, AG; Stauffer, SR; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50531124	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50531124&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	Q1J	6U80	145704699	440739706							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51308106	Oc1ccc(cc1NS(=O)(=O)c1cc(Br)ccc1O)C1(CC1)C#N	InChI=1S/C16H13BrN2O4S/c17-11-2-4-14(21)15(8-11)24(22,23)19-12-7-10(1-3-13(12)20)16(9-18)5-6-16/h1-4,7-8,19-21H,5-6H2	BZJQKWLSPXGRHB-UHFFFAOYSA-N	50531125	CHEMBL4436954	WD repeat-containing protein 5				 852						ChEMBL	10.1021/acs.jmedchem.9b01411	10.7270/Q2B85CM0	31724864			Macdonald, JD; Chacón Simon, S; Han, C; Wang, F; Shaw, JG; Howes, JE; Sai, J; Yuh, JP; Camper, D; Alicie, BM; Alvarado, J; Nikhar, S; Payne, W; Aho, ER; Bauer, JA; Zhao, B; Phan, J; Thomas, LR; Rossanese, OW; Tansey, WP; Waterson, AG; Stauffer, SR; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50531125	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50531125&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			155512250	440739707							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51308107	COc1ccc(Br)cc1S(=O)(=O)Nc1cc(Cl)cc(C(O)=O)c1O	InChI=1S/C14H11BrClNO6S/c1-23-11-3-2-7(15)4-12(11)24(21,22)17-10-6-8(16)5-9(13(10)18)14(19)20/h2-6,17-18H,1H3,(H,19,20)	HLGWNAJQDWZVDI-UHFFFAOYSA-N	50531133	CHEMBL4515727	WD repeat-containing protein 5				 431						ChEMBL	10.1021/acs.jmedchem.9b01411	10.7270/Q2B85CM0	31724864			Macdonald, JD; Chacón Simon, S; Han, C; Wang, F; Shaw, JG; Howes, JE; Sai, J; Yuh, JP; Camper, D; Alicie, BM; Alvarado, J; Nikhar, S; Payne, W; Aho, ER; Bauer, JA; Zhao, B; Phan, J; Thomas, LR; Rossanese, OW; Tansey, WP; Waterson, AG; Stauffer, SR; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50531133	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50531133&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	Q1M	6U8B	145704700	440739715							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51308108	OC(=O)c1c(O)c(NS(=O)(=O)c2cc(Br)ccc2O)cc(C2CC2)c1F	InChI=1S/C16H13BrFNO6S/c17-8-3-4-11(20)12(5-8)26(24,25)19-10-6-9(7-1-2-7)14(18)13(15(10)21)16(22)23/h3-7,19-21H,1-2H2,(H,22,23)	LZQVQCAIOFNYFL-UHFFFAOYSA-N	50531134	CHEMBL4471200	WD repeat-containing protein 5				 122						ChEMBL	10.1021/acs.jmedchem.9b01411	10.7270/Q2B85CM0	31724864			Macdonald, JD; Chacón Simon, S; Han, C; Wang, F; Shaw, JG; Howes, JE; Sai, J; Yuh, JP; Camper, D; Alicie, BM; Alvarado, J; Nikhar, S; Payne, W; Aho, ER; Bauer, JA; Zhao, B; Phan, J; Thomas, LR; Rossanese, OW; Tansey, WP; Waterson, AG; Stauffer, SR; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50531134	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50531134&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	Q1P	6U8L	145704701	440739716							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51308109	OC(=O)c1cc(OC(F)(F)F)cc(NS(=O)(=O)c2cc(Br)cc(Cl)c2O)c1O	InChI=1S/C14H8BrClF3NO7S/c15-5-1-8(16)12(22)10(2-5)28(25,26)20-9-4-6(27-14(17,18)19)3-7(11(9)21)13(23)24/h1-4,20-22H,(H,23,24)	NJAWBWFLAWGPAQ-UHFFFAOYSA-N	50531127	CHEMBL4529202	WD repeat-containing protein 5				 51						ChEMBL	10.1021/acs.jmedchem.9b01411	10.7270/Q2B85CM0	31724864			Macdonald, JD; Chacón Simon, S; Han, C; Wang, F; Shaw, JG; Howes, JE; Sai, J; Yuh, JP; Camper, D; Alicie, BM; Alvarado, J; Nikhar, S; Payne, W; Aho, ER; Bauer, JA; Zhao, B; Phan, J; Thomas, LR; Rossanese, OW; Tansey, WP; Waterson, AG; Stauffer, SR; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50531127	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50531127&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			155545363	440739709							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51308110	OC(=O)c1cc(cc(NS(=O)(=O)c2cc(Br)ccc2O)c1O)C1(CCC1)C#N	InChI=1S/C18H15BrN2O6S/c19-11-2-3-14(22)15(8-11)28(26,27)21-13-7-10(18(9-20)4-1-5-18)6-12(16(13)23)17(24)25/h2-3,6-8,21-23H,1,4-5H2,(H,24,25)	BLJKTQGNFJGAOA-UHFFFAOYSA-N	50531135	CHEMBL4441676	WD repeat-containing protein 5				 67						ChEMBL	10.1021/acs.jmedchem.9b01411	10.7270/Q2B85CM0	31724864			Macdonald, JD; Chacón Simon, S; Han, C; Wang, F; Shaw, JG; Howes, JE; Sai, J; Yuh, JP; Camper, D; Alicie, BM; Alvarado, J; Nikhar, S; Payne, W; Aho, ER; Bauer, JA; Zhao, B; Phan, J; Thomas, LR; Rossanese, OW; Tansey, WP; Waterson, AG; Stauffer, SR; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50531135	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50531135&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			155515379	440739717							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51308111	CNC(=O)c1cc(Cl)cc(NS(=O)(=O)c2cc(Br)cc(Cl)c2O)c1O	InChI=1S/C14H11BrCl2N2O5S/c1-18-14(22)8-4-7(16)5-10(12(8)20)19-25(23,24)11-3-6(15)2-9(17)13(11)21/h2-5,19-21H,1H3,(H,18,22)	ZMZHJGCDYATWCC-UHFFFAOYSA-N	50531136	CHEMBL4535470	WD repeat-containing protein 5				 298						ChEMBL	10.1021/acs.jmedchem.9b01411	10.7270/Q2B85CM0	31724864			Macdonald, JD; Chacón Simon, S; Han, C; Wang, F; Shaw, JG; Howes, JE; Sai, J; Yuh, JP; Camper, D; Alicie, BM; Alvarado, J; Nikhar, S; Payne, W; Aho, ER; Bauer, JA; Zhao, B; Phan, J; Thomas, LR; Rossanese, OW; Tansey, WP; Waterson, AG; Stauffer, SR; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50531136	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50531136&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			155547629	440739718							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51308112	CNC(=O)c1cc(NS(=O)(=O)c2cc(Br)ccc2O)cc(c1)C1(CCC1)C#N	InChI=1S/C19H18BrN3O4S/c1-22-18(25)12-7-13(19(11-21)5-2-6-19)9-15(8-12)23-28(26,27)17-10-14(20)3-4-16(17)24/h3-4,7-10,23-24H,2,5-6H2,1H3,(H,22,25)	HTDHGPQJWJSDGO-UHFFFAOYSA-N	50531081	CHEMBL4593558	WD repeat-containing protein 5				 1080						ChEMBL	10.1021/acs.jmedchem.9b01411	10.7270/Q2B85CM0	31724864			Macdonald, JD; Chacón Simon, S; Han, C; Wang, F; Shaw, JG; Howes, JE; Sai, J; Yuh, JP; Camper, D; Alicie, BM; Alvarado, J; Nikhar, S; Payne, W; Aho, ER; Bauer, JA; Zhao, B; Phan, J; Thomas, LR; Rossanese, OW; Tansey, WP; Waterson, AG; Stauffer, SR; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50531081	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50531081&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			155569685	440739663							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51308113	CNC(=O)c1cc(cc(NS(=O)(=O)c2cc(Br)ccc2O)c1O)C1(CCCCC1)C#N	InChI=1S/C21H22BrN3O5S/c1-24-20(28)15-9-13(21(12-23)7-3-2-4-8-21)10-16(19(15)27)25-31(29,30)18-11-14(22)5-6-17(18)26/h5-6,9-11,25-27H,2-4,7-8H2,1H3,(H,24,28)	CTKLAWJIXCJAIO-UHFFFAOYSA-N	50531137	CHEMBL4583214	WD repeat-containing protein 5				 779						ChEMBL	10.1021/acs.jmedchem.9b01411	10.7270/Q2B85CM0	31724864			Macdonald, JD; Chacón Simon, S; Han, C; Wang, F; Shaw, JG; Howes, JE; Sai, J; Yuh, JP; Camper, D; Alicie, BM; Alvarado, J; Nikhar, S; Payne, W; Aho, ER; Bauer, JA; Zhao, B; Phan, J; Thomas, LR; Rossanese, OW; Tansey, WP; Waterson, AG; Stauffer, SR; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50531137	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50531137&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			155566223	440739719							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51308114	CS(=O)(=O)c1cc(Cl)cc(NS(=O)(=O)c2cc(Br)cc(Cl)c2O)c1	InChI=1S/C13H10BrCl2NO5S2/c1-23(19,20)10-5-8(15)4-9(6-10)17-24(21,22)12-3-7(14)2-11(16)13(12)18/h2-6,17-18H,1H3	WYGIOFXYDQDPBX-UHFFFAOYSA-N	50531130	CHEMBL4534549	WD repeat-containing protein 5				 220						ChEMBL	10.1021/acs.jmedchem.9b01411	10.7270/Q2B85CM0	31724864			Macdonald, JD; Chacón Simon, S; Han, C; Wang, F; Shaw, JG; Howes, JE; Sai, J; Yuh, JP; Camper, D; Alicie, BM; Alvarado, J; Nikhar, S; Payne, W; Aho, ER; Bauer, JA; Zhao, B; Phan, J; Thomas, LR; Rossanese, OW; Tansey, WP; Waterson, AG; Stauffer, SR; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50531130	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50531130&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			155547031	440739712							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51308115	CS(=O)(=O)c1cc(cc(NS(=O)(=O)c2cc(Br)cc(Cl)c2O)c1O)S(F)(F)(F)(F)F	InChI=1S/C13H10BrClF5NO6S3/c1-28(24,25)10-5-7(30(16,17,18,19)20)4-9(13(10)23)21-29(26,27)11-3-6(14)2-8(15)12(11)22/h2-5,21-23H,1H3	VXOKTNHNKMORHH-UHFFFAOYSA-N	50531131	CHEMBL4552035	WD repeat-containing protein 5				 45						ChEMBL	10.1021/acs.jmedchem.9b01411	10.7270/Q2B85CM0	31724864			Macdonald, JD; Chacón Simon, S; Han, C; Wang, F; Shaw, JG; Howes, JE; Sai, J; Yuh, JP; Camper, D; Alicie, BM; Alvarado, J; Nikhar, S; Payne, W; Aho, ER; Bauer, JA; Zhao, B; Phan, J; Thomas, LR; Rossanese, OW; Tansey, WP; Waterson, AG; Stauffer, SR; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50531131	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50531131&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			155555468	440739713							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51308116	COc1ccc(Br)cc1S(=O)(=O)Nc1ccc(Cl)cc1O	InChI=1S/C13H11BrClNO4S/c1-20-12-5-2-8(14)6-13(12)21(18,19)16-10-4-3-9(15)7-11(10)17/h2-7,16-17H,1H3	BZVGTEQHABVNJF-UHFFFAOYSA-N	50531138	CHEMBL4550667	WD repeat-containing protein 5				 27700						ChEMBL	10.1021/acs.jmedchem.9b01411	10.7270/Q2B85CM0	31724864			Macdonald, JD; Chacón Simon, S; Han, C; Wang, F; Shaw, JG; Howes, JE; Sai, J; Yuh, JP; Camper, D; Alicie, BM; Alvarado, J; Nikhar, S; Payne, W; Aho, ER; Bauer, JA; Zhao, B; Phan, J; Thomas, LR; Rossanese, OW; Tansey, WP; Waterson, AG; Stauffer, SR; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50531138	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50531138&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			155555207	440739720							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51308117	CNC(=O)c1cc(cc(NS(=O)(=O)c2cc(Br)cc3cccnc23)c1O)C1(CCC1)C#N	InChI=1S/C22H19BrN4O4S/c1-25-21(29)16-9-14(22(12-24)5-3-6-22)10-17(20(16)28)27-32(30,31)18-11-15(23)8-13-4-2-7-26-19(13)18/h2,4,7-11,27-28H,3,5-6H2,1H3,(H,25,29)	LUHBUKXZMCITBQ-UHFFFAOYSA-N	50531139	CHEMBL4457793	WD repeat-containing protein 5				 825						ChEMBL	10.1021/acs.jmedchem.9b01411	10.7270/Q2B85CM0	31724864			Macdonald, JD; Chacón Simon, S; Han, C; Wang, F; Shaw, JG; Howes, JE; Sai, J; Yuh, JP; Camper, D; Alicie, BM; Alvarado, J; Nikhar, S; Payne, W; Aho, ER; Bauer, JA; Zhao, B; Phan, J; Thomas, LR; Rossanese, OW; Tansey, WP; Waterson, AG; Stauffer, SR; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50531139	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50531139&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			155526271	440739721							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51308118	CCOc1ccc(c(C)c1C)S(=O)(=O)Nc1ccccc1C(O)=O	InChI=1S/C17H19NO5S/c1-4-23-15-9-10-16(12(3)11(15)2)24(21,22)18-14-8-6-5-7-13(14)17(19)20/h5-10,18H,4H2,1-3H3,(H,19,20)	PYUYEJJTRWPEAM-UHFFFAOYSA-N	50531140	CHEMBL4440417	WD repeat-containing protein 5				>125000						ChEMBL	10.1021/acs.jmedchem.9b01411	10.7270/Q2B85CM0	31724864			Macdonald, JD; Chacón Simon, S; Han, C; Wang, F; Shaw, JG; Howes, JE; Sai, J; Yuh, JP; Camper, D; Alicie, BM; Alvarado, J; Nikhar, S; Payne, W; Aho, ER; Bauer, JA; Zhao, B; Phan, J; Thomas, LR; Rossanese, OW; Tansey, WP; Waterson, AG; Stauffer, SR; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50531140	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50531140&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			15944072	440739722							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51308119	CCOc1ccc(c(C)c1C)S(=O)(=O)Nc1ccccc1C(O)=O	InChI=1S/C17H19NO5S/c1-4-23-15-9-10-16(12(3)11(15)2)24(21,22)18-14-8-6-5-7-13(14)17(19)20/h5-10,18H,4H2,1-3H3,(H,19,20)	PYUYEJJTRWPEAM-UHFFFAOYSA-N	50531140	CHEMBL4440417	WD repeat-containing protein 5				>125000						ChEMBL	10.1021/acs.jmedchem.9b01411	10.7270/Q2B85CM0	31724864			Macdonald, JD; Chacón Simon, S; Han, C; Wang, F; Shaw, JG; Howes, JE; Sai, J; Yuh, JP; Camper, D; Alicie, BM; Alvarado, J; Nikhar, S; Payne, W; Aho, ER; Bauer, JA; Zhao, B; Phan, J; Thomas, LR; Rossanese, OW; Tansey, WP; Waterson, AG; Stauffer, SR; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50531140	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50531140&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			15944072	440739722							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51308120	CNC(=O)c1cc(cc(NS(=O)(=O)c2cc(Br)cc(Cl)c2O)c1O)C1(CCCCC1)C#N	InChI=1S/C21H21BrClN3O5S/c1-25-20(29)14-7-12(21(11-24)5-3-2-4-6-21)8-16(18(14)27)26-32(30,31)17-10-13(22)9-15(23)19(17)28/h7-10,26-28H,2-6H2,1H3,(H,25,29)	RFZNGPIYBXOUDK-UHFFFAOYSA-N	50531106	CHEMBL4441794	WD repeat-containing protein 5				 362						ChEMBL	10.1021/acs.jmedchem.9b01411	10.7270/Q2B85CM0	31724864			Macdonald, JD; Chacón Simon, S; Han, C; Wang, F; Shaw, JG; Howes, JE; Sai, J; Yuh, JP; Camper, D; Alicie, BM; Alvarado, J; Nikhar, S; Payne, W; Aho, ER; Bauer, JA; Zhao, B; Phan, J; Thomas, LR; Rossanese, OW; Tansey, WP; Waterson, AG; Stauffer, SR; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50531106	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50531106&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			155515725	440739688							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51308121	CNC(=O)c1cc(cc(NS(=O)(=O)c2cc(Br)cc3cccnc23)c1O)S(F)(F)(F)(F)F	InChI=1S/C17H13BrF5N3O4S2/c1-24-17(28)12-7-11(32(19,20,21,22)23)8-13(16(12)27)26-31(29,30)14-6-10(18)5-9-3-2-4-25-15(9)14/h2-8,26-27H,1H3,(H,24,28)	YJHTXYKBEWYLEI-UHFFFAOYSA-N	50531132	CHEMBL4578283	WD repeat-containing protein 5				 122						ChEMBL	10.1021/acs.jmedchem.9b01411	10.7270/Q2B85CM0	31724864			Macdonald, JD; Chacón Simon, S; Han, C; Wang, F; Shaw, JG; Howes, JE; Sai, J; Yuh, JP; Camper, D; Alicie, BM; Alvarado, J; Nikhar, S; Payne, W; Aho, ER; Bauer, JA; Zhao, B; Phan, J; Thomas, LR; Rossanese, OW; Tansey, WP; Waterson, AG; Stauffer, SR; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50531132	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50531132&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			155564871	440739714							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51308122	OC(=O)c1cc(NS(=O)(=O)c2cc(Br)cc(Cl)c2O)cc(c1)S(F)(F)(F)(F)F	InChI=1S/C13H8BrClF5NO5S2/c14-7-3-10(15)12(22)11(4-7)27(25,26)21-8-1-6(13(23)24)2-9(5-8)28(16,17,18,19)20/h1-5,21-22H,(H,23,24)	WPAFXJRBUSFEDN-UHFFFAOYSA-N	50531141	CHEMBL4446534	WD repeat-containing protein 5				 29						ChEMBL	10.1021/acs.jmedchem.9b01411	10.7270/Q2B85CM0	31724864			Macdonald, JD; Chacón Simon, S; Han, C; Wang, F; Shaw, JG; Howes, JE; Sai, J; Yuh, JP; Camper, D; Alicie, BM; Alvarado, J; Nikhar, S; Payne, W; Aho, ER; Bauer, JA; Zhao, B; Phan, J; Thomas, LR; Rossanese, OW; Tansey, WP; Waterson, AG; Stauffer, SR; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50531141	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50531141&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			155518416	440739723							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51308123	OC(=O)c1cc(NS(=O)(=O)c2cc(Br)cc(Cl)c2O)cc(c1)S(F)(F)(F)(F)F	InChI=1S/C13H8BrClF5NO5S2/c14-7-3-10(15)12(22)11(4-7)27(25,26)21-8-1-6(13(23)24)2-9(5-8)28(16,17,18,19)20/h1-5,21-22H,(H,23,24)	WPAFXJRBUSFEDN-UHFFFAOYSA-N	50531141	CHEMBL4446534	WD repeat-containing protein 5				 29						ChEMBL	10.1021/acs.jmedchem.9b01411	10.7270/Q2B85CM0	31724864			Macdonald, JD; Chacón Simon, S; Han, C; Wang, F; Shaw, JG; Howes, JE; Sai, J; Yuh, JP; Camper, D; Alicie, BM; Alvarado, J; Nikhar, S; Payne, W; Aho, ER; Bauer, JA; Zhao, B; Phan, J; Thomas, LR; Rossanese, OW; Tansey, WP; Waterson, AG; Stauffer, SR; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50531141	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50531141&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			155518416	440739723							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51308124	CNC(=O)c1cc(Cl)cc(NS(=O)(=O)c2cc(Br)cc(Cl)c2O)c1O	InChI=1S/C14H11BrCl2N2O5S/c1-18-14(22)8-4-7(16)5-10(12(8)20)19-25(23,24)11-3-6(15)2-9(17)13(11)21/h2-5,19-21H,1H3,(H,18,22)	ZMZHJGCDYATWCC-UHFFFAOYSA-N	50531136	CHEMBL4535470	WD repeat-containing protein 5				 298						ChEMBL	10.1021/acs.jmedchem.9b01411	10.7270/Q2B85CM0	31724864			Macdonald, JD; Chacón Simon, S; Han, C; Wang, F; Shaw, JG; Howes, JE; Sai, J; Yuh, JP; Camper, D; Alicie, BM; Alvarado, J; Nikhar, S; Payne, W; Aho, ER; Bauer, JA; Zhao, B; Phan, J; Thomas, LR; Rossanese, OW; Tansey, WP; Waterson, AG; Stauffer, SR; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50531136	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50531136&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			155547629	440739718							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51308125	CS(=O)(=O)c1cc(Cl)cc(NS(=O)(=O)c2cc(Br)ccc2O)c1O	InChI=1S/C13H11BrClNO6S2/c1-23(19,20)12-6-8(15)5-9(13(12)18)16-24(21,22)11-4-7(14)2-3-10(11)17/h2-6,16-18H,1H3	PRESXYPRJSJGMN-UHFFFAOYSA-N	50531142	CHEMBL4535863	WD repeat-containing protein 5				 1070						ChEMBL	10.1021/acs.jmedchem.9b01411	10.7270/Q2B85CM0	31724864			Macdonald, JD; Chacón Simon, S; Han, C; Wang, F; Shaw, JG; Howes, JE; Sai, J; Yuh, JP; Camper, D; Alicie, BM; Alvarado, J; Nikhar, S; Payne, W; Aho, ER; Bauer, JA; Zhao, B; Phan, J; Thomas, LR; Rossanese, OW; Tansey, WP; Waterson, AG; Stauffer, SR; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50531142	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50531142&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			155547683	440739724							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51308126	CS(=O)(=O)c1cc(cc(NS(=O)(=O)c2cc(Br)cc(Cl)c2O)c1O)C1(CCC1)C#N	InChI=1S/C18H16BrClN2O6S2/c1-29(25,26)14-6-10(18(9-21)3-2-4-18)5-13(17(14)24)22-30(27,28)15-8-11(19)7-12(20)16(15)23/h5-8,22-24H,2-4H2,1H3	SUJUXKUBROGCLA-UHFFFAOYSA-N	50531112	CHEMBL4573903	WD repeat-containing protein 5				 110						ChEMBL	10.1021/acs.jmedchem.9b01411	10.7270/Q2B85CM0	31724864			Macdonald, JD; Chacón Simon, S; Han, C; Wang, F; Shaw, JG; Howes, JE; Sai, J; Yuh, JP; Camper, D; Alicie, BM; Alvarado, J; Nikhar, S; Payne, W; Aho, ER; Bauer, JA; Zhao, B; Phan, J; Thomas, LR; Rossanese, OW; Tansey, WP; Waterson, AG; Stauffer, SR; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50531112	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50531112&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			155563363	440739694							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51308127	Oc1ccc(Cl)cc1NS(=O)(=O)c1cc(Br)ccc1O	InChI=1S/C12H9BrClNO4S/c13-7-1-3-11(17)12(5-7)20(18,19)15-9-6-8(14)2-4-10(9)16/h1-6,15-17H	NVBGVGWRMDACKA-UHFFFAOYSA-N	50531087	CHEMBL4470230	WD repeat-containing protein 5				 1250						ChEMBL	10.1021/acs.jmedchem.9b01411	10.7270/Q2B85CM0	31724864			Macdonald, JD; Chacón Simon, S; Han, C; Wang, F; Shaw, JG; Howes, JE; Sai, J; Yuh, JP; Camper, D; Alicie, BM; Alvarado, J; Nikhar, S; Payne, W; Aho, ER; Bauer, JA; Zhao, B; Phan, J; Thomas, LR; Rossanese, OW; Tansey, WP; Waterson, AG; Stauffer, SR; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50531087	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50531087&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			155534245	440739669							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51308128	COc1ccc(Br)cc1S(=O)(=O)Nc1cc(Cl)cc(C(O)=O)c1O	InChI=1S/C14H11BrClNO6S/c1-23-11-3-2-7(15)4-12(11)24(21,22)17-10-6-8(16)5-9(13(10)18)14(19)20/h2-6,17-18H,1H3,(H,19,20)	HLGWNAJQDWZVDI-UHFFFAOYSA-N	50531133	CHEMBL4515727	WD repeat-containing protein 5				 431						ChEMBL	10.1021/acs.jmedchem.9b01411	10.7270/Q2B85CM0	31724864			Macdonald, JD; Chacón Simon, S; Han, C; Wang, F; Shaw, JG; Howes, JE; Sai, J; Yuh, JP; Camper, D; Alicie, BM; Alvarado, J; Nikhar, S; Payne, W; Aho, ER; Bauer, JA; Zhao, B; Phan, J; Thomas, LR; Rossanese, OW; Tansey, WP; Waterson, AG; Stauffer, SR; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50531133	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50531133&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	Q1M	6U8B	145704700	440739715							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51308129	OC(=O)c1cc(cc(NS(=O)(=O)c2cc(Br)ccc2O)c1O)S(F)(F)(F)(F)F	InChI=1S/C13H9BrF5NO6S2/c14-6-1-2-10(21)11(3-6)27(25,26)20-9-5-7(28(15,16,17,18)19)4-8(12(9)22)13(23)24/h1-5,20-22H,(H,23,24)	QJKRMFMEFICLPS-UHFFFAOYSA-N	50531097	CHEMBL4544635	WD repeat-containing protein 5				 47						ChEMBL	10.1021/acs.jmedchem.9b01411	10.7270/Q2B85CM0	31724864			Macdonald, JD; Chacón Simon, S; Han, C; Wang, F; Shaw, JG; Howes, JE; Sai, J; Yuh, JP; Camper, D; Alicie, BM; Alvarado, J; Nikhar, S; Payne, W; Aho, ER; Bauer, JA; Zhao, B; Phan, J; Thomas, LR; Rossanese, OW; Tansey, WP; Waterson, AG; Stauffer, SR; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50531097	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50531097&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			155552825	440739679							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51308130	CS(=O)(=O)c1cc(NS(=O)(=O)c2cc(Br)ccc2O)cc(c1)S(F)(F)(F)(F)F	InChI=1S/C13H11BrF5NO5S3/c1-26(22,23)10-5-9(6-11(7-10)28(15,16,17,18)19)20-27(24,25)13-4-8(14)2-3-12(13)21/h2-7,20-21H,1H3	GXKWWSXTDOWSFB-UHFFFAOYSA-N	50531075	CHEMBL4475470	WD repeat-containing protein 5				 511						ChEMBL	10.1021/acs.jmedchem.9b01411	10.7270/Q2B85CM0	31724864			Macdonald, JD; Chacón Simon, S; Han, C; Wang, F; Shaw, JG; Howes, JE; Sai, J; Yuh, JP; Camper, D; Alicie, BM; Alvarado, J; Nikhar, S; Payne, W; Aho, ER; Bauer, JA; Zhao, B; Phan, J; Thomas, LR; Rossanese, OW; Tansey, WP; Waterson, AG; Stauffer, SR; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50531075	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50531075&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	Q0S	6U5M	145704697	440739657							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51308131	OC(=O)c1cc(cc(NS(=O)(=O)c2cc(Br)cc3cccnc23)c1O)C1(CCC1)C#N	InChI=1S/C21H16BrN3O5S/c22-14-7-12-3-1-6-24-18(12)17(10-14)31(29,30)25-16-9-13(21(11-23)4-2-5-21)8-15(19(16)26)20(27)28/h1,3,6-10,25-26H,2,4-5H2,(H,27,28)	YBOXBNDKAUHBOR-UHFFFAOYSA-N	50531143	CHEMBL4528788	WD repeat-containing protein 5				 104						ChEMBL	10.1021/acs.jmedchem.9b01411	10.7270/Q2B85CM0	31724864			Macdonald, JD; Chacón Simon, S; Han, C; Wang, F; Shaw, JG; Howes, JE; Sai, J; Yuh, JP; Camper, D; Alicie, BM; Alvarado, J; Nikhar, S; Payne, W; Aho, ER; Bauer, JA; Zhao, B; Phan, J; Thomas, LR; Rossanese, OW; Tansey, WP; Waterson, AG; Stauffer, SR; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50531143	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50531143&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			155545084	440739725							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51308132	CS(=O)(=O)c1cc(cc(NS(=O)(=O)c2cc(Br)cc3cccnc23)c1O)C1(CCC1)C#N	InChI=1S/C21H18BrN3O5S2/c1-31(27,28)18-10-14(21(12-23)5-3-6-21)9-16(20(18)26)25-32(29,30)17-11-15(22)8-13-4-2-7-24-19(13)17/h2,4,7-11,25-26H,3,5-6H2,1H3	ZMYXSAKLPAHVLY-UHFFFAOYSA-N	50531115	CHEMBL4476737	WD repeat-containing protein 5				 272						ChEMBL	10.1021/acs.jmedchem.9b01411	10.7270/Q2B85CM0	31724864			Macdonald, JD; Chacón Simon, S; Han, C; Wang, F; Shaw, JG; Howes, JE; Sai, J; Yuh, JP; Camper, D; Alicie, BM; Alvarado, J; Nikhar, S; Payne, W; Aho, ER; Bauer, JA; Zhao, B; Phan, J; Thomas, LR; Rossanese, OW; Tansey, WP; Waterson, AG; Stauffer, SR; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50531115	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50531115&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			155538685	440739697							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51308133	Oc1ccc(cc1NS(=O)(=O)c1cc(Br)ccc1O)C1(CCCC1)C#N	InChI=1S/C18H17BrN2O4S/c19-13-4-6-16(23)17(10-13)26(24,25)21-14-9-12(3-5-15(14)22)18(11-20)7-1-2-8-18/h3-6,9-10,21-23H,1-2,7-8H2	IFBNCOFMJUTHRR-UHFFFAOYSA-N	50531126	CHEMBL4434999	WD repeat-containing protein 5				 614						ChEMBL	10.1021/acs.jmedchem.9b01411	10.7270/Q2B85CM0	31724864			Macdonald, JD; Chacón Simon, S; Han, C; Wang, F; Shaw, JG; Howes, JE; Sai, J; Yuh, JP; Camper, D; Alicie, BM; Alvarado, J; Nikhar, S; Payne, W; Aho, ER; Bauer, JA; Zhao, B; Phan, J; Thomas, LR; Rossanese, OW; Tansey, WP; Waterson, AG; Stauffer, SR; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50531126	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50531126&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			155511088	440739708							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51308134	CNC(=O)c1cc(NS(=O)(=O)c2cc(Br)ccc2O)cc(c1)S(F)(F)(F)(F)F	InChI=1S/C14H12BrF5N2O4S2/c1-21-14(24)8-4-10(7-11(5-8)28(16,17,18,19)20)22-27(25,26)13-6-9(15)2-3-12(13)23/h2-7,22-23H,1H3,(H,21,24)	JJPIOPKOYIGQSD-UHFFFAOYSA-N	50531128	CHEMBL4471513	WD repeat-containing protein 5				 848						ChEMBL	10.1021/acs.jmedchem.9b01411	10.7270/Q2B85CM0	31724864			Macdonald, JD; Chacón Simon, S; Han, C; Wang, F; Shaw, JG; Howes, JE; Sai, J; Yuh, JP; Camper, D; Alicie, BM; Alvarado, J; Nikhar, S; Payne, W; Aho, ER; Bauer, JA; Zhao, B; Phan, J; Thomas, LR; Rossanese, OW; Tansey, WP; Waterson, AG; Stauffer, SR; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50531128	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50531128&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			155535349	440739710							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51308135	OC(=O)c1cc(cc(NS(=O)(=O)c2cc(Br)cc3cccnc23)c1O)C1(CCC1)C#N	InChI=1S/C21H16BrN3O5S/c22-14-7-12-3-1-6-24-18(12)17(10-14)31(29,30)25-16-9-13(21(11-23)4-2-5-21)8-15(19(16)26)20(27)28/h1,3,6-10,25-26H,2,4-5H2,(H,27,28)	YBOXBNDKAUHBOR-UHFFFAOYSA-N	50531143	CHEMBL4528788	WD repeat-containing protein 5				 104						ChEMBL	10.1021/acs.jmedchem.9b01411	10.7270/Q2B85CM0	31724864			Macdonald, JD; Chacón Simon, S; Han, C; Wang, F; Shaw, JG; Howes, JE; Sai, J; Yuh, JP; Camper, D; Alicie, BM; Alvarado, J; Nikhar, S; Payne, W; Aho, ER; Bauer, JA; Zhao, B; Phan, J; Thomas, LR; Rossanese, OW; Tansey, WP; Waterson, AG; Stauffer, SR; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50531143	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50531143&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			155545084	440739725							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51308136	COc1ccc(I)cc1S(=O)(=O)Nc1cc(Cl)ccc1O	InChI=1S/C13H11ClINO4S/c1-20-12-5-3-9(15)7-13(12)21(18,19)16-10-6-8(14)2-4-11(10)17/h2-7,16-17H,1H3	LPFIQDGAKMDLDS-UHFFFAOYSA-N	50531122	CHEMBL4443470	WD repeat-containing protein 5				 8390						ChEMBL	10.1021/acs.jmedchem.9b01411	10.7270/Q2B85CM0	31724864			Macdonald, JD; Chacón Simon, S; Han, C; Wang, F; Shaw, JG; Howes, JE; Sai, J; Yuh, JP; Camper, D; Alicie, BM; Alvarado, J; Nikhar, S; Payne, W; Aho, ER; Bauer, JA; Zhao, B; Phan, J; Thomas, LR; Rossanese, OW; Tansey, WP; Waterson, AG; Stauffer, SR; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50531122	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50531122&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			155516611	440739704							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51308137	CS(=O)(=O)c1cc(Cl)cc(NS(=O)(=O)c2cc(Br)ccc2O)c1O	InChI=1S/C13H11BrClNO6S2/c1-23(19,20)12-6-8(15)5-9(13(12)18)16-24(21,22)11-4-7(14)2-3-10(11)17/h2-6,16-18H,1H3	PRESXYPRJSJGMN-UHFFFAOYSA-N	50531142	CHEMBL4535863	WD repeat-containing protein 5				 1070						ChEMBL	10.1021/acs.jmedchem.9b01411	10.7270/Q2B85CM0	31724864			Macdonald, JD; Chacón Simon, S; Han, C; Wang, F; Shaw, JG; Howes, JE; Sai, J; Yuh, JP; Camper, D; Alicie, BM; Alvarado, J; Nikhar, S; Payne, W; Aho, ER; Bauer, JA; Zhao, B; Phan, J; Thomas, LR; Rossanese, OW; Tansey, WP; Waterson, AG; Stauffer, SR; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50531142	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50531142&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			155547683	440739724							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51308138	COc1ccc(Cl)cc1S(=O)(=O)Nc1cc(Cl)ccc1O	InChI=1S/C13H11Cl2NO4S/c1-20-12-5-3-9(15)7-13(12)21(18,19)16-10-6-8(14)2-4-11(10)17/h2-7,16-17H,1H3	GPRUVNBBDBNFJU-UHFFFAOYSA-N	50531085	CHEMBL4457898	WD repeat-containing protein 5				 8410						ChEMBL	10.1021/acs.jmedchem.9b01411	10.7270/Q2B85CM0	31724864			Macdonald, JD; Chacón Simon, S; Han, C; Wang, F; Shaw, JG; Howes, JE; Sai, J; Yuh, JP; Camper, D; Alicie, BM; Alvarado, J; Nikhar, S; Payne, W; Aho, ER; Bauer, JA; Zhao, B; Phan, J; Thomas, LR; Rossanese, OW; Tansey, WP; Waterson, AG; Stauffer, SR; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50531085	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50531085&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			44117786	440739667							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51308139	COc1ccc(Br)cc1S(=O)(=O)Nc1ccccc1O	InChI=1S/C13H12BrNO4S/c1-19-12-7-6-9(14)8-13(12)20(17,18)15-10-4-2-3-5-11(10)16/h2-8,15-16H,1H3	MDXFESLYXHRFDS-UHFFFAOYSA-N	50531086	CHEMBL4445624	WD repeat-containing protein 5				>40000						ChEMBL	10.1021/acs.jmedchem.9b01411	10.7270/Q2B85CM0	31724864			Macdonald, JD; Chacón Simon, S; Han, C; Wang, F; Shaw, JG; Howes, JE; Sai, J; Yuh, JP; Camper, D; Alicie, BM; Alvarado, J; Nikhar, S; Payne, W; Aho, ER; Bauer, JA; Zhao, B; Phan, J; Thomas, LR; Rossanese, OW; Tansey, WP; Waterson, AG; Stauffer, SR; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50531086	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50531086&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			2210942	440739668							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51308140	Oc1ccc(cc1NS(=O)(=O)c1cc(Br)ccc1O)S(F)(F)(F)(F)F	InChI=1S/C12H9BrF5NO4S2/c13-7-1-3-11(21)12(5-7)24(22,23)19-9-6-8(2-4-10(9)20)25(14,15,16,17)18/h1-6,19-21H	ATCYNRMRQJYXTG-UHFFFAOYSA-N	50531089	CHEMBL4569742	WD repeat-containing protein 5				 110						ChEMBL	10.1021/acs.jmedchem.9b01411	10.7270/Q2B85CM0	31724864			Macdonald, JD; Chacón Simon, S; Han, C; Wang, F; Shaw, JG; Howes, JE; Sai, J; Yuh, JP; Camper, D; Alicie, BM; Alvarado, J; Nikhar, S; Payne, W; Aho, ER; Bauer, JA; Zhao, B; Phan, J; Thomas, LR; Rossanese, OW; Tansey, WP; Waterson, AG; Stauffer, SR; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50531089	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50531089&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			155552109	440739671							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51308141	Oc1ccc(cc1NS(=O)(=O)c1cc(Br)ccc1O)C1(CCC1)C#N	InChI=1S/C17H15BrN2O4S/c18-12-3-5-15(22)16(9-12)25(23,24)20-13-8-11(2-4-14(13)21)17(10-19)6-1-7-17/h2-5,8-9,20-22H,1,6-7H2	DMCFTKWJTBOJFX-UHFFFAOYSA-N	50531091	CHEMBL4470498	WD repeat-containing protein 5				 289						ChEMBL	10.1021/acs.jmedchem.9b01411	10.7270/Q2B85CM0	31724864			Macdonald, JD; Chacón Simon, S; Han, C; Wang, F; Shaw, JG; Howes, JE; Sai, J; Yuh, JP; Camper, D; Alicie, BM; Alvarado, J; Nikhar, S; Payne, W; Aho, ER; Bauer, JA; Zhao, B; Phan, J; Thomas, LR; Rossanese, OW; Tansey, WP; Waterson, AG; Stauffer, SR; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50531091	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50531091&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	Q1G	6U8O	145704703	440739673							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51308142	OC(=O)c1cc(Cl)cc(NS(=O)(=O)c2cc(Br)cc(Cl)c2O)c1O	InChI=1S/C13H8BrCl2NO6S/c14-5-1-8(16)12(19)10(2-5)24(22,23)17-9-4-6(15)3-7(11(9)18)13(20)21/h1-4,17-19H,(H,20,21)	GTSWUTVZEJOAKU-UHFFFAOYSA-N	50531093	CHEMBL4518711	WD repeat-containing protein 5				 163						ChEMBL	10.1021/acs.jmedchem.9b01411	10.7270/Q2B85CM0	31724864			Macdonald, JD; Chacón Simon, S; Han, C; Wang, F; Shaw, JG; Howes, JE; Sai, J; Yuh, JP; Camper, D; Alicie, BM; Alvarado, J; Nikhar, S; Payne, W; Aho, ER; Bauer, JA; Zhao, B; Phan, J; Thomas, LR; Rossanese, OW; Tansey, WP; Waterson, AG; Stauffer, SR; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50531093	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50531093&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			155541573	440739675							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51308143	OC(=O)c1c(O)c(NS(=O)(=O)c2cc(Br)ccc2O)cc(C2CC2)c1F	InChI=1S/C16H13BrFNO6S/c17-8-3-4-11(20)12(5-8)26(24,25)19-10-6-9(7-1-2-7)14(18)13(15(10)21)16(22)23/h3-7,19-21H,1-2H2,(H,22,23)	LZQVQCAIOFNYFL-UHFFFAOYSA-N	50531134	CHEMBL4471200	WD repeat-containing protein 5				 122						ChEMBL	10.1021/acs.jmedchem.9b01411	10.7270/Q2B85CM0	31724864			Macdonald, JD; Chacón Simon, S; Han, C; Wang, F; Shaw, JG; Howes, JE; Sai, J; Yuh, JP; Camper, D; Alicie, BM; Alvarado, J; Nikhar, S; Payne, W; Aho, ER; Bauer, JA; Zhao, B; Phan, J; Thomas, LR; Rossanese, OW; Tansey, WP; Waterson, AG; Stauffer, SR; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50531134	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50531134&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	Q1P	6U8L	145704701	440739716							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51308144	OC(=O)c1cc(NS(=O)(=O)c2cc(Br)ccc2O)cc(c1)S(F)(F)(F)(F)F	InChI=1S/C13H9BrF5NO5S2/c14-8-1-2-11(21)12(5-8)26(24,25)20-9-3-7(13(22)23)4-10(6-9)27(15,16,17,18)19/h1-6,20-21H,(H,22,23)	AAJCYJCNQUYQTH-UHFFFAOYSA-N	50531072	CHEMBL4474057	WD repeat-containing protein 5				 64						ChEMBL	10.1021/acs.jmedchem.9b01411	10.7270/Q2B85CM0	31724864			Macdonald, JD; Chacón Simon, S; Han, C; Wang, F; Shaw, JG; Howes, JE; Sai, J; Yuh, JP; Camper, D; Alicie, BM; Alvarado, J; Nikhar, S; Payne, W; Aho, ER; Bauer, JA; Zhao, B; Phan, J; Thomas, LR; Rossanese, OW; Tansey, WP; Waterson, AG; Stauffer, SR; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50531072	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50531072&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			155536666	440739654							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51308145	OC(=O)c1cc(cc(NS(=O)(=O)c2cc(Br)ccc2O)c1O)C1(CCC1)C#N	InChI=1S/C18H15BrN2O6S/c19-11-2-3-14(22)15(8-11)28(26,27)21-13-7-10(18(9-20)4-1-5-18)6-12(16(13)23)17(24)25/h2-3,6-8,21-23H,1,4-5H2,(H,24,25)	BLJKTQGNFJGAOA-UHFFFAOYSA-N	50531135	CHEMBL4441676	WD repeat-containing protein 5				 67						ChEMBL	10.1021/acs.jmedchem.9b01411	10.7270/Q2B85CM0	31724864			Macdonald, JD; Chacón Simon, S; Han, C; Wang, F; Shaw, JG; Howes, JE; Sai, J; Yuh, JP; Camper, D; Alicie, BM; Alvarado, J; Nikhar, S; Payne, W; Aho, ER; Bauer, JA; Zhao, B; Phan, J; Thomas, LR; Rossanese, OW; Tansey, WP; Waterson, AG; Stauffer, SR; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50531135	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50531135&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			155515379	440739717							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51308146	CNC(=O)c1cc(Cl)cc(NS(=O)(=O)c2cc(Br)ccc2O)c1O	InChI=1S/C14H12BrClN2O5S/c1-17-14(21)9-5-8(16)6-10(13(9)20)18-24(22,23)12-4-7(15)2-3-11(12)19/h2-6,18-20H,1H3,(H,17,21)	WREJJQUEKVRFCU-UHFFFAOYSA-N	50531073	CHEMBL4553810	WD repeat-containing protein 5				 746						ChEMBL	10.1021/acs.jmedchem.9b01411	10.7270/Q2B85CM0	31724864			Macdonald, JD; Chacón Simon, S; Han, C; Wang, F; Shaw, JG; Howes, JE; Sai, J; Yuh, JP; Camper, D; Alicie, BM; Alvarado, J; Nikhar, S; Payne, W; Aho, ER; Bauer, JA; Zhao, B; Phan, J; Thomas, LR; Rossanese, OW; Tansey, WP; Waterson, AG; Stauffer, SR; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50531073	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50531073&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			155555585	440739655							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51308147	CNC(=O)c1cc(cc(NS(=O)(=O)c2cc(Br)cc(Cl)c2O)c1O)S(F)(F)(F)(F)F	InChI=1S/C14H11BrClF5N2O5S2/c1-22-14(26)8-4-7(30(17,18,19,20)21)5-10(12(8)24)23-29(27,28)11-3-6(15)2-9(16)13(11)25/h2-5,23-25H,1H3,(H,22,26)	VAZWKKNFRGLKJW-UHFFFAOYSA-N	50531103	CHEMBL4455721	WD repeat-containing protein 5				 190						ChEMBL	10.1021/acs.jmedchem.9b01411	10.7270/Q2B85CM0	31724864			Macdonald, JD; Chacón Simon, S; Han, C; Wang, F; Shaw, JG; Howes, JE; Sai, J; Yuh, JP; Camper, D; Alicie, BM; Alvarado, J; Nikhar, S; Payne, W; Aho, ER; Bauer, JA; Zhao, B; Phan, J; Thomas, LR; Rossanese, OW; Tansey, WP; Waterson, AG; Stauffer, SR; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50531103	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50531103&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			155524406	440739685							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51308148	CNC(=O)c1cc(cc(NS(=O)(=O)c2cc(Br)ccc2O)c1O)C1(CCCCC1)C#N	InChI=1S/C21H22BrN3O5S/c1-24-20(28)15-9-13(21(12-23)7-3-2-4-8-21)10-16(19(15)27)25-31(29,30)18-11-14(22)5-6-17(18)26/h5-6,9-11,25-27H,2-4,7-8H2,1H3,(H,24,28)	CTKLAWJIXCJAIO-UHFFFAOYSA-N	50531137	CHEMBL4583214	WD repeat-containing protein 5				 779						ChEMBL	10.1021/acs.jmedchem.9b01411	10.7270/Q2B85CM0	31724864			Macdonald, JD; Chacón Simon, S; Han, C; Wang, F; Shaw, JG; Howes, JE; Sai, J; Yuh, JP; Camper, D; Alicie, BM; Alvarado, J; Nikhar, S; Payne, W; Aho, ER; Bauer, JA; Zhao, B; Phan, J; Thomas, LR; Rossanese, OW; Tansey, WP; Waterson, AG; Stauffer, SR; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50531137	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50531137&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			155566223	440739719							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51308149	CS(=O)(=O)c1cc(Cl)cc(NS(=O)(=O)c2cc(Br)ccc2O)c1	InChI=1S/C13H11BrClNO5S2/c1-22(18,19)11-6-9(15)5-10(7-11)16-23(20,21)13-4-8(14)2-3-12(13)17/h2-7,16-17H,1H3	OSGUHHXXRHWXPS-UHFFFAOYSA-N	50531108	CHEMBL4456384	WD repeat-containing protein 5				 1880						ChEMBL	10.1021/acs.jmedchem.9b01411	10.7270/Q2B85CM0	31724864			Macdonald, JD; Chacón Simon, S; Han, C; Wang, F; Shaw, JG; Howes, JE; Sai, J; Yuh, JP; Camper, D; Alicie, BM; Alvarado, J; Nikhar, S; Payne, W; Aho, ER; Bauer, JA; Zhao, B; Phan, J; Thomas, LR; Rossanese, OW; Tansey, WP; Waterson, AG; Stauffer, SR; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50531108	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50531108&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			155524907	440739690							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51308150	CS(=O)(=O)c1cc(cc(NS(=O)(=O)c2cc(Br)ccc2O)c1O)S(F)(F)(F)(F)F	InChI=1S/C13H11BrF5NO6S3/c1-27(23,24)12-6-8(29(15,16,17,18)19)5-9(13(12)22)20-28(25,26)11-4-7(14)2-3-10(11)21/h2-6,20-22H,1H3	PUYSPWVTNKPCJD-UHFFFAOYSA-N	50531120	CHEMBL4554506	WD repeat-containing protein 5				 167						ChEMBL	10.1021/acs.jmedchem.9b01411	10.7270/Q2B85CM0	31724864			Macdonald, JD; Chacón Simon, S; Han, C; Wang, F; Shaw, JG; Howes, JE; Sai, J; Yuh, JP; Camper, D; Alicie, BM; Alvarado, J; Nikhar, S; Payne, W; Aho, ER; Bauer, JA; Zhao, B; Phan, J; Thomas, LR; Rossanese, OW; Tansey, WP; Waterson, AG; Stauffer, SR; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50531120	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50531120&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			155556036	440739702							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51308151	COc1ccc(Br)cc1S(=O)(=O)Nc1ccc(Cl)cc1O	InChI=1S/C13H11BrClNO4S/c1-20-12-5-2-8(14)6-13(12)21(18,19)16-10-4-3-9(15)7-11(10)17/h2-7,16-17H,1H3	BZVGTEQHABVNJF-UHFFFAOYSA-N	50531138	CHEMBL4550667	WD repeat-containing protein 5				 27700						ChEMBL	10.1021/acs.jmedchem.9b01411	10.7270/Q2B85CM0	31724864			Macdonald, JD; Chacón Simon, S; Han, C; Wang, F; Shaw, JG; Howes, JE; Sai, J; Yuh, JP; Camper, D; Alicie, BM; Alvarado, J; Nikhar, S; Payne, W; Aho, ER; Bauer, JA; Zhao, B; Phan, J; Thomas, LR; Rossanese, OW; Tansey, WP; Waterson, AG; Stauffer, SR; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50531138	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50531138&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			155555207	440739720							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51308152	CNC(=O)c1cc(cc(NS(=O)(=O)c2cc(Br)ccc2O)c1O)S(F)(F)(F)(F)F	InChI=1S/C14H12BrF5N2O5S2/c1-21-14(25)9-5-8(29(16,17,18,19)20)6-10(13(9)24)22-28(26,27)12-4-7(15)2-3-11(12)23/h2-6,22-24H,1H3,(H,21,25)	UYPDTLHHKDBIQU-UHFFFAOYSA-N	50531119	CHEMBL4523046	WD repeat-containing protein 5				 204						ChEMBL	10.1021/acs.jmedchem.9b01411	10.7270/Q2B85CM0	31724864			Macdonald, JD; Chacón Simon, S; Han, C; Wang, F; Shaw, JG; Howes, JE; Sai, J; Yuh, JP; Camper, D; Alicie, BM; Alvarado, J; Nikhar, S; Payne, W; Aho, ER; Bauer, JA; Zhao, B; Phan, J; Thomas, LR; Rossanese, OW; Tansey, WP; Waterson, AG; Stauffer, SR; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50531119	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50531119&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			155543818	440739701							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51308153	CS(=O)(=O)c1cc(Cl)cc(NS(=O)(=O)c2cc(Br)cc3cccnc23)c1O	InChI=1S/C16H12BrClN2O5S2/c1-26(22,23)14-8-11(18)7-12(16(14)21)20-27(24,25)13-6-10(17)5-9-3-2-4-19-15(9)13/h2-8,20-21H,1H3	HVHOOKABEVVVMP-UHFFFAOYSA-N	50531113	CHEMBL4458101	WD repeat-containing protein 5				 385						ChEMBL	10.1021/acs.jmedchem.9b01411	10.7270/Q2B85CM0	31724864			Macdonald, JD; Chacón Simon, S; Han, C; Wang, F; Shaw, JG; Howes, JE; Sai, J; Yuh, JP; Camper, D; Alicie, BM; Alvarado, J; Nikhar, S; Payne, W; Aho, ER; Bauer, JA; Zhao, B; Phan, J; Thomas, LR; Rossanese, OW; Tansey, WP; Waterson, AG; Stauffer, SR; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50531113	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50531113&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			155526979	440739695							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51308154	CNC(=O)c1cc(cc(NS(=O)(=O)c2cc(Br)ccc2O)c1O)C1(CCC1)C#N	InChI=1S/C19H18BrN3O5S/c1-22-18(26)13-7-11(19(10-21)5-2-6-19)8-14(17(13)25)23-29(27,28)16-9-12(20)3-4-15(16)24/h3-4,7-9,23-25H,2,5-6H2,1H3,(H,22,26)	QNUCCYVBZDQUMB-UHFFFAOYSA-N	50531105	CHEMBL4543629	WD repeat-containing protein 5				 566						ChEMBL	10.1021/acs.jmedchem.9b01411	10.7270/Q2B85CM0	31724864			Macdonald, JD; Chacón Simon, S; Han, C; Wang, F; Shaw, JG; Howes, JE; Sai, J; Yuh, JP; Camper, D; Alicie, BM; Alvarado, J; Nikhar, S; Payne, W; Aho, ER; Bauer, JA; Zhao, B; Phan, J; Thomas, LR; Rossanese, OW; Tansey, WP; Waterson, AG; Stauffer, SR; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50531105	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50531105&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			155552279	440739687							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51308155	CNC(=O)c1cc(cc(NS(=O)(=O)c2cc(Br)cc3cccnc23)c1O)C1(CCC1)C#N	InChI=1S/C22H19BrN4O4S/c1-25-21(29)16-9-14(22(12-24)5-3-6-22)10-17(20(16)28)27-32(30,31)18-11-15(23)8-13-4-2-7-26-19(13)18/h2,4,7-11,27-28H,3,5-6H2,1H3,(H,25,29)	LUHBUKXZMCITBQ-UHFFFAOYSA-N	50531139	CHEMBL4457793	WD repeat-containing protein 5				 825						ChEMBL	10.1021/acs.jmedchem.9b01411	10.7270/Q2B85CM0	31724864			Macdonald, JD; Chacón Simon, S; Han, C; Wang, F; Shaw, JG; Howes, JE; Sai, J; Yuh, JP; Camper, D; Alicie, BM; Alvarado, J; Nikhar, S; Payne, W; Aho, ER; Bauer, JA; Zhao, B; Phan, J; Thomas, LR; Rossanese, OW; Tansey, WP; Waterson, AG; Stauffer, SR; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50531139	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50531139&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			155526271	440739721							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51308156	OC(=O)c1cc(Cl)cc(NS(=O)(=O)c2cc(Br)ccc2O)c1	InChI=1S/C13H9BrClNO5S/c14-8-1-2-11(17)12(5-8)22(20,21)16-10-4-7(13(18)19)3-9(15)6-10/h1-6,16-17H,(H,18,19)	BAFBQLQHLMLBCL-UHFFFAOYSA-N	50531077	CHEMBL4531782	WD repeat-containing protein 5				 2880						ChEMBL	10.1021/acs.jmedchem.9b01411	10.7270/Q2B85CM0	31724864			Macdonald, JD; Chacón Simon, S; Han, C; Wang, F; Shaw, JG; Howes, JE; Sai, J; Yuh, JP; Camper, D; Alicie, BM; Alvarado, J; Nikhar, S; Payne, W; Aho, ER; Bauer, JA; Zhao, B; Phan, J; Thomas, LR; Rossanese, OW; Tansey, WP; Waterson, AG; Stauffer, SR; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50531077	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50531077&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			155546315	440739659							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51308157	Oc1ccc(Br)cc1S(=O)(=O)Nc1cc(cc(Nc2nc[nH]n2)c1O)C1(CCC1)C#N	InChI=1S/C19H17BrN6O4S/c20-12-2-3-15(27)16(8-12)31(29,30)26-14-7-11(19(9-21)4-1-5-19)6-13(17(14)28)24-18-22-10-23-25-18/h2-3,6-8,10,26-28H,1,4-5H2,(H2,22,23,24,25)	FOGZDMZPYDJTOI-UHFFFAOYSA-N	50531129	CHEMBL4450684	WD repeat-containing protein 5				 46						ChEMBL	10.1021/acs.jmedchem.9b01411	10.7270/Q2B85CM0	31724864			Macdonald, JD; Chacón Simon, S; Han, C; Wang, F; Shaw, JG; Howes, JE; Sai, J; Yuh, JP; Camper, D; Alicie, BM; Alvarado, J; Nikhar, S; Payne, W; Aho, ER; Bauer, JA; Zhao, B; Phan, J; Thomas, LR; Rossanese, OW; Tansey, WP; Waterson, AG; Stauffer, SR; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50531129	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50531129&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			155521779	440739711							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51308010	COc1ccc(Br)cc1S(=O)(=O)Nc1cc(Cl)cc(c1O)S(C)(=O)=O	InChI=1S/C14H13BrClNO6S2/c1-23-11-4-3-8(15)5-12(11)25(21,22)17-10-6-9(16)7-13(14(10)18)24(2,19)20/h3-7,17-18H,1-2H3	XSNDBCXTZMGFDN-UHFFFAOYSA-N	50531070	CHEMBL4532703	WD repeat-containing protein 5				 304						ChEMBL	10.1021/acs.jmedchem.9b01411	10.7270/Q2B85CM0	31724864			Macdonald, JD; Chacón Simon, S; Han, C; Wang, F; Shaw, JG; Howes, JE; Sai, J; Yuh, JP; Camper, D; Alicie, BM; Alvarado, J; Nikhar, S; Payne, W; Aho, ER; Bauer, JA; Zhao, B; Phan, J; Thomas, LR; Rossanese, OW; Tansey, WP; Waterson, AG; Stauffer, SR; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50531070	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50531070&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			155547690	440739652							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51308011	OC(=O)c1cc(Cl)cc(NS(=O)(=O)c2cc(Br)ccc2O)c1O	InChI=1S/C13H9BrClNO6S/c14-6-1-2-10(17)11(3-6)23(21,22)16-9-5-7(15)4-8(12(9)18)13(19)20/h1-5,16-18H,(H,19,20)	YKNSJAKLAKAVKH-UHFFFAOYSA-N	50531071	CHEMBL4573789	WD repeat-containing protein 5				 223						ChEMBL	10.1021/acs.jmedchem.9b01411	10.7270/Q2B85CM0	31724864			Macdonald, JD; Chacón Simon, S; Han, C; Wang, F; Shaw, JG; Howes, JE; Sai, J; Yuh, JP; Camper, D; Alicie, BM; Alvarado, J; Nikhar, S; Payne, W; Aho, ER; Bauer, JA; Zhao, B; Phan, J; Thomas, LR; Rossanese, OW; Tansey, WP; Waterson, AG; Stauffer, SR; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50531071	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50531071&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			155563120	440739653							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51308012	OC(=O)c1cc(NS(=O)(=O)c2cc(Br)ccc2O)cc(c1)S(F)(F)(F)(F)F	InChI=1S/C13H9BrF5NO5S2/c14-8-1-2-11(21)12(5-8)26(24,25)20-9-3-7(13(22)23)4-10(6-9)27(15,16,17,18)19/h1-6,20-21H,(H,22,23)	AAJCYJCNQUYQTH-UHFFFAOYSA-N	50531072	CHEMBL4474057	WD repeat-containing protein 5				 64						ChEMBL	10.1021/acs.jmedchem.9b01411	10.7270/Q2B85CM0	31724864			Macdonald, JD; Chacón Simon, S; Han, C; Wang, F; Shaw, JG; Howes, JE; Sai, J; Yuh, JP; Camper, D; Alicie, BM; Alvarado, J; Nikhar, S; Payne, W; Aho, ER; Bauer, JA; Zhao, B; Phan, J; Thomas, LR; Rossanese, OW; Tansey, WP; Waterson, AG; Stauffer, SR; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50531072	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50531072&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			155536666	440739654							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51308013	CNC(=O)c1cc(Cl)cc(NS(=O)(=O)c2cc(Br)ccc2O)c1O	InChI=1S/C14H12BrClN2O5S/c1-17-14(21)9-5-8(16)6-10(13(9)20)18-24(22,23)12-4-7(15)2-3-11(12)19/h2-6,18-20H,1H3,(H,17,21)	WREJJQUEKVRFCU-UHFFFAOYSA-N	50531073	CHEMBL4553810	WD repeat-containing protein 5				 746						ChEMBL	10.1021/acs.jmedchem.9b01411	10.7270/Q2B85CM0	31724864			Macdonald, JD; Chacón Simon, S; Han, C; Wang, F; Shaw, JG; Howes, JE; Sai, J; Yuh, JP; Camper, D; Alicie, BM; Alvarado, J; Nikhar, S; Payne, W; Aho, ER; Bauer, JA; Zhao, B; Phan, J; Thomas, LR; Rossanese, OW; Tansey, WP; Waterson, AG; Stauffer, SR; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50531073	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50531073&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			155555585	440739655							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51308014	CNC(=O)c1cc(cc(NS(=O)(=O)c2cc(Br)cc(Cl)c2O)c1O)C1(CCC1)C#N	InChI=1S/C19H17BrClN3O5S/c1-23-18(27)12-5-10(19(9-22)3-2-4-19)6-14(16(12)25)24-30(28,29)15-8-11(20)7-13(21)17(15)26/h5-8,24-26H,2-4H2,1H3,(H,23,27)	COYGYHFILXAMSQ-UHFFFAOYSA-N	50531074	CHEMBL4472649	WD repeat-containing protein 5				 69						ChEMBL	10.1021/acs.jmedchem.9b01411	10.7270/Q2B85CM0	31724864			Macdonald, JD; Chacón Simon, S; Han, C; Wang, F; Shaw, JG; Howes, JE; Sai, J; Yuh, JP; Camper, D; Alicie, BM; Alvarado, J; Nikhar, S; Payne, W; Aho, ER; Bauer, JA; Zhao, B; Phan, J; Thomas, LR; Rossanese, OW; Tansey, WP; Waterson, AG; Stauffer, SR; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50531074	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50531074&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	Q0M	6U5Y	145704698	440739656							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51308015	CS(=O)(=O)c1cc(NS(=O)(=O)c2cc(Br)ccc2O)cc(c1)S(F)(F)(F)(F)F	InChI=1S/C13H11BrF5NO5S3/c1-26(22,23)10-5-9(6-11(7-10)28(15,16,17,18)19)20-27(24,25)13-4-8(14)2-3-12(13)21/h2-7,20-21H,1H3	GXKWWSXTDOWSFB-UHFFFAOYSA-N	50531075	CHEMBL4475470	WD repeat-containing protein 5				 511						ChEMBL	10.1021/acs.jmedchem.9b01411	10.7270/Q2B85CM0	31724864			Macdonald, JD; Chacón Simon, S; Han, C; Wang, F; Shaw, JG; Howes, JE; Sai, J; Yuh, JP; Camper, D; Alicie, BM; Alvarado, J; Nikhar, S; Payne, W; Aho, ER; Bauer, JA; Zhao, B; Phan, J; Thomas, LR; Rossanese, OW; Tansey, WP; Waterson, AG; Stauffer, SR; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50531075	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50531075&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	Q0S	6U5M	145704697	440739657							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51308016	COc1ccc(Br)cc1S(=O)(=O)Nc1cc(ccc1O)C(C)(C)C	InChI=1S/C17H20BrNO4S/c1-17(2,3)11-5-7-14(20)13(9-11)19-24(21,22)16-10-12(18)6-8-15(16)23-4/h5-10,19-20H,1-4H3	NUCBFUKPFYXFNL-UHFFFAOYSA-N	50531076	CHEMBL4514703	WD repeat-containing protein 5				 3780						ChEMBL	10.1021/acs.jmedchem.9b01411	10.7270/Q2B85CM0	31724864			Macdonald, JD; Chacón Simon, S; Han, C; Wang, F; Shaw, JG; Howes, JE; Sai, J; Yuh, JP; Camper, D; Alicie, BM; Alvarado, J; Nikhar, S; Payne, W; Aho, ER; Bauer, JA; Zhao, B; Phan, J; Thomas, LR; Rossanese, OW; Tansey, WP; Waterson, AG; Stauffer, SR; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50531076	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50531076&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			155539506	440739658							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51308017	OC(=O)c1cc(Cl)cc(NS(=O)(=O)c2cc(Br)ccc2O)c1	InChI=1S/C13H9BrClNO5S/c14-8-1-2-11(17)12(5-8)22(20,21)16-10-4-7(13(18)19)3-9(15)6-10/h1-6,16-17H,(H,18,19)	BAFBQLQHLMLBCL-UHFFFAOYSA-N	50531077	CHEMBL4531782	WD repeat-containing protein 5				 2880						ChEMBL	10.1021/acs.jmedchem.9b01411	10.7270/Q2B85CM0	31724864			Macdonald, JD; Chacón Simon, S; Han, C; Wang, F; Shaw, JG; Howes, JE; Sai, J; Yuh, JP; Camper, D; Alicie, BM; Alvarado, J; Nikhar, S; Payne, W; Aho, ER; Bauer, JA; Zhao, B; Phan, J; Thomas, LR; Rossanese, OW; Tansey, WP; Waterson, AG; Stauffer, SR; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50531077	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50531077&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			155546315	440739659							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51308018	OC(=O)c1cc(OC(F)(F)F)cc(NS(=O)(=O)c2cc(Br)ccc2O)c1O	InChI=1S/C14H9BrF3NO7S/c15-6-1-2-10(20)11(3-6)27(24,25)19-9-5-7(26-14(16,17)18)4-8(12(9)21)13(22)23/h1-5,19-21H,(H,22,23)	HJSHYSJMDZOUAB-UHFFFAOYSA-N	50531078	CHEMBL4575067	WD repeat-containing protein 5				 137						ChEMBL	10.1021/acs.jmedchem.9b01411	10.7270/Q2B85CM0	31724864			Macdonald, JD; Chacón Simon, S; Han, C; Wang, F; Shaw, JG; Howes, JE; Sai, J; Yuh, JP; Camper, D; Alicie, BM; Alvarado, J; Nikhar, S; Payne, W; Aho, ER; Bauer, JA; Zhao, B; Phan, J; Thomas, LR; Rossanese, OW; Tansey, WP; Waterson, AG; Stauffer, SR; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50531078	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50531078&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			155561018	440739660							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51308019	OC(=O)c1cc(cc(NS(=O)(=O)c2cc(Br)ccc2O)c1O)C1(CCCCC1)C#N	InChI=1S/C20H19BrN2O6S/c21-13-4-5-16(24)17(10-13)30(28,29)23-15-9-12(8-14(18(15)25)19(26)27)20(11-22)6-2-1-3-7-20/h4-5,8-10,23-25H,1-3,6-7H2,(H,26,27)	LHQJNKXEQDMDIL-UHFFFAOYSA-N	50531079	CHEMBL4471282	WD repeat-containing protein 5				 195						ChEMBL	10.1021/acs.jmedchem.9b01411	10.7270/Q2B85CM0	31724864			Macdonald, JD; Chacón Simon, S; Han, C; Wang, F; Shaw, JG; Howes, JE; Sai, J; Yuh, JP; Camper, D; Alicie, BM; Alvarado, J; Nikhar, S; Payne, W; Aho, ER; Bauer, JA; Zhao, B; Phan, J; Thomas, LR; Rossanese, OW; Tansey, WP; Waterson, AG; Stauffer, SR; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50531079	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50531079&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			155534803	440739661							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51308020	CCOc1cc(ccc1F)S(=O)(=O)Nc1ccccc1C(O)=O	InChI=1S/C15H14FNO5S/c1-2-22-14-9-10(7-8-12(14)16)23(20,21)17-13-6-4-3-5-11(13)15(18)19/h3-9,17H,2H2,1H3,(H,18,19)	DMIRFYYZRJSZPF-UHFFFAOYSA-N	50531080	CHEMBL4465263	WD repeat-containing protein 5				 71000						ChEMBL	10.1021/acs.jmedchem.9b01411	10.7270/Q2B85CM0	31724864			Macdonald, JD; Chacón Simon, S; Han, C; Wang, F; Shaw, JG; Howes, JE; Sai, J; Yuh, JP; Camper, D; Alicie, BM; Alvarado, J; Nikhar, S; Payne, W; Aho, ER; Bauer, JA; Zhao, B; Phan, J; Thomas, LR; Rossanese, OW; Tansey, WP; Waterson, AG; Stauffer, SR; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50531080	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50531080&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			15943973	440739662							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51308021	CNC(=O)c1cc(NS(=O)(=O)c2cc(Br)ccc2O)cc(c1)C1(CCC1)C#N	InChI=1S/C19H18BrN3O4S/c1-22-18(25)12-7-13(19(11-21)5-2-6-19)9-15(8-12)23-28(26,27)17-10-14(20)3-4-16(17)24/h3-4,7-10,23-24H,2,5-6H2,1H3,(H,22,25)	HTDHGPQJWJSDGO-UHFFFAOYSA-N	50531081	CHEMBL4593558	WD repeat-containing protein 5				 1080						ChEMBL	10.1021/acs.jmedchem.9b01411	10.7270/Q2B85CM0	31724864			Macdonald, JD; Chacón Simon, S; Han, C; Wang, F; Shaw, JG; Howes, JE; Sai, J; Yuh, JP; Camper, D; Alicie, BM; Alvarado, J; Nikhar, S; Payne, W; Aho, ER; Bauer, JA; Zhao, B; Phan, J; Thomas, LR; Rossanese, OW; Tansey, WP; Waterson, AG; Stauffer, SR; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50531081	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50531081&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			155569685	440739663							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51308022	CS(=O)(=O)c1cc(Cl)cc(NS(=O)(=O)c2cc(Br)cc(Cl)c2O)c1O	InChI=1S/C13H10BrCl2NO6S2/c1-24(20,21)10-5-7(15)4-9(13(10)19)17-25(22,23)11-3-6(14)2-8(16)12(11)18/h2-5,17-19H,1H3	DMNYWAGZZMQKRG-UHFFFAOYSA-N	50531082	CHEMBL4455527	WD repeat-containing protein 5				 123						ChEMBL	10.1021/acs.jmedchem.9b01411	10.7270/Q2B85CM0	31724864			Macdonald, JD; Chacón Simon, S; Han, C; Wang, F; Shaw, JG; Howes, JE; Sai, J; Yuh, JP; Camper, D; Alicie, BM; Alvarado, J; Nikhar, S; Payne, W; Aho, ER; Bauer, JA; Zhao, B; Phan, J; Thomas, LR; Rossanese, OW; Tansey, WP; Waterson, AG; Stauffer, SR; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50531082	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50531082&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			155524950	440739664							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981739	Cc1cc(ccc1F)[C@@H](NC(=O)c1cc(CN2CCOC2=N)cc(n1)-c1cn(C)nc1C(F)(F)F)C1CC1	InChI=1S/C26H26F4N6O2/c1-14-9-17(5-6-19(14)27)22(16-3-4-16)33-24(37)21-11-15(12-36-7-8-38-25(36)31)10-20(32-21)18-13-35(2)34-23(18)26(28,29)30/h5-6,9-11,13,16,22,31H,3-4,7-8,12H2,1-2H3,(H,33,37)/t22-/m0/s1	JFCPGTOXKDIFFJ-QFIPXVFZSA-N	473539	US10844044, Example 361	WD repeat-containing protein 5		 0.770								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473539	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473539&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456086	442073747							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981740	Cc1cc(CNC(=O)c2cc(Cn3ccn(C)c3=N)cc(c2)-c2ccc(F)cc2C)ccc1F	InChI=1S/C27H26F2N4O/c1-17-11-23(28)5-6-24(17)21-12-20(16-33-9-8-32(3)27(33)30)13-22(14-21)26(34)31-15-19-4-7-25(29)18(2)10-19/h4-14,30H,15-16H2,1-3H3,(H,31,34)	LEOZOVLOEOWBAL-UHFFFAOYSA-N	50520127	CHEMBL4585441::US10844044, Example 87	WD repeat-containing protein 5		 0.800								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50520127	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50520127&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456497	440728709							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981741	COc1cc(CNC(=O)c2cc(Cn3ccn(C)c3=N)cc(OCC3CC3)c2)cc(OC)c1	InChI=1S/C25H30N4O4/c1-28-6-7-29(25(28)26)15-19-8-20(12-23(11-19)33-16-17-4-5-17)24(30)27-14-18-9-21(31-2)13-22(10-18)32-3/h6-13,17,26H,4-5,14-16H2,1-3H3,(H,27,30)	PNJLXWFUJBKCJP-UHFFFAOYSA-N	473541	US10844044, Example 178	WD repeat-containing protein 5		 3.30								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473541	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473541&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146455881	442073749							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981742	FC(F)Oc1cc(F)ccc1-c1cc(Cn2ccoc2=N)cc(c1)C(=O)N[C@@H](C1CC1)c1ccc(Cl)c(Cl)c1	InChI=1S/C28H22Cl2F3N3O3/c29-22-6-3-17(12-23(22)30)25(16-1-2-16)35-26(37)19-10-15(14-36-7-8-38-28(36)34)9-18(11-19)21-5-4-20(31)13-24(21)39-27(32)33/h3-13,16,25,27,34H,1-2,14H2,(H,35,37)/t25-/m0/s1	NHTFTZSMUWDSFK-VWLOTQADSA-N	473542	US10844044, Example 270	WD repeat-containing protein 5		 0.180								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473542	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473542&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146455955	442073750							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981743	Cc1cc(ccc1F)[C@@H](NC(=O)c1cc(CN2CCCOC2=N)cc(c1)-c1cccnc1C(F)(F)F)C1CC1	InChI=1S/C29H28F4N4O2/c1-17-12-20(7-8-24(17)30)25(19-5-6-19)36-27(38)22-14-18(16-37-10-3-11-39-28(37)34)13-21(15-22)23-4-2-9-35-26(23)29(31,32)33/h2,4,7-9,12-15,19,25,34H,3,5-6,10-11,16H2,1H3,(H,36,38)/t25-/m0/s1	RWDXQFHWSULJBR-VWLOTQADSA-N	473526	US10844044, Example 266::US10844044, Example 362	WD repeat-containing protein 5		 0.720								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473526	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473526&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146455809	442073734							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981744	Cc1cc(F)ccc1-c1cc(Cn2ccn(C)c2=N)cc(c1)C(=O)NCc1cc(F)c(F)c(F)c1	InChI=1S/C26H22F4N4O/c1-15-7-20(27)3-4-21(15)18-8-17(14-34-6-5-33(2)26(34)31)9-19(12-18)25(35)32-13-16-10-22(28)24(30)23(29)11-16/h3-12,31H,13-14H2,1-2H3,(H,32,35)	CGXLRSGFPVWZIJ-UHFFFAOYSA-N	473544	US10844044, Example 88	WD repeat-containing protein 5		 3.40								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473544	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473544&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456313	442073751							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981745	Cc1cc(ccc1F)[C@@H](NC(=O)c1cc(Cn2ccn(C)c2=N)cc(OC(F)(F)F)c1)C1CC1	InChI=1S/C24H24F4N4O2/c1-14-9-17(5-6-20(14)25)21(16-3-4-16)30-22(33)18-10-15(11-19(12-18)34-24(26,27)28)13-32-8-7-31(2)23(32)29/h5-12,16,21,29H,3-4,13H2,1-2H3,(H,30,33)/t21-/m0/s1	QIANIUPSYPZROU-NRFANRHFSA-N	473545	US10844044, Example 179	WD repeat-containing protein 5		<0.100								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473545	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473545&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146455841	442073752							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981746	FC(F)(F)c1ncccc1-c1cc(Cn2ccoc2=N)cc(c1)C(=O)N[C@@H](C1CC1)c1ccc(Cl)c(Cl)c1	InChI=1S/C27H21Cl2F3N4O2/c28-21-6-5-17(13-22(21)29)23(16-3-4-16)35-25(37)19-11-15(14-36-8-9-38-26(36)33)10-18(12-19)20-2-1-7-34-24(20)27(30,31)32/h1-2,5-13,16,23,33H,3-4,14H2,(H,35,37)/t23-/m0/s1	VDEBFQLLNDRPRL-QHCPKHFHSA-N	473546	US10844044, Example 271	WD repeat-containing protein 5		 0.720								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473546	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473546&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456436	442073753							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981747	Cc1cc(ccc1F)[C@@H](NC(=O)c1cc(Cn2cnn(C)c2=N)cc(c1)-c1cn(C)nc1C(F)(F)F)C1CC1	InChI=1S/C27H27F4N7O/c1-15-8-18(6-7-22(15)28)23(17-4-5-17)34-25(39)20-10-16(12-38-14-33-37(3)26(38)32)9-19(11-20)21-13-36(2)35-24(21)27(29,30)31/h6-11,13-14,17,23,32H,4-5,12H2,1-3H3,(H,34,39)/t23-/m0/s1	FOQAOHTWSAZEKH-QHCPKHFHSA-N	473547	US10844044, Example 363	WD repeat-containing protein 5		<0.100								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473547	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473547&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146457320	442073754							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981748	Cc1cc(F)ccc1-c1cc(Cn2ccn(C)c2=N)cc(c1)C(=O)NCc1ccc(F)cc1	InChI=1S/C26H24F2N4O/c1-17-11-23(28)7-8-24(17)20-12-19(16-32-10-9-31(2)26(32)29)13-21(14-20)25(33)30-15-18-3-5-22(27)6-4-18/h3-14,29H,15-16H2,1-2H3,(H,30,33)	BXZUNLOKCRSVHA-UHFFFAOYSA-N	473548	US10844044, Example 89	WD repeat-containing protein 5		 15.0								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473548	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473548&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456394	442073755							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981749	CCOc1cc(Cn2ccn(C)c2=N)cc(c1)C(=O)N[C@@H](C1CC1)c1ccc(F)c(C)c1	InChI=1S/C25H29FN4O2/c1-4-32-21-13-17(15-30-10-9-29(3)25(30)27)12-20(14-21)24(31)28-23(18-5-6-18)19-7-8-22(26)16(2)11-19/h7-14,18,23,27H,4-6,15H2,1-3H3,(H,28,31)/t23-/m0/s1	LKHFYLYLSUWWJI-QHCPKHFHSA-N	473549	US10844044, Example 180	WD repeat-containing protein 5		 0.130								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473549	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473549&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146457313	442073756							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981750	Cc1cc(ccc1F)[C@@H](NC(=O)c1cc(CN2CCOC2=N)cc(c1)-c1ccc(F)cc1C(F)F)C1CC1	InChI=1S/C29H27F4N3O2/c1-16-10-19(4-7-25(16)31)26(18-2-3-18)35-28(37)21-12-17(15-36-8-9-38-29(36)34)11-20(13-21)23-6-5-22(30)14-24(23)27(32)33/h4-7,10-14,18,26-27,34H,2-3,8-9,15H2,1H3,(H,35,37)/t26-/m0/s1	USAARLBJOVHAKH-SANMLTNESA-N	473550	US10844044, Example 272	WD repeat-containing protein 5		<0.100								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473550	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473550&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146455848	442073757							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981751	Cc1ccnc(c1)C(NC(=O)c1cc(Cn2ccn(C)c2=N)cc(c1)-c1ncccc1C(F)(F)F)C1CC1	InChI=1S/C28H27F3N6O/c1-17-7-9-33-23(12-17)25(19-5-6-19)35-26(38)21-14-18(16-37-11-10-36(2)27(37)32)13-20(15-21)24-22(28(29,30)31)4-3-8-34-24/h3-4,7-15,19,25,32H,5-6,16H2,1-2H3,(H,35,38)	PFEQICCQWNQNGD-UHFFFAOYSA-N	473551	US10844044, Example 364	WD repeat-containing protein 5		 4.30								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473551	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473551&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456016	442073758							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981752	Cn1ccn(Cc2cc(cc(c2)-c2ccccc2C(F)(F)F)C(=O)NCc2ccc(Cl)c(Cl)c2)c1=N	InChI=1S/C26H21Cl2F3N4O/c1-34-8-9-35(25(34)32)15-17-10-18(20-4-2-3-5-21(20)26(29,30)31)13-19(11-17)24(36)33-14-16-6-7-22(27)23(28)12-16/h2-13,32H,14-15H2,1H3,(H,33,36)	WKZHBGZDYFHMNP-UHFFFAOYSA-N	473552	US10844044, Example 90	WD repeat-containing protein 5		 0.460								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473552	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473552&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146455741	442073759							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981753	C[C@H](NC(=O)c1cc(Cn2ccn(C)c2=N)cc(OCC2CC2)c1)c1ccc(F)c(C)c1	InChI=1S/C25H29FN4O2/c1-16-10-20(6-7-23(16)26)17(2)28-24(31)21-11-19(14-30-9-8-29(3)25(30)27)12-22(13-21)32-15-18-4-5-18/h6-13,17-18,27H,4-5,14-15H2,1-3H3,(H,28,31)/t17-/m0/s1	DMKJPVBQLQJSPA-KRWDZBQOSA-N	473553	US10844044, Example 181	WD repeat-containing protein 5		 0.350								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473553	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473553&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146455773	442073760							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981754	Cc1cc(ccc1F)[C@@H](NC(=O)c1cc(CN2CCOC2=N)cc(c1)-c1ccc(F)cc1OC(F)F)C1CC1	InChI=1S/C29H27F4N3O3/c1-16-10-19(4-7-24(16)31)26(18-2-3-18)35-27(37)21-12-17(15-36-8-9-38-29(36)34)11-20(13-21)23-6-5-22(30)14-25(23)39-28(32)33/h4-7,10-14,18,26,28,34H,2-3,8-9,15H2,1H3,(H,35,37)/t26-/m0/s1	KMVVRYNPDMOBKR-SANMLTNESA-N	473554	US10844044, Example 273	WD repeat-containing protein 5		<0.100								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473554	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473554&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456794	442073761							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981755	COc1cc(CNC(=O)c2cc(Cn3ccn(C)c3=N)nc(c2)-c2ccc(F)cc2C)cc(OC)c1	InChI=1S/C27H28FN5O3/c1-17-9-20(28)5-6-24(17)25-13-19(12-21(31-25)16-33-8-7-32(2)27(33)29)26(34)30-15-18-10-22(35-3)14-23(11-18)36-4/h5-14,29H,15-16H2,1-4H3,(H,30,34)	ZTRIQPKBTHQSHH-UHFFFAOYSA-N	473555	US10844044, Example 365	WD repeat-containing protein 5		 0.550								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473555	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473555&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456271	442073762							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981756	Cc1ccnc(c1)[C@@H](NC(=O)c1cc(Cn2ccn(C)c2=N)cc(c1)-c1ccc(F)cc1C)C1CC1	InChI=1S/C29H30FN5O/c1-18-8-9-32-26(12-18)27(21-4-5-21)33-28(36)23-15-20(17-35-11-10-34(3)29(35)31)14-22(16-23)25-7-6-24(30)13-19(25)2/h6-16,21,27,31H,4-5,17H2,1-3H3,(H,33,36)/t27-/m0/s1	SSPGQCWIFWWIMQ-MHZLTWQESA-N	473556	US10844044, Example 91	WD repeat-containing protein 5		<0.100								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473556	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473556&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456305	442073763							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981757	Cc1ccnc(c1)[C@@H](NC(=O)c1cc(Cn2ccn(C)c2=N)cc(OCC2CC2)c1)C1CC1	InChI=1S/C26H31N5O2/c1-17-7-8-28-23(11-17)24(20-5-6-20)29-25(32)21-12-19(15-31-10-9-30(2)26(31)27)13-22(14-21)33-16-18-3-4-18/h7-14,18,20,24,27H,3-6,15-16H2,1-2H3,(H,29,32)/t24-/m0/s1	IZYAZQXLASFBOY-DEOSSOPVSA-N	473557	US10844044, Example 182	WD repeat-containing protein 5		 1.000								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473557	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473557&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456046	442073764							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981758	Cc1cc(ccc1F)[C@@H](NC(=O)c1cc(Cn2ccoc2=N)cc(c1)-c1ccc(F)cc1C(F)F)C1CC1	InChI=1S/C29H25F4N3O2/c1-16-10-19(4-7-25(16)31)26(18-2-3-18)35-28(37)21-12-17(15-36-8-9-38-29(36)34)11-20(13-21)23-6-5-22(30)14-24(23)27(32)33/h4-14,18,26-27,34H,2-3,15H2,1H3,(H,35,37)/t26-/m0/s1	RJCLWVUUHSZHSZ-SANMLTNESA-N	473558	US10844044, Example 274	WD repeat-containing protein 5		<0.100								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473558	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473558&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456195	442073765							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981759	COc1ccnc(CNC(=O)c2ccc(F)c(Cn3ccn(C)c3=N)c2)c1	InChI=1S/C19H20FN5O2/c1-24-7-8-25(19(24)21)12-14-9-13(3-4-17(14)20)18(26)23-11-15-10-16(27-2)5-6-22-15/h3-10,21H,11-12H2,1-2H3,(H,23,26)	LWOKPBIVQDLWMM-UHFFFAOYSA-N	473559	US10844044, Example 366	WD repeat-containing protein 5		 13.0								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473559	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473559&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146455986	442073766							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968567	Fc1ccc(c(Cl)c1)-c1cc(CNC2=NCCN2)cc(c1)C(=O)NC(C1CC1)C1CC1	InChI=1S/C24H26ClFN4O/c25-21-12-19(26)5-6-20(21)17-9-14(13-29-24-27-7-8-28-24)10-18(11-17)23(31)30-22(15-1-2-15)16-3-4-16/h5-6,9-12,15-16,22H,1-4,7-8,13H2,(H,30,31)(H2,27,28,29)	IAJHBHHTWPWBQR-UHFFFAOYSA-N	468656	US10807959, Example 2	WD repeat-containing protein 5		 6.00								US Patent		10.7270/Q26Q219X		aid1804926	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468656	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468656&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370880	441570757							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968568	COc1cc(CNC(=O)c2cc(CNC3=NCCN3)cc(c2)-c2ccc(F)cc2Cl)cc(OC)c1	InChI=1S/C26H26ClFN4O3/c1-34-21-9-17(10-22(13-21)35-2)14-31-25(33)19-8-16(15-32-26-29-5-6-30-26)7-18(11-19)23-4-3-20(28)12-24(23)27/h3-4,7-13H,5-6,14-15H2,1-2H3,(H,31,33)(H2,29,30,32)	NCDDOTFEQCIEET-UHFFFAOYSA-N	468657	US10807959, Example 3	WD repeat-containing protein 5		 2.70								US Patent		10.7270/Q26Q219X		aid1804926	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468657	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468657&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370897	441570758							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968569	Clc1cc(Cl)cc(CNC(=O)c2cc(Cl)cc(Cn3ccnc3)c2)c1	InChI=1S/C18H14Cl3N3O/c19-15-6-13(10-24-2-1-22-11-24)3-14(7-15)18(25)23-9-12-4-16(20)8-17(21)5-12/h1-8,11H,9-10H2,(H,23,25)	FQDHIPIENIYXFJ-UHFFFAOYSA-N	468698	US10807959, Example 110	WD repeat-containing protein 5		 33.7								US Patent		10.7270/Q26Q219X		aid1804926	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468698	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468698&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370876	441570799							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968570	COc1cc(CNC(=O)c2cc(Cl)cc(Cn3ccnc3)c2)cc(OC)c1	InChI=1S/C20H20ClN3O3/c1-26-18-7-14(8-19(10-18)27-2)11-23-20(25)16-5-15(6-17(21)9-16)12-24-4-3-22-13-24/h3-10,13H,11-12H2,1-2H3,(H,23,25)	UMMZDUDQWHLSAQ-UHFFFAOYSA-N	468699	US10807959, Example 111	WD repeat-containing protein 5		 135								US Patent		10.7270/Q26Q219X		aid1804926	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468699	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468699&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370871	441570800							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968571	Cc1ccc(CNC(=O)c2cc(Cl)cc(Cn3ccnc3)c2)cc1Cl	InChI=1S/C19H17Cl2N3O/c1-13-2-3-14(8-18(13)21)10-23-19(25)16-6-15(7-17(20)9-16)11-24-5-4-22-12-24/h2-9,12H,10-11H2,1H3,(H,23,25)	GEMSEPIHRWFUHO-UHFFFAOYSA-N	468700	US10807959, Example 112	WD repeat-containing protein 5		 141								US Patent		10.7270/Q26Q219X		aid1804926	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468700	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468700&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370793	441570801							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968572	COc1cc(Cn2ccnc2)cc(c1)C(=O)NCc1ccc(Cl)c(C)c1	InChI=1S/C20H20ClN3O2/c1-14-7-15(3-4-19(14)21)11-23-20(25)17-8-16(9-18(10-17)26-2)12-24-6-5-22-13-24/h3-10,13H,11-12H2,1-2H3,(H,23,25)	ZYLKBLAXINMOCN-UHFFFAOYSA-N	468701	US10807959, Example 113	WD repeat-containing protein 5		 141								US Patent		10.7270/Q26Q219X		aid1804926	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468701	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468701&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370828	441570802							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968573	COC(=O)CC(NC(=O)c1cc(Cl)cc(Cn2ccnc2)c1)c1cccc(Cl)c1	InChI=1S/C21H19Cl2N3O3/c1-29-20(27)11-19(15-3-2-4-17(22)9-15)25-21(28)16-7-14(8-18(23)10-16)12-26-6-5-24-13-26/h2-10,13,19H,11-12H2,1H3,(H,25,28)	KPSYDAWMUQTVFA-UHFFFAOYSA-N	468702	US10807959, Example 114	WD repeat-containing protein 5		 298								US Patent		10.7270/Q26Q219X		aid1804926	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468702	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468702&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370968	441570803							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968574	Cc1cc(CNC(=O)c2cc(Cn3ccnc3)cc(OC3CCCC3)c2)ccc1Cl	InChI=1S/C24H26ClN3O2/c1-17-10-18(6-7-23(17)25)14-27-24(29)20-11-19(15-28-9-8-26-16-28)12-22(13-20)30-21-4-2-3-5-21/h6-13,16,21H,2-5,14-15H2,1H3,(H,27,29)	QANZWSJBKGEFJF-UHFFFAOYSA-N	468703	US10807959, Example 115	WD repeat-containing protein 5		 3.50								US Patent		10.7270/Q26Q219X		aid1804926	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468703	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468703&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370782	441570804							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968575	Fc1ccc(c(Cl)c1)-c1cc(Cn2ccnc2)cc(c1)C(=O)NCc1ccc(Cl)c(Cl)c1	InChI=1S/C24H17Cl3FN3O/c25-21-4-1-15(9-23(21)27)12-30-24(32)18-8-16(13-31-6-5-29-14-31)7-17(10-18)20-3-2-19(28)11-22(20)26/h1-11,14H,12-13H2,(H,30,32)	MLESPKVIRFJOEN-UHFFFAOYSA-N	468704	US10807959, Example 116	WD repeat-containing protein 5		 1.90								US Patent		10.7270/Q26Q219X		aid1804926	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468704	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468704&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370869	441570805							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968576	COc1ccccc1-c1cc(Cn2ccnc2)cc(c1)C(=O)NCc1ccc(Cl)c(Cl)c1	InChI=1S/C25H21Cl2N3O2/c1-32-24-5-3-2-4-21(24)19-10-18(15-30-9-8-28-16-30)11-20(13-19)25(31)29-14-17-6-7-22(26)23(27)12-17/h2-13,16H,14-15H2,1H3,(H,29,31)	ZGHSAUNYSOAFQT-UHFFFAOYSA-N	468705	US10807959, Example 117	WD repeat-containing protein 5		 13.0								US Patent		10.7270/Q26Q219X		aid1804926	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468705	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468705&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370941	441570806							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968577	Clc1ccc(CNC(=O)c2cc(Cn3ccnc3)cc(c2)-c2cccnc2)cc1Cl	InChI=1S/C23H18Cl2N4O/c24-21-4-3-16(10-22(21)25)12-28-23(30)20-9-17(14-29-7-6-27-15-29)8-19(11-20)18-2-1-5-26-13-18/h1-11,13,15H,12,14H2,(H,28,30)	OAMUQCKZKPALOG-UHFFFAOYSA-N	468706	US10807959, Example 118	WD repeat-containing protein 5		 10.3								US Patent		10.7270/Q26Q219X		aid1804926	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468706	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468706&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370845	441570807							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968578	Clc1ccc(CNC(=O)c2cc(Cn3ccnc3)cc(c2)-c2ccco2)cc1Cl	InChI=1S/C22H17Cl2N3O2/c23-19-4-3-15(10-20(19)24)12-26-22(28)18-9-16(13-27-6-5-25-14-27)8-17(11-18)21-2-1-7-29-21/h1-11,14H,12-13H2,(H,26,28)	NSTIDFKHTYHBCL-UHFFFAOYSA-N	468707	US10807959, Example 119	WD repeat-containing protein 5		 3.30								US Patent		10.7270/Q26Q219X		aid1804926	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468707	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468707&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370863	441570808							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968579	COc1cc(CNC(=O)c2cc(Cn3ccnc3)cc(Oc3ccccc3)c2)cc(OC)c1	InChI=1S/C26H25N3O4/c1-31-23-11-19(12-24(15-23)32-2)16-28-26(30)21-10-20(17-29-9-8-27-18-29)13-25(14-21)33-22-6-4-3-5-7-22/h3-15,18H,16-17H2,1-2H3,(H,28,30)	WHVUFHHUSRSPMN-UHFFFAOYSA-N	468708	US10807959, Example 120	WD repeat-containing protein 5		 5.10								US Patent		10.7270/Q26Q219X		aid1804926	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468708	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468708&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370742	441570809							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968580	Cc1ccncc1-c1cc(Cn2ccnc2)cc(c1)C(=O)NCc1ccc(Cl)c(Cl)c1	InChI=1S/C24H20Cl2N4O/c1-16-4-5-27-13-21(16)19-8-18(14-30-7-6-28-15-30)9-20(11-19)24(31)29-12-17-2-3-22(25)23(26)10-17/h2-11,13,15H,12,14H2,1H3,(H,29,31)	YJYBPVLABQABCY-UHFFFAOYSA-N	468709	US10807959, Example 121	WD repeat-containing protein 5		 1.30								US Patent		10.7270/Q26Q219X		aid1804926	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468709	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468709&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146371097	441570810							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968581	Cc1ccc(Cl)c(c1)-c1cc(Cn2ccnc2)cc(c1)C(=O)NCc1ccc(Cl)c(Cl)c1	InChI=1S/C25H20Cl3N3O/c1-16-2-4-22(26)21(8-16)19-9-18(14-31-7-6-29-15-31)10-20(12-19)25(32)30-13-17-3-5-23(27)24(28)11-17/h2-12,15H,13-14H2,1H3,(H,30,32)	BVPOMEXWTCOUOE-UHFFFAOYSA-N	468710	US10807959, Example 122	WD repeat-containing protein 5		 2.20								US Patent		10.7270/Q26Q219X		aid1804926	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468710	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468710&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370729	441570811							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968582	Cc1cc(ccn1)-c1cc(Cn2ccnc2)cc(c1)C(=O)NCc1ccc(Cl)c(Cl)c1	InChI=1S/C24H20Cl2N4O/c1-16-8-19(4-5-28-16)20-9-18(14-30-7-6-27-15-30)10-21(12-20)24(31)29-13-17-2-3-22(25)23(26)11-17/h2-12,15H,13-14H2,1H3,(H,29,31)	PGTCTXLGORKJAN-UHFFFAOYSA-N	468711	US10807959, Example 123	WD repeat-containing protein 5		 8.70								US Patent		10.7270/Q26Q219X		aid1804926	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468711	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468711&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370841	441570812							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968583	FC(F)(F)c1ccccc1-c1cc(Cn2ccnc2)cc(c1)C(=O)NCc1ccc(Cl)c(Cl)c1	InChI=1S/C25H18Cl2F3N3O/c26-22-6-5-16(11-23(22)27)13-32-24(34)19-10-17(14-33-8-7-31-15-33)9-18(12-19)20-3-1-2-4-21(20)25(28,29)30/h1-12,15H,13-14H2,(H,32,34)	GJAMUNKMOBULNL-UHFFFAOYSA-N	468712	US10807959, Example 124	WD repeat-containing protein 5		 1.80								US Patent		10.7270/Q26Q219X		aid1804926	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468712	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468712&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370889	441570813							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968584	Clc1ccc(CNC(=O)c2cc(Cn3ccnc3)cc(c2)-c2ccncc2Cl)cc1Cl	InChI=1S/C23H17Cl3N4O/c24-20-2-1-15(9-21(20)25)11-29-23(31)18-8-16(13-30-6-5-28-14-30)7-17(10-18)19-3-4-27-12-22(19)26/h1-10,12,14H,11,13H2,(H,29,31)	LQJZKPUTDJTISG-UHFFFAOYSA-N	468713	US10807959, Example 125	WD repeat-containing protein 5		 1.90								US Patent		10.7270/Q26Q219X		aid1804926	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468713	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468713&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146371088	441570814							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968585	Cc1nc(F)ccc1-c1cc(Cn2ccnc2)cc(c1)C(=O)NCc1ccc(Cl)c(Cl)c1	InChI=1S/C24H19Cl2FN4O/c1-15-20(3-5-23(27)30-15)18-8-17(13-31-7-6-28-14-31)9-19(11-18)24(32)29-12-16-2-4-21(25)22(26)10-16/h2-11,14H,12-13H2,1H3,(H,29,32)	ZMEHLTRGAHGRAP-UHFFFAOYSA-N	468714	US10807959, Example 126	WD repeat-containing protein 5		<1.000								US Patent		10.7270/Q26Q219X		aid1804926	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468714	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468714&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370781	441570815							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968586	Fc1ccc(-c2cc(Cn3ccnc3)cc(c2)C(=O)NCc2ccc(Cl)c(Cl)c2)c(c1)C(F)(F)F	InChI=1S/C25H17Cl2F4N3O/c26-22-4-1-15(9-23(22)27)12-33-24(35)18-8-16(13-34-6-5-32-14-34)7-17(10-18)20-3-2-19(28)11-21(20)25(29,30)31/h1-11,14H,12-13H2,(H,33,35)	POQSNZTZYBLMPI-UHFFFAOYSA-N	468715	US10807959, Example 127	WD repeat-containing protein 5		<1.000								US Patent		10.7270/Q26Q219X		aid1804926	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468715	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468715&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370769	441570816							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968587	COc1cncc(c1)-c1cc(Cn2ccnc2)cc(c1)C(=O)NCc1ccc(Cl)c(Cl)c1	InChI=1S/C24H20Cl2N4O2/c1-32-21-10-20(12-28-13-21)18-6-17(14-30-5-4-27-15-30)7-19(9-18)24(31)29-11-16-2-3-22(25)23(26)8-16/h2-10,12-13,15H,11,14H2,1H3,(H,29,31)	MMXOBKKQVRAKNU-UHFFFAOYSA-N	468716	US10807959, Example 128	WD repeat-containing protein 5		 2.20								US Patent		10.7270/Q26Q219X		aid1804926	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468716	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468716&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370743	441570817							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968588	COc1cnccc1-c1cc(Cn2ccnc2)cc(c1)C(=O)NCc1ccc(Cl)c(Cl)c1	InChI=1S/C24H20Cl2N4O2/c1-32-23-13-27-5-4-20(23)18-8-17(14-30-7-6-28-15-30)9-19(11-18)24(31)29-12-16-2-3-21(25)22(26)10-16/h2-11,13,15H,12,14H2,1H3,(H,29,31)	OAPFQMOINAKDGH-UHFFFAOYSA-N	468717	US10807959, Example 129	WD repeat-containing protein 5		 5.90								US Patent		10.7270/Q26Q219X		aid1804926	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468717	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468717&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370862	441570818							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968589	COc1cc(CNC(=O)c2cc(Cn3ccnc3)cc(c2)-c2ccoc2C)cc(OC)c1	InChI=1S/C25H25N3O4/c1-17-24(4-7-32-17)20-8-19(15-28-6-5-26-16-28)9-21(12-20)25(29)27-14-18-10-22(30-2)13-23(11-18)31-3/h4-13,16H,14-15H2,1-3H3,(H,27,29)	DOYICUYSNWKLEQ-UHFFFAOYSA-N	468718	US10807959, Example 130	WD repeat-containing protein 5		 2.10								US Patent		10.7270/Q26Q219X		aid1804926	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468718	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468718&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370921	441570819							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968590	Cn1nccc1-c1cc(Cn2ccnc2)cc(c1)C(=O)NCc1ccc(Cl)c(Cl)c1	InChI=1S/C22H19Cl2N5O/c1-28-21(4-5-27-28)17-8-16(13-29-7-6-25-14-29)9-18(11-17)22(30)26-12-15-2-3-19(23)20(24)10-15/h2-11,14H,12-13H2,1H3,(H,26,30)	SSAPHCMBLIIGMI-UHFFFAOYSA-N	468719	US10807959, Example 131	WD repeat-containing protein 5		<1.000								US Patent		10.7270/Q26Q219X		aid1804926	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468719	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468719&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146371020	441570820							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968591	CC(NC(=O)c1cc(Cn2ccnc2)cc(c1)-c1ccc(F)nc1C)C1CCCCC1	InChI=1S/C25H29FN4O/c1-17(20-6-4-3-5-7-20)29-25(31)22-13-19(15-30-11-10-27-16-30)12-21(14-22)23-8-9-24(26)28-18(23)2/h8-14,16-17,20H,3-7,15H2,1-2H3,(H,29,31)	YLXBDLUEVXMJMM-UHFFFAOYSA-N	468720	US10807959, Example 132	WD repeat-containing protein 5		 3.90								US Patent		10.7270/Q26Q219X		aid1804926	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468720	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468720&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370844	441570821							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968592	Cc1nc(F)ccc1-c1cc(Cn2ccnc2)cc(c1)C(=O)NC(C1CC1)C1CC1	InChI=1S/C24H25FN4O/c1-15-21(6-7-22(25)27-15)19-10-16(13-29-9-8-26-14-29)11-20(12-19)24(30)28-23(17-2-3-17)18-4-5-18/h6-12,14,17-18,23H,2-5,13H2,1H3,(H,28,30)	NDWGDICKLLHJRK-UHFFFAOYSA-N	468721	US10807959, Example 133	WD repeat-containing protein 5		 3.50								US Patent		10.7270/Q26Q219X		aid1804926	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468721	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468721&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370840	441570822							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968593	Cc1nccn1Cc1cc(cc(c1)-c1ccc(F)cc1Cl)C(=O)NCc1ccc(Cl)c(Cl)c1	InChI=1S/C25H19Cl3FN3O/c1-15-30-6-7-32(15)14-17-8-18(21-4-3-20(29)12-23(21)27)11-19(9-17)25(33)31-13-16-2-5-22(26)24(28)10-16/h2-12H,13-14H2,1H3,(H,31,33)	UUQJUPSTHIASAJ-UHFFFAOYSA-N	468722	US10807959, Example 134	WD repeat-containing protein 5		 1.60								US Patent		10.7270/Q26Q219X		aid1804926	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468722	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468722&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370927	441570823							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968594	Fc1ccc(c(Cl)c1)-c1cc(Cn2ccnc2C(F)(F)F)cc(c1)C(=O)NCc1ccc(Cl)c(Cl)c1	InChI=1S/C25H16Cl3F4N3O/c26-20-4-1-14(9-22(20)28)12-34-23(36)17-8-15(13-35-6-5-33-24(35)25(30,31)32)7-16(10-17)19-3-2-18(29)11-21(19)27/h1-11H,12-13H2,(H,34,36)	WNCWNJIZHNAUEN-UHFFFAOYSA-N	468723	US10807959, Example 135	WD repeat-containing protein 5		>10000								US Patent		10.7270/Q26Q219X		aid1804926	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468723	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468723&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370919	441570824							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981396	Cc1nc(F)ccc1-c1cc(Cn2ccn(C)c2=N)cc(c1)C(=O)NCc1ccc(Cl)c(Cl)c1	InChI=1S/C25H22Cl2FN5O/c1-15-20(4-6-23(28)31-15)18-9-17(14-33-8-7-32(2)25(33)29)10-19(12-18)24(34)30-13-16-3-5-21(26)22(27)11-16/h3-12,29H,13-14H2,1-2H3,(H,30,34)	ZPVQIJIWGMKMQN-UHFFFAOYSA-N	50520121	CHEMBL4441671::US10844044, Example 1	WD repeat-containing protein 5		<0.100								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50520121	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50520121&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	HLJ	6E23	138319680	440728703							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981397	Cc1ccccc1-c1cc(Cn2ccn(C)c2=N)cc(c1)C(=O)NCc1ccc(Cl)c(Cl)c1	InChI=1S/C26H24Cl2N4O/c1-17-5-3-4-6-22(17)20-11-19(16-32-10-9-31(2)26(32)29)12-21(14-20)25(33)30-15-18-7-8-23(27)24(28)13-18/h3-14,29H,15-16H2,1-2H3,(H,30,33)	RHGYLKDWASNERE-UHFFFAOYSA-N	473191	US10844044, Example 92	WD repeat-containing protein 5		 0.720								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473191	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473191&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456817	442073403							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981398	CCOc1cc(Cn2ccn(C)c2=N)cc(c1)C(=O)NCc1ccc(Cl)c(C)c1	InChI=1S/C22H25ClN4O2/c1-4-29-19-11-17(14-27-8-7-26(3)22(27)24)10-18(12-19)21(28)25-13-16-5-6-20(23)15(2)9-16/h5-12,24H,4,13-14H2,1-3H3,(H,25,28)	SPWRKNPIYYHHOE-UHFFFAOYSA-N	473192	US10844044, Example 183	WD repeat-containing protein 5		 0.710								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473192	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473192&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146455921	442073404							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981399	CC(C)n1cc(c(n1)C(F)(F)F)-c1cc(CN2CCOC2=N)cc(c1)C(=O)N[C@@H](C1CC1)c1ccc(F)c(C)c1	InChI=1S/C29H31F4N5O2/c1-16(2)38-15-23(26(36-38)29(31,32)33)21-11-18(14-37-8-9-40-28(37)34)12-22(13-21)27(39)35-25(19-4-5-19)20-6-7-24(30)17(3)10-20/h6-7,10-13,15-16,19,25,34H,4-5,8-9,14H2,1-3H3,(H,35,39)/t25-/m0/s1	SMCRFJSYTSPBMP-VWLOTQADSA-N	473193	US10844044, Example 275	WD repeat-containing protein 5		<0.100								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473193	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473193&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456160	442073405							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981400	COc1ncc(C)cc1-c1cc(Cn2ccn(C)c2=N)cc(c1)C(=O)NC(C1CC1)c1cc(C)ccn1	InChI=1S/C29H32N6O2/c1-18-7-8-31-25(12-18)26(21-5-6-21)33-27(36)23-14-20(17-35-10-9-34(3)29(35)30)13-22(15-23)24-11-19(2)16-32-28(24)37-4/h7-16,21,26,30H,5-6,17H2,1-4H3,(H,33,36)	JVLGUFGOOHDVOV-UHFFFAOYSA-N	473194	US10844044, Example 2	WD repeat-containing protein 5		<0.100								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473194	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473194&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456935	442073406							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981401	COc1ccnc(c1)[C@H](NC(=O)c1cc(Cn2ccn(C)c2=N)cc(c1)-c1ccc(F)cc1C)C1CC1	InChI=1S/C29H30FN5O2/c1-18-12-23(30)6-7-25(18)21-13-19(17-35-11-10-34(2)29(35)31)14-22(15-21)28(36)33-27(20-4-5-20)26-16-24(37-3)8-9-32-26/h6-16,20,27,31H,4-5,17H2,1-3H3,(H,33,36)/t27-/m1/s1	JMMNYJULKRGWMJ-HHHXNRCGSA-N	473195	US10844044, Example 93	WD repeat-containing protein 5		 1.90								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473195	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473195&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456264	442073407							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981402	COc1cc(c(F)cn1)-c1cc(Cn2ccn(C)c2=N)cc(c1)C(=O)NCc1ccc(Cl)c(Cl)c1	InChI=1S/C25H22Cl2FN5O2/c1-32-5-6-33(25(32)29)14-16-7-17(19-11-23(35-2)30-13-22(19)28)10-18(8-16)24(34)31-12-15-3-4-20(26)21(27)9-15/h3-11,13,29H,12,14H2,1-2H3,(H,31,34)	RKKFZAOPNHOZNW-UHFFFAOYSA-N	473196	US10844044, Example 184	WD repeat-containing protein 5		 0.560								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473196	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473196&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146455708	442073408							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968595	Clc1ccc(CNC(=O)c2cc(Cn3ccnc3)cc(c2)N2CCCC2)cc1Cl	InChI=1S/C22H22Cl2N4O/c23-20-4-3-16(11-21(20)24)13-26-22(29)18-9-17(14-27-8-5-25-15-27)10-19(12-18)28-6-1-2-7-28/h3-5,8-12,15H,1-2,6-7,13-14H2,(H,26,29)	BDOCXEVVVXWIRT-UHFFFAOYSA-N	468724	US10807959, Example 136	WD repeat-containing protein 5		 6.50								US Patent		10.7270/Q26Q219X		aid1804926	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468724	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468724&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370820	441570825							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968596	Cc1ccnc(c1)C(NC(=O)c1cc(Cn2ccnc2)cc(c1)-c1ccc(F)nc1C)C1CC1	InChI=1S/C27H26FN5O/c1-17-7-8-30-24(11-17)26(20-3-4-20)32-27(34)22-13-19(15-33-10-9-29-16-33)12-21(14-22)23-5-6-25(28)31-18(23)2/h5-14,16,20,26H,3-4,15H2,1-2H3,(H,32,34)	UBPIMOHMVJQFFW-UHFFFAOYSA-N	468725	US10807959, Example 137	WD repeat-containing protein 5		<1.000								US Patent		10.7270/Q26Q219X		aid1804926	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468725	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468725&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370915	441570826							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968597	Fc1ccc(c(Cl)c1)-c1cc(Cn2ccnc2)cc(n1)C(=O)NCc1cc(Cl)cc(Cl)c1	InChI=1S/C23H16Cl3FN4O/c24-16-5-14(6-17(25)9-16)11-29-23(32)22-8-15(12-31-4-3-28-13-31)7-21(30-22)19-2-1-18(27)10-20(19)26/h1-10,13H,11-12H2,(H,29,32)	DVTOVXLDZCQPEV-UHFFFAOYSA-N	468726	US10807959, Example 148	WD repeat-containing protein 5		 1.60								US Patent		10.7270/Q26Q219X		aid1804926	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468726	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468726&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370992	441570827							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968598	CC(C)(NC(=O)c1cc(Cn2ccnc2)cc(n1)-c1ccc(F)cc1Cl)C1CC1	InChI=1S/C22H22ClFN4O/c1-22(2,15-3-4-15)27-21(29)20-10-14(12-28-8-7-25-13-28)9-19(26-20)17-6-5-16(24)11-18(17)23/h5-11,13,15H,3-4,12H2,1-2H3,(H,27,29)	JXVNRFPBVYCJFU-UHFFFAOYSA-N	468727	US10807959, Example 149	WD repeat-containing protein 5		 8.60								US Patent		10.7270/Q26Q219X		aid1804926	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468727	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468727&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370784	441570828							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968599	Cc1ccnc(c1)C(NC(=O)c1cc(Cn2ccnc2)cc(n1)-c1ccc(F)cc1Cl)C1CC1	InChI=1S/C26H23ClFN5O/c1-16-6-7-30-23(10-16)25(18-2-3-18)32-26(34)24-12-17(14-33-9-8-29-15-33)11-22(31-24)20-5-4-19(28)13-21(20)27/h4-13,15,18,25H,2-3,14H2,1H3,(H,32,34)	NLWDHZNWWYOXLN-UHFFFAOYSA-N	468728	US10807959, Example 150	WD repeat-containing protein 5		 1.10								US Patent		10.7270/Q26Q219X		aid1804926	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468728	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468728&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146371012	441570829							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968600	Cc1cccc(CNC(=O)c2cc(Cn3ccnc3)cc(n2)-c2ccc(F)cc2Cl)n1	InChI=1S/C23H19ClFN5O/c1-15-3-2-4-18(28-15)12-27-23(31)22-10-16(13-30-8-7-26-14-30)9-21(29-22)19-6-5-17(25)11-20(19)24/h2-11,14H,12-13H2,1H3,(H,27,31)	FCVZKYYPBCCHIA-UHFFFAOYSA-N	468729	US10807959, Example 151	WD repeat-containing protein 5		 8.70								US Patent		10.7270/Q26Q219X		aid1804926	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468729	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468729&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370878	441570830							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968601	CCC(NC(=O)c1cc(Cn2ccnc2)cc(n1)-c1ccc(F)cc1Cl)C1CC1	InChI=1S/C22H22ClFN4O/c1-2-19(15-3-4-15)27-22(29)21-10-14(12-28-8-7-25-13-28)9-20(26-21)17-6-5-16(24)11-18(17)23/h5-11,13,15,19H,2-4,12H2,1H3,(H,27,29)	XFRZUAFNQSJGKI-UHFFFAOYSA-N	468730	US10807959, Example 152	WD repeat-containing protein 5		 13.1								US Patent		10.7270/Q26Q219X		aid1804926	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468730	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468730&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370959	441570831							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968602	Cc1cc(C)cc(CNC(=O)c2cc(Cn3ccnc3)cc(n2)-c2ccc(F)cc2Cl)c1	InChI=1S/C25H22ClFN4O/c1-16-7-17(2)9-18(8-16)13-29-25(32)24-11-19(14-31-6-5-28-15-31)10-23(30-24)21-4-3-20(27)12-22(21)26/h3-12,15H,13-14H2,1-2H3,(H,29,32)	ZWTHKWDWPWZUMG-UHFFFAOYSA-N	468731	US10807959, Example 153	WD repeat-containing protein 5		 4.80								US Patent		10.7270/Q26Q219X		aid1804926	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468731	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468731&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146371024	441570832							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968603	COc1cc(OC)cc(c1)C(C)NC(=O)c1cc(Cn2ccnc2)cc(n1)-c1ccc(F)cc1Cl	InChI=1S/C26H24ClFN4O3/c1-16(18-10-20(34-2)13-21(11-18)35-3)30-26(33)25-9-17(14-32-7-6-29-15-32)8-24(31-25)22-5-4-19(28)12-23(22)27/h4-13,15-16H,14H2,1-3H3,(H,30,33)	QNFRUEXTNWMWRQ-UHFFFAOYSA-N	468732	US10807959, Example 154	WD repeat-containing protein 5		 5.10								US Patent		10.7270/Q26Q219X		aid1804926	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468732	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468732&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370835	441570833							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968604	CC(NC(=O)c1cc(Cn2ccnc2)cc(n1)-c1ccc(F)cc1Cl)c1ccccn1	InChI=1S/C23H19ClFN5O/c1-15(20-4-2-3-7-27-20)28-23(31)22-11-16(13-30-9-8-26-14-30)10-21(29-22)18-6-5-17(25)12-19(18)24/h2-12,14-15H,13H2,1H3,(H,28,31)	FDNOUKNRKBXWJS-UHFFFAOYSA-N	468733	US10807959, Example 155	WD repeat-containing protein 5		 21.9								US Patent		10.7270/Q26Q219X		aid1804926	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468733	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468733&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370849	441570834							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968605	COc1cc(OC)cc(c1)C(C)NC(=O)c1cc(CNC2=NCCN2)cc(c1)-c1ccc(F)cc1C	InChI=1S/C28H31FN4O3/c1-17-9-23(29)5-6-26(17)21-10-19(16-32-28-30-7-8-31-28)11-22(12-21)27(34)33-18(2)20-13-24(35-3)15-25(14-20)36-4/h5-6,9-15,18H,7-8,16H2,1-4H3,(H,33,34)(H2,30,31,32)	VRNHATNYXMZSFL-UHFFFAOYSA-N	468734	US10807959, Example 1	WD repeat-containing protein 5		 0.460								US Patent		10.7270/Q26Q219X		aid1804927	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468734	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468734&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370896	441570835							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968606	COc1ccc(CNC(=O)c2cc(CNC3=NCCN3)cc(c2)-c2ccc(F)nc2C)cc1OC	InChI=1S/C26H28FN5O3/c1-16-21(5-7-24(27)32-16)19-10-18(15-31-26-28-8-9-29-26)11-20(13-19)25(33)30-14-17-4-6-22(34-2)23(12-17)35-3/h4-7,10-13H,8-9,14-15H2,1-3H3,(H,30,33)(H2,28,29,31)	LXKXGQLWYWEGOP-UHFFFAOYSA-N	468735	US10807959, Example 4	WD repeat-containing protein 5		 0.360								US Patent		10.7270/Q26Q219X		aid1804927	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468735	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468735&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370783	441570836							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968607	Cc1cc(CNC(=O)c2cc(CNC3=NCCN3)cc(c2)-c2ccc(F)nc2C)ccc1Cl	InChI=1S/C25H25ClFN5O/c1-15-9-17(3-5-22(15)26)13-30-24(33)20-11-18(14-31-25-28-7-8-29-25)10-19(12-20)21-4-6-23(27)32-16(21)2/h3-6,9-12H,7-8,13-14H2,1-2H3,(H,30,33)(H2,28,29,31)	HYUIOAVDRVFASD-UHFFFAOYSA-N	468736	US10807959, Example 5	WD repeat-containing protein 5		 0.020								US Patent		10.7270/Q26Q219X		aid1804927	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468736	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468736&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370990	441570837							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968608	Cc1cc(C)cc(CNC(=O)c2cc(CNC3=NCCN3)cc(c2)-c2ccc(F)nc2C)c1	InChI=1S/C26H28FN5O/c1-16-8-17(2)10-19(9-16)14-30-25(33)22-12-20(15-31-26-28-6-7-29-26)11-21(13-22)23-4-5-24(27)32-18(23)3/h4-5,8-13H,6-7,14-15H2,1-3H3,(H,30,33)(H2,28,29,31)	XTTCEUVGQFYKBU-UHFFFAOYSA-N	468737	US10807959, Example 6	WD repeat-containing protein 5		 0.140								US Patent		10.7270/Q26Q219X		aid1804927	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468737	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468737&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370861	441570838							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968609	COc1cc(OC)cc(c1)C(C)NC(=O)c1cc(CNC2=NCCN2)cc(c1)-c1ccc(F)nc1C	InChI=1S/C27H30FN5O3/c1-16(19-12-22(35-3)14-23(13-19)36-4)33-26(34)21-10-18(15-31-27-29-7-8-30-27)9-20(11-21)24-5-6-25(28)32-17(24)2/h5-6,9-14,16H,7-8,15H2,1-4H3,(H,33,34)(H2,29,30,31)	OMDNPCMMOWFKGA-UHFFFAOYSA-N	468738	US10807959, Example 7	WD repeat-containing protein 5		 0.110								US Patent		10.7270/Q26Q219X		aid1804927	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468738	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468738&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370938	441570839							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968610	COc1cc(CN(C)C(=O)c2cc(CNC3=NCCN3)cc(c2)-c2ccc(F)nc2C)cc(OC)c1	InChI=1S/C27H30FN5O3/c1-17-24(5-6-25(28)32-17)20-9-18(15-31-27-29-7-8-30-27)10-21(13-20)26(34)33(2)16-19-11-22(35-3)14-23(12-19)36-4/h5-6,9-14H,7-8,15-16H2,1-4H3,(H2,29,30,31)	BCUYZPYONPMNJK-UHFFFAOYSA-N	468739	US10807959, Example 8	WD repeat-containing protein 5		 12.0								US Patent		10.7270/Q26Q219X		aid1804927	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468739	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468739&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370719	441570840							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968611	Cc1ccnc(c1)C(NC(=O)c1cc(CNC2=NCCN2)cc(c1)-c1ccc(F)nc1C)C1CC1	InChI=1S/C27H29FN6O/c1-16-7-8-29-23(11-16)25(19-3-4-19)34-26(35)21-13-18(15-32-27-30-9-10-31-27)12-20(14-21)22-5-6-24(28)33-17(22)2/h5-8,11-14,19,25H,3-4,9-10,15H2,1-2H3,(H,34,35)(H2,30,31,32)	UUOJOOPRBIMZID-UHFFFAOYSA-N	468740	US10807959, Example 9	WD repeat-containing protein 5		<0.100								US Patent		10.7270/Q26Q219X		aid1804927	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468740	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468740&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370826	441570841							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968612	Cc1nc(F)ccc1-c1cc(CNC2=NCCN2)cc(c1)C(=O)NC(C1CC1)C1CC1	InChI=1S/C24H28FN5O/c1-14-20(6-7-21(25)29-14)18-10-15(13-28-24-26-8-9-27-24)11-19(12-18)23(31)30-22(16-2-3-16)17-4-5-17/h6-7,10-12,16-17,22H,2-5,8-9,13H2,1H3,(H,30,31)(H2,26,27,28)	MQTGZGWPCINZPD-UHFFFAOYSA-N	468741	US10807959, Example 10	WD repeat-containing protein 5		 2.90								US Patent		10.7270/Q26Q219X		aid1804927	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468741	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468741&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370846	441570842							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968613	COc1ccnc(CNC(=O)c2cc(CNC3=NCCN3)cc(c2)-c2ccc(F)nc2C)c1	InChI=1S/C24H25FN6O2/c1-15-21(3-4-22(25)31-15)17-9-16(13-30-24-27-7-8-28-24)10-18(11-17)23(32)29-14-19-12-20(33-2)5-6-26-19/h3-6,9-12H,7-8,13-14H2,1-2H3,(H,29,32)(H2,27,28,30)	YMLHYSSHPLNUBK-UHFFFAOYSA-N	468742	US10807959, Example 11	WD repeat-containing protein 5		 0.220								US Patent		10.7270/Q26Q219X		aid1804927	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468742	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468742&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370732	441570843							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968614	Cc1ccncc1-c1cc(CNC2=NCCN2)cc(c1)C(=O)NCc1ccc(Cl)c(Cl)c1	InChI=1S/C24H23Cl2N5O/c1-15-4-5-27-14-20(15)18-8-17(13-31-24-28-6-7-29-24)9-19(11-18)23(32)30-12-16-2-3-21(25)22(26)10-16/h2-5,8-11,14H,6-7,12-13H2,1H3,(H,30,32)(H2,28,29,31)	BZTRCMPRKNFOBP-UHFFFAOYSA-N	468743	US10807959, Example 12	WD repeat-containing protein 5		<0.100								US Patent		10.7270/Q26Q219X		aid1804927	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468743	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468743&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370824	441570844							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968615	COc1cc(CNC(=O)c2cc(CNC3=NCCN3)cc(c2)-c2cnccc2C)cc(OC)c1	InChI=1S/C26H29N5O3/c1-17-4-5-27-16-24(17)20-8-18(15-31-26-28-6-7-29-26)9-21(12-20)25(32)30-14-19-10-22(33-2)13-23(11-19)34-3/h4-5,8-13,16H,6-7,14-15H2,1-3H3,(H,30,32)(H2,28,29,31)	XBNTUXGZTIUACW-UHFFFAOYSA-N	468744	US10807959, Example 13	WD repeat-containing protein 5		 0.530								US Patent		10.7270/Q26Q219X		aid1804927	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468744	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468744&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370906	441570845							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968616	COc1ccc(CNC(=O)c2cc(CNC3=NCCN3)cc(c2)-c2cnccc2C)cc1Cl	InChI=1S/C25H26ClN5O2/c1-16-5-6-27-15-21(16)19-9-18(14-31-25-28-7-8-29-25)10-20(12-19)24(32)30-13-17-3-4-23(33-2)22(26)11-17/h3-6,9-12,15H,7-8,13-14H2,1-2H3,(H,30,32)(H2,28,29,31)	RWCHPXIGOOPYBS-UHFFFAOYSA-N	468745	US10807959, Example 14	WD repeat-containing protein 5		 0.740								US Patent		10.7270/Q26Q219X		aid1804927	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468745	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468745&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370936	441570846							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968617	COc1ccc(CNC(=O)c2cc(CNC3=NCCN3)cc(c2)-c2ccnc(C)c2)cc1OC	InChI=1S/C26H29N5O3/c1-17-10-20(6-7-27-17)21-11-19(16-31-26-28-8-9-29-26)12-22(14-21)25(32)30-15-18-4-5-23(33-2)24(13-18)34-3/h4-7,10-14H,8-9,15-16H2,1-3H3,(H,30,32)(H2,28,29,31)	JOLOCYRJBJFRDB-UHFFFAOYSA-N	468746	US10807959, Example 15	WD repeat-containing protein 5		 1.70								US Patent		10.7270/Q26Q219X		aid1804927	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468746	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468746&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146371268	441570847							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968618	Cc1cc(ccn1)-c1cc(CNC2=NCCN2)cc(c1)C(=O)NCc1cc(F)cc(Cl)c1	InChI=1S/C24H23ClFN5O/c1-15-6-18(2-3-27-15)19-7-16(14-31-24-28-4-5-29-24)8-20(11-19)23(32)30-13-17-9-21(25)12-22(26)10-17/h2-3,6-12H,4-5,13-14H2,1H3,(H,30,32)(H2,28,29,31)	XHUVCOGWSGJBLK-UHFFFAOYSA-N	468747	US10807959, Example 16	WD repeat-containing protein 5		 0.520								US Patent		10.7270/Q26Q219X		aid1804927	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468747	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468747&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370834	441570848							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968619	COc1cc(CNC(=O)c2cc(CNC3=NCCN3)cc(c2)-c2ccnc(C)c2)ccc1Cl	InChI=1S/C25H26ClN5O2/c1-16-9-19(5-6-27-16)20-10-18(15-31-25-28-7-8-29-25)11-21(13-20)24(32)30-14-17-3-4-22(26)23(12-17)33-2/h3-6,9-13H,7-8,14-15H2,1-2H3,(H,30,32)(H2,28,29,31)	MRWCRYFXLRSTJU-UHFFFAOYSA-N	468748	US10807959, Example 17	WD repeat-containing protein 5		 3.20								US Patent		10.7270/Q26Q219X		aid1804927	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468748	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468748&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146371052	441570849							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968620	COc1cc(CNC(=O)c2cc(CNC3=NCCN3)cc(c2)-c2cnccc2C)ccc1Cl	InChI=1S/C25H26ClN5O2/c1-16-5-6-27-15-21(16)19-9-18(14-31-25-28-7-8-29-25)10-20(12-19)24(32)30-13-17-3-4-22(26)23(11-17)33-2/h3-6,9-12,15H,7-8,13-14H2,1-2H3,(H,30,32)(H2,28,29,31)	MVMYWNZMIQCMGI-UHFFFAOYSA-N	468749	US10807959, Example 18	WD repeat-containing protein 5		 3.10								US Patent		10.7270/Q26Q219X		aid1804927	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468749	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468749&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370916	441570850							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968621	COc1ccnc(CNC(=O)c2cc(CNC3=NCCN3)cc(c2)-c2cnccc2C)c1	InChI=1S/C24H26N6O2/c1-16-3-5-25-15-22(16)18-9-17(13-30-24-27-7-8-28-24)10-19(11-18)23(31)29-14-20-12-21(32-2)4-6-26-20/h3-6,9-12,15H,7-8,13-14H2,1-2H3,(H,29,31)(H2,27,28,30)	AREJUAVNDRFWSU-UHFFFAOYSA-N	468750	US10807959, Example 19	WD repeat-containing protein 5		 0.450								US Patent		10.7270/Q26Q219X		aid1804927	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468750	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468750&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370877	441570851							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968622	COc1cc(OC)cc(c1)C(C)NC(=O)c1cc(CNC2=NCCN2)cc(c1)-c1cnccc1C	InChI=1S/C27H31N5O3/c1-17-5-6-28-16-25(17)21-9-19(15-31-27-29-7-8-30-27)10-22(11-21)26(33)32-18(2)20-12-23(34-3)14-24(13-20)35-4/h5-6,9-14,16,18H,7-8,15H2,1-4H3,(H,32,33)(H2,29,30,31)	MSCXJTMDQLDZMM-UHFFFAOYSA-N	468751	US10807959, Example 20	WD repeat-containing protein 5		 0.600								US Patent		10.7270/Q26Q219X		aid1804927	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468751	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468751&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370994	441570852							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968623	COc1ccnc(CNC(=O)c2cc(CNC3=NCCN3)cc(c2)-c2ccnc(C)c2)c1	InChI=1S/C24H26N6O2/c1-16-9-18(3-5-25-16)19-10-17(14-30-24-27-7-8-28-24)11-20(12-19)23(31)29-15-21-13-22(32-2)4-6-26-21/h3-6,9-13H,7-8,14-15H2,1-2H3,(H,29,31)(H2,27,28,30)	DBDCPLDUOVLPLU-UHFFFAOYSA-N	468752	US10807959, Example 21	WD repeat-containing protein 5		 0.390								US Patent		10.7270/Q26Q219X		aid1804927	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468752	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468752&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370904	441570853							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968624	Cc1cc(ccn1)-c1cc(CNC2=NCCN2)cc(c1)C(=O)NCc1cc(Cl)ccn1	InChI=1S/C23H23ClN6O/c1-15-8-17(2-4-25-15)18-9-16(13-30-23-27-6-7-28-23)10-19(11-18)22(31)29-14-21-12-20(24)3-5-26-21/h2-5,8-12H,6-7,13-14H2,1H3,(H,29,31)(H2,27,28,30)	GGCRQQRXJISFDH-UHFFFAOYSA-N	468753	US10807959, Example 22	WD repeat-containing protein 5		 0.280								US Patent		10.7270/Q26Q219X		aid1804927	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468753	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468753&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370791	441570854							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968625	COc1ccc(CNC(=O)c2cc(CNC3=NCCN3)cc(c2)-c2ccnc(C)c2)cc1Cl	InChI=1S/C25H26ClN5O2/c1-16-9-19(5-6-27-16)20-10-18(15-31-25-28-7-8-29-25)11-21(13-20)24(32)30-14-17-3-4-23(33-2)22(26)12-17/h3-6,9-13H,7-8,14-15H2,1-2H3,(H,30,32)(H2,28,29,31)	VBCIFJGPJMOHLD-UHFFFAOYSA-N	468754	US10807959, Example 23	WD repeat-containing protein 5		 1.30								US Patent		10.7270/Q26Q219X		aid1804927	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468754	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468754&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370724	441570855							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968626	Cc1ccncc1-c1cc(CNC2=NCCN2)cc(c1)C(=O)NCc1cc(F)cc(Cl)c1	InChI=1S/C24H23ClFN5O/c1-15-2-3-27-14-22(15)18-6-16(13-31-24-28-4-5-29-24)7-19(10-18)23(32)30-12-17-8-20(25)11-21(26)9-17/h2-3,6-11,14H,4-5,12-13H2,1H3,(H,30,32)(H2,28,29,31)	GVGKNOIQPDRMNV-UHFFFAOYSA-N	468755	US10807959, Example 24	WD repeat-containing protein 5		 0.370								US Patent		10.7270/Q26Q219X		aid1804927	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468755	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468755&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370758	441570856							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968627	Cc1ccnc(c1)C(NC(=O)c1cc(CNC2=NCCN2)cc(c1)-c1cnccc1C)C1CC1	InChI=1S/C27H30N6O/c1-17-5-8-29-24(11-17)25(20-3-4-20)33-26(34)22-13-19(15-32-27-30-9-10-31-27)12-21(14-22)23-16-28-7-6-18(23)2/h5-8,11-14,16,20,25H,3-4,9-10,15H2,1-2H3,(H,33,34)(H2,30,31,32)	YRULKHGFIWOREI-UHFFFAOYSA-N	468756	US10807959, Example 25	WD repeat-containing protein 5		 0.200								US Patent		10.7270/Q26Q219X		aid1804927	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468756	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468756&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370893	441570857							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968628	Cc1ccc(CNC(=O)c2cc(CNC3=NCCN3)cc(c2)-c2ccnc(C)c2)cn1	InChI=1S/C24H26N6O/c1-16-3-4-18(13-28-16)14-29-23(31)22-11-19(15-30-24-26-7-8-27-24)10-21(12-22)20-5-6-25-17(2)9-20/h3-6,9-13H,7-8,14-15H2,1-2H3,(H,29,31)(H2,26,27,30)	CVDYLYARWPZCQA-UHFFFAOYSA-N	468757	US10807959, Example 26	WD repeat-containing protein 5		 3.00								US Patent		10.7270/Q26Q219X		aid1804927	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468757	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468757&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146371022	441570858							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968629	Cc1cc(ccn1)-c1cc(CNC2=NCCN2)cc(c1)C(=O)NCc1ccc(Cl)cn1	InChI=1S/C23H23ClN6O/c1-15-8-17(4-5-25-15)18-9-16(12-30-23-26-6-7-27-23)10-19(11-18)22(31)29-14-21-3-2-20(24)13-28-21/h2-5,8-11,13H,6-7,12,14H2,1H3,(H,29,31)(H2,26,27,30)	OOVKOIOBSWDQNL-UHFFFAOYSA-N	468758	US10807959, Example 27	WD repeat-containing protein 5		 1.50								US Patent		10.7270/Q26Q219X		aid1804927	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468758	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468758&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370767	441570859							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968630	Cc1ccc(CNC(=O)c2cc(CNC3=NCCN3)cc(c2)-c2cnccc2C)cn1	InChI=1S/C24H26N6O/c1-16-5-6-25-15-22(16)20-9-19(14-30-24-26-7-8-27-24)10-21(11-20)23(31)29-13-18-4-3-17(2)28-12-18/h3-6,9-12,15H,7-8,13-14H2,1-2H3,(H,29,31)(H2,26,27,30)	SBKBYEZLIDCKEV-UHFFFAOYSA-N	468759	US10807959, Example 28	WD repeat-containing protein 5		 7.60								US Patent		10.7270/Q26Q219X		aid1804927	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468759	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468759&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370779	441570860							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968631	Cc1ccnc(CNC(=O)c2cc(CNC3=NCCN3)cc(c2)-c2ccnc(C)c2)n1	InChI=1S/C23H25N7O/c1-15-3-5-25-21(30-15)14-28-22(31)20-11-17(13-29-23-26-7-8-27-23)10-19(12-20)18-4-6-24-16(2)9-18/h3-6,9-12H,7-8,13-14H2,1-2H3,(H,28,31)(H2,26,27,29)	AFTFTDWMJRYIBG-UHFFFAOYSA-N	468760	US10807959, Example 29	WD repeat-containing protein 5		 13.0								US Patent		10.7270/Q26Q219X		aid1804927	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468760	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468760&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370954	441570861							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968632	COc1cc(CNC(=O)c2cc(CNC3=NCCN3)cc(c2)-c2cnc(F)c(C)c2)cc(OC)c1	InChI=1S/C26H28FN5O3/c1-16-6-21(15-30-24(16)27)19-7-17(14-32-26-28-4-5-29-26)8-20(11-19)25(33)31-13-18-9-22(34-2)12-23(10-18)35-3/h6-12,15H,4-5,13-14H2,1-3H3,(H,31,33)(H2,28,29,32)	RAOHZPIFDZZFFY-UHFFFAOYSA-N	468761	US10807959, Example 30	WD repeat-containing protein 5		 0.330								US Patent		10.7270/Q26Q219X		aid1804927	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468761	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468761&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370882	441570862							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968633	Cc1cc(CNC(=O)c2cc(CNC3=NCCN3)cc(c2)-c2cnc(F)c(C)c2)ccc1Cl	InChI=1S/C25H25ClFN5O/c1-15-7-17(3-4-22(15)26)12-31-24(33)20-10-18(13-32-25-28-5-6-29-25)9-19(11-20)21-8-16(2)23(27)30-14-21/h3-4,7-11,14H,5-6,12-13H2,1-2H3,(H,31,33)(H2,28,29,32)	ABTRAMXICOTPGZ-UHFFFAOYSA-N	468762	US10807959, Example 31	WD repeat-containing protein 5		<0.100								US Patent		10.7270/Q26Q219X		aid1804927	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468762	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468762&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370738	441570863							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968634	Cc1cccc(Oc2cc(CNC3=NCCN3)cc(c2)C(=O)NCc2ccc(Cl)c(Cl)c2)c1	InChI=1S/C25H24Cl2N4O2/c1-16-3-2-4-20(9-16)33-21-11-18(15-31-25-28-7-8-29-25)10-19(13-21)24(32)30-14-17-5-6-22(26)23(27)12-17/h2-6,9-13H,7-8,14-15H2,1H3,(H,30,32)(H2,28,29,31)	BVPXPBGLNDLCKY-UHFFFAOYSA-N	468763	US10807959, Example 32	WD repeat-containing protein 5		 0.910								US Patent		10.7270/Q26Q219X		aid1804927	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468763	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468763&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370943	441570864							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968635	COc1cc(OC)cc(c1)C(C)NC(=O)c1cc(CNC2=NCCN2)cc(c1)C(F)(F)F	InChI=1S/C22H25F3N4O3/c1-13(15-9-18(31-2)11-19(10-15)32-3)29-20(30)16-6-14(7-17(8-16)22(23,24)25)12-28-21-26-4-5-27-21/h6-11,13H,4-5,12H2,1-3H3,(H,29,30)(H2,26,27,28)	CGMIWHNTSJYOCJ-UHFFFAOYSA-N	468764	US10807959, Example 33	WD repeat-containing protein 5		 8.90								US Patent		10.7270/Q26Q219X		aid1804927	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468764	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468764&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370987	441570865							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968636	COc1cc(CNC(=O)c2cc(CNC3=NCCN3)cc(c2)-c2cnc(OC)c(Cl)c2)cc(OC)c1	InChI=1S/C26H28ClN5O4/c1-34-21-8-17(9-22(12-21)35-2)13-30-24(33)19-7-16(14-32-26-28-4-5-29-26)6-18(10-19)20-11-23(27)25(36-3)31-15-20/h6-12,15H,4-5,13-14H2,1-3H3,(H,30,33)(H2,28,29,32)	VQOYFYDFIKNXMY-UHFFFAOYSA-N	468765	US10807959, Example 34	WD repeat-containing protein 5		 0.370								US Patent		10.7270/Q26Q219X		aid1804927	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468765	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468765&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370961	441570866							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968637	COc1cc(CNC(=O)c2cc(CNC3=NCCN3)cc(c2)-c2cnc(F)c(Cl)c2)cc(OC)c1	InChI=1S/C25H25ClFN5O3/c1-34-20-7-16(8-21(11-20)35-2)12-31-24(33)18-6-15(13-32-25-28-3-4-29-25)5-17(9-18)19-10-22(26)23(27)30-14-19/h5-11,14H,3-4,12-13H2,1-2H3,(H,31,33)(H2,28,29,32)	BXAYLADJSATDIP-UHFFFAOYSA-N	468766	US10807959, Example 35	WD repeat-containing protein 5		 0.360								US Patent		10.7270/Q26Q219X		aid1804927	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468766	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468766&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370837	441570867							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968638	Cc1cnc(CNC(=O)c2cc(CNC3=NCCN3)cc(c2)-c2ccc(F)nc2C)cn1	InChI=1S/C23H24FN7O/c1-14-10-28-19(12-27-14)13-29-22(32)18-8-16(11-30-23-25-5-6-26-23)7-17(9-18)20-3-4-21(24)31-15(20)2/h3-4,7-10,12H,5-6,11,13H2,1-2H3,(H,29,32)(H2,25,26,30)	BIMGNFAJIDRCDN-UHFFFAOYSA-N	468767	US10807959, Example 36	WD repeat-containing protein 5		 2.80								US Patent		10.7270/Q26Q219X		aid1804927	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468767	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468767&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146371245	441570868							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968639	Cc1ncc(CNC(=O)c2cc(CNC3=NCCN3)cc(c2)-c2ccc(F)nc2C)cn1	InChI=1S/C23H24FN7O/c1-14-20(3-4-21(24)31-14)18-7-16(10-30-23-25-5-6-26-23)8-19(9-18)22(32)29-13-17-11-27-15(2)28-12-17/h3-4,7-9,11-12H,5-6,10,13H2,1-2H3,(H,29,32)(H2,25,26,30)	ZSRIWEHLGLHIMK-UHFFFAOYSA-N	468768	US10807959, Example 37	WD repeat-containing protein 5		 2.10								US Patent		10.7270/Q26Q219X		aid1804927	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468768	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468768&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370905	441570869							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968640	Cc1cnc(F)c(c1)-c1cc(CNC2=NCCN2)cc(c1)C(=O)NCc1cc(Cl)ccn1	InChI=1S/C23H22ClFN6O/c1-14-6-20(21(25)29-11-14)16-7-15(12-31-23-27-4-5-28-23)8-17(9-16)22(32)30-13-19-10-18(24)2-3-26-19/h2-3,6-11H,4-5,12-13H2,1H3,(H,30,32)(H2,27,28,31)	LJUDJDLHXPBURH-UHFFFAOYSA-N	468769	US10807959, Example 38	WD repeat-containing protein 5		 0.260								US Patent		10.7270/Q26Q219X		aid1804927	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468769	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468769&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370715	441570870							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968641	Cc1ccnc(c1)C(NC(=O)c1cc(CNC2=NCCN2)cc(c1)-c1cc(C)cnc1F)C1CC1	InChI=1S/C27H29FN6O/c1-16-5-6-29-23(10-16)24(19-3-4-19)34-26(35)21-12-18(15-33-27-30-7-8-31-27)11-20(13-21)22-9-17(2)14-32-25(22)28/h5-6,9-14,19,24H,3-4,7-8,15H2,1-2H3,(H,34,35)(H2,30,31,33)	WWIWXPPDHSNLMK-UHFFFAOYSA-N	468770	US10807959, Example 39	WD repeat-containing protein 5		<0.100								US Patent		10.7270/Q26Q219X		aid1804927	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468770	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468770&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370969	441570871							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968642	CN(C)C(=O)c1cc(CNC2=NCCN2)cc(c1)-c1cc(C)cnc1F	InChI=1S/C19H22FN5O/c1-12-6-16(17(20)23-10-12)14-7-13(11-24-19-21-4-5-22-19)8-15(9-14)18(26)25(2)3/h6-10H,4-5,11H2,1-3H3,(H2,21,22,24)	JATRNMJEBRTXKB-UHFFFAOYSA-N	468771	US10807959, Example 40	WD repeat-containing protein 5		 64.0								US Patent		10.7270/Q26Q219X		aid1804927	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468771	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468771&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370815	441570872							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968643	Cc1cc(cc(C)n1)-c1cc(CNC2=NCCN2)cc(c1)C(=O)NCc1ccc(Cl)c(C)c1	InChI=1S/C26H28ClN5O/c1-16-8-19(4-5-24(16)27)14-30-25(33)23-12-20(15-31-26-28-6-7-29-26)11-22(13-23)21-9-17(2)32-18(3)10-21/h4-5,8-13H,6-7,14-15H2,1-3H3,(H,30,33)(H2,28,29,31)	MTLAEEOCQBVZIW-UHFFFAOYSA-N	468772	US10807959, Example 41	WD repeat-containing protein 5		<0.100								US Patent		10.7270/Q26Q219X		aid1804927	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468772	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468772&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370855	441570873							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968644	Cc1cnc(F)c(c1)-c1cc(CNC2=NCCN2)cc(c1)C(=O)NCc1ccc(Cl)c(C)c1	InChI=1S/C25H25ClFN5O/c1-15-7-21(23(27)30-12-15)19-9-18(14-32-25-28-5-6-29-25)10-20(11-19)24(33)31-13-17-3-4-22(26)16(2)8-17/h3-4,7-12H,5-6,13-14H2,1-2H3,(H,31,33)(H2,28,29,32)	GFEQQEVVCJPEQP-UHFFFAOYSA-N	468773	US10807959, Example 42	WD repeat-containing protein 5		<0.100								US Patent		10.7270/Q26Q219X		aid1804927	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468773	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468773&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370933	441570874							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981403	CCn1cc(c(n1)C(F)(F)F)-c1cc(CN2CCOC2=N)cc(c1)C(=O)N[C@@H](C1CC1)c1ccc(F)c(C)c1	InChI=1S/C28H29F4N5O2/c1-3-37-15-22(25(35-37)28(30,31)32)20-11-17(14-36-8-9-39-27(36)33)12-21(13-20)26(38)34-24(18-4-5-18)19-6-7-23(29)16(2)10-19/h6-7,10-13,15,18,24,33H,3-5,8-9,14H2,1-2H3,(H,34,38)/t24-/m0/s1	PVNNFXRYMGEMDB-DEOSSOPVSA-N	473197	US10844044, Example 276	WD repeat-containing protein 5		<0.100								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473197	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473197&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146455896	442073409							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981404	Cc1ccnc(c1)C(NC(=O)c1cc(Cn2ccn(C)c2=N)cc(c1)-c1ccc(F)nc1C)C1CC1	InChI=1S/C28H29FN6O/c1-17-8-9-31-24(12-17)26(20-4-5-20)33-27(36)22-14-19(16-35-11-10-34(3)28(35)30)13-21(15-22)23-6-7-25(29)32-18(23)2/h6-15,20,26,30H,4-5,16H2,1-3H3,(H,33,36)	RJOWQRHZMOOCGJ-UHFFFAOYSA-N	473198	US10844044, Example 3	WD repeat-containing protein 5		<0.100								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473198	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473198&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456009	442073410							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981405	Cc1cc(ccc1F)[C@@H](NC(=O)c1cc(Cn2ccn(C)c2=N)cc(c1)-c1ncnc2CCCCc12)C1CC1	InChI=1S/C31H33FN6O/c1-19-13-22(9-10-26(19)32)28(21-7-8-21)36-30(39)24-15-20(17-38-12-11-37(2)31(38)33)14-23(16-24)29-25-5-3-4-6-27(25)34-18-35-29/h9-16,18,21,28,33H,3-8,17H2,1-2H3,(H,36,39)/t28-/m0/s1	ROCUMSDYZKAHSN-NDEPHWFRSA-N	473199	US10844044, Example 94	WD repeat-containing protein 5		 36.0								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473199	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473199&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146455914	442073411							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981406	Cc1cc(ccc1F)[C@@H](NC(=O)c1cc(Cn2ccn(C)c2=N)cc(c1)-c1ccc(F)cc1C#N)C1CC1	InChI=1S/C30H27F2N5O/c1-18-11-21(5-8-27(18)32)28(20-3-4-20)35-29(38)23-13-19(17-37-10-9-36(2)30(37)34)12-22(14-23)26-7-6-25(31)15-24(26)16-33/h5-15,20,28,34H,3-4,17H2,1-2H3,(H,35,38)/t28-/m0/s1	DCRBYUPUTDSYIN-NDEPHWFRSA-N	473200	US10844044, Example 185	WD repeat-containing protein 5		<0.100								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473200	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473200&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456481	442073412							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981407	Cc1cc(F)ccc1-c1cc(Cn2ccoc2=N)cc(n1)C(=O)NCc1ccc(Cl)c(Cl)c1	InChI=1S/C24H19Cl2FN4O2/c1-14-8-17(27)3-4-18(14)21-10-16(13-31-6-7-33-24(31)28)11-22(30-21)23(32)29-12-15-2-5-19(25)20(26)9-15/h2-11,28H,12-13H2,1H3,(H,29,32)	WQEDAJCUQKKQFJ-UHFFFAOYSA-N	473201	US10844044, Example 277	WD repeat-containing protein 5		>33.0								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473201	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473201&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146455751	442073413							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981408	COc1ccnc(CNC(=O)c2cc(Cn3ccn(C)c3=N)cc(c2)-c2cc(C)cnc2OC)c1	InChI=1S/C26H28N6O3/c1-17-9-23(25(35-4)30-14-17)19-10-18(16-32-8-7-31(2)26(32)27)11-20(12-19)24(33)29-15-21-13-22(34-3)5-6-28-21/h5-14,27H,15-16H2,1-4H3,(H,29,33)	UQJAMEZWLARBAO-UHFFFAOYSA-N	473202	US10844044, Example 4	WD repeat-containing protein 5		 0.340								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473202	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473202&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456425	442073414							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981409	Cc1ccnc(c1)C(NC(=O)c1cc(Cn2ccn(C)c2=N)cc(c1)-c1ncnc2CCCCc12)C1CC1	InChI=1S/C30H33N7O/c1-19-9-10-32-26(13-19)28(21-7-8-21)35-29(38)23-15-20(17-37-12-11-36(2)30(37)31)14-22(16-23)27-24-5-3-4-6-25(24)33-18-34-27/h9-16,18,21,28,31H,3-8,17H2,1-2H3,(H,35,38)	CIRBGGNVSKVRDD-UHFFFAOYSA-N	473203	US10844044, Example 95	WD repeat-containing protein 5		 20.0								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473203	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473203&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146457146	442073415							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981410	Cn1ccn(Cc2cc(C(=O)NC3(CCC3)c3cccc(Br)c3)c(F)c(c2)-c2ccc(F)cc2C(F)(F)F)c1=N	InChI=1S/C29H24BrF5N4O/c1-38-10-11-39(27(38)36)16-17-12-22(21-7-6-20(31)15-24(21)29(33,34)35)25(32)23(13-17)26(40)37-28(8-3-9-28)18-4-2-5-19(30)14-18/h2,4-7,10-15,36H,3,8-9,16H2,1H3,(H,37,40)	WTOJAMPKAKOIJC-UHFFFAOYSA-N	473204	US10844044, Example 186	WD repeat-containing protein 5		<0.100								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473204	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473204&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146455725	442073416							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981411	CC(C)Cn1cc(c(n1)C(F)(F)F)-c1cc(CN2CCOC2=N)cc(c1)C(=O)N[C@@H](C1CC1)c1ccc(F)c(C)c1	InChI=1S/C30H33F4N5O2/c1-17(2)14-39-16-24(27(37-39)30(32,33)34)22-11-19(15-38-8-9-41-29(38)35)12-23(13-22)28(40)36-26(20-4-5-20)21-6-7-25(31)18(3)10-21/h6-7,10-13,16-17,20,26,35H,4-5,8-9,14-15H2,1-3H3,(H,36,40)/t26-/m0/s1	QHERLUOFQGCXST-SANMLTNESA-N	473205	US10844044, Example 278	WD repeat-containing protein 5		 0.340								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473205	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473205&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456151	442073417							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981412	Cc1cc(F)ccc1-c1cc(Cn2ccn(C)c2=N)cc(n1)C(=O)NCc1ccc(Cl)c(Cl)c1	InChI=1S/C25H22Cl2FN5O/c1-15-9-18(28)4-5-19(15)22-11-17(14-33-8-7-32(2)25(33)29)12-23(31-22)24(34)30-13-16-3-6-20(26)21(27)10-16/h3-12,29H,13-14H2,1-2H3,(H,30,34)	IULMWXZOYMXUER-UHFFFAOYSA-N	473206	US10844044, Example 5	WD repeat-containing protein 5		 0.350								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473206	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473206&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146457653	442073418							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981413	COc1cc(OC)cc(c1)C(NC(=O)c1cc(Cn2ccn(C)c2=N)cc(c1)-c1ncnc2CCCCc12)C1CC1	InChI=1S/C32H36N6O3/c1-37-10-11-38(32(37)33)18-20-12-22(30-27-6-4-5-7-28(27)34-19-35-30)14-24(13-20)31(39)36-29(21-8-9-21)23-15-25(40-2)17-26(16-23)41-3/h10-17,19,21,29,33H,4-9,18H2,1-3H3,(H,36,39)	LWWOVMAPSPWFBM-UHFFFAOYSA-N	473207	US10844044, Example 96	WD repeat-containing protein 5		 27.0								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473207	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473207&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456434	442073419							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981414	Cn1ccn(Cc2cc(cc(c2)-c2ncc(F)cc2C(F)(F)F)C(=O)N[C@@H](C2CC2)c2ccc(Cl)c(Cl)c2)c1=N	InChI=1S/C28H23Cl2F4N5O/c1-38-6-7-39(27(38)35)14-15-8-18(25-21(28(32,33)34)12-20(31)13-36-25)10-19(9-15)26(40)37-24(16-2-3-16)17-4-5-22(29)23(30)11-17/h4-13,16,24,35H,2-3,14H2,1H3,(H,37,40)/t24-/m0/s1	LNETWEXBHUOMLE-DEOSSOPVSA-N	473208	US10844044, Example 187	WD repeat-containing protein 5		<0.100								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473208	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473208&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146455825	442073420							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981415	Cc1cc(ccc1F)[C@@H](NC(=O)c1cc(CN2CCOC2=N)cc(c1)-c1cn(nc1C(F)(F)F)C1CCCC1)C1CC1	InChI=1S/C31H33F4N5O2/c1-18-12-21(8-9-26(18)32)27(20-6-7-20)37-29(41)23-14-19(16-39-10-11-42-30(39)36)13-22(15-23)25-17-40(24-4-2-3-5-24)38-28(25)31(33,34)35/h8-9,12-15,17,20,24,27,36H,2-7,10-11,16H2,1H3,(H,37,41)/t27-/m0/s1	WVQYTCZRTKWTFF-MHZLTWQESA-N	473209	US10844044, Example 279	WD repeat-containing protein 5		 0.610								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473209	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473209&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456136	442073421							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981416	Cc1cc(F)ccc1-c1cc(Cn2cc[nH]c2=N)cc(n1)C(=O)NCc1ccc(Cl)c(Cl)c1	InChI=1S/C24H20Cl2FN5O/c1-14-8-17(27)3-4-18(14)21-10-16(13-32-7-6-29-24(32)28)11-22(31-21)23(33)30-12-15-2-5-19(25)20(26)9-15/h2-11H,12-13H2,1H3,(H2,28,29)(H,30,33)	NYFNPKRIFORSQW-UHFFFAOYSA-N	473210	US10844044, Example 6	WD repeat-containing protein 5		 24.0								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473210	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473210&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456315	442073422							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981417	COc1ccnc(c1)[C@@H](NC(=O)c1cc(Cn2ccn(C)c2=N)cc(c1)-c1ccc(F)cc1C)C1CC1	InChI=1S/C29H30FN5O2/c1-18-12-23(30)6-7-25(18)21-13-19(17-35-11-10-34(2)29(35)31)14-22(15-21)28(36)33-27(20-4-5-20)26-16-24(37-3)8-9-32-26/h6-16,20,27,31H,4-5,17H2,1-3H3,(H,33,36)/t27-/m0/s1	JMMNYJULKRGWMJ-MHZLTWQESA-N	473211	US10844044, Example 97	WD repeat-containing protein 5		 0.140								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473211	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473211&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146455873	442073423							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981418	Cc1cc(ccc1Cl)[C@@H](NC(=O)c1cc(Cn2ccn(C)c2=N)cc(c1)-c1ccc(F)cc1C(F)(F)F)C1CC1	InChI=1S/C30H27ClF4N4O/c1-17-11-20(5-8-26(17)31)27(19-3-4-19)37-28(40)22-13-18(16-39-10-9-38(2)29(39)36)12-21(14-22)24-7-6-23(32)15-25(24)30(33,34)35/h5-15,19,27,36H,3-4,16H2,1-2H3,(H,37,40)/t27-/m0/s1	ZMNRJBOZQHXMLP-MHZLTWQESA-N	473212	US10844044, Example 188	WD repeat-containing protein 5		<0.100								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473212	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473212&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			156022868	442073424							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981419	CCn1cc(c(n1)C(F)(F)F)-c1cc(Cn2ccoc2=N)cc(c1)C(=O)N[C@@H](C1CC1)c1ccc(Cl)c(Cl)c1	InChI=1S/C27H24Cl2F3N5O2/c1-2-37-14-20(24(35-37)27(30,31)32)18-9-15(13-36-7-8-39-26(36)33)10-19(11-18)25(38)34-23(16-3-4-16)17-5-6-21(28)22(29)12-17/h5-12,14,16,23,33H,2-4,13H2,1H3,(H,34,38)/t23-/m0/s1	JCQWZMUTAHGUSH-QHCPKHFHSA-N	473213	US10844044, Example 280	WD repeat-containing protein 5		<0.100								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473213	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473213&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456528	442073425							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981420	Cc1ccnc(c1)C(NC(=O)c1cc(Cn2ccn(C)c2=N)cc(c1)-c1ccnc(C)c1)C1CC1	InChI=1S/C28H30N6O/c1-18-6-8-31-25(12-18)26(21-4-5-21)32-27(35)24-15-20(17-34-11-10-33(3)28(34)29)14-23(16-24)22-7-9-30-19(2)13-22/h6-16,21,26,29H,4-5,17H2,1-3H3,(H,32,35)	LKWYATRPXRPKLX-UHFFFAOYSA-N	473214	US10844044, Example 7	WD repeat-containing protein 5		 0.800								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473214	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473214&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146457659	442073426							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981421	COc1cc(CNC(=O)c2cc(Cn3ccn(C)c3=N)cc(c2)-c2ccc(F)cc2C(F)(F)F)cc(OC)c1	InChI=1S/C28H26F4N4O3/c1-35-6-7-36(27(35)33)16-18-8-19(24-5-4-21(29)13-25(24)28(30,31)32)12-20(9-18)26(37)34-15-17-10-22(38-2)14-23(11-17)39-3/h4-14,33H,15-16H2,1-3H3,(H,34,37)	MXDHGDCQJNHCSE-UHFFFAOYSA-N	473215	US10844044, Example 98	WD repeat-containing protein 5		 0.060								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473215	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473215&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146455726	442073427							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981422	Cn1ccn(Cc2cc(cc(c2)-c2cccnc2C(F)(F)F)C(=O)N[C@@H](C2CC2)c2ccc(F)c(F)c2)c1=N	InChI=1S/C28H24F5N5O/c1-37-9-10-38(27(37)34)15-16-11-19(21-3-2-8-35-25(21)28(31,32)33)13-20(12-16)26(39)36-24(17-4-5-17)18-6-7-22(29)23(30)14-18/h2-3,6-14,17,24,34H,4-5,15H2,1H3,(H,36,39)/t24-/m0/s1	OSHRJYIRFVOIFJ-DEOSSOPVSA-N	473216	US10844044, Example 189	WD repeat-containing protein 5		<0.100								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473216	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473216&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456438	442073428							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981423	CCn1cc(c(n1)C(F)(F)F)-c1cc(CN2CCOC2=N)cc(c1)C(=O)N[C@@H](C1CC1)c1ccc(Cl)c(Cl)c1	InChI=1S/C27H26Cl2F3N5O2/c1-2-37-14-20(24(35-37)27(30,31)32)18-9-15(13-36-7-8-39-26(36)33)10-19(11-18)25(38)34-23(16-3-4-16)17-5-6-21(28)22(29)12-17/h5-6,9-12,14,16,23,33H,2-4,7-8,13H2,1H3,(H,34,38)/t23-/m0/s1	CJDYDKVPBAKDDE-QHCPKHFHSA-N	473217	US10844044, Example 281	WD repeat-containing protein 5		<0.100								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473217	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473217&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146455967	442073429							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981424	COc1ccnc(CNC(=O)c2cc(Cn3ccn(C)c3=N)cc(c2)-c2ccncc2C)c1	InChI=1S/C25H26N6O2/c1-17-14-27-6-5-23(17)19-10-18(16-31-9-8-30(2)25(31)26)11-20(12-19)24(32)29-15-21-13-22(33-3)4-7-28-21/h4-14,26H,15-16H2,1-3H3,(H,29,32)	PZTYPVIWASSISH-UHFFFAOYSA-N	473218	US10844044, Example 8	WD repeat-containing protein 5		 0.270								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473218	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473218&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456249	442073430							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981425	Cc1cc(CNC(=O)c2cc(Cn3ccn(C)c3=N)cc(n2)-c2ccc(F)cc2C(F)(F)F)ccc1Cl	InChI=1S/C26H22ClF4N5O/c1-15-9-16(3-6-21(15)27)13-33-24(37)23-11-17(14-36-8-7-35(2)25(36)32)10-22(34-23)19-5-4-18(28)12-20(19)26(29,30)31/h3-12,32H,13-14H2,1-2H3,(H,33,37)	LRAGULFZSGHIIL-UHFFFAOYSA-N	473219	US10844044, Example 99	WD repeat-containing protein 5		 1.10								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473219	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473219&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456140	442073431							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981426	CCn1cc(c(n1)C(F)(F)F)-c1cc(Cn2ccn(C3CC3)c2=N)cc(c1)C(=O)N[C@@H](C1CC1)c1ccc(F)c(F)c1	InChI=1S/C30H29F5N6O/c1-2-40-16-23(27(38-40)30(33,34)35)20-11-17(15-39-9-10-41(29(39)36)22-6-7-22)12-21(13-20)28(42)37-26(18-3-4-18)19-5-8-24(31)25(32)14-19/h5,8-14,16,18,22,26,36H,2-4,6-7,15H2,1H3,(H,37,42)/t26-/m0/s1	DZSWVPKGQBEOTE-SANMLTNESA-N	473220	US10844044, Example 190	WD repeat-containing protein 5		 0.110								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473220	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473220&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146455993	442073432							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981427	Cc1cc(ccc1F)[C@@H](NC(=O)c1cc(CN2CCOC2=N)cc(c1)-c1ccc(F)cc1C#N)C1CC1	InChI=1S/C29H26F2N4O2/c1-17-10-20(4-7-26(17)31)27(19-2-3-19)34-28(36)22-12-18(16-35-8-9-37-29(35)33)11-21(13-22)25-6-5-24(30)14-23(25)15-32/h4-7,10-14,19,27,33H,2-3,8-9,16H2,1H3,(H,34,36)/t27-/m0/s1	WBIFECZYYGBSBP-MHZLTWQESA-N	473221	US10844044, Example 282	WD repeat-containing protein 5		 0.210								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473221	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473221&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456581	442073433							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981428	Cc1ccnc(c1)C(NC(=O)c1cc(Cn2ccn(C)c2=N)cc(c1)-c1ccc(F)cc1C)C1CC1	InChI=1S/C29H30FN5O/c1-18-8-9-32-26(12-18)27(21-4-5-21)33-28(36)23-15-20(17-35-11-10-34(3)29(35)31)14-22(16-23)25-7-6-24(30)13-19(25)2/h6-16,21,27,31H,4-5,17H2,1-3H3,(H,33,36)	SSPGQCWIFWWIMQ-UHFFFAOYSA-N	473222	US10844044, Example 9	WD repeat-containing protein 5		 0.150								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473222	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473222&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456308	442073434							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981429	COc1cc(CNC(=O)c2cc(Cn3ccn(C)c3=N)cc(n2)-c2ccc(F)cc2C(F)(F)F)cc(OC)c1	InChI=1S/C27H25F4N5O3/c1-35-6-7-36(26(35)32)15-17-10-23(21-5-4-18(28)12-22(21)27(29,30)31)34-24(11-17)25(37)33-14-16-8-19(38-2)13-20(9-16)39-3/h4-13,32H,14-15H2,1-3H3,(H,33,37)	COGIPINVIFHQQN-UHFFFAOYSA-N	473223	US10844044, Example 100	WD repeat-containing protein 5		 0.710								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473223	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473223&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456299	442073435							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981430	CCn1cc(c(n1)C(F)(F)F)-c1cc(Cn2ccn(C)c2=N)cc(c1)C(=O)N[C@@H](C1CC1)c1ccc(F)c(F)c1	InChI=1S/C28H27F5N6O/c1-3-39-15-21(25(36-39)28(31,32)33)19-10-16(14-38-9-8-37(2)27(38)34)11-20(12-19)26(40)35-24(17-4-5-17)18-6-7-22(29)23(30)13-18/h6-13,15,17,24,34H,3-5,14H2,1-2H3,(H,35,40)/t24-/m0/s1	UGYLPQAQOHYWFG-DEOSSOPVSA-N	473224	US10844044, Example 191::US10844044, Example 213	WD repeat-containing protein 5		<0.100								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473224	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473224&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146455858	442073436							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981431	Cc1cc(ccc1F)[C@@H](NC(=O)c1cc(CN2CCOC2=N)cc(c1F)-c1ccc(F)cc1C(F)(F)F)C1CC1	InChI=1S/C29H25F6N3O2/c1-15-10-18(4-7-24(15)31)26(17-2-3-17)37-27(39)22-12-16(14-38-8-9-40-28(38)36)11-21(25(22)32)20-6-5-19(30)13-23(20)29(33,34)35/h4-7,10-13,17,26,36H,2-3,8-9,14H2,1H3,(H,37,39)/t26-/m0/s1	IPKRPNNLBJEMGE-SANMLTNESA-N	473225	US10844044, Example 283	WD repeat-containing protein 5		 0.020								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473225	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473225&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456761	442073437							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981432	COc1ccnc(CNC(=O)c2cc(Cn3ccn(C)c3=N)cc(c2)-c2cc(C)ccc2OC)c1	InChI=1S/C27H29N5O3/c1-18-5-6-25(35-4)24(11-18)20-12-19(17-32-10-9-31(2)27(32)28)13-21(14-20)26(33)30-16-22-15-23(34-3)7-8-29-22/h5-15,28H,16-17H2,1-4H3,(H,30,33)	ARKKNNQSXXBYTE-UHFFFAOYSA-N	473226	US10844044, Example 10	WD repeat-containing protein 5		 1.50								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473226	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473226&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456070	442073438							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981433	Cc1ccnc(c1)C(NC(=O)c1cc(Cn2ccn(C)c2=N)cc(n1)-c1ccc(F)cc1C(F)(F)F)C1CC1	InChI=1S/C28H26F4N6O/c1-16-7-8-34-23(11-16)25(18-3-4-18)36-26(39)24-13-17(15-38-10-9-37(2)27(38)33)12-22(35-24)20-6-5-19(29)14-21(20)28(30,31)32/h5-14,18,25,33H,3-4,15H2,1-2H3,(H,36,39)	UBHBQORFVWTUQH-UHFFFAOYSA-N	473227	US10844044, Example 101	WD repeat-containing protein 5		 0.450								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473227	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473227&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146455715	442073439							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981434	Cc1cc(ccc1F)[C@@H](NC(=O)c1cc(Cn2ccn(C)c2=N)cc(c1)C(=C)C(F)(F)F)C1CC1	InChI=1S/C26H26F4N4O/c1-15-10-19(6-7-22(15)27)23(18-4-5-18)32-24(35)21-12-17(14-34-9-8-33(3)25(34)31)11-20(13-21)16(2)26(28,29)30/h6-13,18,23,31H,2,4-5,14H2,1,3H3,(H,32,35)/t23-/m0/s1	LHVFUUZUTHIXDT-QHCPKHFHSA-N	473228	US10844044, Example 192	WD repeat-containing protein 5		<0.100								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473228	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473228&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146488027	442073440							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981435	Fc1cnc(-c2cc(CN3CCOC3=N)cc(c2)C(=O)N[C@@H](C2CC2)c2ccc(Cl)c(Cl)c2)c(c1)C(F)(F)F	InChI=1S/C27H22Cl2F4N4O2/c28-21-4-3-16(10-22(21)29)23(15-1-2-15)36-25(38)18-8-14(13-37-5-6-39-26(37)34)7-17(9-18)24-20(27(31,32)33)11-19(30)12-35-24/h3-4,7-12,15,23,34H,1-2,5-6,13H2,(H,36,38)/t23-/m0/s1	OYTFOLLSXPJVLL-QHCPKHFHSA-N	473229	US10844044, Example 284	WD repeat-containing protein 5		 0.110								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473229	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473229&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456324	442073441							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981436	Cc1ccnc(c1)C(NC(=O)c1cc(Cn2ccn(C)c2=N)cc(c1)-c1cccn1C)C1CC1	InChI=1S/C27H30N6O/c1-18-8-9-29-23(13-18)25(20-6-7-20)30-26(34)22-15-19(17-33-12-11-32(3)27(33)28)14-21(16-22)24-5-4-10-31(24)2/h4-5,8-16,20,25,28H,6-7,17H2,1-3H3,(H,30,34)	NLNNPCRHBAGSIB-UHFFFAOYSA-N	473230	US10844044, Example 11	WD repeat-containing protein 5		 0.830								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473230	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473230&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456702	442073442							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981437	CC(C)n1nccc1-c1cc(Cn2ccn(C)c2=N)cc(c1)C(=O)N[C@@H](C1CC1)c1ccc(F)c(C)c1	InChI=1S/C29H33FN6O/c1-18(2)36-26(9-10-32-36)23-14-20(17-35-12-11-34(4)29(35)31)15-24(16-23)28(37)33-27(21-5-6-21)22-7-8-25(30)19(3)13-22/h7-16,18,21,27,31H,5-6,17H2,1-4H3,(H,33,37)/t27-/m0/s1	DHSTYPXBBFXIMB-MHZLTWQESA-N	473231	US10844044, Example 102	WD repeat-containing protein 5		 0.320								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473231	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473231&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456214	442073443							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981438	CC(C)n1cc(c(n1)C(F)(F)F)-c1cc(Cn2ccn(C)c2=N)cc(c1)C(=O)N[C@@H](C1CC1)c1ccc(F)c(C)c1	InChI=1S/C30H32F4N6O/c1-17(2)40-16-24(27(37-40)30(32,33)34)22-12-19(15-39-10-9-38(4)29(39)35)13-23(14-22)28(41)36-26(20-5-6-20)21-7-8-25(31)18(3)11-21/h7-14,16-17,20,26,35H,5-6,15H2,1-4H3,(H,36,41)/t26-/m0/s1	RESJAEHDHNZHSW-SANMLTNESA-N	473232	US10844044, Example 193	WD repeat-containing protein 5		<0.100								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473232	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473232&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146457004	442073444							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981439	Cc1cc(ccc1F)[C@@H](NC(=O)c1cc(CN2CCOC2=N)cc(c1)-c1ccc(F)cc1C(F)(F)F)C1CC1	InChI=1S/C29H26F5N3O2/c1-16-10-19(4-7-25(16)31)26(18-2-3-18)36-27(38)21-12-17(15-37-8-9-39-28(37)35)11-20(13-21)23-6-5-22(30)14-24(23)29(32,33)34/h4-7,10-14,18,26,35H,2-3,8-9,15H2,1H3,(H,36,38)/t26-/m0/s1	CXMXPUXGUCTVDZ-SANMLTNESA-N	473233	US10844044, Example 285	WD repeat-containing protein 5		<0.100								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473233	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473233&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456355	442073445							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981440	Cc1ccnc(c1)C(NC(=O)c1cc(Cn2ccn(C)c2=N)cc(c1)-c1ccnn1C)C1CC1	InChI=1S/C26H29N7O/c1-17-6-8-28-22(12-17)24(19-4-5-19)30-25(34)21-14-18(16-33-11-10-31(2)26(33)27)13-20(15-21)23-7-9-29-32(23)3/h6-15,19,24,27H,4-5,16H2,1-3H3,(H,30,34)	YDSAEZVRMMNABM-UHFFFAOYSA-N	473234	US10844044, Example 12	WD repeat-containing protein 5		 1.20								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473234	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473234&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456568	442073446							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981441	CC(C)n1nccc1-c1cc(Cn2ccn(C)c2=N)cc(c1)C(=O)N[C@H](C1CC1)c1cc(C)ccn1	InChI=1S/C28H33N7O/c1-18(2)35-25(8-10-31-35)22-14-20(17-34-12-11-33(4)28(34)29)15-23(16-22)27(36)32-26(21-5-6-21)24-13-19(3)7-9-30-24/h7-16,18,21,26,29H,5-6,17H2,1-4H3,(H,32,36)/t26-/m1/s1	FBGLJMUXIXSIRI-AREMUKBSSA-N	473235	US10844044, Example 103	WD repeat-containing protein 5		 20.0								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473235	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473235&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456286	442073447							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981442	CC(C)n1cc(c(n1)C(F)(F)F)-c1cc(Cn2ccn(C3CC3)c2=N)cc(c1)C(=O)N[C@@H](C1CC1)c1ccc(F)c(C)c1	InChI=1S/C32H34F4N6O/c1-18(2)42-17-26(29(39-42)32(34,35)36)23-13-20(16-40-10-11-41(31(40)37)25-7-8-25)14-24(15-23)30(43)38-28(21-4-5-21)22-6-9-27(33)19(3)12-22/h6,9-15,17-18,21,25,28,37H,4-5,7-8,16H2,1-3H3,(H,38,43)/t28-/m0/s1	FYYHMKSDLAROMQ-NDEPHWFRSA-N	473236	US10844044, Example 194	WD repeat-containing protein 5		<0.100								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473236	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473236&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456364	442073448							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981443	CC(C)n1cc(c(n1)C(F)(F)F)-c1cc(CN2CCOC2=N)cc(c1)C(=O)N[C@@H](C1CC1)c1ccc(F)c(F)c1	InChI=1S/C28H28F5N5O2/c1-15(2)38-14-21(25(36-38)28(31,32)33)19-9-16(13-37-7-8-40-27(37)34)10-20(11-19)26(39)35-24(17-3-4-17)18-5-6-22(29)23(30)12-18/h5-6,9-12,14-15,17,24,34H,3-4,7-8,13H2,1-2H3,(H,35,39)/t24-/m0/s1	CPONQUAVFCMICY-DEOSSOPVSA-N	473237	US10844044, Example 286	WD repeat-containing protein 5		<0.100								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473237	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473237&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456033	442073449							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981444	COc1cnccc1-c1cc(Cn2ccn(C)c2=N)cc(c1)C(=O)NC(C1CC1)c1cc(C)ccn1	InChI=1S/C28H30N6O2/c1-18-6-9-31-24(12-18)26(20-4-5-20)32-27(35)22-14-19(17-34-11-10-33(2)28(34)29)13-21(15-22)23-7-8-30-16-25(23)36-3/h6-16,20,26,29H,4-5,17H2,1-3H3,(H,32,35)	MUVXQFKSYTTWTQ-UHFFFAOYSA-N	473239	US10844044, Example 13	WD repeat-containing protein 5		 2.70								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473239	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473239&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146455893	442073451							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981445	Cn1ccn(Cc2cc(nc(c2)-c2ccc(F)cc2C(F)(F)F)C(=O)NC(CC(O)=O)c2ccc(Cl)c(Cl)c2)c1=N	InChI=1S/C27H21Cl2F4N5O3/c1-37-6-7-38(26(37)34)13-14-8-22(17-4-3-16(30)11-18(17)27(31,32)33)35-23(9-14)25(41)36-21(12-24(39)40)15-2-5-19(28)20(29)10-15/h2-11,21,34H,12-13H2,1H3,(H,36,41)(H,39,40)	UZNDCISOOMRVTD-UHFFFAOYSA-N	473240	US10844044, Example 104	WD repeat-containing protein 5		 0.130								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473240	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473240&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456027	442073452							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981446	CC(c1cc(Cn2ccn(C)c2=N)cc(c1)C(=O)N[C@@H](C1CC1)c1ccc(F)c(C)c1)C(F)(F)F	InChI=1S/C26H28F4N4O/c1-15-10-19(6-7-22(15)27)23(18-4-5-18)32-24(35)21-12-17(14-34-9-8-33(3)25(34)31)11-20(13-21)16(2)26(28,29)30/h6-13,16,18,23,31H,4-5,14H2,1-3H3,(H,32,35)/t16?,23-/m0/s1	XEICHAIGVISICF-KESSSICBSA-N	473241	US10844044, Example 195	WD repeat-containing protein 5		<0.100								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473241	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473241&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456077	442073453							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981447	Cc1cc(ccc1F)[C@@H](NC(=O)c1cc(CN2CCOC2=N)cc(c1)-c1cc(nn1C)C(F)(F)F)C1CC1	InChI=1S/C27H27F4N5O2/c1-15-9-18(5-6-21(15)28)24(17-3-4-17)33-25(37)20-11-16(14-36-7-8-38-26(36)32)10-19(12-20)22-13-23(27(29,30)31)34-35(22)2/h5-6,9-13,17,24,32H,3-4,7-8,14H2,1-2H3,(H,33,37)/t24-/m0/s1	WBUIWRBVNKBOMH-DEOSSOPVSA-N	473242	US10844044, Example 287	WD repeat-containing protein 5		<0.100								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473242	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473242&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456005	442073454							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981448	COc1cc(ccn1)-c1cc(Cn2ccn(C)c2=N)cc(c1)C(=O)NC(C1CC1)c1cc(C)ccn1	InChI=1S/C28H30N6O2/c1-18-6-8-30-24(12-18)26(20-4-5-20)32-27(35)23-14-19(17-34-11-10-33(2)28(34)29)13-22(15-23)21-7-9-31-25(16-21)36-3/h6-16,20,26,29H,4-5,17H2,1-3H3,(H,32,35)	JZYBZUBBUVTZNM-UHFFFAOYSA-N	473243	US10844044, Example 14	WD repeat-containing protein 5		 6.00								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473243	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473243&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146457312	442073455							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981449	Cc1ccnc(c1)C(NC(=O)c1cc(Cn2ccn(C)c2=N)cc(c1F)-c1ccc(F)cc1C(F)(F)F)C1CC1	InChI=1S/C29H26F5N5O/c1-16-7-8-36-24(11-16)26(18-3-4-18)37-27(40)22-13-17(15-39-10-9-38(2)28(39)35)12-21(25(22)31)20-6-5-19(30)14-23(20)29(32,33)34/h5-14,18,26,35H,3-4,15H2,1-2H3,(H,37,40)	XMSBMGGMBZIKEW-UHFFFAOYSA-N	473244	US10844044, Example 105	WD repeat-containing protein 5		<0.100								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473244	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473244&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146455703	442073456							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981450	Cc1cc(ccc1F)[C@@H](NC(=O)c1cc(Cn2ccn(C)c2=N)cc(c1)-c1cc(nn1C)C(F)(F)F)C1CC1	InChI=1S/C28H28F4N6O/c1-16-10-19(6-7-22(16)29)25(18-4-5-18)34-26(39)21-12-17(15-38-9-8-36(2)27(38)33)11-20(13-21)23-14-24(28(30,31)32)35-37(23)3/h6-14,18,25,33H,4-5,15H2,1-3H3,(H,34,39)/t25-/m0/s1	GAXRSNWHWVTFNR-VWLOTQADSA-N	473245	US10844044, Example 196	WD repeat-containing protein 5		<0.100								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473245	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473245&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456153	442073457							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981451	CCn1cc(c(n1)C(F)(F)F)-c1cc(CN2CCOC2=N)cc(c1)C(=O)NCC1CCOCC1	InChI=1S/C23H28F3N5O3/c1-2-31-14-19(20(29-31)23(24,25)26)17-9-16(13-30-5-8-34-22(30)27)10-18(11-17)21(32)28-12-15-3-6-33-7-4-15/h9-11,14-15,27H,2-8,12-13H2,1H3,(H,28,32)	WPHSKEQIKCATRH-UHFFFAOYSA-N	473246	US10844044, Example 288	WD repeat-containing protein 5		 8.70								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473246	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473246&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146455883	442073458							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981452	Cc1ccnc(c1)C(NC(=O)c1cc(Cn2ccn(C)c2=N)cc(c1)-c1cnccc1C)C1CC1	InChI=1S/C28H30N6O/c1-18-6-9-31-25(12-18)26(21-4-5-21)32-27(35)23-14-20(17-34-11-10-33(3)28(34)29)13-22(15-23)24-16-30-8-7-19(24)2/h6-16,21,26,29H,4-5,17H2,1-3H3,(H,32,35)	QKSQBZZZBZBSAF-UHFFFAOYSA-N	473247	US10844044, Example 15	WD repeat-containing protein 5		 2.70								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473247	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473247&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146457015	442073459							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981453	COC(=O)CC(NC(=O)c1cc(Cn2ccn(C)c2=N)cc(n1)-c1ccc(F)cc1C(F)(F)F)c1ccc(Cl)c(Cl)c1	InChI=1S/C28H23Cl2F4N5O3/c1-38-7-8-39(27(38)35)14-15-9-23(18-5-4-17(31)12-19(18)28(32,33)34)36-24(10-15)26(41)37-22(13-25(40)42-2)16-3-6-20(29)21(30)11-16/h3-12,22,35H,13-14H2,1-2H3,(H,37,41)	HFVBGMFXLNTJIC-UHFFFAOYSA-N	473248	US10844044, Example 106	WD repeat-containing protein 5		 0.340								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473248	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473248&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146457559	442073460							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981454	CCn1cc(c(n1)C(F)(F)F)-c1cc(Cn2ccn(C3CC3)c2=N)cc(c1)C(=O)NCc1ccc(F)c(C)c1	InChI=1S/C28H28F4N6O/c1-3-37-16-23(25(35-37)28(30,31)32)20-11-19(15-36-8-9-38(27(36)33)22-5-6-22)12-21(13-20)26(39)34-14-18-4-7-24(29)17(2)10-18/h4,7-13,16,22,33H,3,5-6,14-15H2,1-2H3,(H,34,39)	JDDQROKCFHICFG-UHFFFAOYSA-N	473249	US10844044, Example 197	WD repeat-containing protein 5		<0.100								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473249	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473249&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146455700	442073461							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981455	CCn1cc(c(n1)C(F)(F)F)-c1cc(CN2CCOC2=N)cc(c1)C(=O)NCC1CCCO1	InChI=1S/C22H26F3N5O3/c1-2-30-13-18(19(28-30)22(23,24)25)15-8-14(12-29-5-7-33-21(29)26)9-16(10-15)20(31)27-11-17-4-3-6-32-17/h8-10,13,17,26H,2-7,11-12H2,1H3,(H,27,31)	XNZLNPLIUJBCMN-UHFFFAOYSA-N	473250	US10844044, Example 289	WD repeat-containing protein 5		 31.0								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473250	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473250&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146455943	442073462							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981456	Cc1cc(CNC(=O)c2cc(Cn3ccn(C)c3=N)cc(c2)-c2ccncc2C)ccc1Cl	InChI=1S/C26H26ClN5O/c1-17-10-19(4-5-24(17)27)15-30-25(33)22-12-20(16-32-9-8-31(3)26(32)28)11-21(13-22)23-6-7-29-14-18(23)2/h4-14,28H,15-16H2,1-3H3,(H,30,33)	RTXXOMJYDBCZNP-UHFFFAOYSA-N	473251	US10844044, Example 16	WD repeat-containing protein 5		 0.490								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473251	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473251&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456004	442073463							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981457	Cc1cc(ccc1F)[C@@H](NC(=O)c1cc(Cn2ccn(C)c2=N)cc(n1)-c1ccc(F)cc1C(F)(F)F)C1CC1	InChI=1S/C29H26F5N5O/c1-16-11-19(5-8-23(16)31)26(18-3-4-18)37-27(40)25-13-17(15-39-10-9-38(2)28(39)35)12-24(36-25)21-7-6-20(30)14-22(21)29(32,33)34/h5-14,18,26,35H,3-4,15H2,1-2H3,(H,37,40)/t26-/m0/s1	AKKWACFBGWEIPJ-SANMLTNESA-N	473252	US10844044, Example 107	WD repeat-containing protein 5		 0.230								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473252	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473252&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456190	442073464							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981458	CCn1cc(c(n1)C(F)(F)F)-c1cc(Cn2ccn(C)c2=N)cc(c1)C(=O)NCc1ccc(F)c(C)c1	InChI=1S/C26H26F4N6O/c1-4-36-15-21(23(33-36)26(28,29)30)19-10-18(14-35-8-7-34(3)25(35)31)11-20(12-19)24(37)32-13-17-5-6-22(27)16(2)9-17/h5-12,15,31H,4,13-14H2,1-3H3,(H,32,37)	CKCSDCHTLXSCGT-UHFFFAOYSA-N	473253	US10844044, Example 198	WD repeat-containing protein 5		<0.100								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473253	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473253&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456423	442073465							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968645	CN1CC(=O)N=C1NCc1cc(cc(c1)-c1ccc(F)nc1C)C(=O)NCc1ccc(Cl)c(Cl)c1	InChI=1S/C25H22Cl2FN5O2/c1-14-19(4-6-22(28)31-14)17-7-16(12-30-25-32-23(34)13-33(25)2)8-18(10-17)24(35)29-11-15-3-5-20(26)21(27)9-15/h3-10H,11-13H2,1-2H3,(H,29,35)(H,30,32,34)	RCKPPIBTKTTWGZ-UHFFFAOYSA-N	468774	US10807959, Example 43	WD repeat-containing protein 5		 15.0								US Patent		10.7270/Q26Q219X		aid1804927	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468774	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468774&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370887	441570875							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968646	COc1cc(OC)cc(c1)C(C)NC(=O)c1cc(CNC2=NC(=O)CN2C)cc(c1)-c1ccc(F)nc1C	InChI=1S/C28H30FN5O4/c1-16(19-11-22(37-4)13-23(12-19)38-5)32-27(36)21-9-18(14-30-28-33-26(35)15-34(28)3)8-20(10-21)24-6-7-25(29)31-17(24)2/h6-13,16H,14-15H2,1-5H3,(H,32,36)(H,30,33,35)	ZRRQDAYFOPNWOA-UHFFFAOYSA-N	468775	US10807959, Example 44	WD repeat-containing protein 5		 17.0								US Patent		10.7270/Q26Q219X		aid1804927	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468775	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468775&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370836	441570876							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968647	COc1ccnc(CNC(=O)c2cc(CNC3=NCCN3)cc(c2)-c2cc(ccc2OC)C(C)C)c1	InChI=1S/C28H33N5O3/c1-18(2)20-5-6-26(36-4)25(14-20)21-11-19(16-33-28-30-9-10-31-28)12-22(13-21)27(34)32-17-23-15-24(35-3)7-8-29-23/h5-8,11-15,18H,9-10,16-17H2,1-4H3,(H,32,34)(H2,30,31,33)	QIYWWOLIQXKWRO-UHFFFAOYSA-N	468776	US10807959, Example 45	WD repeat-containing protein 5		 1.01								US Patent		10.7270/Q26Q219X		aid1804927	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468776	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468776&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370720	441570877							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968648	COc1ccnc(CNC(=O)c2cc(CNC3=NCCN3)cc(c2)-c2cc(cnc2OC)C(F)(F)F)c1	InChI=1S/C25H25F3N6O3/c1-36-20-3-4-29-19(11-20)14-32-22(35)17-8-15(12-34-24-30-5-6-31-24)7-16(9-17)21-10-18(25(26,27)28)13-33-23(21)37-2/h3-4,7-11,13H,5-6,12,14H2,1-2H3,(H,32,35)(H2,30,31,34)	YYEYETLLKOSKFX-UHFFFAOYSA-N	468777	US10807959, Example 46	WD repeat-containing protein 5		 0.100								US Patent		10.7270/Q26Q219X		aid1804927	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468777	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468777&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370721	441570878							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968649	COc1ccnc(CNC(=O)c2cc(CNC3=NCCN3)cc(c2)-c2ccc(F)cc2C(F)(F)F)c1	InChI=1S/C25H23F4N5O2/c1-36-20-4-5-30-19(12-20)14-33-23(35)17-9-15(13-34-24-31-6-7-32-24)8-16(10-17)21-3-2-18(26)11-22(21)25(27,28)29/h2-5,8-12H,6-7,13-14H2,1H3,(H,33,35)(H2,31,32,34)	SKZIHBXXYAQMOA-UHFFFAOYSA-N	468778	US10807959, Example 47	WD repeat-containing protein 5		<0.100								US Patent		10.7270/Q26Q219X		aid1804927	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468778	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468778&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370777	441570879							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968650	COc1ccnc(CNC(=O)c2cc(CNC3=NCCN3)cc(c2)-c2cc(F)cnc2OC)c1	InChI=1S/C24H25FN6O3/c1-33-20-3-4-26-19(11-20)14-29-22(32)17-8-15(12-31-24-27-5-6-28-24)7-16(9-17)21-10-18(25)13-30-23(21)34-2/h3-4,7-11,13H,5-6,12,14H2,1-2H3,(H,29,32)(H2,27,28,31)	QHZBQAIIJUWKAB-UHFFFAOYSA-N	468779	US10807959, Example 48	WD repeat-containing protein 5		 0.630								US Patent		10.7270/Q26Q219X		aid1804927	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468779	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468779&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370761	441570880							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968651	COc1ccnc(CNC(=O)c2cc(CNC3=NCCN3)cc(c2)-c2ccc(F)cc2OC)c1	InChI=1S/C25H26FN5O3/c1-33-21-5-6-27-20(13-21)15-30-24(32)18-10-16(14-31-25-28-7-8-29-25)9-17(11-18)22-4-3-19(26)12-23(22)34-2/h3-6,9-13H,7-8,14-15H2,1-2H3,(H,30,32)(H2,28,29,31)	UYQBHFQYLCIJRJ-UHFFFAOYSA-N	468780	US10807959, Example 49	WD repeat-containing protein 5		 0.300								US Patent		10.7270/Q26Q219X		aid1804927	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468780	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468780&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146371094	441570881							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968652	COc1ccnc(CNC(=O)c2cc(CNC3=NCCN3)cc(c2)-c2cc(C)c(F)cc2OC)c1	InChI=1S/C26H28FN5O3/c1-16-8-22(24(35-3)13-23(16)27)18-9-17(14-32-26-29-6-7-30-26)10-19(11-18)25(33)31-15-20-12-21(34-2)4-5-28-20/h4-5,8-13H,6-7,14-15H2,1-3H3,(H,31,33)(H2,29,30,32)	WWCQDRCTKNPKTR-UHFFFAOYSA-N	468781	US10807959, Example 50	WD repeat-containing protein 5		<0.100								US Patent		10.7270/Q26Q219X		aid1804927	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468781	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468781&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370718	441570882							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968653	COc1ccnc(CNC(=O)c2cc(CNC3=NCCN3)cc(c2)-c2cc(C)c(F)cc2C)c1	InChI=1S/C26H28FN5O2/c1-16-9-24(27)17(2)8-23(16)19-10-18(14-32-26-29-6-7-30-26)11-20(12-19)25(33)31-15-21-13-22(34-3)4-5-28-21/h4-5,8-13H,6-7,14-15H2,1-3H3,(H,31,33)(H2,29,30,32)	NYVNYZIFEMAPEX-UHFFFAOYSA-N	468782	US10807959, Example 51	WD repeat-containing protein 5		<0.100								US Patent		10.7270/Q26Q219X		aid1804927	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468782	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468782&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370797	441570883							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968654	COc1ccnc(CNC(=O)c2cc(CNC3=NCCC3)cc(c2)-c2ccc(F)nc2C)c1	InChI=1S/C25H26FN5O2/c1-16-22(5-6-23(26)31-16)18-10-17(14-29-24-4-3-8-28-24)11-19(12-18)25(32)30-15-20-13-21(33-2)7-9-27-20/h5-7,9-13H,3-4,8,14-15H2,1-2H3,(H,28,29)(H,30,32)	LJVLMQXCMQJBFX-UHFFFAOYSA-N	468783	US10807959, Example 53	WD repeat-containing protein 5		 0.530								US Patent		10.7270/Q26Q219X		aid1804927	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468783	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468783&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370819	441570884							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968655	CC(NC(=O)c1cc(CNC2=NCCC2)cc(c1)-c1ccc(F)nc1C)c1cc(C)c(Cl)cn1	InChI=1S/C26H27ClFN5O/c1-15-9-23(30-14-22(15)27)17(3)33-26(34)20-11-18(13-31-25-5-4-8-29-25)10-19(12-20)21-6-7-24(28)32-16(21)2/h6-7,9-12,14,17H,4-5,8,13H2,1-3H3,(H,29,31)(H,33,34)	PYLZSMLKKINSES-UHFFFAOYSA-N	468784	US10807959, Example 54	WD repeat-containing protein 5		 0.310								US Patent		10.7270/Q26Q219X		aid1804927	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468784	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468784&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370800	441570885							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968656	COc1cc(OC)cc(c1)C(C)NC(=O)c1cc(CNC2=NCCC2)cc(c1)-c1ccc(F)nc1C	InChI=1S/C28H31FN4O3/c1-17(20-13-23(35-3)15-24(14-20)36-4)33-28(34)22-11-19(16-31-27-6-5-9-30-27)10-21(12-22)25-7-8-26(29)32-18(25)2/h7-8,10-15,17H,5-6,9,16H2,1-4H3,(H,30,31)(H,33,34)	WZAJNJLKABFEPO-UHFFFAOYSA-N	468785	US10807959, Example 55	WD repeat-containing protein 5		 11.0								US Patent		10.7270/Q26Q219X		aid1804927	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468785	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468785&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370993	441570886							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968657	COc1cc(CN(C)C(=O)c2cc(CNC3=NCCC3)cc(c2)-c2ccc(F)nc2C)cc(OC)c1	InChI=1S/C28H31FN4O3/c1-18-25(7-8-26(29)32-18)21-10-19(16-31-27-6-5-9-30-27)11-22(14-21)28(34)33(2)17-20-12-23(35-3)15-24(13-20)36-4/h7-8,10-15H,5-6,9,16-17H2,1-4H3,(H,30,31)	OERHWRNHHWPRIC-UHFFFAOYSA-N	468786	US10807959, Example 56	WD repeat-containing protein 5		 20.0								US Patent		10.7270/Q26Q219X		aid1804927	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468786	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468786&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370944	441570887							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968658	COc1cc(CNC(=O)c2cc(CNC3=NCCC3)cc(c2)-c2ccnc(C)c2)cc(OC)c1	InChI=1S/C27H30N4O3/c1-18-9-21(6-8-28-18)22-10-19(16-30-26-5-4-7-29-26)11-23(14-22)27(32)31-17-20-12-24(33-2)15-25(13-20)34-3/h6,8-15H,4-5,7,16-17H2,1-3H3,(H,29,30)(H,31,32)	MUPCTRAMZAOVFP-UHFFFAOYSA-N	468787	US10807959, Example 57	WD repeat-containing protein 5		 3.00								US Patent		10.7270/Q26Q219X		aid1804927	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468787	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468787&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370814	441570888							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968659	COc1cc(CNC(=O)c2cc(CNC3=NCCC3)cc(c2)-c2cccn2C)cc(OC)c1	InChI=1S/C26H30N4O3/c1-30-9-5-6-24(30)20-10-18(16-28-25-7-4-8-27-25)11-21(14-20)26(31)29-17-19-12-22(32-2)15-23(13-19)33-3/h5-6,9-15H,4,7-8,16-17H2,1-3H3,(H,27,28)(H,29,31)	GRANRZVBEVTVGZ-UHFFFAOYSA-N	468788	US10807959, Example 58	WD repeat-containing protein 5		 5.80								US Patent		10.7270/Q26Q219X		aid1804927	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468788	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468788&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370790	441570889							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968660	COc1cc(CNC(=O)c2cc(CNC3=NCCC3)cc(c2)-c2ccc(F)cc2C)cc(OC)c1	InChI=1S/C28H30FN3O3/c1-18-9-23(29)6-7-26(18)21-10-19(16-31-27-5-4-8-30-27)11-22(14-21)28(33)32-17-20-12-24(34-2)15-25(13-20)35-3/h6-7,9-15H,4-5,8,16-17H2,1-3H3,(H,30,31)(H,32,33)	NUDFGSDNSJHZDV-UHFFFAOYSA-N	468789	US10807959, Example 59	WD repeat-containing protein 5		 0.740								US Patent		10.7270/Q26Q219X		aid1804927	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468789	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468789&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146371063	441570890							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968661	COc1cc(CNC(=O)c2cc(CNC3=NCCC3)cc(c2)-c2ccc(F)nc2C)cc(OC)c1	InChI=1S/C27H29FN4O3/c1-17-24(6-7-25(28)32-17)20-9-18(15-30-26-5-4-8-29-26)10-21(13-20)27(33)31-16-19-11-22(34-2)14-23(12-19)35-3/h6-7,9-14H,4-5,8,15-16H2,1-3H3,(H,29,30)(H,31,33)	RKWUZLFDEPSXDB-UHFFFAOYSA-N	468790	US10807959, Example 60	WD repeat-containing protein 5		 0.550								US Patent		10.7270/Q26Q219X		aid1804927	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468790	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468790&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370730	441570891							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968662	COc1cc(CNC(=O)c2cc(CNC3=NCCC3)cc(c2)-c2ccncc2C)cc(OC)c1	InChI=1S/C27H30N4O3/c1-18-15-28-8-6-25(18)21-9-19(16-30-26-5-4-7-29-26)10-22(13-21)27(32)31-17-20-11-23(33-2)14-24(12-20)34-3/h6,8-15H,4-5,7,16-17H2,1-3H3,(H,29,30)(H,31,32)	DUYCQNMACVKGGS-UHFFFAOYSA-N	468791	US10807959, Example 61	WD repeat-containing protein 5		 1.80								US Patent		10.7270/Q26Q219X		aid1804927	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468791	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468791&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370755	441570892							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968663	COc1cc(CNC(=O)c2cc(CNC3=NCCC3)cc(c2)-c2cc(C)c(F)cc2C)cc(OC)c1	InChI=1S/C29H32FN3O3/c1-18-9-27(30)19(2)8-26(18)22-10-20(16-32-28-6-5-7-31-28)11-23(14-22)29(34)33-17-21-12-24(35-3)15-25(13-21)36-4/h8-15H,5-7,16-17H2,1-4H3,(H,31,32)(H,33,34)	NMIDLMMZIULQKW-UHFFFAOYSA-N	468792	US10807959, Example 62	WD repeat-containing protein 5		 0.210								US Patent		10.7270/Q26Q219X		aid1804927	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468792	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468792&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370972	441570893							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968664	Cc1cc(CNC(=O)c2cc(CNC3=NCCC3)cc(c2)-c2cccc(CO)c2)ccc1Cl	InChI=1S/C27H28ClN3O2/c1-18-10-19(7-8-25(18)28)15-31-27(33)24-13-21(16-30-26-6-3-9-29-26)12-23(14-24)22-5-2-4-20(11-22)17-32/h2,4-5,7-8,10-14,32H,3,6,9,15-17H2,1H3,(H,29,30)(H,31,33)	FOWSLKMJBVYBPU-UHFFFAOYSA-N	468793	US10807959, Example 63	WD repeat-containing protein 5		 0.880								US Patent		10.7270/Q26Q219X		aid1804927	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468793	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468793&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146371034	441570894							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968665	Cc1cc(CNC(=O)c2cc(CNC3=NCCC3)cc(c2)-c2ccc(F)cc2C)ccc1Cl	InChI=1S/C27H27ClFN3O/c1-17-11-23(29)6-7-24(17)21-12-20(16-31-26-4-3-9-30-26)13-22(14-21)27(33)32-15-19-5-8-25(28)18(2)10-19/h5-8,10-14H,3-4,9,15-16H2,1-2H3,(H,30,31)(H,32,33)	VHFNQVFPFPMQKD-UHFFFAOYSA-N	468794	US10807959, Example 64	WD repeat-containing protein 5		 0.640								US Patent		10.7270/Q26Q219X		aid1804927	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468794	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468794&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146371157	441570895							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968666	Cc1cc(CNC(=O)c2cc(CNC3=NCCC3)cc(c2)-c2ccc(F)c(CO)c2)ccc1Cl	InChI=1S/C27H27ClFN3O2/c1-17-9-18(4-6-24(17)28)14-32-27(34)22-11-19(15-31-26-3-2-8-30-26)10-21(13-22)20-5-7-25(29)23(12-20)16-33/h4-7,9-13,33H,2-3,8,14-16H2,1H3,(H,30,31)(H,32,34)	KXPJSTYSNQVCPB-UHFFFAOYSA-N	468795	US10807959, Example 65	WD repeat-containing protein 5		 4.30								US Patent		10.7270/Q26Q219X		aid1804927	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468795	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468795&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370924	441570896							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968667	Cc1cc(c(C)cc1F)-c1cc(CNC2=NCCC2)cc(c1)C(=O)NCc1ccc(Cl)c(C)c1	InChI=1S/C28H29ClFN3O/c1-17-11-26(30)19(3)10-24(17)22-12-21(16-32-27-5-4-8-31-27)13-23(14-22)28(34)33-15-20-6-7-25(29)18(2)9-20/h6-7,9-14H,4-5,8,15-16H2,1-3H3,(H,31,32)(H,33,34)	XDMGKYVLXNHMAD-UHFFFAOYSA-N	468796	US10807959, Example 66	WD repeat-containing protein 5		 0.380								US Patent		10.7270/Q26Q219X		aid1804927	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468796	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468796&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370945	441570897							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968668	Cc1cc(CNC(=O)c2cc(CNC3=NCCC3)cc(c2)-c2cccnc2C(F)(F)F)ccc1Cl	InChI=1S/C26H24ClF3N4O/c1-16-10-17(6-7-22(16)27)14-34-25(35)20-12-18(15-33-23-5-3-8-31-23)11-19(13-20)21-4-2-9-32-24(21)26(28,29)30/h2,4,6-7,9-13H,3,5,8,14-15H2,1H3,(H,31,33)(H,34,35)	ISGMRSHKUHZIEN-UHFFFAOYSA-N	468797	US10807959, Example 67	WD repeat-containing protein 5		<0.100								US Patent		10.7270/Q26Q219X		aid1804927	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468797	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468797&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146371019	441570898							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968669	Cc1cc(CNC(=O)c2cc(CNC3=NCCC3)cc(c2)-c2ccc(F)cc2C(F)(F)F)ccc1Cl	InChI=1S/C27H24ClF4N3O/c1-16-9-17(4-7-24(16)28)14-35-26(36)20-11-18(15-34-25-3-2-8-33-25)10-19(12-20)22-6-5-21(29)13-23(22)27(30,31)32/h4-7,9-13H,2-3,8,14-15H2,1H3,(H,33,34)(H,35,36)	BYXOHNUQRNOQBC-UHFFFAOYSA-N	468798	US10807959, Example 68	WD repeat-containing protein 5		 0.300								US Patent		10.7270/Q26Q219X		aid1804927	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468798	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468798&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146371228	441570899							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968670	COc1cc(F)c(C)cc1-c1cc(CNC2=NCCC2)cc(c1)C(=O)NCc1ccc(Cl)c(C)c1	InChI=1S/C28H29ClFN3O2/c1-17-9-19(6-7-24(17)29)15-33-28(34)22-12-20(16-32-27-5-4-8-31-27)11-21(13-22)23-10-18(2)25(30)14-26(23)35-3/h6-7,9-14H,4-5,8,15-16H2,1-3H3,(H,31,32)(H,33,34)	GPEQTZRNLVAVIJ-UHFFFAOYSA-N	468799	US10807959, Example 69	WD repeat-containing protein 5		 1.30								US Patent		10.7270/Q26Q219X		aid1804927	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468799	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468799&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370853	441570900							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968671	COc1cc(F)ccc1-c1cc(CNC2=NCCC2)cc(c1)C(=O)NCc1ccc(Cl)c(C)c1	InChI=1S/C27H27ClFN3O2/c1-17-10-18(5-8-24(17)28)15-32-27(33)21-12-19(16-31-26-4-3-9-30-26)11-20(13-21)23-7-6-22(29)14-25(23)34-2/h5-8,10-14H,3-4,9,15-16H2,1-2H3,(H,30,31)(H,32,33)	OWLREWDYINTFQX-UHFFFAOYSA-N	468800	US10807959, Example 70	WD repeat-containing protein 5		 0.500								US Patent		10.7270/Q26Q219X		aid1804927	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468800	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468800&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370830	441570901							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968672	CN1CC(=O)N=C1NCc1cc(cc(c1)-c1ccc(F)nc1C)C(=O)NCc1ccc(Cl)c(C)c1	InChI=1S/C26H25ClFN5O2/c1-15-8-17(4-6-22(15)27)12-29-25(35)20-10-18(13-30-26-32-24(34)14-33(26)3)9-19(11-20)21-5-7-23(28)31-16(21)2/h4-11H,12-14H2,1-3H3,(H,29,35)(H,30,32,34)	VLRXASQOVPPSHK-UHFFFAOYSA-N	468801	US10807959, Example 71	WD repeat-containing protein 5		 6.60								US Patent		10.7270/Q26Q219X		aid1804927	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468801	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468801&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146371005	441570902							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968673	Cc1nc(F)ccc1-c1cc(CNC2=NCCN2)cc(n1)C(=O)NCc1ccc(Cl)c(Cl)c1	InChI=1S/C23H21Cl2FN6O/c1-13-16(3-5-21(26)31-13)19-9-15(12-30-23-27-6-7-28-23)10-20(32-19)22(33)29-11-14-2-4-17(24)18(25)8-14/h2-5,8-10H,6-7,11-12H2,1H3,(H,29,33)(H2,27,28,30)	JJDOYMYROIEHHQ-UHFFFAOYSA-N	468802	US10807959, Example 72	WD repeat-containing protein 5		 0.310								US Patent		10.7270/Q26Q219X		aid1804927	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468802	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468802&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370883	441570903							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968674	Cc1nc(F)ccc1-c1cc(CNC2=NCCN2)cc(n1)C(=O)NCc1ccc(Cl)c(F)c1	InChI=1S/C23H21ClF2N6O/c1-13-16(3-5-21(26)31-13)19-9-15(12-30-23-27-6-7-28-23)10-20(32-19)22(33)29-11-14-2-4-17(24)18(25)8-14/h2-5,8-10H,6-7,11-12H2,1H3,(H,29,33)(H2,27,28,30)	SMSOHNFGNDOORA-UHFFFAOYSA-N	468803	US10807959, Example 73	WD repeat-containing protein 5		 0.430								US Patent		10.7270/Q26Q219X		aid1804927	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468803	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468803&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146371006	441570904							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968675	Cc1cc(CNC(=O)c2cc(CNC3=NCCN3)cc(n2)-c2ccc(F)nc2C)ccc1Cl	InChI=1S/C24H24ClFN6O/c1-14-9-16(3-5-19(14)25)12-29-23(33)21-11-17(13-30-24-27-7-8-28-24)10-20(32-21)18-4-6-22(26)31-15(18)2/h3-6,9-11H,7-8,12-13H2,1-2H3,(H,29,33)(H2,27,28,30)	YNGZZOYPOOUENT-UHFFFAOYSA-N	468804	US10807959, Example 74	WD repeat-containing protein 5		 0.460								US Patent		10.7270/Q26Q219X		aid1804927	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468804	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468804&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146371105	441570905							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968676	COc1cc(OC)cc(c1)C(C)NC(=O)c1cc(CNC2=NCCN2)cc(n1)-c1ccc(F)nc1C	InChI=1S/C26H29FN6O3/c1-15(18-11-19(35-3)13-20(12-18)36-4)32-25(34)23-10-17(14-30-26-28-7-8-29-26)9-22(33-23)21-5-6-24(27)31-16(21)2/h5-6,9-13,15H,7-8,14H2,1-4H3,(H,32,34)(H2,28,29,30)	UTLCNOFBVMSVTB-UHFFFAOYSA-N	468805	US10807959, Example 75	WD repeat-containing protein 5		 0.800								US Patent		10.7270/Q26Q219X		aid1804927	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468805	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468805&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370829	441570906							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968677	Cc1cnc(CNC(=O)c2cc(CNC3=NCCN3)cc(n2)-c2ccc(F)nc2C)cn1	InChI=1S/C22H23FN8O/c1-13-9-27-16(11-26-13)12-28-21(32)19-8-15(10-29-22-24-5-6-25-22)7-18(31-19)17-3-4-20(23)30-14(17)2/h3-4,7-9,11H,5-6,10,12H2,1-2H3,(H,28,32)(H2,24,25,29)	OPXWNWPYUNDGKR-UHFFFAOYSA-N	468806	US10807959, Example 76	WD repeat-containing protein 5		 32.0								US Patent		10.7270/Q26Q219X		aid1804927	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468806	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468806&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146371043	441570907							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968678	Cc1cnc(CNC(=O)c2cc(CNC3=NCCN3)cc(n2)-c2ccc(F)nc2C)nc1	InChI=1S/C22H23FN8O/c1-13-9-26-20(27-10-13)12-28-21(32)18-8-15(11-29-22-24-5-6-25-22)7-17(31-18)16-3-4-19(23)30-14(16)2/h3-4,7-10H,5-6,11-12H2,1-2H3,(H,28,32)(H2,24,25,29)	WSCJNBGFUMPWRO-UHFFFAOYSA-N	468807	US10807959, Example 77	WD repeat-containing protein 5		 33.0								US Patent		10.7270/Q26Q219X		aid1804927	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468807	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468807&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370984	441570908							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968679	COc1cc(CNC(=O)c2cc(CNC3=NCCN3)cc(n2)-c2ccc(F)nc2C)cc(OC)c1	InChI=1S/C25H27FN6O3/c1-15-20(4-5-23(26)31-15)21-10-17(14-30-25-27-6-7-28-25)11-22(32-21)24(33)29-13-16-8-18(34-2)12-19(9-16)35-3/h4-5,8-12H,6-7,13-14H2,1-3H3,(H,29,33)(H2,27,28,30)	FBAQYGSSCZKTFB-UHFFFAOYSA-N	468808	US10807959, Example 78	WD repeat-containing protein 5		 0.720								US Patent		10.7270/Q26Q219X		aid1804927	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468808	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468808&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370923	441570909							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968680	COc1cc(CNC(=O)c2cc(CNC3=NCCN3)cc(n2)-c2ccc(F)nc2C)ccn1	InChI=1S/C23H24FN7O2/c1-14-17(3-4-20(24)30-14)18-9-16(13-29-23-26-7-8-27-23)10-19(31-18)22(32)28-12-15-5-6-25-21(11-15)33-2/h3-6,9-11H,7-8,12-13H2,1-2H3,(H,28,32)(H2,26,27,29)	UFSZXLNXYHEOKQ-UHFFFAOYSA-N	468809	US10807959, Example 79	WD repeat-containing protein 5		 5.74								US Patent		10.7270/Q26Q219X		aid1804927	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468809	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468809&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370747	441570910							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968681	Cc1ncc(CNC(=O)c2cc(CNC3=NCCN3)cc(n2)-c2ccc(F)nc2C)cn1	InChI=1S/C22H23FN8O/c1-13-17(3-4-20(23)30-13)18-7-15(9-29-22-24-5-6-25-22)8-19(31-18)21(32)28-12-16-10-26-14(2)27-11-16/h3-4,7-8,10-11H,5-6,9,12H2,1-2H3,(H,28,32)(H2,24,25,29)	CDLVTAZITFCKQG-UHFFFAOYSA-N	468810	US10807959, Example 80	WD repeat-containing protein 5		 22.0								US Patent		10.7270/Q26Q219X		aid1804927	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468810	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468810&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370734	441570911							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968682	Cc1ccncc1-c1cc(CNC2=NCCN2)cc(n1)C(=O)NCc1ccc(Cl)c(Cl)c1	InChI=1S/C23H22Cl2N6O/c1-14-4-5-26-13-17(14)20-9-16(12-30-23-27-6-7-28-23)10-21(31-20)22(32)29-11-15-2-3-18(24)19(25)8-15/h2-5,8-10,13H,6-7,11-12H2,1H3,(H,29,32)(H2,27,28,30)	OQHOTHAKXDQNAZ-UHFFFAOYSA-N	468811	US10807959, Example 81	WD repeat-containing protein 5		 0.240								US Patent		10.7270/Q26Q219X		aid1804927	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468811	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468811&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370953	441570912							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968683	Cc1cc(ccn1)-c1cc(CNC2=NCCN2)cc(n1)C(=O)NCc1ccc(Cl)c(Cl)c1	InChI=1S/C23H22Cl2N6O/c1-14-8-17(4-5-26-14)20-10-16(13-30-23-27-6-7-28-23)11-21(31-20)22(32)29-12-15-2-3-18(24)19(25)9-15/h2-5,8-11H,6-7,12-13H2,1H3,(H,29,32)(H2,27,28,30)	UDPKLCBGASNKGB-UHFFFAOYSA-N	468812	US10807959, Example 82	WD repeat-containing protein 5		 0.460								US Patent		10.7270/Q26Q219X		aid1804927	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468812	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468812&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370775	441570913							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968684	COc1ncc(C)cc1-c1cc(CNC2=NCCN2)cc(n1)C(=O)NCc1ccc(Cl)c(Cl)c1	InChI=1S/C24H24Cl2N6O2/c1-14-7-17(23(34-2)30-11-14)20-9-16(13-31-24-27-5-6-28-24)10-21(32-20)22(33)29-12-15-3-4-18(25)19(26)8-15/h3-4,7-11H,5-6,12-13H2,1-2H3,(H,29,33)(H2,27,28,31)	REJSOGGUSVXDCM-UHFFFAOYSA-N	468813	US10807959, Example 83	WD repeat-containing protein 5		 0.310								US Patent		10.7270/Q26Q219X		aid1804927	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468813	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468813&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146371014	441570914							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968685	Cc1cnccc1-c1cc(CNC2=NCCN2)cc(n1)C(=O)NCc1ccc(Cl)c(Cl)c1	InChI=1S/C23H22Cl2N6O/c1-14-11-26-5-4-17(14)20-9-16(13-30-23-27-6-7-28-23)10-21(31-20)22(32)29-12-15-2-3-18(24)19(25)8-15/h2-5,8-11H,6-7,12-13H2,1H3,(H,29,32)(H2,27,28,30)	RSPUYJLFVANDQW-UHFFFAOYSA-N	468814	US10807959, Example 84	WD repeat-containing protein 5		 0.150								US Patent		10.7270/Q26Q219X		aid1804927	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468814	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468814&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370895	441570915							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968686	Cc1cc(C)nc(CNC(=O)c2cc(CNC3=NCCN3)cc(n2)-c2ccc(F)nc2C)n1	InChI=1S/C23H25FN8O/c1-13-8-14(2)30-21(29-13)12-27-22(33)19-10-16(11-28-23-25-6-7-26-23)9-18(32-19)17-4-5-20(24)31-15(17)3/h4-5,8-10H,6-7,11-12H2,1-3H3,(H,27,33)(H2,25,26,28)	YNTXURRQDYMXJZ-UHFFFAOYSA-N	468815	US10807959, Example 85	WD repeat-containing protein 5		 0.990								US Patent		10.7270/Q26Q219X		aid1804927	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468815	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468815&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370899	441570916							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968687	COc1ncc(Cl)cc1-c1cc(CNC2=NCCN2)cc(n1)C(=O)NCc1ccc(Cl)c(Cl)c1	InChI=1S/C23H21Cl3N6O2/c1-34-22-16(9-15(24)12-30-22)19-7-14(11-31-23-27-4-5-28-23)8-20(32-19)21(33)29-10-13-2-3-17(25)18(26)6-13/h2-3,6-9,12H,4-5,10-11H2,1H3,(H,29,33)(H2,27,28,31)	PVZXKTDNVPKVTN-UHFFFAOYSA-N	468816	US10807959, Example 86	WD repeat-containing protein 5		<0.100								US Patent		10.7270/Q26Q219X		aid1804927	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468816	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468816&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370958	441570917							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968688	COc1ccc(C)cc1-c1cc(CNC2=NCCN2)cc(n1)C(=O)NCc1ccc(Cl)c(Cl)c1	InChI=1S/C25H25Cl2N5O2/c1-15-3-6-23(34-2)18(9-15)21-11-17(14-31-25-28-7-8-29-25)12-22(32-21)24(33)30-13-16-4-5-19(26)20(27)10-16/h3-6,9-12H,7-8,13-14H2,1-2H3,(H,30,33)(H2,28,29,31)	WVLUIBXSYQJJSQ-UHFFFAOYSA-N	468817	US10807959, Example 87	WD repeat-containing protein 5		<0.100								US Patent		10.7270/Q26Q219X		aid1804927	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468817	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468817&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370762	441570918							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968689	CCOc1ncc(C)cc1-c1cc(CNC2=NCCN2)cc(n1)C(=O)NCc1ccc(Cl)c(Cl)c1	InChI=1S/C25H26Cl2N6O2/c1-3-35-24-18(8-15(2)12-31-24)21-10-17(14-32-25-28-6-7-29-25)11-22(33-21)23(34)30-13-16-4-5-19(26)20(27)9-16/h4-5,8-12H,3,6-7,13-14H2,1-2H3,(H,30,34)(H2,28,29,32)	JMFDWSXRBNSUPQ-UHFFFAOYSA-N	468818	US10807959, Example 88	WD repeat-containing protein 5		 0.120								US Patent		10.7270/Q26Q219X		aid1804927	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468818	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468818&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370974	441570919							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968690	Fc1ccc(-c2cc(CNC3=NCCC3)cc(n2)C(=O)NCc2ccc(Cl)c(Cl)c2)c(c1)C(F)(F)F	InChI=1S/C25H20Cl2F4N4O/c26-19-6-3-14(8-20(19)27)12-34-24(36)22-10-15(13-33-23-2-1-7-32-23)9-21(35-22)17-5-4-16(28)11-18(17)25(29,30)31/h3-6,8-11H,1-2,7,12-13H2,(H,32,33)(H,34,36)	IRCPLZIDFDRNET-UHFFFAOYSA-N	468819	US10807959, Example 89	WD repeat-containing protein 5		 1.90								US Patent		10.7270/Q26Q219X		aid1804927	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468819	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468819&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370929	441570920							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968691	Cc1ccnc(c1)C(NC(=O)c1cc(CNC2=NCCC2)cc(n1)-c1ccc(F)cc1C(F)(F)F)C1CC1	InChI=1S/C28H27F4N5O/c1-16-8-10-33-23(11-16)26(18-4-5-18)37-27(38)24-13-17(15-35-25-3-2-9-34-25)12-22(36-24)20-7-6-19(29)14-21(20)28(30,31)32/h6-8,10-14,18,26H,2-5,9,15H2,1H3,(H,34,35)(H,37,38)	ZJHGOPYSEMEMPG-UHFFFAOYSA-N	468820	US10807959, Example 90	WD repeat-containing protein 5		 1.20								US Patent		10.7270/Q26Q219X		aid1804927	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468820	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468820&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370940	441570921							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968692	COc1cc(CNC(=O)c2cc(CNC3=NCCC3)nc(c2)-c2ccc(F)cc2C(F)(F)F)cc(OC)c1	InChI=1S/C27H26F4N4O3/c1-37-20-8-16(9-21(13-20)38-2)14-34-26(36)17-10-19(15-33-25-4-3-7-32-25)35-24(11-17)22-6-5-18(28)12-23(22)27(29,30)31/h5-6,8-13H,3-4,7,14-15H2,1-2H3,(H,32,33)(H,34,36)	CHOMAKSSNAKZTK-UHFFFAOYSA-N	468821	US10807959, Example 91	WD repeat-containing protein 5		 1.60								US Patent		10.7270/Q26Q219X		aid1804927	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468821	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468821&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146371003	441570922							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968693	C[C@H](NC(=O)c1cc(CNC2=NCCC2)cc(n1)-c1ccc(F)cc1C(F)(F)F)c1ccc(Cl)c(C)c1	InChI=1S/C27H25ClF4N4O/c1-15-10-18(5-8-22(15)28)16(2)35-26(37)24-12-17(14-34-25-4-3-9-33-25)11-23(36-24)20-7-6-19(29)13-21(20)27(30,31)32/h5-8,10-13,16H,3-4,9,14H2,1-2H3,(H,33,34)(H,35,37)/t16-/m0/s1	QPYZZUQOFSOCFY-INIZCTEOSA-N	468822	US10807959, Example 92	WD repeat-containing protein 5		 1.50								US Patent		10.7270/Q26Q219X		aid1804927	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468822	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468822&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146371039	441570923							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968694	COc1cc(OC)cc(c1)C(C)NC(=O)c1cc(CNC2=NCCC2)cc(n1)-c1ccc(F)cc1C(F)(F)F	InChI=1S/C28H28F4N4O3/c1-16(18-11-20(38-2)14-21(12-18)39-3)35-27(37)25-10-17(15-34-26-5-4-8-33-26)9-24(36-25)22-7-6-19(29)13-23(22)28(30,31)32/h6-7,9-14,16H,4-5,8,15H2,1-3H3,(H,33,34)(H,35,37)	CUEPGJAGFNKCLD-UHFFFAOYSA-N	468823	US10807959, Example 93	WD repeat-containing protein 5		 3.30								US Patent		10.7270/Q26Q219X		aid1804927	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468823	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468823&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370745	441570924							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981459	CCn1cc(c(n1)C(F)(F)F)-c1cc(CN2CCOC2=N)cc(c1)C(=O)NCC1CCOC1	InChI=1S/C22H26F3N5O3/c1-2-30-12-18(19(28-30)22(23,24)25)16-7-15(11-29-4-6-33-21(29)26)8-17(9-16)20(31)27-10-14-3-5-32-13-14/h7-9,12,14,26H,2-6,10-11,13H2,1H3,(H,27,31)	DCFAKXBACIFGKK-UHFFFAOYSA-N	473254	US10844044, Example 290	WD repeat-containing protein 5		 20.0								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473254	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473254&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456071	442073466							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981460	Cc1cc(CNC(=O)c2cc(Cn3ccn(C)c3=N)cc(c2)-c2ccnn2C)ccc1Cl	InChI=1S/C24H25ClN6O/c1-16-10-17(4-5-21(16)25)14-27-23(32)20-12-18(15-31-9-8-29(2)24(31)26)11-19(13-20)22-6-7-28-30(22)3/h4-13,26H,14-15H2,1-3H3,(H,27,32)	VVBGZQAPLNVLMF-UHFFFAOYSA-N	473255	US10844044, Example 17	WD repeat-containing protein 5		 0.940								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473255	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473255&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456084	442073467							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981461	COc1cc(CNC(=O)c2cc(Cn3ccn(C)c3=N)cc(c2F)-c2ccc(F)cc2C(F)(F)F)cc(OC)c1	InChI=1S/C28H25F5N4O3/c1-36-6-7-37(27(36)34)15-17-10-22(21-5-4-18(29)12-24(21)28(31,32)33)25(30)23(11-17)26(38)35-14-16-8-19(39-2)13-20(9-16)40-3/h4-13,34H,14-15H2,1-3H3,(H,35,38)	VWZAGEVGWUQNJL-UHFFFAOYSA-N	473256	US10844044, Example 108	WD repeat-containing protein 5		<0.100								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473256	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473256&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456199	442073468							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981462	CCn1cc(c(n1)C(F)(F)F)-c1cc(Cn2ccn(C3CC3)c2=N)cc(c1)C(=O)NCc1ccc(=O)n(C)c1	InChI=1S/C27H28F3N7O2/c1-3-36-16-22(24(33-36)27(28,29)30)19-10-18(15-35-8-9-37(26(35)31)21-5-6-21)11-20(12-19)25(39)32-13-17-4-7-23(38)34(2)14-17/h4,7-12,14,16,21,31H,3,5-6,13,15H2,1-2H3,(H,32,39)	LGXXBAMZIVGJEP-UHFFFAOYSA-N	473257	US10844044, Example 199	WD repeat-containing protein 5		 0.300								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473257	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473257&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146455776	442073469							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981463	CC(C)n1cc(c(n1)C(F)(F)F)-c1cc(Cn2ccoc2=N)cc(c1)C(=O)N[C@@H](C1CC1)c1ccc(F)c(C)c1	InChI=1S/C29H29F4N5O2/c1-16(2)38-15-23(26(36-38)29(31,32)33)21-11-18(14-37-8-9-40-28(37)34)12-22(13-21)27(39)35-25(19-4-5-19)20-6-7-24(30)17(3)10-20/h6-13,15-16,19,25,34H,4-5,14H2,1-3H3,(H,35,39)/t25-/m0/s1	MFKPRJPANTWPHT-VWLOTQADSA-N	473258	US10844044, Example 291	WD repeat-containing protein 5		<0.100								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473258	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473258&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456667	442073470							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981464	Cc1cc(ccn1)-c1cc(Cn2ccn(C)c2=N)cc(c1)C(=O)NCc1ccc(Cl)c(C)c1	InChI=1S/C26H26ClN5O/c1-17-10-19(4-5-24(17)27)15-30-25(33)23-13-20(16-32-9-8-31(3)26(32)28)12-22(14-23)21-6-7-29-18(2)11-21/h4-14,28H,15-16H2,1-3H3,(H,30,33)	FFELOLPQYKXVQJ-UHFFFAOYSA-N	473259	US10844044, Example 18	WD repeat-containing protein 5		 3.50								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473259	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473259&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456654	442073471							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981465	Cc1cc(ccc1F)[C@@H](NC(=O)c1cc(Cn2ccn(C)c2=N)cc(c1F)-c1ccc(F)cc1C(F)(F)F)C1CC1	InChI=1S/C30H26F6N4O/c1-16-11-19(5-8-25(16)32)27(18-3-4-18)38-28(41)23-13-17(15-40-10-9-39(2)29(40)37)12-22(26(23)33)21-7-6-20(31)14-24(21)30(34,35)36/h5-14,18,27,37H,3-4,15H2,1-2H3,(H,38,41)/t27-/m0/s1	NGCXKJBNAVLJAI-MHZLTWQESA-N	473260	US10844044, Example 109	WD repeat-containing protein 5		<0.100								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473260	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473260&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456475	442073472							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981466	CCn1cc(c(n1)C(F)(F)F)-c1cc(Cn2ccn(C)c2=N)cc(c1)C(=O)NCc1ccc(=O)n(C)c1	InChI=1S/C25H26F3N7O2/c1-4-35-15-20(22(31-35)25(26,27)28)18-9-17(14-34-8-7-32(2)24(34)29)10-19(11-18)23(37)30-12-16-5-6-21(36)33(3)13-16/h5-11,13,15,29H,4,12,14H2,1-3H3,(H,30,37)	XDGKYFOWXFYLKC-UHFFFAOYSA-N	473261	US10844044, Example 200	WD repeat-containing protein 5		 0.150								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473261	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473261&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456402	442073473							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981467	CCn1cc(c(n1)C(F)(F)F)-c1cc(Cn2ccoc2=N)cc(c1)C(=O)NCc1ccc(=O)n(C)c1	InChI=1S/C24H23F3N6O3/c1-3-33-14-19(21(30-33)24(25,26)27)17-8-16(13-32-6-7-36-23(32)28)9-18(10-17)22(35)29-11-15-4-5-20(34)31(2)12-15/h4-10,12,14,28H,3,11,13H2,1-2H3,(H,29,35)	FVGWTRMTJJJDQO-UHFFFAOYSA-N	473262	US10844044, Example 292	WD repeat-containing protein 5		 1.10								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473262	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473262&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456133	442073474							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981468	Cc1cc(CNC(=O)c2cc(Cn3cc[nH]c3=N)cc(c2)-c2cccn2C)ccc1Cl	InChI=1S/C24H24ClN5O/c1-16-10-17(5-6-21(16)25)14-28-23(31)20-12-18(15-30-9-7-27-24(30)26)11-19(13-20)22-4-3-8-29(22)2/h3-13H,14-15H2,1-2H3,(H2,26,27)(H,28,31)	SCKVLJFPQFKGDA-UHFFFAOYSA-N	473263	US10844044, Example 19	WD repeat-containing protein 5		 0.350								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473263	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473263&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146457041	442073475							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981469	COC(=O)CC(NC(=O)c1cc(Cn2ccn(C)c2=N)cc(c1F)-c1ccc(F)cc1C(F)(F)F)c1ccc(Cl)c(Cl)c1	InChI=1S/C29H23Cl2F5N4O3/c1-39-7-8-40(28(39)37)14-15-9-19(18-5-4-17(32)12-21(18)29(34,35)36)26(33)20(10-15)27(42)38-24(13-25(41)43-2)16-3-6-22(30)23(31)11-16/h3-12,24,37H,13-14H2,1-2H3,(H,38,42)	BAEBGXJRILNWDE-UHFFFAOYSA-N	473264	US10844044, Example 110	WD repeat-containing protein 5		 0.100								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473264	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473264&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146455927	442073476							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981470	Cc1cc(ccc1F)[C@@H](NC(=O)c1cc(Cn2ccn(C)c2=N)cc(c1)-c1ccccc1C)C1CC1	InChI=1S/C30H31FN4O/c1-19-6-4-5-7-26(19)24-15-21(18-35-13-12-34(3)30(35)32)16-25(17-24)29(36)33-28(22-8-9-22)23-10-11-27(31)20(2)14-23/h4-7,10-17,22,28,32H,8-9,18H2,1-3H3,(H,33,36)/t28-/m0/s1	STFMCBSGCNEJKN-NDEPHWFRSA-N	473265	US10844044, Example 201	WD repeat-containing protein 5		<0.100								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473265	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473265&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456544	442073477							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981471	CCn1cc(c(n1)C(F)(F)F)-c1cc(CN2CCOC2=N)cc(c1)C(=O)NCc1ccc(=O)n(C)c1	InChI=1S/C24H25F3N6O3/c1-3-33-14-19(21(30-33)24(25,26)27)17-8-16(13-32-6-7-36-23(32)28)9-18(10-17)22(35)29-11-15-4-5-20(34)31(2)12-15/h4-5,8-10,12,14,28H,3,6-7,11,13H2,1-2H3,(H,29,35)	NRLVHJIGDXLTNU-UHFFFAOYSA-N	473266	US10844044, Example 293	WD repeat-containing protein 5		 0.540								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473266	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473266&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146455766	442073478							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981472	COc1cnccc1-c1cc(Cn2ccn(C)c2=N)cc(c1)C(=O)NCc1ccc(Cl)c(C)c1	InChI=1S/C26H26ClN5O2/c1-17-10-18(4-5-23(17)27)14-30-25(33)21-12-19(16-32-9-8-31(2)26(32)28)11-20(13-21)22-6-7-29-15-24(22)34-3/h4-13,15,28H,14,16H2,1-3H3,(H,30,33)	FMTWGZGNAPSFOS-UHFFFAOYSA-N	473267	US10844044, Example 20	WD repeat-containing protein 5		 2.50								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473267	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473267&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146455835	442073479							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981473	Cc1cc(CNC(=O)c2cc(Cn3ccn(C)c3=N)cc(c2F)-c2ccc(F)cc2C(F)(F)F)ccc1Cl	InChI=1S/C27H22ClF5N4O/c1-15-9-16(3-6-23(15)28)13-35-25(38)21-11-17(14-37-8-7-36(2)26(37)34)10-20(24(21)30)19-5-4-18(29)12-22(19)27(31,32)33/h3-12,34H,13-14H2,1-2H3,(H,35,38)	JRTJHGXDXCATKI-UHFFFAOYSA-N	473268	US10844044, Example 111	WD repeat-containing protein 5		<0.100								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473268	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473268&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456593	442073480							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981474	CCn1cc(c(n1)C(F)(F)F)-c1cc(Cn2ccn(C3CC3)c2=N)cc(c1)C(=O)N[C@@H](C1CC1)c1ccc(F)c(Cl)c1	InChI=1S/C30H29ClF4N6O/c1-2-40-16-23(27(38-40)30(33,34)35)20-11-17(15-39-9-10-41(29(39)36)22-6-7-22)12-21(13-20)28(42)37-26(18-3-4-18)19-5-8-25(32)24(31)14-19/h5,8-14,16,18,22,26,36H,2-4,6-7,15H2,1H3,(H,37,42)/t26-/m0/s1	VQZPLGHPOFUJHK-SANMLTNESA-N	473269	US10844044, Example 202	WD repeat-containing protein 5		<0.100								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473269	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473269&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456298	442073481							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981475	CCn1cc(c(n1)C(F)(F)F)-c1cc(Cn2ccoc2=N)cc(c1)C(=O)NCc1ccc(F)c(C)c1	InChI=1S/C25H23F4N5O2/c1-3-34-14-20(22(32-34)25(27,28)29)18-9-17(13-33-6-7-36-24(33)30)10-19(11-18)23(35)31-12-16-4-5-21(26)15(2)8-16/h4-11,14,30H,3,12-13H2,1-2H3,(H,31,35)	CWHLAVCHAUHKGC-UHFFFAOYSA-N	473270	US10844044, Example 294	WD repeat-containing protein 5		<0.100								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473270	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473270&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146457651	442073482							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981476	Cn1cccc1-c1cc(Cn2ccn(C)c2=N)cc(c1)C(=O)NCc1ccc(Cl)c(Cl)c1	InChI=1S/C24H23Cl2N5O/c1-29-7-3-4-22(29)18-10-17(15-31-9-8-30(2)24(31)27)11-19(13-18)23(32)28-14-16-5-6-20(25)21(26)12-16/h3-13,27H,14-15H2,1-2H3,(H,28,32)	MLGKWRKTOAWDOO-UHFFFAOYSA-N	473271	US10844044, Example 21	WD repeat-containing protein 5		 0.640								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473271	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473271&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456193	442073483							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981477	Cc1[nH]c(=O)ccc1-c1cc(Cn2ccn(C)c2=N)cc(c1)C(=O)NCc1ccc(Cl)c(Cl)c1	InChI=1S/C25H23Cl2N5O2/c1-15-20(4-6-23(33)30-15)18-9-17(14-32-8-7-31(2)25(32)28)10-19(12-18)24(34)29-13-16-3-5-21(26)22(27)11-16/h3-12,28H,13-14H2,1-2H3,(H,29,34)(H,30,33)	LOBPFOLFDBJDEE-UHFFFAOYSA-N	473272	US10844044, Example 112	WD repeat-containing protein 5		 29.0								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473272	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473272&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			156022869	442073484							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981478	CN1CCN(Cc2cc(cc(c2)-c2cn(C)nc2C(F)(F)F)C(=O)N[C@@H](C2CC2)c2ccc(F)c(C)c2)C1=N	InChI=1S/C28H30F4N6O/c1-16-10-19(6-7-23(16)29)24(18-4-5-18)34-26(39)21-12-17(14-38-9-8-36(2)27(38)33)11-20(13-21)22-15-37(3)35-25(22)28(30,31)32/h6-7,10-13,15,18,24,33H,4-5,8-9,14H2,1-3H3,(H,34,39)/t24-/m0/s1	XFELDXYOLGFGBH-DEOSSOPVSA-N	473273	US10844044, Example 203	WD repeat-containing protein 5		<0.100								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473273	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473273&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146457350	442073485							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981479	CCn1cc(c(n1)C(F)(F)F)-c1cc(CN2CCOC2=N)cc(c1)C(=O)NCc1ccc(F)c(C)c1	InChI=1S/C25H25F4N5O2/c1-3-34-14-20(22(32-34)25(27,28)29)18-9-17(13-33-6-7-36-24(33)30)10-19(11-18)23(35)31-12-16-4-5-21(26)15(2)8-16/h4-5,8-11,14,30H,3,6-7,12-13H2,1-2H3,(H,31,35)	UGLDYEXYEKNIFG-UHFFFAOYSA-N	473274	US10844044, Example 295	WD repeat-containing protein 5		<0.100								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473274	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473274&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146455714	442073486							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981480	Cc1cc(ccn1)-c1cc(Cn2ccn(C)c2=N)cc(c1)C(=O)NCc1ccc(Cl)c(Cl)c1	InChI=1S/C25H23Cl2N5O/c1-16-9-19(5-6-29-16)20-10-18(15-32-8-7-31(2)25(32)28)11-21(13-20)24(33)30-14-17-3-4-22(26)23(27)12-17/h3-13,28H,14-15H2,1-2H3,(H,30,33)	KSAXHZMTSFDGTI-UHFFFAOYSA-N	473276	US10844044, Example 22	WD repeat-containing protein 5		 6.40								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473276	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473276&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456399	442073488							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981481	Cc1cc(ccc1F)[C@@H](NC(=O)c1cc(Cn2ccn(C)c2=N)cc(c1)-c1cnc(F)cc1C)C1CC1	InChI=1S/C29H29F2N5O/c1-17-11-26(31)33-15-24(17)22-12-19(16-36-9-8-35(3)29(36)32)13-23(14-22)28(37)34-27(20-4-5-20)21-6-7-25(30)18(2)10-21/h6-15,20,27,32H,4-5,16H2,1-3H3,(H,34,37)/t27-/m0/s1	WGRHFEXFWAIIGL-MHZLTWQESA-N	473277	US10844044, Example 113	WD repeat-containing protein 5		>33.0								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473277	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473277&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456251	442073489							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981482	Cc1cc(ncc1F)[C@@H](NC(=O)c1cc(Cn2ccn(C3CC3)c2=N)cc(c1)-c1cn(C)nc1C(F)(F)F)C1CC1	InChI=1S/C29H29F4N7O/c1-16-9-24(35-13-23(16)30)25(18-3-4-18)36-27(41)20-11-17(14-39-7-8-40(28(39)34)21-5-6-21)10-19(12-20)22-15-38(2)37-26(22)29(31,32)33/h7-13,15,18,21,25,34H,3-6,14H2,1-2H3,(H,36,41)/t25-/m0/s1	VESLYKRFMKRVBD-VWLOTQADSA-N	473278	US10844044, Example 204	WD repeat-containing protein 5		<0.100								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473278	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473278&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146457700	442073490							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981483	C[C@H]1CN(Cc2cc(cc(c2)-c2cccnc2C(F)(F)F)C(=O)N[C@@H](C2CC2)c2ccc(F)c(C)c2)C(=N)O1	InChI=1S/C29H28F4N4O2/c1-16-10-20(7-8-24(16)30)25(19-5-6-19)36-27(38)22-12-18(15-37-14-17(2)39-28(37)34)11-21(13-22)23-4-3-9-35-26(23)29(31,32)33/h3-4,7-13,17,19,25,34H,5-6,14-15H2,1-2H3,(H,36,38)/t17-,25-/m0/s1	JUFSLJSOTQNBPW-GKVSMKOHSA-N	473279	US10844044, Example 296	WD repeat-containing protein 5		 7.00								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473279	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473279&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146457356	442073491							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981484	COc1cnccc1-c1cc(Cn2ccn(C)c2=N)cc(c1)C(=O)NCc1ccc(Cl)c(Cl)c1	InChI=1S/C25H23Cl2N5O2/c1-31-7-8-32(25(31)28)15-17-9-18(20-5-6-29-14-23(20)34-2)12-19(10-17)24(33)30-13-16-3-4-21(26)22(27)11-16/h3-12,14,28H,13,15H2,1-2H3,(H,30,33)	VSQFBDGGMZKBOO-UHFFFAOYSA-N	473280	US10844044, Example 23	WD repeat-containing protein 5		 5.70								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473280	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473280&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146455940	442073492							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981485	CCn1ccn(Cc2cc(cc(c2)-c2cccnc2C(F)(F)F)C(=O)N[C@@H](C2CC2)c2ccc(F)c(C)c2)c1=N	InChI=1S/C30H29F4N5O/c1-3-38-11-12-39(29(38)35)17-19-14-22(24-5-4-10-36-27(24)30(32,33)34)16-23(15-19)28(40)37-26(20-6-7-20)21-8-9-25(31)18(2)13-21/h4-5,8-16,20,26,35H,3,6-7,17H2,1-2H3,(H,37,40)/t26-/m0/s1	MCGFPQFQBSHHTF-SANMLTNESA-N	473281	US10844044, Example 114	WD repeat-containing protein 5		<0.100								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473281	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473281&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146457022	442073493							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981486	Cc1cc(ncc1F)[C@@H](NC(=O)c1cc(Cn2ccn(C)c2=N)cc(c1)-c1cn(C)nc1C(F)(F)F)C1CC1	InChI=1S/C27H27F4N7O/c1-15-8-22(33-12-21(15)28)23(17-4-5-17)34-25(39)19-10-16(13-38-7-6-36(2)26(38)32)9-18(11-19)20-14-37(3)35-24(20)27(29,30)31/h6-12,14,17,23,32H,4-5,13H2,1-3H3,(H,34,39)/t23-/m0/s1	RWNNXLKTNWWOCP-QHCPKHFHSA-N	473282	US10844044, Example 205	WD repeat-containing protein 5		<0.100								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473282	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473282&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456155	442073494							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981487	C[C@@H]1CN(Cc2cc(cc(c2)-c2cccnc2C(F)(F)F)C(=O)N[C@@H](C2CC2)c2ccc(F)c(C)c2)C(=N)O1	InChI=1S/C29H28F4N4O2/c1-16-10-20(7-8-24(16)30)25(19-5-6-19)36-27(38)22-12-18(15-37-14-17(2)39-28(37)34)11-21(13-22)23-4-3-9-35-26(23)29(31,32)33/h3-4,7-13,17,19,25,34H,5-6,14-15H2,1-2H3,(H,36,38)/t17-,25+/m1/s1	JUFSLJSOTQNBPW-NSYGIPOTSA-N	473283	US10844044, Example 297	WD repeat-containing protein 5		 2.30								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473283	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473283&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146455931	442073495							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981488	COc1cc(ccn1)-c1cc(Cn2ccn(C)c2=N)cc(c1)C(=O)NCc1ccc(Cl)c(Cl)c1	InChI=1S/C25H23Cl2N5O2/c1-31-7-8-32(25(31)28)15-17-9-19(18-5-6-29-23(13-18)34-2)12-20(10-17)24(33)30-14-16-3-4-21(26)22(27)11-16/h3-13,28H,14-15H2,1-2H3,(H,30,33)	XVXHVPJWGIFKLL-UHFFFAOYSA-N	473284	US10844044, Example 24	WD repeat-containing protein 5		 25.0								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473284	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473284&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146455954	442073496							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981489	Cc1cc(ccc1F)[C@@H](NC(=O)c1cc(Cn2ccn(C3CC3)c2=N)cc(c1)-c1cccnc1C(F)(F)F)C1CC1	InChI=1S/C31H29F4N5O/c1-18-13-21(6-9-26(18)32)27(20-4-5-20)38-29(41)23-15-19(17-39-11-12-40(30(39)36)24-7-8-24)14-22(16-23)25-3-2-10-37-28(25)31(33,34)35/h2-3,6,9-16,20,24,27,36H,4-5,7-8,17H2,1H3,(H,38,41)/t27-/m0/s1	LUBSALMJHCMFQI-MHZLTWQESA-N	473285	US10844044, Example 115	WD repeat-containing protein 5		<0.100								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473285	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473285&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146455799	442073497							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981490	Cc1cc(ccc1F)[C@@H](NC(=O)c1cc(Cn2ccn(C)c2=N)cc(c1)N1CCCC1)C1CC1	InChI=1S/C27H32FN5O/c1-18-13-21(7-8-24(18)28)25(20-5-6-20)30-26(34)22-14-19(17-33-12-11-31(2)27(33)29)15-23(16-22)32-9-3-4-10-32/h7-8,11-16,20,25,29H,3-6,9-10,17H2,1-2H3,(H,30,34)/t25-/m0/s1	FCJHBKYAOAOAFF-VWLOTQADSA-N	473286	US10844044, Example 206	WD repeat-containing protein 5		 0.340								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473286	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473286&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456407	442073498							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981491	CCn1cc(c(n1)C(F)(F)F)-c1cc(Cn2ccoc2=N)cc(c1)C(=O)N[C@@H](C1CC1)c1ccc(F)c(Cl)c1	InChI=1S/C27H24ClF4N5O2/c1-2-37-14-20(24(35-37)27(30,31)32)18-9-15(13-36-7-8-39-26(36)33)10-19(11-18)25(38)34-23(16-3-4-16)17-5-6-22(29)21(28)12-17/h5-12,14,16,23,33H,2-4,13H2,1H3,(H,34,38)/t23-/m0/s1	HFUVKGPHYGHZOK-QHCPKHFHSA-N	473287	US10844044, Example 298	WD repeat-containing protein 5		<0.100								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473287	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473287&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456318	442073499							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981492	Cc1cnccc1-c1cc(Cn2ccn(C)c2=N)cc(c1)C(=O)NCc1ccc(Cl)c(Cl)c1	InChI=1S/C25H23Cl2N5O/c1-16-13-29-6-5-21(16)19-9-18(15-32-8-7-31(2)25(32)28)10-20(12-19)24(33)30-14-17-3-4-22(26)23(27)11-17/h3-13,28H,14-15H2,1-2H3,(H,30,33)	HZCXZXADGOSMDP-UHFFFAOYSA-N	473288	US10844044, Example 25	WD repeat-containing protein 5		 1.30								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473288	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473288&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146457379	442073500							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981493	CCn1ccn(Cc2cc(cc(c2)-c2ccc(F)cc2C)C(=O)NCc2cc(OC)cc(OC)c2)c1=N	InChI=1S/C29H31FN4O3/c1-5-33-8-9-34(29(33)31)18-21-11-22(27-7-6-24(30)10-19(27)2)15-23(12-21)28(35)32-17-20-13-25(36-3)16-26(14-20)37-4/h6-16,31H,5,17-18H2,1-4H3,(H,32,35)	NZKQZTCHZGFDHM-UHFFFAOYSA-N	473289	US10844044, Example 116	WD repeat-containing protein 5		 0.400								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473289	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473289&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456288	442073501							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981494	COc1cc(ccc1F)[C@@H](NC(=O)c1cc(Cn2ccn(C)c2=N)cc(c1)-c1cn(C)nc1C(F)(F)F)C1CC1	InChI=1S/C28H28F4N6O2/c1-36-8-9-38(27(36)33)14-16-10-19(21-15-37(2)35-25(21)28(30,31)32)12-20(11-16)26(39)34-24(17-4-5-17)18-6-7-22(29)23(13-18)40-3/h6-13,15,17,24,33H,4-5,14H2,1-3H3,(H,34,39)/t24-/m0/s1	HJTWVFIIZRJPSG-DEOSSOPVSA-N	473290	US10844044, Example 207	WD repeat-containing protein 5		<0.100								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473290	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473290&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456047	442073502							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981495	Cc1cc(ncc1F)[C@@H](NC(=O)c1cc(Cn2ccoc2=N)cc(c1)-c1cn(C)nc1C(F)(F)F)C1CC1	InChI=1S/C26H24F4N6O2/c1-14-7-21(32-11-20(14)27)22(16-3-4-16)33-24(37)18-9-15(12-36-5-6-38-25(36)31)8-17(10-18)19-13-35(2)34-23(19)26(28,29)30/h5-11,13,16,22,31H,3-4,12H2,1-2H3,(H,33,37)/t22-/m0/s1	DPJQFJQSHYISES-QFIPXVFZSA-N	473291	US10844044, Example 299	WD repeat-containing protein 5		<0.100								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473291	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473291&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456166	442073503							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981496	Cn1ccn(Cc2cc(cc(c2)-c2ccnn2C)C(=O)NCc2ccc(Cl)c(Cl)c2)c1=N	InChI=1S/C23H22Cl2N6O/c1-29-7-8-31(23(29)26)14-16-9-17(21-5-6-28-30(21)2)12-18(10-16)22(32)27-13-15-3-4-19(24)20(25)11-15/h3-12,26H,13-14H2,1-2H3,(H,27,32)	ATQLRHVTOPYWGC-UHFFFAOYSA-N	473292	US10844044, Example 26	WD repeat-containing protein 5		 0.720								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473292	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473292&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146455971	442073504							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981497	COc1cc(CNC(=O)c2cc(Cn3ccn(C4CC4)c3=N)cc(c2)-c2ccc(F)cc2C)cc(OC)c1	InChI=1S/C30H31FN4O3/c1-19-10-24(31)4-7-28(19)22-11-21(18-34-8-9-35(30(34)32)25-5-6-25)12-23(15-22)29(36)33-17-20-13-26(37-2)16-27(14-20)38-3/h4,7-16,25,32H,5-6,17-18H2,1-3H3,(H,33,36)	SHSKQHGZMLWEQY-UHFFFAOYSA-N	473293	US10844044, Example 117	WD repeat-containing protein 5		 0.150								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473293	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473293&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456292	442073505							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981498	Cc1cc(ncc1F)[C@@H](NC(=O)c1cc(Cn2ccn(C)c2=N)cc(c1)N1CCCC1)C1CC1	InChI=1S/C26H31FN6O/c1-17-11-23(29-15-22(17)27)24(19-5-6-19)30-25(34)20-12-18(16-33-10-9-31(2)26(33)28)13-21(14-20)32-7-3-4-8-32/h9-15,19,24,28H,3-8,16H2,1-2H3,(H,30,34)/t24-/m0/s1	ORFBPMAZILMILR-DEOSSOPVSA-N	473294	US10844044, Example 208	WD repeat-containing protein 5		 0.590								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473294	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473294&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456777	442073506							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981499	Cc1cc(ncc1F)[C@@H](NC(=O)c1cc(CN2CCOC2=N)cc(c1)-c1cn(C)nc1C(F)(F)F)C1CC1	InChI=1S/C26H26F4N6O2/c1-14-7-21(32-11-20(14)27)22(16-3-4-16)33-24(37)18-9-15(12-36-5-6-38-25(36)31)8-17(10-18)19-13-35(2)34-23(19)26(28,29)30/h7-11,13,16,22,31H,3-6,12H2,1-2H3,(H,33,37)/t22-/m0/s1	IGSGNLFYIDDDCI-QFIPXVFZSA-N	473295	US10844044, Example 300	WD repeat-containing protein 5		<0.100								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473295	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473295&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456411	442073507							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981500	Cc1ccc2[nH]ncc2c1-c1cc(Cn2ccn(C)c2=N)cc(c1)C(=O)NCc1ccc(Cl)c(Cl)c1	InChI=1S/C27H24Cl2N6O/c1-16-3-6-24-21(14-32-33-24)25(16)19-9-18(15-35-8-7-34(2)27(35)30)10-20(12-19)26(36)31-13-17-4-5-22(28)23(29)11-17/h3-12,14,30H,13,15H2,1-2H3,(H,31,36)(H,32,33)	LFLLGKQOTMRFFB-UHFFFAOYSA-N	473296	US10844044, Example 27	WD repeat-containing protein 5		 1.50								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473296	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473296&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146455915	442073508							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981501	COc1cc(OC)cc(c1)C(NC(=O)c1cc(Cn2ccn(C)c2=N)cc(c1)-c1ccnn1C(C)C)C1CC1	InChI=1S/C30H36N6O3/c1-19(2)36-27(8-9-32-36)22-12-20(18-35-11-10-34(3)30(35)31)13-24(14-22)29(37)33-28(21-6-7-21)23-15-25(38-4)17-26(16-23)39-5/h8-17,19,21,28,31H,6-7,18H2,1-5H3,(H,33,37)	DTMLAZNGBSUUKA-UHFFFAOYSA-N	473297	US10844044, Example 118	WD repeat-containing protein 5		 0.830								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473297	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473297&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146455920	442073509							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981502	CCOc1c(cc(Cn2ccn(C)c2=N)cc1-c1cn(C)nc1C(F)(F)F)C(=O)N[C@@H](C)c1ccc(F)c(C)c1	InChI=1S/C28H30F4N6O2/c1-6-40-24-20(22-15-37(5)35-25(22)28(30,31)32)12-18(14-38-10-9-36(4)27(38)33)13-21(24)26(39)34-17(3)19-7-8-23(29)16(2)11-19/h7-13,15,17,33H,6,14H2,1-5H3,(H,34,39)/t17-/m0/s1	HHOAWASKOWIQHK-KRWDZBQOSA-N	473298	US10844044, Example 209	WD repeat-containing protein 5		<0.100								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473298	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473298&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146455739	442073510							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981503	Fc1ccc(c(Cl)c1)-c1cc(CN2CCOC2=N)cc(c1)C(=O)N[C@@H](C1CC1)c1ccc(Cl)c(F)c1	InChI=1S/C27H23Cl2F2N3O2/c28-22-6-3-17(12-24(22)31)25(16-1-2-16)33-26(35)19-10-15(14-34-7-8-36-27(34)32)9-18(11-19)21-5-4-20(30)13-23(21)29/h3-6,9-13,16,25,32H,1-2,7-8,14H2,(H,33,35)/t25-/m0/s1	FPKKFSITUYTLIG-VWLOTQADSA-N	473299	US10844044, Example 301	WD repeat-containing protein 5		<0.100								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473299	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473299&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456114	442073511							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981504	Cc1cc(F)cc(F)c1-c1cc(Cn2ccn(C)c2=N)cc(c1)C(=O)NCc1ccc(Cl)c(Cl)c1	InChI=1S/C26H22Cl2F2N4O/c1-15-7-20(29)12-23(30)24(15)18-8-17(14-34-6-5-33(2)26(34)31)9-19(11-18)25(35)32-13-16-3-4-21(27)22(28)10-16/h3-12,31H,13-14H2,1-2H3,(H,32,35)	ZNCGBLVLEIXOJY-UHFFFAOYSA-N	473300	US10844044, Example 28	WD repeat-containing protein 5		 0.350								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473300	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473300&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146457930	442073512							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981505	Cc1cc(ccc1F)[C@@H](NC(=O)c1cc(Cn2ccn(C)c2=N)cc(n1)-c1cccnc1C(F)(F)F)C1CC1	InChI=1S/C28H26F4N6O/c1-16-12-19(7-8-21(16)29)24(18-5-6-18)36-26(39)23-14-17(15-38-11-10-37(2)27(38)33)13-22(35-23)20-4-3-9-34-25(20)28(30,31)32/h3-4,7-14,18,24,33H,5-6,15H2,1-2H3,(H,36,39)/t24-/m0/s1	WNRXLZREBBUMNM-DEOSSOPVSA-N	473301	US10844044, Example 119	WD repeat-containing protein 5		 0.160								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473301	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473301&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456245	442073513							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981506	CCOc1c(cc(Cn2ccn(C)c2=N)cc1-c1cn(C)nc1C(F)(F)F)C(=O)N[C@@H](C1CC1)c1ccc(F)c(C)c1	InChI=1S/C30H32F4N6O2/c1-5-42-26-21(23-16-39(4)37-27(23)30(32,33)34)13-18(15-40-11-10-38(3)29(40)35)14-22(26)28(41)36-25(19-6-7-19)20-8-9-24(31)17(2)12-20/h8-14,16,19,25,35H,5-7,15H2,1-4H3,(H,36,41)/t25-/m0/s1	IBNCSJDFRUSYMR-VWLOTQADSA-N	473302	US10844044, Example 210	WD repeat-containing protein 5		<0.100								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473302	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473302&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456771	442073514							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981507	CCOc1c(cc(CN2CCOC2=N)cc1-c1cn(C)nc1C(F)(F)F)C(=O)N[C@@H](C)c1ccc(F)c(C)c1	InChI=1S/C27H29F4N5O3/c1-5-38-23-19(21-14-35(4)34-24(21)27(29,30)31)11-17(13-36-8-9-39-26(36)32)12-20(23)25(37)33-16(3)18-6-7-22(28)15(2)10-18/h6-7,10-12,14,16,32H,5,8-9,13H2,1-4H3,(H,33,37)/t16-/m0/s1	YJMQCVVTYQFVHY-INIZCTEOSA-N	473303	US10844044, Example 302	WD repeat-containing protein 5		<0.100								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473303	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473303&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456664	442073515							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981508	C[C@@H](NC(=O)c1cc(Cn2ccn(C)c2=N)cc(c1)-c1ccc(F)cc1C)c1ccc(F)c(C)c1	InChI=1S/C28H28F2N4O/c1-17-12-24(29)6-7-25(17)22-13-20(16-34-10-9-33(4)28(34)31)14-23(15-22)27(35)32-19(3)21-5-8-26(30)18(2)11-21/h5-15,19,31H,16H2,1-4H3,(H,32,35)/t19-/m1/s1	WLJUDWPYHBJUSE-LJQANCHMSA-N	473304	US10844044, Example 29	WD repeat-containing protein 5		 0.280								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473304	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473304&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456564	442073516							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981509	Cc1ccnc(c1)[C@@H](NC(=O)c1cc(Cn2ccn(C)c2=N)cc(c1F)-c1ccc(F)cc1C(F)(F)F)C1CC1	InChI=1S/C29H26F5N5O/c1-16-7-8-36-24(11-16)26(18-3-4-18)37-27(40)22-13-17(15-39-10-9-38(2)28(39)35)12-21(25(22)31)20-6-5-19(30)14-23(20)29(32,33)34/h5-14,18,26,35H,3-4,15H2,1-2H3,(H,37,40)/t26-/m0/s1	XMSBMGGMBZIKEW-SANMLTNESA-N	473305	US10844044, Example 120	WD repeat-containing protein 5		<0.100								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473305	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473305&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146455702	442073517							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981510	Cn1cc(c(n1)C(F)(F)F)-c1cc(Cn2ccn(C)c2=N)cc(c1)C(=O)N[C@@H](C1CC1)c1ccc(Cl)c(Cl)c1	InChI=1S/C27H25Cl2F3N6O/c1-36-7-8-38(26(36)33)13-15-9-18(20-14-37(2)35-24(20)27(30,31)32)11-19(10-15)25(39)34-23(16-3-4-16)17-5-6-21(28)22(29)12-17/h5-12,14,16,23,33H,3-4,13H2,1-2H3,(H,34,39)/t23-/m0/s1	XXBDHHUZDWANQK-QHCPKHFHSA-N	473306	US10844044, Example 157::US10844044, Example 211	WD repeat-containing protein 5		<0.100								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473306	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473306&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456260	442073518							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981511	CCOc1c(cc(CN2CCOC2=N)cc1-c1cn(C)nc1C(F)(F)F)C(=O)N[C@@H](C1CC1)c1ccc(F)c(C)c1	InChI=1S/C29H31F4N5O3/c1-4-40-25-20(22-15-37(3)36-26(22)29(31,32)33)12-17(14-38-9-10-41-28(38)34)13-21(25)27(39)35-24(18-5-6-18)19-7-8-23(30)16(2)11-19/h7-8,11-13,15,18,24,34H,4-6,9-10,14H2,1-3H3,(H,35,39)/t24-/m0/s1	QJKPWBWMBDTKDO-DEOSSOPVSA-N	473307	US10844044, Example 303	WD repeat-containing protein 5		<0.100								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473307	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473307&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456294	442073519							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981512	C[C@H](NC(=O)c1cc(Cn2ccn(C)c2=N)cc(c1)-c1ccc(F)cc1C)c1ccc(F)c(C)c1	InChI=1S/C28H28F2N4O/c1-17-12-24(29)6-7-25(17)22-13-20(16-34-10-9-33(4)28(34)31)14-23(15-22)27(35)32-19(3)21-5-8-26(30)18(2)11-21/h5-15,19,31H,16H2,1-4H3,(H,32,35)/t19-/m0/s1	WLJUDWPYHBJUSE-IBGZPJMESA-N	473308	US10844044, Example 30	WD repeat-containing protein 5		<0.100								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473308	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473308&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456357	442073520							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981513	CC(=O)\N=c1/n(C)ccn1Cc1cc(cc(c1)-c1ccc(F)nc1C)C(=O)NCc1ccc(Cl)c(Cl)c1	InChI=1S/C27H24Cl2FN5O2/c1-16-22(5-7-25(30)32-16)20-10-19(15-35-9-8-34(3)27(35)33-17(2)36)11-21(13-20)26(37)31-14-18-4-6-23(28)24(29)12-18/h4-13H,14-15H2,1-3H3,(H,31,37)/b33-27+	PIGJSXMSIDVRBW-MUGXBBEHSA-N	473309	US10844044, Example 121	WD repeat-containing protein 5		>33.0								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473309	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473309&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456390	442073521							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981514	CCn1cc(c(n1)C(F)(F)F)-c1cc(Cn2ccn(C)c2=N)cc(c1)C(=O)N[C@@H](C1CC1)c1ccc(F)c(C)c1	InChI=1S/C29H30F4N6O/c1-4-39-16-23(26(36-39)29(31,32)33)21-12-18(15-38-10-9-37(3)28(38)34)13-22(14-21)27(40)35-25(19-5-6-19)20-7-8-24(30)17(2)11-20/h7-14,16,19,25,34H,4-6,15H2,1-3H3,(H,35,40)/t25-/m0/s1	SBXCJLHQQJUEHZ-VWLOTQADSA-N	473310	US10844044, Example 212	WD repeat-containing protein 5		<0.100								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473310	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473310&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146487971	442073522							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968695	COc1ccnc(CNC(=O)c2cc(CNC3=NCCC3)cc(n2)-c2ccc(F)cc2C(F)(F)F)c1	InChI=1S/C25H23F4N5O2/c1-36-18-6-8-30-17(12-18)14-33-24(35)22-10-15(13-32-23-3-2-7-31-23)9-21(34-22)19-5-4-16(26)11-20(19)25(27,28)29/h4-6,8-12H,2-3,7,13-14H2,1H3,(H,31,32)(H,33,35)	RHTGRUUBNOQISB-UHFFFAOYSA-N	468824	US10807959, Example 94	WD repeat-containing protein 5		 1.20								US Patent		10.7270/Q26Q219X		aid1804927	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468824	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468824&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370731	441570925							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968696	Cc1ccnc(c1)C(NC(=O)c1cc(CNC2=NCCC2)cc(n1)-c1ccc(F)cc1C)C1CC1	InChI=1S/C28H30FN5O/c1-17-9-11-30-24(12-17)27(20-5-6-20)34-28(35)25-15-19(16-32-26-4-3-10-31-26)14-23(33-25)22-8-7-21(29)13-18(22)2/h7-9,11-15,20,27H,3-6,10,16H2,1-2H3,(H,31,32)(H,34,35)	RBNZNTCSOZINBP-UHFFFAOYSA-N	468825	US10807959, Example 95	WD repeat-containing protein 5		 8.60								US Patent		10.7270/Q26Q219X		aid1804927	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468825	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468825&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370898	441570926							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968697	CC(NC(=O)c1cc(CNC2=NCCC2)cc(n1)-c1ccc(F)cc1C(F)(F)F)c1cc(C)c(Cl)cn1	InChI=1S/C26H24ClF4N5O/c1-14-8-21(33-13-20(14)27)15(2)35-25(37)23-10-16(12-34-24-4-3-7-32-24)9-22(36-23)18-6-5-17(28)11-19(18)26(29,30)31/h5-6,8-11,13,15H,3-4,7,12H2,1-2H3,(H,32,34)(H,35,37)	UTGNODDDCMEOQZ-UHFFFAOYSA-N	468826	US10807959, Example 96	WD repeat-containing protein 5		 1.50								US Patent		10.7270/Q26Q219X		aid1804927	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468826	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468826&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146371158	441570927							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968698	C[C@H](NC(=O)c1cc(CNC2=NCCC2)cc(n1)-c1ccc(F)cc1C)c1ccc(F)c(c1)C(F)(F)F	InChI=1S/C27H25F5N4O/c1-15-10-19(28)6-7-20(15)23-11-17(14-34-25-4-3-9-33-25)12-24(36-23)26(37)35-16(2)18-5-8-22(29)21(13-18)27(30,31)32/h5-8,10-13,16H,3-4,9,14H2,1-2H3,(H,33,34)(H,35,37)/t16-/m0/s1	QZSYHWGTYXPLIC-INIZCTEOSA-N	468827	US10807959, Example 97	WD repeat-containing protein 5		 7.30								US Patent		10.7270/Q26Q219X		aid1804927	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468827	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468827&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146371080	441570928							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968699	Cc1nc(F)ccc1-c1cc(CNC2=NCCN2)cc(n1)C(=O)NCc1ccc(=O)[nH]c1	InChI=1S/C22H22FN7O2/c1-13-16(3-4-19(23)29-13)17-8-15(12-28-22-24-6-7-25-22)9-18(30-17)21(32)27-11-14-2-5-20(31)26-10-14/h2-5,8-10H,6-7,11-12H2,1H3,(H,26,31)(H,27,32)(H2,24,25,28)	ZBXJRWSJCZDGIY-UHFFFAOYSA-N	468828	US10807959, Example 98	WD repeat-containing protein 5		 23.0								US Patent		10.7270/Q26Q219X		aid1804927	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468828	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468828&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			155921719	441570929							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968700	COc1cc(CNC(=O)c2cc(CNC(N)=N)cc(c2)-c2ccnc(C)c2)cc(OC)c1	InChI=1S/C24H27N5O3/c1-15-6-18(4-5-27-15)19-7-16(14-29-24(25)26)8-20(11-19)23(30)28-13-17-9-21(31-2)12-22(10-17)32-3/h4-12H,13-14H2,1-3H3,(H,28,30)(H4,25,26,29)	WTWQHNSVSVXCFJ-UHFFFAOYSA-N	468829	US10807959, Example 99	WD repeat-containing protein 5		 1.10								US Patent		10.7270/Q26Q219X		aid1804927	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468829	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468829&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370963	441570930							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968701	Cc1cc(ccn1)-c1cc(CNC(N)=N)cc(c1)C(=O)NCc1cc(F)cc(Cl)c1	InChI=1S/C22H21ClFN5O/c1-13-4-16(2-3-27-13)17-5-14(12-29-22(25)26)6-18(9-17)21(30)28-11-15-7-19(23)10-20(24)8-15/h2-10H,11-12H2,1H3,(H,28,30)(H4,25,26,29)	YNJKMUFOXNWJRK-UHFFFAOYSA-N	468830	US10807959, Example 100	WD repeat-containing protein 5		 2.40								US Patent		10.7270/Q26Q219X		aid1804927	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468830	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468830&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146371036	441570931							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968702	COc1ccc(CNC(=O)c2cc(CNC(N)=N)cc(c2)-c2ccnc(C)c2)cc1Cl	InChI=1S/C23H24ClN5O2/c1-14-7-17(5-6-27-14)18-8-16(13-29-23(25)26)9-19(11-18)22(30)28-12-15-3-4-21(31-2)20(24)10-15/h3-11H,12-13H2,1-2H3,(H,28,30)(H4,25,26,29)	ZPLOGCMMXPYNQG-UHFFFAOYSA-N	468831	US10807959, Example 101	WD repeat-containing protein 5		 2.10								US Patent		10.7270/Q26Q219X		aid1804927	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468831	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468831&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370727	441570932							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968703	COc1ccnc(CNC(=O)c2cc(CNC(N)=N)cc(c2)-c2ccnc(C)c2)c1	InChI=1S/C22H24N6O2/c1-14-7-16(3-5-25-14)17-8-15(12-28-22(23)24)9-18(10-17)21(29)27-13-19-11-20(30-2)4-6-26-19/h3-11H,12-13H2,1-2H3,(H,27,29)(H4,23,24,28)	QNDBQMWUPDEOCO-UHFFFAOYSA-N	468832	US10807959, Example 102	WD repeat-containing protein 5		 1.000								US Patent		10.7270/Q26Q219X		aid1804927	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468832	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468832&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146371000	441570933							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968704	Cc1cc(ccn1)-c1cc(CNC(N)=N)cc(c1)C(=O)NCc1ccc(Cl)cn1	InChI=1S/C21H21ClN6O/c1-13-6-15(4-5-25-13)16-7-14(10-28-21(23)24)8-17(9-16)20(29)27-12-19-3-2-18(22)11-26-19/h2-9,11H,10,12H2,1H3,(H,27,29)(H4,23,24,28)	GRRHOFOENKFPNM-UHFFFAOYSA-N	468833	US10807959, Example 103	WD repeat-containing protein 5		 3.30								US Patent		10.7270/Q26Q219X		aid1804927	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468833	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468833&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370803	441570934							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968705	Cc1ccc(CNC(=O)c2cc(CNC(N)=N)cc(c2)-c2ccnc(C)c2)cn1	InChI=1S/C22H24N6O/c1-14-3-4-16(11-26-14)12-27-21(29)20-9-17(13-28-22(23)24)8-19(10-20)18-5-6-25-15(2)7-18/h3-11H,12-13H2,1-2H3,(H,27,29)(H4,23,24,28)	VDEPHGQABIOPIZ-UHFFFAOYSA-N	468834	US10807959, Example 104	WD repeat-containing protein 5		 12.0								US Patent		10.7270/Q26Q219X		aid1804927	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468834	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468834&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146371009	441570935							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968706	CCn1cc(c(n1)C(F)(F)F)-c1cc(CNC(=N)C2CC2)cc(c1)C(=O)N[C@@H](C1CC1)c1ccc(F)c(C)c1	InChI=1S/C29H31F4N5O/c1-3-38-15-23(26(37-38)29(31,32)33)21-11-17(14-35-27(34)19-6-7-19)12-22(13-21)28(39)36-25(18-4-5-18)20-8-9-24(30)16(2)10-20/h8-13,15,18-19,25H,3-7,14H2,1-2H3,(H2,34,35)(H,36,39)/t25-/m0/s1	HEHNXNWDOJTUAT-VWLOTQADSA-N	468835	US10807959, Example 105	WD repeat-containing protein 5		<0.100								US Patent		10.7270/Q26Q219X		aid1804927	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468835	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468835&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146388357	441570936							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968707	CCn1cc(c(n1)C(F)(F)F)-c1cc(CNC(=N)C2CCC2)cc(c1)C(=O)N[C@@H](C1CC1)c1ccc(F)c(C)c1	InChI=1S/C30H33F4N5O/c1-3-39-16-24(27(38-39)30(32,33)34)22-12-18(15-36-28(35)20-5-4-6-20)13-23(14-22)29(40)37-26(19-7-8-19)21-9-10-25(31)17(2)11-21/h9-14,16,19-20,26H,3-8,15H2,1-2H3,(H2,35,36)(H,37,40)/t26-/m0/s1	KZSIXXAKNZZHJR-SANMLTNESA-N	468836	US10807959, Example 106	WD repeat-containing protein 5		<0.100								US Patent		10.7270/Q26Q219X		aid1804927	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468836	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468836&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146388344	441570937							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968708	CCn1cc(c(n1)C(F)(F)F)-c1cc(CNC(=N)CC2CC2)cc(c1)C(=O)N[C@@H](C1CC1)c1ccc(F)c(C)c1	InChI=1S/C30H33F4N5O/c1-3-39-16-24(28(38-39)30(32,33)34)22-11-19(15-36-26(35)13-18-4-5-18)12-23(14-22)29(40)37-27(20-6-7-20)21-8-9-25(31)17(2)10-21/h8-12,14,16,18,20,27H,3-7,13,15H2,1-2H3,(H2,35,36)(H,37,40)/t27-/m0/s1	WOCQKLHDXWEVLU-MHZLTWQESA-N	468837	US10807959, Example 107	WD repeat-containing protein 5		 0.150								US Patent		10.7270/Q26Q219X		aid1804927	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468837	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468837&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146388304	441570938							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968709	CCn1cc(c(n1)C(F)(F)F)-c1cc(CNC(=N)C2CCOC2)cc(c1)C(=O)N[C@@H](C1CC1)c1ccc(F)c(C)c1	InChI=1S/C30H33F4N5O2/c1-3-39-15-24(27(38-39)30(32,33)34)22-11-18(14-36-28(35)21-8-9-41-16-21)12-23(13-22)29(40)37-26(19-4-5-19)20-6-7-25(31)17(2)10-20/h6-7,10-13,15,19,21,26H,3-5,8-9,14,16H2,1-2H3,(H2,35,36)(H,37,40)/t21?,26-/m0/s1	XPEWSUMUZIKCHW-UQTORGHUSA-N	468838	US10807959, Example 108	WD repeat-containing protein 5		 2.00								US Patent		10.7270/Q26Q219X		aid1804927	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468838	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468838&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146388306	441570939							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968710	CCn1cc(c(n1)C(F)(F)F)-c1cc(CNC(=N)C2(C)CC2)cc(c1)C(=O)N[C@@H](C1CC1)c1ccc(F)c(C)c1	InChI=1S/C30H33F4N5O/c1-4-39-16-23(26(38-39)30(32,33)34)21-12-18(15-36-28(35)29(3)9-10-29)13-22(14-21)27(40)37-25(19-5-6-19)20-7-8-24(31)17(2)11-20/h7-8,11-14,16,19,25H,4-6,9-10,15H2,1-3H3,(H2,35,36)(H,37,40)/t25-/m0/s1	QGEUHDWFTZDVPL-VWLOTQADSA-N	468839	US10807959, Example 109	WD repeat-containing protein 5		 0.130								US Patent		10.7270/Q26Q219X		aid1804927	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468839	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468839&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146388358	441570940							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968711	Fc1ccc(c(Cl)c1)-c1cc(Cn2ccnc2)cc(c1)C(=O)NCc1ccc(Cl)c(Cl)c1	InChI=1S/C24H17Cl3FN3O/c25-21-4-1-15(9-23(21)27)12-30-24(32)18-8-16(13-31-6-5-29-14-31)7-17(10-18)20-3-2-19(28)11-22(20)26/h1-11,14H,12-13H2,(H,30,32)	MLESPKVIRFJOEN-UHFFFAOYSA-N	468704	US10807959, Example 116	WD repeat-containing protein 5		 1.30								US Patent		10.7270/Q26Q219X		aid1804927	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468704	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468704&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370869	441570805							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968712	Cc1nc(F)ccc1-c1cc(Cn2ccnc2)cc(c1)C(=O)NC(C1CC1)C1CC1	InChI=1S/C24H25FN4O/c1-15-21(6-7-22(25)27-15)19-10-16(13-29-9-8-26-14-29)11-20(12-19)24(30)28-23(17-2-3-17)18-4-5-18/h6-12,14,17-18,23H,2-5,13H2,1H3,(H,28,30)	NDWGDICKLLHJRK-UHFFFAOYSA-N	468721	US10807959, Example 133	WD repeat-containing protein 5		 4.60								US Patent		10.7270/Q26Q219X		aid1804927	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468721	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468721&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370840	441570822							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968713	Cc1nccn1Cc1cc(cc(c1)-c1ccc(F)cc1Cl)C(=O)NCc1ccc(Cl)c(Cl)c1	InChI=1S/C25H19Cl3FN3O/c1-15-30-6-7-32(15)14-17-8-18(21-4-3-20(29)12-23(21)27)11-19(9-17)25(33)31-13-16-2-5-22(26)24(28)10-16/h2-12H,13-14H2,1H3,(H,31,33)	UUQJUPSTHIASAJ-UHFFFAOYSA-N	468722	US10807959, Example 134	WD repeat-containing protein 5		 1.000								US Patent		10.7270/Q26Q219X		aid1804927	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468722	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468722&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370927	441570823							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968714	Cc1ccnc(c1)C(NC(=O)c1cc(Cn2ccnc2)cc(c1)-c1ccc(F)nc1C)C1CC1	InChI=1S/C27H26FN5O/c1-17-7-8-30-24(11-17)26(20-3-4-20)32-27(34)22-13-19(15-33-10-9-29-16-33)12-21(14-22)23-5-6-25(28)31-18(23)2/h5-14,16,20,26H,3-4,15H2,1-2H3,(H,32,34)	UBPIMOHMVJQFFW-UHFFFAOYSA-N	468725	US10807959, Example 137	WD repeat-containing protein 5		 2.00								US Patent		10.7270/Q26Q219X		aid1804927	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468725	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468725&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370915	441570826							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968715	CC1(CCCC1)NC(=O)c1cc(Cn2ccnc2)cc(c1)-c1ccc(F)cc1Cl	InChI=1S/C23H23ClFN3O/c1-23(6-2-3-7-23)27-22(29)18-11-16(14-28-9-8-26-15-28)10-17(12-18)20-5-4-19(25)13-21(20)24/h4-5,8-13,15H,2-3,6-7,14H2,1H3,(H,27,29)	GLIZWTMFVCPOAP-UHFFFAOYSA-N	468840	US10807959, Example 138	WD repeat-containing protein 5		 50.0								US Patent		10.7270/Q26Q219X		aid1804927	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468840	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468840&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370903	441570941							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968716	Cc1nc(F)ccc1-c1cc(Cn2ccnc2C2CC2)cc(c1)C(=O)NCc1ccc(Cl)c(Cl)c1	InChI=1S/C27H23Cl2FN4O/c1-16-22(5-7-25(30)33-16)20-10-18(15-34-9-8-31-26(34)19-3-4-19)11-21(13-20)27(35)32-14-17-2-6-23(28)24(29)12-17/h2,5-13,19H,3-4,14-15H2,1H3,(H,32,35)	WSEHOMFQHDXKIB-UHFFFAOYSA-N	468841	US10807959, Example 139	WD repeat-containing protein 5		 1.60								US Patent		10.7270/Q26Q219X		aid1804927	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468841	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468841&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370851	441570942							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968717	COc1cc(CN(C)C(=O)c2cc(Cn3ccnc3)cc(c2)-c2ccc(F)nc2C)cc(OC)c1	InChI=1S/C27H27FN4O3/c1-18-25(5-6-26(28)30-18)21-9-19(16-32-8-7-29-17-32)10-22(13-21)27(33)31(2)15-20-11-23(34-3)14-24(12-20)35-4/h5-14,17H,15-16H2,1-4H3	DLWOJGDTNINSIY-UHFFFAOYSA-N	468842	US10807959, Example 140	WD repeat-containing protein 5		 95.0								US Patent		10.7270/Q26Q219X		aid1804927	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468842	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468842&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370768	441570943							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968718	FC(F)(F)c1cc(Cn2ccnc2)cc(c1)C(=O)NCc1ccc(Cl)c(Cl)c1	InChI=1S/C19H14Cl2F3N3O/c20-16-2-1-12(7-17(16)21)9-26-18(28)14-5-13(10-27-4-3-25-11-27)6-15(8-14)19(22,23)24/h1-8,11H,9-10H2,(H,26,28)	CIQMNIRMYOOVEL-UHFFFAOYSA-N	468843	US10807959, Example 141	WD repeat-containing protein 5		 10.00								US Patent		10.7270/Q26Q219X		aid1804927	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468843	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468843&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370913	441570944							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968719	Clc1ccc(CNC(=O)c2cc(Cn3ccnc3)cc(OC3CCC3)c2)cc1Cl	InChI=1S/C22H21Cl2N3O2/c23-20-5-4-15(10-21(20)24)12-26-22(28)17-8-16(13-27-7-6-25-14-27)9-19(11-17)29-18-2-1-3-18/h4-11,14,18H,1-3,12-13H2,(H,26,28)	DTAHWVOEJJPJOY-UHFFFAOYSA-N	468844	US10807959, Example 142	WD repeat-containing protein 5		 0.590								US Patent		10.7270/Q26Q219X		aid1804927	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468844	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468844&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146371018	441570945							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968720	Cc1nccn1Cc1cc(OC2CCC2)cc(c1)C(=O)NCc1ccc(Cl)c(Cl)c1	InChI=1S/C23H23Cl2N3O2/c1-15-26-7-8-28(15)14-17-9-18(12-20(10-17)30-19-3-2-4-19)23(29)27-13-16-5-6-21(24)22(25)11-16/h5-12,19H,2-4,13-14H2,1H3,(H,27,29)	RVTRTLHQKXYZGX-UHFFFAOYSA-N	468845	US10807959, Example 143	WD repeat-containing protein 5		 0.430								US Patent		10.7270/Q26Q219X		aid1804927	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468845	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468845&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370879	441570946							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968721	Cc1nccn1Cc1cc(cc(c1)C(=O)NC(C1CC1)c1cc(C)ccn1)N1CCOCC1	InChI=1S/C26H31N5O2/c1-18-5-6-28-24(13-18)25(21-3-4-21)29-26(32)22-14-20(17-31-8-7-27-19(31)2)15-23(16-22)30-9-11-33-12-10-30/h5-8,13-16,21,25H,3-4,9-12,17H2,1-2H3,(H,29,32)	FDWWCCVCFIWJRR-UHFFFAOYSA-N	468846	US10807959, Example 144	WD repeat-containing protein 5		 4.77								US Patent		10.7270/Q26Q219X		aid1804927	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468846	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468846&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370885	441570947							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968722	COc1cc(CNC(=O)c2cc(Cn3ccnc3)cc(c2)-c2ccc(=O)[nH]c2)cc(OC)c1	InChI=1S/C25H24N4O4/c1-32-22-9-17(10-23(12-22)33-2)13-28-25(31)21-8-18(15-29-6-5-26-16-29)7-20(11-21)19-3-4-24(30)27-14-19/h3-12,14,16H,13,15H2,1-2H3,(H,27,30)(H,28,31)	GEJBFDQAFCZDQC-UHFFFAOYSA-N	468847	US10807959, Example 145	WD repeat-containing protein 5		 22.0								US Patent		10.7270/Q26Q219X		aid1804927	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468847	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468847&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			155921720	441570948							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968723	COc1ccnc(CNC(=O)c2cc(C)c(OC)c(Cn3ccnc3C)c2)c1	InChI=1S/C21H24N4O3/c1-14-9-16(21(26)24-12-18-11-19(27-3)5-6-23-18)10-17(20(14)28-4)13-25-8-7-22-15(25)2/h5-11H,12-13H2,1-4H3,(H,24,26)	YWOBCHRDCMXYFR-UHFFFAOYSA-N	468848	US10807959, Example 146	WD repeat-containing protein 5		 500								US Patent		10.7270/Q26Q219X		aid1804927	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468848	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468848&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370822	441570949							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968724	Cc1cncn1Cc1cc(nc(c1)-c1cccc(CO)c1)C(=O)NCc1ccc(Cl)c(Cl)c1	InChI=1S/C25H22Cl2N4O2/c1-16-11-28-15-31(16)13-19-9-23(20-4-2-3-18(7-20)14-32)30-24(10-19)25(33)29-12-17-5-6-21(26)22(27)8-17/h2-11,15,32H,12-14H2,1H3,(H,29,33)	IORMZRXMQGFIHQ-UHFFFAOYSA-N	468849	US10807959, Example 147	WD repeat-containing protein 5		 0.310								US Patent		10.7270/Q26Q219X		aid1804927	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468849	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468849&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146388324	441570950							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968725	Cc1ccnc(c1)C(NC(=O)c1cc(Cn2ccnc2)cc(n1)-c1ccc(F)cc1Cl)C1CC1	InChI=1S/C26H23ClFN5O/c1-16-6-7-30-23(10-16)25(18-2-3-18)32-26(34)24-12-17(14-33-9-8-29-15-33)11-22(31-24)20-5-4-19(28)13-21(20)27/h4-13,15,18,25H,2-3,14H2,1H3,(H,32,34)	NLWDHZNWWYOXLN-UHFFFAOYSA-N	468728	US10807959, Example 150	WD repeat-containing protein 5		 5.71								US Patent		10.7270/Q26Q219X		aid1804927	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468728	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468728&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146371012	441570829							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968726	Cc1cccc(CNC(=O)c2cc(Cn3ccnc3)cc(n2)-c2ccc(F)cc2Cl)n1	InChI=1S/C23H19ClFN5O/c1-15-3-2-4-18(28-15)12-27-23(31)22-10-16(13-30-8-7-26-14-30)9-21(29-22)19-6-5-17(25)11-20(19)24/h2-11,14H,12-13H2,1H3,(H,27,31)	FCVZKYYPBCCHIA-UHFFFAOYSA-N	468729	US10807959, Example 151	WD repeat-containing protein 5		 32.0								US Patent		10.7270/Q26Q219X		aid1804927	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468729	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468729&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370878	441570830							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968727	Cc1nccn1Cc1cc(nc(c1)-c1ccc(F)cc1C)C(=O)NCc1ccc(Cl)c(Cl)c1	InChI=1S/C25H21Cl2FN4O/c1-15-9-19(28)4-5-20(15)23-11-18(14-32-8-7-29-16(32)2)12-24(31-23)25(33)30-13-17-3-6-21(26)22(27)10-17/h3-12H,13-14H2,1-2H3,(H,30,33)	OUAHQXRMIPLGQF-UHFFFAOYSA-N	468850	US10807959, Example 156	WD repeat-containing protein 5		 2.15								US Patent		10.7270/Q26Q219X		aid1804927	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468850	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468850&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370801	441570951							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968728	COc1cc(OC)cc(c1)C(C)NC(=O)c1cc(Cn2ccnc2C)cc(n1)-c1cccc(CO)c1	InChI=1S/C28H30N4O4/c1-18(23-13-24(35-3)15-25(14-23)36-4)30-28(34)27-12-21(16-32-9-8-29-19(32)2)11-26(31-27)22-7-5-6-20(10-22)17-33/h5-15,18,33H,16-17H2,1-4H3,(H,30,34)	ZIGHYWSPTIECGR-UHFFFAOYSA-N	468851	US10807959, Example 157	WD repeat-containing protein 5		 27.0								US Patent		10.7270/Q26Q219X		aid1804927	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468851	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468851&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370776	441570952							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968729	COc1cc(OC)cc(c1)C(C)NC(=O)c1cc(Cn2ccnc2C)cc(n1)-c1ccc(F)cc1OC	InChI=1S/C28H29FN4O4/c1-17(20-12-22(35-3)15-23(13-20)36-4)31-28(34)26-11-19(16-33-9-8-30-18(33)2)10-25(32-26)24-7-6-21(29)14-27(24)37-5/h6-15,17H,16H2,1-5H3,(H,31,34)	XAUBSSBUXMGFIK-UHFFFAOYSA-N	468852	US10807959, Example 158	WD repeat-containing protein 5		 8.00								US Patent		10.7270/Q26Q219X		aid1804927	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468852	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468852&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370920	441570953							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968730	COc1cc(OC)cc(c1)C(C)NC(=O)c1cc(Cn2ccnc2C)cc(n1)-c1ccc(F)nc1C	InChI=1S/C27H28FN5O3/c1-16(20-12-21(35-4)14-22(13-20)36-5)31-27(34)25-11-19(15-33-9-8-29-18(33)3)10-24(32-25)23-6-7-26(28)30-17(23)2/h6-14,16H,15H2,1-5H3,(H,31,34)	YUGGAXKERFSEBA-UHFFFAOYSA-N	468853	US10807959, Example 159	WD repeat-containing protein 5		 3.90								US Patent		10.7270/Q26Q219X		aid1804927	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468853	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468853&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146371017	441570954							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968731	COc1cc(OC)cc(c1)C(C)NC(=O)c1cc(Cn2ccnc2C)cc(n1)-c1cc(ccc1OC)C(F)(F)F	InChI=1S/C29H29F3N4O4/c1-17(20-12-22(38-3)15-23(13-20)39-4)34-28(37)26-11-19(16-36-9-8-33-18(36)2)10-25(35-26)24-14-21(29(30,31)32)6-7-27(24)40-5/h6-15,17H,16H2,1-5H3,(H,34,37)	ZQKIIKZCOYCSCF-UHFFFAOYSA-N	468854	US10807959, Example 160	WD repeat-containing protein 5		>33.0								US Patent		10.7270/Q26Q219X		aid1804927	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468854	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468854&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370808	441570955							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968732	COc1cc(OC)cc(c1)C(C)NC(=O)c1cc(Cn2ccnc2C)cc(n1)-c1ccc(F)c(c1)C(N)=O	InChI=1S/C28H28FN5O4/c1-16(20-11-21(37-3)14-22(12-20)38-4)32-28(36)26-10-18(15-34-8-7-31-17(34)2)9-25(33-26)19-5-6-24(29)23(13-19)27(30)35/h5-14,16H,15H2,1-4H3,(H2,30,35)(H,32,36)	QBLGEMQQNMLGSL-UHFFFAOYSA-N	468855	US10807959, Example 161	WD repeat-containing protein 5		>33.0								US Patent		10.7270/Q26Q219X		aid1804927	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468855	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468855&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146371011	441570956							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968733	COc1ncccc1-c1cc(Cn2ccnc2C)cc(n1)C(=O)NCc1ccc(Cl)c(Cl)c1	InChI=1S/C24H21Cl2N5O2/c1-15-27-8-9-31(15)14-17-11-21(18-4-3-7-28-24(18)33-2)30-22(12-17)23(32)29-13-16-5-6-19(25)20(26)10-16/h3-12H,13-14H2,1-2H3,(H,29,32)	OOLKLCFIJYMSFE-UHFFFAOYSA-N	468856	US10807959, Example 162	WD repeat-containing protein 5		 6.40								US Patent		10.7270/Q26Q219X		aid1804927	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468856	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468856&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146371008	441570957							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968734	COc1cc(OC)cc(c1)C(C)NC(=O)c1cc(Cn2ccnc2C)cc(n1)-c1ccc(F)c(CO)c1	InChI=1S/C28H29FN4O4/c1-17(21-12-23(36-3)14-24(13-21)37-4)31-28(35)27-10-19(15-33-8-7-30-18(33)2)9-26(32-27)20-5-6-25(29)22(11-20)16-34/h5-14,17,34H,15-16H2,1-4H3,(H,31,35)	NXLAOWSJGSQXRG-UHFFFAOYSA-N	468857	US10807959, Example 163	WD repeat-containing protein 5		>33.0								US Patent		10.7270/Q26Q219X		aid1804927	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468857	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468857&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370795	441570958							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968735	Cc1nccn1Cc1cc(nc(c1)-c1ccc(F)nc1C)C(=O)NCc1ccc(Cl)c(Cl)c1	InChI=1S/C24H20Cl2FN5O/c1-14-18(4-6-23(27)30-14)21-10-17(13-32-8-7-28-15(32)2)11-22(31-21)24(33)29-12-16-3-5-19(25)20(26)9-16/h3-11H,12-13H2,1-2H3,(H,29,33)	SAZBBSALDUBDMF-UHFFFAOYSA-N	468858	US10807959, Example 164	WD repeat-containing protein 5		 0.280								US Patent		10.7270/Q26Q219X		aid1804927	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468858	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468858&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370810	441570959							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968736	COc1cc(F)ccc1-c1cc(Cn2ccnc2C)cc(n1)C(=O)NCc1ccc(Cl)c(Cl)c1	InChI=1S/C25H21Cl2FN4O2/c1-15-29-7-8-32(15)14-17-10-22(19-5-4-18(28)12-24(19)34-2)31-23(11-17)25(33)30-13-16-3-6-20(26)21(27)9-16/h3-12H,13-14H2,1-2H3,(H,30,33)	DPMGXNKAXKVVJS-UHFFFAOYSA-N	468859	US10807959, Example 165	WD repeat-containing protein 5		 11.0								US Patent		10.7270/Q26Q219X		aid1804927	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468859	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468859&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370739	441570960							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968737	Cc1nccn1Cc1cc(nc(c1)-c1ccncc1C)C(=O)NCc1ccc(Cl)c(Cl)c1	InChI=1S/C24H21Cl2N5O/c1-15-12-27-6-5-19(15)22-10-18(14-31-8-7-28-16(31)2)11-23(30-22)24(32)29-13-17-3-4-20(25)21(26)9-17/h3-12H,13-14H2,1-2H3,(H,29,32)	ZLSUBDOORBXNEU-UHFFFAOYSA-N	468860	US10807959, Example 166	WD repeat-containing protein 5		 2.44								US Patent		10.7270/Q26Q219X		aid1804927	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468860	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468860&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370778	441570961							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968738	Cc1nccn1Cc1cc(nc(c1)-c1ccc(F)c(c1)C(N)=O)C(=O)NCc1ccc(Cl)c(Cl)c1	InChI=1S/C25H20Cl2FN5O2/c1-14-30-6-7-33(14)13-16-9-22(17-3-5-21(28)18(11-17)24(29)34)32-23(10-16)25(35)31-12-15-2-4-19(26)20(27)8-15/h2-11H,12-13H2,1H3,(H2,29,34)(H,31,35)	ZWSLCWAUHOQXQN-UHFFFAOYSA-N	468861	US10807959, Example 167	WD repeat-containing protein 5		>33.0								US Patent		10.7270/Q26Q219X		aid1804927	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468861	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468861&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370874	441570962							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968739	COc1cc(CNC(=O)c2cc(CNC3=NCCC3)cc(c2N)-c2ccc(F)cc2C)cc(OC)c1	InChI=1S/C28H31FN4O3/c1-17-9-20(29)6-7-23(17)24-12-19(15-32-26-5-4-8-31-26)13-25(27(24)30)28(34)33-16-18-10-21(35-2)14-22(11-18)36-3/h6-7,9-14H,4-5,8,15-16,30H2,1-3H3,(H,31,32)(H,33,34)	YJWXCBCTPSTTMV-UHFFFAOYSA-N	468862	US10807959, Example 168	WD repeat-containing protein 5		 5.20								US Patent		10.7270/Q26Q219X		aid1804927	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468862	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468862&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146371010	441570963							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968740	COc1cc(CNC(=O)c2cc(CNC3=NCCN3)cc(c2N)-c2ccc(F)cc2C)cc(OC)c1	InChI=1S/C27H30FN5O3/c1-16-8-19(28)4-5-22(16)23-11-18(15-33-27-30-6-7-31-27)12-24(25(23)29)26(34)32-14-17-9-20(35-2)13-21(10-17)36-3/h4-5,8-13H,6-7,14-15,29H2,1-3H3,(H,32,34)(H2,30,31,33)	JQEJNYUQONTPIM-UHFFFAOYSA-N	468863	US10807959, Example 169	WD repeat-containing protein 5		 6.10								US Patent		10.7270/Q26Q219X		aid1804927	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468863	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468863&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370890	441570964							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968741	CNc1c(cc(CNC2=NCCC2)cc1-c1ccc(F)cc1C)C(=O)N(C)Cc1cc(OC)cc(OC)c1	InChI=1S/C30H35FN4O3/c1-19-11-22(31)8-9-25(19)26-14-20(17-34-28-7-6-10-33-28)15-27(29(26)32-2)30(36)35(3)18-21-12-23(37-4)16-24(13-21)38-5/h8-9,11-16,32H,6-7,10,17-18H2,1-5H3,(H,33,34)	HHDUETNFQMCWAX-UHFFFAOYSA-N	468864	US10807959, Example 170	WD repeat-containing protein 5		 19.0								US Patent		10.7270/Q26Q219X		aid1804927	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468864	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468864&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370816	441570965							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968742	CNc1c(cc(CNC2=NCCN2)cc1-c1ccc(F)cc1C)C(=O)N(C)Cc1cc(OC)cc(OC)c1	InChI=1S/C29H34FN5O3/c1-18-10-21(30)6-7-24(18)25-13-19(16-34-29-32-8-9-33-29)14-26(27(25)31-2)28(36)35(3)17-20-11-22(37-4)15-23(12-20)38-5/h6-7,10-15,31H,8-9,16-17H2,1-5H3,(H2,32,33,34)	VAICQJHQHOPZKZ-UHFFFAOYSA-N	468865	US10807959, Example 171	WD repeat-containing protein 5		 19.0								US Patent		10.7270/Q26Q219X		aid1804927	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468865	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468865&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370975	441570966							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968743	COc1cc(CNC(=O)c2cc(CNC3=NCCC3)cc(c2NC(C)=O)-c2ccc(F)cc2C)cc(OC)c1	InChI=1S/C30H33FN4O4/c1-18-10-22(31)7-8-25(18)26-13-21(16-33-28-6-5-9-32-28)14-27(29(26)35-19(2)36)30(37)34-17-20-11-23(38-3)15-24(12-20)39-4/h7-8,10-15H,5-6,9,16-17H2,1-4H3,(H,32,33)(H,34,37)(H,35,36)	WDEWZZVHPDLKGJ-UHFFFAOYSA-N	468866	US10807959, Example 172	WD repeat-containing protein 5		 2.10								US Patent		10.7270/Q26Q219X		aid1804927	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468866	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468866&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370934	441570967							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981515	CCOc1c(cc(Cn2ccoc2=N)cc1-c1cn(C)nc1C(F)(F)F)C(=O)N[C@@H](C1CC1)c1ccc(F)c(C)c1	InChI=1S/C29H29F4N5O3/c1-4-40-25-20(22-15-37(3)36-26(22)29(31,32)33)12-17(14-38-9-10-41-28(38)34)13-21(25)27(39)35-24(18-5-6-18)19-7-8-23(30)16(2)11-19/h7-13,15,18,24,34H,4-6,14H2,1-3H3,(H,35,39)/t24-/m0/s1	XUNYMFWBUYKIIF-DEOSSOPVSA-N	473311	US10844044, Example 304	WD repeat-containing protein 5		<0.100								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473311	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473311&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146455711	442073523							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981516	C[C@H](NC(=O)c1cc(Cn2ccn(C)c2=N)cc(c1)-c1ccc(F)cc1C)c1ccc(F)c(c1)C(F)(F)F	InChI=1S/C28H25F5N4O/c1-16-10-22(29)5-6-23(16)20-11-18(15-37-9-8-36(3)27(37)34)12-21(13-20)26(38)35-17(2)19-4-7-25(30)24(14-19)28(31,32)33/h4-14,17,34H,15H2,1-3H3,(H,35,38)/t17-/m0/s1	NVZGYYXYJQXBPR-KRWDZBQOSA-N	473312	US10844044, Example 31	WD repeat-containing protein 5		 0.170								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473312	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473312&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456751	442073524							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981517	CCOC(=O)\N=c1/n(C)ccn1Cc1cc(cc(c1)-c1ccc(F)nc1C)C(=O)NCc1ccc(Cl)c(Cl)c1	InChI=1S/C28H26Cl2FN5O3/c1-4-39-28(38)34-27-35(3)9-10-36(27)16-19-11-20(22-6-8-25(31)33-17(22)2)14-21(12-19)26(37)32-15-18-5-7-23(29)24(30)13-18/h5-14H,4,15-16H2,1-3H3,(H,32,37)/b34-27+	GPLLVQKJANBDJO-DNGXXSEMSA-N	473313	US10844044, Example 122	WD repeat-containing protein 5		>33.0								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473313	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473313&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146487871	442073525							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981518	CCn1cc(c(n1)C(F)(F)F)-c1cc(Cn2ccn(C)c2=N)cc(c1)C(=O)N[C@@H](C1CC1)c1ccc(F)c(F)c1	InChI=1S/C28H27F5N6O/c1-3-39-15-21(25(36-39)28(31,32)33)19-10-16(14-38-9-8-37(2)27(38)34)11-20(12-19)26(40)35-24(17-4-5-17)18-6-7-22(29)23(30)13-18/h6-13,15,17,24,34H,3-5,14H2,1-2H3,(H,35,40)/t24-/m0/s1	UGYLPQAQOHYWFG-DEOSSOPVSA-N	473224	US10844044, Example 191::US10844044, Example 213	WD repeat-containing protein 5		<0.100								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473224	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473224&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146455858	442073436							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981519	COc1cc(ccc1F)[C@@H](NC(=O)c1cc(CN2CCOC2=N)cc(c1)-c1cccnc1C(F)(F)F)C1CC1	InChI=1S/C28H26F4N4O3/c1-38-23-14-18(6-7-22(23)29)24(17-4-5-17)35-26(37)20-12-16(15-36-9-10-39-27(36)33)11-19(13-20)21-3-2-8-34-25(21)28(30,31)32/h2-3,6-8,11-14,17,24,33H,4-5,9-10,15H2,1H3,(H,35,37)/t24-/m0/s1	RNLUQWZNZCSDDV-DEOSSOPVSA-N	473315	US10844044, Example 305	WD repeat-containing protein 5		<0.100								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473315	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473315&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456430	442073526							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981520	C[C@@H](NC(=O)c1cc(Cn2ccn(C)c2=N)cc(c1)-c1ccc(F)cc1C)c1ccc(F)c(c1)C(F)(F)F	InChI=1S/C28H25F5N4O/c1-16-10-22(29)5-6-23(16)20-11-18(15-37-9-8-36(3)27(37)34)12-21(13-20)26(38)35-17(2)19-4-7-25(30)24(14-19)28(31,32)33/h4-14,17,34H,15H2,1-3H3,(H,35,38)/t17-/m1/s1	NVZGYYXYJQXBPR-QGZVFWFLSA-N	473316	US10844044, Example 32	WD repeat-containing protein 5		 0.880								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473316	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473316&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456804	442073527							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981521	Cc1cc(ccc1F)[C@@H](NC(=O)c1cc(Cn2ccn(C)c2=N)cc(c1)-c1cncnc1C(F)(F)F)C1CC1	InChI=1S/C28H26F4N6O/c1-16-9-19(5-6-23(16)29)24(18-3-4-18)36-26(39)21-11-17(14-38-8-7-37(2)27(38)33)10-20(12-21)22-13-34-15-35-25(22)28(30,31)32/h5-13,15,18,24,33H,3-4,14H2,1-2H3,(H,36,39)/t24-/m0/s1	ULKYTQGCBVXHFR-DEOSSOPVSA-N	473317	US10844044, Example 123::US10844044, Example 125	WD repeat-containing protein 5		 0.180								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473317	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473317&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146455728	442073528							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981522	CCn1cc(c(n1)C(F)(F)F)-c1cc(Cn2ccn(C)c2=N)cc(c1)C(=O)N[C@@H](C1CC1)c1ccc(F)c(Cl)c1	InChI=1S/C28H27ClF4N6O/c1-3-39-15-21(25(36-39)28(31,32)33)19-10-16(14-38-9-8-37(2)27(38)34)11-20(12-19)26(40)35-24(17-4-5-17)18-6-7-23(30)22(29)13-18/h6-13,15,17,24,34H,3-5,14H2,1-2H3,(H,35,40)/t24-/m0/s1	UVTOCBFVYBUDLA-DEOSSOPVSA-N	473318	US10844044, Example 214	WD repeat-containing protein 5		<0.100								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473318	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473318&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146487974	442073529							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981523	COc1cc(ccc1F)[C@@H](NC(=O)c1cc(Cn2ccoc2=N)cc(c1)-c1cn(C)nc1C(F)(F)F)C1CC1	InChI=1S/C27H25F4N5O3/c1-35-14-20(24(34-35)27(29,30)31)18-9-15(13-36-7-8-39-26(36)32)10-19(11-18)25(37)33-23(16-3-4-16)17-5-6-21(28)22(12-17)38-2/h5-12,14,16,23,32H,3-4,13H2,1-2H3,(H,33,37)/t23-/m0/s1	QSWDBKDWGTVXGJ-QHCPKHFHSA-N	473319	US10844044, Example 306	WD repeat-containing protein 5		<0.100								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473319	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473319&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146488079	442073530							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981524	Cc1cc(CNC(=O)c2cc(Cn3ccn(C)c3=N)cc(c2)-c2c(C)ccc3[nH]ncc23)ccc1Cl	InChI=1S/C28H27ClN6O/c1-17-4-7-25-23(15-32-33-25)26(17)21-11-20(16-35-9-8-34(3)28(35)30)12-22(13-21)27(36)31-14-19-5-6-24(29)18(2)10-19/h4-13,15,30H,14,16H2,1-3H3,(H,31,36)(H,32,33)	BEFXUTBVOQXEDD-UHFFFAOYSA-N	473320	US10844044, Example 33	WD repeat-containing protein 5		 0.990								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473320	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473320&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456211	442073531							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981525	C[C@H](NC(=O)c1cc(Cn2ccn(C)c2=N)cc(c1)-c1cccnc1C(F)(F)F)c1ccc(F)c(Cl)c1	InChI=1S/C26H22ClF4N5O/c1-15(17-5-6-22(28)21(27)13-17)34-24(37)19-11-16(14-36-9-8-35(2)25(36)32)10-18(12-19)20-4-3-7-33-23(20)26(29,30)31/h3-13,15,32H,14H2,1-2H3,(H,34,37)/t15-/m0/s1	ILFSHERPUGGODW-HNNXBMFYSA-N	473321	US10844044, Example 124	WD repeat-containing protein 5		 1.000								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473321	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473321&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146457572	442073532							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981526	CCn1cc(c(n1)C(F)(F)F)-c1cc(CN2CCN(C)C2=N)cc(c1)C(=O)N[C@@H](C1CC1)c1ccc(F)c(C)c1	InChI=1S/C29H32F4N6O/c1-4-39-16-23(26(36-39)29(31,32)33)21-12-18(15-38-10-9-37(3)28(38)34)13-22(14-21)27(40)35-25(19-5-6-19)20-7-8-24(30)17(2)11-20/h7-8,11-14,16,19,25,34H,4-6,9-10,15H2,1-3H3,(H,35,40)/t25-/m0/s1	QJKWIJZWGMXZCI-VWLOTQADSA-N	473322	US10844044, Example 215	WD repeat-containing protein 5		<0.100								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473322	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473322&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456216	442073533							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981527	COc1cc(CNC(=O)c2cc(Cn3ccsc3=N)cc(c2)-c2ccc(F)cc2C)cc(OC)c1	InChI=1S/C27H26FN3O3S/c1-17-8-22(28)4-5-25(17)20-9-19(16-31-6-7-35-27(31)29)10-21(13-20)26(32)30-15-18-11-23(33-2)14-24(12-18)34-3/h4-14,29H,15-16H2,1-3H3,(H,30,32)	CDTWRLDBXMPKLF-UHFFFAOYSA-N	473323	US10844044, Example 307	WD repeat-containing protein 5		 0.950								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473323	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473323&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456635	442073534							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981528	COc1cc(CN(C)C(=O)c2cc(Cn3ccn(C)c3=N)cc(c2)-c2c(C)ccc3[nH]ncc23)cc(OC)c1	InChI=1S/C30H32N6O3/c1-19-6-7-27-26(16-32-33-27)28(19)22-10-20(18-36-9-8-34(2)30(36)31)11-23(14-22)29(37)35(3)17-21-12-24(38-4)15-25(13-21)39-5/h6-16,31H,17-18H2,1-5H3,(H,32,33)	IQTSAGUPXNPHHI-UHFFFAOYSA-N	473324	US10844044, Example 34	WD repeat-containing protein 5		 16.0								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473324	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473324&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456651	442073535							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981529	Cc1cc(ccc1F)[C@@H](NC(=O)c1cc(Cn2ccn(C)c2=N)cc(c1)-c1cncnc1C(F)(F)F)C1CC1	InChI=1S/C28H26F4N6O/c1-16-9-19(5-6-23(16)29)24(18-3-4-18)36-26(39)21-11-17(14-38-8-7-37(2)27(38)33)10-20(12-21)22-13-34-15-35-25(22)28(30,31)32/h5-13,15,18,24,33H,3-4,14H2,1-2H3,(H,36,39)/t24-/m0/s1	ULKYTQGCBVXHFR-DEOSSOPVSA-N	473317	US10844044, Example 123::US10844044, Example 125	WD repeat-containing protein 5		<0.100								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473317	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473317&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146455728	442073528							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981530	CC(C)n1cc(c(n1)C(F)(F)F)-c1cc(CN2CCN(C)C2=N)cc(c1)C(=O)N[C@@H](C1CC1)c1ccc(F)c(F)c1	InChI=1S/C29H31F5N6O/c1-16(2)40-15-22(26(37-40)29(32,33)34)20-10-17(14-39-9-8-38(3)28(39)35)11-21(12-20)27(41)36-25(18-4-5-18)19-6-7-23(30)24(31)13-19/h6-7,10-13,15-16,18,25,35H,4-5,8-9,14H2,1-3H3,(H,36,41)/t25-/m0/s1	CQZFCQMZIORWIT-VWLOTQADSA-N	473326	US10844044, Example 216	WD repeat-containing protein 5		<0.100								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473326	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473326&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456744	442073536							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981531	COc1cc(CNC(=O)c2cc(CN3CCSC3=N)cc(c2)-c2ccc(F)cc2C)cc(OC)c1	InChI=1S/C27H28FN3O3S/c1-17-8-22(28)4-5-25(17)20-9-19(16-31-6-7-35-27(31)29)10-21(13-20)26(32)30-15-18-11-23(33-2)14-24(12-18)34-3/h4-5,8-14,29H,6-7,15-16H2,1-3H3,(H,30,32)	MCQUKMLWJYVCCV-UHFFFAOYSA-N	473327	US10844044, Example 308	WD repeat-containing protein 5		 0.450								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473327	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473327&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456137	442073537							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981532	COc1cc(CNC(=O)c2cc(Cn3ccn(C)c3=N)cc(c2)-c2c(C)ccc3[nH]ncc23)cc(OC)c1	InChI=1S/C29H30N6O3/c1-18-5-6-26-25(16-32-33-26)27(18)21-9-20(17-35-8-7-34(2)29(35)30)10-22(13-21)28(36)31-15-19-11-23(37-3)14-24(12-19)38-4/h5-14,16,30H,15,17H2,1-4H3,(H,31,36)(H,32,33)	UUICOEPTKOOGCS-UHFFFAOYSA-N	473328	US10844044, Example 35	WD repeat-containing protein 5		 1.30								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473328	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473328&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146455831	442073538							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981533	C[C@H](NC(=O)c1cc(Cn2ccn(C)c2=N)cc(c1)-c1cccnc1C(F)(F)F)c1ccc(cc1)C(F)(F)F	InChI=1S/C27H23F6N5O/c1-16(18-5-7-21(8-6-18)26(28,29)30)36-24(39)20-13-17(15-38-11-10-37(2)25(38)34)12-19(14-20)22-4-3-9-35-23(22)27(31,32)33/h3-14,16,34H,15H2,1-2H3,(H,36,39)/t16-/m0/s1	DLFNCTXJALLRNT-INIZCTEOSA-N	473329	US10844044, Example 126	WD repeat-containing protein 5		 2.50								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473329	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473329&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146455867	442073539							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981534	Cc1cc(ccc1F)[C@@H](NC(=O)c1cc(Cn2ccn(C)c2=N)cc(c1)C1(CC1)C(F)(F)F)C1CC1	InChI=1S/C27H28F4N4O/c1-16-11-19(5-6-22(16)28)23(18-3-4-18)33-24(36)20-12-17(15-35-10-9-34(2)25(35)32)13-21(14-20)26(7-8-26)27(29,30)31/h5-6,9-14,18,23,32H,3-4,7-8,15H2,1-2H3,(H,33,36)/t23-/m0/s1	LUALJLUXAUYSKE-QHCPKHFHSA-N	473330	US10844044, Example 217	WD repeat-containing protein 5		<0.100								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473330	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473330&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146455717	442073540							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981535	FC(F)Oc1cc(F)ccc1-c1cc(CN2CCSC2=N)cc(c1)C(=O)N[C@@H](C1CC1)c1ccc(Cl)c(Cl)c1	InChI=1S/C28H24Cl2F3N3O2S/c29-22-6-3-17(12-23(22)30)25(16-1-2-16)35-26(37)19-10-15(14-36-7-8-39-28(36)34)9-18(11-19)21-5-4-20(31)13-24(21)38-27(32)33/h3-6,9-13,16,25,27,34H,1-2,7-8,14H2,(H,35,37)/t25-/m0/s1	FNUUGBOTXQZDNE-VWLOTQADSA-N	473331	US10844044, Example 309	WD repeat-containing protein 5		 0.770								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473331	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473331&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146457669	442073541							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981536	CN1C(=O)CN(Cc2cc(cc(c2)-c2ccc(F)nc2C)C(=O)NCc2ccc(Cl)c(Cl)c2)C1=N	InChI=1S/C25H22Cl2FN5O2/c1-14-19(4-6-22(28)31-14)17-7-16(12-33-13-23(34)32(2)25(33)29)8-18(10-17)24(35)30-11-15-3-5-20(26)21(27)9-15/h3-10,29H,11-13H2,1-2H3,(H,30,35)	JMUJODDTICNHAB-UHFFFAOYSA-N	473332	US10844044, Example 36	WD repeat-containing protein 5		 8.50								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473332	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473332&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456378	442073542							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981537	Cc1cc(ccc1F)[C@@H](NC(=O)c1cc(Cn2ccn(C)c2=N)cc(c1)-c1cccnc1OC(F)F)C1CC1	InChI=1S/C29H28F3N5O2/c1-17-12-20(7-8-24(17)30)25(19-5-6-19)35-26(38)22-14-18(16-37-11-10-36(2)29(37)33)13-21(15-22)23-4-3-9-34-27(23)39-28(31)32/h3-4,7-15,19,25,28,33H,5-6,16H2,1-2H3,(H,35,38)/t25-/m0/s1	IGYWASSPIALFMK-VWLOTQADSA-N	473333	US10844044, Example 127	WD repeat-containing protein 5		 0.210								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473333	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473333&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146455719	442073543							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981538	Cc1cc(ncc1F)[C@@H](NC(=O)c1cc(Cn2ccn(C)c2=N)cc(c1)C1(CC1)C(F)(F)F)C1CC1	InChI=1S/C26H27F4N5O/c1-15-9-21(32-13-20(15)27)22(17-3-4-17)33-23(36)18-10-16(14-35-8-7-34(2)24(35)31)11-19(12-18)25(5-6-25)26(28,29)30/h7-13,17,22,31H,3-6,14H2,1-2H3,(H,33,36)/t22-/m0/s1	HBWJKRSHEIVLCP-QFIPXVFZSA-N	473334	US10844044, Example 218	WD repeat-containing protein 5		<0.100								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473334	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473334&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146455812	442073544							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981539	Cn1cc(c(n1)C(F)(F)F)-c1cc(CN2CCSC2=N)cc(c1)C(=O)N[C@@H](C1CC1)c1ccc(Cl)c(Cl)c1	InChI=1S/C26H24Cl2F3N5OS/c1-35-13-19(23(34-35)26(29,30)31)17-8-14(12-36-6-7-38-25(36)32)9-18(10-17)24(37)33-22(15-2-3-15)16-4-5-20(27)21(28)11-16/h4-5,8-11,13,15,22,32H,2-3,6-7,12H2,1H3,(H,33,37)/t22-/m0/s1	GIAJJPLQOAXLKE-QFIPXVFZSA-N	473335	US10844044, Example 310	WD repeat-containing protein 5		<0.100								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473335	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473335&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456243	442073545							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981540	Cc1ccnc(c1)C(NC(=O)c1cc(Cn2ccn(C)c2=N)cc(c1)-c1cccnc1C)C1CC1	InChI=1S/C28H30N6O/c1-18-8-10-31-25(13-18)26(21-6-7-21)32-27(35)23-15-20(17-34-12-11-33(3)28(34)29)14-22(16-23)24-5-4-9-30-19(24)2/h4-5,8-16,21,26,29H,6-7,17H2,1-3H3,(H,32,35)	ROCPKWMXNIWONN-UHFFFAOYSA-N	473336	US10844044, Example 37	WD repeat-containing protein 5		 0.400								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473336	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473336&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146455903	442073546							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981541	Cn1ccn(Cc2cc(cc(c2)-c2cccnc2C(F)(F)F)C(=O)N[C@@H](C2CC2)c2ccc(F)cn2)c1=N	InChI=1S/C27H24F4N6O/c1-36-9-10-37(26(36)32)15-16-11-18(21-3-2-8-33-24(21)27(29,30)31)13-19(12-16)25(38)35-23(17-4-5-17)22-7-6-20(28)14-34-22/h2-3,6-14,17,23,32H,4-5,15H2,1H3,(H,35,38)/t23-/m0/s1	NVCZUETUGSJFFU-QHCPKHFHSA-N	473337	US10844044, Example 128	WD repeat-containing protein 5		 23.0								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473337	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473337&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456012	442073547							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981542	CN1CCN(Cc2cc(cc(c2)-c2cccnc2C(F)(F)F)C(=O)N[C@@H](C2CC2)c2ccc(F)c(Cl)c2)C1=N	InChI=1S/C28H26ClF4N5O/c1-37-9-10-38(27(37)34)15-16-11-19(21-3-2-8-35-25(21)28(31,32)33)13-20(12-16)26(39)36-24(17-4-5-17)18-6-7-23(30)22(29)14-18/h2-3,6-8,11-14,17,24,34H,4-5,9-10,15H2,1H3,(H,36,39)/t24-/m0/s1	MPHJLGJFDVZKQQ-DEOSSOPVSA-N	473338	US10844044, Example 219	WD repeat-containing protein 5		<0.100								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473338	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473338&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146455745	442073548							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981543	FC(F)(F)c1ncccc1-c1cc(CN2CCSC2=N)cc(c1)C(=O)N[C@@H](C1CC1)c1ccc(Cl)c(Cl)c1	InChI=1S/C27H23Cl2F3N4OS/c28-21-6-5-17(13-22(21)29)23(16-3-4-16)35-25(37)19-11-15(14-36-8-9-38-26(36)33)10-18(12-19)20-2-1-7-34-24(20)27(30,31)32/h1-2,5-7,10-13,16,23,33H,3-4,8-9,14H2,(H,35,37)/t23-/m0/s1	UGGDRGQJZKQVLY-QHCPKHFHSA-N	473339	US10844044, Example 311	WD repeat-containing protein 5		 1.49								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473339	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473339&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			151998860	442073549							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981544	Cc1cc(CNC(=O)c2cc(Cn3ccn(C)c3=N)cc(c2)-c2cccnc2C)ncn1	InChI=1S/C24H25N7O/c1-16-9-21(29-15-28-16)13-27-23(32)20-11-18(14-31-8-7-30(3)24(31)25)10-19(12-20)22-5-4-6-26-17(22)2/h4-12,15,25H,13-14H2,1-3H3,(H,27,32)	MAEFIYVEVAYABC-UHFFFAOYSA-N	473340	US10844044, Example 38	WD repeat-containing protein 5		 3.70								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473340	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473340&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456183	442073550							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981545	Cn1ccn(Cc2cc(CN[C@H]3CCc4cc(F)ccc34)cc(c2)-c2cccnc2C(F)(F)F)c1=N	InChI=1S/C27H25F4N5/c1-35-9-10-36(26(35)32)16-18-11-17(15-34-24-7-4-19-14-21(28)5-6-22(19)24)12-20(13-18)23-3-2-8-33-25(23)27(29,30)31/h2-3,5-6,8-14,24,32,34H,4,7,15-16H2,1H3/t24-/m0/s1	DVNIUENBLAEGCP-DEOSSOPVSA-N	473341	US10844044, Example 129	WD repeat-containing protein 5		>33.0								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473341	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473341&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146487901	442073551							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981546	Cc1cccc(c1)C1(CCC1)NC(=O)c1cc(Cn2ccn(C)c2=N)cc(c1)-c1cn(C)nc1C(F)(F)F	InChI=1S/C28H29F3N6O/c1-18-6-4-7-22(12-18)27(8-5-9-27)33-25(38)21-14-19(16-37-11-10-35(2)26(37)32)13-20(15-21)23-17-36(3)34-24(23)28(29,30)31/h4,6-7,10-15,17,32H,5,8-9,16H2,1-3H3,(H,33,38)	RPRGZZMBIJZKBP-UHFFFAOYSA-N	473342	US10844044, Example 220	WD repeat-containing protein 5		<0.100								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473342	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473342&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146455752	442073552							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981547	CCn1cc(c(n1)C(F)(F)F)-c1cc(CN2CCSC2=N)cc(c1)C(=O)N[C@@H](C1CC1)c1ccc(F)c(C)c1	InChI=1S/C28H29F4N5OS/c1-3-37-15-22(25(35-37)28(30,31)32)20-11-17(14-36-8-9-39-27(36)33)12-21(13-20)26(38)34-24(18-4-5-18)19-6-7-23(29)16(2)10-19/h6-7,10-13,15,18,24,33H,3-5,8-9,14H2,1-2H3,(H,34,38)/t24-/m0/s1	BULASWCVLAEFGR-DEOSSOPVSA-N	473343	US10844044, Example 312	WD repeat-containing protein 5		<0.100								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473343	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473343&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456496	442073553							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981548	Cc1ncccc1-c1cc(Cn2ccn(C)c2=N)cc(c1)C(=O)NC(C1CC1)C1CC1	InChI=1S/C25H29N5O/c1-16-22(4-3-9-27-16)20-12-17(15-30-11-10-29(2)25(30)26)13-21(14-20)24(31)28-23(18-5-6-18)19-7-8-19/h3-4,9-14,18-19,23,26H,5-8,15H2,1-2H3,(H,28,31)	DOIBVSFRFPYGAI-UHFFFAOYSA-N	473344	US10844044, Example 39	WD repeat-containing protein 5		 17.0								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473344	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473344&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146455806	442073554							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981549	C[C@H](NC(=O)c1cc(Cn2ccn(C)c2=N)cc(c1)-c1cccnc1C(F)(F)F)c1ncc(F)cn1	InChI=1S/C24H21F4N7O/c1-14(21-31-11-18(25)12-32-21)33-22(36)17-9-15(13-35-7-6-34(2)23(35)29)8-16(10-17)19-4-3-5-30-20(19)24(26,27)28/h3-12,14,29H,13H2,1-2H3,(H,33,36)/t14-/m0/s1	MECOIQULWXKNMK-AWEZNQCLSA-N	473345	US10844044, Example 130	WD repeat-containing protein 5		>33.0								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473345	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473345&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456179	442073555							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981550	COc1cc(ncc1F)[C@@H](NC(=O)c1cc(Cn2ccn(C)c2=N)cc(c1)-c1cn(C)nc1C(F)(F)F)C1CC1	InChI=1S/C27H27F4N7O2/c1-36-6-7-38(26(36)32)13-15-8-17(19-14-37(2)35-24(19)27(29,30)31)10-18(9-15)25(39)34-23(16-4-5-16)21-11-22(40-3)20(28)12-33-21/h6-12,14,16,23,32H,4-5,13H2,1-3H3,(H,34,39)/t23-/m0/s1	JTMFUPYUNBGDPN-QHCPKHFHSA-N	473346	US10844044, Example 221	WD repeat-containing protein 5		<0.100								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473346	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473346&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146457359	442073556							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981551	CC(C)Cn1cc(c(n1)C(F)(F)F)-c1cc(CN2CCSC2=N)cc(c1)C(=O)N[C@@H](C1CC1)c1ccc(F)c(C)c1	InChI=1S/C30H33F4N5OS/c1-17(2)14-39-16-24(27(37-39)30(32,33)34)22-11-19(15-38-8-9-41-29(38)35)12-23(13-22)28(40)36-26(20-4-5-20)21-6-7-25(31)18(3)10-21/h6-7,10-13,16-17,20,26,35H,4-5,8-9,14-15H2,1-3H3,(H,36,40)/t26-/m0/s1	YITHLLZIAGVCPM-SANMLTNESA-N	473347	US10844044, Example 313	WD repeat-containing protein 5		 1.20								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473347	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473347&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146455796	442073557							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981552	Cc1ncccc1-c1cc(Cn2ccn(C)c2=N)cc(c1)C(=O)NCc1cncnc1	InChI=1S/C23H23N7O/c1-16-21(4-3-5-27-16)19-8-17(14-30-7-6-29(2)23(30)24)9-20(10-19)22(31)28-13-18-11-25-15-26-12-18/h3-12,15,24H,13-14H2,1-2H3,(H,28,31)	RXQLZDWVIQHJDO-UHFFFAOYSA-N	473348	US10844044, Example 40	WD repeat-containing protein 5		 133								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473348	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473348&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146488005	442073558							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981553	Cc1cc(ccc1F)[C@@H](NC(=O)c1cc(Cn2ccn(C)c2=N)cc(c1F)-c1cccnc1C(F)(F)F)C1CC1	InChI=1S/C29H26F5N5O/c1-16-12-19(7-8-23(16)30)25(18-5-6-18)37-27(40)22-14-17(15-39-11-10-38(2)28(39)35)13-21(24(22)31)20-4-3-9-36-26(20)29(32,33)34/h3-4,7-14,18,25,35H,5-6,15H2,1-2H3,(H,37,40)/t25-/m0/s1	MIZYXICOJODQRY-VWLOTQADSA-N	473349	US10844044, Example 131	WD repeat-containing protein 5		<0.100								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473349	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473349&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146455904	442073559							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981554	Cc1cc(ccc1F)[C@@H](NC(=O)c1cc(Cn2ccn(C)c2=N)cc(c1)N1CCC[C@@H]1C(F)(F)F)C1CC1	InChI=1S/C28H31F4N5O/c1-17-12-20(7-8-23(17)29)25(19-5-6-19)34-26(38)21-13-18(16-36-11-10-35(2)27(36)33)14-22(15-21)37-9-3-4-24(37)28(30,31)32/h7-8,10-15,19,24-25,33H,3-6,9,16H2,1-2H3,(H,34,38)/t24-,25+/m1/s1	UKWBUCJBBQOGSR-RPBOFIJWSA-N	473350	US10844044, Example 222	WD repeat-containing protein 5		 0.330								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473350	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473350&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456266	442073560							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981555	Cc1cc(ccc1F)[C@@H](NC(=O)c1cc(CN2CCSC2=N)cc(c1)-c1cn(nc1C(F)(F)F)C1CCCC1)C1CC1	InChI=1S/C31H33F4N5OS/c1-18-12-21(8-9-26(18)32)27(20-6-7-20)37-29(41)23-14-19(16-39-10-11-42-30(39)36)13-22(15-23)25-17-40(24-4-2-3-5-24)38-28(25)31(33,34)35/h8-9,12-15,17,20,24,27,36H,2-7,10-11,16H2,1H3,(H,37,41)/t27-/m0/s1	RBPBSWXTVDBOLQ-MHZLTWQESA-N	473351	US10844044, Example 314	WD repeat-containing protein 5		 4.00								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473351	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473351&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456207	442073561							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981556	COc1cc(CNC(=O)c2cc(Cn3ccn(C)c3=N)cc(c2)-c2cccnc2C)ccn1	InChI=1S/C25H26N6O2/c1-17-22(5-4-7-27-17)20-11-19(16-31-10-9-30(2)25(31)26)12-21(14-20)24(32)29-15-18-6-8-28-23(13-18)33-3/h4-14,26H,15-16H2,1-3H3,(H,29,32)	IWYMVXNIEXGOMP-UHFFFAOYSA-N	473352	US10844044, Example 41	WD repeat-containing protein 5		 33.0								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473352	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473352&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146455839	442073562							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981557	Cc1ccnc(c1)[C@@H](NC(=O)c1cc(Cn2ccn(C)c2=N)cc(c1F)-c1cccnc1C(F)(F)F)C1CC1	InChI=1S/C28H26F4N6O/c1-16-7-9-34-22(12-16)24(18-5-6-18)36-26(39)21-14-17(15-38-11-10-37(2)27(38)33)13-20(23(21)29)19-4-3-8-35-25(19)28(30,31)32/h3-4,7-14,18,24,33H,5-6,15H2,1-2H3,(H,36,39)/t24-/m0/s1	XIMOTMRTSPVYQT-DEOSSOPVSA-N	473353	US10844044, Example 132	WD repeat-containing protein 5		 0.130								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473353	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473353&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146457381	442073563							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981558	Cc1cc(ccc1F)[C@@H](NC(=O)c1cc(Cn2ccn(C)c2=N)cc(c1)N1CCC[C@H]1C(F)(F)F)C1CC1	InChI=1S/C28H31F4N5O/c1-17-12-20(7-8-23(17)29)25(19-5-6-19)34-26(38)21-13-18(16-36-11-10-35(2)27(36)33)14-22(15-21)37-9-3-4-24(37)28(30,31)32/h7-8,10-15,19,24-25,33H,3-6,9,16H2,1-2H3,(H,34,38)/t24-,25-/m0/s1	UKWBUCJBBQOGSR-DQEYMECFSA-N	473354	US10844044, Example 223	WD repeat-containing protein 5		 1.30								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473354	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473354&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456465	442073564							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981559	Cc1cc(ccc1F)[C@@H](NC(=O)c1cc(CN2CCCSC2=N)cc(c1)-c1cccnc1C(F)(F)F)C1CC1	InChI=1S/C29H28F4N4OS/c1-17-12-20(7-8-24(17)30)25(19-5-6-19)36-27(38)22-14-18(16-37-10-3-11-39-28(37)34)13-21(15-22)23-4-2-9-35-26(23)29(31,32)33/h2,4,7-9,12-15,19,25,34H,3,5-6,10-11,16H2,1H3,(H,36,38)/t25-/m0/s1	XYNPOHAKZWDPSU-VWLOTQADSA-N	473356	US10844044, Example 315	WD repeat-containing protein 5		 1.000								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473356	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473356&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146455968	442073566							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981560	Cc1cc(C)nc(CNC(=O)c2cc(Cn3ccn(C)c3=N)cc(c2)-c2cccnc2C)n1	InChI=1S/C25H27N7O/c1-16-10-17(2)30-23(29-16)14-28-24(33)21-12-19(15-32-9-8-31(4)25(32)26)11-20(13-21)22-6-5-7-27-18(22)3/h5-13,26H,14-15H2,1-4H3,(H,28,33)	DCMVVMSALSWLFY-UHFFFAOYSA-N	473357	US10844044, Example 42	WD repeat-containing protein 5		 10.00								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473357	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473357&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146455923	442073567							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981561	COc1cc(CNC(=O)c2cc(Cn3ccn(CC4CC4)c3=N)cc(c2)-c2ccc(F)cc2C)cc(OC)c1	InChI=1S/C31H33FN4O3/c1-20-10-26(32)6-7-29(20)24-11-23(19-36-9-8-35(31(36)33)18-21-4-5-21)12-25(15-24)30(37)34-17-22-13-27(38-2)16-28(14-22)39-3/h6-16,21,33H,4-5,17-19H2,1-3H3,(H,34,37)	YLUYADFVQAOAPF-UHFFFAOYSA-N	473358	US10844044, Example 133::US10844044, Example 134	WD repeat-containing protein 5		>33.0								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473358	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473358&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146457876	442073568							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981562	Cc1nccn1-c1cc(Cn2ccn(C)c2=N)cc(c1)C(=O)N[C@@H](C1CC1)c1ccc(F)c(C)c1	InChI=1S/C27H29FN6O/c1-17-12-21(6-7-24(17)28)25(20-4-5-20)31-26(35)22-13-19(16-33-11-10-32(3)27(33)29)14-23(15-22)34-9-8-30-18(34)2/h6-15,20,25,29H,4-5,16H2,1-3H3,(H,31,35)/t25-/m0/s1	XQXQBRUTYDCGSF-VWLOTQADSA-N	473359	US10844044, Example 224	WD repeat-containing protein 5		 0.140								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473359	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473359&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146457306	442073569							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981563	Cc1cc(ccc1F)[C@@H](NC(=O)c1cc(CN2CCSC2=N)cc(c1)-c1ccc(F)cc1C#N)C1CC1	InChI=1S/C29H26F2N4OS/c1-17-10-20(4-7-26(17)31)27(19-2-3-19)34-28(36)22-12-18(16-35-8-9-37-29(35)33)11-21(13-22)25-6-5-24(30)14-23(25)15-32/h4-7,10-14,19,27,33H,2-3,8-9,16H2,1H3,(H,34,36)/t27-/m0/s1	GNWJGLNVEIKWEO-MHZLTWQESA-N	473360	US10844044, Example 316	WD repeat-containing protein 5		 0.910								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473360	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473360&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146455837	442073570							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981564	COc1ccnc(CNC(=O)c2cc(Cn3ccn(C)c3=N)cc(c2)-c2cccnc2C)c1	InChI=1S/C25H26N6O2/c1-17-23(5-4-7-27-17)19-11-18(16-31-10-9-30(2)25(31)26)12-20(13-19)24(32)29-15-21-14-22(33-3)6-8-28-21/h4-14,26H,15-16H2,1-3H3,(H,29,32)	RJTPWXYKNYXXCR-UHFFFAOYSA-N	473361	US10844044, Example 43	WD repeat-containing protein 5		 8423								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473361	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473361&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456036	442073571							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981565	COc1cc(CNC(=O)c2cc(Cn3ccn(CC4CC4)c3=N)cc(c2)-c2ccc(F)cc2C)cc(OC)c1	InChI=1S/C31H33FN4O3/c1-20-10-26(32)6-7-29(20)24-11-23(19-36-9-8-35(31(36)33)18-21-4-5-21)12-25(15-24)30(37)34-17-22-13-27(38-2)16-28(14-22)39-3/h6-16,21,33H,4-5,17-19H2,1-3H3,(H,34,37)	YLUYADFVQAOAPF-UHFFFAOYSA-N	473358	US10844044, Example 133::US10844044, Example 134	WD repeat-containing protein 5		 38.0								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473358	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473358&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146457876	442073568							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981566	CCn1cc(c(C)n1)-c1cc(Cn2ccn(C)c2=N)cc(c1)C(=O)N[C@@H](C1CC1)c1ccc(F)c(C)c1	InChI=1S/C29H33FN6O/c1-5-36-17-25(19(3)33-36)23-13-20(16-35-11-10-34(4)29(35)31)14-24(15-23)28(37)32-27(21-6-7-21)22-8-9-26(30)18(2)12-22/h8-15,17,21,27,31H,5-7,16H2,1-4H3,(H,32,37)/t27-/m0/s1	HSEMHGVCDWCOFF-MHZLTWQESA-N	473363	US10844044, Example 225	WD repeat-containing protein 5		<0.100								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473363	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473363&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146455852	442073572							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981567	Fc1cnc(-c2cc(CN3CCSC3=N)cc(c2)C(=O)N[C@@H](C2CC2)c2ccc(Cl)c(Cl)c2)c(c1)C(F)(F)F	InChI=1S/C27H22Cl2F4N4OS/c28-21-4-3-16(10-22(21)29)23(15-1-2-15)36-25(38)18-8-14(13-37-5-6-39-26(37)34)7-17(9-18)24-20(27(31,32)33)11-19(30)12-35-24/h3-4,7-12,15,23,34H,1-2,5-6,13H2,(H,36,38)/t23-/m0/s1	WOSZGYONPOLALF-QHCPKHFHSA-N	473364	US10844044, Example 317	WD repeat-containing protein 5		 0.280								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473364	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473364&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146455885	442073573							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981568	Cc1ncccc1-c1cc(Cn2ccn(C)c2=N)cc(c1)C(=O)NCc1ncc(Cl)cn1	InChI=1S/C23H22ClN7O/c1-15-20(4-3-5-26-15)17-8-16(14-31-7-6-30(2)23(31)25)9-18(10-17)22(32)29-13-21-27-11-19(24)12-28-21/h3-12,25H,13-14H2,1-2H3,(H,29,32)	NGHNHTJDGLSQGM-UHFFFAOYSA-N	473365	US10844044, Example 44	WD repeat-containing protein 5		 9.20								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473365	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473365&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456279	442073574							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981569	Cc1cc(ccc1F)[C@@H](NC(=O)c1cc(Cn2ccn(C)c2=N)cc(c1)-c1cccnc1OCC(F)(F)F)C1CC1	InChI=1S/C30H29F4N5O2/c1-18-12-21(7-8-25(18)31)26(20-5-6-20)37-27(40)23-14-19(16-39-11-10-38(2)29(39)35)13-22(15-23)24-4-3-9-36-28(24)41-17-30(32,33)34/h3-4,7-15,20,26,35H,5-6,16-17H2,1-2H3,(H,37,40)/t26-/m0/s1	BIDWMLNMDVPPLD-SANMLTNESA-N	473366	US10844044, Example 135	WD repeat-containing protein 5		 0.830								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473366	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473366&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146455874	442073575							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981570	C[C@@H]1CCCN1c1cc(Cn2ccn(C)c2=N)cc(c1)C(=O)N[C@@H](C1CC1)c1ccc(F)c(C)c1	InChI=1S/C28H34FN5O/c1-18-13-22(8-9-25(18)29)26(21-6-7-21)31-27(35)23-14-20(17-33-12-11-32(3)28(33)30)15-24(16-23)34-10-4-5-19(34)2/h8-9,11-16,19,21,26,30H,4-7,10,17H2,1-3H3,(H,31,35)/t19-,26+/m1/s1	MMPUFGJSZCUYAD-BCHFMIIMSA-N	473367	US10844044, Example 226	WD repeat-containing protein 5		 7.10								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473367	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473367&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456807	442073576							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968744	COc1cc(CNC(=O)c2cc(CNC3=NCCN3)cc(c2NC(C)=O)-c2ccc(F)cc2C)cc(OC)c1	InChI=1S/C29H32FN5O4/c1-17-9-21(30)5-6-24(17)25-12-20(16-34-29-31-7-8-32-29)13-26(27(25)35-18(2)36)28(37)33-15-19-10-22(38-3)14-23(11-19)39-4/h5-6,9-14H,7-8,15-16H2,1-4H3,(H,33,37)(H,35,36)(H2,31,32,34)	CXUFMXYKXOKBDH-UHFFFAOYSA-N	468867	US10807959, Example 173	WD repeat-containing protein 5		 7.20								US Patent		10.7270/Q26Q219X		aid1804927	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468867	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468867&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370733	441570968							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968745	Clc1cc(Cl)cc(CNC(=O)c2cccc(CNC3=NCCN3)c2)c1	InChI=1S/C18H18Cl2N4O/c19-15-7-13(8-16(20)9-15)11-23-17(25)14-3-1-2-12(6-14)10-24-18-21-4-5-22-18/h1-3,6-9H,4-5,10-11H2,(H,23,25)(H2,21,22,24)	AASGICFZYTUAEO-UHFFFAOYSA-N	468868	US10807959, Example B1	WD repeat-containing protein 5		 18.0								US Patent		10.7270/Q26Q219X		aid1804926	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468868	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468868&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370964	441570969							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968746	CC(C)N(Cc1cccc(Cl)c1)C(=O)c1cccc(CNC2=NCCN2)c1	InChI=1S/C21H25ClN4O/c1-15(2)26(14-17-6-4-8-19(22)12-17)20(27)18-7-3-5-16(11-18)13-25-21-23-9-10-24-21/h3-8,11-12,15H,9-10,13-14H2,1-2H3,(H2,23,24,25)	GCNIMPRJCBTIII-UHFFFAOYSA-N	468869	US10807959, Example B2	WD repeat-containing protein 5		 400								US Patent		10.7270/Q26Q219X		aid1804926	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468869	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468869&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370854	441570970							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968747	Clc1ccc(CNC(=O)c2cccc(CNC3=NCCN3)c2)cc1Cl	InChI=1S/C18H18Cl2N4O/c19-15-5-4-13(9-16(15)20)10-23-17(25)14-3-1-2-12(8-14)11-24-18-21-6-7-22-18/h1-5,8-9H,6-7,10-11H2,(H,23,25)(H2,21,22,24)	DOIDLJPFNQHXFM-UHFFFAOYSA-N	468870	US10807959, Example B3	WD repeat-containing protein 5		 209								US Patent		10.7270/Q26Q219X		aid1804926	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468870	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468870&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146371057	441570971							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968748	Cc1cc(CNC(=O)c2cccc(CNC3=NCCN3)c2)ccc1Cl	InChI=1S/C19H21ClN4O/c1-13-9-15(5-6-17(13)20)11-23-18(25)16-4-2-3-14(10-16)12-24-19-21-7-8-22-19/h2-6,9-10H,7-8,11-12H2,1H3,(H,23,25)(H2,21,22,24)	IKBPIQKPYJVGCZ-UHFFFAOYSA-N	468871	US10807959, Example B4	WD repeat-containing protein 5		 11.9								US Patent		10.7270/Q26Q219X		aid1804926	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468871	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468871&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370960	441570972							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968749	CC(NC(=O)c1cccc(CNC2=NCCN2)c1)c1cccc(Cl)c1	InChI=1S/C19H21ClN4O/c1-13(15-5-3-7-17(20)11-15)24-18(25)16-6-2-4-14(10-16)12-23-19-21-8-9-22-19/h2-7,10-11,13H,8-9,12H2,1H3,(H,24,25)(H2,21,22,23)	ZHGJIKXLESXIHK-UHFFFAOYSA-N	468872	US10807959, Example B5	WD repeat-containing protein 5		 30.8								US Patent		10.7270/Q26Q219X		aid1804926	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468872	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468872&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	HLM	6E1Y	146370875	441570973							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968750	Fc1ccc(cc1CNC1=NCCN1)C(=O)NCc1ccc(Cl)c(Cl)c1	InChI=1S/C18H17Cl2FN4O/c19-14-3-1-11(7-15(14)20)9-24-17(26)12-2-4-16(21)13(8-12)10-25-18-22-5-6-23-18/h1-4,7-8H,5-6,9-10H2,(H,24,26)(H2,22,23,25)	AJSVUDYNQZYABC-UHFFFAOYSA-N	468873	US10807959, Example B6	WD repeat-containing protein 5		 4.01								US Patent		10.7270/Q26Q219X		aid1804926	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468873	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468873&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370937	441570974							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968751	Cc1cc(C)cc(CNC(=O)c2ccc(F)c(CNC3=NCCN3)c2)c1	InChI=1S/C20H23FN4O/c1-13-7-14(2)9-15(8-13)11-24-19(26)16-3-4-18(21)17(10-16)12-25-20-22-5-6-23-20/h3-4,7-10H,5-6,11-12H2,1-2H3,(H,24,26)(H2,22,23,25)	VWCCPJSNKFCTAC-UHFFFAOYSA-N	468874	US10807959, Example B7	WD repeat-containing protein 5		 8.46								US Patent		10.7270/Q26Q219X		aid1804926	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468874	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468874&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370740	441570975							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968752	Clc1cc(CNC2=NCCN2)cc(c1)C(=O)NCc1ccc(Cl)c(Cl)c1	InChI=1S/C18H17Cl3N4O/c19-14-6-12(10-25-18-22-3-4-23-18)5-13(8-14)17(26)24-9-11-1-2-15(20)16(21)7-11/h1-2,5-8H,3-4,9-10H2,(H,24,26)(H2,22,23,25)	VNKABGWHTNAYDI-UHFFFAOYSA-N	468875	US10807959, Example B8	WD repeat-containing protein 5		 10.7								US Patent		10.7270/Q26Q219X		aid1804926	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468875	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468875&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370955	441570976							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968753	Clc1cc(Cl)cc(CNC(=O)c2cc(Cl)cc(CNC3=NCCN3)c2)c1	InChI=1S/C18H17Cl3N4O/c19-14-4-11(10-25-18-22-1-2-23-18)3-13(7-14)17(26)24-9-12-5-15(20)8-16(21)6-12/h3-8H,1-2,9-10H2,(H,24,26)(H2,22,23,25)	SMVOQFYYRZDCDW-UHFFFAOYSA-N	468876	US10807959, Example B9	WD repeat-containing protein 5		 17.4								US Patent		10.7270/Q26Q219X		aid1804926	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468876	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468876&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370772	441570977							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968754	Cc1ccc(CNC(=O)c2cc(Cl)cc(CNC3=NCCN3)c2)cc1Cl	InChI=1S/C19H20Cl2N4O/c1-12-2-3-13(8-17(12)21)10-24-18(26)15-6-14(7-16(20)9-15)11-25-19-22-4-5-23-19/h2-3,6-9H,4-5,10-11H2,1H3,(H,24,26)(H2,22,23,25)	UDIHWAXVJRPUES-UHFFFAOYSA-N	468877	US10807959, Example B10	WD repeat-containing protein 5		 54.5								US Patent		10.7270/Q26Q219X		aid1804926	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468877	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468877&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370770	441570978							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968755	Cc1cc(C)cc(CNC(=O)c2cc(Cl)cc(CNC3=NCCN3)c2)c1	InChI=1S/C20H23ClN4O/c1-13-5-14(2)7-15(6-13)11-24-19(26)17-8-16(9-18(21)10-17)12-25-20-22-3-4-23-20/h5-10H,3-4,11-12H2,1-2H3,(H,24,26)(H2,22,23,25)	KQYSRLCBMFIISB-UHFFFAOYSA-N	468878	US10807959, Example B11	WD repeat-containing protein 5		 46.0								US Patent		10.7270/Q26Q219X		aid1804926	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468878	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468878&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370865	441570979							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968756	CC(NC(=O)c1cc(Cl)cc(CNC2=NCCN2)c1)c1cccc(Cl)c1	InChI=1S/C19H20Cl2N4O/c1-12(14-3-2-4-16(20)9-14)25-18(26)15-7-13(8-17(21)10-15)11-24-19-22-5-6-23-19/h2-4,7-10,12H,5-6,11H2,1H3,(H,25,26)(H2,22,23,24)	KIWLNNWKTKWKSY-UHFFFAOYSA-N	468879	US10807959, Example B12	WD repeat-containing protein 5		 65.1								US Patent		10.7270/Q26Q219X		aid1804926	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468879	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468879&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370914	441570980							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968757	COc1cc(CNC(=O)c2ccc(Cl)c(CNC3=NCCN3)c2)cc(OC)c1	InChI=1S/C20H23ClN4O3/c1-27-16-7-13(8-17(10-16)28-2)11-24-19(26)14-3-4-18(21)15(9-14)12-25-20-22-5-6-23-20/h3-4,7-10H,5-6,11-12H2,1-2H3,(H,24,26)(H2,22,23,25)	SCLMJEWUVAWYAX-UHFFFAOYSA-N	468880	US10807959, Example B13	WD repeat-containing protein 5		 83.0								US Patent		10.7270/Q26Q219X		aid1804926	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468880	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468880&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370942	441570981							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968758	Clc1cc(Cl)cc(CNC(=O)c2ccc(Cl)c(CNC3=NCCN3)c2)c1	InChI=1S/C18H17Cl3N4O/c19-14-5-11(6-15(20)8-14)9-24-17(26)12-1-2-16(21)13(7-12)10-25-18-22-3-4-23-18/h1-2,5-8H,3-4,9-10H2,(H,24,26)(H2,22,23,25)	XOLLIDAEXAZECO-UHFFFAOYSA-N	468881	US10807959, Example B14	WD repeat-containing protein 5		 56.0								US Patent		10.7270/Q26Q219X		aid1804926	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468881	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468881&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370970	441570982							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968759	COc1cc(CNC(=O)c2ccc(F)c(CNC3=NCCN3)c2)cc(OC)c1	InChI=1S/C20H23FN4O3/c1-27-16-7-13(8-17(10-16)28-2)11-24-19(26)14-3-4-18(21)15(9-14)12-25-20-22-5-6-23-20/h3-4,7-10H,5-6,11-12H2,1-2H3,(H,24,26)(H2,22,23,25)	VDAMWMOTTUWVPR-UHFFFAOYSA-N	468882	US10807959, Example B15	WD repeat-containing protein 5		 1.33								US Patent		10.7270/Q26Q219X		aid1804926	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468882	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468882&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	HLS	6E22	138753248	441570983							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968760	Fc1ccc(cc1CNC1=NCCN1)C(=O)NCc1cc(Cl)ccn1	InChI=1S/C17H17ClFN5O/c18-13-3-4-20-14(8-13)10-23-16(25)11-1-2-15(19)12(7-11)9-24-17-21-5-6-22-17/h1-4,7-8H,5-6,9-10H2,(H,23,25)(H2,21,22,24)	MFOVFAFYOPSJAC-UHFFFAOYSA-N	468883	US10807959, Example B16	WD repeat-containing protein 5		 9.05								US Patent		10.7270/Q26Q219X		aid1804926	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468883	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468883&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370831	441570984							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968761	Fc1ccc(cc1CNC1=NCCN1)C(=O)NCc1cc(Cl)cc(Cl)c1	InChI=1S/C18H17Cl2FN4O/c19-14-5-11(6-15(20)8-14)9-24-17(26)12-1-2-16(21)13(7-12)10-25-18-22-3-4-23-18/h1-2,5-8H,3-4,9-10H2,(H,24,26)(H2,22,23,25)	DHFKUHSRJROAEG-UHFFFAOYSA-N	468884	US10807959, Example B17	WD repeat-containing protein 5		 2.47								US Patent		10.7270/Q26Q219X		aid1804926	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468884	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468884&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370827	441570985							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968762	COc1cc(OC)cc(c1)C(C)NC(=O)c1ccc(F)c(CNC2=NCCN2)c1	InChI=1S/C21H25FN4O3/c1-13(15-9-17(28-2)11-18(10-15)29-3)26-20(27)14-4-5-19(22)16(8-14)12-25-21-23-6-7-24-21/h4-5,8-11,13H,6-7,12H2,1-3H3,(H,26,27)(H2,23,24,25)	DTISHQXZUPPLFM-UHFFFAOYSA-N	468885	US10807959, Example B18	WD repeat-containing protein 5		 1.81								US Patent		10.7270/Q26Q219X		aid1804926	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468885	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468885&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146371004	441570986							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968763	COc1ccc(CNC(=O)c2ccc(F)c(CNC3=NCCN3)c2)cc1OC	InChI=1S/C20H23FN4O3/c1-27-17-6-3-13(9-18(17)28-2)11-24-19(26)14-4-5-16(21)15(10-14)12-25-20-22-7-8-23-20/h3-6,9-10H,7-8,11-12H2,1-2H3,(H,24,26)(H2,22,23,25)	LYPQQWFJWPIGAJ-UHFFFAOYSA-N	468886	US10807959, Example B19	WD repeat-containing protein 5		 8.06								US Patent		10.7270/Q26Q219X		aid1804926	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468886	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468886&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370842	441570987							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968764	Cc1ccnc(c1)C(NC(=O)c1ccc(F)c(CNC2=NCCN2)c1)C1CC1	InChI=1S/C21H24FN5O/c1-13-6-7-23-18(10-13)19(14-2-3-14)27-20(28)15-4-5-17(22)16(11-15)12-26-21-24-8-9-25-21/h4-7,10-11,14,19H,2-3,8-9,12H2,1H3,(H,27,28)(H2,24,25,26)	MQPDOSBDHVOUJT-UHFFFAOYSA-N	468887	US10807959, Example B20	WD repeat-containing protein 5		 4.60								US Patent		10.7270/Q26Q219X		aid1804926	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468887	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468887&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146371016	441570988							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968765	COc1cc(CNC(=O)c2cccc(CNC3=NCCN3)c2F)cc(OC)c1	InChI=1S/C20H23FN4O3/c1-27-15-8-13(9-16(10-15)28-2)11-24-19(26)17-5-3-4-14(18(17)21)12-25-20-22-6-7-23-20/h3-5,8-10H,6-7,11-12H2,1-2H3,(H,24,26)(H2,22,23,25)	QDOLMNUEDRBING-UHFFFAOYSA-N	468888	US10807959, Example B21	WD repeat-containing protein 5		 17.8								US Patent		10.7270/Q26Q219X		aid1804926	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468888	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468888&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146371031	441570989							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968766	COc1ccnc(CNC(=O)c2ccc(F)c(CNC3=NCCN3)c2)c1	InChI=1S/C18H20FN5O2/c1-26-15-4-5-20-14(9-15)11-23-17(25)12-2-3-16(19)13(8-12)10-24-18-21-6-7-22-18/h2-5,8-9H,6-7,10-11H2,1H3,(H,23,25)(H2,21,22,24)	RWJBVMFFPMBPMY-UHFFFAOYSA-N	468889	US10807959, Example B22	WD repeat-containing protein 5		 1.50								US Patent		10.7270/Q26Q219X		aid1804926	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468889	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468889&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370750	441570990							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968767	Fc1ccc(cc1CNC1=NCCN1)C(=O)NCc1ccc(Cl)cn1	InChI=1S/C17H17ClFN5O/c18-13-2-3-14(22-9-13)10-23-16(25)11-1-4-15(19)12(7-11)8-24-17-20-5-6-21-17/h1-4,7,9H,5-6,8,10H2,(H,23,25)(H2,20,21,24)	FICZSYPDVDGUJN-UHFFFAOYSA-N	468890	US10807959, Example B23	WD repeat-containing protein 5		 30.3								US Patent		10.7270/Q26Q219X		aid1804926	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468890	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468890&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370973	441570991							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968768	COc1cc(CN(C)C(=O)c2ccc(F)c(CNC3=NCCN3)c2)cc(OC)c1	InChI=1S/C21H25FN4O3/c1-26(13-14-8-17(28-2)11-18(9-14)29-3)20(27)15-4-5-19(22)16(10-15)12-25-21-23-6-7-24-21/h4-5,8-11H,6-7,12-13H2,1-3H3,(H2,23,24,25)	HFFBZGRIISJEED-UHFFFAOYSA-N	468891	US10807959, Example B24	WD repeat-containing protein 5		 49.8								US Patent		10.7270/Q26Q219X		aid1804926	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468891	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468891&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370717	441570992							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968769	COc1cccc(CNC(=O)c2ccc(F)c(CNC3=NCCN3)c2)n1	InChI=1S/C18H20FN5O2/c1-26-16-4-2-3-14(24-16)11-22-17(25)12-5-6-15(19)13(9-12)10-23-18-20-7-8-21-18/h2-6,9H,7-8,10-11H2,1H3,(H,22,25)(H2,20,21,23)	UUORHVYYAMJBMY-UHFFFAOYSA-N	468892	US10807959, Example B25	WD repeat-containing protein 5		 74.2								US Patent		10.7270/Q26Q219X		aid1804926	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468892	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468892&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370949	441570993							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968770	COc1ccc(cc1Cl)C(=O)NCc1ccc(F)c(CNC2=NCCN2)c1	InChI=1S/C19H20ClFN4O2/c1-27-17-5-3-13(9-15(17)20)18(26)24-10-12-2-4-16(21)14(8-12)11-25-19-22-6-7-23-19/h2-5,8-9H,6-7,10-11H2,1H3,(H,24,26)(H2,22,23,25)	UYOSSTIGEJMPEY-UHFFFAOYSA-N	468893	US10807959, Example B26	WD repeat-containing protein 5		 3.24								US Patent		10.7270/Q26Q219X		aid1804926	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468893	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468893&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146388583	441570994							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968771	COc1cc(CNC(=O)c2ccc(OC)c(CNC3=NCCN3)c2)cc(OC)c1	InChI=1S/C21H26N4O4/c1-27-17-8-14(9-18(11-17)28-2)12-24-20(26)15-4-5-19(29-3)16(10-15)13-25-21-22-6-7-23-21/h4-5,8-11H,6-7,12-13H2,1-3H3,(H,24,26)(H2,22,23,25)	GOVNGDRUVCAFTN-UHFFFAOYSA-N	468894	US10807959, Example B27	WD repeat-containing protein 5		 7.52								US Patent		10.7270/Q26Q219X		aid1804926	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468894	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468894&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370752	441570995							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968772	COc1ccc(cc1CNC1=NCCN1)C(=O)NCc1ccc(Cl)c(Cl)c1	InChI=1S/C19H20Cl2N4O2/c1-27-17-5-3-13(9-14(17)11-25-19-22-6-7-23-19)18(26)24-10-12-2-4-15(20)16(21)8-12/h2-5,8-9H,6-7,10-11H2,1H3,(H,24,26)(H2,22,23,25)	ZXFHPIAATGVMAP-UHFFFAOYSA-N	468895	US10807959, Example B28	WD repeat-containing protein 5		 0.622								US Patent		10.7270/Q26Q219X		aid1804926	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468895	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468895&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370948	441570996							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968773	Cc1ccnc(CNC(=O)c2ccc(F)c(CNC3=NCCN3)c2)c1	InChI=1S/C18H20FN5O/c1-12-4-5-20-15(8-12)11-23-17(25)13-2-3-16(19)14(9-13)10-24-18-21-6-7-22-18/h2-5,8-9H,6-7,10-11H2,1H3,(H,23,25)(H2,21,22,24)	DKXXBIFGWXWDPQ-UHFFFAOYSA-N	468896	US10807959, Example B29	WD repeat-containing protein 5		 24.9								US Patent		10.7270/Q26Q219X		aid1804926	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468896	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468896&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370817	441570997							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968774	COc1cc(OC)cc(c1)C(=O)NCc1cc(F)c(F)c(CNC2=NCCN2)c1	InChI=1S/C20H22F2N4O3/c1-28-15-7-13(8-16(9-15)29-2)19(27)25-10-12-5-14(18(22)17(21)6-12)11-26-20-23-3-4-24-20/h5-9H,3-4,10-11H2,1-2H3,(H,25,27)(H2,23,24,26)	LHHKQJQQYAPCPQ-UHFFFAOYSA-N	468897	US10807959, Example B30	WD repeat-containing protein 5		 5.32								US Patent		10.7270/Q26Q219X		aid1804926	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468897	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468897&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146388406	441570998							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968775	Cc1cc(C)cc(CNC(=O)c2cc(F)c(F)c(CNC3=NCCN3)c2)c1	InChI=1S/C20H22F2N4O/c1-12-5-13(2)7-14(6-12)10-25-19(27)15-8-16(18(22)17(21)9-15)11-26-20-23-3-4-24-20/h5-9H,3-4,10-11H2,1-2H3,(H,25,27)(H2,23,24,26)	GYOMWZSGMLUJGB-UHFFFAOYSA-N	468898	US10807959, Example B31	WD repeat-containing protein 5		 8.11								US Patent		10.7270/Q26Q219X		aid1804926	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468898	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468898&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370818	441570999							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968776	COc1ccc(CNC(=O)c2cc(F)c(F)c(CNC3=NCCN3)c2)cc1Cl	InChI=1S/C19H19ClF2N4O2/c1-28-16-3-2-11(6-14(16)20)9-25-18(27)12-7-13(17(22)15(21)8-12)10-26-19-23-4-5-24-19/h2-3,6-8H,4-5,9-10H2,1H3,(H,25,27)(H2,23,24,26)	DQKSHSPITVBLOW-UHFFFAOYSA-N	468899	US10807959, Example B32	WD repeat-containing protein 5		 4.51								US Patent		10.7270/Q26Q219X		aid1804926	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468899	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468899&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370859	441571000							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968777	Fc1cc(cc(CNC2=NCCN2)c1F)C(=O)NCc1ccc(Cl)c(Cl)c1	InChI=1S/C18H16Cl2F2N4O/c19-13-2-1-10(5-14(13)20)8-25-17(27)11-6-12(16(22)15(21)7-11)9-26-18-23-3-4-24-18/h1-2,5-7H,3-4,8-9H2,(H,25,27)(H2,23,24,26)	RNRBPSZZSDNMCH-UHFFFAOYSA-N	468900	US10807959, Example B33	WD repeat-containing protein 5		 0.444								US Patent		10.7270/Q26Q219X		aid1804926	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468900	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468900&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370728	441571001							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968778	COc1ccnc(CNC(=O)c2cc(F)c(F)c(CNC3=NCCN3)c2)c1	InChI=1S/C18H19F2N5O2/c1-27-14-2-3-21-13(8-14)10-24-17(26)11-6-12(16(20)15(19)7-11)9-25-18-22-4-5-23-18/h2-3,6-8H,4-5,9-10H2,1H3,(H,24,26)(H2,22,23,25)	SFUVQDYAADXKJP-UHFFFAOYSA-N	468901	US10807959, Example B34	WD repeat-containing protein 5		 12.0								US Patent		10.7270/Q26Q219X		aid1804926	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468901	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468901&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370868	441571002							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968779	COc1cc(OC)cc(c1)C(C)NC(=O)c1cc(F)c(F)c(CNC2=NCCN2)c1	InChI=1S/C21H24F2N4O3/c1-12(13-7-16(29-2)10-17(8-13)30-3)27-20(28)14-6-15(19(23)18(22)9-14)11-26-21-24-4-5-25-21/h6-10,12H,4-5,11H2,1-3H3,(H,27,28)(H2,24,25,26)	OEHQKPIAMJWIFZ-UHFFFAOYSA-N	468902	US10807959, Example B35	WD repeat-containing protein 5		 4.22								US Patent		10.7270/Q26Q219X		aid1804926	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468902	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468902&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370935	441571003							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968780	Fc1ccc(CNC2=NCCN2)cc1C(=O)NCc1ccc(Cl)c(Cl)c1	InChI=1S/C18H17Cl2FN4O/c19-14-3-1-12(8-15(14)20)9-24-17(26)13-7-11(2-4-16(13)21)10-25-18-22-5-6-23-18/h1-4,7-8H,5-6,9-10H2,(H,24,26)(H2,22,23,25)	UAJYZMHGFGIDCJ-UHFFFAOYSA-N	468903	US10807959, Example B36	WD repeat-containing protein 5		 0.917								US Patent		10.7270/Q26Q219X		aid1804926	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468903	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468903&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370832	441571004							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968781	COc1cc(CNC(=O)c2cc(CNC3=NCCN3)ccc2F)cc(OC)c1	InChI=1S/C20H23FN4O3/c1-27-15-7-14(8-16(10-15)28-2)12-24-19(26)17-9-13(3-4-18(17)21)11-25-20-22-5-6-23-20/h3-4,7-10H,5-6,11-12H2,1-2H3,(H,24,26)(H2,22,23,25)	BQOUKLMEMOPTRU-UHFFFAOYSA-N	468904	US10807959, Example B37	WD repeat-containing protein 5		 8.71								US Patent		10.7270/Q26Q219X		aid1804926	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468904	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468904&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370881	441571005							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968782	COc1cc(CNC(=O)c2ccc(OC)c(CNC3=NCCN3)c2)ccc1Cl	InChI=1S/C20H23ClN4O3/c1-27-17-6-4-14(10-15(17)12-25-20-22-7-8-23-20)19(26)24-11-13-3-5-16(21)18(9-13)28-2/h3-6,9-10H,7-8,11-12H2,1-2H3,(H,24,26)(H2,22,23,25)	OKECICYUSFHJFT-UHFFFAOYSA-N	468905	US10807959, Example B38	WD repeat-containing protein 5		 24.5								US Patent		10.7270/Q26Q219X		aid1804926	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468905	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468905&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370947	441571006							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968783	COc1ccc(cc1CNC1=NCCN1)C(=O)NCc1cc(Cl)ccn1	InChI=1S/C18H20ClN5O2/c1-26-16-3-2-12(8-13(16)10-24-18-21-6-7-22-18)17(25)23-11-15-9-14(19)4-5-20-15/h2-5,8-9H,6-7,10-11H2,1H3,(H,23,25)(H2,21,22,24)	GXHLEJDAHIKZBM-UHFFFAOYSA-N	468906	US10807959, Example B39	WD repeat-containing protein 5		 1.39								US Patent		10.7270/Q26Q219X		aid1804926	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468906	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468906&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370901	441571007							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968784	COc1ccnc(CNC(=O)c2ccc(OC)c(CNC3=NCCN3)c2)c1	InChI=1S/C19H23N5O3/c1-26-16-5-6-20-15(10-16)12-23-18(25)13-3-4-17(27-2)14(9-13)11-24-19-21-7-8-22-19/h3-6,9-10H,7-8,11-12H2,1-2H3,(H,23,25)(H2,21,22,24)	LOPKNASLFQYWJZ-UHFFFAOYSA-N	468907	US10807959, Example B40	WD repeat-containing protein 5		 7.21								US Patent		10.7270/Q26Q219X		aid1804926	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468907	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468907&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146371045	441571008							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968785	COc1ccc(cc1CNC1=NCCN1)C(=O)NCc1ccc(Cl)c(F)c1	InChI=1S/C19H20ClFN4O2/c1-27-17-5-3-13(9-14(17)11-25-19-22-6-7-23-19)18(26)24-10-12-2-4-15(20)16(21)8-12/h2-5,8-9H,6-7,10-11H2,1H3,(H,24,26)(H2,22,23,25)	OFWDZCVBTYIZLG-UHFFFAOYSA-N	468908	US10807959, Example B41	WD repeat-containing protein 5		 1.76								US Patent		10.7270/Q26Q219X		aid1804926	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468908	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468908&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370735	441571009							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968786	COc1ccc(cc1CNC1=NCCN1)C(=O)NCc1ccc(Cl)c(C)c1	InChI=1S/C20H23ClN4O2/c1-13-9-14(3-5-17(13)21)11-24-19(26)15-4-6-18(27-2)16(10-15)12-25-20-22-7-8-23-20/h3-6,9-10H,7-8,11-12H2,1-2H3,(H,24,26)(H2,22,23,25)	RLYIVVQBINPGSS-UHFFFAOYSA-N	468909	US10807959, Example B42	WD repeat-containing protein 5		 1.51								US Patent		10.7270/Q26Q219X		aid1804926	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468909	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468909&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370967	441571010							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968787	COc1cc(OC)cc(c1)C(C)NC(=O)c1ccc(OC)c(CNC2=NCCN2)c1	InChI=1S/C22H28N4O4/c1-14(16-10-18(28-2)12-19(11-16)29-3)26-21(27)15-5-6-20(30-4)17(9-15)13-25-22-23-7-8-24-22/h5-6,9-12,14H,7-8,13H2,1-4H3,(H,26,27)(H2,23,24,25)	RAWBYXWDOHDUBV-UHFFFAOYSA-N	468910	US10807959, Example B43	WD repeat-containing protein 5		 1.82								US Patent		10.7270/Q26Q219X		aid1804926	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468910	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468910&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370866	441571011							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968788	COc1ccc(cc1CNC1=NCCN1)C(=O)NCc1ccc(Cl)cn1	InChI=1S/C18H20ClN5O2/c1-26-16-5-2-12(8-13(16)9-24-18-20-6-7-21-18)17(25)23-11-15-4-3-14(19)10-22-15/h2-5,8,10H,6-7,9,11H2,1H3,(H,23,25)(H2,20,21,24)	NAUUFUAXYBUOER-UHFFFAOYSA-N	468911	US10807959, Example B44	WD repeat-containing protein 5		 20.3								US Patent		10.7270/Q26Q219X		aid1804926	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468911	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468911&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370873	441571012							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968789	Cc1cc(C)nc(CNC(=O)c2ccc(F)c(CNC3=NCCN3)c2)n1	InChI=1S/C18H21FN6O/c1-11-7-12(2)25-16(24-11)10-22-17(26)13-3-4-15(19)14(8-13)9-23-18-20-5-6-21-18/h3-4,7-8H,5-6,9-10H2,1-2H3,(H,22,26)(H2,20,21,23)	VTHWXKRYNMVINZ-UHFFFAOYSA-N	468912	US10807959, Example B45	WD repeat-containing protein 5		 11.3								US Patent		10.7270/Q26Q219X		aid1804926	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468912	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468912&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370989	441571013							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968790	Cc1cnc(CNC(=O)c2ccc(F)c(CNC3=NCCN3)c2)cn1	InChI=1S/C17H19FN6O/c1-11-7-22-14(9-21-11)10-23-16(25)12-2-3-15(18)13(6-12)8-24-17-19-4-5-20-17/h2-3,6-7,9H,4-5,8,10H2,1H3,(H,23,25)(H2,19,20,24)	VJMFKAXDPBOTAD-UHFFFAOYSA-N	468913	US10807959, Example B46	WD repeat-containing protein 5		 3.96								US Patent		10.7270/Q26Q219X		aid1804926	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468913	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468913&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370763	441571014							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968791	Cc1cc(CNC(=O)c2ccc(F)c(CNC3=NCCN3)c2)ccc1Cl	InChI=1S/C19H20ClFN4O/c1-12-8-13(2-4-16(12)20)10-24-18(26)14-3-5-17(21)15(9-14)11-25-19-22-6-7-23-19/h2-5,8-9H,6-7,10-11H2,1H3,(H,24,26)(H2,22,23,25)	DMFIRDHYJGFZMK-UHFFFAOYSA-N	468914	US10807959, Example B47	WD repeat-containing protein 5		 0.189								US Patent		10.7270/Q26Q219X		aid1804926	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468914	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468914&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146371153	441571015							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968792	Cc1ccnc(c1)C(NC(=O)c1cc(CNC2=NCCN2)c(F)cc1F)C1CC1	InChI=1S/C21H23F2N5O/c1-12-4-5-24-18(8-12)19(13-2-3-13)28-20(29)15-9-14(16(22)10-17(15)23)11-27-21-25-6-7-26-21/h4-5,8-10,13,19H,2-3,6-7,11H2,1H3,(H,28,29)(H2,25,26,27)	WCMFJMLYCUGWTD-UHFFFAOYSA-N	468915	US10807959, Example B48	WD repeat-containing protein 5		 2.17								US Patent		10.7270/Q26Q219X		aid1804926	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468915	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468915&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146371116	441571016							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981571	Fc1ccc(cc1F)[C@@H](NC(=O)c1cc(CN2CCSC2=N)cc(c1)-c1cccnc1C(F)(F)F)C1CC1	InChI=1S/C27H23F5N4OS/c28-21-6-5-17(13-22(21)29)23(16-3-4-16)35-25(37)19-11-15(14-36-8-9-38-26(36)33)10-18(12-19)20-2-1-7-34-24(20)27(30,31)32/h1-2,5-7,10-13,16,23,33H,3-4,8-9,14H2,(H,35,37)/t23-/m0/s1	BQLSZABWPPJTRL-QHCPKHFHSA-N	473368	US10844044, Example 318	WD repeat-containing protein 5		 0.290								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473368	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473368&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456021	442073577							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981572	Cc1cc(ccc1F)[C@H](NC(=O)c1cc(Cn2ccn(C)c2=N)cc(c1)-c1ccc(F)cc1C)C(F)(F)F	InChI=1S/C28H25F5N4O/c1-16-11-22(29)5-6-23(16)20-12-18(15-37-9-8-36(3)27(37)34)13-21(14-20)26(38)35-25(28(31,32)33)19-4-7-24(30)17(2)10-19/h4-14,25,34H,15H2,1-3H3,(H,35,38)/t25-/m0/s1	GGHFFQWJGTYANA-VWLOTQADSA-N	473369	US10844044, Example 45	WD repeat-containing protein 5		 0.740								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473369	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473369&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456453	442073578							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981573	Cc1cc(ccc1F)[C@@H](NC(=O)c1cc(Cn2ccn(C)c2=N)cc(c1)-c1ccnc2CCCc12)C1CC1	InChI=1S/C31H32FN5O/c1-19-14-22(8-9-27(19)32)29(21-6-7-21)35-30(38)24-16-20(18-37-13-12-36(2)31(37)33)15-23(17-24)25-10-11-34-28-5-3-4-26(25)28/h8-17,21,29,33H,3-7,18H2,1-2H3,(H,35,38)/t29-/m0/s1	YHRRNNYJLQXTKV-LJAQVGFWSA-N	473370	US10844044, Example 136	WD repeat-containing protein 5		<0.100								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473370	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473370&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456549	442073579							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981574	C[C@@H]1COCCN1c1cc(Cn2ccn(C)c2=N)cc(c1)C(=O)N[C@@H](C1CC1)c1ccc(F)c(C)c1	InChI=1S/C28H34FN5O2/c1-18-12-22(6-7-25(18)29)26(21-4-5-21)31-27(35)23-13-20(16-33-9-8-32(3)28(33)30)14-24(15-23)34-10-11-36-17-19(34)2/h6-9,12-15,19,21,26,30H,4-5,10-11,16-17H2,1-3H3,(H,31,35)/t19-,26+/m1/s1	AUOQQAVNIWBMMF-BCHFMIIMSA-N	473371	US10844044, Example 227	WD repeat-containing protein 5		 2.10								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473371	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473371&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146455753	442073580							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981575	CC(C)n1cc(c(n1)C(F)(F)F)-c1cc(CN2CCSC2=N)cc(c1)C(=O)N[C@@H](C1CC1)c1ccc(F)c(F)c1	InChI=1S/C28H28F5N5OS/c1-15(2)38-14-21(25(36-38)28(31,32)33)19-9-16(13-37-7-8-40-27(37)34)10-20(11-19)26(39)35-24(17-3-4-17)18-5-6-22(29)23(30)12-18/h5-6,9-12,14-15,17,24,34H,3-4,7-8,13H2,1-2H3,(H,35,39)/t24-/m0/s1	LXDRSBABISVMHK-DEOSSOPVSA-N	473372	US10844044, Example 319	WD repeat-containing protein 5		 0.320								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473372	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473372&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146455944	442073581							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981576	Cc1n[nH]c2cccc(-c3cc(Cn4ccn(C)c4=N)cc(c3)C(=O)NCc3ccc(Cl)c(C)c3)c12	InChI=1S/C28H27ClN6O/c1-17-11-19(7-8-24(17)29)15-31-27(36)22-13-20(16-35-10-9-34(3)28(35)30)12-21(14-22)23-5-4-6-25-26(23)18(2)32-33-25/h4-14,30H,15-16H2,1-3H3,(H,31,36)(H,32,33)	GUGKUQIXSPGOLP-UHFFFAOYSA-N	473373	US10844044, Example 46	WD repeat-containing protein 5		 1.30								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473373	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473373&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146455849	442073582							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981577	Cc1cc(ccc1F)[C@@H](NC(=O)c1cc(Cn2ccn(-c3ccccc3)c2=N)cc(c1)-c1cccnc1C(F)(F)F)C1CC1	InChI=1S/C34H29F4N5O/c1-21-16-24(11-12-29(21)35)30(23-9-10-23)41-32(44)26-18-22(17-25(19-26)28-8-5-13-40-31(28)34(36,37)38)20-42-14-15-43(33(42)39)27-6-3-2-4-7-27/h2-8,11-19,23,30,39H,9-10,20H2,1H3,(H,41,44)/t30-/m0/s1	HEHFWWVGJTWHJG-PMERELPUSA-N	473374	US10844044, Example 137	WD repeat-containing protein 5		>33.0								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473374	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473374&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146457354	442073583							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981578	Fc1ccc(c(Cl)c1)-c1cc(Cn2ccoc2=N)cc(c1)C(=O)NCc1ccc(Cl)c(Cl)c1	InChI=1S/C24H17Cl3FN3O2/c25-20-4-1-14(9-22(20)27)12-30-23(32)17-8-15(13-31-5-6-33-24(31)29)7-16(10-17)19-3-2-18(28)11-21(19)26/h1-11,29H,12-13H2,(H,30,32)	JFLTVBBUGYCCEA-UHFFFAOYSA-N	473375	US10844044, Example 228	WD repeat-containing protein 5		>33.0								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473375	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473375&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146488025	442073584							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981579	CCn1cc(c(n1)C(F)(F)F)-c1cc(Cn2ccsc2=N)cc(c1)C(=O)N[C@@H](C1CC1)c1ccc(F)c(C)c1	InChI=1S/C28H27F4N5OS/c1-3-37-15-22(25(35-37)28(30,31)32)20-11-17(14-36-8-9-39-27(36)33)12-21(13-20)26(38)34-24(18-4-5-18)19-6-7-23(29)16(2)10-19/h6-13,15,18,24,33H,3-5,14H2,1-2H3,(H,34,38)/t24-/m0/s1	SUALJMLRSACEMC-DEOSSOPVSA-N	473376	US10844044, Example 320	WD repeat-containing protein 5		<0.100								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473376	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473376&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456773	442073585							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981580	Cc1ccnc(c1)C(NC(=O)c1cc(Cn2ccn(C)c2=N)cc(c1)-c1c(C)ccc2[nH]ncc12)C1CC1			473377	US10844044, Example 47	WD repeat-containing protein 5		 0.880								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473377	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473377&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146455784	442073586							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981581	Cc1cc(ccc1F)[C@@H](NC(=O)c1cc(Cn2ccn(CC3CC3)c2=N)cc(c1)-c1cccnc1C(F)(F)F)C1CC1	InChI=1S/C32H31F4N5O/c1-19-13-23(8-9-27(19)33)28(22-6-7-22)39-30(42)25-15-21(18-41-12-11-40(31(41)37)17-20-4-5-20)14-24(16-25)26-3-2-10-38-29(26)32(34,35)36/h2-3,8-16,20,22,28,37H,4-7,17-18H2,1H3,(H,39,42)/t28-/m0/s1	AQMJUYLNRAQZAV-NDEPHWFRSA-N	473378	US10844044, Example 138	WD repeat-containing protein 5		 1.10								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473378	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473378&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146455866	442073587							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981582	COc1cc(CNC(=O)c2cc(Cn3ccoc3=N)cc(c2)-c2ccc(F)cc2Cl)cc(OC)c1	InChI=1S/C26H23ClFN3O4/c1-33-21-9-16(10-22(13-21)34-2)14-30-25(32)19-8-17(15-31-5-6-35-26(31)29)7-18(11-19)23-4-3-20(28)12-24(23)27/h3-13,29H,14-15H2,1-2H3,(H,30,32)	GECCAYUIPUVEDC-UHFFFAOYSA-N	473379	US10844044, Example 229	WD repeat-containing protein 5		 0.210								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473379	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473379&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146488041	442073588							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981583	Cc1cc(ccc1F)[C@@H](NC(=O)c1cc(Cn2ccsc2=N)cc(c1)-c1cn(C)nc1C(F)(F)F)C1CC1	InChI=1S/C27H25F4N5OS/c1-15-9-18(5-6-22(15)28)23(17-3-4-17)33-25(37)20-11-16(13-36-7-8-38-26(36)32)10-19(12-20)21-14-35(2)34-24(21)27(29,30)31/h5-12,14,17,23,32H,3-4,13H2,1-2H3,(H,33,37)/t23-/m0/s1	LVYKKJMAWCXRFL-QHCPKHFHSA-N	473380	US10844044, Example 321	WD repeat-containing protein 5		<0.100								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473380	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473380&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456338	442073589							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981584	COc1cc(CN(C)C(=O)c2cc(Cn3ccn(C)c3=N)cc(c2)-c2ccnc(C)c2)cc(OC)c1	InChI=1S/C28H31N5O3/c1-19-10-22(6-7-30-19)23-11-20(18-33-9-8-31(2)28(33)29)12-24(15-23)27(34)32(3)17-21-13-25(35-4)16-26(14-21)36-5/h6-16,29H,17-18H2,1-5H3	GWRSVACWJGLTEA-UHFFFAOYSA-N	473381	US10844044, Example 48	WD repeat-containing protein 5		 26.0								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473381	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473381&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146457663	442073590							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981585	Cc1cc(ccc1F)[C@@H](NC(=O)c1cc(Cn2ccn(C)c2=N)cc(c1)C1CC1)C1CC1	InChI=1S/C26H29FN4O/c1-16-11-20(7-8-23(16)27)24(19-5-6-19)29-25(32)22-13-17(12-21(14-22)18-3-4-18)15-31-10-9-30(2)26(31)28/h7-14,18-19,24,28H,3-6,15H2,1-2H3,(H,29,32)/t24-/m0/s1	CRPFOIBKZQMVQL-DEOSSOPVSA-N	473382	US10844044, Example 139	WD repeat-containing protein 5		 0.180								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473382	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473382&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456611	442073591							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981586	C[C@H](NC(=O)c1cc(Cn2ccoc2=N)cc(c1)-c1ccc(F)cc1C)c1ccc(F)c(C)c1	InChI=1S/C27H25F2N3O2/c1-16-11-23(28)5-6-24(16)21-12-19(15-32-8-9-34-27(32)30)13-22(14-21)26(33)31-18(3)20-4-7-25(29)17(2)10-20/h4-14,18,30H,15H2,1-3H3,(H,31,33)/t18-/m0/s1	QYAYPPKUMJPFKD-SFHVURJKSA-N	473383	US10844044, Example 230	WD repeat-containing protein 5		 0.060								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473383	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473383&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456327	442073592							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981587	CC(C)n1cc(c(n1)C(F)(F)F)-c1cc(Cn2ccsc2=N)cc(c1)C(=O)N[C@@H](C1CC1)c1ccc(F)c(C)c1	InChI=1S/C29H29F4N5OS/c1-16(2)38-15-23(26(36-38)29(31,32)33)21-11-18(14-37-8-9-40-28(37)34)12-22(13-21)27(39)35-25(19-4-5-19)20-6-7-24(30)17(3)10-20/h6-13,15-16,19,25,34H,4-5,14H2,1-3H3,(H,35,39)/t25-/m0/s1	ABTVJLKMUOHSNJ-VWLOTQADSA-N	473384	US10844044, Example 322	WD repeat-containing protein 5		<0.100								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473384	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473384&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146455704	442073593							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981588	Cc1cc(ccn1)-c1cc(Cn2ccn(C)c2=N)cc(c1)C(=O)NC(C1CC1)C1CC1	InChI=1S/C25H29N5O/c1-16-11-20(7-8-27-16)21-12-17(15-30-10-9-29(2)25(30)26)13-22(14-21)24(31)28-23(18-3-4-18)19-5-6-19/h7-14,18-19,23,26H,3-6,15H2,1-2H3,(H,28,31)	NDIPAWRSXYHFKR-UHFFFAOYSA-N	473385	US10844044, Example 49	WD repeat-containing protein 5		 22.0								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473385	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473385&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146455727	442073594							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981589	CN(Cc1ccc(Cl)c(Cl)c1)C(=O)c1cc(Cn2ccn(C)c2=N)cc(c1)-c1cnc(F)nc1C	InChI=1S/C25H23Cl2FN6O/c1-15-20(12-30-24(28)31-15)18-8-17(14-34-7-6-32(2)25(34)29)9-19(11-18)23(35)33(3)13-16-4-5-21(26)22(27)10-16/h4-12,29H,13-14H2,1-3H3	FAOXPARZWXTSHZ-UHFFFAOYSA-N	473386	US10844044, Example 140	WD repeat-containing protein 5		 10.00								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473386	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473386&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146488064	442073595							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981590	Cc1cc(ccc1F)[C@H](NC(=O)c1cc(Cn2ccoc2=N)cc(c1)-c1ccc(F)cc1C)C(F)(F)F	InChI=1S/C27H22F5N3O2/c1-15-10-21(28)4-5-22(15)19-11-17(14-35-7-8-37-26(35)33)12-20(13-19)25(36)34-24(27(30,31)32)18-3-6-23(29)16(2)9-18/h3-13,24,33H,14H2,1-2H3,(H,34,36)/t24-/m0/s1	DDSUAKREFLBEDR-DEOSSOPVSA-N	473387	US10844044, Example 231	WD repeat-containing protein 5		 0.620								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473387	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473387&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456320	442073596							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981591	CCn1cc(c(n1)C(F)(F)F)-c1cc(CN2CCSC2=N)cc(c1)C(=O)NCc1ccc(=O)n(C)c1	InChI=1S/C24H25F3N6O2S/c1-3-33-14-19(21(30-33)24(25,26)27)17-8-16(13-32-6-7-36-23(32)28)9-18(10-17)22(35)29-11-15-4-5-20(34)31(2)12-15/h4-5,8-10,12,14,28H,3,6-7,11,13H2,1-2H3,(H,29,35)	FRFOAQCHQYFGSD-UHFFFAOYSA-N	473389	US10844044, Example 323	WD repeat-containing protein 5		 1.80								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473389	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473389&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456391	442073598							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981592	Cc1cc(ccn1)-c1cc(Cn2ccn(C)c2=N)cc(c1)C(=O)NCc1nc(C)cc(C)n1	InChI=1S/C25H27N7O/c1-16-10-20(5-6-27-16)21-11-19(15-32-8-7-31(4)25(32)26)12-22(13-21)24(33)28-14-23-29-17(2)9-18(3)30-23/h5-13,26H,14-15H2,1-4H3,(H,28,33)	PQHRWRKIIPIKDB-UHFFFAOYSA-N	473390	US10844044, Example 50	WD repeat-containing protein 5		 27.0								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473390	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473390&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456646	442073599							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981593	Cc1cc(ccc1F)[C@@H](NC(=O)c1cc(Cn2ccn(C3CC3)c2=N)cc(c1)-c1ccc(F)cc1Cl)C1CC1	InChI=1S/C31H29ClF2N4O/c1-18-12-21(4-9-28(18)34)29(20-2-3-20)36-30(39)23-14-19(17-37-10-11-38(31(37)35)25-6-7-25)13-22(15-23)26-8-5-24(33)16-27(26)32/h4-5,8-16,20,25,29,35H,2-3,6-7,17H2,1H3,(H,36,39)/t29-/m0/s1	JYMBQPRGCVHDNK-LJAQVGFWSA-N	473392	US10844044, Example 141	WD repeat-containing protein 5		<0.100								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473392	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473392&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456115	442073601							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981594	Cc1cc(ccc1F)[C@@H](NC(=O)c1cc(Cn2ccoc2=N)cc(c1)-c1ccc(F)cc1C)C1CC1	InChI=1S/C29H27F2N3O2/c1-17-12-24(30)6-7-25(17)22-13-19(16-34-9-10-36-29(34)32)14-23(15-22)28(35)33-27(20-3-4-20)21-5-8-26(31)18(2)11-21/h5-15,20,27,32H,3-4,16H2,1-2H3,(H,33,35)/t27-/m0/s1	UQVLZOSFEYYOPD-MHZLTWQESA-N	473393	US10844044, Example 232	WD repeat-containing protein 5		 0.060								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473393	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473393&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456031	442073602							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981595	CCn1cc(c(n1)C(F)(F)F)-c1cc(Cn2ccsc2=N)cc(c1)C(=O)N[C@@H](C1CC1)c1ccc(Cl)c(F)c1	InChI=1S/C27H24ClF4N5OS/c1-2-37-14-20(24(35-37)27(30,31)32)18-9-15(13-36-7-8-39-26(36)33)10-19(11-18)25(38)34-23(16-3-4-16)17-5-6-21(28)22(29)12-17/h5-12,14,16,23,33H,2-4,13H2,1H3,(H,34,38)/t23-/m0/s1	WQPKHEIUDCRLIR-QHCPKHFHSA-N	473394	US10844044, Example 324	WD repeat-containing protein 5		<0.100								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473394	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473394&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146457563	442073603							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981596	Cc1cc(ccn1)-c1cc(Cn2ccn(C)c2=N)cc(c1)C(=O)NCc1ncc(Cl)cn1	InChI=1S/C23H22ClN7O/c1-15-7-17(3-4-26-15)18-8-16(14-31-6-5-30(2)23(31)25)9-19(10-18)22(32)29-13-21-27-11-20(24)12-28-21/h3-12,25H,13-14H2,1-2H3,(H,29,32)	YGZFHTOZWQJDMP-UHFFFAOYSA-N	473395	US10844044, Example 51	WD repeat-containing protein 5		 17.0								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473395	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473395&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456142	442073604							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981597	Cc1cc(ccc1F)[C@@H](NC(=O)c1cc(Cn2ccn(C3CC3)c2=N)cc(c1)-c1cn(C)nc1C(F)(F)F)C1CC1	InChI=1S/C30H30F4N6O/c1-17-11-20(5-8-25(17)31)26(19-3-4-19)36-28(41)22-13-18(15-39-9-10-40(29(39)35)23-6-7-23)12-21(14-22)24-16-38(2)37-27(24)30(32,33)34/h5,8-14,16,19,23,26,35H,3-4,6-7,15H2,1-2H3,(H,36,41)/t26-/m0/s1	OMKXOUGNSKUUQD-SANMLTNESA-N	473396	US10844044, Example 142	WD repeat-containing protein 5		<0.100								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473396	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473396&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456060	442073605							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981598	C[C@H](NC(=O)c1cc(Cn2ccoc2=N)cc(c1)-c1ccc(F)cc1C)c1ccc(F)c(c1)C(F)(F)F	InChI=1S/C27H22F5N3O2/c1-15-9-21(28)4-5-22(15)19-10-17(14-35-7-8-37-26(35)33)11-20(12-19)25(36)34-16(2)18-3-6-24(29)23(13-18)27(30,31)32/h3-13,16,33H,14H2,1-2H3,(H,34,36)/t16-/m0/s1	ISSKJNNKHOGDIC-INIZCTEOSA-N	473397	US10844044, Example 233	WD repeat-containing protein 5		 1.50								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473397	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473397&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146455742	442073606							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981599	Cc1cc(ncc1F)[C@@H](NC(=O)c1cc(Cn2ccsc2=N)cc(c1)-c1cn(C)nc1C(F)(F)F)C1CC1	InChI=1S/C26H24F4N6OS/c1-14-7-21(32-11-20(14)27)22(16-3-4-16)33-24(37)18-9-15(12-36-5-6-38-25(36)31)8-17(10-18)19-13-35(2)34-23(19)26(28,29)30/h5-11,13,16,22,31H,3-4,12H2,1-2H3,(H,33,37)/t22-/m0/s1	AESNMGWHBDUKQR-QFIPXVFZSA-N	473398	US10844044, Example 325	WD repeat-containing protein 5		<0.100								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473398	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473398&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456882	442073607							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981600	COc1cc(CNC(=O)c2cc(Cn3ccn(C)c3=N)cc(c2)-c2c(C)cc(F)cc2F)cc(OC)c1	InChI=1S/C28H28F2N4O3/c1-17-7-22(29)13-25(30)26(17)20-8-19(16-34-6-5-33(2)28(34)31)9-21(12-20)27(35)32-15-18-10-23(36-3)14-24(11-18)37-4/h5-14,31H,15-16H2,1-4H3,(H,32,35)	VLIAEHVNDKQOBJ-UHFFFAOYSA-N	473399	US10844044, Example 52	WD repeat-containing protein 5		 0.190								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473399	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473399&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146455942	442073608							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981601	CN1CCN(Cc2cc(cc(c2)-c2cccnc2C(F)(F)F)C(=O)N[C@@H](C2CC2)c2ccc(F)c(C)c2)C1=N	InChI=1S/C29H29F4N5O/c1-17-12-20(7-8-24(17)30)25(19-5-6-19)36-27(39)22-14-18(16-38-11-10-37(2)28(38)34)13-21(15-22)23-4-3-9-35-26(23)29(31,32)33/h3-4,7-9,12-15,19,25,34H,5-6,10-11,16H2,1-2H3,(H,36,39)/t25-/m0/s1	OUJXJWRAPICBTJ-VWLOTQADSA-N	473400	US10844044, Example 143	WD repeat-containing protein 5		<0.100								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473400	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473400&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146455951	442073609							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981602	C[C@H](NC(=O)c1cc(Cn2ccoc2=N)cc(c1)-c1ccc(F)cc1C)c1ccc(Cl)c(C)c1	InChI=1S/C27H25ClFN3O2/c1-16-11-23(29)5-6-24(16)21-12-19(15-32-8-9-34-27(32)30)13-22(14-21)26(33)31-18(3)20-4-7-25(28)17(2)10-20/h4-14,18,30H,15H2,1-3H3,(H,31,33)/t18-/m0/s1	LBSKBVMXIDVPSQ-SFHVURJKSA-N	473401	US10844044, Example 234	WD repeat-containing protein 5		 1.000								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473401	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473401&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456835	442073610							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981603	Cc1cc(ncc1F)[C@@H](NC(=O)c1cc(CN2CCSC2=N)cc(c1)-c1cn(C)nc1C(F)(F)F)C1CC1	InChI=1S/C26H26F4N6OS/c1-14-7-21(32-11-20(14)27)22(16-3-4-16)33-24(37)18-9-15(12-36-5-6-38-25(36)31)8-17(10-18)19-13-35(2)34-23(19)26(28,29)30/h7-11,13,16,22,31H,3-6,12H2,1-2H3,(H,33,37)/t22-/m0/s1	BHGOTVOEUHONCC-QFIPXVFZSA-N	473402	US10844044, Example 326	WD repeat-containing protein 5		<0.100								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473402	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473402&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456801	442073611							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981604	Cc1cc(CNC(=O)c2cc(Cn3ccn(C)c3=N)cc(c2)-c2c(C)cc(F)cc2F)ccc1Cl	InChI=1S/C27H25ClF2N4O/c1-16-8-18(4-5-23(16)28)14-32-26(35)21-11-19(15-34-7-6-33(3)27(34)31)10-20(12-21)25-17(2)9-22(29)13-24(25)30/h4-13,31H,14-15H2,1-3H3,(H,32,35)	CBNDBDPZYFJHRL-UHFFFAOYSA-N	473403	US10844044, Example 53	WD repeat-containing protein 5		 0.560								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473403	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473403&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146457786	442073612							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981605	COc1cc(CNC(=O)c2cc(Cn3ccn(C)c3=N)cc(OC(F)(F)F)c2)cc(OC)c1	InChI=1S/C22H23F3N4O4/c1-28-4-5-29(21(28)26)13-15-6-16(10-19(9-15)33-22(23,24)25)20(30)27-12-14-7-17(31-2)11-18(8-14)32-3/h4-11,26H,12-13H2,1-3H3,(H,27,30)	PBFPKPKAXCZJIC-UHFFFAOYSA-N	473404	US10844044, Example 144	WD repeat-containing protein 5		 1.14								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473404	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473404&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456742	442073613							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981606	COc1cc(OC)cc(c1)C(NC(=O)c1cc(Cn2ccoc2=N)cc(c1)-c1ncccc1C(F)(F)F)C1CC1	InChI=1S/C29H27F3N4O4/c1-38-22-13-20(14-23(15-22)39-2)25(18-5-6-18)35-27(37)21-11-17(16-36-8-9-40-28(36)33)10-19(12-21)26-24(29(30,31)32)4-3-7-34-26/h3-4,7-15,18,25,33H,5-6,16H2,1-2H3,(H,35,37)	MNIZEJTYGAHLDN-UHFFFAOYSA-N	473405	US10844044, Example 235	WD repeat-containing protein 5		 3.50								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473405	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473405&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146455744	442073614							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981607	COc1cc(ccc1F)[C@@H](NC(=O)c1cc(Cn2ccsc2=N)cc(c1)-c1cn(C)nc1C(F)(F)F)C1CC1	InChI=1S/C27H25F4N5O2S/c1-35-14-20(24(34-35)27(29,30)31)18-9-15(13-36-7-8-39-26(36)32)10-19(11-18)25(37)33-23(16-3-4-16)17-5-6-21(28)22(12-17)38-2/h5-12,14,16,23,32H,3-4,13H2,1-2H3,(H,33,37)/t23-/m0/s1	FVWZGJJKHQOJDV-QHCPKHFHSA-N	473406	US10844044, Example 327	WD repeat-containing protein 5		<0.100								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473406	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473406&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456255	442073615							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981608	Cc1cc(ccc1F)[C@@H](NC(=O)c1cc(Cn2ccn(C)c2=N)cc(c1)-c1ccc(F)cc1C)C1CC1	InChI=1S/C30H30F2N4O/c1-18-13-25(31)7-8-26(18)23-14-20(17-36-11-10-35(3)30(36)33)15-24(16-23)29(37)34-28(21-4-5-21)22-6-9-27(32)19(2)12-22/h6-16,21,28,33H,4-5,17H2,1-3H3,(H,34,37)/t28-/m0/s1	CNTZMTRZTREIRC-NDEPHWFRSA-N	473407	US10844044, Example 54	WD repeat-containing protein 5		<0.100								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473407	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473407&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456042	442073616							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981609	Cc1ccnc(c1)C(NC(=O)c1cc(Cn2ccn(C)c2=N)cc(OC(F)(F)F)c1)C1CC1	InChI=1S/C23H24F3N5O2/c1-14-5-6-28-19(9-14)20(16-3-4-16)29-21(32)17-10-15(11-18(12-17)33-23(24,25)26)13-31-8-7-30(2)22(31)27/h5-12,16,20,27H,3-4,13H2,1-2H3,(H,29,32)	GLTBQXGLLMFNRI-UHFFFAOYSA-N	473408	US10844044, Example 145	WD repeat-containing protein 5		 0.950								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473408	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473408&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456041	442073617							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981610	COc1cc(OC)cc(c1)C(NC(=O)c1cc(Cn2ccoc2=N)cc(c1)-c1ccc(F)cc1OC(F)F)C1CC1	InChI=1S/C30H28F3N3O5/c1-38-23-12-20(13-24(15-23)39-2)27(18-3-4-18)35-28(37)21-10-17(16-36-7-8-40-30(36)34)9-19(11-21)25-6-5-22(31)14-26(25)41-29(32)33/h5-15,18,27,29,34H,3-4,16H2,1-2H3,(H,35,37)	AXBAJKQKDKOEFG-UHFFFAOYSA-N	473409	US10844044, Example 236	WD repeat-containing protein 5		 0.160								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473409	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473409&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456083	442073618							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981611	CCn1cc(c(n1)C(F)(F)F)-c1cc(Cn2ccsc2=N)cc(c1)C(=O)N[C@@H](C1CC1)c1ccc(F)c(OC)c1	InChI=1S/C28H27F4N5O2S/c1-3-37-15-21(25(35-37)28(30,31)32)19-10-16(14-36-8-9-40-27(36)33)11-20(12-19)26(38)34-24(17-4-5-17)18-6-7-22(29)23(13-18)39-2/h6-13,15,17,24,33H,3-5,14H2,1-2H3,(H,34,38)/t24-/m0/s1	ATIXNZXSOBXEAZ-DEOSSOPVSA-N	473410	US10844044, Example 328	WD repeat-containing protein 5		<0.100								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473410	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473410&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456345	442073619							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981612	CC(NC(=O)c1cc(Cn2ccn(C)c2=N)cc(n1)-c1ccc(F)cc1C)c1cc(C)c(Cl)cn1	InChI=1S/C26H26ClFN6O/c1-15-9-19(28)5-6-20(15)23-11-18(14-34-8-7-33(4)26(34)29)12-24(32-23)25(35)31-17(3)22-10-16(2)21(27)13-30-22/h5-13,17,29H,14H2,1-4H3,(H,31,35)	VGNKYNRRDSPVQH-UHFFFAOYSA-N	473411	US10844044, Example 55	WD repeat-containing protein 5		 1.80								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473411	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473411&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456030	442073620							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981613	Cn1ccn(Cc2cc(OC(F)(F)F)cc(c2)C(=O)N[C@@H](CC(O)=O)c2cccc(c2)C(F)(F)F)c1=N	InChI=1S/C23H20F6N4O4/c1-32-5-6-33(21(32)30)12-13-7-15(10-17(8-13)37-23(27,28)29)20(36)31-18(11-19(34)35)14-3-2-4-16(9-14)22(24,25)26/h2-10,18,30H,11-12H2,1H3,(H,31,36)(H,34,35)/t18-/m0/s1	HQGOEWNJEQICNL-SFHVURJKSA-N	473412	US10844044, Example 146	WD repeat-containing protein 5		 10.00								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473412	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473412&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456409	442073621							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981614	Cc1ccnc(c1)C(NC(=O)c1cc(Cn2ccoc2=N)cc(c1)-c1ncccc1C(F)(F)F)C1CC1	InChI=1S/C27H24F3N5O2/c1-16-6-8-32-22(11-16)24(18-4-5-18)34-25(36)20-13-17(15-35-9-10-37-26(35)31)12-19(14-20)23-21(27(28,29)30)3-2-7-33-23/h2-3,6-14,18,24,31H,4-5,15H2,1H3,(H,34,36)	HMJYCTGVPOBEJW-UHFFFAOYSA-N	473413	US10844044, Example 237	WD repeat-containing protein 5		 7.50								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473413	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473413&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146455713	442073622							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981615	COc1cc(ccc1F)[C@@H](NC(=O)c1cc(CN2CCSC2=N)cc(c1)-c1cccnc1C(F)(F)F)C1CC1	InChI=1S/C28H26F4N4O2S/c1-38-23-14-18(6-7-22(23)29)24(17-4-5-17)35-26(37)20-12-16(15-36-9-10-39-27(36)33)11-19(13-20)21-3-2-8-34-25(21)28(30,31)32/h2-3,6-8,11-14,17,24,33H,4-5,9-10,15H2,1H3,(H,35,37)/t24-/m0/s1	NDMYXJINPZVCKD-DEOSSOPVSA-N	473414	US10844044, Example 330	WD repeat-containing protein 5		 0.220								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473414	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473414&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146455788	442073623							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981616	Cc1cc(CNC(=O)c2cc(Cn3ccn(C)c3=N)cc(n2)-c2ccc(F)cc2C)ccc1Cl	InChI=1S/C26H25ClFN5O/c1-16-11-20(28)5-6-21(16)23-12-19(15-33-9-8-32(3)26(33)29)13-24(31-23)25(34)30-14-18-4-7-22(27)17(2)10-18/h4-13,29H,14-15H2,1-3H3,(H,30,34)	CBIKRUBKRFXACN-UHFFFAOYSA-N	473415	US10844044, Example 56	WD repeat-containing protein 5		 1.20								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473415	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473415&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146455738	442073624							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981617	Cc1cc(CNC(=O)c2cc(Cn3ccn(C)c3=N)cc(OC(F)(F)F)c2)ccc1Cl	InChI=1S/C21H20ClF3N4O2/c1-13-7-14(3-4-18(13)22)11-27-19(30)16-8-15(9-17(10-16)31-21(23,24)25)12-29-6-5-28(2)20(29)26/h3-10,26H,11-12H2,1-2H3,(H,27,30)	HZXNVVCPWNIAED-UHFFFAOYSA-N	473416	US10844044, Example 147	WD repeat-containing protein 5		 0.370								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473416	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473416&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456101	442073625							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981618	COc1cc(CNC(=O)c2cc(Cn3ccoc3=N)cc(c2)-c2ncc(F)cc2C)cc(OC)c1	InChI=1S/C26H25FN4O4/c1-16-6-21(27)14-29-24(16)19-7-18(15-31-4-5-35-26(31)28)8-20(11-19)25(32)30-13-17-9-22(33-2)12-23(10-17)34-3/h4-12,14,28H,13,15H2,1-3H3,(H,30,32)	BQTKKMQHOOUHRL-UHFFFAOYSA-N	473417	US10844044, Example 238	WD repeat-containing protein 5		 2.90								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473417	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473417&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146455888	442073626							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981619	Cc1nc(F)ccc1-c1cc(CN2CCCC2=N)cc(c1)C(=O)NCc1ccc(Cl)c(Cl)c1	InChI=1S/C25H23Cl2FN4O/c1-15-20(5-7-23(28)31-15)18-9-17(14-32-8-2-3-24(32)29)10-19(12-18)25(33)30-13-16-4-6-21(26)22(27)11-16/h4-7,9-12,29H,2-3,8,13-14H2,1H3,(H,30,33)	BZOGQEZICWJLJG-UHFFFAOYSA-N	473419	US10844044, Example 331	WD repeat-containing protein 5		 0.300								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473419	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473419&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456303	442073628							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981620	Cc1cc(F)ccc1-c1cc(Cn2ccn(C)c2=N)cc(c1)C(=O)Nc1nc2ccccc2s1	InChI=1S/C26H22FN5OS/c1-16-11-20(27)7-8-21(16)18-12-17(15-32-10-9-31(2)25(32)28)13-19(14-18)24(33)30-26-29-22-5-3-4-6-23(22)34-26/h3-14,28H,15H2,1-2H3,(H,29,30,33)	GVZUNXSGVIXLTP-UHFFFAOYSA-N	473420	US10844044, Example 57	WD repeat-containing protein 5		>33.0								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473420	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473420&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146457906	442073629							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981621	Cn1ccn(Cc2cc(C(=O)N[C@@H](CC(O)=O)c3cccc(c3)C(F)(F)F)c(F)c(c2)-c2ccc(F)cc2C(F)(F)F)c1=N	InChI=1S/C29H22F8N4O3/c1-40-7-8-41(27(40)38)14-15-9-20(19-6-5-18(30)12-22(19)29(35,36)37)25(31)21(10-15)26(44)39-23(13-24(42)43)16-3-2-4-17(11-16)28(32,33)34/h2-12,23,38H,13-14H2,1H3,(H,39,44)(H,42,43)/t23-/m0/s1	GZSDPPWFWPRISX-QHCPKHFHSA-N	473421	US10844044, Example 148	WD repeat-containing protein 5		 0.290								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473421	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473421&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146455929	442073630							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981622	Cc1ccnc(c1)C(NC(=O)c1cc(Cn2ccoc2=N)cc(c1)-c1ncc(F)cc1C)C1CC1	InChI=1S/C27H26FN5O2/c1-16-5-6-30-23(9-16)25(19-3-4-19)32-26(34)21-12-18(15-33-7-8-35-27(33)29)11-20(13-21)24-17(2)10-22(28)14-31-24/h5-14,19,25,29H,3-4,15H2,1-2H3,(H,32,34)	UYMWVRRXZMTIQC-UHFFFAOYSA-N	473422	US10844044, Example 239	WD repeat-containing protein 5		 5.30								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473422	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473422&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146457645	442073631							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981623	Cc1cc(c(C)cc1F)-c1cc(CN2CCCC2=N)cc(c1)C(=O)NCc1ccc(Cl)c(Cl)c1	InChI=1S/C27H26Cl2FN3O/c1-16-9-25(30)17(2)8-22(16)20-10-19(15-33-7-3-4-26(33)31)11-21(13-20)27(34)32-14-18-5-6-23(28)24(29)12-18/h5-6,8-13,31H,3-4,7,14-15H2,1-2H3,(H,32,34)	MZGTVDSJTZRYAM-UHFFFAOYSA-N	473423	US10844044, Example 332	WD repeat-containing protein 5		 19.0								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473423	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473423&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146455891	442073632							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981624	C[C@@H](NC(=O)c1cc(Cn2ccn(C)c2=N)cc(n1)-c1ccc(F)cc1C)c1ccc(Cl)c(Cl)c1	InChI=1S/C26H24Cl2FN5O/c1-15-10-19(29)5-6-20(15)23-11-17(14-34-9-8-33(3)26(34)30)12-24(32-23)25(35)31-16(2)18-4-7-21(27)22(28)13-18/h4-13,16,30H,14H2,1-3H3,(H,31,35)/t16-/m1/s1	BWYOIODDAPEQOB-MRXNPFEDSA-N	473424	US10844044, Example 58	WD repeat-containing protein 5		 0.930								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473424	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473424&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456258	442073633							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981625	Cc1ccnc(c1)[C@@H](NC(=O)c1cc(Cn2ccn(C)c2=N)cc(OC(F)(F)F)c1)C1CC1	InChI=1S/C23H24F3N5O2/c1-14-5-6-28-19(9-14)20(16-3-4-16)29-21(32)17-10-15(11-18(12-17)33-23(24,25)26)13-31-8-7-30(2)22(31)27/h5-12,16,20,27H,3-4,13H2,1-2H3,(H,29,32)/t20-/m0/s1	GLTBQXGLLMFNRI-FQEVSTJZSA-N	473425	US10844044, Example 149	WD repeat-containing protein 5		 0.560								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473425	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473425&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456039	442073634							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981626	Cc1cc(ccc1F)[C@@H](NC(=O)c1cc(Cn2ccoc2=N)cc(c1)-c1ncc(F)cc1C)C1CC1	InChI=1S/C28H26F2N4O2/c1-16-9-20(5-6-24(16)30)26(19-3-4-19)33-27(35)22-12-18(15-34-7-8-36-28(34)31)11-21(13-22)25-17(2)10-23(29)14-32-25/h5-14,19,26,31H,3-4,15H2,1-2H3,(H,33,35)/t26-/m0/s1	HDLNUTIGFBFGFB-SANMLTNESA-N	473426	US10844044, Example 240	WD repeat-containing protein 5		 10.00								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473426	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473426&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146455758	442073635							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968793	COc1cc(OC)cc(c1)C(C)NC(=O)c1cc(CNC2=NCCN2)c(F)cc1F	InChI=1S/C21H24F2N4O3/c1-12(13-6-15(29-2)9-16(7-13)30-3)27-20(28)17-8-14(18(22)10-19(17)23)11-26-21-24-4-5-25-21/h6-10,12H,4-5,11H2,1-3H3,(H,27,28)(H2,24,25,26)	GWKWTDUQHRORGA-UHFFFAOYSA-N	468916	US10807959, Example B49	WD repeat-containing protein 5		 1.06								US Patent		10.7270/Q26Q219X		aid1804926	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468916	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468916&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370766	441571017							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968794	CCOc1ccc(cc1CNC1=NCCN1)C(=O)NC(C1CC1)c1cc(C)ccn1	InChI=1S/C23H29N5O2/c1-3-30-20-7-6-17(13-18(20)14-27-23-25-10-11-26-23)22(29)28-21(16-4-5-16)19-12-15(2)8-9-24-19/h6-9,12-13,16,21H,3-5,10-11,14H2,1-2H3,(H,28,29)(H2,25,26,27)	LGUBRHURHQEMPA-UHFFFAOYSA-N	468917	US10807959, Example B50	WD repeat-containing protein 5		 12.4								US Patent		10.7270/Q26Q219X		aid1804926	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468917	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468917&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370774	441571018							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968795	CCOc1ccc(cc1CNC1=NCCN1)C(=O)NC(C)c1cc(OC)cc(OC)c1	InChI=1S/C23H30N4O4/c1-5-31-21-7-6-16(10-18(21)14-26-23-24-8-9-25-23)22(28)27-15(2)17-11-19(29-3)13-20(12-17)30-4/h6-7,10-13,15H,5,8-9,14H2,1-4H3,(H,27,28)(H2,24,25,26)	JUWGYXCESNDPPV-UHFFFAOYSA-N	468918	US10807959, Example B51	WD repeat-containing protein 5		 9.77								US Patent		10.7270/Q26Q219X		aid1804926	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468918	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468918&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370891	441571019							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968796	COc1cc(OC)cc(c1)C(C)NC(=O)c1ccc(OC(C)C)c(CNC2=NCCN2)c1	InChI=1S/C24H32N4O4/c1-15(2)32-22-7-6-17(10-19(22)14-27-24-25-8-9-26-24)23(29)28-16(3)18-11-20(30-4)13-21(12-18)31-5/h6-7,10-13,15-16H,8-9,14H2,1-5H3,(H,28,29)(H2,25,26,27)	IILFFOCGRIXDME-UHFFFAOYSA-N	468919	US10807959, Example B52	WD repeat-containing protein 5		 33.0								US Patent		10.7270/Q26Q219X		aid1804926	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468919	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468919&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370932	441571020							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968797	CC(C)Oc1ccc(cc1CNC1=NCCN1)C(=O)NCc1ccc(Cl)c(Cl)c1	InChI=1S/C21H24Cl2N4O2/c1-13(2)29-19-6-4-15(10-16(19)12-27-21-24-7-8-25-21)20(28)26-11-14-3-5-17(22)18(23)9-14/h3-6,9-10,13H,7-8,11-12H2,1-2H3,(H,26,28)(H2,24,25,27)	SHVCQPLJGMAYFL-UHFFFAOYSA-N	468920	US10807959, Example B53	WD repeat-containing protein 5		 40.9								US Patent		10.7270/Q26Q219X		aid1804926	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468920	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468920&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370918	441571021							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968798	Fc1ccc(c(Cl)c1)-c1cc(CNC2=NCCN2)cc(c1)C(=O)NCc1ccc(Cl)c(Cl)c1	InChI=1S/C24H20Cl3FN4O/c25-20-4-1-14(9-22(20)27)12-31-23(33)17-8-15(13-32-24-29-5-6-30-24)7-16(10-17)19-3-2-18(28)11-21(19)26/h1-4,7-11H,5-6,12-13H2,(H,31,33)(H2,29,30,32)	CYQGIBVRUPZKTF-UHFFFAOYSA-N	468921	US10807959, Example B54	WD repeat-containing protein 5		 1.12								US Patent		10.7270/Q26Q219X		aid1804926	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468921	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468921&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370771	441571022							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968799	Cc1cc(C)cc(CNC(=O)c2cc(CNC3=NCCN3)cc(c2)-c2ccc(F)cc2Cl)c1	InChI=1S/C26H26ClFN4O/c1-16-7-17(2)9-18(8-16)14-31-25(33)21-11-19(15-32-26-29-5-6-30-26)10-20(12-21)23-4-3-22(28)13-24(23)27/h3-4,7-13H,5-6,14-15H2,1-2H3,(H,31,33)(H2,29,30,32)	HSMFVHUXDLSKLX-UHFFFAOYSA-N	468922	US10807959, Example B55	WD repeat-containing protein 5		 1.27								US Patent		10.7270/Q26Q219X		aid1804926	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468922	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468922&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370931	441571023							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968800	Cc1cc(CNC(=O)c2cc(CNC3=NCCN3)cc(c2)-c2ccc(F)cc2Cl)ccc1Cl	InChI=1S/C25H23Cl2FN4O/c1-15-8-16(2-5-22(15)26)13-31-24(33)19-10-17(14-32-25-29-6-7-30-25)9-18(11-19)21-4-3-20(28)12-23(21)27/h2-5,8-12H,6-7,13-14H2,1H3,(H,31,33)(H2,29,30,32)	KHUCUHUFENFFTJ-UHFFFAOYSA-N	468923	US10807959, Example B58	WD repeat-containing protein 5		 2.06								US Patent		10.7270/Q26Q219X		aid1804926	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468923	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468923&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370962	441571024							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968801	COc1cc(CNC(=O)c2cc(CNC3=NCCN3)cc(c2)-c2ccc(F)nc2C)cc(OC)c1	InChI=1S/C26H28FN5O3/c1-16-23(4-5-24(27)32-16)19-8-17(15-31-26-28-6-7-29-26)9-20(12-19)25(33)30-14-18-10-21(34-2)13-22(11-18)35-3/h4-5,8-13H,6-7,14-15H2,1-3H3,(H,30,33)(H2,28,29,31)	FBFIUNWMMTUQQO-UHFFFAOYSA-N	468924	US10807959, Example B63	WD repeat-containing protein 5		 0.131								US Patent		10.7270/Q26Q219X		aid1804926	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468924	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468924&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370760	441571025							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968802	Cc1nc(F)ccc1-c1cc(CNC2=NCCN2)cc(c1)C(=O)NCc1ccc(Cl)c(Cl)c1	InChI=1S/C24H22Cl2FN5O/c1-14-19(3-5-22(27)32-14)17-8-16(13-31-24-28-6-7-29-24)9-18(11-17)23(33)30-12-15-2-4-20(25)21(26)10-15/h2-5,8-11H,6-7,12-13H2,1H3,(H,30,33)(H2,28,29,31)	RQCCOXNZCYISHV-UHFFFAOYSA-N	468925	US10807959, Example B64	WD repeat-containing protein 5		 0.021								US Patent		10.7270/Q26Q219X		aid1804926	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468925	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468925&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370821	441571026							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968803	COc1cc(CNC(=O)c2cc(CNC3=NCCN3)cc(c2)-c2ccnc(C)c2)cc(OC)c1	InChI=1S/C26H29N5O3/c1-17-8-20(4-5-27-17)21-9-18(16-31-26-28-6-7-29-26)10-22(13-21)25(32)30-15-19-11-23(33-2)14-24(12-19)34-3/h4-5,8-14H,6-7,15-16H2,1-3H3,(H,30,32)(H2,28,29,31)	JNGAZPQYKBUCDK-UHFFFAOYSA-N	468926	US10807959, Example B72	WD repeat-containing protein 5		 0.634								US Patent		10.7270/Q26Q219X		aid1804926	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468926	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468926&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370716	441571027							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968804	Cc1cc(ccn1)-c1cc(CNC2=NCCN2)cc(c1)C(=O)NCc1ccc(Cl)c(Cl)c1	InChI=1S/C24H23Cl2N5O/c1-15-8-18(4-5-27-15)19-9-17(14-31-24-28-6-7-29-24)10-20(12-19)23(32)30-13-16-2-3-21(25)22(26)11-16/h2-5,8-12H,6-7,13-14H2,1H3,(H,30,32)(H2,28,29,31)	VSNKYTAOGVJICV-UHFFFAOYSA-N	468927	US10807959, Example B74	WD repeat-containing protein 5		 0.031								US Patent		10.7270/Q26Q219X		aid1804926	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468927	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468927&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370909	441571028							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968805	Cc1cc(ccn1)-c1cc(CNC2=NCCN2)cc(c1)C(=O)NCc1cc(Cl)cc(Cl)c1	InChI=1S/C24H23Cl2N5O/c1-15-6-18(2-3-27-15)19-7-16(14-31-24-28-4-5-29-24)8-20(11-19)23(32)30-13-17-9-21(25)12-22(26)10-17/h2-3,6-12H,4-5,13-14H2,1H3,(H,30,32)(H2,28,29,31)	MYNLOOJXVUZZJO-UHFFFAOYSA-N	468928	US10807959, Example B81	WD repeat-containing protein 5		 0.033								US Patent		10.7270/Q26Q219X		aid1804926	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468928	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468928&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370748	441571029							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968806	Cc1cc(ccn1)-c1cc(CNC2=NCCN2)cc(c1)C(=O)NCc1ccc(Cl)c(C)c1	InChI=1S/C25H26ClN5O/c1-16-9-18(3-4-23(16)26)14-30-24(32)22-12-19(15-31-25-28-7-8-29-25)11-21(13-22)20-5-6-27-17(2)10-20/h3-6,9-13H,7-8,14-15H2,1-2H3,(H,30,32)(H2,28,29,31)	VBZCTAVYGIBEOE-UHFFFAOYSA-N	468929	US10807959, Example B84	WD repeat-containing protein 5		 0.118								US Patent		10.7270/Q26Q219X		aid1804926	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468929	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468929&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370926	441571030							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968807	Cc1ccncc1-c1cc(CNC2=NCCN2)cc(c1)C(=O)NCc1cc(Cl)cc(Cl)c1	InChI=1S/C24H23Cl2N5O/c1-15-2-3-27-14-22(15)18-6-16(13-31-24-28-4-5-29-24)7-19(10-18)23(32)30-12-17-8-20(25)11-21(26)9-17/h2-3,6-11,14H,4-5,12-13H2,1H3,(H,30,32)(H2,28,29,31)	YPIMYOAKPMWDPY-UHFFFAOYSA-N	468930	US10807959, Example B87	WD repeat-containing protein 5		 0.198								US Patent		10.7270/Q26Q219X		aid1804926	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468930	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468930&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370726	441571031							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968808	Cc1cc(CNC(=O)c2cc(CNC3=NCCN3)cc(c2)-c2cnccc2C)ccc1Cl	InChI=1S/C25H26ClN5O/c1-16-5-6-27-15-22(16)20-10-19(14-31-25-28-7-8-29-25)11-21(12-20)24(32)30-13-18-3-4-23(26)17(2)9-18/h3-6,9-12,15H,7-8,13-14H2,1-2H3,(H,30,32)(H2,28,29,31)	KSXRRLKDFXBULD-UHFFFAOYSA-N	468931	US10807959, Example B88	WD repeat-containing protein 5		 0.115								US Patent		10.7270/Q26Q219X		aid1804926	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468931	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468931&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370928	441571032							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968809	Cc1ccncc1-c1cc(CNC2=NCCN2)cc(c1)C(=O)NCc1cccc(F)n1	InChI=1S/C23H23FN6O/c1-15-5-6-25-14-20(15)17-9-16(12-29-23-26-7-8-27-23)10-18(11-17)22(31)28-13-19-3-2-4-21(24)30-19/h2-6,9-11,14H,7-8,12-13H2,1H3,(H,28,31)(H2,26,27,29)	RKTZSLKBHKADAX-UHFFFAOYSA-N	468932	US10807959, Example B89	WD repeat-containing protein 5		 4.39								US Patent		10.7270/Q26Q219X		aid1804926	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468932	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468932&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146371119	441571033							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968810	Cc1cc(C)cc(CNC(=O)c2cc(CNC3=NCCN3)cc(c2)-c2ccnc(C)c2)c1	InChI=1S/C26H29N5O/c1-17-8-18(2)10-20(9-17)15-30-25(32)24-13-21(16-31-26-28-6-7-29-26)12-23(14-24)22-4-5-27-19(3)11-22/h4-5,8-14H,6-7,15-16H2,1-3H3,(H,30,32)(H2,28,29,31)	VGFXTXQXAQWYHT-UHFFFAOYSA-N	468933	US10807959, Example B90	WD repeat-containing protein 5		 0.115								US Patent		10.7270/Q26Q219X		aid1804926	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468933	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468933&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370976	441571034							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968811	Cc1ccncc1-c1cc(CNC2=NCCN2)cc(c1)C(=O)NC(C1CC1)C1CC1	InChI=1S/C24H29N5O/c1-15-6-7-25-14-21(15)19-10-16(13-28-24-26-8-9-27-24)11-20(12-19)23(30)29-22(17-2-3-17)18-4-5-18/h6-7,10-12,14,17-18,22H,2-5,8-9,13H2,1H3,(H,29,30)(H2,26,27,28)	FSKCSXSVOVFUQT-UHFFFAOYSA-N	468934	US10807959, Example B93	WD repeat-containing protein 5		 0.759								US Patent		10.7270/Q26Q219X		aid1804926	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468934	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468934&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370870	441571035							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968812	Cc1cc(ccn1)-c1cc(CNC2=NCCN2)cc(c1)C(=O)NCc1cccc(F)n1	InChI=1S/C23H23FN6O/c1-15-9-17(5-6-25-15)18-10-16(13-29-23-26-7-8-27-23)11-19(12-18)22(31)28-14-20-3-2-4-21(24)30-20/h2-6,9-12H,7-8,13-14H2,1H3,(H,28,31)(H2,26,27,29)	MANJSKBUMZZKMP-UHFFFAOYSA-N	468935	US10807959, Example B95	WD repeat-containing protein 5		 6.10								US Patent		10.7270/Q26Q219X		aid1804926	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468935	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468935&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146371013	441571036							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968813	Cc1cc(cnc1F)-c1cc(CNC2=NCCN2)cc(c1)C(=O)NCc1ccc(Cl)c(Cl)c1	InChI=1S/C24H22Cl2FN5O/c1-14-6-19(13-30-22(14)27)17-7-16(12-32-24-28-4-5-29-24)8-18(10-17)23(33)31-11-15-2-3-20(25)21(26)9-15/h2-3,6-10,13H,4-5,11-12H2,1H3,(H,31,33)(H2,28,29,32)	XOTCGPMVFVNIDY-UHFFFAOYSA-N	468936	US10807959, Example B99	WD repeat-containing protein 5		 0.087								US Patent		10.7270/Q26Q219X		aid1804926	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468936	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468936&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370966	441571037							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968814	COc1ccc(CNC(=O)c2cc(CNC3=NCCN3)cc(c2)-c2cc(C)cnc2F)cc1OC	InChI=1S/C26H28FN5O3/c1-16-8-21(24(27)30-13-16)19-9-18(15-32-26-28-6-7-29-26)10-20(12-19)25(33)31-14-17-4-5-22(34-2)23(11-17)35-3/h4-5,8-13H,6-7,14-15H2,1-3H3,(H,31,33)(H2,28,29,32)	SUOUCMZYAGVKLI-UHFFFAOYSA-N	468937	US10807959, Example B107	WD repeat-containing protein 5		 0.097								US Patent		10.7270/Q26Q219X		aid1804926	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468937	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468937&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370979	441571038							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968815	COc1cc(CNC(=O)c2cc(CNC3=NCCN3)cc(c2)-c2cc(C)cnc2F)cc(OC)c1	InChI=1S/C26H28FN5O3/c1-16-6-23(24(27)30-13-16)19-7-17(15-32-26-28-4-5-29-26)8-20(11-19)25(33)31-14-18-9-21(34-2)12-22(10-18)35-3/h6-13H,4-5,14-15H2,1-3H3,(H,31,33)(H2,28,29,32)	LGWORMOAOLQTNI-UHFFFAOYSA-N	468938	US10807959, Example B109	WD repeat-containing protein 5		 0.038								US Patent		10.7270/Q26Q219X		aid1804926	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468938	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468938&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370756	441571039							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968816	Cc1cc(cc(C)n1)-c1cc(CNC2=NCCN2)cc(c1)C(=O)NCc1cc(Cl)ccn1	InChI=1S/C24H25ClN6O/c1-15-7-18(8-16(2)31-15)19-9-17(13-30-24-27-5-6-28-24)10-20(11-19)23(32)29-14-22-12-21(25)3-4-26-22/h3-4,7-12H,5-6,13-14H2,1-2H3,(H,29,32)(H2,27,28,30)	ULPDCSQAHIVFTA-UHFFFAOYSA-N	468939	US10807959, Example B111	WD repeat-containing protein 5		 0.087								US Patent		10.7270/Q26Q219X		aid1804926	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468939	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468939&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370852	441571040							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968817	COc1ccnc(CNC(=O)c2cc(CNC3=NCCN3)cc(c2)-c2ccc(F)cc2C)c1	InChI=1S/C25H26FN5O2/c1-16-9-20(26)3-4-23(16)18-10-17(14-31-25-28-7-8-29-25)11-19(12-18)24(32)30-15-21-13-22(33-2)5-6-27-21/h3-6,9-13H,7-8,14-15H2,1-2H3,(H,30,32)(H2,28,29,31)	RBDYJTGVBGRXOI-UHFFFAOYSA-N	468940	US10807959, Example B114	WD repeat-containing protein 5		 0.228								US Patent		10.7270/Q26Q219X		aid1804926	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468940	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468940&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370725	441571041							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968818	COc1ccnc(CNC(=O)c2cc(CNC3=NCCN3)cc(c2)-c2cc(OC)ccc2OC)c1	InChI=1S/C26H29N5O4/c1-33-21-4-5-24(35-3)23(14-21)18-10-17(15-31-26-28-8-9-29-26)11-19(12-18)25(32)30-16-20-13-22(34-2)6-7-27-20/h4-7,10-14H,8-9,15-16H2,1-3H3,(H,30,32)(H2,28,29,31)	HXNKXTZUPVGJSO-UHFFFAOYSA-N	468941	US10807959, Example B115	WD repeat-containing protein 5		 0.480								US Patent		10.7270/Q26Q219X		aid1804926	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468941	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468941&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370864	441571042							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968819	COc1ccnc(CNC(=O)c2cc(CNC3=NCCN3)cc(c2)-c2cc(Cl)ccc2OC)c1	InChI=1S/C25H26ClN5O3/c1-33-21-5-6-27-20(13-21)15-30-24(32)18-10-16(14-31-25-28-7-8-29-25)9-17(11-18)22-12-19(26)3-4-23(22)34-2/h3-6,9-13H,7-8,14-15H2,1-2H3,(H,30,32)(H2,28,29,31)	JKVKEQANQLVEIS-UHFFFAOYSA-N	468942	US10807959, Example B116	WD repeat-containing protein 5		 0.106								US Patent		10.7270/Q26Q219X		aid1804926	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468942	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468942&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146371061	441571043							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968820	COc1cc(OC)cc(c1)C(C)NC(=O)c1ccc(OC(C)C)c(CNC2=NCCC2)c1	InChI=1S/C25H33N3O4/c1-16(2)32-23-9-8-18(11-20(23)15-27-24-7-6-10-26-24)25(29)28-17(3)19-12-21(30-4)14-22(13-19)31-5/h8-9,11-14,16-17H,6-7,10,15H2,1-5H3,(H,26,27)(H,28,29)	LTXPBSNXQVNGBR-UHFFFAOYSA-N	468943	US10807959, Example B124	WD repeat-containing protein 5		>33.0								US Patent		10.7270/Q26Q219X		aid1804926	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468943	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468943&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370825	441571044							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968821	CC(C)Oc1ccc(cc1CNC1=NCCC1)C(=O)NCc1ccc(Cl)c(Cl)c1	InChI=1S/C22H25Cl2N3O2/c1-14(2)29-20-8-6-16(11-17(20)13-26-21-4-3-9-25-21)22(28)27-12-15-5-7-18(23)19(24)10-15/h5-8,10-11,14H,3-4,9,12-13H2,1-2H3,(H,25,26)(H,27,28)	LLQPMPAZRYLPOP-UHFFFAOYSA-N	468944	US10807959, Example B125	WD repeat-containing protein 5		>33.0								US Patent		10.7270/Q26Q219X		aid1804926	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468944	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468944&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370872	441571045							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968822	Cc1cc(CNC(=O)c2cc(CNC3=NCCC3)cc(c2)-c2ccc(F)nc2C)ccc1Cl	InChI=1S/C26H26ClFN4O/c1-16-10-18(5-7-23(16)27)14-31-26(33)21-12-19(15-30-25-4-3-9-29-25)11-20(13-21)22-6-8-24(28)32-17(22)2/h5-8,10-13H,3-4,9,14-15H2,1-2H3,(H,29,30)(H,31,33)	YBNBCZJVTIFSTL-UHFFFAOYSA-N	468945	US10807959, Example B129	WD repeat-containing protein 5		 0.089								US Patent		10.7270/Q26Q219X		aid1804926	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468945	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468945&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146371168	441571046							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968823	Fc1ccc(c(F)n1)-c1cc(CNC2=NCCN2)cc(n1)C(=O)NCc1ccc(Cl)c(Cl)c1	InChI=1S/C22H18Cl2F2N6O/c23-15-3-1-12(7-16(15)24)10-29-21(33)18-9-13(11-30-22-27-5-6-28-22)8-17(31-18)14-2-4-19(25)32-20(14)26/h1-4,7-9H,5-6,10-11H2,(H,29,33)(H2,27,28,30)	QASSMQFVSUYLIL-UHFFFAOYSA-N	468946	US10807959, Example C2	WD repeat-containing protein 5		 0.311								US Patent		10.7270/Q26Q219X		aid1804926	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468946	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468946&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370813	441571047							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968824	COc1cc(OC)cc(c1)C(C)NC(=O)c1cc(CNC2=NCCN2)ccn1	InChI=1S/C20H25N5O3/c1-13(15-9-16(27-2)11-17(10-15)28-3)25-19(26)18-8-14(4-5-21-18)12-24-20-22-6-7-23-20/h4-5,8-11,13H,6-7,12H2,1-3H3,(H,25,26)(H2,22,23,24)	IXZVYJPMBFWEGA-UHFFFAOYSA-N	468947	US10807959, Example C20	WD repeat-containing protein 5		 30.3								US Patent		10.7270/Q26Q219X		aid1804926	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468947	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468947&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370995	441571048							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968825	COc1cc(OC)cc(c1)C(C)NC(=O)c1cc(CNC2=NCCC2)ccn1	InChI=1S/C21H26N4O3/c1-14(16-10-17(27-2)12-18(11-16)28-3)25-21(26)19-9-15(6-8-22-19)13-24-20-5-4-7-23-20/h6,8-12,14H,4-5,7,13H2,1-3H3,(H,23,24)(H,25,26)	CYKGGYCIEPLUOT-UHFFFAOYSA-N	468948	US10807959, Example C21	WD repeat-containing protein 5		 33.0								US Patent		10.7270/Q26Q219X		aid1804926	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468948	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468948&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370839	441571049							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968826	Cc1cc(F)ccc1-c1cc(CNC2=NCCC2)cc(n1)C(=O)NCc1ccc(Cl)c(Cl)c1	InChI=1S/C25H23Cl2FN4O/c1-15-9-18(28)5-6-19(15)22-11-17(14-30-24-3-2-8-29-24)12-23(32-22)25(33)31-13-16-4-7-20(26)21(27)10-16/h4-7,9-12H,2-3,8,13-14H2,1H3,(H,29,30)(H,31,33)	VLDBYDNLSBWNGR-UHFFFAOYSA-N	468949	US10807959, Example C22	WD repeat-containing protein 5		 0.132								US Patent		10.7270/Q26Q219X		aid1804926	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468949	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468949&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370857	441571050							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968827	Cc1cc(CNC(=O)c2cc(CNC3=NCCC3)cc(n2)-c2ccc(F)cc2C)ccc1Cl	InChI=1S/C26H26ClFN4O/c1-16-11-20(28)6-7-21(16)23-12-19(15-30-25-4-3-9-29-25)13-24(32-23)26(33)31-14-18-5-8-22(27)17(2)10-18/h5-8,10-13H,3-4,9,14-15H2,1-2H3,(H,29,30)(H,31,33)	KLAPDQDOOFQMED-UHFFFAOYSA-N	468950	US10807959, Example C23	WD repeat-containing protein 5		 3.13								US Patent		10.7270/Q26Q219X		aid1804926	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468950	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468950&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370922	441571051							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968828	COc1cc(CNC(=O)c2cc(CNC3=NCCC3)cc(n2)-c2ccc(F)cc2C)cc(OC)c1	InChI=1S/C27H29FN4O3/c1-17-9-20(28)6-7-23(17)24-12-19(15-30-26-5-4-8-29-26)13-25(32-24)27(33)31-16-18-10-21(34-2)14-22(11-18)35-3/h6-7,9-14H,4-5,8,15-16H2,1-3H3,(H,29,30)(H,31,33)	DKSNUXWYZDDWQQ-UHFFFAOYSA-N	468951	US10807959, Example C24	WD repeat-containing protein 5		 11.7								US Patent		10.7270/Q26Q219X		aid1804926	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468951	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468951&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370951	441571052							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968829	COc1cc(CNC(=O)c2cc(CNC3=NCCC3)cc(n2)-c2ccc(F)cc2C(F)(F)F)cc(OC)c1	InChI=1S/C27H26F4N4O3/c1-37-19-8-16(9-20(13-19)38-2)15-34-26(36)24-11-17(14-33-25-4-3-7-32-25)10-23(35-24)21-6-5-18(28)12-22(21)27(29,30)31/h5-6,8-13H,3-4,7,14-15H2,1-2H3,(H,32,33)(H,34,36)	RCVOAEXGASLDFS-UHFFFAOYSA-N	468952	US10807959, Example C27	WD repeat-containing protein 5		 1.58								US Patent		10.7270/Q26Q219X		aid1804926	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468952	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468952&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370780	441571053							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968830	CC(NC(=O)c1cc(CNC2=NCCC2)cc(n1)-c1ccc(F)cc1C(F)(F)F)c1cc(Cl)c(C)cn1	InChI=1S/C26H24ClF4N5O/c1-14-12-33-21(11-20(14)27)15(2)35-25(37)23-9-16(13-34-24-4-3-7-32-24)8-22(36-23)18-6-5-17(28)10-19(18)26(29,30)31/h5-6,8-12,15H,3-4,7,13H2,1-2H3,(H,32,34)(H,35,37)	GGNJNUANYNKKTH-UHFFFAOYSA-N	468953	US10807959, Example C32	WD repeat-containing protein 5		 1.54								US Patent		10.7270/Q26Q219X		aid1804926	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468953	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468953&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370833	441571054							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968831	COc1cc(OC)cc(c1)C(C)NC(=O)c1ccnc(CNC2=NCCN2)c1	InChI=1S/C20H25N5O3/c1-13(15-9-17(27-2)11-18(10-15)28-3)25-19(26)14-4-5-21-16(8-14)12-24-20-22-6-7-23-20/h4-5,8-11,13H,6-7,12H2,1-3H3,(H,25,26)(H2,22,23,24)	MIOAPNYQUINMCL-UHFFFAOYSA-N	468954	US10807959, Example C34	WD repeat-containing protein 5		 32.5								US Patent		10.7270/Q26Q219X		aid1804926	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468954	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468954&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370977	441571055							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
968832	COc1cc(OC)cc(c1)C(C)NC(=O)c1ccnc(CNC2=NCCC2)c1	InChI=1S/C21H26N4O3/c1-14(16-10-18(27-2)12-19(11-16)28-3)25-21(26)15-6-8-22-17(9-15)13-24-20-5-4-7-23-20/h6,8-12,14H,4-5,7,13H2,1-3H3,(H,23,24)(H,25,26)	BUZLFLQVPAQLMZ-UHFFFAOYSA-N	468955	US10807959, Example C35	WD repeat-containing protein 5		 44.1								US Patent		10.7270/Q26Q219X		aid1804926	US10807959	Gogliotti, RD; Stauffer, SR; Jeon, K; Salovich, JM; Macdonald, JD; Mills, JJ; Meyers, KM; Alvarado, JR; Han, C; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468955	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468955&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146370811	441571056							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981627	Cc1cc(ccc1F)[C@@H](NC(=O)c1cc(CN2CCCC2=N)cc(c1)-c1ccc(F)cc1C#N)C1CC1	InChI=1S/C30H28F2N4O/c1-18-11-21(6-9-27(18)32)29(20-4-5-20)35-30(37)23-13-19(17-36-10-2-3-28(36)34)12-22(14-23)26-8-7-25(31)15-24(26)16-33/h6-9,11-15,20,29,34H,2-5,10,17H2,1H3,(H,35,37)/t29-/m0/s1	REZJSVQUKQTLGY-LJAQVGFWSA-N	473427	US10844044, Example 333	WD repeat-containing protein 5		 0.390								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473427	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473427&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146457758	442073636							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981628	Cc1cc(CNC(=O)c2cc(Cn3ccn(C)c3=N)cc(c2)-c2c(C)cc(F)cc2C)ccc1Cl	InChI=1S/C28H28ClFN4O/c1-17-9-20(5-6-25(17)29)15-32-27(35)23-13-21(16-34-8-7-33(4)28(34)31)12-22(14-23)26-18(2)10-24(30)11-19(26)3/h5-14,31H,15-16H2,1-4H3,(H,32,35)	ZVARUBKVNDTQCA-UHFFFAOYSA-N	473428	US10844044, Example 59	WD repeat-containing protein 5		 0.580								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473428	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473428&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146457641	442073637							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981629	Cn1ccn(Cc2cc(cc(c2)-c2ccc(F)cc2OC(F)F)C(=O)N[C@@H](C2CC2)c2ccc(Cl)c(Cl)c2)c1=N	InChI=1S/C29H25Cl2F3N4O2/c1-37-8-9-38(29(37)35)15-16-10-19(22-6-5-21(32)14-25(22)40-28(33)34)12-20(11-16)27(39)36-26(17-2-3-17)18-4-7-23(30)24(31)13-18/h4-14,17,26,28,35H,2-3,15H2,1H3,(H,36,39)/t26-/m0/s1	ILEAUHIFGBSRKK-SANMLTNESA-N	473429	US10844044, Example 150	WD repeat-containing protein 5		 0.130								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473429	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473429&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456241	442073638							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981630	Cc1cc(ccc1F)[C@@H](NC(=O)c1cc(Cn2ccoc2=N)cc(c1)-c1ncc(F)cc1C(F)(F)F)C1CC1	InChI=1S/C28H23F5N4O2/c1-15-8-18(4-5-23(15)30)24(17-2-3-17)36-26(38)20-10-16(14-37-6-7-39-27(37)34)9-19(11-20)25-22(28(31,32)33)12-21(29)13-35-25/h4-13,17,24,34H,2-3,14H2,1H3,(H,36,38)/t24-/m0/s1	OYLPPMAEYXOWRU-DEOSSOPVSA-N	473430	US10844044, Example 241	WD repeat-containing protein 5		 6.00								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473430	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473430&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146455723	442073639							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981631	Cc1cc(ccc1F)[C@@H](NC(=O)c1cc(CN2CCCC2=N)cc(c1)-c1cccnc1C(F)(F)F)C1CC1	InChI=1S/C29H28F4N4O/c1-17-12-20(8-9-24(17)30)26(19-6-7-19)36-28(38)22-14-18(16-37-11-3-5-25(37)34)13-21(15-22)23-4-2-10-35-27(23)29(31,32)33/h2,4,8-10,12-15,19,26,34H,3,5-7,11,16H2,1H3,(H,36,38)/t26-/m0/s1	UXMPAEDRDCLWDA-SANMLTNESA-N	473431	US10844044, Example 334	WD repeat-containing protein 5		<0.100								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473431	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473431&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456213	442073640							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981632	Cc1cc(ccc1F)[C@@H](NC(=O)c1cc(Cn2ccn(C)c2=N)cc(c1)-c1cccnc1C(F)(F)F)C1CC1	InChI=1S/C29H27F4N5O/c1-17-12-20(7-8-24(17)30)25(19-5-6-19)36-27(39)22-14-18(16-38-11-10-37(2)28(38)34)13-21(15-22)23-4-3-9-35-26(23)29(31,32)33/h3-4,7-15,19,25,34H,5-6,16H2,1-2H3,(H,36,39)/t25-/m0/s1	SGNRQWMFJWIFSN-VWLOTQADSA-N	473432	US10844044, Example 60	WD repeat-containing protein 5		<0.100								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473432	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473432&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456640	442073641							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981633	FC(F)Oc1cc(F)ccc1-c1cc(Cn2ccn(C3CC3)c2=N)cc(c1)C(=O)N[C@@H](C1CC1)c1ccc(Cl)c(Cl)c1	InChI=1S/C31H27Cl2F3N4O2/c32-25-8-3-19(14-26(25)33)28(18-1-2-18)38-29(41)21-12-17(16-39-9-10-40(31(39)37)23-5-6-23)11-20(13-21)24-7-4-22(34)15-27(24)42-30(35)36/h3-4,7-15,18,23,28,30,37H,1-2,5-6,16H2,(H,38,41)/t28-/m0/s1	CWMNWRNMZSVIAE-NDEPHWFRSA-N	473433	US10844044, Example 151	WD repeat-containing protein 5		 0.590								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473433	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473433&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456626	442073642							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981634	Cc1cc(ccc1F)[C@@H](NC(=O)c1cc(Cn2ccoc2=N)cc(c1)-c1ccc(F)cc1OC(F)F)C1CC1	InChI=1S/C29H25F4N3O3/c1-16-10-19(4-7-24(16)31)26(18-2-3-18)35-27(37)21-12-17(15-36-8-9-38-29(36)34)11-20(13-21)23-6-5-22(30)14-25(23)39-28(32)33/h4-14,18,26,28,34H,2-3,15H2,1H3,(H,35,37)/t26-/m0/s1	UJSYVEZBFLFOKK-SANMLTNESA-N	473434	US10844044, Example 242	WD repeat-containing protein 5		<0.100								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473434	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473434&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456018	442073643							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981635	Cc1cc(ccc1F)[C@@H](NC(=O)c1cc(CN2CCCC2=N)cc(c1)-c1ccc(F)cc1C(F)(F)F)C1CC1	InChI=1S/C30H28F5N3O/c1-17-11-20(6-9-26(17)32)28(19-4-5-19)37-29(39)22-13-18(16-38-10-2-3-27(38)36)12-21(14-22)24-8-7-23(31)15-25(24)30(33,34)35/h6-9,11-15,19,28,36H,2-5,10,16H2,1H3,(H,37,39)/t28-/m0/s1	NZCKPPNHSKBSRH-NDEPHWFRSA-N	473435	US10844044, Example 335	WD repeat-containing protein 5		<0.100								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473435	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473435&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146455900	442073644							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981636	COc1cc(OC)cc(c1)C(NC(=O)c1cc(Cn2ccn(C)c2=N)cc(c1)-c1ncccc1C(F)(F)F)C1CC1	InChI=1S/C30H30F3N5O3/c1-37-9-10-38(29(37)34)17-18-11-20(27-25(30(31,32)33)5-4-8-35-27)13-22(12-18)28(39)36-26(19-6-7-19)21-14-23(40-2)16-24(15-21)41-3/h4-5,8-16,19,26,34H,6-7,17H2,1-3H3,(H,36,39)	VUYWIXWYXGOUCX-UHFFFAOYSA-N	473436	US10844044, Example 61	WD repeat-containing protein 5		 2.80								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473436	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473436&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146455899	442073645							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981637	COc1cc(CNC(=O)c2cc(CN3CCN(C)C3=N)cc(c2)-c2ccc(F)cc2C(N)=O)cc(OC)c1	InChI=1S/C28H30FN5O4/c1-33-6-7-34(28(33)31)16-18-8-19(24-5-4-21(29)13-25(24)26(30)35)12-20(9-18)27(36)32-15-17-10-22(37-2)14-23(11-17)38-3/h4-5,8-14,31H,6-7,15-16H2,1-3H3,(H2,30,35)(H,32,36)	BPAWGPCRDIVHJR-UHFFFAOYSA-N	473437	US10844044, Example 152	WD repeat-containing protein 5		 8.90								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473437	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473437&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146488137	442073646							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981638	Cc1cc(ccc1F)[C@@H](NC(=O)c1cc(Cn2ccoc2=N)cc(c1)-c1cccnc1C(F)(F)F)C1CC1	InChI=1S/C28H24F4N4O2/c1-16-11-19(6-7-23(16)29)24(18-4-5-18)35-26(37)21-13-17(15-36-9-10-38-27(36)33)12-20(14-21)22-3-2-8-34-25(22)28(30,31)32/h2-3,6-14,18,24,33H,4-5,15H2,1H3,(H,35,37)/t24-/m0/s1	GWWDUHVBMCFSGI-DEOSSOPVSA-N	473438	US10844044, Example 243	WD repeat-containing protein 5		<0.100								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473438	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473438&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456689	442073647							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981639	CC(C)n1cc(c(n1)C(F)(F)F)-c1cc(CN2CCCC2=N)cc(c1)C(=O)N[C@@H](C1CC1)c1ccc(F)c(C)c1	InChI=1S/C30H33F4N5O/c1-17(2)39-16-24(28(37-39)30(32,33)34)22-12-19(15-38-10-4-5-26(38)35)13-23(14-22)29(40)36-27(20-6-7-20)21-8-9-25(31)18(3)11-21/h8-9,11-14,16-17,20,27,35H,4-7,10,15H2,1-3H3,(H,36,40)/t27-/m0/s1	PQZMAGZYXLBTIG-MHZLTWQESA-N	473439	US10844044, Example 336	WD repeat-containing protein 5		<0.100								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473439	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473439&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146455830	442073648							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981640	COc1cc(CNC(=O)c2cc(Cn3ccn(C)c3=N)cc(c2)-c2ccc(F)cc2OC(F)F)cc(OC)c1	InChI=1S/C28H27F3N4O4/c1-34-6-7-35(28(34)32)16-18-8-19(24-5-4-21(29)13-25(24)39-27(30)31)12-20(9-18)26(36)33-15-17-10-22(37-2)14-23(11-17)38-3/h4-14,27,32H,15-16H2,1-3H3,(H,33,36)	AWOCAJBZUOFJRD-UHFFFAOYSA-N	473440	US10844044, Example 62	WD repeat-containing protein 5		 0.290								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473440	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473440&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146455800	442073649							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981641	Cn1ccn(Cc2cc(cc(c2)-c2cccnc2C(F)(F)F)C(=O)N[C@@H](C2CC2)c2ccc(Cl)c(Cl)c2)c1=N	InChI=1S/C28H24Cl2F3N5O/c1-37-9-10-38(27(37)34)15-16-11-19(21-3-2-8-35-25(21)28(31,32)33)13-20(12-16)26(39)36-24(17-4-5-17)18-6-7-22(29)23(30)14-18/h2-3,6-14,17,24,34H,4-5,15H2,1H3,(H,36,39)/t24-/m0/s1	GKPIIXJEQYEOKD-DEOSSOPVSA-N	473441	US10844044, Example 153	WD repeat-containing protein 5		 0.330								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473441	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473441&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146455894	442073650							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981642	COc1cc(CNC(=O)c2cc(Cn3ccoc3=N)cc(c2)-c2cccnc2C(F)(F)F)cc(OC)c1	InChI=1S/C26H23F3N4O4/c1-35-20-10-16(11-21(13-20)36-2)14-32-24(34)19-9-17(15-33-6-7-37-25(33)30)8-18(12-19)22-4-3-5-31-23(22)26(27,28)29/h3-13,30H,14-15H2,1-2H3,(H,32,34)	WJMWNKWEATWYRG-UHFFFAOYSA-N	473442	US10844044, Example 244	WD repeat-containing protein 5		<0.100								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473442	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473442&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146455820	442073651							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981643	Cc1cc(ccc1F)[C@@H](NC(=O)c1cc(CN2CCCC2=N)cc(c1)-c1cn(C)nc1C(F)(F)F)C1CC1	InChI=1S/C28H29F4N5O/c1-16-10-19(7-8-23(16)29)25(18-5-6-18)34-27(38)21-12-17(14-37-9-3-4-24(37)33)11-20(13-21)22-15-36(2)35-26(22)28(30,31)32/h7-8,10-13,15,18,25,33H,3-6,9,14H2,1-2H3,(H,34,38)/t25-/m0/s1	LOOUMNIFSXYYJY-VWLOTQADSA-N	473443	US10844044, Example 337	WD repeat-containing protein 5		<0.100								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473443	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473443&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146455937	442073652							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981644	COc1cc(OC)cc(c1)C(NC(=O)c1cc(Cn2ccn(C)c2=N)cc(c1)-c1ccc(F)cc1OC(F)F)C1CC1	InChI=1S/C31H31F3N4O4/c1-37-8-9-38(31(37)35)17-18-10-20(26-7-6-23(32)15-27(26)42-30(33)34)12-22(11-18)29(39)36-28(19-4-5-19)21-13-24(40-2)16-25(14-21)41-3/h6-16,19,28,30,35H,4-5,17H2,1-3H3,(H,36,39)	UPYQUJZTFXEWMR-UHFFFAOYSA-N	473444	US10844044, Example 63	WD repeat-containing protein 5		 0.100								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473444	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473444&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146455833	442073653							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981645	Cc1cc(ccc1F)[C@@H](NC(=O)c1cc(Cn2ccn(C)c2=N)cc(c1)-c1ccc(F)cc1C(F)F)C1CC1	InChI=1S/C30H28F4N4O/c1-17-11-20(5-8-26(17)32)27(19-3-4-19)36-29(39)22-13-18(16-38-10-9-37(2)30(38)35)12-21(14-22)24-7-6-23(31)15-25(24)28(33)34/h5-15,19,27-28,35H,3-4,16H2,1-2H3,(H,36,39)/t27-/m0/s1	FKEDSTGSVSSBBI-MHZLTWQESA-N	473445	US10844044, Example 154	WD repeat-containing protein 5		<0.100								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473445	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473445&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146455769	442073654							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981646	COc1cc(OC)cc(c1)C(NC(=O)c1cc(Cn2ccoc2=N)cc(c1)-c1cccnc1C(F)(F)F)C1CC1	InChI=1S/C29H27F3N4O4/c1-38-22-13-20(14-23(15-22)39-2)25(18-5-6-18)35-27(37)21-11-17(16-36-8-9-40-28(36)33)10-19(12-21)24-4-3-7-34-26(24)29(30,31)32/h3-4,7-15,18,25,33H,5-6,16H2,1-2H3,(H,35,37)	WTIDKCAWSGFSIE-UHFFFAOYSA-N	473446	US10844044, Example 245	WD repeat-containing protein 5		<0.100								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473446	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473446&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456869	442073655							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981647	CCn1cc(c(n1)C(F)(F)F)-c1cc(CN2CCCC2=N)cc(c1)C(=O)N[C@@H](C1CC1)c1ccc(F)c(Cl)c1	InChI=1S/C28H28ClF4N5O/c1-2-38-15-21(26(36-38)28(31,32)33)19-10-16(14-37-9-3-4-24(37)34)11-20(12-19)27(39)35-25(17-5-6-17)18-7-8-23(30)22(29)13-18/h7-8,10-13,15,17,25,34H,2-6,9,14H2,1H3,(H,35,39)/t25-/m0/s1	GBODVALIPVDSSV-VWLOTQADSA-N	473447	US10844044, Example 338	WD repeat-containing protein 5		<0.100								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473447	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473447&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146455736	442073656							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981648	Cc1cc(ccc1F)[C@@H](NC(=O)c1cc(Cn2ccn(C)c2=N)cc(c1)-c1ncccc1C(F)(F)F)C1CC1	InChI=1S/C29H27F4N5O/c1-17-12-20(7-8-24(17)30)25(19-5-6-19)36-27(39)22-14-18(16-38-11-10-37(2)28(38)34)13-21(15-22)26-23(29(31,32)33)4-3-9-35-26/h3-4,7-15,19,25,34H,5-6,16H2,1-2H3,(H,36,39)/t25-/m0/s1	TTWKUXCHTKWRNP-VWLOTQADSA-N	473448	US10844044, Example 64	WD repeat-containing protein 5		 0.590								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473448	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473448&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146455933	442073657							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981649	FC(F)(F)c1ncccc1-c1cc(Cn2ccn(C3CC3)c2=N)cc(c1)C(=O)N[C@@H](C1CC1)c1ccc(Cl)c(Cl)c1	InChI=1S/C30H26Cl2F3N5O/c31-24-8-5-19(15-25(24)32)26(18-3-4-18)38-28(41)21-13-17(16-39-10-11-40(29(39)36)22-6-7-22)12-20(14-21)23-2-1-9-37-27(23)30(33,34)35/h1-2,5,8-15,18,22,26,36H,3-4,6-7,16H2,(H,38,41)/t26-/m0/s1	VLPHQBIZSYBWOX-SANMLTNESA-N	473449	US10844044, Example 155	WD repeat-containing protein 5		 1.40								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473449	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473449&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146455760	442073658							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981650	Cc1cc(F)ccc1-c1cc(Cn2ccoc2=N)cc(c1)C(=O)NCc1ccc(F)cc1	InChI=1S/C25H21F2N3O2/c1-16-10-22(27)6-7-23(16)19-11-18(15-30-8-9-32-25(30)28)12-20(13-19)24(31)29-14-17-2-4-21(26)5-3-17/h2-13,28H,14-15H2,1H3,(H,29,31)	GTHLFECYAKIOBB-UHFFFAOYSA-N	473450	US10844044, Example 246	WD repeat-containing protein 5		 182								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473450	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473450&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146455771	442073659							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981651	COc1cc(ccc1F)[C@@H](NC(=O)c1cc(CN2CCCC2=N)cc(c1)-c1cn(C)nc1C(F)(F)F)C1CC1	InChI=1S/C28H29F4N5O2/c1-36-15-21(26(35-36)28(30,31)32)19-10-16(14-37-9-3-4-24(37)33)11-20(12-19)27(38)34-25(17-5-6-17)18-7-8-22(29)23(13-18)39-2/h7-8,10-13,15,17,25,33H,3-6,9,14H2,1-2H3,(H,34,38)/t25-/m0/s1	MOGMWQNFULMKHJ-VWLOTQADSA-N	473451	US10844044, Example 339	WD repeat-containing protein 5		<0.100								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473451	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473451&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146455877	442073660							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981652	COc1cc(CNC(=O)c2cc(Cn3ccn(C)c3=N)cc(c2)-c2c(C)cc(F)cc2C)cc(OC)c1	InChI=1S/C29H31FN4O3/c1-18-8-24(30)9-19(2)27(18)22-10-21(17-34-7-6-33(3)29(34)31)11-23(14-22)28(35)32-16-20-12-25(36-4)15-26(13-20)37-5/h6-15,31H,16-17H2,1-5H3,(H,32,35)	XJZNKYPGIBYVEP-UHFFFAOYSA-N	473452	US10844044, Example 65	WD repeat-containing protein 5		 0.630								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473452	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473452&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456911	442073661							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981653	Cc1cc(ccc1F)[C@@H](NC(=O)c1cc(Cn2ccn(C3CC3)c2=N)cc(c1)-c1ccc(F)cc1OC(F)F)C1CC1	InChI=1S/C32H30F4N4O2/c1-18-12-21(4-9-27(18)34)29(20-2-3-20)38-30(41)23-14-19(17-39-10-11-40(32(39)37)25-6-7-25)13-22(15-23)26-8-5-24(33)16-28(26)42-31(35)36/h4-5,8-16,20,25,29,31,37H,2-3,6-7,17H2,1H3,(H,38,41)/t29-/m0/s1	LEQVYIWJXDYGSU-LJAQVGFWSA-N	473453	US10844044, Example 156	WD repeat-containing protein 5		<0.100								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473453	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473453&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146457664	442073662							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981654	Cc1ccnc(c1)[C@@H](NC(=O)c1cc(Cn2ccoc2=N)cc(c1)-c1ccc(F)cc1C)C1CC1	InChI=1S/C28H27FN4O2/c1-17-7-8-31-25(11-17)26(20-3-4-20)32-27(34)22-14-19(16-33-9-10-35-28(33)30)13-21(15-22)24-6-5-23(29)12-18(24)2/h5-15,20,26,30H,3-4,16H2,1-2H3,(H,32,34)/t26-/m0/s1	VZRQXNCQAZNAPQ-SANMLTNESA-N	473454	US10844044, Example 247	WD repeat-containing protein 5		 0.140								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473454	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473454&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456693	442073663							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981655	Fc1ccc(cc1Cl)[C@@H](NC(=O)c1cc(CN2CCCC2=N)cc(c1)-c1cccnc1C(F)(F)F)C1CC1	InChI=1S/C28H25ClF4N4O/c29-22-14-18(7-8-23(22)30)25(17-5-6-17)36-27(38)20-12-16(15-37-10-2-4-24(37)34)11-19(13-20)21-3-1-9-35-26(21)28(31,32)33/h1,3,7-9,11-14,17,25,34H,2,4-6,10,15H2,(H,36,38)/t25-/m0/s1	YFXVXPBFEUAGCL-VWLOTQADSA-N	473455	US10844044, Example 340	WD repeat-containing protein 5		<0.100								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473455	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473455&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146455730	442073664							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981656	Cc1cc(ccc1F)[C@@H](NC(=O)c1cc(Cn2ccn(C)c2=N)cc(c1)-c1ncc(F)cc1C)C1CC1	InChI=1S/C29H29F2N5O/c1-17-10-21(6-7-25(17)31)27(20-4-5-20)34-28(37)23-13-19(16-36-9-8-35(3)29(36)32)12-22(14-23)26-18(2)11-24(30)15-33-26/h6-15,20,27,32H,4-5,16H2,1-3H3,(H,34,37)/t27-/m0/s1	CGDWGNCJPSMSRS-MHZLTWQESA-N	473456	US10844044, Example 66	WD repeat-containing protein 5		 0.120								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473456	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473456&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146457578	442073665							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981657	Cn1cc(c(n1)C(F)(F)F)-c1cc(Cn2ccn(C)c2=N)cc(c1)C(=O)N[C@@H](C1CC1)c1ccc(Cl)c(Cl)c1	InChI=1S/C27H25Cl2F3N6O/c1-36-7-8-38(26(36)33)13-15-9-18(20-14-37(2)35-24(20)27(30,31)32)11-19(10-15)25(39)34-23(16-3-4-16)17-5-6-21(28)22(29)12-17/h5-12,14,16,23,33H,3-4,13H2,1-2H3,(H,34,39)/t23-/m0/s1	XXBDHHUZDWANQK-QHCPKHFHSA-N	473306	US10844044, Example 157::US10844044, Example 211	WD repeat-containing protein 5		<0.100								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473306	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473306&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456260	442073518							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981658	Cc1cc(ccc1F)[C@@H](NC(=O)c1cc(Cn2ccoc2=N)cc(c1)-c1ccc(F)cc1Cl)C1CC1	InChI=1S/C28H24ClF2N3O2/c1-16-10-19(4-7-25(16)31)26(18-2-3-18)33-27(35)21-12-17(15-34-8-9-36-28(34)32)11-20(13-21)23-6-5-22(30)14-24(23)29/h4-14,18,26,32H,2-3,15H2,1H3,(H,33,35)/t26-/m0/s1	DUUWVNRYTWFKKS-SANMLTNESA-N	473458	US10844044, Example 248	WD repeat-containing protein 5		<0.100								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473458	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473458&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456119	442073666							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981659	Cn1cc(c(n1)C(F)(F)F)-c1cc(CN2CCCC2=N)cc(c1)C(=O)N[C@@H](C1CC1)c1ccc(F)c(F)c1	InChI=1S/C27H26F5N5O/c1-36-14-20(25(35-36)27(30,31)32)18-9-15(13-37-8-2-3-23(37)33)10-19(11-18)26(38)34-24(16-4-5-16)17-6-7-21(28)22(29)12-17/h6-7,9-12,14,16,24,33H,2-5,8,13H2,1H3,(H,34,38)/t24-/m0/s1	DPXMABMSVGGUBP-DEOSSOPVSA-N	473459	US10844044, Example 341	WD repeat-containing protein 5		 0.350								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473459	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473459&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146455975	442073667							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981660	COc1cc(CNC(=O)c2cc(Cn3ccn(C)c3=N)cc(c2)-c2ncc(F)cc2C)cc(OC)c1	InChI=1S/C27H28FN5O3/c1-17-7-22(28)15-30-25(17)20-8-19(16-33-6-5-32(2)27(33)29)9-21(12-20)26(34)31-14-18-10-23(35-3)13-24(11-18)36-4/h5-13,15,29H,14,16H2,1-4H3,(H,31,34)	XOILHYOBVIIZAD-UHFFFAOYSA-N	473460	US10844044, Example 67	WD repeat-containing protein 5		 3.90								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473460	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473460&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456208	442073668							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981661	Cc1cc(ccc1F)[C@@H](NC(=O)c1cc(Cn2ccn(C3CC3)c2=N)cc(c1)-c1ccc(F)cc1C(F)F)C1CC1	InChI=1S/C32H30F4N4O/c1-18-12-21(4-9-28(18)34)29(20-2-3-20)38-31(41)23-14-19(17-39-10-11-40(32(39)37)25-6-7-25)13-22(15-23)26-8-5-24(33)16-27(26)30(35)36/h4-5,8-16,20,25,29-30,37H,2-3,6-7,17H2,1H3,(H,38,41)/t29-/m0/s1	KOWVTLHTXOKLBE-LJAQVGFWSA-N	473461	US10844044, Example 158	WD repeat-containing protein 5		<0.100								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473461	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473461&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146457599	442073669							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981662	COc1cc(OC)cc(c1)[C@@H](NC(=O)c1cc(Cn2ccoc2=N)cc(c1)-c1ccc(F)cc1Cl)C1CC1	InChI=1S/C29H27ClFN3O4/c1-36-23-12-20(13-24(15-23)37-2)27(18-3-4-18)33-28(35)21-10-17(16-34-7-8-38-29(34)32)9-19(11-21)25-6-5-22(31)14-26(25)30/h5-15,18,27,32H,3-4,16H2,1-2H3,(H,33,35)/t27-/m0/s1	FOGXPJTXBQLIJC-MHZLTWQESA-N	473462	US10844044, Example 249	WD repeat-containing protein 5		<0.100								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473462	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473462&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146488071	442073670							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981663	Cc1cc(ccc1F)[C@@H](NC(=O)c1cc(Cn2ccccc2=N)cc(c1)-c1cccnc1C(F)(F)F)C1CC1	InChI=1S/C30H26F4N4O/c1-18-13-21(9-10-25(18)31)27(20-7-8-20)37-29(39)23-15-19(17-38-12-3-2-6-26(38)35)14-22(16-23)24-5-4-11-36-28(24)30(32,33)34/h2-6,9-16,20,27,35H,7-8,17H2,1H3,(H,37,39)/t27-/m0/s1	QDLSYEFQYLCDRD-MHZLTWQESA-N	473463	US10844044, Example 342	WD repeat-containing protein 5		<0.100								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473463	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473463&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146455795	442073671							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981664	COc1cc(OC)cc(c1)C(NC(=O)c1cc(Cn2ccn(C)c2=N)cc(c1)-c1ncc(F)cc1C)C1CC1	InChI=1S/C30H32FN5O3/c1-18-9-24(31)16-33-27(18)21-10-19(17-36-8-7-35(2)30(36)32)11-23(12-21)29(37)34-28(20-5-6-20)22-13-25(38-3)15-26(14-22)39-4/h7-16,20,28,32H,5-6,17H2,1-4H3,(H,34,37)	LKDDJMIQNDTUER-UHFFFAOYSA-N	473464	US10844044, Example 68	WD repeat-containing protein 5		 0.350								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473464	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473464&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456837	442073672							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981665	Cn1cc(c(n1)C(F)(F)F)-c1cc(Cn2ccn(C3CC3)c2=N)cc(c1)C(=O)N[C@@H](C1CC1)c1ccc(Cl)c(Cl)c1	InChI=1S/C29H27Cl2F3N6O/c1-38-15-22(26(37-38)29(32,33)34)19-10-16(14-39-8-9-40(28(39)35)21-5-6-21)11-20(12-19)27(41)36-25(17-2-3-17)18-4-7-23(30)24(31)13-18/h4,7-13,15,17,21,25,35H,2-3,5-6,14H2,1H3,(H,36,41)/t25-/m0/s1	DDTPVLWBWABVCK-VWLOTQADSA-N	473465	US10844044, Example 159	WD repeat-containing protein 5		<0.100								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473465	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473465&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456862	442073673							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981666	Cc1cn(Cc2cc(cc(c2)-c2cccnc2C(F)(F)F)C(=O)N[C@@H](C2CC2)c2ccc(F)c(C)c2)c(=N)o1	InChI=1S/C29H26F4N4O2/c1-16-10-20(7-8-24(16)30)25(19-5-6-19)36-27(38)22-12-18(15-37-14-17(2)39-28(37)34)11-21(13-22)23-4-3-9-35-26(23)29(31,32)33/h3-4,7-14,19,25,34H,5-6,15H2,1-2H3,(H,36,38)/t25-/m0/s1	GTAXNVHXDZGRPI-VWLOTQADSA-N	473466	US10844044, Example 250	WD repeat-containing protein 5		 0.400								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473466	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473466&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146455802	442073674							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981667	Cc1cc(ccc1F)[C@@H](NC(=O)c1cc(Cn2cccc(C)c2=N)cc(c1)-c1cccnc1C(F)(F)F)C1CC1	InChI=1S/C31H28F4N4O/c1-18-5-4-12-39(29(18)36)17-20-14-23(25-6-3-11-37-28(25)31(33,34)35)16-24(15-20)30(40)38-27(21-7-8-21)22-9-10-26(32)19(2)13-22/h3-6,9-16,21,27,36H,7-8,17H2,1-2H3,(H,38,40)/t27-/m0/s1	MOZDLJWPFJKYMU-MHZLTWQESA-N	473467	US10844044, Example 343	WD repeat-containing protein 5		 0.510								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473467	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473467&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456307	442073675							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981668	Cc1ccnc(c1)C(NC(=O)c1cc(Cn2ccn(C)c2=N)cc(c1)-c1ncc(F)cc1C)C1CC1	InChI=1S/C28H29FN6O/c1-17-6-7-31-24(10-17)26(20-4-5-20)33-27(36)22-13-19(16-35-9-8-34(3)28(35)30)12-21(14-22)25-18(2)11-23(29)15-32-25/h6-15,20,26,30H,4-5,16H2,1-3H3,(H,33,36)	LDGUOTOZOKQTEP-UHFFFAOYSA-N	473468	US10844044, Example 69	WD repeat-containing protein 5		 2.40								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473468	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473468&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146455747	442073676							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981669	CCn1cc(c(n1)C(F)(F)F)-c1cc(Cn2ccn(C3CC3)c2=N)cc(c1)C(=O)N[C@@H](C1CC1)c1ccc(F)c(C)c1	InChI=1S/C31H32F4N6O/c1-3-40-17-25(28(38-40)31(33,34)35)22-13-19(16-39-10-11-41(30(39)36)24-7-8-24)14-23(15-22)29(42)37-27(20-4-5-20)21-6-9-26(32)18(2)12-21/h6,9-15,17,20,24,27,36H,3-5,7-8,16H2,1-2H3,(H,37,42)/t27-/m0/s1	ZHFRZJNBNLFRLW-MHZLTWQESA-N	473469	US10844044, Example 160	WD repeat-containing protein 5		<0.100								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473469	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473469&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456063	442073677							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981670	CCc1cn(Cc2cc(cc(c2)-c2cccnc2C(F)(F)F)C(=O)N[C@@H](C2CC2)c2ccc(F)c(C)c2)c(=N)o1	InChI=1S/C30H28F4N4O2/c1-3-23-16-38(29(35)40-23)15-18-12-21(24-5-4-10-36-27(24)30(32,33)34)14-22(13-18)28(39)37-26(19-6-7-19)20-8-9-25(31)17(2)11-20/h4-5,8-14,16,19,26,35H,3,6-7,15H2,1-2H3,(H,37,39)/t26-/m0/s1	NKRZATRXQOEPTO-SANMLTNESA-N	473470	US10844044, Example 251	WD repeat-containing protein 5		 1.24								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473470	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473470&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456272	442073678							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981671	Cc1ccn(Cc2cc(cc(c2)-c2cccnc2C(F)(F)F)C(=O)N[C@@H](C2CC2)c2ccc(F)c(C)c2)c(=N)c1	InChI=1S/C31H28F4N4O/c1-18-9-11-39(27(36)12-18)17-20-14-23(25-4-3-10-37-29(25)31(33,34)35)16-24(15-20)30(40)38-28(21-5-6-21)22-7-8-26(32)19(2)13-22/h3-4,7-16,21,28,36H,5-6,17H2,1-2H3,(H,38,40)/t28-/m0/s1	QGAYZTNDDHKOGN-NDEPHWFRSA-N	473471	US10844044, Example 344	WD repeat-containing protein 5		 0.480								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473471	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473471&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456252	442073679							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981672	Cc1cc(CNC(=O)c2cc(Cn3ccn(C)c3=N)cc(c2)-c2ncc(F)cc2C)ccc1Cl	InChI=1S/C26H25ClFN5O/c1-16-8-18(4-5-23(16)27)13-31-25(34)21-11-19(15-33-7-6-32(3)26(33)29)10-20(12-21)24-17(2)9-22(28)14-30-24/h4-12,14,29H,13,15H2,1-3H3,(H,31,34)	PZTHPCUVWNDPSU-UHFFFAOYSA-N	473472	US10844044, Example 70	WD repeat-containing protein 5		 1.10								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473472	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473472&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146455844	442073680							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981673	CCn1cc(c(n1)C(F)(F)F)-c1cc(Cn2ccn(C)c2=N)cc(c1)C(=O)N[C@@H](C1CC1)c1ccc(Cl)c(Cl)c1	InChI=1S/C28H27Cl2F3N6O/c1-3-39-15-21(25(36-39)28(31,32)33)19-10-16(14-38-9-8-37(2)27(38)34)11-20(12-19)26(40)35-24(17-4-5-17)18-6-7-22(29)23(30)13-18/h6-13,15,17,24,34H,3-5,14H2,1-2H3,(H,35,40)/t24-/m0/s1	QDZRJBVVJJUHAF-DEOSSOPVSA-N	473473	US10844044, Example 161	WD repeat-containing protein 5		<0.100								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473473	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473473&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456472	442073681							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981674	Cc1coc(=N)n1Cc1cc(cc(c1)-c1cccnc1C(F)(F)F)C(=O)N[C@@H](C1CC1)c1ccc(F)c(C)c1	InChI=1S/C29H26F4N4O2/c1-16-10-20(7-8-24(16)30)25(19-5-6-19)36-27(38)22-12-18(14-37-17(2)15-39-28(37)34)11-21(13-22)23-4-3-9-35-26(23)29(31,32)33/h3-4,7-13,15,19,25,34H,5-6,14H2,1-2H3,(H,36,38)/t25-/m0/s1	OHJFJZQPPVFZHL-VWLOTQADSA-N	473474	US10844044, Example 252	WD repeat-containing protein 5		 21.0								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473474	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473474&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456458	442073682							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981675	Cc1cc(ccc1F)[C@@H](NC(=O)c1cc(Cn2cccc(F)c2=N)cc(c1)-c1cc(nn1C)C(F)(F)F)C1CC1	InChI=1S/C29H26F5N5O/c1-16-10-19(7-8-22(16)30)26(18-5-6-18)36-28(40)21-12-17(15-39-9-3-4-23(31)27(39)35)11-20(13-21)24-14-25(29(32,33)34)37-38(24)2/h3-4,7-14,18,26,35H,5-6,15H2,1-2H3,(H,36,40)/t26-/m0/s1	WGGJFQLELLVUIO-SANMLTNESA-N	473475	US10844044, Example 345	WD repeat-containing protein 5		 2.40								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473475	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473475&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146457631	442073683							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981676	Cc1ccnc(c1)C(NC(=O)c1cc(Cn2ccn(C)c2=N)cc(c1)-c1ccc(F)cc1OC(F)F)C1CC1	InChI=1S/C29H28F3N5O2/c1-17-7-8-34-24(11-17)26(19-3-4-19)35-27(38)21-13-18(16-37-10-9-36(2)29(37)33)12-20(14-21)23-6-5-22(30)15-25(23)39-28(31)32/h5-15,19,26,28,33H,3-4,16H2,1-2H3,(H,35,38)	PHVGBGABFFUVGV-UHFFFAOYSA-N	473476	US10844044, Example 71	WD repeat-containing protein 5		 0.330								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473476	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473476&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456333	442073684							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981677	CCn1cc(c(n1)C(F)(F)F)-c1cc(Cn2ccn(C3CC3)c2=N)cc(c1)C(=O)N[C@@H](C1CC1)c1ccc(Cl)c(Cl)c1	InChI=1S/C30H29Cl2F3N6O/c1-2-40-16-23(27(38-40)30(33,34)35)20-11-17(15-39-9-10-41(29(39)36)22-6-7-22)12-21(13-20)28(42)37-26(18-3-4-18)19-5-8-24(31)25(32)14-19/h5,8-14,16,18,22,26,36H,2-4,6-7,15H2,1H3,(H,37,42)/t26-/m0/s1	JAOXZFQPIARIJX-SANMLTNESA-N	473477	US10844044, Example 162	WD repeat-containing protein 5		<0.100								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473477	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473477&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146455780	442073685							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981678	Cc1cc(ccc1F)[C@@H](NC(=O)c1cc(CN2CCOC2=N)cc(c1)-c1cccnc1C(F)(F)F)C1CC1	InChI=1S/C28H26F4N4O2/c1-16-11-19(6-7-23(16)29)24(18-4-5-18)35-26(37)21-13-17(15-36-9-10-38-27(36)33)12-20(14-21)22-3-2-8-34-25(22)28(30,31)32/h2-3,6-8,11-14,18,24,33H,4-5,9-10,15H2,1H3,(H,35,37)/t24-/m0/s1	LIHADAJRNWQKGW-DEOSSOPVSA-N	473478	US10844044, Example 253	WD repeat-containing protein 5		<0.100								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473478	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473478&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146457394	442073686							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981679	Cc1cc(ccc1F)[C@@H](NC(=O)c1cc(Cn2ccccc2=N)cc(c1)-c1cc(nn1C)C(F)(F)F)C1CC1	InChI=1S/C29H27F4N5O/c1-17-11-20(8-9-23(17)30)27(19-6-7-19)35-28(39)22-13-18(16-38-10-4-3-5-26(38)34)12-21(14-22)24-15-25(29(31,32)33)36-37(24)2/h3-5,8-15,19,27,34H,6-7,16H2,1-2H3,(H,35,39)/t27-/m0/s1	RTZIMKFLOLUPFO-MHZLTWQESA-N	473479	US10844044, Example 346	WD repeat-containing protein 5		 1.60								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473479	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473479&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146488055	442073687							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981680	Cc1cc(ccc1F)[C@@H](NC(=O)c1cc(Cn2ccn(C)c2=N)cc(c1)-c1ncc(F)cc1C(F)(F)F)C1CC1	InChI=1S/C29H26F5N5O/c1-16-9-19(5-6-24(16)31)25(18-3-4-18)37-27(40)21-11-17(15-39-8-7-38(2)28(39)35)10-20(12-21)26-23(29(32,33)34)13-22(30)14-36-26/h5-14,18,25,35H,3-4,15H2,1-2H3,(H,37,40)/t25-/m0/s1	DYWNHPXPZBCRPK-VWLOTQADSA-N	473480	US10844044, Example 72	WD repeat-containing protein 5		 0.050								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473480	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473480&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456670	442073688							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981681	CC(C)Cn1cc(c(n1)C(F)(F)F)-c1cc(Cn2ccn(C3CC3)c2=N)cc(c1)C(=O)N[C@@H](C1CC1)c1ccc(F)c(C)c1	InChI=1S/C33H36F4N6O/c1-19(2)16-42-18-27(30(40-42)33(35,36)37)24-13-21(17-41-10-11-43(32(41)38)26-7-8-26)14-25(15-24)31(44)39-29(22-4-5-22)23-6-9-28(34)20(3)12-23/h6,9-15,18-19,22,26,29,38H,4-5,7-8,16-17H2,1-3H3,(H,39,44)/t29-/m0/s1	IWODPEVBQNSVSK-LJAQVGFWSA-N	473481	US10844044, Example 163	WD repeat-containing protein 5		 0.680								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473481	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473481&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456311	442073689							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981682	COc1cc(CNC(=O)c2cc(CN3CCOC3=N)cc(c2)-c2ccc(F)cc2C)cc(OC)c1	InChI=1S/C27H28FN3O4/c1-17-8-22(28)4-5-25(17)20-9-19(16-31-6-7-35-27(31)29)10-21(13-20)26(32)30-15-18-11-23(33-2)14-24(12-18)34-3/h4-5,8-14,29H,6-7,15-16H2,1-3H3,(H,30,32)	FNJBPMDBHNPGLU-UHFFFAOYSA-N	473482	US10844044, Example 254	WD repeat-containing protein 5		 0.120								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473482	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473482&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456509	442073690							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981683	CCOc1c(cc(Cn2ccccc2=N)cc1-c1cn(C)nc1C(F)(F)F)C(=O)N[C@@H](C1CC1)c1ccc(F)c(C)c1	InChI=1S/C31H31F4N5O2/c1-4-42-28-22(24-17-39(3)38-29(24)31(33,34)35)14-19(16-40-12-6-5-7-26(40)36)15-23(28)30(41)37-27(20-8-9-20)21-10-11-25(32)18(2)13-21/h5-7,10-15,17,20,27,36H,4,8-9,16H2,1-3H3,(H,37,41)/t27-/m0/s1	NXOBTXPUNSOYEU-MHZLTWQESA-N	473483	US10844044, Example 347	WD repeat-containing protein 5		<0.100								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473483	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473483&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456898	442073691							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981684	Cc1cc(ccc1F)[C@@H](NC(=O)c1cc(Cn2ccn(C)c2=N)cc(c1)-c1ccc(F)cc1OC(F)F)C1CC1	InChI=1S/C30H28F4N4O2/c1-17-11-20(5-8-25(17)32)27(19-3-4-19)36-28(39)22-13-18(16-38-10-9-37(2)30(38)35)12-21(14-22)24-7-6-23(31)15-26(24)40-29(33)34/h5-15,19,27,29,35H,3-4,16H2,1-2H3,(H,36,39)/t27-/m0/s1	CAZZIDBMTPAUGG-MHZLTWQESA-N	473484	US10844044, Example 73	WD repeat-containing protein 5		 0.140								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473484	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473484&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456282	442073692							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981685	Cc1cc(ccc1F)[C@@H](NC(=O)c1cc(Cn2ccn(C3CC3)c2=N)cc(c1)-c1cn(nc1C(F)(F)F)C1CCCC1)C1CC1	InChI=1S/C34H36F4N6O/c1-20-14-23(8-11-29(20)35)30(22-6-7-22)40-32(45)25-16-21(18-42-12-13-43(33(42)39)26-9-10-26)15-24(17-25)28-19-44(27-4-2-3-5-27)41-31(28)34(36,37)38/h8,11-17,19,22,26-27,30,39H,2-7,9-10,18H2,1H3,(H,40,45)/t30-/m0/s1	QYNKLVOWPIWPAS-PMERELPUSA-N	473485	US10844044, Example 164	WD repeat-containing protein 5		 1.40								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473485	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473485&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146455880	442073693							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981686	Cc1cc(ccc1F)[C@@H](NC(=O)c1cc(Cn2ccoc2=N)cc(c1)-c1cncnc1C(F)(F)F)C1CC1	InChI=1S/C27H23F4N5O2/c1-15-8-18(4-5-22(15)28)23(17-2-3-17)35-25(37)20-10-16(13-36-6-7-38-26(36)32)9-19(11-20)21-12-33-14-34-24(21)27(29,30)31/h4-12,14,17,23,32H,2-3,13H2,1H3,(H,35,37)/t23-/m0/s1	MVTLNPBBIFSXHY-QHCPKHFHSA-N	473486	US10844044, Example 255	WD repeat-containing protein 5		 0.620								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473486	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473486&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146457697	442073694							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981687	CCOc1c(cc(Cn2cccc(F)c2=N)cc1C1=CN(C)NC1C(F)(F)F)C(=O)N[C@@H](C1CC1)c1ccc(F)c(C)c1	InChI=1S/C31H32F5N5O2/c1-4-43-27-21(23-16-40(3)39-28(23)31(34,35)36)13-18(15-41-11-5-6-25(33)29(41)37)14-22(27)30(42)38-26(19-7-8-19)20-9-10-24(32)17(2)12-20/h5-6,9-14,16,19,26,28,37,39H,4,7-8,15H2,1-3H3,(H,38,42)/t26-,28?/m0/s1	MKYKXQBPWNMYNE-QODXOHEASA-N	473487	US10844044, Example 348	WD repeat-containing protein 5		<0.100								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473487	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473487&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146487992	442073695							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981688	COc1cc(OC)cc(c1)C(NC(=O)c1cc(Cn2ccn(C)c2=N)cc(c1)-c1ncc(F)cc1C(F)(F)F)C1CC1	InChI=1S/C30H29F4N5O3/c1-38-6-7-39(29(38)35)16-17-8-19(27-25(30(32,33)34)13-22(31)15-36-27)10-21(9-17)28(40)37-26(18-4-5-18)20-11-23(41-2)14-24(12-20)42-3/h6-15,18,26,35H,4-5,16H2,1-3H3,(H,37,40)	KBQZVFHNXFUGGQ-UHFFFAOYSA-N	473488	US10844044, Example 74	WD repeat-containing protein 5		 0.640								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473488	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473488&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456022	442073696							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981689	CC(C)Cn1cc(c(n1)C(F)(F)F)-c1cc(Cn2ccn(C)c2=N)cc(c1)C(=O)N[C@@H](C1CC1)c1ccc(F)c(C)c1	InChI=1S/C31H34F4N6O/c1-18(2)15-41-17-25(28(38-41)31(33,34)35)23-12-20(16-40-10-9-39(4)30(40)36)13-24(14-23)29(42)37-27(21-5-6-21)22-7-8-26(32)19(3)11-22/h7-14,17-18,21,27,36H,5-6,15-16H2,1-4H3,(H,37,42)/t27-/m0/s1	YPQZSRCVXTYTLL-MHZLTWQESA-N	473489	US10844044, Example 165	WD repeat-containing protein 5		 0.140								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473489	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473489&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146455822	442073697							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981690	CCc1coc(=N)n1Cc1cc(cc(c1)-c1cccnc1C(F)(F)F)C(=O)N[C@@H](C1CC1)c1ccc(F)c(C)c1	InChI=1S/C30H28F4N4O2/c1-3-23-16-40-29(35)38(23)15-18-12-21(24-5-4-10-36-27(24)30(32,33)34)14-22(13-18)28(39)37-26(19-6-7-19)20-8-9-25(31)17(2)11-20/h4-5,8-14,16,19,26,35H,3,6-7,15H2,1-2H3,(H,37,39)/t26-/m0/s1	IPVTYKZELOSEOZ-SANMLTNESA-N	473490	US10844044, Example 256	WD repeat-containing protein 5		 2.70								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473490	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473490&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456469	442073698							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981691	CCOc1c(cc(Cn2cc(F)ccc2=N)cc1-c1cn(C)nc1C(F)(F)F)C(=O)N[C@@H](C1CC1)c1ccc(F)c(C)c1	InChI=1S/C31H30F5N5O2/c1-4-43-28-22(24-16-40(3)39-29(24)31(34,35)36)12-18(14-41-15-21(32)8-10-26(41)37)13-23(28)30(42)38-27(19-5-6-19)20-7-9-25(33)17(2)11-20/h7-13,15-16,19,27,37H,4-6,14H2,1-3H3,(H,38,42)/t27-/m0/s1	BTRXRRBPNXEIGB-MHZLTWQESA-N	473491	US10844044, Example 349	WD repeat-containing protein 5		<0.100								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473491	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473491&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146457363	442073699							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981692	Cc1ccnc(c1)C(NC(=O)c1cc(Cn2ccn(C)c2=N)cc(c1)-c1ncc(F)cc1C(F)(F)F)C1CC1	InChI=1S/C28H26F4N6O/c1-16-5-6-34-23(9-16)25(18-3-4-18)36-26(39)20-11-17(15-38-8-7-37(2)27(38)33)10-19(12-20)24-22(28(30,31)32)13-21(29)14-35-24/h5-14,18,25,33H,3-4,15H2,1-2H3,(H,36,39)	FMOSGWYRJHCSRR-UHFFFAOYSA-N	473492	US10844044, Example 75	WD repeat-containing protein 5		 1.20								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473492	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473492&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146457635	442073700							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981693	Cc1cc(ccc1F)[C@@H](NC(=O)c1cc(Cn2ccn(C)c2=N)cc(c1)C1CCC1)C1CC1	InChI=1S/C27H31FN4O/c1-17-12-21(8-9-24(17)28)25(20-6-7-20)30-26(33)23-14-18(13-22(15-23)19-4-3-5-19)16-32-11-10-31(2)27(32)29/h8-15,19-20,25,29H,3-7,16H2,1-2H3,(H,30,33)/t25-/m0/s1	NZTXHLUCMNIEHS-VWLOTQADSA-N	473493	US10844044, Example 166	WD repeat-containing protein 5		<0.100								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473493	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473493&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456358	442073701							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981694	C[C@H](NC(=O)c1cc(Cn2ccoc2=N)cc(c1)-c1cccnc1C(F)(F)F)c1ccc(F)c(Cl)c1	InChI=1S/C25H19ClF4N4O2/c1-14(16-4-5-21(27)20(26)12-16)33-23(35)18-10-15(13-34-7-8-36-24(34)31)9-17(11-18)19-3-2-6-32-22(19)25(28,29)30/h2-12,14,31H,13H2,1H3,(H,33,35)/t14-/m0/s1	FRNNWCWURRPFGG-AWEZNQCLSA-N	473494	US10844044, Example 257	WD repeat-containing protein 5		 2.00								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473494	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473494&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146457132	442073702							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981695	Cc1cc(ccc1F)[C@@H](NC(=O)c1cc(Cn2cccc(F)c2=N)cc(c1)-c1cccnc1C(F)(F)F)C1CC1	InChI=1S/C30H25F5N4O/c1-17-12-20(8-9-24(17)31)26(19-6-7-19)38-29(40)22-14-18(16-39-11-3-5-25(32)28(39)36)13-21(15-22)23-4-2-10-37-27(23)30(33,34)35/h2-5,8-15,19,26,36H,6-7,16H2,1H3,(H,38,40)/t26-/m0/s1	SJVSMZLCKVMSHW-SANMLTNESA-N	473495	US10844044, Example 350	WD repeat-containing protein 5		 0.120								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473495	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473495&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146455706	442073703							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981696	Cc1cc(CNC(=O)c2cc(Cn3ccn(C)c3=N)cc(c2)-c2cccnc2C(F)(F)F)ccc1Cl	InChI=1S/C26H23ClF3N5O/c1-16-10-17(5-6-22(16)27)14-33-24(36)20-12-18(15-35-9-8-34(2)25(35)31)11-19(13-20)21-4-3-7-32-23(21)26(28,29)30/h3-13,31H,14-15H2,1-2H3,(H,33,36)	YDHPEKHYIWUSFK-UHFFFAOYSA-N	473496	US10844044, Example 76	WD repeat-containing protein 5		<0.100								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473496	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473496&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146455792	442073704							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981697	Cc1cc(F)ccc1-c1cc(Cn2ccn(C)c2=N)cc(c1)C(=O)NC(C1CC1)c1ccc(F)c(C)n1	InChI=1S/C29H29F2N5O/c1-17-12-23(30)6-7-24(17)21-13-19(16-36-11-10-35(3)29(36)32)14-22(15-21)28(37)34-27(20-4-5-20)26-9-8-25(31)18(2)33-26/h6-15,20,27,32H,4-5,16H2,1-3H3,(H,34,37)	MFBPRMLNAJNSLT-UHFFFAOYSA-N	473497	US10844044, Example 167	WD repeat-containing protein 5		 0.210								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473497	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473497&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456909	442073705							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981698	C[C@H](NC(=O)c1cc(Cn2ccoc2=N)cc(c1)-c1cccnc1C(F)(F)F)c1ccc(cc1)C(F)(F)F	InChI=1S/C26H20F6N4O2/c1-15(17-4-6-20(7-5-17)25(27,28)29)35-23(37)19-12-16(14-36-9-10-38-24(36)33)11-18(13-19)21-3-2-8-34-22(21)26(30,31)32/h2-13,15,33H,14H2,1H3,(H,35,37)/t15-/m0/s1	QWMUJAWZSYPVPB-HNNXBMFYSA-N	473498	US10844044, Example 258	WD repeat-containing protein 5		 5.80								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473498	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473498&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456369	442073706							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981699	Cc1cc(ccc1F)[C@@H](NC(=O)c1cc(Cn2cccc(F)c2=N)cc(c1)-c1cn(C)nc1C(F)(F)F)C1CC1	InChI=1S/C29H26F5N5O/c1-16-10-19(7-8-23(16)30)25(18-5-6-18)36-28(40)21-12-17(14-39-9-3-4-24(31)27(39)35)11-20(13-21)22-15-38(2)37-26(22)29(32,33)34/h3-4,7-13,15,18,25,35H,5-6,14H2,1-2H3,(H,36,40)/t25-/m0/s1	CIKKRXNFSNBVPK-VWLOTQADSA-N	473499	US10844044, Example 351	WD repeat-containing protein 5		<0.100								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473499	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473499&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146455948	442073707							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981700	Cc1ccnc(c1)C(NC(=O)c1cc(Cn2ccn(C)c2=N)cc(c1)-c1cccnc1C(F)(F)F)C1CC1	InChI=1S/C28H27F3N6O/c1-17-7-9-33-23(12-17)24(19-5-6-19)35-26(38)21-14-18(16-37-11-10-36(2)27(37)32)13-20(15-21)22-4-3-8-34-25(22)28(29,30)31/h3-4,7-15,19,24,32H,5-6,16H2,1-2H3,(H,35,38)	FKYOQFRQGKFSPS-UHFFFAOYSA-N	473500	US10844044, Example 77	WD repeat-containing protein 5		 0.180								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473500	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473500&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456531	442073708							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981701	Cn1ccn(Cc2cc(cc(c2)-c2cccc3OC(F)(F)Oc23)C(=O)NCc2ccc(Cl)c(Cl)c2)c1=N	InChI=1S/C26H20Cl2F2N4O3/c1-33-7-8-34(25(33)31)14-16-9-17(19-3-2-4-22-23(19)37-26(29,30)36-22)12-18(10-16)24(35)32-13-15-5-6-20(27)21(28)11-15/h2-12,31H,13-14H2,1H3,(H,32,35)	JPDNVRPEGMZHFG-UHFFFAOYSA-N	473501	US10844044, Example 168	WD repeat-containing protein 5		 27.0								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473501	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473501&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146455814	442073709							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981702	Cc1cc(ccc1F)C(NC(=O)c1cc(Cn2ccoc2=N)cc(c1)-c1cn(C)nc1C(F)(F)F)C1CC1	InChI=1S/C27H25F4N5O2/c1-15-9-18(5-6-22(15)28)23(17-3-4-17)33-25(37)20-11-16(13-36-7-8-38-26(36)32)10-19(12-20)21-14-35(2)34-24(21)27(29,30)31/h5-12,14,17,23,32H,3-4,13H2,1-2H3,(H,33,37)	RJPRXTSKPNPRPK-UHFFFAOYSA-N	473502	US10844044, Example 259	WD repeat-containing protein 5		<0.100								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473502	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473502&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456527	442073710							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981703	Cc1cc(ccc1F)[C@@H](NC(=O)c1cc(Cn2ccccc2=N)cc(c1)-c1cn(C)nc1C(F)(F)F)C1CC1	InChI=1S/C29H27F4N5O/c1-17-11-20(8-9-24(17)30)26(19-6-7-19)35-28(39)22-13-18(15-38-10-4-3-5-25(38)34)12-21(14-22)23-16-37(2)36-27(23)29(31,32)33/h3-5,8-14,16,19,26,34H,6-7,15H2,1-2H3,(H,35,39)/t26-/m0/s1	HNXGJVLCSCJPDK-SANMLTNESA-N	473503	US10844044, Example 352	WD repeat-containing protein 5		<0.100								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473503	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473503&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146457628	442073711							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981704	COc1cc(CNC(=O)c2cc(Cn3ccn(C)c3=N)cc(c2)-c2cnc(F)cc2C)cc(OC)c1	InChI=1S/C27H28FN5O3/c1-17-7-25(28)30-15-24(17)20-8-19(16-33-6-5-32(2)27(33)29)9-21(12-20)26(34)31-14-18-10-22(35-3)13-23(11-18)36-4/h5-13,15,29H,14,16H2,1-4H3,(H,31,34)	UKRLFTUMBIRDBO-UHFFFAOYSA-N	473504	US10844044, Example 78	WD repeat-containing protein 5		 5.90								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473504	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473504&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456715	442073712							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981705	COc1cccc(n1)-c1cc(Cn2ccn(C)c2=N)cc(c1)C(=O)NCc1ccc(Cl)c(Cl)n1	InChI=1S/C24H22Cl2N6O2/c1-31-8-9-32(24(31)27)14-15-10-16(20-4-3-5-21(30-20)34-2)12-17(11-15)23(33)28-13-18-6-7-19(25)22(26)29-18/h3-12,27H,13-14H2,1-2H3,(H,28,33)	TUZXHFVKFFOLPH-UHFFFAOYSA-N	473505	US10844044, Example 169	WD repeat-containing protein 5		 23.0								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473505	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473505&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146488066	442073713							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981706	C[C@H](NC(=O)c1cc(Cn2ccoc2=N)cc(c1)-c1cccnc1C(F)(F)F)c1ccc(F)cc1	InChI=1S/C25H20F4N4O2/c1-15(17-4-6-20(26)7-5-17)32-23(34)19-12-16(14-33-9-10-35-24(33)30)11-18(13-19)21-3-2-8-31-22(21)25(27,28)29/h2-13,15,30H,14H2,1H3,(H,32,34)/t15-/m0/s1	HZCBNCPSFQPVNE-HNNXBMFYSA-N	473506	US10844044, Example 260	WD repeat-containing protein 5		 25.0								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473506	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473506&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456285	442073714							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981707	Cc1cc(ccc1F)[C@@H](NC(=O)c1cc(Cn2cc(F)ccc2=N)cc(c1)-c1cn(C)nc1C(F)(F)F)C1CC1	InChI=1S/C29H26F5N5O/c1-16-9-19(5-7-24(16)31)26(18-3-4-18)36-28(40)21-11-17(13-39-14-22(30)6-8-25(39)35)10-20(12-21)23-15-38(2)37-27(23)29(32,33)34/h5-12,14-15,18,26,35H,3-4,13H2,1-2H3,(H,36,40)/t26-/m0/s1	PZYOVBHLNSTCLL-SANMLTNESA-N	473507	US10844044, Example 353	WD repeat-containing protein 5		<0.100								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473507	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473507&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146457404	442073715							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981708	Cc1cc(CNC(=O)c2cc(Cn3ccn(C)c3=N)cc(c2)-c2cnc(F)cc2C)ccc1Cl	InChI=1S/C26H25ClFN5O/c1-16-9-24(28)30-14-22(16)20-10-19(15-33-7-6-32(3)26(33)29)11-21(12-20)25(34)31-13-18-4-5-23(27)17(2)8-18/h4-12,14,29H,13,15H2,1-3H3,(H,31,34)	KYMBIPZCWZELSQ-UHFFFAOYSA-N	473508	US10844044, Example 79	WD repeat-containing protein 5		 4.30								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473508	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473508&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146455886	442073716							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981709	C[C@H](NC(=O)c1cc(Cn2ccn(C)c2=N)cc(OC(F)(F)F)c1)c1ccc(F)c(C)c1	InChI=1S/C22H22F4N4O2/c1-13-8-16(4-5-19(13)23)14(2)28-20(31)17-9-15(10-18(11-17)32-22(24,25)26)12-30-7-6-29(3)21(30)27/h4-11,14,27H,12H2,1-3H3,(H,28,31)/t14-/m0/s1	KCBVUZFANIJJHK-AWEZNQCLSA-N	473509	US10844044, Example 170	WD repeat-containing protein 5		 0.220								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473509	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473509&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146455821	442073717							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981710	Cc1cc(ccc1F)[C@@H](NC(=O)c1cc(Cn2ccoc2=N)cc(c1)-c1cccnc1OC(F)F)C1CC1	InChI=1S/C28H25F3N4O3/c1-16-11-19(6-7-23(16)29)24(18-4-5-18)34-25(36)21-13-17(15-35-9-10-37-28(35)32)12-20(14-21)22-3-2-8-33-26(22)38-27(30)31/h2-3,6-14,18,24,27,32H,4-5,15H2,1H3,(H,34,36)/t24-/m0/s1	QLYVRBCTRZJMLI-DEOSSOPVSA-N	473510	US10844044, Example 261	WD repeat-containing protein 5		 0.280								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473510	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473510&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146455803	442073718							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981711	Cc1cc(ccc1F)[C@@H](NC(=O)c1cc(Cn2cc(F)ccc2=N)cc(c1)-c1cccnc1C(F)(F)F)C1CC1	InChI=1S/C30H25F5N4O/c1-17-11-20(6-8-25(17)32)27(19-4-5-19)38-29(40)22-13-18(15-39-16-23(31)7-9-26(39)36)12-21(14-22)24-3-2-10-37-28(24)30(33,34)35/h2-3,6-14,16,19,27,36H,4-5,15H2,1H3,(H,38,40)/t27-/m0/s1	HGMVVDMGLLCVRR-MHZLTWQESA-N	473511	US10844044, Example 354	WD repeat-containing protein 5		<0.100								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473511	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473511&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456864	442073719							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981712	Cc1cc(CNC(=O)c2cc(Cn3ccn(C)c3=N)cc(c2)-c2ccc(=O)[nH]c2C)ccc1Cl	InChI=1S/C26H26ClN5O2/c1-16-10-18(4-6-23(16)27)14-29-25(34)21-12-19(15-32-9-8-31(3)26(32)28)11-20(13-21)22-5-7-24(33)30-17(22)2/h4-13,28H,14-15H2,1-3H3,(H,29,34)(H,30,33)	DTXKSJUFWTVDGH-UHFFFAOYSA-N	473512	US10844044, Example 80	WD repeat-containing protein 5		 20.0								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473512	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473512&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			156022870	442073720							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981713	C[C@H](NC(=O)c1cc(Cn2ccn(C)c2=N)cc(c1F)-c1ccccn1C(F)(F)F)c1ccc(F)c(C)n1			473513	US10844044, Example 171	WD repeat-containing protein 5		 0.130								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473513	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473513&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			156022871	442073721							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981714	C[C@H](NC(=O)c1cc(Cn2ccoc2=N)cc(c1)-c1cccnc1C(F)(F)F)c1ncc(F)cn1	InChI=1S/C23H18F4N6O2/c1-13(20-30-10-17(24)11-31-20)32-21(34)16-8-14(12-33-5-6-35-22(33)28)7-15(9-16)18-3-2-4-29-19(18)23(25,26)27/h2-11,13,28H,12H2,1H3,(H,32,34)/t13-/m0/s1	SLGSRTNYPATMQF-ZDUSSCGKSA-N	473514	US10844044, Example 262	WD repeat-containing protein 5		>33.0								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473514	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473514&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456395	442073722							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981715	COc1cc(OC)cc(c1)C(C)NC(=O)c1cc(Cn2ccn(C)c2=N)cc(n1)-c1ccc(F)cc1C	InChI=1S/C28H30FN5O3/c1-17-10-21(29)6-7-24(17)25-11-19(16-34-9-8-33(3)28(34)30)12-26(32-25)27(35)31-18(2)20-13-22(36-4)15-23(14-20)37-5/h6-15,18,30H,16H2,1-5H3,(H,31,35)	FJCGXCMOXMFYBW-UHFFFAOYSA-N	473515	US10844044, Example 355	WD repeat-containing protein 5		 3.57								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473515	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473515&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146488049	442073723							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981716	COc1cc(CNC(=O)c2cc(Cn3ccn(C)c3=N)cc(c2)-c2c[nH]c(=O)cc2C)cc(OC)c1	InChI=1S/C27H29N5O4/c1-17-7-25(33)29-15-24(17)20-8-19(16-32-6-5-31(2)27(32)28)9-21(12-20)26(34)30-14-18-10-22(35-3)13-23(11-18)36-4/h5-13,15,28H,14,16H2,1-4H3,(H,29,33)(H,30,34)	KUGOCEVEYMAAHD-UHFFFAOYSA-N	473516	US10844044, Example 81	WD repeat-containing protein 5		 13.0								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473516	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473516&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			156022872	442073724							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981717	C[C@H](NC(=O)c1cc(Cn2ccn(C)c2=N)cc(c1F)-c1ccc(F)cn1C(F)(F)F)c1ccc(F)c(C)c1			473517	US10844044, Example 172	WD repeat-containing protein 5		<0.100								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473517	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473517&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			156022873	442073725							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981718	Cc1cc(ccc1F)[C@@H](NC(=O)c1cc(Cn2ccoc2=N)cc(c1)-c1cccnc1OCC(F)(F)F)C1CC1	InChI=1S/C29H26F4N4O3/c1-17-11-20(6-7-24(17)30)25(19-4-5-19)36-26(38)22-13-18(15-37-9-10-39-28(37)34)12-21(14-22)23-3-2-8-35-27(23)40-16-29(31,32)33/h2-3,6-14,19,25,34H,4-5,15-16H2,1H3,(H,36,38)/t25-/m0/s1	HIEFRFOCSXTOBM-VWLOTQADSA-N	473518	US10844044, Example 263	WD repeat-containing protein 5		 0.290								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473518	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473518&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456289	442073726							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981719	Cc1ccnc(c1)C(NC(=O)c1cc(Cn2ccn(C)c2=N)cc(n1)-c1ccc(F)cc1C)C1CC1	InChI=1S/C28H29FN6O/c1-17-8-9-31-24(12-17)26(20-4-5-20)33-27(36)25-15-19(16-35-11-10-34(3)28(35)30)14-23(32-25)22-7-6-21(29)13-18(22)2/h6-15,20,26,30H,4-5,16H2,1-3H3,(H,33,36)	ZEOWBJYBYFWPKZ-UHFFFAOYSA-N	473519	US10844044, Example 356	WD repeat-containing protein 5		 182								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473519	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473519&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456669	442073727							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981720	Cc1cc(=O)[nH]cc1-c1cc(Cn2ccn(C)c2=N)cc(c1)C(=O)NCc1ccc(Cl)c(Cl)c1	InChI=1S/C25H23Cl2N5O2/c1-15-7-23(33)29-13-20(15)18-8-17(14-32-6-5-31(2)25(32)28)9-19(11-18)24(34)30-12-16-3-4-21(26)22(27)10-16/h3-11,13,28H,12,14H2,1-2H3,(H,29,33)(H,30,34)	LABPWZXYVYJWFK-UHFFFAOYSA-N	473520	US10844044, Example 82	WD repeat-containing protein 5		 20.0								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473520	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473520&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			156022874	442073728							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981721	Cc1cc(F)ccc1-c1cc(Cn2ccn(C)c2=N)cc(c1)C(=O)N[C@@H](C1CC1)c1ccc(F)c(C)n1	InChI=1S/C29H29F2N5O/c1-17-12-23(30)6-7-24(17)21-13-19(16-36-11-10-35(3)29(36)32)14-22(15-21)28(37)34-27(20-4-5-20)26-9-8-25(31)18(2)33-26/h6-15,20,27,32H,4-5,16H2,1-3H3,(H,34,37)/t27-/m0/s1	MFBPRMLNAJNSLT-MHZLTWQESA-N	473521	US10844044, Example 173	WD repeat-containing protein 5		 0.890								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473521	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473521&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146488031	442073729							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981722	Cc1cc(ccc1F)[C@@H](NC(=O)c1cc(Cn2ccoc2=N)cc(c1)C1CC1)C1CC1	InChI=1S/C25H26FN3O2/c1-15-10-19(6-7-22(15)26)23(18-4-5-18)28-24(30)21-12-16(11-20(13-21)17-2-3-17)14-29-8-9-31-25(29)27/h6-13,17-18,23,27H,2-5,14H2,1H3,(H,28,30)/t23-/m0/s1	IPHOSFFTFPOWJV-QHCPKHFHSA-N	473522	US10844044, Example 265	WD repeat-containing protein 5		 0.780								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473522	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473522&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146455956	442073730							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981723	COc1ccnc(CNC(=O)c2cc(Cn3ccn(C)c3=N)cc(n2)-c2ccc(F)cc2C)c1	InChI=1S/C25H25FN6O2/c1-16-10-18(26)4-5-21(16)22-11-17(15-32-9-8-31(2)25(32)27)12-23(30-22)24(33)29-14-19-13-20(34-3)6-7-28-19/h4-13,27H,14-15H2,1-3H3,(H,29,33)	GTIASNBJNBYVDX-UHFFFAOYSA-N	473523	US10844044, Example 357	WD repeat-containing protein 5		 1.30								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473523	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473523&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456154	442073731							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981724	Cc1cc(CNC(=O)c2cc(Cn3ccn(C)c3=N)cc(c2)-c2c[nH]c(=O)cc2C)ccc1Cl	InChI=1S/C26H26ClN5O2/c1-16-9-24(33)29-14-22(16)20-10-19(15-32-7-6-31(3)26(32)28)11-21(12-20)25(34)30-13-18-4-5-23(27)17(2)8-18/h4-12,14,28H,13,15H2,1-3H3,(H,29,33)(H,30,34)	QSENASCPVNBYRG-UHFFFAOYSA-N	473524	US10844044, Example 83	WD repeat-containing protein 5		 7.10								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473524	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473524&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			156022875	442073732							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981725	Cc1cc(ncc1F)[C@@H](NC(=O)c1cc(Cn2ccn(C)c2=N)cc(c1)-c1ccc(F)cc1Cl)C1CC1	InChI=1S/C28H26ClF2N5O/c1-16-9-25(33-14-24(16)31)26(18-3-4-18)34-27(37)20-11-17(15-36-8-7-35(2)28(36)32)10-19(12-20)22-6-5-21(30)13-23(22)29/h5-14,18,26,32H,3-4,15H2,1-2H3,(H,34,37)/t26-/m0/s1	BFVJBRFZHKNUBS-SANMLTNESA-N	473525	US10844044, Example 174	WD repeat-containing protein 5		<0.100								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473525	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473525&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146487898	442073733							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981726	Cc1cc(ccc1F)[C@@H](NC(=O)c1cc(CN2CCCOC2=N)cc(c1)-c1cccnc1C(F)(F)F)C1CC1	InChI=1S/C29H28F4N4O2/c1-17-12-20(7-8-24(17)30)25(19-5-6-19)36-27(38)22-14-18(16-37-10-3-11-39-28(37)34)13-21(15-22)23-4-2-9-35-26(23)29(31,32)33/h2,4,7-9,12-15,19,25,34H,3,5-6,10-11,16H2,1H3,(H,36,38)/t25-/m0/s1	RWDXQFHWSULJBR-VWLOTQADSA-N	473526	US10844044, Example 266::US10844044, Example 362	WD repeat-containing protein 5		 16.0								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473526	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473526&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146455809	442073734							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981727	Cc1cc(F)ccc1-c1cc(Cn2ccn(C)c2=N)cc(n1)C(=O)NCc1ncc(Cl)cn1	InChI=1S/C23H21ClFN7O/c1-14-7-17(25)3-4-18(14)19-8-15(13-32-6-5-31(2)23(32)26)9-20(30-19)22(33)29-12-21-27-10-16(24)11-28-21/h3-11,26H,12-13H2,1-2H3,(H,29,33)	ICWJQRRRNDDDPI-UHFFFAOYSA-N	473527	US10844044, Example 358	WD repeat-containing protein 5		 5.50								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473527	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473527&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146457692	442073735							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981728	Cn1ccn(Cc2cc(cc(c2)-c2ccc(F)cc2C(F)(F)F)C(=O)NC(CC(O)=O)c2ccc(Cl)c(Cl)c2)c1=N	InChI=1S/C28H22Cl2F4N4O3/c1-37-6-7-38(27(37)35)14-15-8-17(20-4-3-19(31)12-21(20)28(32,33)34)10-18(9-15)26(41)36-24(13-25(39)40)16-2-5-22(29)23(30)11-16/h2-12,24,35H,13-14H2,1H3,(H,36,41)(H,39,40)	RAQJSTXWZYZUAB-UHFFFAOYSA-N	473528	US10844044, Example 84	WD repeat-containing protein 5		 0.120								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473528	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473528&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146455984	442073736							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981729	Cc1cc(ccc1F)[C@@H](NC(=O)c1cc(Cn2ccn(C)c2=N)cc(OCC2CC2)c1)C1CC1	InChI=1S/C27H31FN4O2/c1-17-11-21(7-8-24(17)28)25(20-5-6-20)30-26(33)22-12-19(15-32-10-9-31(2)27(32)29)13-23(14-22)34-16-18-3-4-18/h7-14,18,20,25,29H,3-6,15-16H2,1-2H3,(H,30,33)/t25-/m0/s1	YRPQVWISIYLPEG-VWLOTQADSA-N	473529	US10844044, Example 175	WD repeat-containing protein 5		 0.110								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473529	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473529&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146455862	442073737							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981730	FC(F)Oc1cc(F)ccc1-c1cc(CN2CCOC2=N)cc(c1)C(=O)N[C@@H](C1CC1)c1ccc(Cl)c(Cl)c1	InChI=1S/C28H24Cl2F3N3O3/c29-22-6-3-17(12-23(22)30)25(16-1-2-16)35-26(37)19-10-15(14-36-7-8-38-28(36)34)9-18(11-19)21-5-4-20(31)13-24(21)39-27(32)33/h3-6,9-13,16,25,27,34H,1-2,7-8,14H2,(H,35,37)/t25-/m0/s1	ODCAPKBRAXBICC-VWLOTQADSA-N	473530	US10844044, Example 267	WD repeat-containing protein 5		 0.180								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473530	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473530&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456132	442073738							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981731	Cc1cc(F)ccc1-c1cc(Cn2ccn(C)c2=N)cc(n1)C(=O)NCc1ccc(Cl)c(F)c1	InChI=1S/C25H22ClF2N5O/c1-15-9-18(27)4-5-19(15)22-11-17(14-33-8-7-32(2)25(33)29)12-23(31-22)24(34)30-13-16-3-6-20(26)21(28)10-16/h3-12,29H,13-14H2,1-2H3,(H,30,34)	BZHLONLNVCBWPX-UHFFFAOYSA-N	473531	US10844044, Example 359	WD repeat-containing protein 5		 8.70								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473531	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473531&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146457637	442073739							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981732	CCC(=O)CNC(=O)CC(NC(=O)c1cc(Cn2ccn(C)c2=N)cc(c1)-c1ccc(F)cc1C(F)(F)F)c1ccc(Cl)c(Cl)c1	InChI=1S/C32H29Cl2F4N5O3/c1-3-23(44)16-40-29(45)15-28(19-4-7-26(33)27(34)13-19)41-30(46)21-11-18(17-43-9-8-42(2)31(43)39)10-20(12-21)24-6-5-22(35)14-25(24)32(36,37)38/h4-14,28,39H,3,15-17H2,1-2H3,(H,40,45)(H,41,46)	JRSHGFVWYWHAEP-UHFFFAOYSA-N	473532	US10844044, Example 85	WD repeat-containing protein 5		<0.100								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473532	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473532&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456020	442073740							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981733	CCOc1cc(Cn2ccn(C)c2=N)cc(c1)C(=O)N[C@@H](C)c1ccc(F)c(C)c1	InChI=1S/C23H27FN4O2/c1-5-30-20-12-17(14-28-9-8-27(4)23(28)25)11-19(13-20)22(29)26-16(3)18-6-7-21(24)15(2)10-18/h6-13,16,25H,5,14H2,1-4H3,(H,26,29)/t16-/m0/s1	SAHMXGVBUHLXOZ-INIZCTEOSA-N	473533	US10844044, Example 176	WD repeat-containing protein 5		 0.500								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473533	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473533&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146455768	442073741							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981734	Cn1cc(c(n1)C(F)(F)F)-c1cc(Cn2ccoc2=N)cc(c1)C(=O)N[C@@H](C1CC1)c1ccc(Cl)c(Cl)c1	InChI=1S/C26H22Cl2F3N5O2/c1-35-13-19(23(34-35)26(29,30)31)17-8-14(12-36-6-7-38-25(36)32)9-18(10-17)24(37)33-22(15-2-3-15)16-4-5-20(27)21(28)11-16/h4-11,13,15,22,32H,2-3,12H2,1H3,(H,33,37)/t22-/m0/s1	RDJSRYLDRVEGFC-QFIPXVFZSA-N	473534	US10844044, Example 268	WD repeat-containing protein 5		<0.100								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473534	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473534&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146455845	442073742							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981735	C[C@@H](NC(=O)c1cc(Cn2ccn(C)c2=N)cc(n1)-c1ccc(F)cc1C)c1ccc(F)c(c1)C(F)(F)F	InChI=1S/C27H24F5N5O/c1-15-10-19(28)5-6-20(15)23-11-17(14-37-9-8-36(3)26(37)33)12-24(35-23)25(38)34-16(2)18-4-7-22(29)21(13-18)27(30,31)32/h4-13,16,33H,14H2,1-3H3,(H,34,38)/t16-/m1/s1	MXNOTMDQXCUSJW-MRXNPFEDSA-N	473535	US10844044, Example 360	WD repeat-containing protein 5		 1.000								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473535	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473535&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146455779	442073743							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981736	COc1cc(CNC(=O)CC(NC(=O)c2cc(Cn3ccn(C)c3=N)cc(c2)-c2ccc(F)cc2C(F)(F)F)c2ccc(Cl)c(Cl)c2)cc(OC)c1	InChI=1S/C37H33Cl2F4N5O4/c1-47-8-9-48(36(47)44)20-22-10-24(29-6-5-26(40)16-30(29)37(41,42)43)14-25(11-22)35(50)46-33(23-4-7-31(38)32(39)15-23)18-34(49)45-19-21-12-27(51-2)17-28(13-21)52-3/h4-17,33,44H,18-20H2,1-3H3,(H,45,49)(H,46,50)	KLZGTJNZLKUHAA-UHFFFAOYSA-N	473536	US10844044, Example 86	WD repeat-containing protein 5		 0.110								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473536	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473536&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146456352	442073744							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981737	CCOc1cc(Cn2ccn(C)c2=N)cc(c1)C(=O)NCc1cc(OC)cc(OC)c1	InChI=1S/C23H28N4O4/c1-5-31-21-11-17(15-27-7-6-26(2)23(27)24)8-18(12-21)22(28)25-14-16-9-19(29-3)13-20(10-16)30-4/h6-13,24H,5,14-15H2,1-4H3,(H,25,28)	MXEMLIYWLKECMZ-UHFFFAOYSA-N	473537	US10844044, Example 177	WD repeat-containing protein 5		 3.90								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473537	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473537&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146457642	442073745							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
981738	Cn1cc(c(n1)C(F)(F)F)-c1cc(CN2CCOC2=N)cc(c1)C(=O)N[C@@H](C1CC1)c1ccc(Cl)c(Cl)c1	InChI=1S/C26H24Cl2F3N5O2/c1-35-13-19(23(34-35)26(29,30)31)17-8-14(12-36-6-7-38-25(36)32)9-18(10-17)24(37)33-22(15-2-3-15)16-4-5-20(27)21(28)11-16/h4-5,8-11,13,15,22,32H,2-3,6-7,12H2,1H3,(H,33,37)/t22-/m0/s1	GSBNPUGOFDRXIP-QFIPXVFZSA-N	473538	US10844044, Example 269	WD repeat-containing protein 5		<0.100								US Patent		10.7270/Q21R6TKB		aid1805048	US10844044	Alvarado, JR; Stauffer, SR; Gogliotti, RD; Han, C; Meyers, KM; Tian, J; Macdonald, JD; Fesik, SW; Lee, T	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=473538	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=473538&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146455734	442073746							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51329908	Oc1c(Cl)cc(Br)cc1S(=O)(=O)Nc1cn(cn1)C1CCCCC1	InChI=1S/C15H17BrClN3O3S/c16-10-6-12(17)15(21)13(7-10)24(22,23)19-14-8-20(9-18-14)11-4-2-1-3-5-11/h6-9,11,19,21H,1-5H2	FZZVAOWEPRLNJJ-UHFFFAOYSA-N	50538275	CHEMBL4633122	WD repeat-containing protein 5				 1000						ChEMBL	10.1021/acs.jmedchem.0c00224	10.7270/Q20G3PNC	32223236			Chacón Simon, S; Wang, F; Thomas, LR; Phan, J; Zhao, B; Olejniczak, ET; Macdonald, JD; Shaw, JG; Schlund, C; Payne, W; Creighton, J; Stauffer, SR; Waterson, AG; Tansey, WP; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50538275	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50538275&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			156010175	442139838							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51329909	Oc1c(Cl)cc(Br)cc1S(=O)(=O)Nc1cn(cn1)-c1ccccc1	InChI=1S/C15H11BrClN3O3S/c16-10-6-12(17)15(21)13(7-10)24(22,23)19-14-8-20(9-18-14)11-4-2-1-3-5-11/h1-9,19,21H	XMFFLMGSEPXKEH-UHFFFAOYSA-N	50538276	CHEMBL4634425	WD repeat-containing protein 5				 3200						ChEMBL	10.1021/acs.jmedchem.0c00224	10.7270/Q20G3PNC	32223236			Chacón Simon, S; Wang, F; Thomas, LR; Phan, J; Zhao, B; Olejniczak, ET; Macdonald, JD; Shaw, JG; Schlund, C; Payne, W; Creighton, J; Stauffer, SR; Waterson, AG; Tansey, WP; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50538276	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50538276&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			156009733	442139839							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51329910	Oc1c(Cl)cc(Br)cc1S(=O)(=O)Nc1cn(cn1)-c1ccccc1C(F)(F)F	InChI=1S/C16H10BrClF3N3O3S/c17-9-5-11(18)15(25)13(6-9)28(26,27)23-14-7-24(8-22-14)12-4-2-1-3-10(12)16(19,20)21/h1-8,23,25H	AKZGUJQADWDMGW-UHFFFAOYSA-N	50538277	CHEMBL4647265	WD repeat-containing protein 5				 4000						ChEMBL	10.1021/acs.jmedchem.0c00224	10.7270/Q20G3PNC	32223236			Chacón Simon, S; Wang, F; Thomas, LR; Phan, J; Zhao, B; Olejniczak, ET; Macdonald, JD; Shaw, JG; Schlund, C; Payne, W; Creighton, J; Stauffer, SR; Waterson, AG; Tansey, WP; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50538277	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50538277&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			156021686	442139840							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51329911	CC(C)CCn1cnc(NS(=O)(=O)c2cc(Br)cc(Cl)c2O)c1	InChI=1S/C14H17BrClN3O3S/c1-9(2)3-4-19-7-13(17-8-19)18-23(21,22)12-6-10(15)5-11(16)14(12)20/h5-9,18,20H,3-4H2,1-2H3	XGIJWWJNPQPKBI-UHFFFAOYSA-N	50538278	CHEMBL4641551	WD repeat-containing protein 5				 5200						ChEMBL	10.1021/acs.jmedchem.0c00224	10.7270/Q20G3PNC	32223236			Chacón Simon, S; Wang, F; Thomas, LR; Phan, J; Zhao, B; Olejniczak, ET; Macdonald, JD; Shaw, JG; Schlund, C; Payne, W; Creighton, J; Stauffer, SR; Waterson, AG; Tansey, WP; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50538278	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50538278&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			156016842	442139841							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51329912	Oc1c(Cl)cc(Br)cc1S(=O)(=O)Nc1cn(cn1)C(C1CC1)C1CC1	InChI=1S/C16H17BrClN3O3S/c17-11-5-12(18)16(22)13(6-11)25(23,24)20-14-7-21(8-19-14)15(9-1-2-9)10-3-4-10/h5-10,15,20,22H,1-4H2	KMTMRKUFHUQWTN-UHFFFAOYSA-N	50538279	CHEMBL4645526	WD repeat-containing protein 5				 1200						ChEMBL	10.1021/acs.jmedchem.0c00224	10.7270/Q20G3PNC	32223236			Chacón Simon, S; Wang, F; Thomas, LR; Phan, J; Zhao, B; Olejniczak, ET; Macdonald, JD; Shaw, JG; Schlund, C; Payne, W; Creighton, J; Stauffer, SR; Waterson, AG; Tansey, WP; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50538279	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50538279&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			156019544	442139842							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51329913	CC(C)n1cnc(NS(=O)(=O)c2cc(Br)cc(Cl)c2O)c1	InChI=1S/C12H13BrClN3O3S/c1-7(2)17-5-11(15-6-17)16-21(19,20)10-4-8(13)3-9(14)12(10)18/h3-7,16,18H,1-2H3	GBSCURWKEPCSPX-UHFFFAOYSA-N	50538280	CHEMBL4636991	WD repeat-containing protein 5				 5500						ChEMBL	10.1021/acs.jmedchem.0c00224	10.7270/Q20G3PNC	32223236			Chacón Simon, S; Wang, F; Thomas, LR; Phan, J; Zhao, B; Olejniczak, ET; Macdonald, JD; Shaw, JG; Schlund, C; Payne, W; Creighton, J; Stauffer, SR; Waterson, AG; Tansey, WP; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50538280	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50538280&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			156011251	442139843							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51329914	Oc1c(Cl)cc(Br)cc1S(=O)(=O)Nc1cn(cn1)C1CC1	InChI=1S/C12H11BrClN3O3S/c13-7-3-9(14)12(18)10(4-7)21(19,20)16-11-5-17(6-15-11)8-1-2-8/h3-6,8,16,18H,1-2H2	YEVKDDIKGMTEBP-UHFFFAOYSA-N	50538281	CHEMBL4634759	WD repeat-containing protein 5				 4000						ChEMBL	10.1021/acs.jmedchem.0c00224	10.7270/Q20G3PNC	32223236			Chacón Simon, S; Wang, F; Thomas, LR; Phan, J; Zhao, B; Olejniczak, ET; Macdonald, JD; Shaw, JG; Schlund, C; Payne, W; Creighton, J; Stauffer, SR; Waterson, AG; Tansey, WP; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50538281	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50538281&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			156014769	442139844							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51329915	Oc1c(Cl)cc(Br)cc1S(=O)(=O)Nc1cn(cn1)C1CCC1	InChI=1S/C13H13BrClN3O3S/c14-8-4-10(15)13(19)11(5-8)22(20,21)17-12-6-18(7-16-12)9-2-1-3-9/h4-7,9,17,19H,1-3H2	PJAVKNBPZPRFPY-UHFFFAOYSA-N	50538282	CHEMBL4638849	WD repeat-containing protein 5				 400						ChEMBL	10.1021/acs.jmedchem.0c00224	10.7270/Q20G3PNC	32223236			Chacón Simon, S; Wang, F; Thomas, LR; Phan, J; Zhao, B; Olejniczak, ET; Macdonald, JD; Shaw, JG; Schlund, C; Payne, W; Creighton, J; Stauffer, SR; Waterson, AG; Tansey, WP; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50538282	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50538282&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			156012870	442139845							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51329916	Oc1c(Cl)cc(Br)cc1S(=O)(=O)Nc1cn(cn1)C1CCCC1	InChI=1S/C14H15BrClN3O3S/c15-9-5-11(16)14(20)12(6-9)23(21,22)18-13-7-19(8-17-13)10-3-1-2-4-10/h5-8,10,18,20H,1-4H2	RWBIWQQGKHMDCL-UHFFFAOYSA-N	50538283	CHEMBL4633372	WD repeat-containing protein 5				 400						ChEMBL	10.1021/acs.jmedchem.0c00224	10.7270/Q20G3PNC	32223236			Chacón Simon, S; Wang, F; Thomas, LR; Phan, J; Zhao, B; Olejniczak, ET; Macdonald, JD; Shaw, JG; Schlund, C; Payne, W; Creighton, J; Stauffer, SR; Waterson, AG; Tansey, WP; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50538283	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50538283&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	Q8M	6UIK	146019257	442139846							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51329917	Oc1c(Cl)cc(Br)cc1S(=O)(=O)Nc1cn(cn1)C1CCNC1	InChI=1S/C13H14BrClN4O3S/c14-8-3-10(15)13(20)11(4-8)23(21,22)18-12-6-19(7-17-12)9-1-2-16-5-9/h3-4,6-7,9,16,18,20H,1-2,5H2	GGQZIACXEPHTRW-UHFFFAOYSA-N	50538284	CHEMBL4641549	WD repeat-containing protein 5				 11000						ChEMBL	10.1021/acs.jmedchem.0c00224	10.7270/Q20G3PNC	32223236			Chacón Simon, S; Wang, F; Thomas, LR; Phan, J; Zhao, B; Olejniczak, ET; Macdonald, JD; Shaw, JG; Schlund, C; Payne, W; Creighton, J; Stauffer, SR; Waterson, AG; Tansey, WP; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50538284	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50538284&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			156016770	442139847							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51329918	Oc1c(Cl)cc(Br)cc1S(=O)(=O)Nc1cn(CC2CC2)cn1	InChI=1S/C13H13BrClN3O3S/c14-9-3-10(15)13(19)11(4-9)22(20,21)17-12-6-18(7-16-12)5-8-1-2-8/h3-4,6-8,17,19H,1-2,5H2	CMFUFHNCKKLBPA-UHFFFAOYSA-N	50538285	CHEMBL4648697	WD repeat-containing protein 5				 2100						ChEMBL	10.1021/acs.jmedchem.0c00224	10.7270/Q20G3PNC	32223236			Chacón Simon, S; Wang, F; Thomas, LR; Phan, J; Zhao, B; Olejniczak, ET; Macdonald, JD; Shaw, JG; Schlund, C; Payne, W; Creighton, J; Stauffer, SR; Waterson, AG; Tansey, WP; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50538285	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50538285&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			156020624	442139848							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51329919	Oc1c(Cl)cc(Br)cc1S(=O)(=O)Nc1cn(CC2CCC2)cn1	InChI=1S/C14H15BrClN3O3S/c15-10-4-11(16)14(20)12(5-10)23(21,22)18-13-7-19(8-17-13)6-9-2-1-3-9/h4-5,7-9,18,20H,1-3,6H2	VHXYZRGTMOTLLX-UHFFFAOYSA-N	50538286	CHEMBL4633432	WD repeat-containing protein 5				 4500						ChEMBL	10.1021/acs.jmedchem.0c00224	10.7270/Q20G3PNC	32223236			Chacón Simon, S; Wang, F; Thomas, LR; Phan, J; Zhao, B; Olejniczak, ET; Macdonald, JD; Shaw, JG; Schlund, C; Payne, W; Creighton, J; Stauffer, SR; Waterson, AG; Tansey, WP; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50538286	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50538286&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			156010983	442139849							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51329920	Oc1c(Cl)cc(Br)cc1S(=O)(=O)Nc1cn(CC2CCCC2)cn1	InChI=1S/C15H17BrClN3O3S/c16-11-5-12(17)15(21)13(6-11)24(22,23)19-14-8-20(9-18-14)7-10-3-1-2-4-10/h5-6,8-10,19,21H,1-4,7H2	JCNFDVNFZYOCKC-UHFFFAOYSA-N	50538287	CHEMBL4648074	WD repeat-containing protein 5				 3400						ChEMBL	10.1021/acs.jmedchem.0c00224	10.7270/Q20G3PNC	32223236			Chacón Simon, S; Wang, F; Thomas, LR; Phan, J; Zhao, B; Olejniczak, ET; Macdonald, JD; Shaw, JG; Schlund, C; Payne, W; Creighton, J; Stauffer, SR; Waterson, AG; Tansey, WP; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50538287	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50538287&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			156021747	442139850							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51329921	Oc1c(Cl)cc(Br)cc1S(=O)(=O)Nc1cn(CC2CCCO2)cn1	InChI=1S/C14H15BrClN3O4S/c15-9-4-11(16)14(20)12(5-9)24(21,22)18-13-7-19(8-17-13)6-10-2-1-3-23-10/h4-5,7-8,10,18,20H,1-3,6H2	UALDIBGYNTXQLJ-UHFFFAOYSA-N	50538288	CHEMBL4635124	WD repeat-containing protein 5				 8000						ChEMBL	10.1021/acs.jmedchem.0c00224	10.7270/Q20G3PNC	32223236			Chacón Simon, S; Wang, F; Thomas, LR; Phan, J; Zhao, B; Olejniczak, ET; Macdonald, JD; Shaw, JG; Schlund, C; Payne, W; Creighton, J; Stauffer, SR; Waterson, AG; Tansey, WP; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50538288	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50538288&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			156013859	442139851							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51329922	Oc1c(Cl)cc(Br)cc1S(=O)(=O)Nc1cn(cn1)C(=O)C1CCC1	InChI=1S/C14H13BrClN3O4S/c15-9-4-10(16)13(20)11(5-9)24(22,23)18-12-6-19(7-17-12)14(21)8-2-1-3-8/h4-8,18,20H,1-3H2	FVJKMFGFDGVUDM-UHFFFAOYSA-N	50538289	CHEMBL4643031	WD repeat-containing protein 5				 38000						ChEMBL	10.1021/acs.jmedchem.0c00224	10.7270/Q20G3PNC	32223236			Chacón Simon, S; Wang, F; Thomas, LR; Phan, J; Zhao, B; Olejniczak, ET; Macdonald, JD; Shaw, JG; Schlund, C; Payne, W; Creighton, J; Stauffer, SR; Waterson, AG; Tansey, WP; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50538289	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50538289&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			156016897	442139852							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51329923	Oc1c(Cl)cc(Br)cc1S(=O)(=O)Nc1cn(cn1)C(=O)C1CCCC1	InChI=1S/C15H15BrClN3O4S/c16-10-5-11(17)14(21)12(6-10)25(23,24)19-13-7-20(8-18-13)15(22)9-3-1-2-4-9/h5-9,19,21H,1-4H2	XXPSSVTZQXENQC-UHFFFAOYSA-N	50538290	CHEMBL4637280	WD repeat-containing protein 5				>40000						ChEMBL	10.1021/acs.jmedchem.0c00224	10.7270/Q20G3PNC	32223236			Chacón Simon, S; Wang, F; Thomas, LR; Phan, J; Zhao, B; Olejniczak, ET; Macdonald, JD; Shaw, JG; Schlund, C; Payne, W; Creighton, J; Stauffer, SR; Waterson, AG; Tansey, WP; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50538290	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50538290&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			156012444	442139853							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51329924	Oc1c(Cl)cc(Br)cc1S(=O)(=O)Nc1ncn(n1)C1CCCC1	InChI=1S/C13H14BrClN4O3S/c14-8-5-10(15)12(20)11(6-8)23(21,22)18-13-16-7-19(17-13)9-3-1-2-4-9/h5-7,9,20H,1-4H2,(H,17,18)	ZTNASIJCJJOEPJ-UHFFFAOYSA-N	50538291	CHEMBL4638610	WD repeat-containing protein 5				 6500						ChEMBL	10.1021/acs.jmedchem.0c00224	10.7270/Q20G3PNC	32223236			Chacón Simon, S; Wang, F; Thomas, LR; Phan, J; Zhao, B; Olejniczak, ET; Macdonald, JD; Shaw, JG; Schlund, C; Payne, W; Creighton, J; Stauffer, SR; Waterson, AG; Tansey, WP; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50538291	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50538291&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			156012057	442139854							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51329925	Oc1c(Cl)cc(Br)cc1S(=O)(=O)Nc1cc([nH]n1)C1CCCC1	InChI=1S/C14H15BrClN3O3S/c15-9-5-10(16)14(20)12(6-9)23(21,22)19-13-7-11(17-18-13)8-3-1-2-4-8/h5-8,20H,1-4H2,(H2,17,18,19)	FGOJVAFRJXBUNV-UHFFFAOYSA-N	50538292	CHEMBL4643054	WD repeat-containing protein 5				 10000						ChEMBL	10.1021/acs.jmedchem.0c00224	10.7270/Q20G3PNC	32223236			Chacón Simon, S; Wang, F; Thomas, LR; Phan, J; Zhao, B; Olejniczak, ET; Macdonald, JD; Shaw, JG; Schlund, C; Payne, W; Creighton, J; Stauffer, SR; Waterson, AG; Tansey, WP; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50538292	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50538292&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			156017157	442139855							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51329926	Oc1c(Cl)cc(Br)cc1S(=O)(=O)Nc1ccn(n1)C1CCCC1	InChI=1S/C14H15BrClN3O3S/c15-9-7-11(16)14(20)12(8-9)23(21,22)18-13-5-6-19(17-13)10-3-1-2-4-10/h5-8,10,20H,1-4H2,(H,17,18)	XDCWMSIPCXCWPV-UHFFFAOYSA-N	50538293	CHEMBL4646306	WD repeat-containing protein 5				 2800						ChEMBL	10.1021/acs.jmedchem.0c00224	10.7270/Q20G3PNC	32223236			Chacón Simon, S; Wang, F; Thomas, LR; Phan, J; Zhao, B; Olejniczak, ET; Macdonald, JD; Shaw, JG; Schlund, C; Payne, W; Creighton, J; Stauffer, SR; Waterson, AG; Tansey, WP; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50538293	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50538293&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			156019250	442139856							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51329927	Oc1c(Cl)cc(Br)cc1S(=O)(=O)Nc1cnn(c1)C1CCCC1	InChI=1S/C14H15BrClN3O3S/c15-9-5-12(16)14(20)13(6-9)23(21,22)18-10-7-17-19(8-10)11-3-1-2-4-11/h5-8,11,18,20H,1-4H2	RHSXBKMORBGXGZ-UHFFFAOYSA-N	50538294	CHEMBL4638448	WD repeat-containing protein 5				 500						ChEMBL	10.1021/acs.jmedchem.0c00224	10.7270/Q20G3PNC	32223236			Chacón Simon, S; Wang, F; Thomas, LR; Phan, J; Zhao, B; Olejniczak, ET; Macdonald, JD; Shaw, JG; Schlund, C; Payne, W; Creighton, J; Stauffer, SR; Waterson, AG; Tansey, WP; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50538294	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50538294&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			156011626	442139857							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51329928	Oc1c(Cl)cc(Br)cc1S(=O)(=O)Nc1cnc(s1)C1CCCC1	InChI=1S/C14H14BrClN2O3S2/c15-9-5-10(16)13(19)11(6-9)23(20,21)18-12-7-17-14(22-12)8-3-1-2-4-8/h5-8,18-19H,1-4H2	LDAQTKBEYCKNFI-UHFFFAOYSA-N	50538295	CHEMBL4635166	WD repeat-containing protein 5				 600						ChEMBL	10.1021/acs.jmedchem.0c00224	10.7270/Q20G3PNC	32223236			Chacón Simon, S; Wang, F; Thomas, LR; Phan, J; Zhao, B; Olejniczak, ET; Macdonald, JD; Shaw, JG; Schlund, C; Payne, W; Creighton, J; Stauffer, SR; Waterson, AG; Tansey, WP; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50538295	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50538295&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			156014182	442139858							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51329929	Oc1c(Cl)cc(Br)cc1S(=O)(=O)Nc1nc2ccccc2s1	InChI=1S/C13H8BrClN2O3S2/c14-7-5-8(15)12(18)11(6-7)22(19,20)17-13-16-9-3-1-2-4-10(9)21-13/h1-6,18H,(H,16,17)	JWKJZSDYBFIOAA-UHFFFAOYSA-N	50538296	CHEMBL4632873	WD repeat-containing protein 5				 32000						ChEMBL	10.1021/acs.jmedchem.0c00224	10.7270/Q20G3PNC	32223236			Chacón Simon, S; Wang, F; Thomas, LR; Phan, J; Zhao, B; Olejniczak, ET; Macdonald, JD; Shaw, JG; Schlund, C; Payne, W; Creighton, J; Stauffer, SR; Waterson, AG; Tansey, WP; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50538296	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50538296&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			156009484	442139859							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51329930	Cc1nc(NS(=O)(=O)c2cc(Br)cc(Cl)c2O)cn1C1CCCC1	InChI=1S/C15H17BrClN3O3S/c1-9-18-14(8-20(9)11-4-2-3-5-11)19-24(22,23)13-7-10(16)6-12(17)15(13)21/h6-8,11,19,21H,2-5H2,1H3	WOKCPJTYIUMFPY-UHFFFAOYSA-N	50538297	CHEMBL4637994	WD repeat-containing protein 5				 170						ChEMBL	10.1021/acs.jmedchem.0c00224	10.7270/Q20G3PNC	32223236			Chacón Simon, S; Wang, F; Thomas, LR; Phan, J; Zhao, B; Olejniczak, ET; Macdonald, JD; Shaw, JG; Schlund, C; Payne, W; Creighton, J; Stauffer, SR; Waterson, AG; Tansey, WP; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50538297	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50538297&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	Q8S	6UJ4	146019258	442139860							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51329931	CCc1nc(NS(=O)(=O)c2cc(Br)cc(Cl)c2O)cn1C1CCCC1	InChI=1S/C16H19BrClN3O3S/c1-2-15-19-14(9-21(15)11-5-3-4-6-11)20-25(23,24)13-8-10(17)7-12(18)16(13)22/h7-9,11,20,22H,2-6H2,1H3	VBUFZLSUDGCPNO-UHFFFAOYSA-N	50538298	CHEMBL4633333	WD repeat-containing protein 5				 220						ChEMBL	10.1021/acs.jmedchem.0c00224	10.7270/Q20G3PNC	32223236			Chacón Simon, S; Wang, F; Thomas, LR; Phan, J; Zhao, B; Olejniczak, ET; Macdonald, JD; Shaw, JG; Schlund, C; Payne, W; Creighton, J; Stauffer, SR; Waterson, AG; Tansey, WP; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50538298	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50538298&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			156011093	442139861							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51329932	CCOC(=O)c1nc(NS(=O)(=O)c2cc(Br)cc(Cl)c2O)cn1C1CCCC1	InChI=1S/C17H19BrClN3O5S/c1-2-27-17(24)16-20-14(9-22(16)11-5-3-4-6-11)21-28(25,26)13-8-10(18)7-12(19)15(13)23/h7-9,11,21,23H,2-6H2,1H3	OMVJLLWQQVXLOS-UHFFFAOYSA-N	50538299	CHEMBL4648241	WD repeat-containing protein 5				 110						ChEMBL	10.1021/acs.jmedchem.0c00224	10.7270/Q20G3PNC	32223236			Chacón Simon, S; Wang, F; Thomas, LR; Phan, J; Zhao, B; Olejniczak, ET; Macdonald, JD; Shaw, JG; Schlund, C; Payne, W; Creighton, J; Stauffer, SR; Waterson, AG; Tansey, WP; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50538299	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50538299&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			156020175	442139862							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51329933	OC(=O)c1nc(NS(=O)(=O)c2cc(Br)cc(Cl)c2O)cn1C1CCCC1	InChI=1S/C15H15BrClN3O5S/c16-8-5-10(17)13(21)11(6-8)26(24,25)19-12-7-20(9-3-1-2-4-9)14(18-12)15(22)23/h5-7,9,19,21H,1-4H2,(H,22,23)	AWBDBLSUZBKJLN-UHFFFAOYSA-N	50538300	CHEMBL4644171	WD repeat-containing protein 5				 700						ChEMBL	10.1021/acs.jmedchem.0c00224	10.7270/Q20G3PNC	32223236			Chacón Simon, S; Wang, F; Thomas, LR; Phan, J; Zhao, B; Olejniczak, ET; Macdonald, JD; Shaw, JG; Schlund, C; Payne, W; Creighton, J; Stauffer, SR; Waterson, AG; Tansey, WP; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50538300	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50538300&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			156018573	442139863							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51329934	CNC(=O)c1nc(NS(=O)(=O)c2cc(Br)cc(Cl)c2O)cn1C1CCCC1	InChI=1S/C16H18BrClN4O4S/c1-19-16(24)15-20-13(8-22(15)10-4-2-3-5-10)21-27(25,26)12-7-9(17)6-11(18)14(12)23/h6-8,10,21,23H,2-5H2,1H3,(H,19,24)	KXQTXSQWNIVQDX-UHFFFAOYSA-N	50538301	CHEMBL4641743	WD repeat-containing protein 5				 170						ChEMBL	10.1021/acs.jmedchem.0c00224	10.7270/Q20G3PNC	32223236			Chacón Simon, S; Wang, F; Thomas, LR; Phan, J; Zhao, B; Olejniczak, ET; Macdonald, JD; Shaw, JG; Schlund, C; Payne, W; Creighton, J; Stauffer, SR; Waterson, AG; Tansey, WP; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50538301	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50538301&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	Q8P	6UIF	146019256	442139864							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51329935	Oc1c(Cl)cc(Br)cc1S(=O)(=O)Nc1cn(C2CCCC2)c(n1)C(=O)N1CCC(CC1)C1CCCN1	InChI=1S/C24H31BrClN5O4S/c25-16-12-18(26)22(32)20(13-16)36(34,35)29-21-14-31(17-4-1-2-5-17)23(28-21)24(33)30-10-7-15(8-11-30)19-6-3-9-27-19/h12-15,17,19,27,29,32H,1-11H2	CHSPMECAFQPIHC-UHFFFAOYSA-N	50538302	CHEMBL4645266	WD repeat-containing protein 5				 5000						ChEMBL	10.1021/acs.jmedchem.0c00224	10.7270/Q20G3PNC	32223236			Chacón Simon, S; Wang, F; Thomas, LR; Phan, J; Zhao, B; Olejniczak, ET; Macdonald, JD; Shaw, JG; Schlund, C; Payne, W; Creighton, J; Stauffer, SR; Waterson, AG; Tansey, WP; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50538302	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50538302&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			156017981	442139865							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51329936	COCCN1CCN(CC1)C(=O)c1nc(NS(=O)(=O)c2cc(Br)cc(Cl)c2O)cn1C1CCCC1	InChI=1S/C22H29BrClN5O5S/c1-34-11-10-27-6-8-28(9-7-27)22(31)21-25-19(14-29(21)16-4-2-3-5-16)26-35(32,33)18-13-15(23)12-17(24)20(18)30/h12-14,16,26,30H,2-11H2,1H3	OOJJVYVRJMFBEG-UHFFFAOYSA-N	50538303	CHEMBL4637200	WD repeat-containing protein 5				 1100						ChEMBL	10.1021/acs.jmedchem.0c00224	10.7270/Q20G3PNC	32223236			Chacón Simon, S; Wang, F; Thomas, LR; Phan, J; Zhao, B; Olejniczak, ET; Macdonald, JD; Shaw, JG; Schlund, C; Payne, W; Creighton, J; Stauffer, SR; Waterson, AG; Tansey, WP; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50538303	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50538303&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			156011783	442139866							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51329937	Oc1c(Cl)cc(Br)cc1S(=O)(=O)Nc1cn(C2CCCC2)c(n1)C(=O)N1CC2(CNC2)C1	InChI=1S/C20H23BrClN5O4S/c21-12-5-14(22)17(28)15(6-12)32(30,31)25-16-7-27(13-3-1-2-4-13)18(24-16)19(29)26-10-20(11-26)8-23-9-20/h5-7,13,23,25,28H,1-4,8-11H2	YXSSAEISOLMROH-UHFFFAOYSA-N	50538304	CHEMBL4647872	WD repeat-containing protein 5				 2300						ChEMBL	10.1021/acs.jmedchem.0c00224	10.7270/Q20G3PNC	32223236			Chacón Simon, S; Wang, F; Thomas, LR; Phan, J; Zhao, B; Olejniczak, ET; Macdonald, JD; Shaw, JG; Schlund, C; Payne, W; Creighton, J; Stauffer, SR; Waterson, AG; Tansey, WP; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50538304	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50538304&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			156020009	442139867							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51329938	CS(=O)(=O)c1nc(NS(=O)(=O)c2cc(Br)cc(Cl)c2O)cn1C1CCCC1	InChI=1S/C15H17BrClN3O5S2/c1-26(22,23)15-18-13(8-20(15)10-4-2-3-5-10)19-27(24,25)12-7-9(16)6-11(17)14(12)21/h6-8,10,19,21H,2-5H2,1H3	ZBIVDOJYQHNICX-UHFFFAOYSA-N	50538305	CHEMBL4645862	WD repeat-containing protein 5				 100						ChEMBL	10.1021/acs.jmedchem.0c00224	10.7270/Q20G3PNC	32223236			Chacón Simon, S; Wang, F; Thomas, LR; Phan, J; Zhao, B; Olejniczak, ET; Macdonald, JD; Shaw, JG; Schlund, C; Payne, W; Creighton, J; Stauffer, SR; Waterson, AG; Tansey, WP; Fesik, SW	Vanderbilt University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50538305	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50538305&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	QF1	6UOZ	146019259	442139868							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1110989	CN1CCN(CC1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cccc(CN2CCOCC2)c1	InChI=1S/C29H32F3N5O3/c1-35-7-9-37(10-8-35)26-6-5-22(21-4-2-3-20(15-21)19-36-11-13-40-14-12-36)16-25(26)34-28(39)23-18-33-27(38)17-24(23)29(30,31)32/h2-6,15-18H,7-14,19H2,1H3,(H,33,38)(H,34,39)	DJOVLOYCGXNVPI-UHFFFAOYSA-N	50164794	CHEMBL3798846::US11174250, Example Table4.1.1::US11319299, Comp. No. 57	WD repeat-containing protein 5				 36.0						US Patent		10.7270/Q2C53Q0K		aid1806103	US11174250	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50164794	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50164794&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	35Q	4QL1	91623360	341097539		CHEMBL3798846					1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1110991	CN1CCN(CC1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cc(CN2CCOCC2)ccc1F	InChI=1S/C29H31F4N5O3/c1-36-6-8-38(9-7-36)26-5-3-20(21-14-19(2-4-24(21)30)18-37-10-12-41-13-11-37)15-25(26)35-28(40)22-17-34-27(39)16-23(22)29(31,32)33/h2-5,14-17H,6-13,18H2,1H3,(H,34,39)(H,35,40)	HJPMPWYSTRBBLP-UHFFFAOYSA-N	525575	US11174250, Example 2::US11174250, Example Table4.1.2::US11174250, Example Table4.3.2	WD repeat-containing protein 5				 11.0						US Patent		10.7270/Q2C53Q0K		aid1806103	US11174250	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=525575	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=525575&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			163199813	463789229							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1110993	CN1CCN(CC1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cccc(CN2CCC(F)CC2)c1	InChI=1S/C30H33F4N5O2/c1-37-11-13-39(14-12-37)27-6-5-22(21-4-2-3-20(15-21)19-38-9-7-23(31)8-10-38)16-26(27)36-29(41)24-18-35-28(40)17-25(24)30(32,33)34/h2-6,15-18,23H,7-14,19H2,1H3,(H,35,40)(H,36,41)	KKEXEXDHWKMRQV-UHFFFAOYSA-N	525577	US11174250, Example Table4.2.1	WD repeat-containing protein 5				 30.0						US Patent		10.7270/Q2C53Q0K		aid1806103	US11174250	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=525577	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=525577&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			163199814	463789231							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1110994	CN1CCN(CC1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cc(CN2CCC(F)CC2)ccc1F	InChI=1S/C30H32F5N5O2/c1-38-10-12-40(13-11-38)27-5-3-20(22-14-19(2-4-25(22)32)18-39-8-6-21(31)7-9-39)15-26(27)37-29(42)23-17-36-28(41)16-24(23)30(33,34)35/h2-5,14-17,21H,6-13,18H2,1H3,(H,36,41)(H,37,42)	LCHGERIHAPDZCU-UHFFFAOYSA-N	525578	US11174250, Example 73::US11174250, Example Table4.2.2	WD repeat-containing protein 5				 11.0						US Patent		10.7270/Q2C53Q0K		aid1806103	US11174250	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=525578	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=525578&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			163199815	463789232							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1110996	CN1CCN(CC1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cc(CN2CCOCC2)ccc1Cl	InChI=1S/C29H31ClF3N5O3/c1-36-6-8-38(9-7-36)26-5-3-20(21-14-19(2-4-24(21)30)18-37-10-12-41-13-11-37)15-25(26)35-28(40)22-17-34-27(39)16-23(22)29(31,32)33/h2-5,14-17H,6-13,18H2,1H3,(H,34,39)(H,35,40)	FOAUMOZOTVHACR-UHFFFAOYSA-N	525579	US11174250, Example 86::US11174250, Example Table4.3.1	WD repeat-containing protein 5				 34.5						US Patent		10.7270/Q2C53Q0K		aid1806103	US11174250	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=525579	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=525579&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			163199816	463789233							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1110997	CN1CCN(CC1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cc(CN2CCOCC2)ccc1F	InChI=1S/C29H31F4N5O3/c1-36-6-8-38(9-7-36)26-5-3-20(21-14-19(2-4-24(21)30)18-37-10-12-41-13-11-37)15-25(26)35-28(40)22-17-34-27(39)16-23(22)29(31,32)33/h2-5,14-17H,6-13,18H2,1H3,(H,34,39)(H,35,40)	HJPMPWYSTRBBLP-UHFFFAOYSA-N	525575	US11174250, Example 2::US11174250, Example Table4.1.2::US11174250, Example Table4.3.2	WD repeat-containing protein 5				 11.0						US Patent		10.7270/Q2C53Q0K		aid1806103	US11174250	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=525575	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=525575&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			163199813	463789229							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1110999	CN1CCN(CC1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cc(ccc1Cl)C(=O)NC1CCCCC1	InChI=1S/C31H33ClF3N5O3/c1-39-11-13-40(14-12-39)27-10-8-19(16-26(27)38-30(43)23-18-36-28(41)17-24(23)31(33,34)35)22-15-20(7-9-25(22)32)29(42)37-21-5-3-2-4-6-21/h7-10,15-18,21H,2-6,11-14H2,1H3,(H,36,41)(H,37,42)(H,38,43)	QYUSSNJDVILCJQ-UHFFFAOYSA-N	525581	US11174250, Example 116::US11174250, Example Table4.4.1	WD repeat-containing protein 5				 13.2						US Patent		10.7270/Q2C53Q0K		aid1806103	US11174250	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=525581	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=525581&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			163199817	463789234							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1111000	CN1CCN(CC1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cc(ccc1F)C(=O)NC1CCCCC1	InChI=1S/C31H33F4N5O3/c1-39-11-13-40(14-12-39)27-10-8-19(16-26(27)38-30(43)23-18-36-28(41)17-24(23)31(33,34)35)22-15-20(7-9-25(22)32)29(42)37-21-5-3-2-4-6-21/h7-10,15-18,21H,2-6,11-14H2,1H3,(H,36,41)(H,37,42)(H,38,43)	GLHJOTVYVUCLQO-UHFFFAOYSA-N	525582	US11174250, Example 32::US11174250, Example Table4.4.2	WD repeat-containing protein 5				 6.00						US Patent		10.7270/Q2C53Q0K		aid1806103	US11174250	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=525582	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=525582&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			163199818	463789235							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1111001	C[C@H]1CN(Cc2ccc(F)c(c2)-c2ccc(N3CCN(C)CC3)c(NC(=O)c3c[nH]c(=O)cc3C(F)(F)F)c2)C[C@@H](C)O1			525583	US11174250, Example 1	WD repeat-containing protein 5				 17.0						US Patent		10.7270/Q2C53Q0K		aid1806103	US11174250	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=525583	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=525583&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			163199819	463789236							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1111003	CN1CCN(CC1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cc(CN2CCOCC2)ccc1F	InChI=1S/C29H31F4N5O3/c1-36-6-8-38(9-7-36)26-5-3-20(21-14-19(2-4-24(21)30)18-37-10-12-41-13-11-37)15-25(26)35-28(40)22-17-34-27(39)16-23(22)29(31,32)33/h2-5,14-17H,6-13,18H2,1H3,(H,34,39)(H,35,40)	HJPMPWYSTRBBLP-UHFFFAOYSA-N	525575	US11174250, Example 2::US11174250, Example Table4.1.2::US11174250, Example Table4.3.2	WD repeat-containing protein 5				 11.0						US Patent		10.7270/Q2C53Q0K		aid1806103	US11174250	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=525575	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=525575&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			163199813	463789229							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1111005	COCOc1cc(F)c(cc1C(=O)NC(C)(C)CC(C)(C)C)-c1ccc(N2CCN(C)CC2)c(NC(=O)c2c[nH]c(=O)cc2C(F)(F)F)c1	InChI=1S/C35H43F4N5O5/c1-33(2,3)19-34(4,5)42-32(47)23-15-22(26(36)17-29(23)49-20-48-7)21-8-9-28(44-12-10-43(6)11-13-44)27(14-21)41-31(46)24-18-40-30(45)16-25(24)35(37,38)39/h8-9,14-18H,10-13,19-20H2,1-7H3,(H,40,45)(H,41,46)(H,42,47)	YOZWQAYOZCWKIG-UHFFFAOYSA-N	525585	US11174250, Example 3	WD repeat-containing protein 5				 11.0						US Patent		10.7270/Q2C53Q0K		aid1806103	US11174250	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=525585	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=525585&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			163199820	463789237							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1111007	CN1CCN(CC1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cc(C(N)=O)c(O)cc1F	InChI=1S/C25H23F4N5O4/c1-33-4-6-34(7-5-33)20-3-2-13(14-9-15(23(30)37)21(35)11-18(14)26)8-19(20)32-24(38)16-12-31-22(36)10-17(16)25(27,28)29/h2-3,8-12,35H,4-7H2,1H3,(H2,30,37)(H,31,36)(H,32,38)	CVIREEPRCSCSPK-UHFFFAOYSA-N	525586	US11174250, Example 4	WD repeat-containing protein 5				 86.0						US Patent		10.7270/Q2C53Q0K		aid1806103	US11174250	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=525586	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=525586&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			163199821	463789238							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1111008	CN1CCN(CC1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cc(OC(F)(F)F)ccc1F	InChI=1S/C25H21F7N4O3/c1-35-6-8-36(9-7-35)21-5-2-14(16-11-15(3-4-19(16)26)39-25(30,31)32)10-20(21)34-23(38)17-13-33-22(37)12-18(17)24(27,28)29/h2-5,10-13H,6-9H2,1H3,(H,33,37)(H,34,38)	YKVYRIFLGNVFKL-UHFFFAOYSA-N	525587	US11174250, Example 5	WD repeat-containing protein 5				 29.0						US Patent		10.7270/Q2C53Q0K		aid1806103	US11174250	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=525587	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=525587&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			163199822	463789239							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1111009	CC(C)COc1ccc(F)c(c1)-c1ccc(N2CCN(C)CC2)c(NC(=O)c2c[nH]c(=O)cc2C(F)(F)F)c1	InChI=1S/C28H30F4N4O3/c1-17(2)16-39-19-5-6-23(29)20(13-19)18-4-7-25(36-10-8-35(3)9-11-36)24(12-18)34-27(38)21-15-33-26(37)14-22(21)28(30,31)32/h4-7,12-15,17H,8-11,16H2,1-3H3,(H,33,37)(H,34,38)	ZXGPMNRFVXJEBT-UHFFFAOYSA-N	525588	US11174250, Example 6	WD repeat-containing protein 5				 76.0						US Patent		10.7270/Q2C53Q0K		aid1806103	US11174250	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=525588	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=525588&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			163199823	463789240							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1111011	CN1CCN(CC1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cc(CNC2CCCCC2)ccc1F	InChI=1S/C31H35F4N5O2/c1-39-11-13-40(14-12-39)28-10-8-21(23-15-20(7-9-26(23)32)18-36-22-5-3-2-4-6-22)16-27(28)38-30(42)24-19-37-29(41)17-25(24)31(33,34)35/h7-10,15-17,19,22,36H,2-6,11-14,18H2,1H3,(H,37,41)(H,38,42)	SYLSWCJVGKVJRP-UHFFFAOYSA-N	525589	US11174250, Example 7	WD repeat-containing protein 5				 4.00						US Patent		10.7270/Q2C53Q0K		aid1806103	US11174250	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=525589	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=525589&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			163199824	463789241							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1111013	CN1CCN(CC1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(OC2CCOCC2)nc1F	InChI=1S/C28H29F4N5O4/c1-36-8-10-37(11-9-36)23-4-2-17(19-3-5-25(35-26(19)29)41-18-6-12-40-13-7-18)14-22(23)34-27(39)20-16-33-24(38)15-21(20)28(30,31)32/h2-5,14-16,18H,6-13H2,1H3,(H,33,38)(H,34,39)	BKPFEHCOJLAUMD-UHFFFAOYSA-N	525590	US11174250, Example 8	WD repeat-containing protein 5				 5.00						US Patent		10.7270/Q2C53Q0K		aid1806103	US11174250	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=525590	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=525590&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			163199825	463789242							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1111015	CN1CCN(CC1)c1ccc(cc1NC(=O)c1ccc(=O)[nH]n1)-c1cc(CN2CCOCC2)ccc1F	InChI=1S/C27H31FN6O3/c1-32-8-10-34(11-9-32)25-6-3-20(17-24(25)29-27(36)23-5-7-26(35)31-30-23)21-16-19(2-4-22(21)28)18-33-12-14-37-15-13-33/h2-7,16-17H,8-15,18H2,1H3,(H,29,36)(H,31,35)	XSDWUEUWCFEPKR-UHFFFAOYSA-N	525591	US11174250, Example 9	WD repeat-containing protein 5				 1600						US Patent		10.7270/Q2C53Q0K		aid1806103	US11174250	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=525591	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=525591&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			163199826	463789243							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1111016	COc1cccc(c1)C(=O)Nc1cc(ccc1N1CCN(C)CC1)-c1cc(CN2CCOCC2)ccc1F	InChI=1S/C30H35FN4O3/c1-33-10-12-35(13-11-33)29-9-7-23(20-28(29)32-30(36)24-4-3-5-25(19-24)37-2)26-18-22(6-8-27(26)31)21-34-14-16-38-17-15-34/h3-9,18-20H,10-17,21H2,1-2H3,(H,32,36)	YISLEUASYBXZOU-UHFFFAOYSA-N	525592	US11174250, Example 10	WD repeat-containing protein 5				 1000						US Patent		10.7270/Q2C53Q0K		aid1806103	US11174250	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=525592	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=525592&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138558056	463789244							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1111017	CN1CCN(CC1)c1ccc(cc1NC(=O)c1cc(C)c(F)c(C)c1)-c1cc(CN2CCOCC2)ccc1F	InChI=1S/C31H36F2N4O2/c1-21-16-25(17-22(2)30(21)33)31(38)34-28-19-24(5-7-29(28)37-10-8-35(3)9-11-37)26-18-23(4-6-27(26)32)20-36-12-14-39-15-13-36/h4-7,16-19H,8-15,20H2,1-3H3,(H,34,38)	CRJVRDBFAYGWJT-UHFFFAOYSA-N	525593	US11174250, Example 11	WD repeat-containing protein 5				 6.00						US Patent		10.7270/Q2C53Q0K		aid1806103	US11174250	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=525593	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=525593&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			137376385	463789245							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1111019	CN1CCN(CC1)c1ccc(cc1NC(=O)c1ccc(F)c(C)c1Cl)-c1cc(CN2CCOCC2)ccc1F	InChI=1S/C30H33ClF2N4O2/c1-20-25(32)7-5-23(29(20)31)30(38)34-27-18-22(4-8-28(27)37-11-9-35(2)10-12-37)24-17-21(3-6-26(24)33)19-36-13-15-39-16-14-36/h3-8,17-18H,9-16,19H2,1-2H3,(H,34,38)	GNGFABMWVXAILW-UHFFFAOYSA-N	525594	US11174250, Example 12	WD repeat-containing protein 5				 93.0						US Patent		10.7270/Q2C53Q0K		aid1806103	US11174250	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=525594	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=525594&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			137376624	463789246							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1111020	CN1CCN(CC1)c1ccc(cc1NC(=O)c1cn(C)c(=O)cc1C(F)(F)F)-c1cc(CN2CCOCC2)ccc1F	InChI=1S/C30H33F4N5O3/c1-36-7-9-39(10-8-36)27-6-4-21(22-15-20(3-5-25(22)31)18-38-11-13-42-14-12-38)16-26(27)35-29(41)23-19-37(2)28(40)17-24(23)30(32,33)34/h3-6,15-17,19H,7-14,18H2,1-2H3,(H,35,41)	KYEHLKFNXJSZRC-UHFFFAOYSA-N	525595	US11174250, Example 13	WD repeat-containing protein 5				 15.0						US Patent		10.7270/Q2C53Q0K		aid1806103	US11174250	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=525595	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=525595&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			137376569	463789247							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1111022	COC(=O)c1ccc(F)c(c1)-c1ccc(N2CCN(C)CC2)c(NC(=O)c2c[nH]c(=O)cc2C(F)(F)F)c1	InChI=1S/C26H24F4N4O4/c1-33-7-9-34(10-8-33)22-6-4-15(17-11-16(25(37)38-2)3-5-20(17)27)12-21(22)32-24(36)18-14-31-23(35)13-19(18)26(28,29)30/h3-6,11-14H,7-10H2,1-2H3,(H,31,35)(H,32,36)	NCLMJGKDCMDFOZ-UHFFFAOYSA-N	525596	US11174250, Example 14	WD repeat-containing protein 5				 26.0						US Patent		10.7270/Q2C53Q0K		aid1806103	US11174250	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=525596	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=525596&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			163199827	463789248							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1111023	CN1CCN(CC1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cc(OCC2CC2)ncc1F	InChI=1S/C27H27F4N5O3/c1-35-6-8-36(9-7-35)23-5-4-17(18-11-25(33-14-21(18)28)39-15-16-2-3-16)10-22(23)34-26(38)19-13-32-24(37)12-20(19)27(29,30)31/h4-5,10-14,16H,2-3,6-9,15H2,1H3,(H,32,37)(H,34,38)	MCGJZXZCEBZTRU-UHFFFAOYSA-N	525597	US11174250, Example 15	WD repeat-containing protein 5				 9.00						US Patent		10.7270/Q2C53Q0K		aid1806103	US11174250	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=525597	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=525597&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			163199828	463789249							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1111025	CN1CCN(CC1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(OCC2CC2)nc1F	InChI=1S/C27H27F4N5O3/c1-35-8-10-36(11-9-35)22-6-4-17(18-5-7-24(34-25(18)28)39-15-16-2-3-16)12-21(22)33-26(38)19-14-32-23(37)13-20(19)27(29,30)31/h4-7,12-14,16H,2-3,8-11,15H2,1H3,(H,32,37)(H,33,38)	LRFLJHLBEGFWNW-UHFFFAOYSA-N	525598	US11174250, Example 16	WD repeat-containing protein 5				 10.00						US Patent		10.7270/Q2C53Q0K		aid1806103	US11174250	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=525598	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=525598&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			163199829	463789250							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1111027	CN1CCN(CC1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cc(CNC2CC2)ccc1F	InChI=1S/C28H29F4N5O2/c1-36-8-10-37(11-9-36)25-7-3-18(20-12-17(2-6-23(20)29)15-33-19-4-5-19)13-24(25)35-27(39)21-16-34-26(38)14-22(21)28(30,31)32/h2-3,6-7,12-14,16,19,33H,4-5,8-11,15H2,1H3,(H,34,38)(H,35,39)	HOCSMKQNXKCYNP-UHFFFAOYSA-N	525599	US11174250, Example 17	WD repeat-containing protein 5				 14.0						US Patent		10.7270/Q2C53Q0K		aid1806103	US11174250	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=525599	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=525599&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			163199830	463789251							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1111028	CN1CCN(CC1)c1ccc(cc1NC(=O)c1cc(C)c(F)c(C)c1)-c1cc(CNC2CCCCC2)ccc1F	InChI=1S/C33H40F2N4O/c1-22-17-26(18-23(2)32(22)35)33(40)37-30-20-25(10-12-31(30)39-15-13-38(3)14-16-39)28-19-24(9-11-29(28)34)21-36-27-7-5-4-6-8-27/h9-12,17-20,27,36H,4-8,13-16,21H2,1-3H3,(H,37,40)	VMFLEEZZDJFXSN-UHFFFAOYSA-N	525600	US11174250, Example 18	WD repeat-containing protein 5				 27.0						US Patent		10.7270/Q2C53Q0K		aid1806103	US11174250	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=525600	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=525600&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			137376297	463789252							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1111029	CN1CCN(CC1)c1ccc(cc1NC(=O)c1cc(C)c(F)c(C)c1)-c1ccc(OC2CCOCC2)nc1F	InChI=1S/C30H34F2N4O3/c1-19-16-22(17-20(2)28(19)31)30(37)33-25-18-21(4-6-26(25)36-12-10-35(3)11-13-36)24-5-7-27(34-29(24)32)39-23-8-14-38-15-9-23/h4-7,16-18,23H,8-15H2,1-3H3,(H,33,37)	SELRACPBIBUEEF-UHFFFAOYSA-N	525601	US11174250, Example 19	WD repeat-containing protein 5				 71.0						US Patent		10.7270/Q2C53Q0K		aid1806103	US11174250	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=525601	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=525601&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			137376265	463789253							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1111030	CCOc1cc(c(nn1)C(=O)Nc1cc(ccc1N1CCN(C)CC1)-c1cc(CN2CCOCC2)ccc1F)C(F)(F)F	InChI=1S/C30H34F4N6O3/c1-3-43-27-18-23(30(32,33)34)28(37-36-27)29(41)35-25-17-21(5-7-26(25)40-10-8-38(2)9-11-40)22-16-20(4-6-24(22)31)19-39-12-14-42-15-13-39/h4-7,16-18H,3,8-15,19H2,1-2H3,(H,35,41)	JRYDJOKWCMXIJP-UHFFFAOYSA-N	525602	US11174250, Example 20	WD repeat-containing protein 5				 76.0						US Patent		10.7270/Q2C53Q0K		aid1806103	US11174250	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=525602	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=525602&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			137376333	463789254							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1111031	CN1CCN(CC1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cc(OCC2CC2)c(F)cc1F	InChI=1S/C28H27F5N4O3/c1-36-6-8-37(9-7-36)24-5-4-17(18-11-25(22(30)13-21(18)29)40-15-16-2-3-16)10-23(24)35-27(39)19-14-34-26(38)12-20(19)28(31,32)33/h4-5,10-14,16H,2-3,6-9,15H2,1H3,(H,34,38)(H,35,39)	VXJQBCFPOAUKDT-UHFFFAOYSA-N	525603	US11174250, Example 21	WD repeat-containing protein 5				 19.0						US Patent		10.7270/Q2C53Q0K		aid1806103	US11174250	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=525603	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=525603&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			163199831	463789255							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1111032	CN1CCN(CC1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(nc1F)N1CCCC1	InChI=1S/C27H28F4N6O2/c1-35-10-12-36(13-11-35)22-6-4-17(18-5-7-23(34-25(18)28)37-8-2-3-9-37)14-21(22)33-26(39)19-16-32-24(38)15-20(19)27(29,30)31/h4-7,14-16H,2-3,8-13H2,1H3,(H,32,38)(H,33,39)	BNEXOFUXQOASJO-UHFFFAOYSA-N	525604	US11174250, Example 22	WD repeat-containing protein 5				 17.0						US Patent		10.7270/Q2C53Q0K		aid1806103	US11174250	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=525604	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=525604&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			163199832	463789256							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1111033	CN1CCN(CC1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cccc(CN2CCOCC2)c1F	InChI=1S/C29H31F4N5O3/c1-36-7-9-38(10-8-36)25-6-5-19(21-4-2-3-20(27(21)30)18-37-11-13-41-14-12-37)15-24(25)35-28(40)22-17-34-26(39)16-23(22)29(31,32)33/h2-6,15-17H,7-14,18H2,1H3,(H,34,39)(H,35,40)	GZJGZRQNIYCCKJ-UHFFFAOYSA-N	525605	US11174250, Example 23	WD repeat-containing protein 5				 79.0						US Patent		10.7270/Q2C53Q0K		aid1806103	US11174250	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=525605	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=525605&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			163199833	463789257							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1111034	CN1CCN(CC1)c1ccc(cc1NC(=O)c1cccc(C)c1)-c1cc(CN2CCOCC2)ccc1F	InChI=1S/C30H35FN4O2/c1-22-4-3-5-25(18-22)30(36)32-28-20-24(7-9-29(28)35-12-10-33(2)11-13-35)26-19-23(6-8-27(26)31)21-34-14-16-37-17-15-34/h3-9,18-20H,10-17,21H2,1-2H3,(H,32,36)	XZDAYUHSZSKJGF-UHFFFAOYSA-N	525606	US11174250, Example 24	WD repeat-containing protein 5				 5030						US Patent		10.7270/Q2C53Q0K		aid1806103	US11174250	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=525606	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=525606&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138558045	463789258							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1111035	CN1CCN(CC1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccccc1F	InChI=1S/C24H22F4N4O2/c1-31-8-10-32(11-9-31)21-7-6-15(16-4-2-3-5-19(16)25)12-20(21)30-23(34)17-14-29-22(33)13-18(17)24(26,27)28/h2-7,12-14H,8-11H2,1H3,(H,29,33)(H,30,34)	BZGTYEKCVKLBKA-UHFFFAOYSA-N	525607	US11174250, Example 25	WD repeat-containing protein 5				 102						US Patent		10.7270/Q2C53Q0K		aid1806103	US11174250	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=525607	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=525607&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			163199834	463789259							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1111036	CC1CN(CCN1C)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cc(CN2CCOCC2)ccc1F			525608	US11174250, Example 26	WD repeat-containing protein 5				 9.00						US Patent		10.7270/Q2C53Q0K		aid1806103	US11174250	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=525608	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=525608&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			163199835	463789260							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1111038	C[C@H]1CN(C[C@@H](C)N1C)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cc(CN2CCOCC2)ccc1F			525609	US11174250, Example 27	WD repeat-containing protein 5				 8.00						US Patent		10.7270/Q2C53Q0K		aid1806103	US11174250	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=525609	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=525609&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			163199836	463789261							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1111040	C[C@H]1CN(C)CCN1c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cc(CN2CCOCC2)ccc1F			525610	US11174250, Example 104::US11174250, Example 28	WD repeat-containing protein 5				 4000						US Patent		10.7270/Q2C53Q0K		aid1806103	US11174250	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=525610	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=525610&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			163199837	463789262							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1111041	CN1CCN(CC1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C)-c1cc(CN2CCOCC2)ccc1F	InChI=1S/C29H34FN5O3/c1-20-15-28(36)31-18-24(20)29(37)32-26-17-22(4-6-27(26)35-9-7-33(2)8-10-35)23-16-21(3-5-25(23)30)19-34-11-13-38-14-12-34/h3-6,15-18H,7-14,19H2,1-2H3,(H,31,36)(H,32,37)	VWJOEOAQIKTGBE-UHFFFAOYSA-N	525611	US11174250, Example 29	WD repeat-containing protein 5				 262						US Patent		10.7270/Q2C53Q0K		aid1806103	US11174250	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=525611	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=525611&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			163199838	463789263							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1111043	CN1CCN(CC1)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cc(CN2CCOCC2)ccc1F	InChI=1S/C29H30F5N5O3/c1-37-4-6-39(7-5-37)26-15-24(31)20(19-12-18(2-3-23(19)30)17-38-8-10-42-11-9-38)13-25(26)36-28(41)21-16-35-27(40)14-22(21)29(32,33)34/h2-3,12-16H,4-11,17H2,1H3,(H,35,40)(H,36,41)	JYVWWLIWJLNTAD-UHFFFAOYSA-N	525612	US11174250, Example 30::US11319299, Example 43	WD repeat-containing protein 5				 20.0						US Patent		10.7270/Q2C53Q0K		aid1806103	US11174250	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=525612	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=525612&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			163199839	463789264							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1111045	CN1CCN(CC1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cc(OC2CCOCC2)ncc1F	InChI=1S/C28H29F4N5O4/c1-36-6-8-37(9-7-36)24-3-2-17(19-13-26(34-16-22(19)29)41-18-4-10-40-11-5-18)12-23(24)35-27(39)20-15-33-25(38)14-21(20)28(30,31)32/h2-3,12-16,18H,4-11H2,1H3,(H,33,38)(H,35,39)	ACXYOZFCRYNCTJ-UHFFFAOYSA-N	525613	US11174250, Example 31	WD repeat-containing protein 5				 9.00						US Patent		10.7270/Q2C53Q0K		aid1806103	US11174250	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=525613	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=525613&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			163199840	463789265							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1111047	CN1CCN(CC1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cc(ccc1F)C(=O)NC1CCCCC1	InChI=1S/C31H33F4N5O3/c1-39-11-13-40(14-12-39)27-10-8-19(16-26(27)38-30(43)23-18-36-28(41)17-24(23)31(33,34)35)22-15-20(7-9-25(22)32)29(42)37-21-5-3-2-4-6-21/h7-10,15-18,21H,2-6,11-14H2,1H3,(H,36,41)(H,37,42)(H,38,43)	GLHJOTVYVUCLQO-UHFFFAOYSA-N	525582	US11174250, Example 32::US11174250, Example Table4.4.2	WD repeat-containing protein 5				 6.00						US Patent		10.7270/Q2C53Q0K		aid1806103	US11174250	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=525582	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=525582&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			163199818	463789235							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1111049	CN1CCN(CC1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(CNC2CCCC2)cc1F	InChI=1S/C30H33F4N5O2/c1-38-10-12-39(13-11-38)27-9-7-20(22-8-6-19(14-25(22)31)17-35-21-4-2-3-5-21)15-26(27)37-29(41)23-18-36-28(40)16-24(23)30(32,33)34/h6-9,14-16,18,21,35H,2-5,10-13,17H2,1H3,(H,36,40)(H,37,41)	HEBOREHIASXCQK-UHFFFAOYSA-N	525615	US11174250, Example 33	WD repeat-containing protein 5				 23.0						US Patent		10.7270/Q2C53Q0K		aid1806103	US11174250	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=525615	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=525615&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			163199841	463789266							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1111051	CN1CCN(CC1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(CNC2CCCCC2)cc1F	InChI=1S/C31H35F4N5O2/c1-39-11-13-40(14-12-39)28-10-8-21(23-9-7-20(15-26(23)32)18-36-22-5-3-2-4-6-22)16-27(28)38-30(42)24-19-37-29(41)17-25(24)31(33,34)35/h7-10,15-17,19,22,36H,2-6,11-14,18H2,1H3,(H,37,41)(H,38,42)	BWGYDAIKRMRFTQ-UHFFFAOYSA-N	525616	US11174250, Example 34	WD repeat-containing protein 5				 21.0						US Patent		10.7270/Q2C53Q0K		aid1806103	US11174250	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=525616	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=525616&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			163199842	463789267							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1111053	CN1CCN(CC1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cc(CNC(C)(C)C)ccc1F	InChI=1S/C29H33F4N5O2/c1-28(2,3)35-16-18-5-7-23(30)20(13-18)19-6-8-25(38-11-9-37(4)10-12-38)24(14-19)36-27(40)21-17-34-26(39)15-22(21)29(31,32)33/h5-8,13-15,17,35H,9-12,16H2,1-4H3,(H,34,39)(H,36,40)	KFTPIHQLXRHCSW-UHFFFAOYSA-N	525617	US11174250, Example 35	WD repeat-containing protein 5				 9.00						US Patent		10.7270/Q2C53Q0K		aid1806103	US11174250	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=525617	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=525617&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			163199843	463789268							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1111055	CN1CCN(CC1)c1ccc(cc1NC(=O)c1ccc(F)c(C)c1)-c1cc(CN2CCOCC2)ccc1F	InChI=1S/C30H34F2N4O2/c1-21-17-24(4-7-26(21)31)30(37)33-28-19-23(5-8-29(28)36-11-9-34(2)10-12-36)25-18-22(3-6-27(25)32)20-35-13-15-38-16-14-35/h3-8,17-19H,9-16,20H2,1-2H3,(H,33,37)	KQIMORZBKVLGNE-UHFFFAOYSA-N	525618	US11174250, Example 36	WD repeat-containing protein 5				 4.00						US Patent		10.7270/Q2C53Q0K		aid1806103	US11174250	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=525618	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=525618&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			137376652	463789269							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1111057	CN1CCN(CC1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cc(CNC2CCOCC2)ccc1F	InChI=1S/C30H33F4N5O3/c1-38-8-10-39(11-9-38)27-5-3-20(22-14-19(2-4-25(22)31)17-35-21-6-12-42-13-7-21)15-26(27)37-29(41)23-18-36-28(40)16-24(23)30(32,33)34/h2-5,14-16,18,21,35H,6-13,17H2,1H3,(H,36,40)(H,37,41)	AVUKHGKRUAUGJG-UHFFFAOYSA-N	525619	US11174250, Example 37	WD repeat-containing protein 5				 6.00						US Patent		10.7270/Q2C53Q0K		aid1806103	US11174250	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=525619	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=525619&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			163199844	463789270							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1111059	CN1CCN(CC1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(CN2CCOCC2)cc1F	InChI=1S/C29H31F4N5O3/c1-36-6-8-38(9-7-36)26-5-3-20(21-4-2-19(14-24(21)30)18-37-10-12-41-13-11-37)15-25(26)35-28(40)22-17-34-27(39)16-23(22)29(31,32)33/h2-5,14-17H,6-13,18H2,1H3,(H,34,39)(H,35,40)	RZMHVRYMGMZVQU-UHFFFAOYSA-N	525620	US11174250, Example 38	WD repeat-containing protein 5				 8.00						US Patent		10.7270/Q2C53Q0K		aid1806103	US11174250	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=525620	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=525620&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			163199845	463789271							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1111061	CN1CCN(CC1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccnc(N2CCOCC2)c1F	InChI=1S/C27H28F4N6O3/c1-35-6-8-36(9-7-35)22-3-2-17(18-4-5-32-25(24(18)28)37-10-12-40-13-11-37)14-21(22)34-26(39)19-16-33-23(38)15-20(19)27(29,30)31/h2-5,14-16H,6-13H2,1H3,(H,33,38)(H,34,39)	LPAXCQJMGILCNC-UHFFFAOYSA-N	525621	US11174250, Example 39	WD repeat-containing protein 5				 28.0						US Patent		10.7270/Q2C53Q0K		aid1806103	US11174250	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=525621	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=525621&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			163199846	463789272							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1111063	CN(C)Cc1ccc(F)c(c1)-c1ccc(N2CCN(C)CC2)c(NC(=O)c2c[nH]c(=O)cc2C(F)(F)F)c1	InChI=1S/C27H29F4N5O2/c1-34(2)16-17-4-6-22(28)19(12-17)18-5-7-24(36-10-8-35(3)9-11-36)23(13-18)33-26(38)20-15-32-25(37)14-21(20)27(29,30)31/h4-7,12-15H,8-11,16H2,1-3H3,(H,32,37)(H,33,38)	GXQQAULZONMYCT-UHFFFAOYSA-N	525622	US11174250, Example 40	WD repeat-containing protein 5				 9.00						US Patent		10.7270/Q2C53Q0K		aid1806103	US11174250	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=525622	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=525622&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			163199847	463789273							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1111065	CN1CCN(CC1)c1ccc(cc1NC(=O)c1cc(C)c(F)c(c1)C(F)(F)F)-c1cc(CN2CCOCC2)ccc1F	InChI=1S/C31H33F5N4O2/c1-20-15-23(17-25(29(20)33)31(34,35)36)30(41)37-27-18-22(4-6-28(27)40-9-7-38(2)8-10-40)24-16-21(3-5-26(24)32)19-39-11-13-42-14-12-39/h3-6,15-18H,7-14,19H2,1-2H3,(H,37,41)	BOVKVTDVQGJRCJ-UHFFFAOYSA-N	525623	US11174250, Example 41	WD repeat-containing protein 5				 55.0						US Patent		10.7270/Q2C53Q0K		aid1806103	US11174250	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=525623	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=525623&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			137376698	463789274							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1111067	CN1CCN(CC1)c1ccc(cc1NC(=O)c1cnc(OCC[Si](C)(C)C)cc1C(F)(F)F)-c1cc(CNC2CCC(F)(F)CC2)ccc1F	InChI=1S/C36H45F6N5O2Si/c1-46-13-15-47(16-14-46)32-8-6-25(27-19-24(5-7-30(27)37)22-43-26-9-11-35(38,39)12-10-26)20-31(32)45-34(48)28-23-44-33(21-29(28)36(40,41)42)49-17-18-50(2,3)4/h5-8,19-21,23,26,43H,9-18,22H2,1-4H3,(H,45,48)	HGPCPTVSTUVIQI-UHFFFAOYSA-N	525624	US11174250, Example 42	WD repeat-containing protein 5				 5.00						US Patent		10.7270/Q2C53Q0K		aid1806103	US11174250	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=525624	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=525624&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			141655775	463789275							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1111069	CN(Cc1ccc(F)c(c1)-c1ccc(N2CCN(C)CC2)c(NC(=O)c2c[nH]c(=O)cc2C(F)(F)F)c1)C1COC1	InChI=1S/C29H31F4N5O3/c1-36-7-9-38(10-8-36)26-6-4-19(21-11-18(3-5-24(21)30)15-37(2)20-16-41-17-20)12-25(26)35-28(40)22-14-34-27(39)13-23(22)29(31,32)33/h3-6,11-14,20H,7-10,15-17H2,1-2H3,(H,34,39)(H,35,40)	RZGVKGLIYMLVJM-UHFFFAOYSA-N	525625	US11174250, Example 43	WD repeat-containing protein 5				 7.00						US Patent		10.7270/Q2C53Q0K		aid1806103	US11174250	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=525625	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=525625&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			163199848	463789276							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1111071	CN1CCN(CC1)c1ccc(cc1NC(=O)c1ccc(O)cc1C(F)(F)F)-c1cc(CN2CCOCC2)ccc1F	InChI=1S/C30H32F4N4O3/c1-36-8-10-38(11-9-36)28-7-3-21(24-16-20(2-6-26(24)31)19-37-12-14-41-15-13-37)17-27(28)35-29(40)23-5-4-22(39)18-25(23)30(32,33)34/h2-7,16-18,39H,8-15,19H2,1H3,(H,35,40)	GDXSDWNVMRVNLW-UHFFFAOYSA-N	525626	US11174250, Example 44	WD repeat-containing protein 5				 69.0						US Patent		10.7270/Q2C53Q0K		aid1806103	US11174250	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=525626	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=525626&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			137376359	463789277							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1111073	C[C@H]1CN(C[C@@H](C)N1C)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cc(CNC2CCCCC2)ccc1F			525627	US11174250, Example 45	WD repeat-containing protein 5				 2.00						US Patent		10.7270/Q2C53Q0K		aid1806103	US11174250	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=525627	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=525627&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			163199849	463789278							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1111075	C[C@H]1CN(C[C@@H](C)N1C)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cc(ccc1F)C(=O)NC1CCCCC1			525628	US11174250, Example 46	WD repeat-containing protein 5				 0.950						US Patent		10.7270/Q2C53Q0K		aid1806103	US11174250	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=525628	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=525628&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			163199850	463789279							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1111077	C[C@H]1CN(C[C@@H](C)N1C)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cc(ccc1F)C(=O)N1CCOCC1			525629	US11174250, Example 47	WD repeat-containing protein 5				 8.00						US Patent		10.7270/Q2C53Q0K		aid1806103	US11174250	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=525629	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=525629&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			163199851	463789280							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1111079	CN1CCN(CC1)c1ccc(cc1NC(=O)c1cc(O)cc(F)c1F)-c1cc(CN2CCOCC2)ccc1F	InChI=1S/C29H31F3N4O3/c1-34-6-8-36(9-7-34)27-5-3-20(15-26(27)33-29(38)23-16-21(37)17-25(31)28(23)32)22-14-19(2-4-24(22)30)18-35-10-12-39-13-11-35/h2-5,14-17,37H,6-13,18H2,1H3,(H,33,38)	LDZZELJKEFFULJ-UHFFFAOYSA-N	525630	US11174250, Example 48	WD repeat-containing protein 5				 93.0						US Patent		10.7270/Q2C53Q0K		aid1806103	US11174250	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=525630	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=525630&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			137376704	463789281							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1111081	CN1CCN(CC1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)F)-c1cc(CN2CCOCC2)ccc1F	InChI=1S/C29H32F3N5O3/c1-35-6-8-37(9-7-35)26-5-3-20(21-14-19(2-4-24(21)30)18-36-10-12-40-13-11-36)15-25(26)34-29(39)23-17-33-27(38)16-22(23)28(31)32/h2-5,14-17,28H,6-13,18H2,1H3,(H,33,38)(H,34,39)	SNSKIDONUPQTCE-UHFFFAOYSA-N	525631	US11174250, Example 49	WD repeat-containing protein 5				 7.00						US Patent		10.7270/Q2C53Q0K		aid1806103	US11174250	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=525631	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=525631&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			163199852	463789282							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1111083	C[C@H]1CN(C[C@@H](C)N1C)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cc(OCC2CC2)ncc1F			525632	US11174250, Example 50	WD repeat-containing protein 5				 4.00						US Patent		10.7270/Q2C53Q0K		aid1806103	US11174250	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=525632	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=525632&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			163199853	463789283							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1111085	COc1cc(c(cn1)C(=O)Nc1cc(ccc1N1CCN(C)CC1)-c1cc(C=O)ccc1F)C(F)(F)F	InChI=1S/C26H24F4N4O3/c1-33-7-9-34(10-8-33)23-6-4-17(18-11-16(15-35)3-5-21(18)27)12-22(23)32-25(36)19-14-31-24(37-2)13-20(19)26(28,29)30/h3-6,11-15H,7-10H2,1-2H3,(H,32,36)	JGDUXPQQVSSJAG-UHFFFAOYSA-N	525633	US11174250, Example 51	WD repeat-containing protein 5				>200						US Patent		10.7270/Q2C53Q0K		aid1806103	US11174250	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=525633	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=525633&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			137376356	463789284							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1111086	COc1cc(c(cn1)C(=O)Nc1cc(ccc1N1CCN(C)CC1)-c1cc(CN2CCC(CC2)N2CCOCC2)ccc1F)C(F)(F)F	InChI=1S/C35H42F4N6O3/c1-42-11-13-45(14-12-42)32-6-4-25(20-31(32)41-34(46)28-22-40-33(47-2)21-29(28)35(37,38)39)27-19-24(3-5-30(27)36)23-43-9-7-26(8-10-43)44-15-17-48-18-16-44/h3-6,19-22,26H,7-18,23H2,1-2H3,(H,41,46)	LSYNGTFUYRULPD-UHFFFAOYSA-N	525634	US11174250, Example 52	WD repeat-containing protein 5				>200						US Patent		10.7270/Q2C53Q0K		aid1806103	US11174250	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=525634	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=525634&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			137376354	463789285							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1111087	COc1cc(c(cn1)C(=O)Nc1cc(ccc1N1CCN(C)CC1)-c1cc(CN2CC[C@H](C2)C(C)C)ccc1F)C(F)(F)F	InChI=1S/C33H39F4N5O2/c1-21(2)24-9-10-41(20-24)19-22-5-7-28(34)25(15-22)23-6-8-30(42-13-11-40(3)12-14-42)29(16-23)39-32(43)26-18-38-31(44-4)17-27(26)33(35,36)37/h5-8,15-18,21,24H,9-14,19-20H2,1-4H3,(H,39,43)/t24-/m1/s1	OMVDNRLZCSQGNL-XMMPIXPASA-N	525635	US11174250, Example 53	WD repeat-containing protein 5				>200						US Patent		10.7270/Q2C53Q0K		aid1806103	US11174250	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=525635	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=525635&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			137376301	463789286							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1111088	COc1cc(c(cn1)C(=O)Nc1cc(ccc1N1CCN(C)CC1)-c1cc(CN2CCN(CC2)C(C)=O)ccc1F)C(F)(F)F	InChI=1S/C32H36F4N6O3/c1-21(43)41-14-10-40(11-15-41)20-22-4-6-27(33)24(16-22)23-5-7-29(42-12-8-39(2)9-13-42)28(17-23)38-31(44)25-19-37-30(45-3)18-26(25)32(34,35)36/h4-7,16-19H,8-15,20H2,1-3H3,(H,38,44)	MLAYYWSYGKSRBO-UHFFFAOYSA-N	525636	US11174250, Example 54	WD repeat-containing protein 5				>200						US Patent		10.7270/Q2C53Q0K		aid1806103	US11174250	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=525636	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=525636&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			137376288	463789287							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1111089	COc1cc(c(cn1)C(=O)Nc1cc(ccc1N1CCN(C)CC1)-c1cc(CN2CCC(F)CC2)ccc1F)C(F)(F)F	InChI=1S/C31H34F5N5O2/c1-39-11-13-41(14-12-39)28-6-4-21(23-15-20(3-5-26(23)33)19-40-9-7-22(32)8-10-40)16-27(28)38-30(42)24-18-37-29(43-2)17-25(24)31(34,35)36/h3-6,15-18,22H,7-14,19H2,1-2H3,(H,38,42)	OZSFVNHGPLWHND-UHFFFAOYSA-N	525637	US11174250, Example 55	WD repeat-containing protein 5				>200						US Patent		10.7270/Q2C53Q0K		aid1806103	US11174250	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=525637	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=525637&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			137376289	463789288							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1111090	COc1cc(c(cn1)C(=O)Nc1cc(ccc1N1CCN(C)CC1)-c1cc(CN2C3CC2COC3)ccc1F)C(F)(F)F	InChI=1S/C31H33F4N5O3/c1-38-7-9-39(10-8-38)28-6-4-20(23-11-19(3-5-26(23)32)16-40-21-13-22(40)18-43-17-21)12-27(28)37-30(41)24-15-36-29(42-2)14-25(24)31(33,34)35/h3-6,11-12,14-15,21-22H,7-10,13,16-18H2,1-2H3,(H,37,41)	KWJLATYORDQAOJ-UHFFFAOYSA-N	525638	US11174250, Example 56	WD repeat-containing protein 5				>200						US Patent		10.7270/Q2C53Q0K		aid1806103	US11174250	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=525638	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=525638&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			137376318	463789289							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1111091	COc1cc(c(cn1)C(=O)Nc1cc(ccc1N1CCN(C)CC1)-c1cc(CN2CCC(C2)S(C)(=O)=O)ccc1F)C(F)(F)F	InChI=1S/C31H35F4N5O4S/c1-38-10-12-40(13-11-38)28-7-5-21(15-27(28)37-30(41)24-17-36-29(44-2)16-25(24)31(33,34)35)23-14-20(4-6-26(23)32)18-39-9-8-22(19-39)45(3,42)43/h4-7,14-17,22H,8-13,18-19H2,1-3H3,(H,37,41)	RZQVYLYINRBCQA-UHFFFAOYSA-N	525639	US11174250, Example 57	WD repeat-containing protein 5				>200						US Patent		10.7270/Q2C53Q0K		aid1806103	US11174250	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=525639	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=525639&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138558101	463789290							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1111092	COc1cc(c(cn1)C(=O)Nc1cc(ccc1N1CCN(C)CC1)-c1cc(CN(C)[C@H]2CCOC2)ccc1F)C(F)(F)F	InChI=1S/C31H35F4N5O3/c1-38-9-11-40(12-10-38)28-7-5-21(23-14-20(4-6-26(23)32)18-39(2)22-8-13-43-19-22)15-27(28)37-30(41)24-17-36-29(42-3)16-25(24)31(33,34)35/h4-7,14-17,22H,8-13,18-19H2,1-3H3,(H,37,41)/t22-/m0/s1	QHDOOYLHJSZHCX-QFIPXVFZSA-N	525640	US11174250, Example 58	WD repeat-containing protein 5				>200						US Patent		10.7270/Q2C53Q0K		aid1806103	US11174250	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=525640	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=525640&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			137376440	463789291							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1111093	COc1cc(c(cn1)C(=O)Nc1cc(ccc1N1CCN(C)CC1)-c1cc(CN2CCOC(C)(C)C2)ccc1F)C(F)(F)F	InChI=1S/C32H37F4N5O3/c1-31(2)20-40(13-14-44-31)19-21-5-7-26(33)23(15-21)22-6-8-28(41-11-9-39(3)10-12-41)27(16-22)38-30(42)24-18-37-29(43-4)17-25(24)32(34,35)36/h5-8,15-18H,9-14,19-20H2,1-4H3,(H,38,42)	BJMLVUKERJEGKD-UHFFFAOYSA-N	525641	US11174250, Example 59	WD repeat-containing protein 5				>200						US Patent		10.7270/Q2C53Q0K		aid1806103	US11174250	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=525641	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=525641&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			137376366	463789292							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1111094	C[C@H]1CN(C[C@@H](C)N1C)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cc(CN2CCOCC2)cnc1F			525642	US11174250, Example 60	WD repeat-containing protein 5				 7.00						US Patent		10.7270/Q2C53Q0K		aid1806103	US11174250	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=525642	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=525642&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			163199854	463789293							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1111096	CN1CCN(CC1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cc(CN2CCOCC2)cnc1F	InChI=1S/C28H30F4N6O3/c1-36-4-6-38(7-5-36)24-3-2-19(20-12-18(15-34-26(20)29)17-37-8-10-41-11-9-37)13-23(24)35-27(40)21-16-33-25(39)14-22(21)28(30,31)32/h2-3,12-16H,4-11,17H2,1H3,(H,33,39)(H,35,40)	FZVHYHVJNVOCCK-UHFFFAOYSA-N	525643	US11174250, Example 61	WD repeat-containing protein 5				 7.00						US Patent		10.7270/Q2C53Q0K		aid1806103	US11174250	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=525643	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=525643&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			163199855	463789294							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1111098	CCN1CCN(CC1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cc(CN2CCOCC2)ccc1F	InChI=1S/C30H33F4N5O3/c1-2-37-7-9-39(10-8-37)27-6-4-21(22-15-20(3-5-25(22)31)19-38-11-13-42-14-12-38)16-26(27)36-29(41)23-18-35-28(40)17-24(23)30(32,33)34/h3-6,15-18H,2,7-14,19H2,1H3,(H,35,40)(H,36,41)	BEWURZMFMJZRIA-UHFFFAOYSA-N	525644	US11174250, Example 62	WD repeat-containing protein 5				>200						US Patent		10.7270/Q2C53Q0K		aid1806103	US11174250	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=525644	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=525644&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			163199856	463789295							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1111100	CCN1CCN(CC1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cc(CNC2CCCCC2)ccc1F	InChI=1S/C32H37F4N5O2/c1-2-40-12-14-41(15-13-40)29-11-9-22(24-16-21(8-10-27(24)33)19-37-23-6-4-3-5-7-23)17-28(29)39-31(43)25-20-38-30(42)18-26(25)32(34,35)36/h8-11,16-18,20,23,37H,2-7,12-15,19H2,1H3,(H,38,42)(H,39,43)	CGMHUMFZWIFNAO-UHFFFAOYSA-N	525645	US11174250, Example 63	WD repeat-containing protein 5				>200						US Patent		10.7270/Q2C53Q0K		aid1806103	US11174250	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=525645	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=525645&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			163199857	463789296							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1111102	CN1CCN(CC1COC(=O)C(C)(C)C)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cc(CN2CCOCC2)ccc1F			525646	US11174250, Example 64	WD repeat-containing protein 5				 102						US Patent		10.7270/Q2C53Q0K		aid1806103	US11174250	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=525646	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=525646&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138558072	463789297							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1111103	CN1CCN(CC1CO)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cc(CN2CCOCC2)ccc1F			525647	US11174250, Example 65	WD repeat-containing protein 5				 9.40						US Patent		10.7270/Q2C53Q0K		aid1806103	US11174250	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=525647	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=525647&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			163199858	463789298							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1111105	CN1CCN(CC1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cc(CN2CCN(CC3CC3)CC2)ccc1F	InChI=1S/C33H38F4N6O2/c1-40-8-14-43(15-9-40)30-7-5-24(17-29(30)39-32(45)26-19-38-31(44)18-27(26)33(35,36)37)25-16-23(4-6-28(25)34)21-42-12-10-41(11-13-42)20-22-2-3-22/h4-7,16-19,22H,2-3,8-15,20-21H2,1H3,(H,38,44)(H,39,45)	UCIMUGNNMDZMDT-UHFFFAOYSA-N	525648	US11174250, Example 66	WD repeat-containing protein 5				 7.20						US Patent		10.7270/Q2C53Q0K		aid1806103	US11174250	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=525648	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=525648&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			163199859	463789299							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1111107	CN(Cc1ccc(F)c(c1)-c1ccc(N2CCN(C)CC2)c(NC(=O)c2c[nH]c(=O)cc2C(F)(F)F)c1)C1CCCCC1	InChI=1S/C32H37F4N5O2/c1-39-12-14-41(15-13-39)29-11-9-22(17-28(29)38-31(43)25-19-37-30(42)18-26(25)32(34,35)36)24-16-21(8-10-27(24)33)20-40(2)23-6-4-3-5-7-23/h8-11,16-19,23H,3-7,12-15,20H2,1-2H3,(H,37,42)(H,38,43)	KZGBALJQZBEHNW-UHFFFAOYSA-N	525649	US11174250, Example 67	WD repeat-containing protein 5				 3.20						US Patent		10.7270/Q2C53Q0K		aid1806103	US11174250	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=525649	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=525649&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			163199860	463789300							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1111109	CN1CCN(CC1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cc(CN2CCN(Cc3ccc(F)cc3)CC2)ccc1F	InChI=1S/C36H37F5N6O2/c1-44-10-16-47(17-11-44)33-9-5-26(19-32(33)43-35(49)29-21-42-34(48)20-30(29)36(39,40)41)28-18-25(4-8-31(28)38)23-46-14-12-45(13-15-46)22-24-2-6-27(37)7-3-24/h2-9,18-21H,10-17,22-23H2,1H3,(H,42,48)(H,43,49)	MSVYPKVNSDNBMD-UHFFFAOYSA-N	525650	US11174250, Example 68	WD repeat-containing protein 5				 7.70						US Patent		10.7270/Q2C53Q0K		aid1806103	US11174250	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=525650	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=525650&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			163199861	463789301							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1111111	CN1CCN(CC1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cc(CN2CC[C@@H](O)C2)ccc1F			525651	US11174250, Example 69	WD repeat-containing protein 5				 5.40						US Patent		10.7270/Q2C53Q0K		aid1806103	US11174250	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=525651	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=525651&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			163199862	463789302							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1111113	CN1CCN(CC1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cc(CN2CCC(CC2)N2CCOCC2)ccc1F	InChI=1S/C34H40F4N6O3/c1-41-10-12-44(13-11-41)31-5-3-24(19-30(31)40-33(46)27-21-39-32(45)20-28(27)34(36,37)38)26-18-23(2-4-29(26)35)22-42-8-6-25(7-9-42)43-14-16-47-17-15-43/h2-5,18-21,25H,6-17,22H2,1H3,(H,39,45)(H,40,46)	ZXQPWVCTBWBJLE-UHFFFAOYSA-N	525652	US11174250, Example 70	WD repeat-containing protein 5				 4.40						US Patent		10.7270/Q2C53Q0K		aid1806103	US11174250	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=525652	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=525652&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			163199863	463789303							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1111115	CN(C)[C@@H]1CCN(Cc2ccc(F)c(c2)-c2ccc(N3CCN(C)CC3)c(NC(=O)c3c[nH]c(=O)cc3C(F)(F)F)c2)C1			525653	US11174250, Example 71	WD repeat-containing protein 5				 4.80						US Patent		10.7270/Q2C53Q0K		aid1806103	US11174250	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=525653	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=525653&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			163199864	463789304							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1111117	CN1CCN(CC1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cc(CN2CCNCC2)ccc1F	InChI=1S/C29H32F4N6O2/c1-37-10-12-39(13-11-37)26-5-3-20(21-14-19(2-4-24(21)30)18-38-8-6-34-7-9-38)15-25(26)36-28(41)22-17-35-27(40)16-23(22)29(31,32)33/h2-5,14-17,34H,6-13,18H2,1H3,(H,35,40)(H,36,41)	RDIJFNQKWLWKCS-UHFFFAOYSA-N	525654	US11174250, Example 72	WD repeat-containing protein 5				 5.10						US Patent		10.7270/Q2C53Q0K		aid1806103	US11174250	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=525654	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=525654&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			163199865	463789305							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1111119	CN1CCN(CC1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cc(CN2CCC(F)CC2)ccc1F	InChI=1S/C30H32F5N5O2/c1-38-10-12-40(13-11-38)27-5-3-20(22-14-19(2-4-25(22)32)18-39-8-6-21(31)7-9-39)15-26(27)37-29(42)23-17-36-28(41)16-24(23)30(33,34)35/h2-5,14-17,21H,6-13,18H2,1H3,(H,36,41)(H,37,42)	LCHGERIHAPDZCU-UHFFFAOYSA-N	525578	US11174250, Example 73::US11174250, Example Table4.2.2	WD repeat-containing protein 5				 4.20						US Patent		10.7270/Q2C53Q0K		aid1806103	US11174250	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=525578	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=525578&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			163199815	463789232							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1111121	CN1CCN(CC1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cc(CN2C3CC2COC3)ccc1F			525656	US11174250, Example 74	WD repeat-containing protein 5				 4.80						US Patent		10.7270/Q2C53Q0K		aid1806103	US11174250	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=525656	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=525656&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			163199866	463789306							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1111123	CN1CCN(CC1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cc(CN2CC[C@H](C2)S(C)(=O)=O)ccc1F			525657	US11174250, Example 75	WD repeat-containing protein 5				 5.90						US Patent		10.7270/Q2C53Q0K		aid1806103	US11174250	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=525657	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=525657&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			163199867	463789307							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1111125	CN(Cc1ccc(F)c(c1)-c1ccc(N2CCN(C)CC2)c(NC(=O)c2c[nH]c(=O)cc2C(F)(F)F)c1)[C@H]1CCOC1			525658	US11174250, Example 76	WD repeat-containing protein 5				 5.50						US Patent		10.7270/Q2C53Q0K		aid1806103	US11174250	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=525658	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=525658&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			163199868	463789308							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1111127	CN1CCN(CC1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cc(CN2CCOC(C)(C)C2)ccc1F	InChI=1S/C31H35F4N5O3/c1-30(2)19-39(12-13-43-30)18-20-4-6-25(32)22(14-20)21-5-7-27(40-10-8-38(3)9-11-40)26(15-21)37-29(42)23-17-36-28(41)16-24(23)31(33,34)35/h4-7,14-17H,8-13,18-19H2,1-3H3,(H,36,41)(H,37,42)	XXBPCORNASWFLI-UHFFFAOYSA-N	525659	US11174250, Example 77	WD repeat-containing protein 5				 4.50						US Patent		10.7270/Q2C53Q0K		aid1806103	US11174250	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=525659	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=525659&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			163199869	463789309							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1111129	C[C@H]1CN(C[C@@H](C)N1C)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1c(F)ccc(C#N)c1F			525660	US11174250, Example 78	WD repeat-containing protein 5				 39.0						US Patent		10.7270/Q2C53Q0K		aid1806103	US11174250	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=525660	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=525660&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			163199870	463789310							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1111130	C[C@H]1CN(C[C@@H](C)N1C)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cc(CNC2CCCCC2)c(F)cc1F			525661	US11174250, Example 79	WD repeat-containing protein 5				 2.50						US Patent		10.7270/Q2C53Q0K		aid1806103	US11174250	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=525661	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=525661&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			163199871	463789311							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1111131	CN1CCN(CC1=O)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cc(ccc1F)C(=O)NC1CCCCC1	InChI=1S/C31H31F4N5O4/c1-39-11-12-40(17-28(39)42)26-10-8-18(14-25(26)38-30(44)22-16-36-27(41)15-23(22)31(33,34)35)21-13-19(7-9-24(21)32)29(43)37-20-5-3-2-4-6-20/h7-10,13-16,20H,2-6,11-12,17H2,1H3,(H,36,41)(H,37,43)(H,38,44)	AJEAVPDKUNNESV-UHFFFAOYSA-N	525662	US11174250, Example 80	WD repeat-containing protein 5				 14.0						US Patent		10.7270/Q2C53Q0K		aid1806103	US11174250	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=525662	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=525662&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			163199872	463789312							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1111133	CC1CN(CCN1C)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cc(ccc1F)C(=O)NC1CCCCC1			525663	US11174250, Example 81	WD repeat-containing protein 5				 17.5						US Patent		10.7270/Q2C53Q0K		aid1806103	US11174250	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=525663	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=525663&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			163199873	463789313							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1111135	C[C@H]1CN(C[C@@H](C)N1C)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(OCC2CC2)nc1F			525664	US11174250, Example 82	WD repeat-containing protein 5				 0.700						US Patent		10.7270/Q2C53Q0K		aid1806103	US11174250	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=525664	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=525664&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			163199874	463789314							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1111137	C[C@H]1CN(C[C@@H](C)N1C)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(F)c(CNC2CCCCC2)c1F			525665	US11174250, Example 83	WD repeat-containing protein 5				 10.3						US Patent		10.7270/Q2C53Q0K		aid1806103	US11174250	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=525665	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=525665&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			163199875	463789315							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1111138	CN1CCN(CC1)c1ncc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cc(CN2CCOCC2)ccc1F	InChI=1S/C28H30F4N6O3/c1-36-4-6-38(7-5-36)26-24(35-27(40)21-16-33-25(39)14-22(21)28(30,31)32)13-19(15-34-26)20-12-18(2-3-23(20)29)17-37-8-10-41-11-9-37/h2-3,12-16H,4-11,17H2,1H3,(H,33,39)(H,35,40)	UOZGJWWPIWCEJI-UHFFFAOYSA-N	525666	US11174250, Example 84	WD repeat-containing protein 5				 22.0						US Patent		10.7270/Q2C53Q0K		aid1806103	US11174250	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=525666	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=525666&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			163199876	463789316							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1111140	CN1CCN(CC1)c1ncc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cc(CNC2CCCCC2)ccc1F	InChI=1S/C30H34F4N6O2/c1-39-9-11-40(12-10-39)28-26(38-29(42)23-18-36-27(41)15-24(23)30(32,33)34)14-20(17-37-28)22-13-19(7-8-25(22)31)16-35-21-5-3-2-4-6-21/h7-8,13-15,17-18,21,35H,2-6,9-12,16H2,1H3,(H,36,41)(H,38,42)	KMZWIGDLQWYHNE-UHFFFAOYSA-N	525667	US11174250, Example 85	WD repeat-containing protein 5				 14.8						US Patent		10.7270/Q2C53Q0K		aid1806103	US11174250	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=525667	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=525667&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			163199877	463789317							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1111141	CN1CCN(CC1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cc(CN2CCOCC2)ccc1Cl	InChI=1S/C29H31ClF3N5O3/c1-36-6-8-38(9-7-36)26-5-3-20(21-14-19(2-4-24(21)30)18-37-10-12-41-13-11-37)15-25(26)35-28(40)22-17-34-27(39)16-23(22)29(31,32)33/h2-5,14-17H,6-13,18H2,1H3,(H,34,39)(H,35,40)	FOAUMOZOTVHACR-UHFFFAOYSA-N	525579	US11174250, Example 86::US11174250, Example Table4.3.1	WD repeat-containing protein 5				 34.5						US Patent		10.7270/Q2C53Q0K		aid1806103	US11174250	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=525579	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=525579&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			163199816	463789233							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1111142	CN(C)C1CCN(C1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cc(CN2CCOCC2)ccc1F			525669	US11174250, Example 87	WD repeat-containing protein 5				 12.0						US Patent		10.7270/Q2C53Q0K		aid1806103	US11174250	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=525669	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=525669&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			163199878	463789318							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1111144	CN1CCCN(CC1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cc(CN2CCOCC2)ccc1F	InChI=1S/C30H33F4N5O3/c1-37-7-2-8-39(10-9-37)27-6-4-21(22-15-20(3-5-25(22)31)19-38-11-13-42-14-12-38)16-26(27)36-29(41)23-18-35-28(40)17-24(23)30(32,33)34/h3-6,15-18H,2,7-14,19H2,1H3,(H,35,40)(H,36,41)	HUNQCTSTGWMXHS-UHFFFAOYSA-N	525670	US11174250, Example 88	WD repeat-containing protein 5				 18.0						US Patent		10.7270/Q2C53Q0K		aid1806103	US11174250	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=525670	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=525670&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			163199879	463789319							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1111145	CN1CCCN(CC1)c1ccc(cc1NC(=O)c1cn(C)c(=O)cc1C(F)(F)F)-c1cc(CN2CCOCC2)ccc1F	InChI=1S/C31H35F4N5O3/c1-37-8-3-9-40(11-10-37)28-7-5-22(23-16-21(4-6-26(23)32)19-39-12-14-43-15-13-39)17-27(28)36-30(42)24-20-38(2)29(41)18-25(24)31(33,34)35/h4-7,16-18,20H,3,8-15,19H2,1-2H3,(H,36,42)	XYQKOKXWCZHAJW-UHFFFAOYSA-N	525671	US11174250, Example 89	WD repeat-containing protein 5				 235						US Patent		10.7270/Q2C53Q0K		aid1806103	US11174250	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=525671	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=525671&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			137377325	463789320							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1111146	CNC(=O)c1ccc(F)c(c1)-c1ccc(N2C[C@H](C)N(C)[C@H](C)C2)c(NC(=O)c2c[nH]c(=O)cc2C(F)(F)F)c1			525672	US11174250, Example 90	WD repeat-containing protein 5				 6.40						US Patent		10.7270/Q2C53Q0K		aid1806103	US11174250	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=525672	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=525672&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			163199880	463789321							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1111148	CN(C)C1CCN(C1)c1ccc(cc1NC(=O)c1cc(C)c(F)c(C)c1)-c1cc(CN2CCOCC2)ccc1F	InChI=1S/C32H38F2N4O2/c1-21-15-25(16-22(2)31(21)34)32(39)35-29-18-24(6-8-30(29)38-10-9-26(20-38)36(3)4)27-17-23(5-7-28(27)33)19-37-11-13-40-14-12-37/h5-8,15-18,26H,9-14,19-20H2,1-4H3,(H,35,39)	SMKWFQLMCHIGQB-UHFFFAOYSA-N	525673	US11174250, Example 91	WD repeat-containing protein 5				 316						US Patent		10.7270/Q2C53Q0K		aid1806103	US11174250	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=525673	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=525673&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138558107	463789322							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1111149	CN1CCCN(CC1)c1ccc(cc1NC(=O)c1cc(C)c(F)c(C)c1)-c1cc(CN2CCOCC2)ccc1F	InChI=1S/C32H38F2N4O2/c1-22-17-26(18-23(2)31(22)34)32(39)35-29-20-25(6-8-30(29)38-10-4-9-36(3)11-12-38)27-19-24(5-7-28(27)33)21-37-13-15-40-16-14-37/h5-8,17-20H,4,9-16,21H2,1-3H3,(H,35,39)	GHKWSNRRDKKPLQ-UHFFFAOYSA-N	525674	US11174250, Example 92	WD repeat-containing protein 5				 394						US Patent		10.7270/Q2C53Q0K		aid1806103	US11174250	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=525674	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=525674&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			137376507	463789323							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1111150	C[C@H]1CN(C[C@@H](C)N1C)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cc(ccc1F)C(=O)NC1CC1			525675	US11174250, Example 93	WD repeat-containing protein 5				 3.00						US Patent		10.7270/Q2C53Q0K		aid1806103	US11174250	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=525675	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=525675&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			163199881	463789324							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1111152	CN1CC2CN(CC2C1)c1ccc(cc1NC(=O)c1cc(C)c(F)c(C)c1)-c1cc(CN2CCOCC2)ccc1F	InChI=1S/C33H38F2N4O2/c1-21-12-25(13-22(2)32(21)35)33(40)36-30-15-24(5-7-31(30)39-19-26-17-37(3)18-27(26)20-39)28-14-23(4-6-29(28)34)16-38-8-10-41-11-9-38/h4-7,12-15,26-27H,8-11,16-20H2,1-3H3,(H,36,40)	FPFQFUXPTOREAD-UHFFFAOYSA-N	525676	US11174250, Example 94	WD repeat-containing protein 5				>200						US Patent		10.7270/Q2C53Q0K		aid1806103	US11174250	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=525676	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=525676&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138558079	463789325							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1111153	Cc1cc(cc(C)c1F)C(=O)Nc1cc(ccc1N1CCN(CC(F)(F)F)CC1)-c1cc(CN2CCOCC2)ccc1F	InChI=1S/C32H35F5N4O2/c1-21-15-25(16-22(2)30(21)34)31(42)38-28-18-24(4-6-29(28)41-9-7-40(8-10-41)20-32(35,36)37)26-17-23(3-5-27(26)33)19-39-11-13-43-14-12-39/h3-6,15-18H,7-14,19-20H2,1-2H3,(H,38,42)	DHCLLDQUEBPRCB-UHFFFAOYSA-N	525677	US11174250, Example 95	WD repeat-containing protein 5				>200						US Patent		10.7270/Q2C53Q0K		aid1806103	US11174250	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=525677	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=525677&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			137376420	463789326							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1111154	C[C@H]1CN(CCN1C)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ncccc1F			525678	US11174250, Example 96	WD repeat-containing protein 5				 3.00						US Patent		10.7270/Q2C53Q0K		aid1806103	US11174250	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=525678	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=525678&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			137376461	463789327							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1111156	Fc1ccc(CN2CCOCC2)cc1-c1ccc(N2CCN(CC(F)(F)F)CC2)c(NC(=O)c2c[nH]c(=O)cc2C(F)(F)F)c1	InChI=1S/C30H30F7N5O3/c31-24-3-1-19(17-40-9-11-45-12-10-40)13-21(24)20-2-4-26(42-7-5-41(6-8-42)18-29(32,33)34)25(14-20)39-28(44)22-16-38-27(43)15-23(22)30(35,36)37/h1-4,13-16H,5-12,17-18H2,(H,38,43)(H,39,44)	VUXNDTHYMVUCTO-UHFFFAOYSA-N	525679	US11174250, Example 97	WD repeat-containing protein 5				>200						US Patent		10.7270/Q2C53Q0K		aid1806103	US11174250	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=525679	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=525679&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			163199882	463789328							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1111157	CN1CCN(CC1)c1c(F)cc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cc(CN2CCOCC2)ccc1F	InChI=1S/C29H30F5N5O3/c1-37-4-6-39(7-5-37)27-24(31)13-19(20-12-18(2-3-23(20)30)17-38-8-10-42-11-9-38)14-25(27)36-28(41)21-16-35-26(40)15-22(21)29(32,33)34/h2-3,12-16H,4-11,17H2,1H3,(H,35,40)(H,36,41)	FNMIGKXNLZEIGZ-UHFFFAOYSA-N	525680	US11174250, Example 98	WD repeat-containing protein 5				 17.0						US Patent		10.7270/Q2C53Q0K		aid1806103	US11174250	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=525680	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=525680&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			163199883	463789329							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1111159	CN1CCN(CC1)c1ccc(c(F)c1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cc(CN2CCOCC2)ccc1F	InChI=1S/C29H30F5N5O3/c1-37-6-8-39(9-7-37)24-5-3-19(20-14-18(2-4-23(20)30)17-38-10-12-42-13-11-38)26(31)27(24)36-28(41)21-16-35-25(40)15-22(21)29(32,33)34/h2-5,14-16H,6-13,17H2,1H3,(H,35,40)(H,36,41)	PEHSNIFVIAESBC-UHFFFAOYSA-N	525681	US11174250, Example 99	WD repeat-containing protein 5				 14.0						US Patent		10.7270/Q2C53Q0K		aid1806103	US11174250	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=525681	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=525681&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			163199884	463789330							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1111161	CN1CC2CN(CC2C1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cc(CN2CCOCC2)ccc1F			525682	US11174250, Example 100	WD repeat-containing protein 5				 5930						US Patent		10.7270/Q2C53Q0K		aid1806103	US11174250	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=525682	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=525682&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			163199885	463789331							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1111162	CN(C)C1CCN(C1)c1ccc(cc1NC(=O)c1cn(C)c(=O)cc1C(F)(F)F)-c1cc(CN2CCOCC2)ccc1F	InChI=1S/C31H35F4N5O3/c1-37(2)22-8-9-40(18-22)28-7-5-21(23-14-20(4-6-26(23)32)17-39-10-12-43-13-11-39)15-27(28)36-30(42)24-19-38(3)29(41)16-25(24)31(33,34)35/h4-7,14-16,19,22H,8-13,17-18H2,1-3H3,(H,36,42)	YKWQWMBSYUCMLT-UHFFFAOYSA-N	525683	US11174250, Example 101	WD repeat-containing protein 5				 2274						US Patent		10.7270/Q2C53Q0K		aid1806103	US11174250	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=525683	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=525683&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			137376764	463789332							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1111163	CN1CCN(CC1)c1ccc(cc1NC(=O)c1cc(F)cc2[nH]cnc12)-c1cc(CN2CCOCC2)ccc1F	InChI=1S/C30H32F2N6O2/c1-36-6-8-38(9-7-36)28-5-3-21(23-14-20(2-4-25(23)32)18-37-10-12-40-13-11-37)15-26(28)35-30(39)24-16-22(31)17-27-29(24)34-19-33-27/h2-5,14-17,19H,6-13,18H2,1H3,(H,33,34)(H,35,39)	ZONWONWYQRHXFI-UHFFFAOYSA-N	525684	US11174250, Example 102	WD repeat-containing protein 5				>200						US Patent		10.7270/Q2C53Q0K		aid1806103	US11174250	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=525684	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=525684&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			137376400	463789333							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1111164	CN1CCN(CC1)c1ccc(cc1NC(=O)c1nc2ccccc2[nH]1)-c1cc(CN2CCOCC2)ccc1F	InChI=1S/C30H33FN6O2/c1-35-10-12-37(13-11-35)28-9-7-22(23-18-21(6-8-24(23)31)20-36-14-16-39-17-15-36)19-27(28)34-30(38)29-32-25-4-2-3-5-26(25)33-29/h2-9,18-19H,10-17,20H2,1H3,(H,32,33)(H,34,38)	IVRANXJUYMIUKO-UHFFFAOYSA-N	525685	US11174250, Example 103	WD repeat-containing protein 5				>200						US Patent		10.7270/Q2C53Q0K		aid1806103	US11174250	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=525685	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=525685&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138558106	463789334							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1111165	C[C@H]1CN(C)CCN1c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cc(CN2CCOCC2)ccc1F			525610	US11174250, Example 104::US11174250, Example 28	WD repeat-containing protein 5				 4000						US Patent		10.7270/Q2C53Q0K		aid1806103	US11174250	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=525610	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=525610&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			163199837	463789262							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1111166	CN1CCN(CC1)c1ccc(cc1NC(=O)c1ccc(=O)[nH]c1)-c1cc(CN2CCOCC2)ccc1F	InChI=1S/C28H32FN5O3/c1-32-8-10-34(11-9-32)26-6-3-21(17-25(26)31-28(36)22-4-7-27(35)30-18-22)23-16-20(2-5-24(23)29)19-33-12-14-37-15-13-33/h2-7,16-18H,8-15,19H2,1H3,(H,30,35)(H,31,36)	UMGLYFUYPLXUEU-UHFFFAOYSA-N	525687	US11174250, Example 105	WD repeat-containing protein 5				 1950						US Patent		10.7270/Q2C53Q0K		aid1806103	US11174250	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=525687	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=525687&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			163199886	463789335							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1111167	CN1CCN(CC1)c1ccc(cc1NC(=O)c1cnc(NC(C)=O)cc1C)-c1cc(CN2CCOCC2)ccc1F	InChI=1S/C31H37FN6O3/c1-21-16-30(34-22(2)39)33-19-26(21)31(40)35-28-18-24(5-7-29(28)38-10-8-36(3)9-11-38)25-17-23(4-6-27(25)32)20-37-12-14-41-15-13-37/h4-7,16-19H,8-15,20H2,1-3H3,(H,35,40)(H,33,34,39)	FSZYZDCGGYNVDQ-UHFFFAOYSA-N	525688	US11174250, Example 106	WD repeat-containing protein 5				 829						US Patent		10.7270/Q2C53Q0K		aid1806103	US11174250	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=525688	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=525688&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			137376745	463789336							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1111168	COc1cc(c(cn1)C(=O)Nc1cc(ccc1N1CCN(C)CC1)-c1cc(CN2CCN(CC3CC3)CC2)ccc1F)C(F)(F)F	InChI=1S/C34H40F4N6O2/c1-41-9-15-44(16-10-41)31-8-6-25(18-30(31)40-33(45)27-20-39-32(46-2)19-28(27)34(36,37)38)26-17-24(5-7-29(26)35)22-43-13-11-42(12-14-43)21-23-3-4-23/h5-8,17-20,23H,3-4,9-16,21-22H2,1-2H3,(H,40,45)	HHZIAOCNJDXBOK-UHFFFAOYSA-N	525689	US11174250, Example 107	WD repeat-containing protein 5				>200						US Patent		10.7270/Q2C53Q0K		aid1806103	US11174250	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=525689	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=525689&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			137376466	463789337							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1111169	CNc1cc(c(cn1)C(=O)Nc1cc(ccc1N1CCN(C)CC1)-c1cc(CN2CCOCC2)ccc1F)C(F)(F)F	InChI=1S/C30H34F4N6O2/c1-35-28-17-24(30(32,33)34)23(18-36-28)29(41)37-26-16-21(4-6-27(26)40-9-7-38(2)8-10-40)22-15-20(3-5-25(22)31)19-39-11-13-42-14-12-39/h3-6,15-18H,7-14,19H2,1-2H3,(H,35,36)(H,37,41)	AKPOZBSWTYUTFS-UHFFFAOYSA-N	525690	US11174250, Example 108	WD repeat-containing protein 5				>200						US Patent		10.7270/Q2C53Q0K		aid1806103	US11174250	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=525690	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=525690&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			137377548	463789338							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1111170	CN1CCN(CC1)c1ccc(cc1NC(=O)c1cnc(N)cc1C(F)(F)F)-c1cc(CN2CCOCC2)ccc1F	InChI=1S/C29H32F4N6O2/c1-37-6-8-39(9-7-37)26-5-3-20(21-14-19(2-4-24(21)30)18-38-10-12-41-13-11-38)15-25(26)36-28(40)22-17-35-27(34)16-23(22)29(31,32)33/h2-5,14-17H,6-13,18H2,1H3,(H2,34,35)(H,36,40)	NHGMXRRRHPDJNK-UHFFFAOYSA-N	525691	US11174250, Example 109	WD repeat-containing protein 5				>200						US Patent		10.7270/Q2C53Q0K		aid1806103	US11174250	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=525691	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=525691&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			137376399	463789339							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1111171	CN(C1CCCCC1)C(=O)c1ccc(F)c(c1)-c1ccc(N2CCN(C)CC2)c(NC(=O)c2c[nH]c(=O)cc2C(F)(F)F)c1	InChI=1S/C32H35F4N5O3/c1-39-12-14-41(15-13-39)28-11-9-20(17-27(28)38-30(43)24-19-37-29(42)18-25(24)32(34,35)36)23-16-21(8-10-26(23)33)31(44)40(2)22-6-4-3-5-7-22/h8-11,16-19,22H,3-7,12-15H2,1-2H3,(H,37,42)(H,38,43)	LSSYDYCCKSSRBW-UHFFFAOYSA-N	525692	US11174250, Example 110	WD repeat-containing protein 5				 4.00						US Patent		10.7270/Q2C53Q0K		aid1806103	US11174250	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=525692	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=525692&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			163199887	463789340							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1111173	C[C@H]1CN(C[C@@H](C)N1C)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cc(ccc1F)C(=O)N(C)C1CCCCC1			525693	US11174250, Example 111	WD repeat-containing protein 5				 24.0						US Patent		10.7270/Q2C53Q0K		aid1806103	US11174250	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=525693	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=525693&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			163199888	463789341							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1111175	C[C@H]1CN(C[C@@H](C)N1C)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(F)c(CN(C)C2COC2)c1F			525694	US11174250, Example 112	WD repeat-containing protein 5				 23.0						US Patent		10.7270/Q2C53Q0K		aid1806103	US11174250	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=525694	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=525694&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			163199889	463789342							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1111176	C[C@H]1CN(C[C@@H](C)N1C)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cc(CN(C)C2COC2)c(F)cc1F			525695	US11174250, Example 113	WD repeat-containing protein 5				 8.00						US Patent		10.7270/Q2C53Q0K		aid1806103	US11174250	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=525695	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=525695&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			163199890	463789343							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1111178	C[C@H]1CN(C[C@@H](C)N1C)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1c(F)ccc(CNC2CCCCC2)c1F			525696	US11174250, Example 114	WD repeat-containing protein 5				 13.0						US Patent		10.7270/Q2C53Q0K		aid1806103	US11174250	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=525696	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=525696&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			163199891	463789344							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1111180	C[C@H]1CN(C[C@@H](C)N1C)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1c(F)cc(CNC2CCCCC2)cc1F			525697	US11174250, Example 115	WD repeat-containing protein 5				 55.0						US Patent		10.7270/Q2C53Q0K		aid1806103	US11174250	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=525697	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=525697&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			163199892	463789345							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1111181	CN1CCN(CC1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cc(ccc1Cl)C(=O)NC1CCCCC1	InChI=1S/C31H33ClF3N5O3/c1-39-11-13-40(14-12-39)27-10-8-19(16-26(27)38-30(43)23-18-36-28(41)17-24(23)31(33,34)35)22-15-20(7-9-25(22)32)29(42)37-21-5-3-2-4-6-21/h7-10,15-18,21H,2-6,11-14H2,1H3,(H,36,41)(H,37,42)(H,38,43)	QYUSSNJDVILCJQ-UHFFFAOYSA-N	525581	US11174250, Example 116::US11174250, Example Table4.4.1	WD repeat-containing protein 5				 13.0						US Patent		10.7270/Q2C53Q0K		aid1806103	US11174250	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=525581	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=525581&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			163199817	463789234							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1111183	C[C@H]1CN(C[C@@H](C)N1C)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(cc1F)C(N)=O			525699	US11174250, Example 117	WD repeat-containing protein 5				 1.60						US Patent		10.7270/Q2C53Q0K		aid1806103	US11174250	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=525699	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=525699&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138558083	463789346							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1111184	C[C@H]1CN(C[C@@H](C)N1C)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(cc1F)N1CCOCC1			525700	US11174250, Example 118	WD repeat-containing protein 5				 6.00						US Patent		10.7270/Q2C53Q0K		aid1806103	US11174250	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=525700	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=525700&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138558068	463789347							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1111185	C[C@H]1CN(C[C@@H](C)N1C)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cc(ccc1F)C(N)=O			525701	US11174250, Example 119	WD repeat-containing protein 5				 4.00						US Patent		10.7270/Q2C53Q0K		aid1806103	US11174250	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=525701	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=525701&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			163199893	463789348							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1111186	C[C@H]1CN(C[C@@H](C)N1C)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cc(C(=O)NC(C)(C)CC(C)(C)C)c(F)cc1F			525702	US11174250, Example 120	WD repeat-containing protein 5				 6.00						US Patent		10.7270/Q2C53Q0K		aid1806103	US11174250	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=525702	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=525702&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			137376362	463789349							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1111187	C[C@H]1CN(C[C@@H](C)N1C)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cc(C(N)=O)c(F)cc1F			525703	US11174250, Example 121	WD repeat-containing protein 5				 9.00						US Patent		10.7270/Q2C53Q0K		aid1806103	US11174250	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=525703	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=525703&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			163199894	463789350							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1111188	C[C@H]1CN(C[C@@H](C)N1C)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(C(=O)NC(C)(C)CC(C)(C)C)c(F)c1F			525704	US11174250, Example 122	WD repeat-containing protein 5				 8.00						US Patent		10.7270/Q2C53Q0K		aid1806103	US11174250	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=525704	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=525704&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			163199895	463789351							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1111189	C[C@H]1CN(C[C@@H](C)N1C)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(C(N)=O)c(F)c1F			525705	US11174250, Example 123	WD repeat-containing protein 5				 4.00						US Patent		10.7270/Q2C53Q0K		aid1806103	US11174250	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=525705	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=525705&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			163199896	463789352							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1111190	CC1CN(CC(C)N1C)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cc(ccc1F)C(=O)NC1CCCCC1			525706	US11174250, Example 124	WD repeat-containing protein 5				 1.70						US Patent		10.7270/Q2C53Q0K		aid1806103	US11174250	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=525706	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=525706&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			163199897	463789353							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1111192	C[C@H]1CN(C[C@@H](C)N1C)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1nc(ncc1F)N1CCOCC1			525707	US11174250, Example 125	WD repeat-containing protein 5				 3.10						US Patent		10.7270/Q2C53Q0K		aid1806103	US11174250	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=525707	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=525707&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			137376401	463789354							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167143	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCN(C1)c1ncc(CN2CCOCC2)cn1			553383	N-[4-fluoro-5-[1-[5- (morpholin-4- ylmethyl)pyrimidin-2-yl]- 2,5-dihydropyrrol-3-yl]- 2-[rac-(3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 458	WD repeat-containing protein 5				 0.474						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553383	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553383&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608091	469797248							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167144	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCN(C1)c1ncc(CN2CCN(C)CC2)cn1			553384	N-[4-fluoro-5-[1-[5-[(4- methylpiperazin-1- yl)methyl]pyrimidin-2- yl]-2,5-dihydropyrrol-3- yl]-2-[rac-(3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 459	WD repeat-containing protein 5				 0.392						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553384	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553384&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608092	469797249							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167145	C[C@@H]1CN(CCO1)c1ncc(cn1)-c1cc(NC(=O)c2cn(C)c(=O)cc2C(F)F)c(cc1F)N1CCN(C)[C@@H](C)C1	InChI=1S/C29H34F3N7O3/c1-17-14-38(6-5-36(17)3)25-11-23(30)20(19-12-33-29(34-13-19)39-7-8-42-18(2)15-39)9-24(25)35-28(41)22-16-37(4)26(40)10-21(22)27(31)32/h9-13,16-18,27H,5-8,14-15H2,1-4H3,(H,35,41)/t17-,18+/m0/s1	YVMPDRKPFAFZNO-ZWKOTPCHSA-N	553385	4-(difluoromethyl)-N-[4- fluoro-2-[rac-(3S)-3,4- dimethylpiperazin-1-yl]- 5-[2-[rac-(2R)-2- methylmorpholin-4- yl]pyrimidin-5- yl]phenyl]-1-methyl-6- oxopyridine-3- carboxamide::US11319299, Example 460	WD repeat-containing protein 5				 3.43						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553385	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553385&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			137376736	469797250							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167146	C[C@@H]1CN(CCO1)c1ncc(cn1)-c1cc(NC(=O)c2cn(C)c(=O)cc2C(F)F)c(cc1F)N1C[C@H](C)N(C)[C@H](C)C1	InChI=1S/C30H36F3N7O3/c1-17-13-40(14-18(2)38(17)5)26-10-24(31)21(20-11-34-30(35-12-20)39-6-7-43-19(3)15-39)8-25(26)36-29(42)23-16-37(4)27(41)9-22(23)28(32)33/h8-12,16-19,28H,6-7,13-15H2,1-5H3,(H,36,42)/t17-,18+,19-/m1/s1	OCXIOXDNHHZKMM-CEXWTWQISA-N	553386	4-(difluoromethyl)-N-[4- fluoro-5-[2-[rac-(2R)-2- methylmorpholin-4- yl]pyrimidin-5-yl]-2-[rac- (3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-1-methyl-6- oxopyridine-3-carboxamide::US11319299, Example 461	WD repeat-containing protein 5				 4.93						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553386	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553386&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			137377251	469797251							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167147	C[C@H]1CN(C[C@@H](C)O1)c1ncc(cn1)-c1cc(NC(=O)c2cn(C)c(=O)cc2C(F)F)c(cc1F)N1C[C@H](C)N(C)[C@H](C)C1	InChI=1S/C31H38F3N7O3/c1-17-12-40(13-18(2)39(17)6)27-9-25(32)22(21-10-35-31(36-11-21)41-14-19(3)44-20(4)15-41)7-26(27)37-30(43)24-16-38(5)28(42)8-23(24)29(33)34/h7-11,16-20,29H,12-15H2,1-6H3,(H,37,43)/t17-,18+,19-,20+	UPMSAXBMORZPKO-FGYAAKKASA-N	553387	4-(difluoromethyl)-N-[4- fluoro-5-[2-[rac-(2R,6S)- 2,6-dimethylmorpholin-4- yl]pyrimidin-5-yl]-2-[rac- (3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-1-methyl-6- oxopyridine-3-carboxamide::US11319299, Example 462	WD repeat-containing protein 5				 3.70						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553387	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553387&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138541778	469797252							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167148	Fc1cc(N2C[C@@H]3CCN[C@@H]3C2)c(NC(=O)c2c[nH]c(=O)cc2C(F)(F)F)cc1-c1cnc(nc1)N1CCOCC1			553388	N-[4-fluoro-5-(2- morpholin-4-ylpyrimidin- 5-yl)-2-[rac-(3aR,6aR)- 2,3,3a,4,6,6a-hexahydro- 1H-pyrrolo[2,3-c]pyrrol- 5-yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 463	WD repeat-containing protein 5				 168						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553388	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553388&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608093	469797253							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167149	C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1cn(C)c(=O)cc1C(F)(F)F)-c1cnc(nc1)N1CCNCC1	InChI=1S/C28H32F4N8O2/c1-17-15-40(9-8-37(17)2)24-12-22(29)19(18-13-34-27(35-14-18)39-6-4-33-5-7-39)10-23(24)36-26(42)20-16-38(3)25(41)11-21(20)28(30,31)32/h10-14,16-17,33H,4-9,15H2,1-3H3,(H,36,42)/t17-/m0/s1	HNFLATTUKOKKPM-KRWDZBQOSA-N	553389	N-[4-fluoro-5-(2- piperazin-1-ylpyrimidin- 5-yl)-2-[rac-(3R)-3,4- dimethylpiperazin-1- yl]phenyl]-1-methyl-6- oxo-4-(trifluoromethyl)pyridine- 3-carboxamide::US11319299, Example 464	WD repeat-containing protein 5				 2.21						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553389	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553389&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138551480	469797254							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167150	CC(C)N1CCN(CC1)c1ncc(cn1)-c1cc(NC(=O)c2ccc(F)cc2C(F)(F)F)c(cc1F)N1CCN(C)[C@@H](C)C1	InChI=1S/C31H36F5N7O/c1-19(2)41-9-11-42(12-10-41)30-37-16-21(17-38-30)24-14-27(28(15-26(24)33)43-8-7-40(4)20(3)18-43)39-29(44)23-6-5-22(32)13-25(23)31(34,35)36/h5-6,13-17,19-20H,7-12,18H2,1-4H3,(H,39,44)/t20-/m0/s1	RWLKJZIFMVGSSG-FQEVSTJZSA-N	553390	4-fluoro-N-[4-fluoro-5-[2- (4-propan-2-ylpiperazin-1- yl)pyrimidin-5-yl]-2-[rac- (3R)-3,4-dimethylpiperazin-1- yl]phenyl]-2-(trifluoromethyl) benzamide::US11319299, Example 465	WD repeat-containing protein 5				 1.77						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553390	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553390&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138551335	469797255							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167151	CC(C)N1CCN(CC1)c1ncc(cn1)-c1cc(NC(=O)c2ccc(F)cc2C(F)(F)F)c(cc1F)N1C[C@H](C)N(C)[C@H](C)C1	InChI=1S/C32H38F5N7O/c1-19(2)42-8-10-43(11-9-42)31-38-15-22(16-39-31)25-13-28(29(14-27(25)34)44-17-20(3)41(5)21(4)18-44)40-30(45)24-7-6-23(33)12-26(24)32(35,36)37/h6-7,12-16,19-21H,8-11,17-18H2,1-5H3,(H,40,45)/t20-,21+	RCUDLUQSPHPFBA-OYRHEFFESA-N	553391	4-fluoro-N-[4-fluoro-5- [2-(4-propan-2- ylpiperazin-1- yl)pyrimidin-5-yl]-2-[rac- (3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-2- (trifluoromethyl)benzamide::US11319299, Example 466	WD repeat-containing protein 5				 2.28						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553391	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553391&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			137376735	469797256							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167152	CC(C)N1CCN(CC1)c1ncc(cn1)-c1cc(NC(=O)c2cn(C)c(=O)cc2C(F)(F)F)c(cc1F)N1CCN(C)[C@@H](C)C1	InChI=1S/C31H38F4N8O2/c1-19(2)41-8-10-42(11-9-41)30-36-15-21(16-37-30)22-12-26(27(14-25(22)32)43-7-6-39(4)20(3)17-43)38-29(45)23-18-40(5)28(44)13-24(23)31(33,34)35/h12-16,18-20H,6-11,17H2,1-5H3,(H,38,45)/t20-/m0/s1	PNNXHDIJLRCCHS-FQEVSTJZSA-N	553392	N-[4-fluoro-5-[2-(4- propan-2-ylpiperazin-1- yl)pyrimidin-5-yl]-2-[rac- (3R)-3,4-dimethylpiperazin-1- yl]phenyl]-1-methyl-6- oxo-4-(trifluoromethyl) pyridine-3-carboxamide::US11319299, Example 467	WD repeat-containing protein 5				 2.54						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553392	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553392&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138551582	469797257							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167153	C[C@@H]1COCCN1c1ncc(cn1)-c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)(F)F)c(cc1F)N1CCN(C)[C@@H](C)C1			553393	N-[4-fluoro-2-[rac-(3S)- 3,4-dimethylpiperazin-1- yl]-5-[2-[rac-(3R)-3- methylmorpholin-4-yl] pyrimidin-5-yl]phenyl]-6- oxo-4-(trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 468	WD repeat-containing protein 5				 2.28						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553393	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553393&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608094	469797258							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167154	C[C@@H]1COCCN1c1ncc(cn1)-c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)(F)F)c(cc1F)N1C[C@H](C)N(C)[C@H](C)C1			553394	N-[4-fluoro-5-[2-[rac- (3R)-3-methylmorpholin- 4-yl]pyrimidin-5-yl]-2- [rac-(3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 469	WD repeat-containing protein 5				 5.64						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553394	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553394&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608095	469797259							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167155	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCN(CC1)C(=O)OC1(C)CCC1			553395	(1-methylcyclobutyl) 4- [2-fluoro-5-[[6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carbonyl]amino]- 4-[rac-(3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-3,6-dihydro- 2H-pyridine-1-carboxylate::US11319299, Example 470	WD repeat-containing protein 5				 4.27						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553395	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553395&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608096	469797260							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167156	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCCN(C1)C(=O)OC1(C)CCC1			553396	(1-methylcyclobutyl) 5- [2-fluoro-5-[[6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carbonyl]amino]- 4-[rac-(3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-3,6-dihydro- 2H-pyridine-1-carboxylate::US11319299, Example 471	WD repeat-containing protein 5				 0.494						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553396	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553396&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608097	469797261							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167157	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCN(C1)C(=O)OC1(C)CCC1			553397	(1-methylcyclobutyl) 3- [2-fluoro-5-[[6-oxo-4- (trifluoromethyl)-1H- pyridine-3- carbonyl]amino]-4-[rac- (3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-2,5- dihydropyrrole-1- carboxylate::US11319299, Example 472	WD repeat-containing protein 5				 0.407						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553397	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553397&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608098	469797262							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167158	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cccc(n1)N1CCOCC1			553398	N-[4-fluoro-5-(6- morpholin-4-ylpyridin-2- yl)-2-[rac-(3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 473	WD repeat-containing protein 5				 0.533						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553398	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553398&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608099	469797263							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167159	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cncc(n1)N1CCOCC1			553399	N-[4-fluoro-5-(6- morpholin-4-ylpyrazin-2- yl)-2-[rac-(3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 474	WD repeat-containing protein 5				 1.20						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553399	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553399&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608100	469797264							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167160	C[C@H]1COCCN1c1ncc(cn1)-c1cc(NC(=O)c2cn(C)c(=O)cc2C(F)F)c(cc1F)N1C[C@H](C)N(C)[C@H](C)C1	InChI=1S/C30H36F3N7O3/c1-17-13-39(14-18(2)38(17)5)26-10-24(31)21(20-11-34-30(35-12-20)40-6-7-43-16-19(40)3)8-25(26)36-29(42)23-15-37(4)27(41)9-22(23)28(32)33/h8-12,15,17-19,28H,6-7,13-14,16H2,1-5H3,(H,36,42)/t17-,18+,19-/m0/s1	ARRGSKGNSFDJAS-OTWHNJEPSA-N	553400	4-(difluoromethyl)-N-[4- fluoro-5-[2-[rac-(3R)-3- methylmorpholin-4- yl]pyrimidin-5-yl]-2-[rac- (3S,5R)-3,4,5- trimethylpiperazin-1- yl]phenyl]-1-methyl-6- oxopyridine-3-carboxamide::US11319299, Example 475	WD repeat-containing protein 5				 3.52						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553400	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553400&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138551482	469797265							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167161	CCCN1CC[C@H]2CN(C[C@@H]12)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cnc(nc1)N1CCOCC1			553401	N-[4-fluoro-5-(2- morpholin-4-ylpyrimidin- 5-yl)-2-[rac-(3aR,6aR)-1- propyl-2,3,3a,4,6,6a- hexahydropyrrolo[2,3-c] pyrrol-5-yl]phenyl]-6- oxo-4-(trifluoromethyl)- 1H-pyridine-3-carboxamide::US11319299, Example 476	WD repeat-containing protein 5				 9.71						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553401	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553401&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608101	469797266							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167162	CN1CC[C@H]2CN(C[C@@H]12)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cnc(nc1)N1CCOCC1			553402	N-[4-fluoro-5-(2- morpholin-4-ylpyrimidin- 5-yl)-2-[rac-(3aR,6aR)-1- methyl-2,3,3a,4,6,6a- hexahydropyrrolo[2,3-c] pyrrol-5-yl]phenyl]-6- oxo-4-(trifluoromethyl)- 1H-pyridine-3-carboxamide::US11319299, Example 477	WD repeat-containing protein 5				 24.2						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553402	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553402&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608102	469797267							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167163	C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1cn(C)c(=O)cc1C(F)F)-c1ccc(N2CCOCC2)c(F)c1	InChI=1S/C30H33F4N5O3/c1-18-16-39(7-6-36(18)2)27-15-23(31)20(19-4-5-26(24(32)12-19)38-8-10-42-11-9-38)13-25(27)35-30(41)22-17-37(3)28(40)14-21(22)29(33)34/h4-5,12-15,17-18,29H,6-11,16H2,1-3H3,(H,35,41)/t18-/m0/s1	DIBDVTPTCCSFFI-SFHVURJKSA-N	553403	4-(difluoromethyl)-N-[4- fluoro-5-(3-fluoro-4- morpholin-4-ylphenyl)-2- [rac-(3R)-3,4-dimethylpiperazin- 1-yl]phenyl]-1-methyl-6- oxopyridine-3-carboxamide::US11319299, Example 478	WD repeat-containing protein 5				 5.32						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553403	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553403&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138542047	469797268							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167164	C[C@H]1CN(CC[N+]1(C)C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cnc(nc1)N1CCOCC1			553404	N-[4-fluoro-5-(2- morpholin-4-ylpyrimidin- 5-yl)-2-[rac-(3R,5S)- 3,4,4,5-tetramethylpiperazin-4- ium-1-yl]phenyl]-6-oxo- 4-(trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 479	WD repeat-containing protein 5				 3.54						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553404	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553404&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608103	469797269							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167165	C[C@H]1CN(CCO1)c1ncc(cn1)-c1cc(NC(=O)c2cn(C)c(=O)cc2C(F)F)c(cc1F)N1CCN(C)[C@@H](C)C1	InChI=1S/C29H34F3N7O3/c1-17-14-38(6-5-36(17)3)25-11-23(30)20(19-12-33-29(34-13-19)39-7-8-42-18(2)15-39)9-24(25)35-28(41)22-16-37(4)26(40)10-21(22)27(31)32/h9-13,16-18,27H,5-8,14-15H2,1-4H3,(H,35,41)/t17-,18-/m0/s1	YVMPDRKPFAFZNO-ROUUACIJSA-N	553405	4-(difluoromethyl)-N-[4- fluoro-2-[rac-(3R)-3,4- dimethylpiperazin-1-yl)- 5-[2-[rac-(2R)-2- methylmorpholin-4- yl]pyrimidin-5- yl]phenyl]-1-methyl-6- oxopyridine-3-carboxamide::US11319299, Example 480::US11319299, Example 481	WD repeat-containing protein 5				 2.15						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553405	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553405&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138551497	469797270							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167166	C[C@H]1CN(CCO1)c1ncc(cn1)-c1cc(NC(=O)c2cn(C)c(=O)cc2C(F)F)c(cc1F)N1CCN(C)[C@@H](C)C1	InChI=1S/C29H34F3N7O3/c1-17-14-38(6-5-36(17)3)25-11-23(30)20(19-12-33-29(34-13-19)39-7-8-42-18(2)15-39)9-24(25)35-28(41)22-16-37(4)26(40)10-21(22)27(31)32/h9-13,16-18,27H,5-8,14-15H2,1-4H3,(H,35,41)/t17-,18-/m0/s1	YVMPDRKPFAFZNO-ROUUACIJSA-N	553405	4-(difluoromethyl)-N-[4- fluoro-2-[rac-(3R)-3,4- dimethylpiperazin-1-yl)- 5-[2-[rac-(2R)-2- methylmorpholin-4- yl]pyrimidin-5- yl]phenyl]-1-methyl-6- oxopyridine-3-carboxamide::US11319299, Example 480::US11319299, Example 481	WD repeat-containing protein 5				 4.89						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553405	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553405&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138551497	469797270							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167167	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1nc(cs1)C(=O)NCC1CC1			553407	N-(cyclopropylmethyl)-2- [2-fluoro-5-[[6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carbonyl] amino]-4-[rac-(3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-1,3-thiazole-4- carboxamide::US11319299, Example 482	WD repeat-containing protein 5				 1.75						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553407	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553407&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608104	469797271							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167168	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1nc(cs1)C(=O)N(C)CC1CC1			553408	N-(cyclopropylmethyl)-2- [2-fluoro-5-[[6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carbonyl] amino]-4-[rac-(3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-N-methyl-1,3- thiazole-4-carboxamide::US11319299, Example 483	WD repeat-containing protein 5				 3.97						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553408	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553408&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608105	469797272							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167169	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1nc(cs1)C(=O)NC1CCCCC1			553409	N-cyclohexyl-2-[2- fluoro-5-[[6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carbonyl] amino]-4-[rac- (3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-1,3-thiazole-4- carboxamide::US11319299, Example 484	WD repeat-containing protein 5				 3.07						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553409	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553409&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608106	469797273							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167170	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1nc(cs1)C(=O)N(C)C1CCCCC1			553410	N-cyclohexyl-2-[2- fluoro-5-[[6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carbonyl] amino]-4-[rac-(3R,5S)- 3,4,5-trimethylpiperazin-1- yl]phenyl]-N-methyl-1,3- thiazole-4-carboxamide::US11319299, Example 485	WD repeat-containing protein 5				 2.21						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553410	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553410&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608107	469797274							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167171	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1nc(cs1)C(=O)N1CCOCC1			553411	N-[4-fluoro-5-[4- (morpholine-4-carbonyl)- 1,3-thiazol-2-yl]-2-[rac- (3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 486	WD repeat-containing protein 5				 2.44						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553411	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553411&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608108	469797275							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167172	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1nc(cs1)C(=O)N1CCN(C)CC1			553412	N-[4-fluoro-5-[4-(4- methylpiperazine-1- carbonyl)-1,3-thiazol-2- yl]-2-[rac-(3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 487	WD repeat-containing protein 5				 2.81						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553412	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553412&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608109	469797276							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167173	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCN(CC1)C(=O)OC1(C)COC1			553413	(3-methyloxetan-3-yl) 4- [2-fluoro-5-[[6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carbonyl]amino]- 4-[rac-(3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-3,6-dihydro- 2H-pyridine-1-carboxylate::US11319299, Example 488	WD repeat-containing protein 5				 4.87						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553413	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553413&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608110	469797277							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167174	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCCN(C1)C(=O)OC1(C)COC1			553414	(3-methyloxetan-3-yl) 5- [2-fluoro-5-[[6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carbonyl]amino]- 4-[rac-(3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-3,6-dihydro- 2H-pyridine-1-carboxylate::US11319299, Example 489	WD repeat-containing protein 5				 2.74						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553414	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553414&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608111	469797278							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167175	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCN(C1)C(=O)OC1(C)COC1			553415	(3-methyloxetan-3-yl) 3- [2-fluoro-5-[[6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carbonyl]amino]- 4-[rac-(3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-2,5- dihydropyrrole-1-carboxylate::US11319299, Example 490	WD repeat-containing protein 5				 3.24						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553415	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553415&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608112	469797279							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167176	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(CN2CCOCC2)s1			553416	N-[4-fluoro-5-[5- (morpholin-4-ylmethyl) thiophen-2-yl]-2-[rac- (3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 491	WD repeat-containing protein 5				 3.59						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553416	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553416&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608113	469797280							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167177	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cccs1			553417	N-[4-fluoro-2-[rac- (3R,5S)-3,4,5- trimethylpiperazin-1-yl]- 5-thiophen-2-ylphenyl]-6- oxo-4-(trifluoromethyl)- 1H-pyridine-3-carboxamide::US11319299, Example 492	WD repeat-containing protein 5				 3.35						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553417	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553417&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608114	469797281							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167178	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccsc1			553418	N-[4-fluoro-2-[rac- (3R,5S)-3,4,5- trimethylpiperazin-1-yl]- 5-thiophen-3-ylphenyl]-6- oxo-4-(trifluoromethyl)- 1H-pyridine-3-carboxamide::US11319299, Example 493	WD repeat-containing protein 5				 2.86						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553418	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553418&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608115	469797282							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167179	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1csc(CN2CCOCC2)c1			553419	N-[4-fluoro-5-[5- (morpholin-4-ylmethyl) thiophen-3-yl]-2-[rac- (3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 494	WD repeat-containing protein 5				 3.01						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553419	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553419&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608116	469797283							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167180	C\[O]=c1\[nH]cc(cc1C(F)(F)F)C(=O)Nc1cc(c(F)cc1N1CCN(C)[C@@H](C)C1)-c1cnc(nc1)N1CCOCC1			553420	N-[4-fluoro-5-(2- morpholin-4-ylpyrimidin- 5-yl)-2-[rac-(3R)-3,4- dimethylpiperazin-1- yl]phenyl]-6-oxo-5- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 495	WD repeat-containing protein 5				 24.9						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553420	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553420&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138551576	469797284							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167181	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ncc(s1)C(=O)NCC1CC1			553421	N-(cyclopropylmethyl)-2- [2-fluoro-5-[[6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carbonyl]amino]- 4-[rac-(3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-1,3-thiazole-5- carboxamide::US11319299, Example 496	WD repeat-containing protein 5				 3.03						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553421	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553421&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608117	469797285							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167182	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ncc(s1)C(=O)N(C)CC1CC1			553422	N-(cyclopropylmethyl)-2- [2-fluoro-5-[[6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carbonyl]amino]- 4-[rac-(3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-N-methyl-1,3- thiazole-5-carboxamide::US11319299, Example 497	WD repeat-containing protein 5				 2.59						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553422	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553422&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608118	469797286							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167183	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=[S]C(=CN1)C(=O)NC1CCCCC1			553423	N-cyclohexyl-2-[2- fluoro-5-[[6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carbonyl]amino]- 4-[rac-(3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-1,3-thiazole-5- carboxamide::US11319299, Example 498	WD repeat-containing protein 5				 1.47						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553423	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553423&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164885350	469797287							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167184	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=[S]C(=CN1)C(=O)N(C)C1CCCCC1			553424	N-cyclohexyl-2-[2- fluoro-5-[[6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carbonyl]amino]- 4-[rac-(3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-N-methyl-1,3- thiazolc-5-carboxamide::US11319299, Example 499	WD repeat-containing protein 5				 3.40						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553424	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553424&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164885351	469797288							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167185	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=[S]C(=CN1)C(=O)N1CCOCC1			553425	N-[4-fluoro-5-[5- (morpholine-4-carbonyl)- 1,3-thiazol-2-yl]-2-[rac- (3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 500	WD repeat-containing protein 5				 1.85						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553425	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553425&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164885352	469797289							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167186	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=[S]C(=CN1)C(=O)N1CCN(C)CC1			553426	N-[4-fluoro-5-[5-(4- methylpiperazine-1- carbonyl)-1,3-thiazol-2- yl]-2-[rac-(3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 501	WD repeat-containing protein 5				 3.44						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553426	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553426&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164885353	469797290							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167187	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1cc(N)c(F)cc1C(F)(F)F)-c1cnc(nc1)N1CCOCC1	InChI=1S/C29H32F5N7O2/c1-16-14-41(15-17(2)39(16)3)26-11-22(30)19(18-12-36-28(37-13-18)40-4-6-43-7-5-40)9-25(26)38-27(42)20-8-24(35)23(31)10-21(20)29(32,33)34/h8-13,16-17H,4-7,14-15,35H2,1-3H3,(H,38,42)/t16-,17+	RDYGVKWQXOWEFO-CALCHBBNSA-N	553427	5-amino-4-fluoro-N-[4- fluoro-5-(2-morpholin-4- ylpyrimidin-5-yl)-2-[rac- (3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-2-(trifluoromethyl) benzamide::US11319299, Example 502	WD repeat-containing protein 5				 1.15						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553427	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553427&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138541753	469797291							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167188	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCN(CC1)c1ccc(nn1)C1CC1			553428	N-[5-[1-(6- cyclopropylpyridazin-3- yl)-3,6-dihydro-2H- pyridin-4-yl]-4-fluoro-2- [rac-(3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 503	WD repeat-containing protein 5				 2.44						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553428	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553428&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608119	469797292							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167189	CCc1ccc(nn1)N1CCC(=CC1)c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)(F)F)c(cc1F)N1C[C@H](C)N(C)[C@H](C)C1			553429	N-[5-[1-(6-ethylpyridazin- 3-yl)-3,6-dihydro-2H-pyridin- 4-yl]-4-fluoro-2-[rac-(3R,5S)- 3,4,5-trimethylpiperazin- 1-yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 504	WD repeat-containing protein 5				 2.44						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553429	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553429&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608120	469797293							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167190	COc1cc(c(cn1)C(=O)Nc1cc(c(F)cc1N1C[C@H](C)N(C)[C@H](C)C1)-c1cnc(nc1)N1CCOCC1)C(F)(F)F	InChI=1S/C29H33F4N7O3/c1-17-15-40(16-18(2)38(17)3)25-11-23(30)20(19-12-35-28(36-13-19)39-5-7-43-8-6-39)9-24(25)37-27(41)21-14-34-26(42-4)10-22(21)29(31,32)33/h9-14,17-18H,5-8,15-16H2,1-4H3,(H,37,41)/t17-,18+	NSMLWLULIDTGPK-HDICACEKSA-N	553430	N-[4-fluoro-5-(2- morpholin-4-ylpyrimidin- 5-yl)-2-[rac-(3R,5S)- 3,4,5-trimethylpiperazin- 1-yl]phenyl]-6-methoxy- 4-(trifluoromethyl)pyridine- 3-carboxamide::US11319299, Example 506	WD repeat-containing protein 5				 354						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553430	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553430&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138541755	469797294							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167191	C[C@H]1CN(CCO1)c1ccc(cn1)-c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)F)c(cc1F)N1CCN(C)[C@@H](C)C1			553431	4-(difluoromethyl)-N-[4- fluoro-2-[rac-(3R)-3,4- dimethylpiperazin-1-yl]- 5-[6-[rac-(2R)-2- methylmorpholin-4- yl]Pyridin-3-yl]phenyl]-6- oxo-1H-pyridine-3-carboxamide::US11319299, Example 507	WD repeat-containing protein 5				 1.76						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553431	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553431&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608121	469797295							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167192	C[C@@H]1CN(CCO1)c1ccc(cn1)-c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)F)c(cc1F)N1C[C@H](C)N(C)[C@H](C)C1			553432	4-(difluoromethyl)-N-[4- fluoro-5-[6-[rac-(2R)-2- methylmorpholin-4- yl]pyridin-3-yl)-2-[rac- (3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-6-oxo-1H- pyridine-3-carboxamide::US11319299, Example 508	WD repeat-containing protein 5				 2.66						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553432	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553432&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608122	469797296							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167193	C[C@@H]1CN(CCO1)c1ccc(cn1)-c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)F)c(cc1F)N1CCN(C)[C@@H](C)C1			553433	4-(difluoromethyl)-N-[4- fluoro-2-[rac-(3S)-3,4- dimethylpiperazin-1-yl]- 5-[6-[rac-(2R)-2- methylmorpholin-4- yl]pyridin-3-yl]phenyl]-6- oxo-1H-pyridine-3- carboxamide::US11319299, Example 509	WD repeat-containing protein 5				 0.947						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553433	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553433&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608123	469797297							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167194	C[C@H]1CN(CCO1)c1ccc(cn1)-c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)F)c(cc1F)N1C[C@H](C)N(C)[C@H](C)C1			553434	4-(difluoromethyl)-N-[4- fluoro-5-[6-[rac-(2R)-2- methylmorpholin-4- yl]pyridin-3-yl]-2-[rac- (3S,5R)-3,4,5- trimethylpiperazin-1- yl]phenyl]-6-oxo-1H- pyridine-3-carboxamide::US11319299, Example 510	WD repeat-containing protein 5				 0.623						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553434	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553434&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608124	469797298							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167195	C[C@H]1CN(C[C@@H](C)O1)c1ccc(cn1)-c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)F)c(cc1F)N1C[C@H](C)N(C)[C@H](C)C1			553435	4-(difluoromethyl)-N-[4- fluoro-5-[6-[rac-(2R,6S)- 2,6-dimethylmorpholin-4- yl]pyridin-3-yl]-2-[rac- (3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-6-oxo-1H- pyridine-3-carboxamide::US11319299, Example 511	WD repeat-containing protein 5				 0.779						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553435	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553435&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608125	469797299							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167196	C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1cc(N)c(F)cc1C(F)(F)F)-c1cnc(nc1)N1CCOCC1	InChI=1S/C28H30F5N7O2/c1-16-15-40(4-3-38(16)2)25-12-21(29)18(17-13-35-27(36-14-17)39-5-7-42-8-6-39)10-24(25)37-26(41)19-9-23(34)22(30)11-20(19)28(31,32)33/h9-14,16H,3-8,15,34H2,1-2H3,(H,37,41)/t16-/m0/s1	QTUYXFOWBHITSC-INIZCTEOSA-N	553436	5-amino-4-fluoro-N-[4- fluoro-5-(2-morpholin-4- ylpyrimidin-5-yl)-2-[rac- (3R)-3,4-dimethylpiperazin-1- yl]phenyl]-2-(trifluoromethyl) benzamide::US11319299, Example 512	WD repeat-containing protein 5				 0.711						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553436	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553436&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138551581	469797300							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167197	CCN1CC[C@H]2CN(C[C@@H]12)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cnc(nc1)N1CCOCC1			553437	N-[4-fluoro-5-(2- morpholin-4-ylpyrimidin- 5-yl)-2-[rac-(3aR,6aR)-1- ethyl-2,3,3a,4,6,6a- hexahydropyrrolo[2,3-c] pyrrol-5-yl]phenyl]-6- oxo-4-(trifluoromethyl)- 1H-pyridine-3-carboxamide::US11319299, Example 513	WD repeat-containing protein 5				 9.90						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553437	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553437&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608126	469797301							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167198	C[C@H]1CN(C[C@@H](C)O1)c1ccc(cn1)-c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)F)c(cc1F)N1CCN(C)[C@@H](C)C1			553438	4-(difluoromethyl)-N-[4- fluoro-5-[6-[rac-(2R,6S)- 2,6-dimethylmorpholin-4- yl]pyridin-3-yl]-2-[rac- (3S)-3,4-dimethylpiperazin-1- yl]phenyl]-6-oxo-1H- pyridine-3-carboxamide::US11319299, Example 514	WD repeat-containing protein 5				 0.959						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553438	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553438&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608127	469797302							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167199	C[C@H]1CN(C[C@@H](C)O1)c1ccc(cn1)-c1cc(NC(=O)c2cn(C)c(=O)cc2C(F)F)c(cc1F)N1CCN(C)[C@@H](C)C1	InChI=1S/C31H37F3N6O3/c1-18-14-39(9-8-37(18)4)27-12-25(32)22(21-6-7-28(35-13-21)40-15-19(2)43-20(3)16-40)10-26(27)36-31(42)24-17-38(5)29(41)11-23(24)30(33)34/h6-7,10-13,17-20,30H,8-9,14-16H2,1-5H3,(H,36,42)/t18-,19-,20+/m0/s1	BQVIODKCWLYNLR-SLFFLAALSA-N	553439	4-(difluoromethyl)-N-[4- fluoro-5-[6-[rac-(2R,6S)- 2,6-dimethylmorpholin-4- yl]pyridin-3-yl]-2-[rac- (3S)-3,4-dimethylpiperazin-1- yl]phenyl]-1-methyl-6- oxopyridine-3-carboxamide::US11319299, Example 515	WD repeat-containing protein 5				 4.09						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553439	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553439&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138541701	469797303							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167200	C[C@@H]1CN(CCO1)c1ccc(cn1)-c1cc(NC(=O)c2cn(C)c(=O)cc2C(F)F)c(cc1F)N1CCN(C)[C@@H](C)C1	InChI=1S/C30H35F3N6O3/c1-18-15-38(8-7-36(18)3)26-13-24(31)21(20-5-6-27(34-14-20)39-9-10-42-19(2)16-39)11-25(26)35-30(41)23-17-37(4)28(40)12-22(23)29(32)33/h5-6,11-14,17-19,29H,7-10,15-16H2,1-4H3,(H,35,41)/t18-,19+/m0/s1	GUMGGQGWDFBAJZ-RBUKOAKNSA-N	553440	4-(difluoromethyl)-N-[4- fluoro-2-[rac-(3S)-3,4- dimethylpiperazin-1-yl]- 5-[6-[rac-(2R)-2- methylmorpholin-4- yl]pyridin-3-yl]phenyl]-1- methyl-6-oxopyridine-3- carboxamide::US11319299, Example 516	WD repeat-containing protein 5				 4.00						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553440	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553440&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			137377171	469797304							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167201	C[C@H]1CN(CCO1)c1ccc(cn1)-c1cc(NC(=O)c2cn(C)c(=O)cc2C(F)F)c(cc1F)N1C[C@H](C)N(C)[C@H](C)C1	InChI=1S/C31H37F3N6O3/c1-18-14-40(15-19(2)38(18)5)27-12-25(32)22(21-6-7-28(35-13-21)39-8-9-43-20(3)16-39)10-26(27)36-31(42)24-17-37(4)29(41)11-23(24)30(33)34/h6-7,10-13,17-20,30H,8-9,14-16H2,1-5H3,(H,36,42)/t18-,19+,20-/m0/s1	JPAMAMFUQDMPRD-ZCNNSNEGSA-N	553441	4-(difluoromethyl)-N-[4- fluoro-5-[6-[rac-(2R)-2- methylmorpholin-4- yl]pyridin-3-yl]-2-[rac- (3S,5R)-3,4,5- trimethylpiperazin-1- yl]phenyl]-1-methyl-6- oxopyridine-3-carboxamide::US11319299, Example 517	WD repeat-containing protein 5				 5.97						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553441	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553441&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138542513	469797305							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167202	C[C@H]1CN(C[C@@H](C)O1)c1ccc(cn1)-c1cc(NC(=O)c2cn(C)c(=O)cc2C(F)F)c(cc1F)N1C[C@H](C)N(C)[C@H](C)C1	InChI=1S/C32H39F3N6O3/c1-18-13-40(14-19(2)39(18)6)28-11-26(33)23(22-7-8-29(36-12-22)41-15-20(3)44-21(4)16-41)9-27(28)37-32(43)25-17-38(5)30(42)10-24(25)31(34)35/h7-12,17-21,31H,13-16H2,1-6H3,(H,37,43)/t18-,19+,20-,21+	MJBDOBUCPDQIEC-FXELSEDVSA-N	553442	4-(difluoromethyl)-N-[4- fluoro-5-[6-[rac-(2R,6S)- 2,6-dimethylmorpholin-4- yl]pyridin-3-yl]-2-[rac- (3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-1-methyl-6- oxopyridine-3-carboxamide::US11319299, Example 518	WD repeat-containing protein 5				 3.41						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553442	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553442&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138541685	469797306							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167203	C[C@H]1CN(CCO1)c1ccc(cn1)-c1cc(NC(=O)c2cn(C)c(=O)cc2C(F)F)c(cc1F)N1CCN(C)[C@@H](C)C1	InChI=1S/C30H35F3N6O3/c1-18-15-38(8-7-36(18)3)26-13-24(31)21(20-5-6-27(34-14-20)39-9-10-42-19(2)16-39)11-25(26)35-30(41)23-17-37(4)28(40)12-22(23)29(32)33/h5-6,11-14,17-19,29H,7-10,15-16H2,1-4H3,(H,35,41)/t18-,19-/m0/s1	GUMGGQGWDFBAJZ-OALUTQOASA-N	553443	4-(difluoromethyl)-N-[4- fluoro-2-[rac-(3R)-3,4- dimethylpiperazin-1-yl]- 5-[6-[rac-(2R)-2- methylmorpholin-4- yl]pyridin-3-yl]phenyl]-1- methyl-6-oxopyridine-3- carboxamide::US11319299, Example 519	WD repeat-containing protein 5				 3.39						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553443	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553443&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138542481	469797307							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167204	C[C@H]1COCCN1c1ncc(cn1)-c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)F)c(cc1F)N1CCN(C)[C@@H](C)C1			553444	4-(difluoromethyl)-N-[4- fluoro-5-[2-[rac-(3R)-3- methylmorpholin-4- yl]pyrimidin-5-yl]-2-[rac- (3S,5R)-3,4,5- trimethylpiperazin-1- yl]phenyl]-6-oxo-1H- pyridine-3-carboxamide::US11319299, Example 521::US11319299, Example 628	WD repeat-containing protein 5				 0.579						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553444	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553444&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608128	469797308							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167205	C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1cn(C)c(=O)cc1C(F)(F)F)-c1ccc(OCC2CC2)nc1	InChI=1S/C29H31F4N5O3/c1-17-14-38(9-8-36(17)2)25-12-23(30)20(19-6-7-26(34-13-19)41-16-18-4-5-18)10-24(25)35-28(40)21-15-37(3)27(39)11-22(21)29(31,32)33/h6-7,10-13,15,17-18H,4-5,8-9,14,16H2,1-3H3,(H,35,40)/t17-/m0/s1	LGLGPJVPAOVCOA-KRWDZBQOSA-N	553445	N-[5-[6-(cyclopropylmethoxy) pyridin-3-yl]-4-fluoro-2-[rac- (3R)-3,4-dimethylpiperazin-1- yl]phenyl]-1-methyl-6- oxo-4-(trifluoromethyl) pyridine-3-carboxamide::US11319299, Example 522	WD repeat-containing protein 5				 5.62						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553445	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553445&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138542597	469797309							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167206	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1cn(C)c(=O)cc1C(F)(F)F)-c1csc(n1)C(=O)NCC1CC1	InChI=1S/C29H32F4N6O3S/c1-15-11-39(12-16(2)38(15)4)24-9-21(30)18(23-14-43-28(36-23)27(42)34-10-17-5-6-17)7-22(24)35-26(41)19-13-37(3)25(40)8-20(19)29(31,32)33/h7-9,13-17H,5-6,10-12H2,1-4H3,(H,34,42)(H,35,41)/t15-,16+	XKFXVWTTZHPMSW-IYBDPMFKSA-N	553446	N-(cyclopropylmethyl)-4- [2-fluoro-5-[[1-methyl-6- oxo-4-(trifluoromethyl) pyridine-3-carbonyl]amino]-4- [rac-(3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-1,3-thiazole-2- carboxamide::US11319299, Example 523	WD repeat-containing protein 5				 4.59						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553446	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553446&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			137377226	469797310							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167207	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1cn(C)c(=O)cc1C(F)(F)F)-c1csc(n1)C(=O)N(C)CC1CC1	InChI=1S/C30H34F4N6O3S/c1-16-11-40(12-17(2)39(16)5)25-10-22(31)19(24-15-44-28(36-24)29(43)38(4)13-18-6-7-18)8-23(25)35-27(42)20-14-37(3)26(41)9-21(20)30(32,33)34/h8-10,14-18H,6-7,11-13H2,1-5H3,(H,35,42)/t16-,17+	HLWJDWJTXLGGCJ-CALCHBBNSA-N	553447	N-(cyclopropylmethyl)-4- [2-fluoro-5-[[1-methyl-6- oxo-4-(trifluoromethyl) pyridine-3-carbonyl]amino]-4- [rac-(3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-N-methyl-1,3- thiazole-2-carboxamide::US11319299, Example 524	WD repeat-containing protein 5				 5.03						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553447	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553447&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			137376801	469797311							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167208	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1cn(C)c(=O)cc1C(F)(F)F)-c1csc(n1)C(=O)NC1CCCCC1	InChI=1S/C31H36F4N6O3S/c1-17-13-41(14-18(2)40(17)4)26-12-23(32)20(25-16-45-30(38-25)29(44)36-19-8-6-5-7-9-19)10-24(26)37-28(43)21-15-39(3)27(42)11-22(21)31(33,34)35/h10-12,15-19H,5-9,13-14H2,1-4H3,(H,36,44)(H,37,43)/t17-,18+	BQSBVEONZMXQGE-HDICACEKSA-N	553448	N-cyclohexyl-4-[2- fluoro-5-[[1-methyl-6- oxo-4-(trifluoromethyl) pyridine-3-carbonyl]amino]-4- [rac-(3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-1,3-thiazole-2- carboxamide::US11319299, Example 525	WD repeat-containing protein 5				 5.42						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553448	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553448&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			137377422	469797312							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167209	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1cn(C)c(=O)cc1C(F)(F)F)-c1csc(n1)C(=O)N(C)C1CCCCC1	InChI=1S/C32H38F4N6O3S/c1-18-14-42(15-19(2)40(18)4)27-13-24(33)21(26-17-46-30(38-26)31(45)41(5)20-9-7-6-8-10-20)11-25(27)37-29(44)22-16-39(3)28(43)12-23(22)32(34,35)36/h11-13,16-20H,6-10,14-15H2,1-5H3,(H,37,44)/t18-,19+	SCMNLMDUWQDRHX-KDURUIRLSA-N	553449	N-cyclohexyl-4-[2- fluoro-5-[[1-methyl-6- oxo-4-(trifluoromethyl) pyridine-3-carbonyl]amino]- 4-[rac-(3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-N-methyl-1,3- thiazole-2-carboxamide::US11319299, Example 526	WD repeat-containing protein 5				 4.89						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553449	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553449&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			137377292	469797313							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167210	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1cn(C)c(=O)cc1C(F)(F)F)-c1csc(n1)C(=O)N1CCOCC1	InChI=1S/C29H32F4N6O4S/c1-16-12-39(13-17(2)37(16)4)24-11-21(30)18(23-15-44-27(35-23)28(42)38-5-7-43-8-6-38)9-22(24)34-26(41)19-14-36(3)25(40)10-20(19)29(31,32)33/h9-11,14-17H,5-8,12-13H2,1-4H3,(H,34,41)/t16-,17+	LOTZOUXGDXHJKA-CALCHBBNSA-N	553450	N-[4-fluoro-5-[2- (morpholine-4-carbonyl)- 1,3-thiazol-4-yl]-2-[rac- (3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-1-methyl-6- oxo-4-(trifluoromethyl) pyridine-3-carboxamide::US11319299, Example 527	WD repeat-containing protein 5				 5.66						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553450	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553450&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			137376940	469797314							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167211	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1cn(C)c(=O)cc1C(F)(F)F)-c1csc(n1)C(=O)N1CCN(C)CC1	InChI=1S/C30H35F4N7O3S/c1-17-13-41(14-18(2)39(17)5)25-12-22(31)19(24-16-45-28(36-24)29(44)40-8-6-37(3)7-9-40)10-23(25)35-27(43)20-15-38(4)26(42)11-21(20)30(32,33)34/h10-12,15-18H,6-9,13-14H2,1-5H3,(H,35,43)/t17-,18+	OGQDCUJPQMPAIM-HDICACEKSA-N	553451	N-[4-fluoro-5-[2-(4- methylpiperazine-1- carbonyl)-1,3-thiazol-4- yl]-2-[rac-(3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-1-methyl-6- oxo-4-(trifluoromethyl) pyridine-3-carboxamide::US11319299, Example 528	WD repeat-containing protein 5				 4.05						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553451	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553451&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138541808	469797315							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167212	C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1ccc(F)cc1C(F)(F)F)-c1ccc(cc1)N1CCNCC1	InChI=1S/C30H32F5N5O/c1-19-18-40(14-13-38(19)2)28-17-26(32)24(20-3-6-22(7-4-20)39-11-9-36-10-12-39)16-27(28)37-29(41)23-8-5-21(31)15-25(23)30(33,34)35/h3-8,15-17,19,36H,9-14,18H2,1-2H3,(H,37,41)/t19-/m0/s1	BLPJPUPAZTVKIQ-IBGZPJMESA-N	553452	4-fluoro-N-[4-fluoro-5-(4- piperazin-1-ylphenyl)-2- [rac-(3R)-3,4- dimethylpiperazin-1- yl]phenyl]-2-(trifluoromethyl) benzamide::US11319299, Example 529	WD repeat-containing protein 5				 2.92						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553452	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553452&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138551467	469797316							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167213	C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1ccc(F)cc1C(F)(F)F)-c1ccc(nc1)N1CCNCC1	InChI=1S/C29H31F5N6O/c1-18-17-40(12-11-38(18)2)26-15-24(31)22(19-3-6-27(36-16-19)39-9-7-35-8-10-39)14-25(26)37-28(41)21-5-4-20(30)13-23(21)29(32,33)34/h3-6,13-16,18,35H,7-12,17H2,1-2H3,(H,37,41)/t18-/m0/s1	DCMCFPHKSHIZQQ-SFHVURJKSA-N	553453	4-fluoro-N-[4-fluoro-5-(6- piperazin-1-ylpyridin-3- yl)-2-[rac-(3R)-3,4- dimethylpiperazin-1- yl]phenyl]-2- (trifluoromethyl)benzamide::US11319299, Example 530	WD repeat-containing protein 5				 2.16						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553453	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553453&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138551583	469797317							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167214	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1csc(n1)C(=O)NCC1CC1			553454	N-(cyclopropylmethyl)-4- [2-fluoro-5-[[6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carbonyl]amino]- 4-[rac-(3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-1,3-thiazole-2- carboxamide::US11319299, Example 531	WD repeat-containing protein 5				 1.06						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553454	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553454&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608129	469797318							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167215	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1csc(n1)C(=O)N(C)CC1CC1			553455	N-(cyclopropylmethyl)-4- [2-fluoro-5-[[6-oxo-4- (trifluoromethyl)-1H- pyridine-3- carbonyl]amino]-4-[rac- (3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-N-methyl-1,3- thiazole-2-carboxamide::US11319299, Example 532	WD repeat-containing protein 5				 0.694						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553455	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553455&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608130	469797319							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167216	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1csc(n1)C(=O)NC1CCCCC1			553456	N-cyclohexyl-4-[2- fluoro-5-[[6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carbonyl]amino]- 4-[rac-(3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-1,3-thiazole-2- carboxamide::US11319299, Example 533	WD repeat-containing protein 5				 1.98						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553456	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553456&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608131	469797320							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167217	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1csc(n1)C(=O)N(C)C1CCCCC1			553457	N-cyclohexyl-4-[2- fluoro-5-[[6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carbonyl]amino]- 4-[rac-(3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-N-methyl-1,3- thiazole-2-carboxamide::US11319299, Example 534	WD repeat-containing protein 5				 1.31						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553457	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553457&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608132	469797321							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167218	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1csc(n1)C(=O)N1CCOCC1			553458	N-[4-fluoro-5-[2- (morpholine-4-carbonyl)- 1,3-thiazol-4-yl]-2-[rac- (3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 535	WD repeat-containing protein 5				 2.80						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553458	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553458&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608133	469797322							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167219	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1csc(n1)C(=O)N1CCN(C)CC1			553459	N-[4-fluoro-5-[2-(4- methylpiperazine-1- carbonyl)-1,3-thiazol-4- yl]-2-[rac-(3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 536	WD repeat-containing protein 5				 1.03						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553459	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553459&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608134	469797323							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167220	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccnc(NC2CCCCC2)n1			553460	N-[5-[2-(cyclohexylamino) pyrimidin-4-yl]-4-fluoro-2-[rac- (3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 537	WD repeat-containing protein 5				 0.944						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553460	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553460&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608135	469797324							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167221	CNc1nccc(n1)-c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)(F)F)c(cc1F)N1C[C@H](C)N(C)[C@H](C)C1			553461	N-[4-fluoro-5-[2- (methylamino)pyrimidin- 4-yl]-2-[rac-(3R,5S)- 3,4,5-trimethylpiperazin- 1-yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 538	WD repeat-containing protein 5				 3.02						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553461	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553461&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608136	469797325							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167222	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccnc(n1)C#N			553462	N-[5-(2-cyanopyrimidin- 4-yl)-4-fluoro-2-[rac- (3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 539	WD repeat-containing protein 5				 2.56						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553462	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553462&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608137	469797326							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167223	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccnc(n1)N(C)C			553463	N-[5-[2-(dimethylamino) pyrimidin-4-yl]-4-fluoro- 2-[rac-(3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 540	WD repeat-containing protein 5				 1.10						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553463	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553463&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608138	469797327							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167224	CNC1CCN(CC1)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cnc(nc1)N1CCOCC1	InChI=1S/C27H29F4N7O3/c1-32-17-2-4-37(5-3-17)23-12-21(28)18(16-13-34-26(35-14-16)38-6-8-41-9-7-38)10-22(23)36-25(40)19-15-33-24(39)11-20(19)27(29,30)31/h10-15,17,32H,2-9H2,1H3,(H,33,39)(H,36,40)	NDSVXXWYDJFFLM-UHFFFAOYSA-N	553464	N-[4-fluoro-2-[4- (methylamino)piperidin- 1-yl]-5-(2-morpholin-4- ylpyrimidin-5-yl)phenyl]- 6-oxo-4-(trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 541	WD repeat-containing protein 5				 7.44						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553464	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553464&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608139	469797328							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167225	C[C@@H]1CN(CCO1)c1ccc(cn1)-c1cc(NC(=O)c2cn(C)c(=O)cc2C(F)F)c(cc1F)N1C[C@H](C)N(C)[C@H](C)C1	InChI=1S/C31H37F3N6O3/c1-18-14-40(15-19(2)38(18)5)27-12-25(32)22(21-6-7-28(35-13-21)39-8-9-43-20(3)16-39)10-26(27)36-31(42)24-17-37(4)29(41)11-23(24)30(33)34/h6-7,10-13,17-20,30H,8-9,14-16H2,1-5H3,(H,36,42)/t18-,19+,20-/m1/s1	JPAMAMFUQDMPRD-HSALFYBXSA-N	553465	4-(difluoromethyl)-N-[4- fluoro-5-[6-[rac-(2R)-2- methylmorpholin-4- yl]pyridin-3-yl]-2-[rac- (3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-1-methyl-6- oxopyridine-3-carboxamide::US11319299, Example 542	WD repeat-containing protein 5				 5.53						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553465	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553465&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			137377047	469797329							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167226	C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1cn(C)c(=O)cc1C(F)F)-c1ccc(OCC2CC2)nc1	InChI=1S/C29H32F3N5O3/c1-17-14-37(9-8-35(17)2)25-12-23(30)20(19-6-7-26(33-13-19)40-16-18-4-5-18)10-24(25)34-29(39)22-15-36(3)27(38)11-21(22)28(31)32/h6-7,10-13,15,17-18,28H,4-5,8-9,14,16H2,1-3H3,(H,34,39)/t17-/m0/s1	QSRBIBQPRKNDSR-KRWDZBQOSA-N	553466	N-[5-[6-(cyclopropylmethoxy) pyridin-3-yl]-4-fluoro-2-[rac- (3R)-3,4-dimethylpiperazin-1- yl]phenyl]-4-(difluoromethyl)- 1-methyl-6-oxopyridine-3- carboxamide::US11319299, Example 543	WD repeat-containing protein 5				 8.21						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553466	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553466&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138551685	469797330							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167227	C[C@@H]1CN(CCO1)c1ncc(cn1)-c1cc(NC(=O)c2cn(C)c(=O)cc2C(F)(F)F)c(cc1F)N1CCN(C)[C@@H](C)C1	InChI=1S/C29H33F4N7O3/c1-17-14-39(6-5-37(17)3)25-11-23(30)20(19-12-34-28(35-13-19)40-7-8-43-18(2)15-40)9-24(25)36-27(42)21-16-38(4)26(41)10-22(21)29(31,32)33/h9-13,16-18H,5-8,14-15H2,1-4H3,(H,36,42)/t17-,18+/m0/s1	UQOLIVLMQOQTBL-ZWKOTPCHSA-N	553467	N-[4-fluoro-2-[rac-(3S)- 3,4-dimethylpiperazin-1- yl]-5-[2-[rac-(2R)-2- methylmorpholin-4- yl]pyrimidin-5-yl]phenyl]- 1-methyl-6-oxo-4- (trifluoromethyl)pyridine- 3-carboxamide::US11319299, Example 544	WD repeat-containing protein 5				 1.80						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553467	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553467&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			137377296	469797331							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167228	C[C@@H]1CN(CCO1)c1ncc(cn1)-c1cc(NC(=O)c2ccc(F)cc2C(F)(F)F)c(cc1F)N1C[C@H](C)N(C)[C@H](C)C1	InChI=1S/C30H33F5N6O2/c1-17-14-41(15-18(2)39(17)4)27-11-25(32)23(20-12-36-29(37-13-20)40-7-8-43-19(3)16-40)10-26(27)38-28(42)22-6-5-21(31)9-24(22)30(33,34)35/h5-6,9-13,17-19H,7-8,14-16H2,1-4H3,(H,38,42)/t17-,18+,19-/m1/s1	YHRUDJMQAFXZEQ-CEXWTWQISA-N	553468	4-fluoro-N-[4-fluoro-5- [2-[rac-(2R)-2- methylmorpholin-4- yl]pyrimidin-5-yl]-2-[rac- (3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-2- (trifluoromethyl)benzamide::US11319299, Example 545	WD repeat-containing protein 5				 3.40						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553468	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553468&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			137377681	469797332							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167229	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1ccc(F)cc1C(F)(F)F)-c1cnc(nc1)N1CCNCC1	InChI=1S/C29H32F5N7O/c1-17-15-41(16-18(2)39(17)3)26-12-24(31)22(19-13-36-28(37-14-19)40-8-6-35-7-9-40)11-25(26)38-27(42)21-5-4-20(30)10-23(21)29(32,33)34/h4-5,10-14,17-18,35H,6-9,15-16H2,1-3H3,(H,38,42)/t17-,18+	PHGWBZCYPVTWQV-HDICACEKSA-N	553469	4-fluoro-N-[4-fluoro-5- (2-piperazin-1-ylpyrimidin- 5-yl)-2-[rac-(3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-2-(trifluoromethyl) benzamide::US11319299, Example 546	WD repeat-containing protein 5				 2.10						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553469	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553469&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			137376849	469797333							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167230	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1ccc(F)cc1C(F)(F)F)-c1ccc(nc1)N1CCOCC1	InChI=1S/C30H32F5N5O2/c1-18-16-40(17-19(2)38(18)3)27-14-25(32)23(20-4-7-28(36-15-20)39-8-10-42-11-9-39)13-26(27)37-29(41)22-6-5-21(31)12-24(22)30(33,34)35/h4-7,12-15,18-19H,8-11,16-17H2,1-3H3,(H,37,41)/t18-,19+	BBHLHXUXGHZBSQ-KDURUIRLSA-N	553470	4-fluoro-N-[4-fluoro-5- (6-morpholin-4-ylpyridin- 3-yl)-2-[rac-(3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-2-(trifluoromethyl) benzamide::US11319299, Example 547	WD repeat-containing protein 5				 1.50						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553470	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553470&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			137377067	469797334							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167231	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(nc1)N1CCNCC1			553471	N-[4-fluoro-5-(6- piperazin-1-ylpyridin-3- yl)-2-[rac-(3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 548	WD repeat-containing protein 5				 0.500						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553471	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553471&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608140	469797335							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167232	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(cc1)N1CCNCC1			553472	N-[4-fluoro-5-(4- piperazin-1-ylphenyl)-2- [rac-(3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 549	WD repeat-containing protein 5				 0.800						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553472	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553472&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608141	469797336							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167233	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(F)c(c1)C(N)=O			553473	N-[5-(3-carbamoyl-4- fluorophenyl)-4-fluoro-2- [rac-(3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 550	WD repeat-containing protein 5				 2.50						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553473	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553473&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608142	469797337							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167234	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(C(N)=O)c(F)c1			553474	N-[5-(4-carbamoyl-3- fluorophenyl)-4-fluoro-2- [rac-(3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 551	WD repeat-containing protein 5				 0.600						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553474	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553474&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608143	469797338							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167235	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)F)-c1ccc(F)c(c1)C(N)=O			553475	N-[5-(3-carbamoyl-4- fluorophenyl)-4-fluoro-2- [rac-(3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-4- (difluoromethyl)-6-oxo- 1H-pyridine-3-carboxamide::US11319299, Example 552	WD repeat-containing protein 5				 3.10						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553475	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553475&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608144	469797339							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167236	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)F)-c1ccc(C(N)=O)c(F)c1			553476	N-[5-(4-carbamoyl-3- fluorophenyl)-4-fluoro-2- [rac-(3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-4-(difluoromethyl)- 6-oxo-1H-pyridine-3- carboxamide::US11319299, Example 553	WD repeat-containing protein 5				 1.000						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553476	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553476&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608145	469797340							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167237	C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1ccc(F)cc1C(F)(F)F)-c1ccc(F)c(c1)C(N)=O	InChI=1S/C27H24F6N4O2/c1-14-13-37(8-7-36(14)2)24-12-22(30)18(15-3-6-21(29)19(9-15)25(34)38)11-23(24)35-26(39)17-5-4-16(28)10-20(17)27(31,32)33/h3-6,9-12,14H,7-8,13H2,1-2H3,(H2,34,38)(H,35,39)/t14-/m0/s1	WMXFUBIWWNJHTQ-AWEZNQCLSA-N	553477	2-fluoro-5-[2-fluoro-5- [[4-fluoro-2-(trifluoromethyl) benzoyl]amino]-4-[rac-(3R)- 3,4-dimethylpiperazin-1- yl]phenyl]benzamide::US11319299, Example 554	WD repeat-containing protein 5				 5.30						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553477	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553477&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138551379	469797341							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167238	C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1ccc(F)cc1C(F)(F)F)-c1ccc(C(N)=O)c(F)c1	InChI=1S/C27H24F6N4O2/c1-14-13-37(8-7-36(14)2)24-12-22(30)19(15-3-5-18(25(34)38)21(29)9-15)11-23(24)35-26(39)17-6-4-16(28)10-20(17)27(31,32)33/h3-6,9-12,14H,7-8,13H2,1-2H3,(H2,34,38)(H,35,39)/t14-/m0/s1	NGFYKPPLHCYJGM-AWEZNQCLSA-N	553478	2-fluoro-4-[2-fluoro-5- [[4-fluoro-2- (trifluoromethyl)benzoyl] amino]-4-[rac-(3R)-3,4- dimethylpiperazin-1- yl]phenyl]benzamide::US11319299, Example 555	WD repeat-containing protein 5				 2.94						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553478	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553478&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138551487	469797342							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167239	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1ccc(F)cc1C(F)(F)F)-c1ccc(F)c(c1)C(N)=O	InChI=1S/C28H26F6N4O2/c1-14-12-38(13-15(2)37(14)3)25-11-23(31)19(16-4-7-22(30)20(8-16)26(35)39)10-24(25)36-27(40)18-6-5-17(29)9-21(18)28(32,33)34/h4-11,14-15H,12-13H2,1-3H3,(H2,35,39)(H,36,40)/t14-,15+	CGGRRNPZYDEUQD-GASCZTMLSA-N	553479	2-fluoro-5-[2-fluoro-5- [[4-fluoro-2- (trifluoromethyl)benzoyl] amino]-4-[rac-(3R,5S)- 3,4,5-trimethylpiperazin- 1-yl]phenyl]benzamide::US11319299, Example 556	WD repeat-containing protein 5				 10.4						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553479	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553479&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138541727	469797343							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167240	C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1ccc(F)cc1C(F)(F)F)-c1cnc(nc1)N1CCN(CC1)C(C)(C)C	InChI=1S/C32H38F5N7O/c1-20-19-43(9-8-41(20)5)28-16-26(34)24(15-27(28)40-29(45)23-7-6-22(33)14-25(23)32(35,36)37)21-17-38-30(39-18-21)42-10-12-44(13-11-42)31(2,3)4/h6-7,14-18,20H,8-13,19H2,1-5H3,(H,40,45)/t20-/m0/s1	FECYEYRJVWGNAQ-FQEVSTJZSA-N	553480	N-[5-[2-(4-tert- butylpiperazin-1- yl)pyrimidin-5-yl]-4- fluoro-2-[rac-(3R)-3,4- dimethylpiperazin-1- yl]phenyl]-4-fluoro-2- (trifluoromethyl)benzamide::US11319299, Example 557	WD repeat-containing protein 5				 1.09						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553480	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553480&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138551474	469797344							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167241	C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1ccc(F)cc1C(F)(F)F)-c1cnc(nc1)N1CCOC(C)(C)C1	InChI=1S/C30H33F5N6O2/c1-18-16-40(8-7-39(18)4)26-13-24(32)22(19-14-36-28(37-15-19)41-9-10-43-29(2,3)17-41)12-25(26)38-27(42)21-6-5-20(31)11-23(21)30(33,34)35/h5-6,11-15,18H,7-10,16-17H2,1-4H3,(H,38,42)/t18-/m0/s1	YRXOMHVWDNWURK-SFHVURJKSA-N	553481	N-[5-[2-(2,2- dimethylmorpholin-4- yl)pyrimidin-5-yl]-4- fluoro-2-[rac-(3R)-3,4- dimethylpiperazin-1- yl]phenyl]-4-fluoro-2- (trifluoromethyl)benzamide::US11319299, Example 558	WD repeat-containing protein 5				 3.78						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553481	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553481&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138551494	469797345							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167242	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1ccc(F)cc1C(F)(F)F)-c1cnc(nc1)N1CCOC(C)(C)C1	InChI=1S/C31H35F5N6O2/c1-18-15-42(16-19(2)40(18)5)27-12-25(33)23(20-13-37-29(38-14-20)41-8-9-44-30(3,4)17-41)11-26(27)39-28(43)22-7-6-21(32)10-24(22)31(34,35)36/h6-7,10-14,18-19H,8-9,15-17H2,1-5H3,(H,39,43)/t18-,19+	YWOYODRMXPTJIB-KDURUIRLSA-N	553482	N-[5-[2-(2,2- dimethylmorpholin-4- yl)pyrimidin-5-yl]-4- fluoro-2-[rac-(3R,5S)- 3,4,5-trimethylpiperazin-1- yl]phenyl]-4-fluoro-2- (trifluoromethyl)benzamide::US11319299, Example 559	WD repeat-containing protein 5				 2.92						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553482	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553482&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138541826	469797346							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167243	C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1ccc(F)cc1C(F)(F)F)-c1ccc(nc1)N1CCN(CC2CC2)CC1	InChI=1S/C33H37F5N6O/c1-21-19-44(12-9-41(21)2)30-17-28(35)26(16-29(30)40-32(45)25-7-6-24(34)15-27(25)33(36,37)38)23-5-8-31(39-18-23)43-13-10-42(11-14-43)20-22-3-4-22/h5-8,15-18,21-22H,3-4,9-14,19-20H2,1-2H3,(H,40,45)/t21-/m0/s1	SPXQNSHYQNJIIQ-NRFANRHFSA-N	553483	N-[5-[2-[4- (cyclopropylmethyl)piperazin- 1-yl]pyrimidin-5-yl]- 4-fluoro-2-[rac-(3R)-3,4- dimethylpiperazin-1- yl]phenyl]-4-fluoro-2- (trifluoromethyl)benzamide::US11319299, Example 560	WD repeat-containing protein 5				 1.12						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553483	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553483&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138551858	469797347							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167244	Fc1cc(N2CCN(CC2)C2CC2)c(NC(=O)c2c[nH]c(=O)cc2C(F)(F)F)cc1-c1cnc(nc1)N1CCOCC1	InChI=1S/C28H29F4N7O3/c29-22-13-24(38-5-3-37(4-6-38)18-1-2-18)23(36-26(41)20-16-33-25(40)12-21(20)28(30,31)32)11-19(22)17-14-34-27(35-15-17)39-7-9-42-10-8-39/h11-16,18H,1-10H2,(H,33,40)(H,36,41)	RONIYNCQOSAEOQ-UHFFFAOYSA-N	553484	N-[2-(4- cyclopropylpiperazin-1- yl)-4-fluoro-5-(2- morpholin-4-ylpyrimidin- 5-yl)phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 561	WD repeat-containing protein 5				 23.5						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553484	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553484&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608146	469797348							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167245	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1c[nH]c(=O)c(F)c1			553485	N-[4-fluoro-5-(5-fluoro- 6-oxo-1H-pyridin-3-yl)- 2-[rac-(3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 562	WD repeat-containing protein 5				 0.904						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553485	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553485&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608147	469797349							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167246	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cncc(NC(=O)OCc2ccccc2)c1			553486	US11319299, Example 563::benzyl N-[5-[2-fluoro-5- [[6-oxo-4-(trifluoromethyl)- 1H-pyridine-3-carbonyl] amino]-4-[rac-(3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]pyridin-3-yl] carbamate	WD repeat-containing protein 5				 3.32						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553486	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553486&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608148	469797350							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167247	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cc(F)c(=O)n(C)c1			553487	N-[4-fluoro-5-(5-fluoro- 1-methyl-6-oxopyridin-3- yl)-2-[rac-(3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 564	WD repeat-containing protein 5				 1.52						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553487	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553487&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608149	469797351							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167248	COc1ccc(cc1)C(=O)N1CCC(=CC1)c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)(F)F)c(cc1F)N1C[C@H](C)N(C)[C@H](C)C1			553488	N-[4-fluoro-5-[1-(4- methoxybenzoyl)-3,6- dihydro-2H-pyridin-4-yl]- 2-[rac-(3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 565	WD repeat-containing protein 5				 0.943						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553488	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553488&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608150	469797352							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167249	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cnc2NC(=O)Cc2c1			553489	N-[4-fluoro-5-(2-oxo-1,3- dihydropyrrolo[2,3-b] pyridin-5-yl)-2-[rac-(3R,5S)- 3,4,5-trimethylpiperazin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 566	WD repeat-containing protein 5				 0.896						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553489	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553489&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608151	469797353							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167250	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccn(C)c(=O)c1			553490	N-[4-fluoro-5-(1-methyl- 2-oxopyridin-4-yl)-2- [rac-(3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 567	WD repeat-containing protein 5				 1.18						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553490	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553490&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608152	469797354							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167251	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(=O)n(C)c1			553491	N-[4-fluoro-5-(1-methyl- 6-oxopyridin-3-yl)-2- [rac-(3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 568	WD repeat-containing protein 5				 4.58						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553491	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553491&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608153	469797355							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167252	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCN(CC1)C(=O)C1CCCCC1			553492	N-[5-[1- (cyclohexanecarbonyl)- 3,6-dihydro-2H-pyridin- 4-yl]-4-fluoro-2-[rac- (3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 569	WD repeat-containing protein 5				 1.99						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553492	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553492&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608154	469797356							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167253	COCCCN(C)C1CCN(C1)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cnc(nc1)N1CCOCC1			553493	N-[4-fluoro-2-[3-[3- methoxypropyl(methyl) amino]pyrrolidin-1-yl]-5- (2-morpholin-4-ylpyrimidin- 5-yl)phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 572	WD repeat-containing protein 5				 113						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553493	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553493&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608155	469797357							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167254	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCN(CC1)C(=O)c1cnccn1			553494	N-[4-fluoro-5-[1- (pyrazine-2-carbonyl)- 3,6-dihydro-2H-pyridin- 4-yl]-2-[rac-(3R,5S)- 3,4,5-trimethylpiperazin- 1-yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 573	WD repeat-containing protein 5				 2.19						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553494	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553494&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608156	469797358							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167255	COCCN(C)[C@@H]1CCN(C1)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cnc(nc1)N1CCOCC1			553495	N-[4-fluoro-5-(2- morpholin-4-ylpyrimidin- 5-yl)-2-[rac-(3R)-3-[2- methoxyethyl(methyl) amino]pyrrolidin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 578	WD repeat-containing protein 5				 16.9						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553495	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553495&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608157	469797359							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167256	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(nc1)S(C)(=O)=O			553496	N-[4-fluoro-5-(6- methylsulfonylpyridin-3- yl)-2-[rac-(3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 581	WD repeat-containing protein 5				 0.768						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553496	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553496&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608158	469797360							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167257	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cnc(NS(C)(=O)=O)nc1			553497	N-[4-fluoro-5-[2- (methanesulfonamido) pyrimidin-5-yl]-2-[rac- (3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 582	WD repeat-containing protein 5				 5.78						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553497	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553497&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608159	469797361							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167258	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCCN(C1)c1ncc(cn1)C#N			553498	N-[5-[1-(5- cyanopyrimdin-2-yl)-3,6- dihydro-2H-pyridin-5-yl]- 4-fluoro-2-[rac-(3R,5S)- 3,4,5-trimethylpiperazin- 1-yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 583	WD repeat-containing protein 5				 0.877						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553498	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553498&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608160	469797362							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167259	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCCN(C1)S(C)(=O)=O			553499	N-[4-fluoro-5-(1- methylsulfonyl-3,6- dihydro-2H-pyridin-5-yl)- 2-[rac-(3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 584	WD repeat-containing protein 5				 1.21						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553499	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553499&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608161	469797363							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167260	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCN(CC1)S(C)(=O)=O			553500	N-[4-fluoro-5-(1- methylsulfonyl-3,6- dihydro-2H-pyridin-4-yl)- 2-[rac-(3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 585	WD repeat-containing protein 5				 0.829						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553500	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553500&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608162	469797364							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167261	CN(CC1CC1)[C@@H]1CCN(C1)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cnc(nc1)N1CCOCC1			553501	N-[4-fluoro-5-(2- morpholin-4-ylpyrimidin- 5-yl)-2-[rac-(3R)-3- [cyclopropylmethyl (methyl)amino]pyrrolidin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 586	WD repeat-containing protein 5				 15.5						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553501	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553501&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608163	469797365							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167262	CN(CC1CC1)[C@@H]1CCN(C1)c1cc(F)c(cc1NC(=O)c1cn(C)c(=O)cc1C(F)(F)F)-c1cnc(nc1)N1CCOCC1	InChI=1S/C31H35F4N7O3/c1-39(16-19-3-4-19)21-5-6-42(17-21)27-13-25(32)22(20-14-36-30(37-15-20)41-7-9-45-10-8-41)11-26(27)38-29(44)23-18-40(2)28(43)12-24(23)31(33,34)35/h11-15,18-19,21H,3-10,16-17H2,1-2H3,(H,38,44)/t21-/m1/s1	RMVKDRWLQONYMP-OAQYLSRUSA-N	553502	N-[4-fluoro-5-(2- morpholin-4-ylpyrimidin- 5-yl)-2-[rac-(3R)-3- [cyclopropylmethyl (methyl)amino]pyrrolidin-1- yl]phenyl]-1-methyl-6- oxo-4-(trifluoromethyl) pyridine-3-carboxamide::US11319299, Example 587	WD repeat-containing protein 5				 253						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553502	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553502&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			137377102	469797366							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167263	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCN(C1)c1ncc(cn1)C#N			553503	N-[5-[1-(5-cyanopyrimidin- 2-yl)-2,5-dihydropyrrol-3-yl]- 4-fluoro-2-[rac-(3R,5S)- 3,4,5-trimethylpiperazin- 1-yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 588	WD repeat-containing protein 5				 1.72						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553503	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553503&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608164	469797367							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167264	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1cn(C)c(=O)cc1C(F)(F)F)-c1ccc(F)c(c1)C(N)=O	InChI=1S/C28H28F5N5O3/c1-14-11-38(12-15(2)37(14)4)24-10-22(30)17(16-5-6-21(29)18(7-16)26(34)40)8-23(24)35-27(41)19-13-36(3)25(39)9-20(19)28(31,32)33/h5-10,13-15H,11-12H2,1-4H3,(H2,34,40)(H,35,41)/t14-,15+	AKGJASQJRQYWMS-GASCZTMLSA-N	553504	N-[5-(3-carbamoyl-4- fluorophenyl)-4-fluoro-2- [rac-(3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-1-methyl-6- oxo-4-(trifluoromethyl) pyridine-3-carboxamide::US11319299, Example 589	WD repeat-containing protein 5				 7.46						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553504	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553504&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			137377099	469797368							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167265	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1cn(C)c(=O)cc1C(F)(F)F)-c1ccc(C(N)=O)c(F)c1	InChI=1S/C28H28F5N5O3/c1-14-11-38(12-15(2)37(14)4)24-10-22(30)18(16-5-6-17(26(34)40)21(29)7-16)8-23(24)35-27(41)19-13-36(3)25(39)9-20(19)28(31,32)33/h5-10,13-15H,11-12H2,1-4H3,(H2,34,40)(H,35,41)/t14-,15+	UURKMMIPYQNGSH-GASCZTMLSA-N	553505	N-[5-(4-carbamoyl-3- fluorophenyl)-4-fluoro-2- [rac-(3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-1-methyl-6- oxo-4-(trifluoromethyl) pyridine-3-carboxamide::US11319299, Example 590	WD repeat-containing protein 5				 3.32						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553505	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553505&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			137377155	469797369							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167266	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1cn(C)c(=O)cc1C(F)F)-c1ccc(F)c(c1)C(N)=O	InChI=1S/C28H29F4N5O3/c1-14-11-37(12-15(2)36(14)4)24-10-22(30)17(16-5-6-21(29)19(7-16)27(33)39)8-23(24)34-28(40)20-13-35(3)25(38)9-18(20)26(31)32/h5-10,13-15,26H,11-12H2,1-4H3,(H2,33,39)(H,34,40)/t14-,15+	JRHFVEXVDLYRTB-GASCZTMLSA-N	553506	N-[5-(3-carbamoyl-4- fluorophenyl)-4-fluoro-2- [rac-(3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-4-(difluoromethyl)- 1-methyl-6-oxopyridine-3- carboxamide::US11319299, Example 591	WD repeat-containing protein 5				 15.5						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553506	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553506&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			137376828	469797370							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167267	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1cn(C)c(=O)cc1C(F)F)-c1ccc(C(N)=O)c(F)c1	InChI=1S/C28H29F4N5O3/c1-14-11-37(12-15(2)36(14)4)24-10-22(30)18(16-5-6-17(27(33)39)21(29)7-16)8-23(24)34-28(40)20-13-35(3)25(38)9-19(20)26(31)32/h5-10,13-15,26H,11-12H2,1-4H3,(H2,33,39)(H,34,40)/t14-,15+	NWWYQJMLOGIQFP-GASCZTMLSA-N	553507	N-[5-(4-carbamoyl-3- fluorophenyl)-4-fluoro-2- [rac-(3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-4-(difluoromethyl)- 1-methyl-6-oxopyridine-3- carboxamide::US11319299, Example 592	WD repeat-containing protein 5				 6.80						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553507	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553507&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			137377284	469797371							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167268	C[C@H]1CN(CCO1)c1nccc(n1)-c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)(F)F)c(cc1F)N1CCN(C)[C@@H](C)C1			553508	N-[4-fluoro-2-[rac-(3R)- 3,4-dimethylpiperazin-1- yl]-5-[2-[rac-(2R)-2- methylmorpholin-4- yl]pyrimidin-4- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 593	WD repeat-containing protein 5				 0.737						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553508	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553508&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608165	469797372							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167269	C[C@H]1CN(CCO1)c1nccc(n1)-c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)(F)F)c(cc1F)N1C[C@H](C)N(C)[C@H](C)C1			553509	N-[4-fluoro-5-[2-[rac- (2R)-2-methylmorpholin- 4-yl]pyrimidin-4-yl]-2- [rac-(3S,5R)-3,4,5- trimethylpiperazin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 594	WD repeat-containing protein 5				 0.712						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553509	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553509&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608166	469797373							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167270	C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)F)-c1ccc(C(N)=O)c(F)c1			553510	N-[5-(4-carbamoyl-3- fluorophenyl)-4-fluoro-2- [rac-(3R)-3,4- dimethylpiperazin-1- yl]phenyl]-4- (difluoromethyl)-6-oxo- 1H-pyridine-3-carboxamide::US11319299, Example 595	WD repeat-containing protein 5				 1.18						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553510	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553510&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608167	469797374							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167271	C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)F)-c1ccc(F)c(c1)C(N)=O			553511	N-[5-(3-carbamoyl-4- fluorophenyl)-4-fluoro-2- [rac-(3R)-3,4- dimethylpiperazin-1- yl]phenyl]-4-(difluoromethyl)- 6-oxo-1H-pyridine-3- carboxamide::US11319299, Example 596	WD repeat-containing protein 5				 4.03						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553511	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553511&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608168	469797375							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167272	CNC(=O)c1ccc(cc1F)-c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)F)c(cc1F)N1CCN(C)[C@@H](C)C1			553512	4-(difluoromethyl)-N-[4- fluoro-5-[3-fluoro-4- (methylcarbamoyl)phenyl]- 2-[rac-(3R)-3,4- dimethylpiperazin-1- yl]phenyl]-6-oxo-1H- pyridine-3-carboxamide::US11319299, Example 597	WD repeat-containing protein 5				 0.711						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553512	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553512&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608169	469797376							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167273	CNC(=O)c1cc(ccc1F)-c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)F)c(cc1F)N1CCN(C)[C@@H](C)C1			553513	4-(difluoromethyl)-N-[4- fluoro-5-[4-fluoro-3- (methylcarbamoyl)phenyl]- 2-[rac-(3R)-3,4- dimethylpiperazin-1- yl]phenyl]-6-oxo-1H- pyridine-3-carboxamide::US11319299, Example 598	WD repeat-containing protein 5				 1.51						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553513	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553513&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608170	469797377							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167274	C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1nccc(n1)N1CCOCC1			553514	N-[4-fluoro-5-(4- morpholin-4-ylpyrimidin- 2-yl)-2-[rac-(3R)-3,4- dimethylpiperazin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 599	WD repeat-containing protein 5				 4.18						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553514	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553514&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608171	469797378							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167275	CC(C)OC(=O)N1CC=C(C1)c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)(F)F)c(cc1F)N1C[C@H](C)N(C)[C@H](C)C1			553515	US11319299, Example 600::propan-2-yl 3-[2-fluoro- 5-[[6-oxo-4-(trifluoromethyl)- 1H-pyridine-3-carbonyl] amino]-4-[rac-(3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-2,5- dihydropyrrole-1-carboxylate	WD repeat-containing protein 5				 0.779						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553515	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553515&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608172	469797379							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167276	CC(C)OC(=O)N1CCC=C(C1)c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)(F)F)c(cc1F)N1C[C@H](C)N(C)[C@H](C)C1			553516	US11319299, Example 601::propan-2-yl 5-[2-fluoro- 5-[[6-oxo-4-(trifluoromethyl)- 1H-pyridine-3-carbonyl] amino]-4-[rac-(3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-3,6-dihydro- 2H-pyridine-1-carboxylate	WD repeat-containing protein 5				 0.271						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553516	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553516&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608173	469797380							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167277	CC(C)OC(=O)N1CCC(=CC1)c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)(F)F)c(cc1F)N1C[C@H](C)N(C)[C@H](C)C1			553517	US11319299, Example 602::propan-2-yl 4-[2-fluoro- 5-[[6-oxo-4-(trifluoromethyl)- 1H-pyridine-3- carbonyl]amino]-4-[rac- (3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-3,6-dihydro- 2H-pyridine-1-carboxylate	WD repeat-containing protein 5				 0.475						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553517	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553517&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608174	469797381							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167278	CNC(=O)c1ccc(cc1F)-c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)(F)F)c(cc1F)N1C[C@H](C)N(C)[C@H](C)C1			553518	N-[4-fluoro-5-[3-fluoro- 4-(methylcarbamoyl)phenyl]- 2-[rac-(3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 603	WD repeat-containing protein 5				 1.09						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553518	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553518&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608175	469797382							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167279	CNC(=O)c1cc(ccc1F)-c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)(F)F)c(cc1F)N1C[C@H](C)N(C)[C@H](C)C1			553519	N-[4-fluoro-5-[4-fluoro- 3-(methylcarbamoyl)phenyl]- 2-[rac-(3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 604	WD repeat-containing protein 5				 1.71						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553519	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553519&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608176	469797383							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167280	CNC(=O)c1ccc(cc1F)-c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)F)c(cc1F)N1C[C@H](C)N(C)[C@H](C)C1			553520	4-(difluoromethyl)-N-[4- fluoro-5-[3-fluoro-4- (methylcarbamoyl)phenyl]- 2-[rac-(3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-6-oxo-1H- pyridine-3-carboxamide::US11319299, Example 605	WD repeat-containing protein 5				 0.600						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553520	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553520&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608177	469797384							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167281	CNC(=O)c1cc(ccc1F)-c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)F)c(cc1F)N1C[C@H](C)N(C)[C@H](C)C1			553521	4-(difluoromethyl)-N-[4- fluoro-5-[4-fluoro-3- (methylcarbamoyl)phenyl]- 2-[rac-(3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-6-oxo-1H- pyridine-3-carboxamide::US11319299, Example 606	WD repeat-containing protein 5				 1.86						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553521	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553521&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608178	469797385							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167282	C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1cn(C)c(=O)cc1C(F)F)-c1cnc(nc1)N1CCOC[C@@H]1C	InChI=1S/C29H34F3N7O3/c1-17-14-38(6-5-36(17)3)25-11-23(30)20(19-12-33-29(34-13-19)39-7-8-42-16-18(39)2)9-24(25)35-28(41)22-15-37(4)26(40)10-21(22)27(31)32/h9-13,15,17-18,27H,5-8,14,16H2,1-4H3,(H,35,41)/t17-,18-/m0/s1	LLGTXXNCAFAYRE-ROUUACIJSA-N	553522	4-(difluoromethyl)-N-[4- fluoro-2-[rac-(3R)-3,4- dimethylpiperazin-1-yl]- 5-[2-[rac-(3R)-3- methylmorpholin-4- yl]pyrimidin-5- yl]phenyl]-1-methyl-6- oxopyridine-3-carboxamide::US11319299, Example 607	WD repeat-containing protein 5				 1.53						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553522	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553522&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138551543	469797386							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167283	C[C@H]1COCCN1c1ncc(cn1)-c1cc(NC(=O)c2cn(C)c(=O)cc2C(F)(F)F)c(cc1F)N1CCN(C)[C@@H](C)C1	InChI=1S/C29H33F4N7O3/c1-17-14-39(6-5-37(17)3)25-11-23(30)20(19-12-34-28(35-13-19)40-7-8-43-16-18(40)2)9-24(25)36-27(42)21-15-38(4)26(41)10-22(21)29(31,32)33/h9-13,15,17-18H,5-8,14,16H2,1-4H3,(H,36,42)/t17-,18-/m0/s1	IUDDJAKLCFILIJ-ROUUACIJSA-N	553523	N-[4-fluoro-2-[rac-(3R)- 3,4-dimethylpiperazin-1- yl]-5-[2-[rac-(3R)-3- methylmorpholin-4- yl]pyrimidin-5- yl]phenyl]-1-methyl-6- oxo-4-(trifluoromethyl) pyridine-3-carboxamide::US11319299, Example 608	WD repeat-containing protein 5				 0.977						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553523	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553523&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138551592	469797387							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167284	C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cccc(F)n1			553524	N-[4-fluoro-5-(6- fluoropyridin-2-yl)-2- [rac-(3R)-3,4- dimethylpiperazin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 609	WD repeat-containing protein 5				 0.774						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553524	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553524&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608179	469797388							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167285	C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cccc(n1)C(F)(F)F			553525	N-[-4-fluoro-2-[rac-(3R)- 3,4-dimethylpiperazin-1- yl]-5-[6-(trifluoromethyl) pyridin-2-yl]phenyl]-6-oxo- 4-(trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 610	WD repeat-containing protein 5				 0.552						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553525	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553525&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608180	469797389							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167286	C[C@H]1CN(CCO1)c1ncc(cn1)-c1cc(NC(=O)c2cc(C)c(F)c(C)c2)c(cc1F)N1C[C@H](C)N(C)[C@H](C)C1	InChI=1S/C31H38F2N6O2/c1-18-9-23(10-19(2)29(18)33)30(40)36-27-11-25(24-13-34-31(35-14-24)38-7-8-41-22(5)17-38)26(32)12-28(27)39-15-20(3)37(6)21(4)16-39/h9-14,20-22H,7-8,15-17H2,1-6H3,(H,36,40)/t20-,21+,22-/m0/s1	GTTCDOFHAWTLKM-BDTNDASRSA-N	553526	4-fluoro-N-[4-fluoro-5- [2-[rac-(2R)-2- methylmorpholin-4- yl]pyrimidin-5-yl]-2-[rac- (3S,5R)-3,4,5- trimethylpiperazin-1- yl]phenyl]-3,5- dimethylbenzamide::US11319299, Example 611	WD repeat-containing protein 5				 1.55						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553526	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553526&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138551704	469797390							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167287	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)F)C1=CCN(C1)C(=O)N1CCCC1			553527	4-(Difluoromethyl)-N-(4- fluoro-5-(1-(pyrrolidine- 1-carbonyl)-2,5-dihydro- 1H-pyrrol-3-yl)-2- ((3S,5R)-3,4,5- trimethylpiperazin-1- yl)phenyl)-6-oxo-1,6- dihydropyridine-3- carboxamide::US11319299, Example 612	WD repeat-containing protein 5				 1.94						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553527	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553527&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608181	469797391							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167288	C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1ccc(F)cc1C(F)(F)F)-c1cnc(nc1)N1CCC(C)(O)CC1	InChI=1S/C30H33F5N6O2/c1-18-17-41(11-10-39(18)3)26-14-24(32)22(19-15-36-28(37-16-19)40-8-6-29(2,43)7-9-40)13-25(26)38-27(42)21-5-4-20(31)12-23(21)30(33,34)35/h4-5,12-16,18,43H,6-11,17H2,1-3H3,(H,38,42)/t18-/m0/s1	FVURXINPUBJJQU-SFHVURJKSA-N	553528	4-fluoro-N-[4-fluoro-5- [2-(4-hydroxy-4- methylpiperidin-1- yl)pyrimidin-5-yl]-2-[rac- (3R)-3,4- dimethylpiperazin-1- yl]phenyl]-2- (trifluoromethyl)benzamide::US11319299, Example 613	WD repeat-containing protein 5				 0.922						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553528	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553528&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138551435	469797392							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167289	C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1ccc(F)cc1C(F)(F)F)-c1ccnc(n1)N1CCOCC1	InChI=1S/C28H29F5N6O2/c1-17-16-39(8-7-37(17)2)25-15-22(30)20(23-5-6-34-27(36-23)38-9-11-41-12-10-38)14-24(25)35-26(40)19-4-3-18(29)13-21(19)28(31,32)33/h3-6,13-15,17H,7-12,16H2,1-2H3,(H,35,40)/t17-/m0/s1	CVFYDFNHNNEKOE-KRWDZBQOSA-N	553529	4-fluoro-N-[4-fluoro-5- (2-morpholin-4- ylpyrimidin-4-yl)-2-[rac- (3R)-3,4- dimethylpiperazin-1- yl]phenyl]-2- (trifluoromethyl)benzamide::US11319299, Example 614	WD repeat-containing protein 5				 0.733						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553529	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553529&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138551504	469797393							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167290	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCCN(C1)c1ncc(s1)C#N			553530	N-[5-[1-(5-cyano-1,3- thiazol-2-yl)-3,6-dihydro- 2H-pyridin-5-yl]-4- fluoro-2-[rac-(3R,5S)- 3,4,5-trimethylpiperazin- 1-yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 615	WD repeat-containing protein 5				 0.375						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553530	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553530&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608182	469797394							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167291	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1csc(n1)N1CCOCC1			553531	N-[4-fluoro-5-(2- morpholin-4-yl-1,3- thiazol-4-yl)-2-[rac- (3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 616	WD repeat-containing protein 5				 0.748						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553531	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553531&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608183	469797395							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167292	C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1csc(n1)N1CCOCC1			553532	N-[4-fluoro-5-(2- morpholin-4-yl-1,3- thiazol-4-yl)-2-[rac-(3R)- 3,4-dimethylpiperazin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 617	WD repeat-containing protein 5				 558000						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553532	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553532&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608184	469797396							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167293	C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cnc(s1)N1CCOCC1			553533	N-[4-fluoro-5-(2-morpholin- 4-yl-1,3-thiazol-5-yl)-2-[rac- (3R)-3,4-dimethylpiperazin- 1-yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 618	WD repeat-containing protein 5				 1.13						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553533	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553533&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608185	469797397							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167294	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cnc(s1)N1CCOCC1			553534	N-[4-fluoro-5-(2- morpholin-4-yl-1,3- thiazol-5-yl)-2-[rac- (3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 619	WD repeat-containing protein 5				 0.948						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553534	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553534&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608186	469797398							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167295	C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1cn(C)c(=O)cc1C(F)F)-c1csc(n1)N1CCOCC1	InChI=1S/C27H31F3N6O3S/c1-16-13-36(5-4-33(16)2)23-12-20(28)18(22-15-40-27(32-22)35-6-8-39-9-7-35)10-21(23)31-26(38)19-14-34(3)24(37)11-17(19)25(29)30/h10-12,14-16,25H,4-9,13H2,1-3H3,(H,31,38)/t16-/m0/s1	WFABOJKYQGFVRX-INIZCTEOSA-N	553535	4-(difluoromethyl)-N-[4- fluoro-5-(2-morpholin-4- yl-1,3-thiazol-4-yl)-2- [rac-(3R)-3,4- dimethylpiperazin-1- yl]phenyl]-1-methyl-6- oxopyridine-3-carboxamide::US11319299, Example 620	WD repeat-containing protein 5				 4.19						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553535	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553535&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138551538	469797399							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167296	C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1cn(C)c(=O)cc1C(F)F)-c1cnc(s1)N1CCOCC1	InChI=1S/C27H31F3N6O3S/c1-16-14-36(5-4-33(16)2)22-12-20(28)18(23-13-31-27(40-23)35-6-8-39-9-7-35)10-21(22)32-26(38)19-15-34(3)24(37)11-17(19)25(29)30/h10-13,15-16,25H,4-9,14H2,1-3H3,(H,32,38)/t16-/m0/s1	XMZRSQJISAITCD-INIZCTEOSA-N	553536	4-(difluoromethyl)-N-[4- fluoro-5-(2-morpholin-4- yl-1,3-thiazol-5-yl)-2- [rac-(3R)-3,4- dimethylpiperazin-1- yl]phenyl]-1-methyl-6- oxopyridine-3- carboxamide::US11319299, Example 621	WD repeat-containing protein 5				 4.84						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553536	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553536&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138551620	469797400							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167297	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1cn(C)c(=O)cc1C(F)F)-c1csc(n1)N1CCOCC1	InChI=1S/C28H33F3N6O3S/c1-16-12-37(13-17(2)35(16)4)24-11-21(29)19(23-15-41-28(33-23)36-5-7-40-8-6-36)9-22(24)32-27(39)20-14-34(3)25(38)10-18(20)26(30)31/h9-11,14-17,26H,5-8,12-13H2,1-4H3,(H,32,39)/t16-,17+	JLRJKTXPSSWJBZ-CALCHBBNSA-N	553537	4-(difluoromethyl)-N-[4- fluoro-5-(2-morpholin-4- yl-1,3-thiazol-4-yl)-2- [rac-(3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-1-methyl-6- oxopyridine-3- carboxamide::US11319299, Example 622	WD repeat-containing protein 5				 5.15						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553537	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553537&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138541795	469797401							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167298	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1cn(C)c(=O)cc1C(F)F)-c1cnc(s1)N1CCOCC1	InChI=1S/C28H33F3N6O3S/c1-16-13-37(14-17(2)35(16)4)23-11-21(29)19(24-12-32-28(41-24)36-5-7-40-8-6-36)9-22(23)33-27(39)20-15-34(3)25(38)10-18(20)26(30)31/h9-12,15-17,26H,5-8,13-14H2,1-4H3,(H,33,39)/t16-,17+	FRVACQLTROJXIT-CALCHBBNSA-N	553538	4-(difluoromethyl)-N-[4- fluoro-5-(2-morpholin-4- yl-1,3-thiazol-5-yl)-2- [rac-(3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-1-methyl-6- oxopyridine-3-carboxamide::US11319299, Example 623	WD repeat-containing protein 5				 5.57						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553538	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553538&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138541743	469797402							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167299	C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1ccc(F)cc1C(F)(F)F)-c1cc(C(=O)NC(C)(C)CC(C)(C)C)c(F)cc1F	InChI=1S/C35H39F7N4O2/c1-19-17-46(11-10-45(19)7)30-16-28(39)23(14-29(30)43-31(47)21-9-8-20(36)12-25(21)35(40,41)42)22-13-24(27(38)15-26(22)37)32(48)44-34(5,6)18-33(2,3)4/h8-9,12-16,19H,10-11,17-18H2,1-7H3,(H,43,47)(H,44,48)/t19-/m0/s1	SDQHUFLHQPNFLC-IBGZPJMESA-N	553539	2,4-difluoro-5-[2-fluoro- 5-[[4-fluoro-2- (trifluoromethyl)benzoyl] amino]-4-[rac-(3R)-3,4- dimethylpiperazin-1- yl]phenyl]-N-(2,4,4- trimethylpentan-2- yl)benzamide::US11319299, Example 625	WD repeat-containing protein 5				 172						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553539	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553539&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138551410	469797403							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167300	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cc(C(=O)NC(C)(C)CC(C)(C)C)c(F)cc1F			553540	N-[5-[2,4-difluoro-5- (2,4,4-trimethylpentan-2- ylcarbamoyl)phenyl]-4- fluoro-2-[rac-(3R,5S)- 3,4,5-trimethylpiperazin- 1-yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 626	WD repeat-containing protein 5				 5.24						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553540	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553540&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608187	469797404							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167301	C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)F)-c1cc(C(=O)NC(C)(C)CC(C)(C)C)c(F)cc1F			553541	4-(difluoromethyl)-N-[5- [2,4-difluoro-5-(2,4,4- trimethylpentan-2- ylcarbamoyl)phenyl]-4- fluoro-2-[rac-(3R,5S)- 3,4,5-trimethylpiperazin- 1-yl]phenyl]-6-oxo-1H- pyridine-3-carboxamide::US11319299, Example 627	WD repeat-containing protein 5				 23.3						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553541	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553541&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608188	469797405							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167302	C[C@H]1COCCN1c1ncc(cn1)-c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)F)c(cc1F)N1CCN(C)[C@@H](C)C1			553444	4-(difluoromethyl)-N-[4- fluoro-5-[2-[rac-(3R)-3- methylmorpholin-4- yl]pyrimidin-5-yl]-2-[rac- (3S,5R)-3,4,5- trimethylpiperazin-1- yl]phenyl]-6-oxo-1H- pyridine-3-carboxamide::US11319299, Example 521::US11319299, Example 628	WD repeat-containing protein 5				 1.25						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553444	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553444&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608128	469797308							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167303	C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)F)C1=CCN(C1)C(=O)N1CCCC1			553543	(S)-4-(Sifluoromethyl)-N- (2-(3,4- dimethylpiperazin-1-yl)- 4-fluoro-5-(1-(pyrrolidine- 1-carbonyl)-2,5-dihydro- 1H-pyrrol-3-yl)phenyl)- 6-oxo-1,6- dihydropyridine-3- carboxamide::US11319299, Example 629	WD repeat-containing protein 5				 2.22						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553543	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553543&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608189	469797406							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167304	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)F)C1=CCN(C1)C(=O)OC1(C)CCC1			553544	1-Methylcyclobutyl 3-(5- (4-(difluoromethyl)-6- oxo-1,6-dihydropyridine- 3-carboxamido)-2-fluoro- 4-((3S,5R)-3,4,5- trimethylpiperazin-1- yl)phenyl)-2,5-dihydro- 1H-pyrrole-1-carboxylate::US11319299, Example 630	WD repeat-containing protein 5				 1.98						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553544	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553544&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608190	469797407							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167305	C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)F)C1=CCN(C1)C(=O)OC1(C)CCC1			553545	1-Methylcyclobutyl (S)- 3-(5-(4-(difluoromethyl)- 6-oxo-1,6-dihydropyridine-3- carboxamido)-4-(3,4- dimethylpiperazin-1-yl)- 2-fluorophenyl)-2,5- dihydro-1H-pyrrole-1- carboxylate::US11319299, Example 631	WD repeat-containing protein 5				 2.65						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553545	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553545&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608191	469797408							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167306	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cc(C(N)=O)c(F)cc1F			553546	N-[5-(5-carbamoyl-2,4- difluorophenyl)-4-fluoro- 2-[rac-(3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 632	WD repeat-containing protein 5				 11.4						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553546	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553546&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608192	469797409							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167307	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)F)-c1cc(C(N)=O)c(F)cc1F			553547	N-[5-(5-carbamoyl-2,4- difluorophenyl)-4-fluoro- 2-[rac-(3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-4- (difluoromethyl)-6-oxo- 1H-pyridine-3-carboxamide::US11319299, Example 633	WD repeat-containing protein 5				 11.9						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553547	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553547&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608193	469797410							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167308	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1ccc(F)cc1C(F)(F)F)-c1cc(C(N)=O)c(F)cc1F	InChI=1S/C28H25F7N4O2/c1-13-11-39(12-14(2)38(13)3)25-10-23(32)18(17-7-19(26(36)40)22(31)9-21(17)30)8-24(25)37-27(41)16-5-4-15(29)6-20(16)28(33,34)35/h4-10,13-14H,11-12H2,1-3H3,(H2,36,40)(H,37,41)/t13-,14+	MHDIYAYCWAPWKU-OKILXGFUSA-N	553548	2,4-difluoro-5-[2-fluoro- 5-[[4-fluoro-2- (trifluoromethyl)benzoyl] amino]-4-[rac-(3R,5S)- 3,4,5-trimethylpiperazin- 1-yl]phenyl]benzamide::US11319299, Example 634	WD repeat-containing protein 5				 69.5						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553548	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553548&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			137377406	469797411							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167309	C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1ccc(F)cc1C(F)(F)F)-c1cc(C(N)=O)c(F)cc1F	InChI=1S/C27H23F7N4O2/c1-13-12-38(6-5-37(13)2)24-11-22(31)17(16-8-18(25(35)39)21(30)10-20(16)29)9-23(24)36-26(40)15-4-3-14(28)7-19(15)27(32,33)34/h3-4,7-11,13H,5-6,12H2,1-2H3,(H2,35,39)(H,36,40)/t13-/m0/s1	DDDNHKGJKKBMHG-ZDUSSCGKSA-N	553549	2,4-difluoro-5-[2-fluoro- 5-[[4-fluoro-2- (trifluoromethyl)benzoyl] amino]-4-[rac-(3R)-3,4- dimethylpiperazin-1- yl]phenyl]benzamide::US11319299, Example 635	WD repeat-containing protein 5				 66.9						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553549	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553549&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138551503	469797412							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167310	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1ccc(F)cc1C(F)(F)F)-c1cnc(nc1)N1CCC(C)(O)CC1	InChI=1S/C31H35F5N6O2/c1-18-16-42(17-19(2)40(18)4)27-13-25(33)23(20-14-37-29(38-15-20)41-9-7-30(3,44)8-10-41)12-26(27)39-28(43)22-6-5-21(32)11-24(22)31(34,35)36/h5-6,11-15,18-19,44H,7-10,16-17H2,1-4H3,(H,39,43)/t18-,19+	XGLNLFUCFFWRFI-KDURUIRLSA-N	553550	4-fluoro-N-[4-fluoro-5- [2-(4-hydroxy-4- methylpiperidin-1- yl)pyrimidin-5-yl]-2-[rac- (3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-2- (trifluoromethyl)benzamide::US11319299, Example 636	WD repeat-containing protein 5				 1.42						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553550	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553550&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			137376762	469797413							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167311	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)F)C1=CCN(C1)C(=O)OC1CC(F)(F)C1			553551	3,3-Difluorocyclobutyl 3- (5-(4-(difluoromethyl)-6- oxo-1,6-dihydropyridine- 3-carboxamido)-2-fluoro- 4-((3S,5R)-3,4,5- trimethylpiperazin-1- yl)phenyl)-2,5-dihydro- 1H-pyrrole-1-carboxylate::US11319299, Example 637	WD repeat-containing protein 5				 2.26						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553551	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553551&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608194	469797414							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167312	C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)F)C1=CCN(C1)C(=O)OC1CC(F)(F)C1			553552	3,3-Difluorocyclobutyl (S)-3-(5-(4- (difluoromethyl)-6-oxo- 1,6-dihydropyridine-3- carboxamido)-4-(3,4- dimethylpiperazin-1-yl)- 2-fluorophenyl)-2,5- dihydro-1H-pyrrole-1- carboxylate::US11319299, Example 638	WD repeat-containing protein 5				 2.27						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553552	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553552&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608195	469797415							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167313	C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)F)C1=CCN(CC1)c1cnc(nc1)C#N			553553	(S)-N-(5-(1-(2- cyanopyrimidin-5-yl)- 1,2,3,6-tetrahydropyridin- 4-yl)-2-(3,4- dimethylpiperazin-1-yl)- 4-fluorophenyl)-4- (difluoromethyl)-6-oxo- 1,6-dihydropyridine-3- carboxamide::US11319299, Example 639	WD repeat-containing protein 5				 4.97						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553553	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553553&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608196	469797416							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167314	C[C@@H]1CN(CCO1)c1ncc(cn1)-c1cc(NC(=O)c2cn(C)c(=O)cc2C(F)(F)F)c(cc1F)N1C[C@H](C)N(C)[C@H](C)C1	InChI=1S/C30H35F4N7O3/c1-17-13-41(14-18(2)39(17)5)26-10-24(31)21(20-11-35-29(36-12-20)40-6-7-44-19(3)15-40)8-25(26)37-28(43)22-16-38(4)27(42)9-23(22)30(32,33)34/h8-12,16-19H,6-7,13-15H2,1-5H3,(H,37,43)/t17-,18+,19-/m1/s1	LGIULJQHFBTTOT-CEXWTWQISA-N	553554	N-[4-fluoro-5-[2-[rac- (2R)-2-methylmorpholin- 4-yl]pyrimidin-5-yl]-2- [rac-(3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-1-methyl-6- oxo-4-(trifluoromethyl) pyridine-3-carboxamide::US11319299, Example 640	WD repeat-containing protein 5				 1.74						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553554	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553554&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138541636	469797417							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167315	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1cn(C)c(=O)cc1C(F)(F)F)-c1cnc(nc1)N1CCC(C)(O)CC1	InChI=1S/C31H37F4N7O3/c1-18-15-42(16-19(2)40(18)5)26-12-24(32)21(20-13-36-29(37-14-20)41-8-6-30(3,45)7-9-41)10-25(26)38-28(44)22-17-39(4)27(43)11-23(22)31(33,34)35/h10-14,17-19,45H,6-9,15-16H2,1-5H3,(H,38,44)/t18-,19+	WSMLVDYZBINLDJ-KDURUIRLSA-N	553555	N-[4-fluoro-5-[2-(4- hydroxy-4-methylpiperidin- 1-yl)pyrimidin-5-yl]-2-[rac- (3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-1-methyl-6- oxo-4-(trifluoromethyl) pyridine-3-carboxamide::US11319299, Example 641	WD repeat-containing protein 5				 1.92						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553555	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553555&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			137377157	469797418							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167316	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCCN(C1)c1nc(cs1)C#N			553556	N-[5-[1-(4-cyano-1,3- thiazol-2-yl)-3,6-dihydro- 2H-pyridin-5-yl]-4- fluoro-2-[rac-(3R,5S)- 3,4,5-trimethylpiperazin- 1-yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 642	WD repeat-containing protein 5				 1.30						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553556	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553556&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608197	469797419							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167317	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCCN(C1)c1ncco1			553557	N-[4-fluoro-5-[1-(1,3- oxazol-2-yl)-3,6-dihydro- 2H-pyridin-5-yl]-2-[rac- (3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 643	WD repeat-containing protein 5				 1.26						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553557	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553557&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608198	469797420							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167318	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCCN(C1)c1ncccn1			553268	N-[4-fluoro-5-(1-pyrimidin-2- yl-3,6-dihydro-2H-pyridin-5-yl)- 2-[rac-(3R,5S)-3,4,5- trimethylpiperazin-1-yl]phenyl]- 6-oxo-4-(trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 334::US11319299, Example 644	WD repeat-containing protein 5				 1.32						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553268	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553268&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608007	469797134							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167319	COc1cnc(nc1)N1CCC=C(C1)c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)F)c(cc1F)N1C[C@H](C)N(C)[C@H](C)C1			553559	4-(difluoromethyl)-N-[4- fluoro-5-[1-(5- methoxypyrimidin-2-yl)- 3,6-dihydro-2H-pyridin- 5-yl]-2-[rac-(3R,5S)- 3,4,5-trimethylpiperazin- 1-yl]phenyl]-6-oxo-1H- pyridine-3-carboxamide::US11319299, Example 645	WD repeat-containing protein 5				 1.41						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553559	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553559&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608199	469797421							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167320	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)F)C1=CCN(CC1)c1ncc(C=O)cn1			553560	4-(difluoromethyl)-N-[4- fluoro-5-[1-(5- formylpyrimidin-2-yl)- 3,6-dihydro-2H-pyridin- 4-yl]-2-[rac-(3R,5S)- 3,4,5-trimethylpiperazin- 1-yl]phenyl]-6-oxo-1H- pyridine-3-carboxamide::US11319299, Example 646	WD repeat-containing protein 5				 1.41						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553560	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553560&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608200	469797422							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167321	COc1cc(ncn1)N1CCC(=CC1)c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)F)c(cc1F)N1C[C@H](C)N(C)[C@H](C)C1			553561	4-(difluoromethyl)-N-[4- fluoro-5-[1-(6- methoxypyrimidin-4-yl)- 3,6-dihydro-2H-pyridin- 4-yl]-2-[rac-(3R,5S)- 3,4,5-trimethylpiperazin- 1-yl]phenyl]-6-oxo-1H- pyridine-3-carboxamide::US11319299, Example 647	WD repeat-containing protein 5				 1.59						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553561	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553561&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608201	469797423							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167322	CCOC(=O)N1CCC=C(C1)c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)F)c(cc1F)N1C[C@H](C)N(C)[C@H](C)C1			553562	US11319299, Example 648::ethyl 5-[5-[[4- ((difluoromethyl)-6-oxo- 1H-pyridine-3- carbonyl]amino]-2- fluoro-4-[rac-(3R,5S)- 3,4,5-trimethylpiperazin- 1-yl]phenyl]-3,6-dihydro- 2H-pyridine-1-carboxylate	WD repeat-containing protein 5				 1.97						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553562	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553562&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608202	469797424							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167323	C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1ccc(F)cc1C(F)(F)F)C1=CCCN(C1)c1ncccn1	InChI=1S/C29H29F5N6O/c1-18-16-39(12-11-38(18)2)26-15-24(31)22(19-5-3-10-40(17-19)28-35-8-4-9-36-28)14-25(26)37-27(41)21-7-6-20(30)13-23(21)29(32,33)34/h4-9,13-15,18H,3,10-12,16-17H2,1-2H3,(H,37,41)/t18-/m0/s1	NDBMEBIYKBQTPR-SFHVURJKSA-N	553563	4-fluoro-N-[4-fluoro-5- (1-pyrimidin-2-yl-3,6- dihydro-2H-pyridin-5-yl)- 2-[rac-(3R)-3,4- dimethylpiperazin-1- yl]phenyl]-2- (trifluoromethyl)benzamide::US11319299, Example 649	WD repeat-containing protein 5				 1.87						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553563	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553563&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138551498	469797425							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167324	C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1ccc(F)cc1C(F)(F)F)C1=CCCN(C1)c1ncc(C=O)cn1	InChI=1S/C30H29F5N6O2/c1-18-15-40(9-8-39(18)2)27-12-25(32)23(20-4-3-7-41(16-20)29-36-13-19(17-42)14-37-29)11-26(27)38-28(43)22-6-5-21(31)10-24(22)30(33,34)35/h4-6,10-14,17-18H,3,7-9,15-16H2,1-2H3,(H,38,43)/t18-/m0/s1	SWYOOGSBHDBRPO-SFHVURJKSA-N	553564	4-fluoro-N-[4-fluoro-5- [1-(5-formylpyrimidin-2- yl)-3,6-dihydro-2H- pyridin-5-yl]-2-[rac-(3R)- 3,4-dimethylpiperazin-1- yl]phenyl]-2- (trifluoromethyl)benzamide::US11319299, Example 650	WD repeat-containing protein 5				 5.18						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553564	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553564&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138551556	469797426							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167325	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)F)C1=CCN(CC1)C(=O)OC1(C)CCC1			553565	(1-methylcyclobutyl) 4- [5-[[4-(difluoromethyl)-6- oxo-1H-pyridine-3- carbonyl]amino]-2- fluoro-4-[rac-(3R,5S)- 3,4,5-trimethylpiperazin- 1-yl]phenyl]-3,6-dihydro- 2H-pyridine-1-carboxylate::US11319299, Example 651	WD repeat-containing protein 5				 0.897						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553565	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553565&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608203	469797427							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167326	C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1cn(C)c(=O)cc1C(F)F)-c1ccc(C(N)=O)c(F)c1	InChI=1S/C27H27F4N5O3/c1-14-12-36(7-6-34(14)2)23-11-21(29)17(15-4-5-16(26(32)38)20(28)8-15)9-22(23)33-27(39)19-13-35(3)24(37)10-18(19)25(30)31/h4-5,8-11,13-14,25H,6-7,12H2,1-3H3,(H2,32,38)(H,33,39)/t14-/m0/s1	OQWKUYHMUPOMGP-AWEZNQCLSA-N	553566	N-[5-(4-carbamoyl-3- fluorophenyl)-4-fluoro-2- [rac-(3R)-3,4- dimethylpiperazin-1- yl]phenyl]-4- (difluoromethyl)-1- methyl-6-oxopyridine-3- carboxamide::US11319299, Example 652	WD repeat-containing protein 5				 5.29						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553566	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553566&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138551605	469797428							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167327	CNC(=O)c1ccc(cc1F)-c1cc(NC(=O)c2cn(C)c(=O)cc2C(F)F)c(cc1F)N1CCN(C)[C@@H](C)C1	InChI=1S/C28H29F4N5O3/c1-15-13-37(8-7-35(15)3)24-12-22(30)18(16-5-6-17(21(29)9-16)27(39)33-2)10-23(24)34-28(40)20-14-36(4)25(38)11-19(20)26(31)32/h5-6,9-12,14-15,26H,7-8,13H2,1-4H3,(H,33,39)(H,34,40)/t15-/m0/s1	VRZYCPJNWZMXJL-HNNXBMFYSA-N	553567	4-(difluoromethyl)-N-[4- fluoro-5-[3-fluoro-4- (methylcarbamoyl)phenyl]- 2-[rac-(3R)-3,4- dimethylpiperazin-1- yl]phenyl]-1-methyl-6- oxopyridine-3-carboxamide::US11319299, Example 653	WD repeat-containing protein 5				 3.43						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553567	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553567&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138551550	469797429							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167328	C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1ccc(F)cc1C(F)F)-c1ccnc(n1)N1CCOCC1	InChI=1S/C28H30F4N6O2/c1-17-16-38(8-7-36(17)2)25-15-22(30)21(23-5-6-33-28(35-23)37-9-11-40-12-10-37)14-24(25)34-27(39)19-4-3-18(29)13-20(19)26(31)32/h3-6,13-15,17,26H,7-12,16H2,1-2H3,(H,34,39)/t17-/m0/s1	WJENCDAKRUHLEZ-KRWDZBQOSA-N	553568	2-(difluoromethyl)-4- fluoro-N-[4-fluoro-5-(2- morpholin-4-ylpyrimidin- 4-yl)-2-[rac-(3R)-3,4- dimethylpiperazin-1- yl]phenyl]benzamide::US11319299, Example 655	WD repeat-containing protein 5				 1.06						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553568	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553568&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138551510	469797430							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167329	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1ccc(F)cc1C(F)(F)F)-c1cc(F)c(C(N)=O)c(F)c1	InChI=1S/C28H25F7N4O2/c1-13-11-39(12-14(2)38(13)3)24-10-20(30)18(15-6-21(31)25(26(36)40)22(32)7-15)9-23(24)37-27(41)17-5-4-16(29)8-19(17)28(33,34)35/h4-10,13-14H,11-12H2,1-3H3,(H2,36,40)(H,37,41)/t13-,14+	KUHYFJZINUKCCY-OKILXGFUSA-N	553569	2,6-difluoro-4-[2-fluoro- 5-[[4-fluoro-2- (trifluoromethyl)benzoyl] amino]-4-[rac-(3R,5S)- 3,4,5-trimethylpiperazin- 1-yl]phenyl]benzamide::US11319299, Example 656	WD repeat-containing protein 5				 5.44						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553569	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553569&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			137376755	469797431							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167330	C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1ccc(F)cc1C(F)(F)F)-c1cc(F)c(C(N)=O)c(F)c1	InChI=1S/C27H23F7N4O2/c1-13-12-38(6-5-37(13)2)23-11-19(29)17(14-7-20(30)24(25(35)39)21(31)8-14)10-22(23)36-26(40)16-4-3-15(28)9-18(16)27(32,33)34/h3-4,7-11,13H,5-6,12H2,1-2H3,(H2,35,39)(H,36,40)/t13-/m0/s1	RWYZRWUXIQDFEC-ZDUSSCGKSA-N	553570	2,6-difluoro-4-[2-fluoro- 5-[[4-fluoro-2- (trifluoromethyl)benzoyl] amino]-4-[rac-(3R)-3,4- dimethylpiperazin-1- yl]phenyl]benzamide::US11319299, Example 657	WD repeat-containing protein 5				 4.69						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553570	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553570&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138551635	469797432							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167331	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cc(F)c(C(N)=O)c(F)c1			553571	N-[5-(4-carbamoyl-3,5- difluorophenyl)-4-fluoro- 2-[rac-(3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 658	WD repeat-containing protein 5				 1.88						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553571	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553571&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608204	469797433							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167332	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)F)-c1cc(F)c(C(N)=O)c(F)c1			553572	N-[5-(4-carbamoyl-3,5- difluorophenyl)-4-fluoro- 2-[rac-(3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-4- (difluoromethyl)-6-oxo- 1H-pyridine-3-carboxamide::US11319299, Example 659	WD repeat-containing protein 5				 1.93						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553572	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553572&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608205	469797434							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167333	C[C@H]1CN(CCO1)c1nccc(n1)-c1cc(NC(=O)c2ccc(F)cc2C(F)(F)F)c(cc1F)N1CCN(C)[C@@H](C)C1	InChI=1S/C29H31F5N6O2/c1-17-15-39(9-8-38(17)3)26-14-23(31)21(24-6-7-35-28(37-24)40-10-11-42-18(2)16-40)13-25(26)36-27(41)20-5-4-19(30)12-22(20)29(32,33)34/h4-7,12-14,17-18H,8-11,15-16H2,1-3H3,(H,36,41)/t17-,18-/m0/s1	SVTZVEIUYZSBTJ-ROUUACIJSA-N	553573	4-fluoro-N-[4-fluoro-2- [rac-(3R)-3,4- dimethylpiperazin-1-yl]-5- [2-[rac-(3R)-3- methylmorpholin-4- yl]pyrimidin-5-yl]phenyl]- 2-(trifluoromethyl)benzamide::US11319299, Example 660	WD repeat-containing protein 5				 0.290						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553573	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553573&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138551409	469797435							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167334	CC(C)N1CCN(CC1)c1ncc(cn1)-c1cc(NC(=O)c2cn(C)c(=O)cc2C(F)(F)F)c(cc1F)N1C[C@H](C)N(C)[C@H](C)C1	InChI=1S/C32H40F4N8O2/c1-19(2)42-7-9-43(10-8-42)31-37-14-22(15-38-31)23-11-27(28(13-26(23)33)44-16-20(3)41(6)21(4)17-44)39-30(46)24-18-40(5)29(45)12-25(24)32(34,35)36/h11-15,18-21H,7-10,16-17H2,1-6H3,(H,39,46)/t20-,21+	LVPOPXOSFNEIJZ-OYRHEFFESA-N	553574	N-[4-fluoro-5-[2-(4- propan-2-ylpiperazin-1- yl)pyrimidin-5-yl]-2-[rac- (3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-1-methyl-6- oxo-4-(trifluoromethyl) pyridine-3-carboxamide::US11319299, Example 661	WD repeat-containing protein 5				 3.23						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553574	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553574&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			137376831	469797436							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167335	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1cn(C)c(=O)cc1C(F)(F)F)-c1cnc(nc1)N1CCOC(C)(C)C1	InChI=1S/C31H37F4N7O3/c1-18-14-42(15-19(2)40(18)6)26-11-24(32)21(20-12-36-29(37-13-20)41-7-8-45-30(3,4)17-41)9-25(26)38-28(44)22-16-39(5)27(43)10-23(22)31(33,34)35/h9-13,16,18-19H,7-8,14-15,17H2,1-6H3,(H,38,44)/t18-,19+	BNYMXOIMQOEKAG-KDURUIRLSA-N	553575	N-[5-[2-(2,2- dimethylmorpholin-4- yl)pyrimidin-5-yl]-4- fluoro-2-[rac-(3R,5S)- 3,4,5-trimethylpiperazin-1- yl]phenyl]-1-methyl-6- oxo-4-(trifluoromethyl) pyridine-3-carboxamide::US11319299, Example 662	WD repeat-containing protein 5				 2.29						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553575	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553575&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138541741	469797437							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167336	C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1cn(C)c(=O)cc1C(F)(F)F)-c1ccnc(n1)N1CCOCC1	InChI=1S/C28H31F4N7O3/c1-17-15-39(7-6-36(17)2)24-14-21(29)18(22-4-5-33-27(35-22)38-8-10-42-11-9-38)12-23(24)34-26(41)19-16-37(3)25(40)13-20(19)28(30,31)32/h4-5,12-14,16-17H,6-11,15H2,1-3H3,(H,34,41)/t17-/m0/s1	CNVUXKCKLCZWJO-KRWDZBQOSA-N	553576	N-[4-fluoro-5-(2- morpholin-4-ylpyrimidin- 4-yl)-2-[rac-(3R)-3,4- dimethylpiperazin-1- yl]phenyl]-1-methyl-6- oxo-4-(trifluoromethyl) pyridine-3-carboxamide::US11319299, Example 663	WD repeat-containing protein 5				 2.50						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553576	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553576&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138551637	469797438							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167337	C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1cn(C)c(=O)cc1C(F)F)-c1ccnc(n1)N1CCOCC1	InChI=1S/C28H32F3N7O3/c1-17-15-38(7-6-35(17)2)24-14-21(29)19(22-4-5-32-28(34-22)37-8-10-41-11-9-37)12-23(24)33-27(40)20-16-36(3)25(39)13-18(20)26(30)31/h4-5,12-14,16-17,26H,6-11,15H2,1-3H3,(H,33,40)/t17-/m0/s1	DMASMZSAJVGUFG-KRWDZBQOSA-N	553577	4-(difluoromethyl)-N-[4- fluoro-5-(2-morpholin-4- ylpyrimidin-4-yl)-2-[rac- (3R)-3,4- dimethylpiperazin-1- yl]phenyl]-1-methyl-6- oxopyridine-3-carboxamide::US11319299, Example 664	WD repeat-containing protein 5				 2.68						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553577	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553577&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138551413	469797439							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167338	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1ccc(F)cc1C(F)(F)F)-c1ccc(C(=O)NC(C)(C)CC(C)(C)C)c(F)c1F	InChI=1S/C36H41F7N4O2/c1-19-16-47(17-20(2)46(19)8)29-15-27(38)25(14-28(29)44-32(48)23-10-9-21(37)13-26(23)36(41,42)43)22-11-12-24(31(40)30(22)39)33(49)45-35(6,7)18-34(3,4)5/h9-15,19-20H,16-18H2,1-8H3,(H,44,48)(H,45,49)/t19-,20+	LZCDZZIVYHQEBO-BGYRXZFFSA-N	553578	2,3-difluoro-4-[2-fluoro- 5-[[4-fluoro-2- (trifluoromethyl)benzoyl] amino]-4-[rac-(3R,5S)- 3,4,5-trimethylpiperazin- 1-yl]phenyl]-N-(2,4,4- trimethylpentan-2- yl)benzamide::US11319299, Example 665	WD repeat-containing protein 5				 151						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553578	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553578&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138541600	469797440							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167339	C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1ccc(F)cc1C(F)(F)F)-c1ccc(C(=O)NC(C)(C)CC(C)(C)C)c(F)c1F	InChI=1S/C35H39F7N4O2/c1-19-17-46(13-12-45(19)7)28-16-26(37)24(15-27(28)43-31(47)22-9-8-20(36)14-25(22)35(40,41)42)21-10-11-23(30(39)29(21)38)32(48)44-34(5,6)18-33(2,3)4/h8-11,14-16,19H,12-13,17-18H2,1-7H3,(H,43,47)(H,44,48)/t19-/m0/s1	ZIECMLNHYHKEON-IBGZPJMESA-N	553579	2,3-difluoro-4-[2-fluoro- 5-[[4-fluoro-2- (trifluoromethyl)benzoyl] amino]-4-[rac-(3R)-3,4- dimethylpiperazin-1- yl]phenyl]-N-(2,4,4- trimethylpentan-2- yl)benzamide::US11319299, Example 666	WD repeat-containing protein 5				 117						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553579	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553579&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138551551	469797441							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167340	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1ccc(F)cc1C(F)(F)F)-c1ccc(C(N)=O)c(F)c1F	InChI=1S/C28H25F7N4O2/c1-13-11-39(12-14(2)38(13)3)23-10-21(30)19(16-6-7-18(26(36)40)25(32)24(16)31)9-22(23)37-27(41)17-5-4-15(29)8-20(17)28(33,34)35/h4-10,13-14H,11-12H2,1-3H3,(H2,36,40)(H,37,41)/t13-,14+	VQEMKXJSIRMEOQ-OKILXGFUSA-N	553580	2,3-difluoro-4-[2-fluoro- 5-[[4-fluoro-2- (trifluoromethyl)benzoyl] amino]-4-[rac-(3R,5S)- 3,4,5-trimethylpiperazin- 1-yl]phenyl]benzamide::US11319299, Example 667	WD repeat-containing protein 5				 9.65						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553580	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553580&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			137376799	469797442							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167341	C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1ccc(F)cc1C(F)(F)F)-c1ccc(C(N)=O)c(F)c1F	InChI=1S/C27H23F7N4O2/c1-13-12-38(8-7-37(13)2)22-11-20(29)18(15-5-6-17(25(35)39)24(31)23(15)30)10-21(22)36-26(40)16-4-3-14(28)9-19(16)27(32,33)34/h3-6,9-11,13H,7-8,12H2,1-2H3,(H2,35,39)(H,36,40)/t13-/m0/s1	UZTVZBZQXJSLHV-ZDUSSCGKSA-N	553581	2,3-difluoro-4-[2-fluoro- 5-[[4-fluoro-2- (trifluoromethyl)benzoyl] amino]-4-[rac-(3R)-3,4- dimethylpiperazin-1- yl]phenyl]benzamide::US11319299, Example 668	WD repeat-containing protein 5				 18.3						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553581	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553581&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138551397	469797443							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167342	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(C(=O)NC(C)(C)CC(C)(C)C)c(F)c1F			553582	N-[5-[2,3-difluoro-4- (2,4,4-trimethylpentan-2- ylcarbamoyl)phenyl]-4- fluoro-2-[rac-(3R,5S)- 3,4,5-trimethylpiperazin- 1-yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 669	WD repeat-containing protein 5				 9.71						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553582	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553582&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608206	469797444							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167343	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(C(N)=O)c(F)c1F			553583	N-[5-(4-carbamoyl-2,3- difluorophenyl)-4-fluoro- 2-[rac-(3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 670	WD repeat-containing protein 5				 3.85						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553583	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553583&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608207	469797445							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167344	C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1cn(C)c(=O)cc1C(F)(F)F)-c1cccc(n1)N1CCOCC1	InChI=1S/C29H32F4N6O3/c1-18-16-39(8-7-36(18)2)25-15-22(30)19(23-5-4-6-26(34-23)38-9-11-42-12-10-38)13-24(25)35-28(41)20-17-37(3)27(40)14-21(20)29(31,32)33/h4-6,13-15,17-18H,7-12,16H2,1-3H3,(H,35,41)/t18-/m0/s1	NEZSOVSCMFBPEB-SFHVURJKSA-N	553584	N-[4-fluoro-5-(6- morpholin-4-ylpyridin-2- yl)-2-[rac-(3R)-3,4- dimethylpiperazin-1- yl]phenyl]-1-methyl-6- oxo-4-(trifluoromethyl) pyridine-3-carboxamide::US11319299, Example 671	WD repeat-containing protein 5				 4.42						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553584	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553584&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138551505	469797446							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167345	C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1cn(C)c(=O)cc1C(F)F)-c1cccc(n1)N1CCOCC1	InChI=1S/C29H33F3N6O3/c1-18-16-38(8-7-35(18)2)25-15-22(30)20(23-5-4-6-26(33-23)37-9-11-41-12-10-37)13-24(25)34-29(40)21-17-36(3)27(39)14-19(21)28(31)32/h4-6,13-15,17-18,28H,7-12,16H2,1-3H3,(H,34,40)/t18-/m0/s1	NYCSQXJDHCCERG-SFHVURJKSA-N	553585	4-(difluoromethyl)-N-[4- fluoro-5-(6-morpholin-4- ylpyridin-2-yl)-2-[rac- (3R)-3,4-dimethylpiperazin- 1-yl]phenyl]-1-methyl-6- oxopyridine-3-carboxamide::US11319299, Example 672	WD repeat-containing protein 5				 5.02						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553585	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553585&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138551709	469797447							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167346	C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1ccc(F)cc1C(F)(F)F)-c1cccc(n1)N1CCOCC1	InChI=1S/C29H30F5N5O2/c1-18-17-39(9-8-37(18)2)26-16-23(31)21(24-4-3-5-27(35-24)38-10-12-41-13-11-38)15-25(26)36-28(40)20-7-6-19(30)14-22(20)29(32,33)34/h3-7,14-16,18H,8-13,17H2,1-2H3,(H,36,40)/t18-/m0/s1	MEGOJCORCRBAMD-SFHVURJKSA-N	553586	4-fluoro-N-[4-fluoro-5-(6- morpholin-4-ylpyridin-2- yl)-2-[rac-(3R)-3,4- dimethylpiperazin-1- yl]phenyl]-2- (trifluoromethyl)benzamide::US11319299, Example 673	WD repeat-containing protein 5				 3.18						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553586	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553586&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138551418	469797448							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167347	CC(C)OC(=O)N1CCC=C(CC1)c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)(F)F)c(cc1F)N1C[C@H](C)N(C)[C@H](C)C1			553587	US11319299, Example 674::propan-2-yl 4-[2-fluoro- 5-[[6-oxo-4-(trifluoromethyl)- 1H-pyridine-3- carbonyl]amino]-4-[rac- (3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-2,3,6,7- tetrahydroazepine-1- carboxylate	WD repeat-containing protein 5				 4.94						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553587	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553587&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608208	469797449							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167348	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc2n(C)cnc2c1			553588	N-[4-fluoro-5-(1- methylbenzimidazol-5- yl)-2-[rac-(3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 675	WD repeat-containing protein 5				 1.97						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553588	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553588&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608209	469797450							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167349	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc2ncn(C)c2c1			553589	N-[4-fluoro-5-(3- methylbenzimidazol-5- yl)-2-[rac-(3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 676	WD repeat-containing protein 5				 4.39						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553589	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553589&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608210	469797451							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167350	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cccc2scnc12			553590	N-[5-(1,3-benzothiazol-4- yl)-4-fluoro-2-[rac- (3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 677	WD repeat-containing protein 5				 5.29						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553590	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553590&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608211	469797452							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167351	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc2scnc2c1			553591	N-[5-(1,3-benzothiazol-5- yl)-4-fluoro-2-[rac- (3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 678	WD repeat-containing protein 5				 3.26						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553591	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553591&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608212	469797453							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167352	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc2ncsc2c1			553592	N-[5-(1,3-benzothiazol-6- yl)-4-fluoro-2-[rac- (3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 679	WD repeat-containing protein 5				 2.97						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553592	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553592&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608213	469797454							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167353	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1cn(C)c(=O)cc1C(F)F)-c1ccc2n(C)cnc2c1	InChI=1S/C29H31F3N6O2/c1-16-12-38(13-17(2)37(16)5)26-11-22(30)19(18-6-7-25-23(8-18)33-15-36(25)4)9-24(26)34-29(40)21-14-35(3)27(39)10-20(21)28(31)32/h6-11,14-17,28H,12-13H2,1-5H3,(H,34,40)/t16-,17+	BRPUXYOFGUISKQ-CALCHBBNSA-N	553593	4-(difluoromethyl)-N-[4- fluoro-5-(1- methylbenzimidazol-5- yl)-2-[rac-(3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-1-methyl-6- oxopyridine-3-carboxamide::US11319299, Example 680	WD repeat-containing protein 5				 58.2						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553593	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553593&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138541620	469797455							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167354	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1cn(C)c(=O)cc1C(F)F)-c1ccc2ncn(C)c2c1	InChI=1S/C29H31F3N6O2/c1-16-12-38(13-17(2)37(16)5)26-11-22(30)19(18-6-7-23-25(8-18)36(4)15-33-23)9-24(26)34-29(40)21-14-35(3)27(39)10-20(21)28(31)32/h6-11,14-17,28H,12-13H2,1-5H3,(H,34,40)/t16-,17+	FOCBALIXURLRRG-CALCHBBNSA-N	553594	4-(difluoromethyl)-N-[4- fluoro-5-(3- methylbenzimidazol-5- yl)-2-[rac-(3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-1-methyl-6- oxopyridine-3-carboxamide::US11319299, Example 681	WD repeat-containing protein 5				 39.3						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553594	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553594&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138541615	469797456							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167355	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1cn(C)c(=O)cc1C(F)F)-c1cccc2scnc12	InChI=1S/C28H28F3N5O2S/c1-15-11-36(12-16(2)35(15)4)23-10-21(29)18(17-6-5-7-24-26(17)32-14-39-24)8-22(23)33-28(38)20-13-34(3)25(37)9-19(20)27(30)31/h5-10,13-16,27H,11-12H2,1-4H3,(H,33,38)/t15-,16+	FZARTRWQXUZUKL-IYBDPMFKSA-N	553595	N-[5-(1,3-benzothiazol-4- yl)-4-fluoro-2-[rac- (3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-4- (difluoromethyl)-1- methyl-6-oxopyridine-3- carboxamide::US11319299, Example 682	WD repeat-containing protein 5				 20.4						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553595	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553595&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			137377100	469797457							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167356	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1cn(C)c(=O)cc1C(F)F)-c1ccc2scnc2c1	InChI=1S/C28H28F3N5O2S/c1-15-11-36(12-16(2)35(15)4)24-10-21(29)18(17-5-6-25-23(7-17)32-14-39-25)8-22(24)33-28(38)20-13-34(3)26(37)9-19(20)27(30)31/h5-10,13-16,27H,11-12H2,1-4H3,(H,33,38)/t15-,16+	KTJMDQNIBQYZPW-IYBDPMFKSA-N	553596	N-[5-(1,3-benzothiazol-5- yl)-4-fluoro-2-[rac- (3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-4- (difluoromethyl)-1- methyl-6-oxopyridine-3- carboxamide::US11319299, Example 683	WD repeat-containing protein 5				 12.3						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553596	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553596&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			137377237	469797458							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167357	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1cn(C)c(=O)cc1C(F)F)-c1ccc2ncsc2c1	InChI=1S/C28H28F3N5O2S/c1-15-11-36(12-16(2)35(15)4)24-10-21(29)18(17-5-6-22-25(7-17)39-14-32-22)8-23(24)33-28(38)20-13-34(3)26(37)9-19(20)27(30)31/h5-10,13-16,27H,11-12H2,1-4H3,(H,33,38)/t15-,16+	QXFVWTNXGFVXME-IYBDPMFKSA-N	553597	N-[5-(1,3-benzothiazol-6- yl)-4-fluoro-2-[rac- (3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-4- (difluoromethyl)-1- methyl-6-oxopyridine-3- carboxamide::US11319299, Example 684	WD repeat-containing protein 5				 7.82						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553597	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553597&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			137376826	469797459							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167358	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)F)C1=CCN(CC1)c1ncc(s1)C#N			553598	N-[5-[1-(5-cyano-1,3- thiazol-2-yl)-3,6-dihydro- 2H-pyridin-4-yl]-4- fluoro-2-[rac-(3R,5S)- 3,4,5-trimethylpiperazin- 1-yl]phenyl]-4- (difluoromethyl)-6-oxo- 1H-pyridine-3-carboxamide::US11319299, Example 685	WD repeat-containing protein 5				 2.23						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553598	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553598&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608214	469797460							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167359	C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)F)C1=CCN(CC1)c1ncc(s1)C#N			553599	N-[5-[1-(5-cyano-1,3- thiazol-2-yl)-3,6-dihydro- 2H-pyridin-4-yl]-4- fluoro-2-[rac-(3R)-3,4- dimethylpiperazin-1- yl]phenyl]-4- (difluoromethyl)-6-oxo- 1H-pyridine-3-carboxamide::US11319299, Example 686	WD repeat-containing protein 5				 1.99						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553599	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553599&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608215	469797461							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167360	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)F)C1=CCCN(C1)c1ncc(s1)C#N			553600	N-[5-[1-(5-cyano-1,3- thiazol-2-yl)-3,6-dihydro- 2H-pyridin-5-yl]-4- fluoro-2-[rac-(3R,5S)- 3,4,5-trimethylpiperazin- 1-yl]phenyl]-4- (difluoromethyl)-6-oxo- 1H-pyridine-3- carboxamide::US11319299, Example 687	WD repeat-containing protein 5				 1.84						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553600	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553600&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608216	469797462							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167361	C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)F)C1=CCCN(C1)c1ncc(s1)C#N			553601	N-[5-[1-(5-cyano-1,3- thiazol-2-yl)-3,6-dihydro- 2H-pyridin-5-yl]-4- fluoro-2-[rac-(3R)-3,4- dimethylpiperazin-1- yl]phenyl]-4- (difluoromethyl)-6-oxo- 1H-pyridine-3- carboxamide::US11319299, Example 688	WD repeat-containing protein 5				 2.49						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553601	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553601&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608217	469797463							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167362	C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1ccc(F)cc1C(F)(F)F)C1=CCCN(C1)c1ncc(s1)C#N	InChI=1S/C29H27F5N6OS/c1-17-15-39(9-8-38(17)2)26-12-24(31)22(18-4-3-7-40(16-18)28-36-14-20(13-35)42-28)11-25(26)37-27(41)21-6-5-19(30)10-23(21)29(32,33)34/h4-6,10-12,14,17H,3,7-9,15-16H2,1-2H3,(H,37,41)/t17-/m0/s1	TWYJGPSUHHTCJT-KRWDZBQOSA-N	553602	N-[5-[1-(5-cyano-1,3- thiazol-2-yl)-3,6-dihydro- 2H-pyridin-5-yl]-4-fluoro- 2-[rac-(3R)-3,4- dimethylpiperazin-1- yl]phenyl]-4-fluoro-2- (trifluoromethyl)benzamide::US11319299, Example 689	WD repeat-containing protein 5				 6.28						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553602	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553602&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138551708	469797464							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167363	C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCN(CC1)c1ncc(s1)C#N			553603	N-[5-[1-(5-cyano-1,3- diazol-2-yl)-3,6-dihydro- 2H-pyridin-4-yl]-4-fluoro- 2-[rac-(3R)-3,4- dimethylpiperazin-1- yl]phenyl]-4-fluoro-2- (trifluoromethyl)benzamide::US11319299, Example 690	WD repeat-containing protein 5				 4.17						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553603	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553603&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608218	469797465							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167364	C[C@@H]1CN(CCO1)c1nccc(n1)-c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)(F)F)c(cc1F)N1C[C@H](C)N(C)[C@H](C)C1			553604	N-[4-fluoro-5-[2-[rac- (2R)-2-methylmorpholin- 4-yl]pyrimidin-4-yl]-2- [rac-(3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 691	WD repeat-containing protein 5				 1.31						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553604	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553604&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608219	469797466							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167365	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)F)-c1ccnc(n1)N1CCOCC1			553605	4-(difluoromethyl)-N-[4- fluoro-5-(2-morpholin-4- ylpyrimidin-4-yl)-2-[rac- (3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-6-oxo-1H- pyridine-3-carboxamide::US11319299, Example 692	WD repeat-containing protein 5				 2.40						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553605	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553605&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608220	469797467							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167366	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1cn(C)c(=O)cc1C(F)(F)F)-c1ccnc(n1)N1CCOCC1	InChI=1S/C29H33F4N7O3/c1-17-14-40(15-18(2)38(17)4)25-13-22(30)19(23-5-6-34-28(36-23)39-7-9-43-10-8-39)11-24(25)35-27(42)20-16-37(3)26(41)12-21(20)29(31,32)33/h5-6,11-13,16-18H,7-10,14-15H2,1-4H3,(H,35,42)/t17-,18+	QGUKAPKZYAOCAM-HDICACEKSA-N	553606	N-[4-fluoro-5-(2- morpholin-4-ylpyrimidin- 4-yl)-2-[rac-(3R,5S)- 3,4,5-trimethylpiperazin- 1-yl]phenyl]-1-methyl-6- oxo-4- (trifluoromethyl)pyridine- 3-carboxamide::US11319299, Example 693	WD repeat-containing protein 5				 4.79						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553606	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553606&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			137377181	469797468							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167367	C[C@H]1CN(CCO1)c1nccc(n1)-c1cc(NC(=O)c2cn(C)c(=O)cc2C(F)(F)F)c(cc1F)N1C[C@H](C)N(C)[C@H](C)C1	InChI=1S/C30H35F4N7O3/c1-17-13-41(14-18(2)39(17)5)26-12-23(31)20(24-6-7-35-29(37-24)40-8-9-44-19(3)15-40)10-25(26)36-28(43)21-16-38(4)27(42)11-22(21)30(32,33)34/h6-7,10-12,16-19H,8-9,13-15H2,1-5H3,(H,36,43)/t17-,18+,19-/m0/s1	WEXWXCNLXCNZLK-OTWHNJEPSA-N	553607	N-[4-fluoro-5-[2-[rac- (2R)-2-methylmorpholin- 4-yl]pyrimidin-4-yl]-2- [rac-(3S,5R)-3,4,5- trimethylpiperazin-1- yl]phenyl]-1-methyl-6- oxo-4-(trifluoromethyl) pyridine-3-carboxamide::US11319299, Example 694	WD repeat-containing protein 5				 4.92						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553607	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553607&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138551707	469797469							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167368	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccnc(OC2CCOCC2)n1			553608	N-[4-fluoro-5-[2-(oxan-4- yloxy)pyrimidin-4-yl]-2- [rac-(3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 695	WD repeat-containing protein 5				 2.53						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553608	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553608&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608221	469797470							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167369	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCN(CC1)c1ncc(s1)C#N			553609	N-[5-[1-(5-cyano-1,3- thiazol-2-yl)-3,6-dihydro- 2H-pyridin-4-yl]-4- fluoro-2-[rac-(3R,5S)- 3,4,5-trimethylpiperazin- 1-yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 696	WD repeat-containing protein 5				 1.31						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553609	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553609&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608222	469797471							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167370	C[C@H]1CN(C[C@@H](C)O1)c1nccc(n1)-c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)(F)F)c(cc1F)N1CCN(C)[C@@H](C)C1			553610	N-[4-fluoro-5-[2-[rac- (2R,6S)-2,6- dimethylmorpholin-4- yl]pyrimidin-4-yl]-2-[rac- (3R)-3,4- dimethylpiperazin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 698	WD repeat-containing protein 5				 1.59						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553610	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553610&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608223	469797472							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167371	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCCN(CC1)C(=O)OC1(C)CCC1			553611	(1-methylcyclobutyl) 4- [2-fluoro-5-[[6-oxo-4- (trifluoromethyl)-1H- pyridine-3- carbonyl]amino]-4-[rac- (3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-2,3,6,7- tetrahydroazepine-1- carboxylate::US11319299, Example 699	WD repeat-containing protein 5				 3.70						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553611	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553611&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608224	469797473							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167372	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCCN(CC1)c1ncc(s1)C#N			553612	N-[5-[1-(5-cyano-1,3- thiazol-2-yl)-2,3,6,7- tetrahydroazepin-4-yl]-4- fluoro-2-[rac-(3R,5S)- 3,4,5-trimethylpiperazin- 1-yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 700	WD repeat-containing protein 5				 7.31						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553612	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553612&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608225	469797474							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167373	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCCN(C1)c1ccnc(n1)C#N			553613	N-[5-[1-(2- cyanopyrimidin-4-yl)-3,6- dihydro-2H-pyridin-5-yl]- 4-fluoro-2-[rac-(3R,5S)- 3,4,5-trimethylpiperazin- 1-yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 701	WD repeat-containing protein 5				 1.73						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553613	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553613&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608226	469797475							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167374	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)F)C1=CCN(CC1)C(=O)OC1CC(F)(F)C1			553614	(3,3-difluorocyclobutyl) 4-[5-[[4-(difluoromethyl)- 6-oxo-1H-pyridine-3- carbonyl]amino]-2- fluoro-4-[rac-(3R,5S)- 3,4,5-trimethylpiperazin- 1-yl]phenyl]-3,6-dihydro- 2H-pyridine-1-carboxylate::US11319299, Example 702	WD repeat-containing protein 5				 3.47						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553614	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553614&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608227	469797476							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167375	C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)F)C1=CCN(CC1)C(=O)OC1CC(F)(F)C1			553615	(3,3-difluorocyclobutyl) 4-[5-[[4-(difluoromethyl)- 6-oxo-1H-pyridine-3- carbonyl]amino]-2- fluoro-4-[rac-(3R)-3,4- dimethylpiperazin-1- yl]phenyl]-3,6-dihydro- 2H-pyridine-1-carboxylate::US11319299, Example 703	WD repeat-containing protein 5				 1.03						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553615	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553615&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608228	469797477							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167376	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)F)C1=CCCN(C1)C(=O)OC1CC(F)(F)C1			553616	(3,3-difluorocyclobutyl) 5-[5-[[4-(difluoromethyl)- 6-oxo-1H-pyridine-3- carbonyl]amino]-2- fluoro-4-[rac-(3R,5S)- 3,4,5-trimethylpiperazin- 1-yl]phenyl]-3,6-dihydro- 2H-pyridine-1-carboxylate::US11319299, Example 704	WD repeat-containing protein 5				 2.72						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553616	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553616&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608229	469797478							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167377	C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)F)C1=CCCN(C1)C(=O)OC1CC(F)(F)C1			553617	(3,3-difluorocyclobutyl) 5-[5-[[4-(difluoromethyl)- 6-oxo-1H-pyridine-3- carbonyl]amino]-2- fluoro-4-[rac-(3R)-3,4- dimethylpiperazin-1- yl]phenyl]-3,6-dihydro- 2H-pyridine-1-carboxylate::US11319299, Example 705	WD repeat-containing protein 5				 2.02						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553617	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553617&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608230	469797479							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167378	C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1ccc(F)cc1C(F)(F)F)C1=CCCN(C1)C(=O)OC1CC(F)(F)C1	InChI=1S/C30H31F7N4O3/c1-17-15-40(9-8-39(17)2)26-12-24(32)22(18-4-3-7-41(16-18)28(43)44-20-13-29(33,34)14-20)11-25(26)38-27(42)21-6-5-19(31)10-23(21)30(35,36)37/h4-6,10-12,17,20H,3,7-9,13-16H2,1-2H3,(H,38,42)/t17-/m0/s1	HAOYBNIUIBWCFJ-KRWDZBQOSA-N	553618	(3,3-difluorocyclobutyl) 5-[2-fluoro-5-[[4-fluoro- 2-(trifluoromethyl)benzoyl] amino]-4-[rac-(3R)-3,4- dimethylpiperazin-1- yl]phenyl]-3,6-dihydro- 2H-pyridine-1-carboxylate::US11319299, Example 706	WD repeat-containing protein 5				 3.81						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553618	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553618&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138551641	469797480							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167379	C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1ccc(F)cc1C(F)(F)F)C1=CCN(CC1)C(=O)OC1CC(F)(F)C1	InChI=1S/C30H31F7N4O3/c1-17-16-41(10-9-39(17)2)26-13-24(32)22(18-5-7-40(8-6-18)28(43)44-20-14-29(33,34)15-20)12-25(26)38-27(42)21-4-3-19(31)11-23(21)30(35,36)37/h3-5,11-13,17,20H,6-10,14-16H2,1-2H3,(H,38,42)/t17-/m0/s1	BOAUEVZUXZRORU-KRWDZBQOSA-N	553619	(3,3-difluorocyclobutyl) 4-[2-fluoro-5-[[4-fluoro- 2-(trifluoromethyl)benzoyl] amino]-4-[rac-(3R)-3,4- dimethylpiperazin-1- yl]phenyl]-3,6-dihydro- 2H-pyridine-1-carboxylate::US11319299, Example 707	WD repeat-containing protein 5				 2.16						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553619	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553619&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138551446	469797481							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167380	C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)F)C1=CCN(CC1)c1ccnc(n1)C#N			553620	N-[5-[1-(2- cyanopyrimidin-4-yl)-3,6- dihydro-2H-pyridin-4-yl]- 4-fluoro-2-[rac-(3R)-3,4- dimethylpiperazin-1- yl]phenyl]-4- (difluoromethyl)-6-oxo- 1H-pyridine-3-carboxamide::US11319299, Example 708	WD repeat-containing protein 5				 0.580						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553620	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553620&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608231	469797482							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167381	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCN(CC1)c1ccnc(n1)C#N			553621	N-[5-[1-(2- cyanopyrimidin-4-yl)-3,6- dihydro-2H-pyridin-4-yl]- 4-fluoro-2-[rac-(3R,5S)- 3,4,5-trimethylpiperazin- 1-yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 709	WD repeat-containing protein 5				 0.720						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553621	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553621&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608232	469797483							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167382	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cc(F)c(C(=O)NC2CCCCC2)c(F)c1			553622	N-[5-[4- (cyclohexylcarbamoyl)- 3,5-difluorophenyl]-4- fluoro-2-[rac-(3R,5S)- 3,4,5-trimethylpiperazin- 1-yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 710	WD repeat-containing protein 5				 2.03						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553622	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553622&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608233	469797484							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167383	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cc(F)c(C(=O)NC2CCCCC2(C)C)c(F)c1			553623	N-[5-[4-[(2,2- dimethylcyclohexyl) carbamoyl]-3,5- difluorophenyl]-4-fluoro- 2-[rac-(3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 711	WD repeat-containing protein 5				 3.17						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553623	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553623&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608234	469797485							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167384	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cc(F)c(C(=O)NCC2CC2)c(F)c1			553624	N-[5-[4- (cyclopropylmethylcarbamoyl)- 3,5-difluorophenyl]-4-fluoro- 2-[rac-(3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 712	WD repeat-containing protein 5				 2.23						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553624	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553624&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608235	469797486							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167385	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1csc(CN2CCOCC2)n1			553625	N-[4-fluoro-5-[2- (morpholin-4-ylmethyl)- 1,3-thiazol-4-yl]-2-[rac- (3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 713	WD repeat-containing protein 5				 2.59						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553625	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553625&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608236	469797487							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167386	C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cnn(CCN2CCOCC2)c1			553626	N-[4-fluoro-5-[1-(2- morpholin-4- ylethyl)pyrazol-4-yl]-2- [rac-(3R)-3,4- dimethylpiperazin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 714	WD repeat-containing protein 5				 2.76						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553626	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553626&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608237	469797488							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167387	C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1cn(C)c(=O)cc1C(F)F)-c1cnn(CCN2CCOCC2)c1	InChI=1S/C29H36F3N7O3/c1-19-16-38(6-4-35(19)2)26-14-24(30)21(20-15-33-39(17-20)7-5-37-8-10-42-11-9-37)12-25(26)34-29(41)23-18-36(3)27(40)13-22(23)28(31)32/h12-15,17-19,28H,4-11,16H2,1-3H3,(H,34,41)/t19-/m0/s1	RVZIRFGDVGNDSW-IBGZPJMESA-N	553627	4-(difluoromethyl)-N-[4- fluoro-5-[1-(2-morpholin- 4-ylethyl)pyrazol-4-yl]-2- [rac-(3R)-3,4- dimethylpiperazin-1- yl]phenyl]-1-methyl-6- oxopyridine-3-carboxamide::US11319299, Example 715	WD repeat-containing protein 5				 10.9						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553627	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553627&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138551517	469797489							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167388	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cnn(CCN2CCOCC2)c1			553628	N-[4-fluoro-5-[1-(2- morpholin-4- ylethyl)pyrazol-4-yl]-2- [rac-(3R,5S)-3,4?5- trimethylpiperazin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 716	WD repeat-containing protein 5				 2.42						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553628	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553628&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608238	469797490							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167389	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1cn(C)c(=O)cc1C(F)F)-c1cnn(CCN2CCOCC2)c1	InChI=1S/C30H38F3N7O3/c1-19-15-39(16-20(2)37(19)4)27-13-25(31)22(21-14-34-40(17-21)6-5-38-7-9-43-10-8-38)11-26(27)35-30(42)24-18-36(3)28(41)12-23(24)29(32)33/h11-14,17-20,29H,5-10,15-16H2,1-4H3,(H,35,42)/t19-,20+	QWMFKMARCSBQKA-BGYRXZFFSA-N	553629	4-(difluoromethyl)-N-[4- fluoro-5-[1-(2-morpholin- 4-ylethyl)pyrazol-4-yl]-2- [rac-(3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-1-methyl-6- oxopyridine-3-carboxamide::US11319299, Example 717	WD repeat-containing protein 5				 21.6						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553629	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553629&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			137377608	469797491							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167390	C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccnc(n1)N1CCOCC1			553630	N-[4-fluoro-5-(2- morpholin-4-ylpyrimidin- 4-yl)-2-[rac-(3R)-3,4- dimethylpiperazin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 718	WD repeat-containing protein 5				 1.09						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553630	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553630&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608239	469797492							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167391	C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cccc(n1)N1CCOCC1			553631	N-[4-fluoro-5-(6- morpholin-4-ylpyridin-2- yl)-2-[rac-(3R)-3,4- dimethylpiperazin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 719	WD repeat-containing protein 5				 1.18						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553631	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553631&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608240	469797493							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167392	C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)F)-c1ccnc(n1)N1CCOCC1			553632	4-(difluoromethyl)-N-[4- fluoro-5-(2-morpholin-4- ylpyrimidin-4-yl)-2-[rac- (3R)-3,4- dimethylpiperazin-1- yl]phenyl]-6-oxo-1H- pyridine-3-carboxamide::US11319299, Example 720	WD repeat-containing protein 5				 1.31						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553632	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553632&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608241	469797494							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167393	C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)F)-c1cccc(n1)N1CCOCC1			553633	4-(difluoromethyl)-N-[4- fluoro-5-(6-morpholin-4- ylpyridin-2-yl)-2-[rac- (3R)-3,4- dimethylpiperazin-1- yl]phenyl]-6-oxo-1H- pyridine-3-carboxamide::US11319299, Example 721	WD repeat-containing protein 5				 1.62						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553633	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553633&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608242	469797495							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167394	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1ccc(F)cc1C(F)F)-c1cnc(nc1)N1CCOCC1	InChI=1S/C29H32F4N6O2/c1-17-15-39(16-18(2)37(17)3)26-12-24(31)22(19-13-34-29(35-14-19)38-6-8-41-9-7-38)11-25(26)36-28(40)21-5-4-20(30)10-23(21)27(32)33/h4-5,10-14,17-18,27H,6-9,15-16H2,1-3H3,(H,36,40)/t17-,18+	ONWHNLJLIQBGSA-HDICACEKSA-N	553634	2-(difluoromethyl)-4- fluoro-N-[4-fluoro-5-(2- morpholin-4-ylpyrimidin- 5-yl)-2-[rac-(3R,5S)- 3,4,5-trimethylpiperazin- 1-yl]phenyl]benzamide::US11319299, Example 722	WD repeat-containing protein 5				 1.36						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553634	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553634&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138542036	469797496							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167395	CC(C)OC(=O)N1CCC=C(CC1)c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)F)c(cc1F)N1C[C@H](C)N(C)[C@H](C)C1			553635	US11319299, Example 723::propan-2-yl 4-[5-[[4- (difluoromethyl)-6-oxo- 1H-pyridine-3- carbonyl]amino]-2- fluoro-4-[rac-(3R,5S)- 3,4,5-trimethylpiperazin- 1-yl]phenyl]-2,3,6,7- tetrahydroazepine-1- carboxylate	WD repeat-containing protein 5				 3.12						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553635	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553635&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608243	469797497							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167396	CC(C)OC(=O)N1CCC(=CC1)c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)F)c(cc1F)N1CCN(C)[C@@H](C)C1			553636	US11319299, Example 724::propan-2-yl 4-[5-[[4- (difluoromethyl)-6-oxo- 1H-pyridine-3- carbonyl]amino]-2- fluoro-4-[rac-(3R)-3,4- dimethylpiperazin-1- yl]phenyl]-3,6-dihydro- 2H-pyridine-1-carboxylate	WD repeat-containing protein 5				 2.82						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553636	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553636&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608244	469797498							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167397	CC(C)OC(=O)N1CCC=C(C1)c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)F)c(cc1F)N1C[C@H](C)N(C)[C@H](C)C1			553637	US11319299, Example 725::propan-2-yl 5-[5-[[4- (difluoromethyl)-6-oxo- 1H-pyridine-3- carbonyl]amino]-2- fluoro-4-[rac-(3R,5S)- 3,4,5-trimethylpiperazin- 1-yl]phenyl]-3,6-dihydro- 2H-pyridine-1-carboxylate	WD repeat-containing protein 5				 1.59						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553637	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553637&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608245	469797499							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167398	CC(C)OC(=O)N1CCC=C(C1)c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)F)c(cc1F)N1CCN(C)[C@@H](C)C1			553638	US11319299, Example 726::propan-2-yl 5-[5-[[4- (difluoromethyl)-6-oxo- 1H-pyridine-3- carbonyl]amino]-2- fluoro-4-[rac-(3R)-3,4- dimethylpiperazin-1- yl]phenyl]-3,6-dihydro- 2H-pyridine-1-carboxylate	WD repeat-containing protein 5				 2.10						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553638	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553638&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608246	469797500							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167399	CC(C)OC(=O)N1CCC(=CC1)c1cc(NC(=O)c2ccc(F)cc2C(F)(F)F)c(cc1F)N1CCN(C)[C@@H](C)C1	InChI=1S/C29H33F5N4O3/c1-17(2)41-28(40)37-9-7-19(8-10-37)22-14-25(26(15-24(22)31)38-12-11-36(4)18(3)16-38)35-27(39)21-6-5-20(30)13-23(21)29(32,33)34/h5-7,13-15,17-18H,8-12,16H2,1-4H3,(H,35,39)/t18-/m0/s1	FPHQKXFJUXCMGE-SFHVURJKSA-N	553639	US11319299, Example 727::propan-2-yl 4-[2-fluoro- 5-[[4-fluoro-2- (trifluoromethyl)benzoyl] amino]-4-[rac-(3R)-3,4- dimethylpiperazin-1- yl]phenyl]-3,6-dihydro- 2H-pyridine-1-carboxylate	WD repeat-containing protein 5				 2.46						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553639	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553639&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138551674	469797501							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167400	CC(C)OC(=O)N1CCC=C(C1)c1cc(NC(=O)c2ccc(F)cc2C(F)(F)F)c(cc1F)N1CCN(C)[C@@H](C)C1	InChI=1S/C29H33F5N4O3/c1-17(2)41-28(40)38-9-5-6-19(16-38)22-13-25(26(14-24(22)31)37-11-10-36(4)18(3)15-37)35-27(39)21-8-7-20(30)12-23(21)29(32,33)34/h6-8,12-14,17-18H,5,9-11,15-16H2,1-4H3,(H,35,39)/t18-/m0/s1	VWFZJHLHORFOES-SFHVURJKSA-N	553640	US11319299, Example 728::propan-2-yl 5-[2-fluoro- 5-[[4-fluoro-2- (trifluoromethyl)benzoyl] amino]-4-[rac-(3R)-3,4- dimethylpiperazin-1- yl]phenyl]-3,6-dihydro- 2H-pyridine-1-carboxylate	WD repeat-containing protein 5				 3.55						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553640	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553640&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138551662	469797502							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167401	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)F)C1=CCCN(CC1)C(=O)OC1(C)CCC1			553641	(1-methylcyclobutyl) 4- [5-[[4-(difluoromethyl)-6- oxo-1H-pyridine-3- carbonyl]amino]-2- fluoro-4-[rac-(3R,5S)- 3,4,5-trimethylpiperazin- 1-yl]phenyl]-2,3,6,7- tetrahydroazepine-1- carboxylate::US11319299, Example 729	WD repeat-containing protein 5				 3.11						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553641	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553641&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608247	469797503							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167402	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)F)C1=CCCN(CC1)C(=O)OC1CC(F)(F)C1			553642	(3,3-difluorocyclobutyl) 4-[5-[[4-(difluoromethyl)- 6-oxo-1H-pyridine-3- carbonyl]amino]-2- fluoro-4-[rac-(3R,5S)- 3,4,5-trimethylpiperazin- 1-yl]phenyl]-2,3,6,7- tetrahydroazepine-1- carboxylate::US11319299, Example 730	WD repeat-containing protein 5				 7.99						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553642	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553642&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608248	469797504							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167403	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)F)C1=CCCN(CC1)c1ncc(s1)C#N			553643	N-[5-[1-(5-cyano-1,3- thiazol-2-yl)-2,3,6,7- tetrahydroazepin-4-yl]-4- fluoro-2-[rac-(3R,5S)- 3,4,5-trimethylpiperazin- 1-yl]phenyl]-4- (difluoromethyl)-6-oxo- 1H-pyridine-3-carboxamide::US11319299, Example 731	WD repeat-containing protein 5				 7.61						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553643	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553643&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608249	469797505							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167404	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(C(=O)NC2CCCCC2)c(F)c1			553644	N-[5-[4- (cyclohexylcarbamoyl)-3- fluorophenyl]-4-fluoro-2- [rac-(3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 732	WD repeat-containing protein 5				 2.76						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553644	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553644&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608250	469797506							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167405	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(C(=O)N(C)CC2CC2)c(F)c1			553645	N-[5-[4- [cyclopropylmethyl(meth yl)carbamoyl]-3- fluorophenyl]-4-fluoro-2- [rac-(3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 733	WD repeat-containing protein 5				 1.29						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553645	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553645&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608251	469797507							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167406	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(C(=O)NC2CCC(F)(F)CC2)c(F)c1			553646	N-[5-[4-[(4,4- difluorocyclohexyl) carbamoyl]-3-fluorophenyl]- 4-fluoro-2-[rac-(3R,5S)- 3,4,5-trimethylpiperazin- 1-yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 734	WD repeat-containing protein 5				 4.13						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553646	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553646&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608252	469797508							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167407	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(C(=O)NCC2CC2)c(F)c1			553647	N-[5-[4- (cyclopropylmethylcarbamoyl)- 3-fluorophenyl]-4- fluoro-2-[rac-(3R,5S)- 3,4,5-trimethylpiperazin- 1-yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 735	WD repeat-containing protein 5				 4.23						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553647	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553647&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608253	469797509							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167408	C[C@H]1COCCN1c1ncc(cn1)-c1cc(NC(=O)c2ccc(F)cc2C(F)(F)F)c(cc1F)N1CCN(C)[C@@H](C)C1	InChI=1S/C29H31F5N6O2/c1-17-15-39(7-6-38(17)3)26-12-24(31)22(19-13-35-28(36-14-19)40-8-9-42-16-18(40)2)11-25(26)37-27(41)21-5-4-20(30)10-23(21)29(32,33)34/h4-5,10-14,17-18H,6-9,15-16H2,1-3H3,(H,37,41)/t17-,18-/m0/s1	IOMHUFLGWGXOMU-ROUUACIJSA-N	553648	4-fluoro-N-[4-fluoro-2- [rac-(3R)-3,4- dimethylpiperazin-1-yl]-5- [2-[rac-(2R)-2- methylmorpholin-4- yl]pyrimidin-4-yl]phenyl]- 2-(trifluoromethyl)benzamide::US11319299, Example 736	WD repeat-containing protein 5				 0.290						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553648	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553648&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138551454	469797510							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167409	C[C@@H]1COCCN1c1ncc(cn1)-c1cc(NC(=O)c2ccc(F)cc2C(F)(F)F)c(cc1F)N1CCN(C)[C@@H](C)C1	InChI=1S/C29H31F5N6O2/c1-17-15-39(7-6-38(17)3)26-12-24(31)22(19-13-35-28(36-14-19)40-8-9-42-16-18(40)2)11-25(26)37-27(41)21-5-4-20(30)10-23(21)29(32,33)34/h4-5,10-14,17-18H,6-9,15-16H2,1-3H3,(H,37,41)/t17-,18+/m0/s1	IOMHUFLGWGXOMU-ZWKOTPCHSA-N	553649	4-fluoro-N-[4-fluoro-2- [rac-(3S)-3,4- dimethylpiperazin-1-yl]-5- [2-[rac-(3R)-3- methylmorpholin-4- yl]pyrimidin-5-yl]phenyl]- 2-(trifluoromethyl)benzamide::US11319299, Example 737	WD repeat-containing protein 5				 4.61						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553649	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553649&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138541825	469797511							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167410	C[C@@H]1CN(CCO1)c1nccc(n1)-c1cc(NC(=O)c2ccc(F)cc2C(F)(F)F)c(cc1F)N1CCN(C)[C@@H](C)C1	InChI=1S/C29H31F5N6O2/c1-17-15-39(9-8-38(17)3)26-14-23(31)21(24-6-7-35-28(37-24)40-10-11-42-18(2)16-40)13-25(26)36-27(41)20-5-4-19(30)12-22(20)29(32,33)34/h4-7,12-14,17-18H,8-11,15-16H2,1-3H3,(H,36,41)/t17-,18+/m0/s1	SVTZVEIUYZSBTJ-ZWKOTPCHSA-N	553650	4-fluoro-N-[4-fluoro-2- [rac-(3S)-3,4- dimethylpiperazin-1-yl]-5- [2-[rac-(2R)-2- methylmorpholin-4- yl]pyriimdin-4-yl]phenyl]- 2-(trifluoromethyl)benzamide::US11319299, Example 738	WD repeat-containing protein 5				 4.00						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553650	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553650&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			137376926	469797512							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167411	C[C@H]1CN(C[C@@H](C)O1)c1nccc(n1)-c1cc(NC(=O)c2ccc(F)cc2C(F)(F)F)c(cc1F)N1CCN(C)[C@@H](C)C1	InChI=1S/C30H33F5N6O2/c1-17-14-40(10-9-39(17)4)27-13-24(32)22(25-7-8-36-29(38-25)41-15-18(2)43-19(3)16-41)12-26(27)37-28(42)21-6-5-20(31)11-23(21)30(33,34)35/h5-8,11-13,17-19H,9-10,14-16H2,1-4H3,(H,37,42)/t17-,18-,19+/m0/s1	RUZCPNUCVFVJFU-GBESFXJTSA-N	553651	4-fluoro-N-[4-fluoro-5-[2- [rac-(2R,6S)-2,6- dimethylmorpholin-4- yl]pyrimidin-4-yl]-2-[rac- (3R)-3,4- dimethylpiperazin-1- yl]phenyl]-2- (trifluoromethyl)benzamide::US11319299, Example 739	WD repeat-containing protein 5				 3.00						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553651	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553651&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138551411	469797513							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167412	C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)F)C1=CCCN(C1)c1ccnc(n1)C#N			553652	N-[5-[1-(2- cyanopyrimidin-4-yl)-3,6- dihydro-2H-pyridin-5-yl]- 4-fluoro-2-[rac-(3R)-3,4- dimethylpiperazin-1- yl]phenyl]-4- (difluoromethyl)-6-oxo- 1H-pyridine-3-carboxamide::US11319299, Example 740	WD repeat-containing protein 5				 4.47						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553652	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553652&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608254	469797514							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167413	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1cn(C)c(=O)cc1C(F)F)-c1nc(CN2CCOCC2)cs1	InChI=1S/C29H35F3N6O3S/c1-17-12-38(13-18(2)36(17)4)25-11-23(30)21(29-33-19(16-42-29)14-37-5-7-41-8-6-37)9-24(25)34-28(40)22-15-35(3)26(39)10-20(22)27(31)32/h9-11,15-18,27H,5-8,12-14H2,1-4H3,(H,34,40)/t17-,18+	SMRSGCKOWDGOSO-HDICACEKSA-N	553653	4-(difluoromethyl)-N-[4- fluoro-5-[4-(morpholin-4- ylmethyl)-1,3-thiazol-2- yl]-2-[rac-(3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-1-methyl-6- oxopyridine-3-carboxamide::US11319299, Example 741	WD repeat-containing protein 5				 6.75						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553653	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553653&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			137377529	469797515							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167414	C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cccc(n1)N1CCNCC1			553654	N-[4-fluoro-5-(6- piperazin-1-ylpyridin-2- yl)-2-[rac-(3R)-3,4- dimethylpiperazin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 742	WD repeat-containing protein 5				 2.87						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553654	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553654&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608255	469797516							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167415	C[C@H]1CN(C[C@@H](C)O1)c1nccc(n1)-c1cc(NC(=O)c2cn(C)c(=O)cc2C(F)(F)F)c(cc1F)N1C[C@H](C)N(C)[C@H](C)C1	InChI=1S/C31H37F4N7O3/c1-17-12-41(13-18(2)40(17)6)27-11-24(32)21(25-7-8-36-30(38-25)42-14-19(3)45-20(4)15-42)9-26(27)37-29(44)22-16-39(5)28(43)10-23(22)31(33,34)35/h7-11,16-20H,12-15H2,1-6H3,(H,37,44)/t17-,18+,19-,20+	RJMONIVAVAQPFW-FGYAAKKASA-N	553655	N-[4-fluoro-5-[2-[rac- (2R,6S)-2,6- dimethylmorpholin-4- yl]pyrimidin-4-yl]-2-[rac- (3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-1-methyl-6- oxo-4-(trifluoromethyl) pyridine-3-carboxamide::US11319299, Example 743::US11319299, Example 745	WD repeat-containing protein 5				 5.22						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553655	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553655&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138541750	469797517							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167416	C[C@H]1CN(C[C@@H](C)O1)c1nccc(n1)-c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)F)c(cc1F)N1C[C@H](C)N(C)[C@H](C)C1			553656	4-(difluoromethyl)-N-[4- fluoro-5-[2-[rac-(2R,6S)- 2,6-dimethylmorpholin-4- yl]pyrimidin-4-yl]-2-[rac- (3S,5R)-3,4,5- trimethylpiperazin-1- yl]phenyl]-6-oxo-1H- pyridine-3-carboxamide::US11319299, Example 744	WD repeat-containing protein 5				 2.76						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553656	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553656&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608256	469797518							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167417	C[C@H]1CN(C[C@@H](C)O1)c1nccc(n1)-c1cc(NC(=O)c2cn(C)c(=O)cc2C(F)(F)F)c(cc1F)N1C[C@H](C)N(C)[C@H](C)C1	InChI=1S/C31H37F4N7O3/c1-17-12-41(13-18(2)40(17)6)27-11-24(32)21(25-7-8-36-30(38-25)42-14-19(3)45-20(4)15-42)9-26(27)37-29(44)22-16-39(5)28(43)10-23(22)31(33,34)35/h7-11,16-20H,12-15H2,1-6H3,(H,37,44)/t17-,18+,19-,20+	RJMONIVAVAQPFW-FGYAAKKASA-N	553655	N-[4-fluoro-5-[2-[rac- (2R,6S)-2,6- dimethylmorpholin-4- yl]pyrimidin-4-yl]-2-[rac- (3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-1-methyl-6- oxo-4-(trifluoromethyl) pyridine-3-carboxamide::US11319299, Example 743::US11319299, Example 745	WD repeat-containing protein 5				 5.60						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553655	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553655&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138541750	469797517							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167418	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1cn(C)c(=O)cc1C(F)F)-c1ccnc(n1)N1CCOCC1	InChI=1S/C29H34F3N7O3/c1-17-14-39(15-18(2)37(17)4)25-13-22(30)20(23-5-6-33-29(35-23)38-7-9-42-10-8-38)11-24(25)34-28(41)21-16-36(3)26(40)12-19(21)27(31)32/h5-6,11-13,16-18,27H,7-10,14-15H2,1-4H3,(H,34,41)/t17-,18+	CMIXAWGKXZPGTB-HDICACEKSA-N	553658	4-(difluoromethyl)-N-[4- fluoro-5-(2-morpholin-4- ylpyrimidin-4-yl)-2-[rac- (3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-1-methyl-6- oxopyridine-3-carboxamide::US11319299, Example 746	WD repeat-containing protein 5				 13565000						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553658	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553658&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138541762	469797519							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166713	CN1CCN(CC1)c1cc(F)c(cc1NC(=O)c1cc(C)c(F)c(C)c1)-c1cccc(CN2CCOCC2)c1	InChI=1S/C31H36F2N4O2/c1-21-15-25(16-22(2)30(21)33)31(38)34-28-18-26(27(32)19-29(28)37-9-7-35(3)8-10-37)24-6-4-5-23(17-24)20-36-11-13-39-14-12-36/h4-6,15-19H,7-14,20H2,1-3H3,(H,34,38)	PXTYRLCEWAUNKF-UHFFFAOYSA-N	552932	4-fluoro-N-[4-fluoro-2- (4-methylpiperazin-1-yl)- 5-[3-(morpholin-4- ylmethyl)phenyl]phenyl]- 3,5-dimethylbenzamide::US11319299, Example 1	WD repeat-containing protein 5				 84.0						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=552932	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=552932&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			137376792	469796801							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166714	CN1CCN(CC1)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cccc(CN2CCOCC2)c1	InChI=1S/C29H31F4N5O3/c1-36-5-7-38(8-6-36)26-16-24(30)21(20-4-2-3-19(13-20)18-37-9-11-41-12-10-37)14-25(26)35-28(40)22-17-34-27(39)15-23(22)29(31,32)33/h2-4,13-17H,5-12,18H2,1H3,(H,34,39)(H,35,40)	GVIBWIRSZYKTTI-UHFFFAOYSA-N	552933	N-[4-fluoro-2-(4- methylpiperazin-1-yl)-5- [3-(morpholin-4- ylmethyl)phenyl]phenyl]- 6-oxo-4-(trifluoromethyl)- 1H-pyridine-3-carboxamide::US11319299, Comp. No. 2::US11319299, Example 2	WD repeat-containing protein 5				 11.0						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=552933	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=552933&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607803	469796802							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166715	CN1CCN(CC1)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cnc(nc1)N1CCOCC1	InChI=1S/C26H27F4N7O3/c1-35-2-4-36(5-3-35)22-12-20(27)17(16-13-32-25(33-14-16)37-6-8-40-9-7-37)10-21(22)34-24(39)18-15-31-23(38)11-19(18)26(28,29)30/h10-15H,2-9H2,1H3,(H,31,38)(H,34,39)	QNEXYXLSJZBQJZ-UHFFFAOYSA-N	552948	N-[4-fluoro-2-(4- methylpiperazin-1-yl)-5- (2-morpholin-4- ylpyrimidin-5-yl)phenyl]- 6-oxo-4-(trifluoromethyl)- 1H-pyridine-3-carboxamide::US11319299, Comp. No. 3::US11319299, Example 3	WD repeat-containing protein 5				 2.00						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=552948	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=552948&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607804	469796817							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166716	CN1CCN(CC1)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(nc1)N1CCOCC1	InChI=1S/C27H28F4N6O3/c1-35-4-6-36(7-5-35)23-14-21(28)18(17-2-3-24(32-15-17)37-8-10-40-11-9-37)12-22(23)34-26(39)19-16-33-25(38)13-20(19)27(29,30)31/h2-3,12-16H,4-11H2,1H3,(H,33,38)(H,34,39)	IDXURNUKWGSUOE-UHFFFAOYSA-N	552949	N-[4-fluoro-2-(4- methylpiperazin-1-yl)-5- (6-morpholin-4-ylpyridin- 3-yl)phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 4	WD repeat-containing protein 5				 4.00						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=552949	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=552949&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607805	469796818							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166717	CN1CCN(CC1)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc2OCOc2c1	InChI=1S/C25H22F4N4O4/c1-32-4-6-33(7-5-32)20-11-18(26)15(14-2-3-21-22(8-14)37-13-36-21)9-19(20)31-24(35)16-12-30-23(34)10-17(16)25(27,28)29/h2-3,8-12H,4-7,13H2,1H3,(H,30,34)(H,31,35)	WOROKLNMCVXIBS-UHFFFAOYSA-N	552950	N-[5-(1,3-benzodioxol-5- yl)-4-fluoro-2-(4- methylpiperazin-1- yl)phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 5	WD repeat-containing protein 5				 33.0						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=552950	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=552950&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607806	469796819							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166718	C[C@@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cnc(nc1)N1CCOCC1			552951	N-[2-[(3R)-3,4- dimethylpiperazin-1-yl]- 4-fluoro-5-(2-morpholin- 4-ylpyrimidin-5- yl)phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 6	WD repeat-containing protein 5				 3.00						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=552951	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=552951&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607807	469796820							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166719	C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cnc(nc1)N1CCOCC1			552952	N-[2-[(3S)-3,4- dimethylpiperazin-1-yl]- 4-fluoro-5-(2-morpholin- 4-ylpyrimidin-5- yl)phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 7	WD repeat-containing protein 5				 0.060						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=552952	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=552952&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607808	469796821							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166720	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cnc(nc1)N1CCOCC1			552953	N-[4-fluoro-5-(2- morpholin-4-ylpyrimidin- 5-yl)-2-[(3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299,  Example Table6.8::US11319299, Comp. No. 8::US11319299, Example 8	WD repeat-containing protein 5				 0.300						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=552953	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=552953&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607809	469796822							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166721	CN1CCN(CC1)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cnc(nc1)N1CCCC1	InChI=1S/C26H27F4N7O2/c1-35-6-8-36(9-7-35)22-12-20(27)17(16-13-32-25(33-14-16)37-4-2-3-5-37)10-21(22)34-24(39)18-15-31-23(38)11-19(18)26(28,29)30/h10-15H,2-9H2,1H3,(H,31,38)(H,34,39)	HUCHWMVKXDSHCR-UHFFFAOYSA-N	552954	N-[4-fluoro-2-(4- methylpiperazin-1-yl)-5- (2-pyrrolidin-1-ylpyrimidin- 5-yl)phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 9	WD repeat-containing protein 5				 5.00						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=552954	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=552954&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607810	469796823							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166722	CN1CCN(CC1)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cnc(NC2CC2)nc1	InChI=1S/C25H25F4N7O2/c1-35-4-6-36(7-5-35)21-10-19(26)16(14-11-31-24(32-12-14)33-15-2-3-15)8-20(21)34-23(38)17-13-30-22(37)9-18(17)25(27,28)29/h8-13,15H,2-7H2,1H3,(H,30,37)(H,34,38)(H,31,32,33)	XHGDUSOCGSBMTC-UHFFFAOYSA-N	552955	N-[5-[2-(cyclopropylamino) pyrimidin-5-yl]-4-fluoro-2- (4-methylpiperazin-1- yl)phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 10	WD repeat-containing protein 5				 13.0						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=552955	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=552955&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607811	469796824							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166723	CN1CCN(CC1)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cnc(NC2CCCCC2)nc1	InChI=1S/C28H31F4N7O2/c1-38-7-9-39(10-8-38)24-13-22(29)19(17-14-34-27(35-15-17)36-18-5-3-2-4-6-18)11-23(24)37-26(41)20-16-33-25(40)12-21(20)28(30,31)32/h11-16,18H,2-10H2,1H3,(H,33,40)(H,37,41)(H,34,35,36)	RRQBQDOLKJVCNU-UHFFFAOYSA-N	552956	N-[5-[2-(cyclohexylamino) pyrimidin-5-yl]-4-fluoro-2- (4-methylpiperazin-1- yl)phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 11	WD repeat-containing protein 5				 5.00						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=552956	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=552956&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607812	469796825							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166724	CCOc1ncc(cn1)-c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)(F)F)c(cc1F)N1CCN(C)CC1	InChI=1S/C24H24F4N6O3/c1-3-37-23-30-11-14(12-31-23)15-8-19(20(10-18(15)25)34-6-4-33(2)5-7-34)32-22(36)16-13-29-21(35)9-17(16)24(26,27)28/h8-13H,3-7H2,1-2H3,(H,29,35)(H,32,36)	OFLSDQKDUXBXCT-UHFFFAOYSA-N	552957	N-[5-(2-ethoxypyrimidin- 5-yl)-4-fluoro-2-(4- methylpiperazin-1- yl)phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 12	WD repeat-containing protein 5				 5.00						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=552957	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=552957&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607813	469796826							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166725	CN1CCN(CC1)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cnc(C)nc1	InChI=1S/C23H22F4N6O2/c1-13-28-10-14(11-29-13)15-7-19(20(9-18(15)24)33-5-3-32(2)4-6-33)31-22(35)16-12-30-21(34)8-17(16)23(25,26)27/h7-12H,3-6H2,1-2H3,(H,30,34)(H,31,35)	MONYSZXYDXDGEK-UHFFFAOYSA-N	552958	N-[4-fluoro-2-(4- methylpiperazin-1-yl)-5- (2-methylpyrimidin-5- yl)phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 13	WD repeat-containing protein 5				 4.00						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=552958	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=552958&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607814	469796827							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166726	CN1CCN(CC1)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(NC2CCCCC2)nc1	InChI=1S/C29H32F4N6O2/c1-38-9-11-39(12-10-38)25-15-23(30)20(18-7-8-26(34-16-18)36-19-5-3-2-4-6-19)13-24(25)37-28(41)21-17-35-27(40)14-22(21)29(31,32)33/h7-8,13-17,19H,2-6,9-12H2,1H3,(H,34,36)(H,35,40)(H,37,41)	KCOMOZYHSDZIRW-UHFFFAOYSA-N	552959	N-[5-[6-(cyclohexylamino) pyridin-3-yl]-4-fluoro-2- (4-methylpiperazin-1- yl)phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 14	WD repeat-containing protein 5				 5.00						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=552959	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=552959&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607815	469796828							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166727	CN1CCN(CC1)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cnc(O)nc1	InChI=1S/C22H20F4N6O3/c1-31-2-4-32(5-3-31)18-8-16(23)13(12-9-28-21(35)29-10-12)6-17(18)30-20(34)14-11-27-19(33)7-15(14)22(24,25)26/h6-11H,2-5H2,1H3,(H,27,33)(H,30,34)(H,28,29,35)	XXSLMFWASLUDIS-UHFFFAOYSA-N	552960	N-[4-fluoro-5-(2- hydroxypyrimidin-5-yl)- 2-(4-methylpiperazin-1- yl)phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 15	WD repeat-containing protein 5				 26.0						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=552960	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=552960&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607816	469796829							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166728	CN1CCN(CC1)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cnc(nc1)C#N	InChI=1S/C23H19F4N7O2/c1-33-2-4-34(5-3-33)19-8-17(24)14(13-10-29-20(9-28)30-11-13)6-18(19)32-22(36)15-12-31-21(35)7-16(15)23(25,26)27/h6-8,10-12H,2-5H2,1H3,(H,31,35)(H,32,36)	CDBKROHOJVKZNJ-UHFFFAOYSA-N	552962	N-[5-(2-cyanopyrimidin- 5-yl)-4-fluoro-2-(4- methylpiperazin-1- yl)phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 16	WD repeat-containing protein 5				 2.00						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=552962	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=552962&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607818	469796831							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167419	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)F)-c1ccc(C(=O)NC2CCCCC2(C)C)c(F)c1			553659	N-[5-[4-[(2,2- dimethylcyclohexyl) carbamoyl]-3-fluorophenyl]-4- fluoro-2-[rac-(3R,5S)- 3,4,5-trimethylpiperazin- 1-yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 747	WD repeat-containing protein 5				 4.85						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553659	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553659&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608257	469797520							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167420	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1cn(C)c(=O)cc1C(F)F)-c1ncc(CN2CCOCC2)s1	InChI=1S/C29H35F3N6O3S/c1-17-13-38(14-18(2)36(17)4)25-11-23(30)21(29-33-12-19(42-29)15-37-5-7-41-8-6-37)9-24(25)34-28(40)22-16-35(3)26(39)10-20(22)27(31)32/h9-12,16-18,27H,5-8,13-15H2,1-4H3,(H,34,40)/t17-,18+	JWFOXMORBRAWCC-HDICACEKSA-N	553660	4-(difluoromethyl)-N-[4- fluoro-5-[5-(morpholin-4- ylmethyl)-1,3-thiazol-2- yl]-2-[rac-(3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-1-methyl-6- oxopyridine-3-carboxamide::US11319299, Example 748	WD repeat-containing protein 5				 51.8						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553660	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553660&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138541647	469797521							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167421	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1cn(C)c(=O)cc1C(F)F)-c1csc(CN2CCOCC2)n1	InChI=1S/C29H35F3N6O3S/c1-17-12-38(13-18(2)36(17)4)25-11-22(30)20(24-16-42-26(33-24)15-37-5-7-41-8-6-37)9-23(25)34-29(40)21-14-35(3)27(39)10-19(21)28(31)32/h9-11,14,16-18,28H,5-8,12-13,15H2,1-4H3,(H,34,40)/t17-,18+	IRJSMHYFJVNAGT-HDICACEKSA-N	553661	4-(difluoromethyl)-N-[4- fluoro-5-[2-(morpholin-4- ylmethyl)-1,3-thiazol-4- yl]-2-[rac-(3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-1-methyl-6- oxopyridine-3-carboxamide::US11319299, Example 749	WD repeat-containing protein 5				 10.6						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553661	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553661&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138541744	469797522							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167422	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1nc(CN2CCOCC2)cs1			553662	N-[4-fluoro-5-[4- (morpholin-4-ylmethyl)- 1,3-thiazol-2-yl]-2-[rac- (3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 750	WD repeat-containing protein 5				 1.71						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553662	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553662&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608258	469797523							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167423	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ncc(CN2CCOCC2)s1			553663	N-[4-fluoro-5-[5- (morpholin-4-ylmethyl)- 1,3-thiazol-2-yl]-2-[rac- (3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 751	WD repeat-containing protein 5				 8.27						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553663	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553663&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608259	469797524							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167424	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cc(F)c(C(=O)N(C)C2CCCCC2)c(F)c1			553664	N-(4'-(cyclohexyl (methyl)carbamoyl)-3',5', 6-trifluoro-4-((3S,5R)-3,4,5- trimethylpiperazin-1-yl)- [1,1'-biphenyl]-3-yl)-6- oxo-4-(trifluoromethyl)- 1,6-dihydropyridine-3- carboxamide::US11319299, Example 760	WD repeat-containing protein 5				 2.00						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553664	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553664&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608260	469797525							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167425	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cc(F)c(C(=O)N(C)C2CCCC2)c(F)c1			553665	N-(4'-(cyclopentyl (methyl)carbamoyl)-3',5',6- trifluoro-4-((3S,5R)-3,4,5- trimethylpiperazin-1-yl)- [1,1'-biphenyl]-3-yl)-6- oxo-4-(trifluoromethyl)- 1,6-dihydropyridine-3- carboxamide::US11319299, Example 761	WD repeat-containing protein 5				 2.00						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553665	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553665&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608261	469797526							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167426	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cc(F)c(C(=O)N[C@@H]2CCOC2)c(F)c1			553666	6-oxo-N-(3',5',6-trifluoro- 4'-(((R)-tetrahydrofuran- 3-yl)carbamoyl)-4- ((3S,5R)-3,4,5- trimethylpiperazin-1-yl)- [1,1'-biphenyl]-3-yl)-4- (trifluoromethyl)-1,6- dihydropyridine-3- carboxamide::US11319299, Example 762	WD repeat-containing protein 5				 0.900						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553666	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553666&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608262	469797527							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167427	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cc(F)c(C(=O)N(C)C2COC2)c(F)c1			553667	6-oxo-N-(3',5',6-trifluoro- 4'-(methyl(oxetan-3- yl)carbamoyl)-4- ((3S,5R)-3,4,5- trimethylpiperazin-1-yl)- [1,1'-biphenyl]-3-yl)-4- (trifluoromethyl)-1,6- dihydropyridine-3- carboxamide::US11319299, Example 763	WD repeat-containing protein 5				 0.700						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553667	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553667&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608263	469797528							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166729	CN1CCN(CC1)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cnc(OCC(F)(F)F)nc1	InChI=1S/C24H21F7N6O3/c1-36-2-4-37(5-3-36)19-8-17(25)14(13-9-33-22(34-10-13)40-12-23(26,27)28)6-18(19)35-21(39)15-11-32-20(38)7-16(15)24(29,30)31/h6-11H,2-5,12H2,1H3,(H,32,38)(H,35,39)	YIGUOFOBBBPQLX-UHFFFAOYSA-N	552963	N-[4-fluoro-2-(4- methylpiperazin-1-yl)-5- [2-(2,2,2-trifluoroethoxy) pyrimidin-5-yl]phenyl]-6- oxo-4-(trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 17	WD repeat-containing protein 5				 6.00						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=552963	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=552963&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607819	469796832							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166730	CN1CCN(CC1)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cncnc1	InChI=1S/C22H20F4N6O2/c1-31-2-4-32(5-3-31)19-8-17(23)14(13-9-27-12-28-10-13)6-18(19)30-21(34)15-11-29-20(33)7-16(15)22(24,25)26/h6-12H,2-5H2,1H3,(H,29,33)(H,30,34)	QGDHQOJSPUAKSA-UHFFFAOYSA-N	552964	N-[4-fluoro-2-(4- methylpiperazin-1-yl)-5- pyrimidin-5-ylphenyl]-6- oxo-4-(trifluoromethyl)- 1H-pyridine-3-carboxamide::US11319299, Example 18	WD repeat-containing protein 5				 9.00						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=552964	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=552964&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607820	469796833							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166731	COc1ncc(c(OC)n1)-c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)(F)F)c(cc1F)N1CCN(C)CC1	InChI=1S/C24H24F4N6O4/c1-33-4-6-34(7-5-33)19-10-17(25)13(14-11-30-23(38-3)32-22(14)37-2)8-18(19)31-21(36)15-12-29-20(35)9-16(15)24(26,27)28/h8-12H,4-7H2,1-3H3,(H,29,35)(H,31,36)	NXSYJUANRFWWGT-UHFFFAOYSA-N	552965	N-[5-(2,4- dimethoxypyrimidin-5- yl)-4-fluoro-2-(4- methylpiperazin-1- yl)phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 19	WD repeat-containing protein 5				 4.00						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=552965	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=552965&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607821	469796834							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166732	CN1CCN(CC1)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)F)-c1cnc(nc1)N1CCOCC1	InChI=1S/C26H28F3N7O3/c1-34-2-4-35(5-3-34)22-12-20(27)17(16-13-31-26(32-14-16)36-6-8-39-9-7-36)10-21(22)33-25(38)19-15-30-23(37)11-18(19)24(28)29/h10-15,24H,2-9H2,1H3,(H,30,37)(H,33,38)	UJCBRBGSYIDHKB-UHFFFAOYSA-N	552966	4-(difluoromethyl)-N-[4- fluoro-2-(4-methylpiperazin- 1-yl)-5-(2-morpholin-4- ylpyrimidin-5-yl)phenyl]- 6-oxo-1H-pyridine-3- carboxamide::US11319299, Example 20	WD repeat-containing protein 5				 2.00						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=552966	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=552966&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607822	469796835							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166733	CN(C)C1CCN(C1)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cnc(nc1)N1CCOCC1			552967	N-[2-[3-(dimethylamino) pyrrolidin-1-yl]-4-fluoro-5- (2-morpholin-4-ylpyrimidin- 5-yl)phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 21	WD repeat-containing protein 5				 0.900						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=552967	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=552967&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607823	469796836							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166734	CN1CCN(CC1)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCOCC1	InChI=1S/C23H24F4N4O3/c1-30-4-6-31(7-5-30)20-12-18(24)15(14-2-8-34-9-3-14)10-19(20)29-22(33)16-13-28-21(32)11-17(16)23(25,26)27/h2,10-13H,3-9H2,1H3,(H,28,32)(H,29,33)	MCKHRDBCHQEZEN-UHFFFAOYSA-N	552968	N-[5-(3,6-dihydro-2H- pyran-4-yl)-4-fluoro-2- (4-methylpiperazin-1- yl)phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 22	WD repeat-containing protein 5				 7.60						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=552968	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=552968&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607824	469796837							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166735	CN1CCN(CC1)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCNCC1	InChI=1S/C23H25F4N5O2/c1-31-6-8-32(9-7-31)20-12-18(24)15(14-2-4-28-5-3-14)10-19(20)30-22(34)16-13-29-21(33)11-17(16)23(25,26)27/h2,10-13,28H,3-9H2,1H3,(H,29,33)(H,30,34)	LBCCPUPFKKIKMY-UHFFFAOYSA-N	552969	N-[4-fluoro-2-(4- methylpiperazin-1-yl)-5- (1,2,3,6-tetrahydropyridin- 4-yl)phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 23	WD repeat-containing protein 5				 17.1						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=552969	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=552969&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607825	469796838							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166736	CN1CCN(CC1)c1cc(F)ccc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F	InChI=1S/C18H18F4N4O2/c1-25-4-6-26(7-5-25)15-8-11(19)2-3-14(15)24-17(28)12-10-23-16(27)9-13(12)18(20,21)22/h2-3,8-10H,4-7H2,1H3,(H,23,27)(H,24,28)	LWTXKPMUOFWYDS-UHFFFAOYSA-N	552970	N-[4-fluoro-2-(4- methylpiperazin-1- yl)phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 24	WD repeat-containing protein 5				 75.6						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=552970	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=552970&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607826	469796839							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166737	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1ccc(F)c(C)c1)-c1cnc(nc1)N1CCOCC1	InChI=1S/C29H34F2N6O2/c1-18-11-21(5-6-24(18)30)28(38)34-26-12-23(22-14-32-29(33-15-22)36-7-9-39-10-8-36)25(31)13-27(26)37-16-19(2)35(4)20(3)17-37/h5-6,11-15,19-20H,7-10,16-17H2,1-4H3,(H,34,38)/t19-,20+	CRLXCSCPDXUEGK-BGYRXZFFSA-N	552971	4-fluoro-N-[4-fluoro-5- (2-morpholin-4- ylpyrimidin-5-yl)-2- [(3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-3- methylbenzamide::US11319299, Example 25	WD repeat-containing protein 5				 8.50						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=552971	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=552971&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			137376879	469796840							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166738	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)ccc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F			552972	N-[4-fluoro-2-[(3R,5S)- 3,4,5-trimethylpiperazin- 1-yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 26	WD repeat-containing protein 5				 42.5						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=552972	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=552972&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607827	469796841							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166739	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1cnc(NC(C)=O)cc1C(F)(F)F)-c1cnc(nc1)N1CCOCC1	InChI=1S/C30H34F4N8O3/c1-17-15-42(16-18(2)40(17)4)26-11-24(31)21(20-12-36-29(37-13-20)41-5-7-45-8-6-41)9-25(26)39-28(44)22-14-35-27(38-19(3)43)10-23(22)30(32,33)34/h9-14,17-18H,5-8,15-16H2,1-4H3,(H,39,44)(H,35,38,43)/t17-,18+	WEPWHMCRXBMMJW-HDICACEKSA-N	552976	6-acetamido-N-[4-fluoro- 5-(2-morpholin-4- ylpyrimidin-5-yl)-2- [(3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-4- (trifluoromethyl)pyridine- 3-carboxamide::US11319299, Example 27	WD repeat-containing protein 5				 294						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=552976	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=552976&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138542084	469796844							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166740	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1cc(C)c(F)c(C)c1)-c1cnc(nc1)N1CCOCC1	InChI=1S/C30H36F2N6O2/c1-18-10-22(11-19(2)28(18)32)29(39)35-26-12-24(23-14-33-30(34-15-23)37-6-8-40-9-7-37)25(31)13-27(26)38-16-20(3)36(5)21(4)17-38/h10-15,20-21H,6-9,16-17H2,1-5H3,(H,35,39)/t20-,21+	HZHCCOARFZTFNJ-OYRHEFFESA-N	552977	4-fluoro-N-[4-fluoro-5- (2-morpholin-4- ylpyrimidin-5-yl)-2- [(3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-3,5- dimethylbenzamide::US11319299, Example 28	WD repeat-containing protein 5				 1.50						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=552977	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=552977&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			137377101	469796845							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166741	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(cc1)N1CCOCC1			552978	N-[4-fluoro-5-(4- morpholin-4-ylphenyl)-2- [(3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 29	WD repeat-containing protein 5				 0.900						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=552978	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=552978&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607829	469796846							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166742	CN1CCN(CC1)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(OC2CCOCC2)nc1	InChI=1S/C28H29F4N5O4/c1-36-6-8-37(9-7-36)24-14-22(29)19(17-2-3-26(34-15-17)41-18-4-10-40-11-5-18)12-23(24)35-27(39)20-16-33-25(38)13-21(20)28(30,31)32/h2-3,12-16,18H,4-11H2,1H3,(H,33,38)(H,35,39)	ZXNZFLDTEWCDMC-UHFFFAOYSA-N	552980	N-[4-fluoro-2-(4- methylpiperazin-1-yl)-5- [6-(oxan-4-yloxy)pyridin- 3-yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 30	WD repeat-containing protein 5				 3.20						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=552980	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=552980&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607831	469796848							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166743	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cnc(nc1)C#N			552981	N-[5-(2-cyanopyrimidin- 5-yl)-4-fluoro-2-[(3S,5R)- 3,4,5-trimethylpiperazin- 1-yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 31	WD repeat-containing protein 5				 1.40						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=552981	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=552981&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607832	469796849							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166744	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(nc1)N1CCOCC1			552982	N-[4-fluoro-5-(6- morpholin-4-ylpyridin-3- yl)-2-[(3S,5R)-3,4,5- trimethylpiperazin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 32	WD repeat-containing protein 5				 0.400						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=552982	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=552982&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607833	469796850							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166745	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cnc(C)nc1			552983	N-[4-fluoro-5-(2- methylpyrimidin-5-yl)-2- [(3S,5R)-3,4,5- trimethylpiperazin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 33	WD repeat-containing protein 5				 0.500						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=552983	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=552983&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607834	469796851							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166746	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)F)-c1cnc(nc1)N1CCOCC1			552984	4-(difluoromethyl)-N-[4- fluoro-5-(2-morpholin-4- ylpyrimidin-5-yl)-2- [(3S,5R)-3,4,5- trimethylpiperazin-1- yl]phenyl]-6-oxo-1H- pyridine-3-carboxamide::US11319299, Example 34	WD repeat-containing protein 5				 0.100						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=552984	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=552984&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607835	469796852							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166747	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cccnc1			552985	N-[4-fluoro-5-pyridin-3- yl-2-[(3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 35	WD repeat-containing protein 5				 2.60						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=552985	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=552985&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607836	469796853							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166748	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccncc1			552986	N-[4-fluoro-5-pyridin-4- yl-2-[(3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 36	WD repeat-containing protein 5				 2.20						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=552986	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=552986&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607837	469796854							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166749	CN(C)[C@@H]1CCN(C1)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cnc(nc1)N1CCOCC1			552987	N-[2-[(3R)-3- (dimethylamino)pyrrolidin- 1-yl]-4-fluoro-5-(2- morpholin-4-ylpyrimidin- 5-yl)phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 37	WD repeat-containing protein 5				 0.200						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=552987	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=552987&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607838	469796855							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166750	CN(C)[C@H]1CCN(C1)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cnc(nc1)N1CCOCC1			552988	N-[2-[(3S)-3- (dimethylamino)pyrrolidin- 1-yl]-4-fluoro-5-(2- morpholin-4-ylpyrimidin- 5-yl)phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 38	WD repeat-containing protein 5				 3.80						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=552988	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=552988&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607839	469796856							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166751	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(OCC2CC2)nc1			552989	N-[5-[6- (cyclopropylmethoxy) pyridin-3-yl]-4-fluoro-2- [(3S,5R)-3,4,5- trimethylpiperazin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 39	WD repeat-containing protein 5				 0.300						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=552989	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=552989&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607840	469796857							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166752	CN(C)c1ncc(cn1)-c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)(F)F)c(cc1F)N1CCN(C)CC1	InChI=1S/C24H25F4N7O2/c1-33(2)23-30-11-14(12-31-23)15-8-19(20(10-18(15)25)35-6-4-34(3)5-7-35)32-22(37)16-13-29-21(36)9-17(16)24(26,27)28/h8-13H,4-7H2,1-3H3,(H,29,36)(H,32,37)	ZHYKLPAWOLFHNY-UHFFFAOYSA-N	552990	N-[5-[2- (dimethylamino)pyrimidin- 5-yl]-4-fluoro-2-(4- methylpiperazin-1- yl)phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 40	WD repeat-containing protein 5				 7.80						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=552990	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=552990&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607841	469796858							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166753	CN1CCN(CC1)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(CN2CCOCC2)nc1	InChI=1S/C28H30F4N6O3/c1-36-4-6-38(7-5-36)25-14-23(29)20(18-2-3-19(33-15-18)17-37-8-10-41-11-9-37)12-24(25)35-27(40)21-16-34-26(39)13-22(21)28(30,31)32/h2-3,12-16H,4-11,17H2,1H3,(H,34,39)(H,35,40)	VJABKHXVGPQFCN-UHFFFAOYSA-N	552991	N-[4-fluoro-2-(4- methylpiperazin-1-yl)-5- [6-(morpholin-4- ylmethyl)pyridin-3- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 41	WD repeat-containing protein 5				 8.60						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=552991	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=552991&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607842	469796859							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166754	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]nc1C(F)(F)F)-c1cnc(nc1)N1CCOCC1			552992	N-[4-fluoro-5-(2- morpholin-4- ylpyrimidin-5-yl)-2- [(3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-3- (trifluoromethyl)-1H- pyrazole-4-carboxamide::US11319299, Example 42	WD repeat-containing protein 5				 9.00						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=552992	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=552992&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			137377675	469796860							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166755	CN1CCN(CC1)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cc(CN2CCOCC2)ccc1F	InChI=1S/C29H30F5N5O3/c1-37-4-6-39(7-5-37)26-15-24(31)20(19-12-18(2-3-23(19)30)17-38-8-10-42-11-9-38)13-25(26)36-28(41)21-16-35-27(40)14-22(21)29(32,33)34/h2-3,12-16H,4-11,17H2,1H3,(H,35,40)(H,36,41)	JYVWWLIWJLNTAD-UHFFFAOYSA-N	525612	US11174250, Example 30::US11319299, Example 43	WD repeat-containing protein 5				 20.0						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=525612	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=525612&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			163199839	463789264							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166756	CN1CCN(CC1)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cccc(CNC2CCCC2)c1	InChI=1S/C30H33F4N5O2/c1-38-9-11-39(12-10-38)27-16-25(31)22(20-6-4-5-19(13-20)17-35-21-7-2-3-8-21)14-26(27)37-29(41)23-18-36-28(40)15-24(23)30(32,33)34/h4-6,13-16,18,21,35H,2-3,7-12,17H2,1H3,(H,36,40)(H,37,41)	MKLAJKBTIBKWMV-UHFFFAOYSA-N	552994	N-(3'-((cyclopentylamino) methyl)-6-fluoro-4-(4- methylpiperazin-1-yl)- [1,1'-biphenyl]-3-yl)-6- oxo-4-(trifluoromethyl)- 1,6-dihydropyridine-3- carboxamide::US11319299, Example 44	WD repeat-containing protein 5				 5.00						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=552994	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=552994&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607843	469796862							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166757	CC1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cccc(CN2CCOCC2)c1			552995	N-(4-(3,4-dimethylpiperazin- 1-yl)-6-fluoro-3'- (morpholinomethyl)-[1,1'- biphenyl]-3-yl)-6-oxo-4- (trifluoromethyl)-1,6- dihydropyridine-3- carboxamide::US11319299, Example 45	WD repeat-containing protein 5				 9.00						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=552995	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=552995&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607844	469796863							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166758	CN1CCN(CC1)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccnc(c1)N1CCOCC1	InChI=1S/C27H28F4N6O3/c1-35-4-6-36(7-5-35)23-15-21(28)18(17-2-3-32-24(12-17)37-8-10-40-11-9-37)13-22(23)34-26(39)19-16-33-25(38)14-20(19)27(29,30)31/h2-3,12-16H,4-11H2,1H3,(H,33,38)(H,34,39)	IIHUZGGGNFKXJX-UHFFFAOYSA-N	552996	N-(4-fluoro-2-(4- methylpiperazin-1-yl)-5- (2-morpholinopyridin-4- yl)phenyl)-6-oxo-4- (trifluoromethyl)-1,6- dihydropyridine-3- carboxamide::US11319299, Example 46::US11319299, Example 60	WD repeat-containing protein 5				 5.00						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=552996	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=552996&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607845	469796864							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166759	CN1CCN(CC1)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cncc(CN2CCOCC2)c1	InChI=1S/C28H30F4N6O3/c1-36-2-4-38(5-3-36)25-13-23(29)20(19-10-18(14-33-15-19)17-37-6-8-41-9-7-37)11-24(25)35-27(40)21-16-34-26(39)12-22(21)28(30,31)32/h10-16H,2-9,17H2,1H3,(H,34,39)(H,35,40)	JLYOQMKXQGIXGN-UHFFFAOYSA-N	552997	N-(4-fluoro-2-(4- methylpiperazin-1-yl)-5- (5-(morpholinomethyl) pyridin-3-yl)phenyl)-6- oxo-4-(trifluoromethyl)-1,6- dihydropyridine-3- carboxamide::US11319299, Example 47	WD repeat-containing protein 5				 19.0						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=552997	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=552997&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607846	469796865							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166760	CN1CCN(CC1)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cncc(CNC2CCOCC2)c1	InChI=1S/C29H32F4N6O3/c1-38-4-6-39(7-5-38)26-13-24(30)21(19-10-18(14-34-16-19)15-35-20-2-8-42-9-3-20)11-25(26)37-28(41)22-17-36-27(40)12-23(22)29(31,32)33/h10-14,16-17,20,35H,2-9,15H2,1H3,(H,36,40)(H,37,41)	CFABCGCXJQFLAB-UHFFFAOYSA-N	552998	N-(4-fluoro-2-(4- methylpiperazin-1-yl)-5- (5-(((tetrahydro-2H-pyran- 4-yl)amino)methyl)pyridin- 3-yl)phenyl)-6-oxo-4- (trifluoromethyl)-1,6- dihydropyridine-3- carboxamide::US11319299, Example 48	WD repeat-containing protein 5				 15.0						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=552998	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=552998&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607847	469796866							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166761	CN1CCN(CC1)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cncc(CNC2CCOC2)c1			552999	(R)-N-(4-fluoro-2-(4- methylpiperazin-1-yl)-5- (5-(((tetrahydrofuran-3- yl)amino)methyl)pyridin- 3-yl)phenyl)-6-oxo-4- (trifluoromethyl)-1,6- dihydropyridine-3- carboxamide::US11319299, Example 49	WD repeat-containing protein 5				 14.0						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=552999	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=552999&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607848	469796867							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166762	C[C@@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cccc(CN2CCOCC2)c1			553000	(R)-N-(4-(3,4- dimethylpiperazin-1-yl)-6- fluoro-3'- (morpholinomethyl)-[1,1'- biphenyl]-3-yl)-6-oxo-4- (trifluoromethyl)-1,6- dihydropyridine-3- carboxamide::US11319299, Example 50	WD repeat-containing protein 5				 12.0						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553000	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553000&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607849	469796868							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166763	C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cccc(CN2CCOCC2)c1			553001	(S)-N-(4-(3,4- dimethylpiperazin-1-yl)-6- fluoro-3'- (morpholinomethyl)-[1,1'- biphenyl]-3-yl)-6-oxo-4- (trifluoromethyl)-1,6- dihydropyridine-3- carboxamide::US11319299, Example 51	WD repeat-containing protein 5				 7.00						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553001	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553001&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607850	469796869							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166764	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cccc(CN2CCOCC2)c1			553002	N-(6-fluoro-3'- (morpholinomethyl)-4- ((3R,5S)-3,4,5- trimethylpiperazin-1-yl)- [1,1-biphenyl]-3-yl)-6- oxo-4-(trifluoromethyl)- 1,6-dihydropyridine-3- carboxamide::US11319299, Example 52	WD repeat-containing protein 5				 6.00						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553002	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553002&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607851	469796870							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166765	CN(C)C1CCN(C1)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cccc(CN2CCOCC2)c1			553003	N-(4-(3-(dimethylamino) pyrrolidin-1-yl)-6-fluoro-3'- (morpholinomethyl)-[1,1'- biphenyl]-3-yl)-6-oxo-4- (trifluoromethyl)-1,6- dihydropyridine-3- carboxamide::US11319299, Example 53	WD repeat-containing protein 5				 5.70						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553003	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553003&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607852	469796871							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166766	CN1CCN(CC1)c1cc(Cl)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cccc(CN2CCOCC2)c1	InChI=1S/C29H31ClF3N5O3/c1-36-5-7-38(8-6-36)26-16-24(30)21(20-4-2-3-19(13-20)18-37-9-11-41-12-10-37)14-25(26)35-28(40)22-17-34-27(39)15-23(22)29(31,32)33/h2-4,13-17H,5-12,18H2,1H3,(H,34,39)(H,35,40)	LQOMVNOXBXIXGZ-UHFFFAOYSA-N	553004	N-(6-chloro-4-(4- methylpiperazin-1-yl)-3'- (morpholinomethyl)-[1,1- biphenyl]-3-yl)-6-oxo-4- (trifluoromethy1)-1,6- dihydropyridine-3- carboxamide::US11319299, Example 54	WD repeat-containing protein 5				 51.0						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553004	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553004&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607853	469796872							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166767	COc1cc(N2C[C@H](C)N(C)[C@H](C)C2)c(NC(=O)c2c[nH]c(=O)cc2C(F)(F)F)cc1-c1cnc(nc1)N1CCOCC1			553005	N-[4-methoxy-5-(2- morpholin-4- ylpyrimidin-5-yl)-2-[rac- (3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299,  Example Table6.593::US11319299, Example 55	WD repeat-containing protein 5				>200						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553005	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553005&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607854	469796873							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166768	CN1CCN(CC1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cnc(nc1)N1CCOCC1	InChI=1S/C26H28F3N7O3/c1-34-4-6-35(7-5-34)22-3-2-17(18-14-31-25(32-15-18)36-8-10-39-11-9-36)12-21(22)33-24(38)19-16-30-23(37)13-20(19)26(27,28)29/h2-3,12-16H,4-11H2,1H3,(H,30,37)(H,33,38)	QNXFOPYFFZOHCX-UHFFFAOYSA-N	553006	N-(2-(4-methylpiperazin- 1-yl)-5-(2- morpholinopyrimidin-5- yl)phenyl)-6-oxo-4- (trifluoromethyl)-1,6- dihydropyridine-3- carboxamide::US11319299, Comp. No. 56::US11319299, Example 56	WD repeat-containing protein 5				 17.5						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553006	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553006&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607855	469796874							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166769	CN1CCN(CC1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cccc(CN2CCOCC2)c1	InChI=1S/C29H32F3N5O3/c1-35-7-9-37(10-8-35)26-6-5-22(21-4-2-3-20(15-21)19-36-11-13-40-14-12-36)16-25(26)34-28(39)23-18-33-27(38)17-24(23)29(30,31)32/h2-6,15-18H,7-14,19H2,1H3,(H,33,38)(H,34,39)	DJOVLOYCGXNVPI-UHFFFAOYSA-N	50164794	CHEMBL3798846::US11174250, Example Table4.1.1::US11319299, Comp. No. 57	WD repeat-containing protein 5				 36.0						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50164794	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50164794&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	35Q	4QL1	91623360	341097539		CHEMBL3798846					1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166770	C[C@H]1CN(C[C@@H](C)N1C)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cnc(nc1)N1CCOCC1			553008	N-(5-(2- morpholinopyrimidin-5- yl)-2-((3R,5S)-3,4,5- trimethylpiperazin-1- yl)phenyl)-6-oxo-4- (trifluoromethyl)-1,6- dihydropyridine-3- carboxamide::US11319299,  Example Table6.58::US11319299, Comp. No. 58::US11319299, Example 58	WD repeat-containing protein 5				 3.50						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553008	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553008&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607856	469796876							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166771	C[C@H]1CN(C[C@@H](C)N1C)c1cc(c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cnc(nc1)N1CCOCC1)C(F)(F)F			553009	N-[5-(2-morpholin-4- ylpyrimidin-5-yl)-2-[rac- (3R,5S)-3,4,5- trimethylpiperazin-1-yl]- 4-(trifluoromethyl)phenyl]- 6-oxo-4-(trifluoromethyl)- 1H-pyridine-3-carboxamide::US11319299,  Example Table6.592::US11319299, Example 59	WD repeat-containing protein 5				>200						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553009	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553009&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607857	469796877							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166772	CN1CCN(CC1)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccnc(c1)N1CCOCC1	InChI=1S/C27H28F4N6O3/c1-35-4-6-36(7-5-35)23-15-21(28)18(17-2-3-32-24(12-17)37-8-10-40-11-9-37)13-22(23)34-26(39)19-16-33-25(38)14-20(19)27(29,30)31/h2-3,12-16H,4-11H2,1H3,(H,33,38)(H,34,39)	IIHUZGGGNFKXJX-UHFFFAOYSA-N	552996	N-(4-fluoro-2-(4- methylpiperazin-1-yl)-5- (2-morpholinopyridin-4- yl)phenyl)-6-oxo-4- (trifluoromethyl)-1,6- dihydropyridine-3- carboxamide::US11319299, Example 46::US11319299, Example 60	WD repeat-containing protein 5				 4.79						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=552996	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=552996&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607845	469796864							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166773	C[C@H]1CN(C[C@@H](C)N1C)c1cc(C)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cnc(nc1)N1CCOCC1			553011	N-[4-methyl-5-(2- morpholin-4-ylpyrimidin- 5-yl)-2-[rac-(3R,5S)- 3,4,5-trimethylpiperazin- 1-yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299,  Example Table6.591::US11319299, Example 61	WD repeat-containing protein 5				 26.0						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553011	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553011&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607858	469796878							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166774	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc2OCOc2c1			553012	N-[5-(1,3-benzodioxol-5- yl)4-fluoro-2-[rac- (3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 63	WD repeat-containing protein 5				 0.694						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553012	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553012&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607859	469796879							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166775	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(NC(C)=O)nc1			553013	N-[5-(6-acetamidopyridin- 3-yl)-4-fluoro-2-[rac-(3R,5S)- 3,4,5-trimethylpiperazin- 1-yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 64	WD repeat-containing protein 5				 0.199						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553013	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553013&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607860	469796880							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166776	COc1cc(=O)[nH]cc1C(=O)Nc1cc(c(F)cc1N1C[C@H](C)N(C)[C@H](C)C1)-c1cnc(nc1)N1CCOCC1			553014	N-[4-fluoro-5-(2- morpholin-4-ylpyrimidin- 5-yl)-2-[rac-(3R,5S)- 3,4,5-trimethylpiperazin- 1-yl]phenyl]-4-methoxy- 6-oxo-1H-pyridine-3- carboxamide::US11319299, Example 65	WD repeat-containing protein 5				 57.2						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553014	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553014&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607861	469796881							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166777	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccnc(OCC2CC2)c1			553016	N-[5-[2- (cyclopropylmethoxy) pyridin-4-yl]-4-fluoro-2- [rac-(3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 66	WD repeat-containing protein 5				 1.16						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553016	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553016&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607862	469796883							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166778	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccccc1CNC1CCCCC1			553017	N-[5-[2- (cyclohexylamino) methyl]phenyl]-4-fluoro-2- [rac-(3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 67	WD repeat-containing protein 5				 4.82						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553017	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553017&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607863	469796884							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166779	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(N2CCOCC2)c(Cl)c1			553018	N-[5-(3-chloro-4- morpholin-4-ylphenyl)-4- fluoro-2-[rac-(3R,5S)- 3,4,5-trimethylpiperazin- 1-yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 68	WD repeat-containing protein 5				 1.34						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553018	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553018&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607864	469796885							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166780	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc2OCCCOc2c1			553019	N-[5-(3,4-dihydro-2H- 1,5-benzodioxepin-7-yl)- 4-fluoro-2-[rac-(3R,5S)- 3,4,5-trimethylpiperazin- 1-yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 69	WD repeat-containing protein 5				 0.225						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553019	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553019&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607865	469796886							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166781	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc2OCCOc2c1			553020	N-[5-(2,3-dihydro-1,4- benzodioxin-6-yl)-4- fluoro-2-[rac-(3R,5S)- 3,4,5-trimethylpiperazin- 1-yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 70	WD repeat-containing protein 5				 0.429						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553020	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553020&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607866	469796887							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166782	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc2N(C)CCOc2c1			553021	N-[4-fluoro-5-(4-methyl- 2,3-dihydro-1,4- benzoxazin-7-yl)-2-[rac- (3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 71	WD repeat-containing protein 5				 0.623						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553021	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553021&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607867	469796888							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166783	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cnc(NC(C)=O)nc1			553022	N-[5-(2- acetamidopyrimidin-5- yl)-4-fluoro-2-[rac- (3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 72	WD repeat-containing protein 5				 0.823						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553022	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553022&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607868	469796889							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166784	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCN(CC1)c1ccccc1			553023	N-[4-fluoro-5-(1-phenyl- 3,6-dihydro-2H-pyridin- 4-yl)-2-[rac-(3R,5S)- 3,4,5-trimethylpiperazin- 1-yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 73	WD repeat-containing protein 5				 3.63						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553023	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553023&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607869	469796890							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166785	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1ccccc1)-c1cnc(nc1)N1CCOCC1	InChI=1S/C28H33FN6O2/c1-19-17-35(18-20(2)33(19)3)26-14-24(29)23(13-25(26)32-27(36)21-7-5-4-6-8-21)22-15-30-28(31-16-22)34-9-11-37-12-10-34/h4-8,13-16,19-20H,9-12,17-18H2,1-3H3,(H,32,36)/t19-,20+	YQFNSMANDGRLTE-BGYRXZFFSA-N	553024	N-[4-fluoro-5-(2- morpholin-4-ylpyrimidin- 5-yl)-2-[rac-(3R,5S)- 3,4,5-trimethylpiperazin- 1-yl]phenyl]benzamide::US11319299, Example 74	WD repeat-containing protein 5				 253						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553024	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553024&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138541780	469796891							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166786	COc1cc(ccc1F)C(=O)Nc1cc(c(F)cc1N1C[C@H](C)N(C)[C@H](C)C1)-c1cnc(nc1)N1CCOCC1	InChI=1S/C29H34F2N6O3/c1-18-16-37(17-19(2)35(18)3)26-13-24(31)22(21-14-32-29(33-15-21)36-7-9-40-10-8-36)12-25(26)34-28(38)20-5-6-23(30)27(11-20)39-4/h5-6,11-15,18-19H,7-10,16-17H2,1-4H3,(H,34,38)/t18-,19+	AUTAOAUKUDQTNY-KDURUIRLSA-N	553025	4-fluoro-N-[4-fluoro-5- (2-morpholin-4- ylpyrimidin-5-yl)-2-[rac- (3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-3- methoxybenzamide::US11319299, Example 75	WD repeat-containing protein 5				 40.9						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553025	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553025&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			137377106	469796892							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166787	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1cc(Cl)cc(Cl)c1)-c1cnc(nc1)N1CCOCC1	InChI=1S/C28H31Cl2FN6O2/c1-17-15-37(16-18(2)35(17)3)26-12-24(31)23(20-13-32-28(33-14-20)36-4-6-39-7-5-36)11-25(26)34-27(38)19-8-21(29)10-22(30)9-19/h8-14,17-18H,4-7,15-16H2,1-3H3,(H,34,38)/t17-,18+	FULWLPHLUKCSAQ-HDICACEKSA-N	553026	3,5-dichloro-N-[4-fluoro- 5-(2-morpholin-4- ylpyrimidin-5-yl)-2-[rac- (3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]benzamide::US11319299, Example 76	WD repeat-containing protein 5				 2.07						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553026	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553026&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138541616	469796893							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166788	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1n[nH]c(=O)cc1C(F)(F)F)-c1cnc(nc1)N1CCOCC1			553027	N-[4-fluoro-5-(2- morpholin-4-ylpyrimidin- 5-yl)-2-[rac-(3R,5S)- 3,4,5-trimethylpiperazin- 1-yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridazine-3-carboxamide::US11319299, Example 77	WD repeat-containing protein 5				 4.43						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553027	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553027&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607870	469796894							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166789	C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1ccccc1)-c1cnc(nc1)N1CCOCC1	InChI=1S/C27H31FN6O2/c1-19-18-34(9-8-32(19)2)25-15-23(28)22(14-24(25)31-26(35)20-6-4-3-5-7-20)21-16-29-27(30-17-21)33-10-12-36-13-11-33/h3-7,14-17,19H,8-13,18H2,1-2H3,(H,31,35)/t19-/m0/s1	LXSJNAPOPPRPNG-IBGZPJMESA-N	553028	N-[4-fluoro-5-(2- morpholin-4-ylpyrimidin- 5-yl)-2-[rac-(3R)-3,4- dimethylpiperazin-1- yl]phenyl]benzamide::US11319299, Example 78	WD repeat-containing protein 5				 17.9						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553028	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553028&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			137377400	469796895							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166790	C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1ccco1)-c1cnc(nc1)N1CCOCC1	InChI=1S/C25H29FN6O3/c1-17-16-32(6-5-30(17)2)22-13-20(26)19(12-21(22)29-24(33)23-4-3-9-35-23)18-14-27-25(28-15-18)31-7-10-34-11-8-31/h3-4,9,12-15,17H,5-8,10-11,16H2,1-2H3,(H,29,33)/t17-/m0/s1	MBGVGLVZOTWFQD-KRWDZBQOSA-N	553029	N-[4-fluoro-5-(2- morpholin-4-ylpyrimidin- 5-yl)-2-[rac-(3R)-3,4- dimethylpiperazin-1- yl]phenyl]furan-2- carboxamide::US11319299, Example 79	WD repeat-containing protein 5				>200						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553029	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553029&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138551477	469796896							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166791	C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1cccnc1)-c1cnc(nc1)N1CCOCC1	InChI=1S/C26H30FN7O2/c1-18-17-34(7-6-32(18)2)24-13-22(27)21(12-23(24)31-25(35)19-4-3-5-28-14-19)20-15-29-26(30-16-20)33-8-10-36-11-9-33/h3-5,12-16,18H,6-11,17H2,1-2H3,(H,31,35)/t18-/m0/s1	BDGULTBESBEFNG-SFHVURJKSA-N	553030	N-[4-fluoro-5-(2- morpholin-4-ylpyrimidin- 5-yl)-2-[rac-(3R)-3,4- dimethylpiperazin-1- yl]phenyl]pyridine-3- carboxamide::US11319299, Example 80	WD repeat-containing protein 5				>200						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553030	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553030&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138551357	469796897							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166792	C[C@H]1CN(CCN1C)c1cc(Cl)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cnc(nc1)N1CCOCC1			553031	N-[4-chloro-5-(2- morpholin-4-ylpyrimidin- 5-yl)-2-[rac-(3R)-3,4- dimethylpiperazin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 81	WD repeat-containing protein 5				 11.1						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553031	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553031&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607871	469796898							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166793	C[C@H]1CN(C[C@@H](C)N1C)c1cc(Cl)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cnc(nc1)N1CCOCC1			553032	N-[4-chloro-5-(2- morpholin-4-ylpyrimidin- 5-yl)-2-[rac-(3R,5S)- 3,4,5-trimethylpiperazin- 1-yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299,  Example Table6.82::US11319299, Example 82	WD repeat-containing protein 5				 10.6						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553032	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553032&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607872	469796899							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166794	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccnc(c1)N1CCOCC1			553033	N-[4-fluoro-5-(2- morpholin-4-ylpyridin-4- yl)-2-[rac-(3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 83	WD repeat-containing protein 5				 0.391						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553033	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553033&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607873	469796900							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166795	COCCOc1ccc(cn1)-c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)(F)F)c(cc1F)N1C[C@H](C)N(C)[C@H](C)C1			553034	N-[4-fluoro-5-[6-(2- methoxyethoxy)pyridin- 3-yl]-2-[rac-(3R,5S)- 3,4,5-trimethylpiperazin- 1-yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 84	WD repeat-containing protein 5				 0.338						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553034	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553034&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607874	469796901							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166796	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cccc(c1)N1CCOCC1			553035	N-[4-fluoro-5-(3-morpholin- 4-ylphenyl)-2-[rac-(3R,5S)- 3,4,5-trimethylpiperazin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 85	WD repeat-containing protein 5				 0.703						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553035	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553035&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607875	469796902							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166797	COc1ccccc1C(=O)Nc1cc(c(F)cc1N1C[C@H](C)N(C)[C@H](C)C1)-c1cnc(nc1)N1CCOCC1	InChI=1S/C29H35FN6O3/c1-19-17-36(18-20(2)34(19)3)26-14-24(30)23(21-15-31-29(32-16-21)35-9-11-39-12-10-35)13-25(26)33-28(37)22-7-5-6-8-27(22)38-4/h5-8,13-16,19-20H,9-12,17-18H2,1-4H3,(H,33,37)/t19-,20+	KWCHDMIGMKTOPV-BGYRXZFFSA-N	553036	N-[4-fluoro-5-(2- morpholin-4-ylpyrimidin- 5-yl)-2-[rac-(3R,5S)- 3,4,5-trimethylpiperazin- 1-yl]phenyl]-2- methoxybenzamide::US11319299, Example 86	WD repeat-containing protein 5				 204						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553036	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553036&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			137377514	469796903							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166798	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1ccc(F)cc1Cl)-c1cnc(nc1)N1CCOCC1	InChI=1S/C28H31ClF2N6O2/c1-17-15-37(16-18(2)35(17)3)26-12-24(31)22(19-13-32-28(33-14-19)36-6-8-39-9-7-36)11-25(26)34-27(38)21-5-4-20(30)10-23(21)29/h4-5,10-14,17-18H,6-9,15-16H2,1-3H3,(H,34,38)/t17-,18+	OHHYLCGVVMQZEM-HDICACEKSA-N	553037	2-chloro-4-fluoro-N-[4- fluoro-5-(2-morpholin-4- ylpyrimidin-5-yl)-2-[rac- (3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]benzamide::US11319299, Example 87	WD repeat-containing protein 5				 8.21						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553037	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553037&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138541641	469796904							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166799	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1cc(F)ccc1C(F)(F)F)-c1cnc(nc1)N1CCOCC1	InChI=1S/C29H31F5N6O2/c1-17-15-40(16-18(2)38(17)3)26-12-24(31)21(19-13-35-28(36-14-19)39-6-8-42-9-7-39)11-25(26)37-27(41)22-10-20(30)4-5-23(22)29(32,33)34/h4-5,10-14,17-18H,6-9,15-16H2,1-3H3,(H,37,41)/t17-,18+	BEDPKUFFMNDEMS-HDICACEKSA-N	553038	5-fluoro-N-[4-fluoro-5- (2-morpholin-4- ylpyrimidin-5-yl)-2-[rac- (3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-2-(trifluoromethyl) benzamide::US11319299, Example 88	WD repeat-containing protein 5				 24.1						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553038	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553038&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			137376898	469796905							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166800	COc1cccc(c1)C(=O)Nc1cc(c(F)cc1N1C[C@H](C)N(C)[C@H](C)C1)-c1cnc(nc1)N1CCOCC1	InChI=1S/C29H35FN6O3/c1-19-17-36(18-20(2)34(19)3)27-14-25(30)24(22-15-31-29(32-16-22)35-8-10-39-11-9-35)13-26(27)33-28(37)21-6-5-7-23(12-21)38-4/h5-7,12-16,19-20H,8-11,17-18H2,1-4H3,(H,33,37)/t19-,20+	OOLSQXVQUZSLSY-BGYRXZFFSA-N	553039	N-[4-fluoro-5-(2- morpholin-4-ylpyrimidin- 5-yl)-2-[rac-(3R,5S)- 3,4,5-trimethylpiperazin- 1-yl]phenyl]-3- methoxybenzamide::US11319299, Example 89	WD repeat-containing protein 5				 33.8						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553039	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553039&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			137377064	469796906							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166801	COCCOc1ccc(cc1)-c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)(F)F)c(cc1F)N1C[C@H](C)N(C)[C@H](C)C1			553040	N-[4-fluoro-5-[4-(2- methoxyethoxy)phenyl]- 2-[rac-(3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 90	WD repeat-containing protein 5				 0.441						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553040	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553040&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607876	469796907							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166802	CC(C)COc1ncc(cc1Cl)-c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)(F)F)c(cc1F)N1C[C@H](C)N(C)[C@H](C)C1			553041	N-[5-[5-chloro-6-(2- methylpropoxy)pyridin-3- yl]-4-fluoro-2-[rac- (3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 91	WD repeat-containing protein 5				 4.47						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553041	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553041&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607877	469796908							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166803	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(OCC2CC2)c(Cl)c1			553042	N-[5-[3-chloro-4- (cyclopropylmethoxy) phenyl]-4-fluoro-2-[rac- (3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 92	WD repeat-containing protein 5				 10.9						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553042	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553042&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607878	469796909							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166804	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1cn(C)c(=O)cc1C(F)(F)F)-c1cnc(nc1)N1CCOCC1	InChI=1S/C29H33F4N7O3/c1-17-14-40(15-18(2)38(17)4)25-11-23(30)20(19-12-34-28(35-13-19)39-5-7-43-8-6-39)9-24(25)36-27(42)21-16-37(3)26(41)10-22(21)29(31,32)33/h9-13,16-18H,5-8,14-15H2,1-4H3,(H,36,42)/t17-,18+	NNAMONHIEIUUHG-HDICACEKSA-N	553043	N-[4-fluoro-5-(2- morpholin-4-ylpyrimidin- 5-yl)-2-[rac-(3R,5S)- 3,4,5-trimethylpiperazin- 1-yl]phenyl]-1-methyl-6- oxo-4-(trifluoromethyl) pyridine-3-carboxamide::US11319299, Example 93	WD repeat-containing protein 5				 2.17						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553043	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553043&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			137376930	469796910							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166805	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCOCC1			553044	N-[5-(3,6-dihydro-2H- pyran-4-yl)-4-fluoro-2- [rac-(3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 94	WD repeat-containing protein 5				 4.06						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553044	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553044&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607879	469796911							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166806	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCNCC1			553045	N-[4-fluoro-2-[rac-(3R,5S)- 3,4,5-trimethylpiperazin-1- yl]-5-(1,2,3,6- tetrahydropyridin-4- yl)phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 95	WD repeat-containing protein 5				 7.18						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553045	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553045&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607880	469796912							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166807	C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1c[nH]nc1C(F)(F)F)-c1cnc(nc1)N1CCOCC1			553046	N-[4-fluoro-5-(2- morpholin-4-ylpyrimidin- 5-yl)-2-[rac-(3R)-3,4- dimethylpiperazin-1- yl]phenyl]-3- (trifluoromethyl)-1H- pyrazole-4-carboxamide::US11319299, Example 96	WD repeat-containing protein 5				 7.71						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553046	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553046&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138551433	469796913							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166808	C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1cc(C)c(F)c(C)c1)-c1cnc(nc1)N1CCOCC1	InChI=1S/C29H34F2N6O2/c1-18-11-21(12-19(2)27(18)31)28(38)34-25-13-23(22-15-32-29(33-16-22)36-7-9-39-10-8-36)24(30)14-26(25)37-6-5-35(4)20(3)17-37/h11-16,20H,5-10,17H2,1-4H3,(H,34,38)/t20-/m0/s1	QTPUIDDNZCGPCD-FQEVSTJZSA-N	553047	4-fluoro-N-[4-fluoro-5- (2-morpholin-4- ylpyrimidin-5-yl)-2-[rac- (3R)-3,4- dimethylpiperazin-1- yl]phenyl]-3,5- dimethylbenzamide::US11319299, Example 97	WD repeat-containing protein 5				 2.21						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553047	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553047&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138551314	469796914							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166809	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cc(Cl)c(O)c(c1)C#N			553048	N-[5-(3-chloro-5-cyano- 4-hydroxyphenyl)-4- fluoro-2-[rac-(3R,5S)- 3,4,5-trimethylpiperazin- 1-yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 98	WD repeat-containing protein 5				 19.5						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553048	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553048&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607881	469796915							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166810	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cnc(OCc2ccccc2)c(c1)C#N			553049	N-[5-(5-cyano-6- phenylmethoxypyridin-3- yl)-4-fluoro-2-[rac- (3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 99	WD repeat-containing protein 5				 11.1						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553049	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553049&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607882	469796916							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166811	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(cc1)C#N			553050	N-[5-(4-cyanophenyl)-4- fluoro-2-[rac-(3R,5S)- 3,4,5-trimethylpiperazin- 1-yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 100	WD repeat-containing protein 5				 0.508						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553050	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553050&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607883	469796917							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166812	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(OC2CCOCC2)nc1			553051	N-[4-fluoro-5-[6-(oxan-4- yloxy)pyridin-3-yl]-2- [rac-(3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 101	WD repeat-containing protein 5				 0.320						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553051	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553051&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607884	469796918							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166813	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cccc(c1)C#N			553052	N-[5-(3-cyanophenyl)-4- fluoro-2-[rac-(3R,5S)- 3,4,5-trimethylpiperazin- 1-yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 102	WD repeat-containing protein 5				 2.08						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553052	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553052&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607885	469796919							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166814	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cnc(nc1)N(C)C			553053	N-[5-[2-(dimethylamino) pyrimidin-5-yl]-4-fluoro-2- [rac-(3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 103	WD repeat-containing protein 5				 0.168						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553053	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553053&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607886	469796920							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166815	COc1cc(cnc1OC)-c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)(F)F)c(cc1F)N1C[C@H](C)N(C)[C@H](C)C1			553054	N-[5-(5,6- dimethoxypyridin-3-yl)- 4-fluoro-2-[rac-(3R,5S)- 3,4,5-trimethylpiperazin- 1-yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 104	WD repeat-containing protein 5				 2.41						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553054	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553054&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607887	469796921							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166816	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1cccc2OCOc12)-c1cnc(nc1)N1CCOCC1	InChI=1S/C29H33FN6O4/c1-18-15-36(16-19(2)34(18)3)25-12-23(30)22(20-13-31-29(32-14-20)35-7-9-38-10-8-35)11-24(25)33-28(37)21-5-4-6-26-27(21)40-17-39-26/h4-6,11-14,18-19H,7-10,15-17H2,1-3H3,(H,33,37)/t18-,19+	FAJAAYYRXGYELC-KDURUIRLSA-N	553055	N-[4-fluoro-5-(2- morpholin-4-ylpyrimidin- 5-yl)-2-[rac-(3R,5S)- 3,4,5-trimethylpiperazin- 1-yl]phenyl]-1,3- benzodioxole-4-carboxamide::US11319299, Example 105	WD repeat-containing protein 5				 466						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553055	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553055&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138541651	469796922							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166817	COc1ccc(cc1)C(=O)Nc1cc(c(F)cc1N1C[C@H](C)N(C)[C@H](C)C1)-c1cnc(nc1)N1CCOCC1	InChI=1S/C29H35FN6O3/c1-19-17-36(18-20(2)34(19)3)27-14-25(30)24(22-15-31-29(32-16-22)35-9-11-39-12-10-35)13-26(27)33-28(37)21-5-7-23(38-4)8-6-21/h5-8,13-16,19-20H,9-12,17-18H2,1-4H3,(H,33,37)/t19-,20+	NSSDRFOXNAVQTL-BGYRXZFFSA-N	553056	N-[4-fluoro-5-(2- morpholin-4-ylpyrimidin- 5-yl)-2-[rac-(3R,5S)- 3,4,5-trimethylpiperazin- 1-yl]phenyl]-4- methoxybenzamide::US11319299, Example 106	WD repeat-containing protein 5				 5400						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553056	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553056&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138541931	469796923							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166818	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1ccc(F)cc1)-c1cnc(nc1)N1CCOCC1	InChI=1S/C28H32F2N6O2/c1-18-16-36(17-19(2)34(18)3)26-13-24(30)23(12-25(26)33-27(37)20-4-6-22(29)7-5-20)21-14-31-28(32-15-21)35-8-10-38-11-9-35/h4-7,12-15,18-19H,8-11,16-17H2,1-3H3,(H,33,37)/t18-,19+	RPYOPIZSDSNFQO-KDURUIRLSA-N	553057	4-fluoro-N-[4-fluoro-5- (2-morpholin-4- ylpyrimidin-5-yl)-2-[rac- (3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]benzamide::US11319299, Example 107	WD repeat-containing protein 5				 137						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553057	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553057&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			137376932	469796924							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166819	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cc(F)cc(c1)N1CCOCC1			553058	N-[4-fluoro-5-(3-fluoro- 5-morpholin-4-ylphenyl)- 2-[rac-(3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 108	WD repeat-containing protein 5				 3.91						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553058	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553058&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607888	469796925							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166820	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1ccccc1Cl)-c1cnc(nc1)N1CCOCC1	InChI=1S/C28H32ClFN6O2/c1-18-16-36(17-19(2)34(18)3)26-13-24(30)22(12-25(26)33-27(37)21-6-4-5-7-23(21)29)20-14-31-28(32-15-20)35-8-10-38-11-9-35/h4-7,12-15,18-19H,8-11,16-17H2,1-3H3,(H,33,37)/t18-,19+	SFNOCEQUUVRJGE-KDURUIRLSA-N	553059	2-chloro-N-[4-fluoro-5- (2-morpholin-4- ylpyrimidin-5-yl)-2-[rac- (3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]benzamide::US11319299, Example 109	WD repeat-containing protein 5				 175						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553059	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553059&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			137376811	469796926							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167541	CN1CCN(CC1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cnc(nc1)N1CCOCC1	InChI=1S/C26H28F3N7O3/c1-34-4-6-35(7-5-34)22-3-2-17(18-14-31-25(32-15-18)36-8-10-39-11-9-36)12-21(22)33-24(38)19-16-30-23(37)13-20(19)26(27,28)29/h2-3,12-16H,4-11H2,1H3,(H,30,37)(H,33,38)	QNXFOPYFFZOHCX-UHFFFAOYSA-N	553006	N-(2-(4-methylpiperazin- 1-yl)-5-(2- morpholinopyrimidin-5- yl)phenyl)-6-oxo-4- (trifluoromethyl)-1,6- dihydropyridine-3- carboxamide::US11319299, Comp. No. 56::US11319299, Example 56	WD repeat-containing protein 5				 17.5						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553006	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553006&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607855	469796874							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167542	CN1CCN(CC1)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cnc(nc1)N1CCOCC1	InChI=1S/C26H27F4N7O3/c1-35-2-4-36(5-3-35)22-12-20(27)17(16-13-32-25(33-14-16)37-6-8-40-9-7-37)10-21(22)34-24(39)18-15-31-23(38)11-19(18)26(28,29)30/h10-15H,2-9H2,1H3,(H,31,38)(H,34,39)	QNEXYXLSJZBQJZ-UHFFFAOYSA-N	552948	N-[4-fluoro-2-(4- methylpiperazin-1-yl)-5- (2-morpholin-4- ylpyrimidin-5-yl)phenyl]- 6-oxo-4-(trifluoromethyl)- 1H-pyridine-3-carboxamide::US11319299, Comp. No. 3::US11319299, Example 3	WD repeat-containing protein 5				 1.50						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=552948	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=552948&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607804	469796817							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167544	CN1CCN(CC1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cccc(CN2CCOCC2)c1	InChI=1S/C29H32F3N5O3/c1-35-7-9-37(10-8-35)26-6-5-22(21-4-2-3-20(15-21)19-36-11-13-40-14-12-36)16-25(26)34-28(39)23-18-33-27(38)17-24(23)29(30,31)32/h2-6,15-18H,7-14,19H2,1H3,(H,33,38)(H,34,39)	DJOVLOYCGXNVPI-UHFFFAOYSA-N	50164794	CHEMBL3798846::US11174250, Example Table4.1.1::US11319299, Comp. No. 57	WD repeat-containing protein 5				 36.0						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50164794	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50164794&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	35Q	4QL1	91623360	341097539		CHEMBL3798846					1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167545	CN1CCN(CC1)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cccc(CN2CCOCC2)c1	InChI=1S/C29H31F4N5O3/c1-36-5-7-38(8-6-36)26-16-24(30)21(20-4-2-3-19(13-20)18-37-9-11-41-12-10-37)14-25(26)35-28(40)22-17-34-27(39)15-23(22)29(31,32)33/h2-4,13-17H,5-12,18H2,1H3,(H,34,39)(H,35,40)	GVIBWIRSZYKTTI-UHFFFAOYSA-N	552933	N-[4-fluoro-2-(4- methylpiperazin-1-yl)-5- [3-(morpholin-4- ylmethyl)phenyl]phenyl]- 6-oxo-4-(trifluoromethyl)- 1H-pyridine-3-carboxamide::US11319299, Comp. No. 2::US11319299, Example 2	WD repeat-containing protein 5				 11.0						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=552933	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=552933&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607803	469796802							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167547	C[C@H]1CN(C[C@@H](C)N1C)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cnc(nc1)N1CCOCC1			553008	N-(5-(2- morpholinopyrimidin-5- yl)-2-((3R,5S)-3,4,5- trimethylpiperazin-1- yl)phenyl)-6-oxo-4- (trifluoromethyl)-1,6- dihydropyridine-3- carboxamide::US11319299,  Example Table6.58::US11319299, Comp. No. 58::US11319299, Example 58	WD repeat-containing protein 5				 3.50						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553008	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553008&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607856	469796876							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167548	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cnc(nc1)N1CCOCC1			552953	N-[4-fluoro-5-(2- morpholin-4-ylpyrimidin- 5-yl)-2-[(3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299,  Example Table6.8::US11319299, Comp. No. 8::US11319299, Example 8	WD repeat-containing protein 5				 0.323						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=552953	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=552953&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607809	469796822							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166821	COc1cccc(C(=O)Nc2cc(c(F)cc2N2C[C@H](C)N(C)[C@H](C)C2)-c2cnc(nc2)N2CCOCC2)c1F	InChI=1S/C29H34F2N6O3/c1-18-16-37(17-19(2)35(18)3)25-13-23(30)22(20-14-32-29(33-15-20)36-8-10-40-11-9-36)12-24(25)34-28(38)21-6-5-7-26(39-4)27(21)31/h5-7,12-15,18-19H,8-11,16-17H2,1-4H3,(H,34,38)/t18-,19+	OVOXAOOAEWEYMJ-KDURUIRLSA-N	553060	2-fluoro-N-[4-fluoro-5- (2-morpholin-4- ylpyrimidin-5-yl)-2-[rac- (3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-3- methoxybenzamide::US11319299, Example 110	WD repeat-containing protein 5				 1730						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553060	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553060&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			137377604	469796927							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166822	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1ccc(F)c(F)c1)-c1cnc(nc1)N1CCOCC1	InChI=1S/C28H31F3N6O2/c1-17-15-37(16-18(2)35(17)3)26-12-23(30)21(20-13-32-28(33-14-20)36-6-8-39-9-7-36)11-25(26)34-27(38)19-4-5-22(29)24(31)10-19/h4-5,10-14,17-18H,6-9,15-16H2,1-3H3,(H,34,38)/t17-,18+	ODUGGTLVMXHSCS-HDICACEKSA-N	553061	3,4-difluoro-N-[4-fluoro- 5-(2-morpholin-4- ylpyrimidin-5-yl)-2-[rac- (3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]benzamide::US11319299, Example 111	WD repeat-containing protein 5				 70.6						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553061	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553061&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138541593	469796928							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166823	COc1ccc(cc1)-c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)(F)F)c(cc1F)N1C[C@H](C)N(C)[C@H](C)C1			553062	N-[4-fluoro-5-(4- methoxyphenyl)-2-[rac- (3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 112	WD repeat-containing protein 5				 2.44						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553062	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553062&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607889	469796929							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166824	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(OCC2CC2)cc1			553063	N-[5-[4- (cyclopropylmethoxy) phenyl]-4-fluoro-2-[rac- (3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 113	WD repeat-containing protein 5				 0.858						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553063	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553063&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607890	469796930							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166825	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(cc1)N1CCCC1			553064	N-[4-fluoro-5-(4- pyrrolidin-1-ylphenyl)-2- [rac-(3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 114	WD repeat-containing protein 5				 4.06						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553064	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553064&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607891	469796931							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166826	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1cccc(NC(C)=O)c1)-c1cnc(nc1)N1CCOCC1	InChI=1S/C30H36FN7O3/c1-19-17-38(18-20(2)36(19)4)28-14-26(31)25(23-15-32-30(33-16-23)37-8-10-41-11-9-37)13-27(28)35-29(40)22-6-5-7-24(12-22)34-21(3)39/h5-7,12-16,19-20H,8-11,17-18H2,1-4H3,(H,34,39)(H,35,40)/t19-,20+	KQPFDVCEDGWLHG-BGYRXZFFSA-N	553066	3-acetamido-N-[4-fluoro- 5-(2-morpholin-4- ylpyrimidin-5-yl)-2-[rac- (3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]benzamide::US11319299, Example 115	WD repeat-containing protein 5				>200						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553066	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553066&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138541766	469796933							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166827	C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1nn(C)c2ccccc12)-c1cnc(nc1)N1CCOCC1	InChI=1S/C29H33FN8O2/c1-19-18-38(9-8-35(19)2)26-15-23(30)22(20-16-31-29(32-17-20)37-10-12-40-13-11-37)14-24(26)33-28(39)27-21-6-4-5-7-25(21)36(3)34-27/h4-7,14-17,19H,8-13,18H2,1-3H3,(H,33,39)/t19-/m0/s1	AWVUBEKBYVCYAU-IBGZPJMESA-N	553067	N-[4-fluoro-5-(2- morpholin-4-ylpyrimidin- 5-yl)-2-[rac-(3R)-3,4- dimethylpiperazin-1- yl]phenyl]-1- methylindazole-3- carboxamide::US11319299, Example 116	WD repeat-containing protein 5				 76.8						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553067	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553067&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138551369	469796934							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166828	C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1nn(C)c2ccccc12)-c1ccc(cc1)N1CCOCC1	InChI=1S/C31H35FN6O2/c1-21-20-38(13-12-35(21)2)29-19-26(32)25(22-8-10-23(11-9-22)37-14-16-40-17-15-37)18-27(29)33-31(39)30-24-6-4-5-7-28(24)36(3)34-30/h4-11,18-19,21H,12-17,20H2,1-3H3,(H,33,39)/t21-/m0/s1	OTTVJSRLQRMGRM-NRFANRHFSA-N	553068	N-[4-fluoro-5-(4- morpholin-4-ylphenyl)-2- [rac-(3R)-3,4- dimethylpiperazin-1- yl]phenyl]-1- methylindazole-3- carboxamide::US11319299, Example 117	WD repeat-containing protein 5				 42.8						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553068	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553068&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138551372	469796935							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166829	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cccc(CN(C)C2COC2)c1			553069	N-[4-fluoro-5-[3- [[methyl(oxetan-3-yl) amino]methyl]phenyl]- 2-[rac-(3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 118	WD repeat-containing protein 5				 4.53						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553069	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553069&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607892	469796936							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166830	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cccc(CN2CCC(F)CC2)c1			553070	N-[4-fluoro-5-[3-[(4- fluoropiperidin-1- yl)methyl]phenyl]-2-[rac- (3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 119	WD repeat-containing protein 5				 5.12						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553070	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553070&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607893	469796937							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166831	Fc1cc(N2CCN3CCOCC3C2)c(NC(=O)c2c[nH]c(=O)cc2C(F)(F)F)cc1-c1cnc(nc1)N1CCOCC1			553071	N-[2-(3,4,6,7,9,9a- hexahydro-1H-pyrazino [2,1-c][1,4]oxazin-8-yl)- 4-fluoro-5-(2-morpholin-4- ylpyrimidin-5-yl)phenyl]- 6-oxo-4-(trifluoromethyl)- 1H-pyridine-3-carboxamide::US11319299, Example 120	WD repeat-containing protein 5				>200						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553071	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553071&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607894	469796938							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166832	C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1cnn(C)c1)-c1cnc(nc1)N1CCOCC1	InChI=1S/C25H31FN8O2/c1-17-15-34(5-4-31(17)2)23-11-21(26)20(10-22(23)30-24(35)19-14-29-32(3)16-19)18-12-27-25(28-13-18)33-6-8-36-9-7-33/h10-14,16-17H,4-9,15H2,1-3H3,(H,30,35)/t17-/m0/s1	FCMGRGPJJVKGQL-KRWDZBQOSA-N	553072	N-[4-fluoro-5-(2- morpholin-4-ylpyrimidin- 5-yl)-2-[rac-(3R)-3,4- dimethylpiperazin-1- yl]phenyl]-1- methylpyrazole-4- carboxamide::US11319299, Example 121	WD repeat-containing protein 5				 33.4						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553072	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553072&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138551414	469796939							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166833	C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1cnn(C)c1)-c1ccc(cc1)N1CCOCC1	InChI=1S/C27H33FN6O2/c1-19-17-34(9-8-31(19)2)26-15-24(28)23(14-25(26)30-27(35)21-16-29-32(3)18-21)20-4-6-22(7-5-20)33-10-12-36-13-11-33/h4-7,14-16,18-19H,8-13,17H2,1-3H3,(H,30,35)/t19-/m0/s1	YIPFNRRSQBRXIB-IBGZPJMESA-N	553073	N-[4-fluoro-5-(4- morpholin-4-ylphenyl)-2- [rac-(3R)-3,4- dimethylpiperazin-1- yl]phenyl]-1- methylpyrazole-4- carboxamide::US11319299, Example 122	WD repeat-containing protein 5				 70.2						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553073	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553073&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138551366	469796940							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166834	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cnc(O)c(c1)C#N			553074	N-[5-(5-cyano-6- hydroxypyridin-3-yl)-4- fluoro-2-[rac-(3R,5S)- 3,4,5-trimethylpiperazin- 1-yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 123	WD repeat-containing protein 5				 9.88						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553074	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553074&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607895	469796941							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166835	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(N2CCOCC2)c(F)c1			553075	N-[4-fluoro-5-(3-fluoro- 4-morpholin-4-ylphenyl)- 2-[rac-(3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 124	WD repeat-containing protein 5				 0.439						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553075	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553075&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607896	469796942							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166836	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cccc(OCC2CC2)c1			553076	N-[5-[3- (cyclopropylmethoxy) phenyl]-4-fluoro-2-[rac- (3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 125	WD repeat-containing protein 5				 10.9						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553076	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553076&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607897	469796943							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166837	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1cccc(c1)N(C)C)-c1cnc(nc1)N1CCOCC1	InChI=1S/C30H38FN7O2/c1-20-18-38(19-21(2)36(20)5)28-15-26(31)25(23-16-32-30(33-17-23)37-9-11-40-12-10-37)14-27(28)34-29(39)22-7-6-8-24(13-22)35(3)4/h6-8,13-17,20-21H,9-12,18-19H2,1-5H3,(H,34,39)/t20-,21+	VREFXFONEXZPNJ-OYRHEFFESA-N	553077	3-(dimethylamino)-N-[4- fluoro-5-(2-morpholin-4- ylpyrimidin-5-yl)-2-[rac- (3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]benzamide::US11319299, Example 126	WD repeat-containing protein 5				 3500						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553077	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553077&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138541794	469796944							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166838	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1cocn1)-c1cnc(nc1)N1CCOCC1	InChI=1S/C25H30FN7O3/c1-16-12-33(13-17(2)31(16)3)23-9-20(26)19(8-21(23)30-24(34)22-14-36-15-29-22)18-10-27-25(28-11-18)32-4-6-35-7-5-32/h8-11,14-17H,4-7,12-13H2,1-3H3,(H,30,34)/t16-,17+	HFFYDYCECLNSNX-CALCHBBNSA-N	553078	N-[4-fluoro-5-(2- morpholin-4-ylpyrimidin- 5-yl)-2-[rac-(3R,5S)- 3,4,5-trimethylpiperazin- 1-yl]pheny]-1,3-oxazole- 4-carboxamide::US11319299, Example 127	WD repeat-containing protein 5				>200						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553078	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553078&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			137377222	469796945							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166839	C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1cn(C)c(=O)cc1C(F)(F)F)-c1cnc(nc1)N1CCOCC1	InChI=1S/C28H31F4N7O3/c1-17-15-39(5-4-36(17)2)24-12-22(29)19(18-13-33-27(34-14-18)38-6-8-42-9-7-38)10-23(24)35-26(41)20-16-37(3)25(40)11-21(20)28(30,31)32/h10-14,16-17H,4-9,15H2,1-3H3,(H,35,41)/t17-/m0/s1	CGLBRJYXTDVSFE-KRWDZBQOSA-N	553079	N-[4-fluoro-5-(2- morpholin-4-ylpyrimidin- 5-yl)-2-[rac-(3R)-3,4- dimethylpiperazin-1- yl]phenyl]-1-methyl-6- oxo-4-(trifluoromethyl) pyridine-3-carboxamide::US11319299, Example 128	WD repeat-containing protein 5				 6.36						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553079	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553079&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138551373	469796946							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166840	C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1cn(C)c(=O)cc1C(F)(F)F)-c1ccc(cc1)N1CCOCC1	InChI=1S/C30H33F4N5O3/c1-19-17-39(9-8-36(19)2)27-16-25(31)22(20-4-6-21(7-5-20)38-10-12-42-13-11-38)14-26(27)35-29(41)23-18-37(3)28(40)15-24(23)30(32,33)34/h4-7,14-16,18-19H,8-13,17H2,1-3H3,(H,35,41)/t19-/m0/s1	LVEWQKTYQLEZCT-IBGZPJMESA-N	553080	N-[4-fluoro-5-(4- morpholin-4-ylphenyl)-2- [rac-(3R)-3,4- dimethylpiperazin-1- yl]phenyl]-1-methyl-6- oxo-4-(trifluoromethyl) pyridine-3-carboxamide::US11319299, Example 129	WD repeat-containing protein 5				 12.9						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553080	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553080&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138551547	469796947							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166841	CC(C)Oc1ncc(cn1)-c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)(F)F)c(cc1F)N1C[C@H](C)N(C)[C@H](C)C1			553081	N-[4-fluoro-5-(2-propan- 2-yloxypyrimidin-5-yl)-2- [rac-(3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 130	WD repeat-containing protein 5				 0.656						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553081	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553081&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607898	469796948							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166842	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(nc1)C#N			553082	N-[5-(6-cyanopyridin-3- yl)-4-fluoro-2-[rac- (3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 131	WD repeat-containing protein 5				 2.43						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553082	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553082&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607899	469796949							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166843	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cnc(C#N)c(C)c1			553083	N-[5-(6-cyano-5- methylpyridin-3-yl)-4- fluoro-2-[rac-(3R,5S)- 3,4,5-trimethylpiperazin- 1-yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 132	WD repeat-containing protein 5				 1.40						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553083	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553083&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607900	469796950							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166844	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccnc(c1)C#N			553084	N-[5-(2-cyanopyridin-4- yl)-4-fluoro-2-[rac- (3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 133	WD repeat-containing protein 5				 1.33						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553084	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553084&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607901	469796951							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166845	COc1cc(cc(n1)C(F)(F)F)-c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)(F)F)c(cc1F)N1C[C@H](C)N(C)[C@H](C)C1			553085	N-[4-fluoro-5-[2- methoxy-6-(trifluoromethyl) pyridin-4-yl]-2-[rac-(3R,5S)- 3,4,5-trimethylpiperazin- 1-yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 134	WD repeat-containing protein 5				 1.01						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553085	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553085&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607902	469796952							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166846	COc1cc(cc(C)n1)-c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)(F)F)c(cc1F)N1C[C@H](C)N(C)[C@H](C)C1			553086	N-[4-fluoro-5-(2- methoxy-6- methylpyridin-4-yl)-2- [rac-(3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 135	WD repeat-containing protein 5				 2.81						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553086	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553086&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607903	469796953							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166847	COc1ncc(cc1C(F)(F)F)-c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)(F)F)c(cc1F)N1C[C@H](C)N(C)[C@H](C)C1			553087	N-[4-fluoro-5-[6- methoxy-5-(trifluoromethyl) pyridin-3-yl]-2-[rac-(3R,5S)- 3,4,5-trimethylpiperazin- 1-yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 136	WD repeat-containing protein 5				 0.463						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553087	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553087&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607904	469796954							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166848	COc1cc(C#N)c(cn1)C(=O)Nc1cc(c(F)cc1N1C[C@H](C)N(C)[C@H](C)C1)-c1cnc(nc1)N1CCOCC1	InChI=1S/C29H33FN8O3/c1-18-16-38(17-19(2)36(18)3)26-11-24(30)22(21-13-33-29(34-14-21)37-5-7-41-8-6-37)10-25(26)35-28(39)23-15-32-27(40-4)9-20(23)12-31/h9-11,13-15,18-19H,5-8,16-17H2,1-4H3,(H,35,39)/t18-,19+	VDIMFVDCAXCMDQ-KDURUIRLSA-N	553088	4-cyano-N-[4-fluoro-5- (2-morpholin-4- ylpyrimidin-5-yl)-2-[rac- (3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-6- methoxypyridine-3- carboxamide::US11319299, Example 137	WD repeat-containing protein 5				 19.7						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553088	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553088&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			137377130	469796955							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166849	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1cccc(Cl)c1)-c1cnc(nc1)N1CCOCC1	InChI=1S/C28H32ClFN6O2/c1-18-16-36(17-19(2)34(18)3)26-13-24(30)23(12-25(26)33-27(37)20-5-4-6-22(29)11-20)21-14-31-28(32-15-21)35-7-9-38-10-8-35/h4-6,11-15,18-19H,7-10,16-17H2,1-3H3,(H,33,37)/t18-,19+	OLDYACLPQYPFEF-KDURUIRLSA-N	553089	3-chloro-N-[4-fluoro-5- (2-morpholin-4- ylpyrimidin-5-yl)-2-[rac- (3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]benzamide::US11319299, Example 138	WD repeat-containing protein 5				 11.3						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553089	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553089&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			137376760	469796956							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166850	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c(Cl)cccc1Cl)-c1cnc(nc1)N1CCOCC1	InChI=1S/C28H31Cl2FN6O2/c1-17-15-37(16-18(2)35(17)3)25-12-23(31)20(19-13-32-28(33-14-19)36-7-9-39-10-8-36)11-24(25)34-27(38)26-21(29)5-4-6-22(26)30/h4-6,11-14,17-18H,7-10,15-16H2,1-3H3,(H,34,38)/t17-,18+	JADSUCOKLXUVPD-HDICACEKSA-N	553090	2,6-dichloro-N-[4-fluoro- 5-(2-morpholin-4- ylpyrimidin-5-yl)-2-[rac- (3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]benzamide::US11319299, Example 139	WD repeat-containing protein 5				 5.86						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553090	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553090&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			137377485	469796957							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166851	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1cccc(Cl)c1F)-c1cnc(nc1)N1CCOCC1	InChI=1S/C28H31ClF2N6O2/c1-17-15-37(16-18(2)35(17)3)25-12-23(30)21(19-13-32-28(33-14-19)36-7-9-39-10-8-36)11-24(25)34-27(38)20-5-4-6-22(29)26(20)31/h4-6,11-14,17-18H,7-10,15-16H2,1-3H3,(H,34,38)/t17-,18+	WNJWEGPRXFMJHB-HDICACEKSA-N	553091	3-chloro-2-fluoro-N-[4- fluoro-5-(2-morpholin-4- ylpyrimidin-5-yl)-2-[rac- (3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]benzamide::US11319299, Example 140	WD repeat-containing protein 5				 18.8						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553091	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553091&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138541777	469796958							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166852	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1ccccc1C(F)(F)F)-c1cnc(nc1)N1CCOCC1	InChI=1S/C29H32F4N6O2/c1-18-16-39(17-19(2)37(18)3)26-13-24(30)22(20-14-34-28(35-15-20)38-8-10-41-11-9-38)12-25(26)36-27(40)21-6-4-5-7-23(21)29(31,32)33/h4-7,12-15,18-19H,8-11,16-17H2,1-3H3,(H,36,40)/t18-,19+	MGPGDGUJGAWPOJ-KDURUIRLSA-N	553092	N-[4-fluoro-5-(2- morpholin-4-ylpyrimidin- 5-yl)-2-[rac-(3R,5S)- 3,4,5-trimethylpiperazin- 1-yl]phenyl]-2- (trifluoromethyl)benzamide::US11319299, Example 141	WD repeat-containing protein 5				 16.2						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553092	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553092&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			137376854	469796959							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166853	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(nc1)N(C)C			553093	N-[5-[6- (dimethylamino)pyridin- 3-yl]-4-fluoro-2-[rac- (3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 142	WD repeat-containing protein 5				 0.985						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553093	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553093&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607905	469796960							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166854	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCN(CC1)C(=O)OC(C)(C)C			553094	US11319299, Example 143::tert-butyl 4-[2-fluoro-5- [[6-oxo-4-(trifluoromethyl)- 1H-pyridine-3-carbonyl] amino]-4-[rac-(3R,5S)-3,4,5- trimethylpiperazin-1-yl] phenyl]-3,6-dihydro-2H- pyridine-1-carboxylate	WD repeat-containing protein 5				 1.24						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553094	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553094&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607906	469796961							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166855	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(cc1)C(F)(F)F			553095	N-[4-fluoro-2-[rac- (3R,5S)-3,4,5- trimethylpiperazin-1-yl]- 5-[4-(trifluoromethyl) phenyl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 144	WD repeat-containing protein 5				 6.06						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553095	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553095&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607907	469796962							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166856	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(OC(F)(F)F)cc1			553096	N-[4-fluoro-2-[rac- (3R,5S)-3,4,5- trimethylpiperazin-1-yl]- 5-[4-(trifluoromethoxy) phenyl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 145	WD repeat-containing protein 5				 6.83						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553096	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553096&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607908	469796963							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166857	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccccc1			553097	N-[4-fluoro-5-phenyl-2- [rac-(3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 146	WD repeat-containing protein 5				 6.02						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553097	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553097&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607909	469796964							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166858	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(Cl)cc1			553098	N-[5-(4-chlorophenyl)-4- fluoro-2-[rac-(3R,5S)- 3,4,5-trimethylpiperazin- 1-yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 147	WD repeat-containing protein 5				 4.44						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553098	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553098&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607910	469796965							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166859	COc1ccc(CN2CCC(=CC2)c2cc(NC(=O)c3c[nH]c(=O)cc3C(F)(F)F)c(cc2F)N2C[C@H](C)N(C)[C@H](C)C2)cc1			553099	N-[4-fluoro-5-[1-[(4- methoxyphenyl)methyl]- 3,6-dihydro-2H-pyridin- 4-yl]-2-[rac-(3R,5S)- 3,4,5-trimethylpiperazin- 1-yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 148	WD repeat-containing protein 5				 0.540						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553099	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553099&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607911	469796966							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166860	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cnnc(C)c1			553100	N-[4-fluoro-5-(6- methylpyridazin-4-yl)-2- [rac-(3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 149	WD repeat-containing protein 5				 4.65						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553100	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553100&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607912	469796967							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166861	CC(C)CN1CCC(=CC1)c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)(F)F)c(cc1F)N1C[C@H](C)N(C)[C@H](C)C1			553101	N-[4-fluoro-5-[1-(2- methylpropyl)-3,6- dihydro-2H-pyridin-4-yl]- 2-[rac-(3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 150	WD repeat-containing protein 5				 9.00						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553101	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553101&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607913	469796968							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166862	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCN(CC2CC2)CC1			553102	N-[5-[1-(cyclopropylmethyl)- 3,6-dihydro-2H-pyridin-4-yl]- 4-fluoro-2-[rac-(3R,5S)- 3,4,5-trimethylpiperazin- 1-yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 151	WD repeat-containing protein 5				 7.46						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553102	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553102&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607914	469796969							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166863	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCN(CCC(F)(F)F)CC1			553103	N-[4-fluoro-2-[rac-(3R,5S)- 3,4,5-trimethylpiperazin-1- yl]-5-[1-(3,3,3-trifluoropropyl)- 3,6-dihydro-2H-pyridin-4- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 152	WD repeat-containing protein 5				 6.33						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553103	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553103&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607915	469796970							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166864	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCN(Cc2ccc(F)cc2)CC1			553104	N-[4-fluoro-5-[1-[(4- fluorophenyl)methyl]-3,6- dihydro-2H-pyridin-4-yl]- 2-[rac-(3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 153	WD repeat-containing protein 5				 1.08						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553104	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553104&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607916	469796971							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166865	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCN(Cc2cccnc2)CC1			553105	N-[4-fluoro-5-[1- (pyridin-3-ylmethyl)-3,6- dihydro-2H-pyridin-4-yl]- 2-[rac-(3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 154	WD repeat-containing protein 5				 5.46						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553105	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553105&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607917	469796972							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166866	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCN(Cc2ccsc2)CC1			553106	N-[4-fluoro-2-[rac-(3R,5S)- 3,4,5-trimethylpiperazin-1- yl]-5-[1-(thiophen-3-ylmethyl)- 3,6-dihydro-2H-pyridin-4-yl] phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 155	WD repeat-containing protein 5				 4.76						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553106	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553106&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607918	469796973							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166867	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cncc(OCC2CC2)c1			553107	N-[5-[5- (cyclopropylmethoxy) pyridin-3-yl]-4-fluoro-2-[rac- (3R,5S)-3,4,5- trimethylpiperazin-1-yl] phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 156	WD repeat-containing protein 5				 8.61						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553107	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553107&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607919	469796974							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166868	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(O)nc1			553108	N-[4-fluoro-5-(6- hydroxypyridin-3-yl)-2- [rac-(3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 157	WD repeat-containing protein 5				 2.16						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553108	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553108&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607920	469796975							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166869	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cnc(nc1)N1CCNCC1			553109	N-[4-fluoro-5-(2- piperazin-1-ylpyrimidin- 5-yl)-2-[rac-(3R,5S)- 3,4,5-trimethylpiperazin- 1-yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 158	WD repeat-containing protein 5				 0.345						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553109	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553109&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607921	469796976							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166870	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1cc(F)cc(Cl)c1)-c1cnc(nc1)N1CCOCC1	InChI=1S/C28H31ClF2N6O2/c1-17-15-37(16-18(2)35(17)3)26-12-24(31)23(20-13-32-28(33-14-20)36-4-6-39-7-5-36)11-25(26)34-27(38)19-8-21(29)10-22(30)9-19/h8-14,17-18H,4-7,15-16H2,1-3H3,(H,34,38)/t17-,18+	CKGNOGCUSZOQTO-HDICACEKSA-N	553110	3-chloro-5-fluoro-N-[4- fluoro-5-(2-morpholin-4- ylpyrimidin-5-yl)-2-[rac- (3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]benzamide::US11319299, Example 159	WD repeat-containing protein 5				 29.0						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553110	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553110&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138541925	469796977							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166871	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1cc(F)cc(F)c1)-c1cnc(nc1)N1CCOCC1	InChI=1S/C28H31F3N6O2/c1-17-15-37(16-18(2)35(17)3)26-12-24(31)23(20-13-32-28(33-14-20)36-4-6-39-7-5-36)11-25(26)34-27(38)19-8-21(29)10-22(30)9-19/h8-14,17-18H,4-7,15-16H2,1-3H3,(H,34,38)/t17-,18+	CQLFTMLQRLXTEG-HDICACEKSA-N	553111	3,5-difluoro-N-[4-fluoro- 5-(2-morpholin-4- ylpyrimidin-5-yl)-2-[rac- (3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]benzamide::US11319299, Example 160	WD repeat-containing protein 5				 26.8						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553111	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553111&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138541982	469796978							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166872	C[C@H]1CN(C[C@@H](C)O1)c1ncc(cn1)-c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)(F)F)c(cc1F)N1C[C@H](C)N(C)[C@H](C)C1			553112	N-[4-fluoro-5-[2-[rac- (2R,6S)-2,6- dimethylmorpholin-4- yl]pyrimidin-5-yl]-2-[rac- (3S,5R)-3,4,5- trimethylpiperazin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 161	WD repeat-containing protein 5				 1.000						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553112	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553112&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607922	469796979							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166873	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCN(Cc2nccs2)CC1			553113	N-[4-fluoro-2-[rac-(3R,5S)- 3,4,5-trimethylpiperazin-1- yl]-5-[1-(1,3-thiazol-2- ylmethyl)-3,6-dihydro- 2H-pyridin-4-yl]phenyl]- 6-oxo-4-(trifluoromethyl)- 1H-pyridine-3-carboxamide::US11319299, Example 162	WD repeat-containing protein 5				 2.83						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553113	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553113&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607923	469796980							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166874	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCN(Cc2cnc(C)o2)CC1			553114	N-[4-fluoro-5-[1-[(2- methyl-1,3-oxazol-5- yl)methyl]-3,6-dihydro- 2H-pyridin-4-yl]-2-[rac- (3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 163	WD repeat-containing protein 5				 4.05						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553114	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553114&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607924	469796981							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166875	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCN(Cc2cnn(C)c2)CC1			553115	N-[4-fluoro-5-[1-[(1- methylpyrazol-4- yl)methyl]-3,6-dihydro- 2H-pyridin-4-yl]-2-[rac- (3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 164	WD repeat-containing protein 5				 1.43						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553115	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553115&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607925	469796982							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166876	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCN(Cc2ccc(cc2)N2CCOCC2)CC1			553116	N-[4-fluoro-5-[1-[(4- morpholin-4-ylphenyl) methyl]-3,6-dihydro-2H- pyridin-4-yl]-2-[rac- (3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 165	WD repeat-containing protein 5				 6.28						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553116	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553116&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607926	469796983							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166877	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCN(Cc2ccc(cc2)N2CCN(C)CC2)CC1			553117	N-[4-fluoro-5-[1-[[4-(4- methylpiperazin-1- yl)phenyl]methyl]-3,6- dihydro-2H-pyridin-4-yl]- 2-[rac-(3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 166	WD repeat-containing protein 5				 0.230						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553117	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553117&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607927	469796984							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166878	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCN(CC2CCOCC2)CC1			553118	N-[4-fluoro-5-[1-(oxan-4- ylmethyl)-3,6-dihydro- 2H-pyridin-4-yl]-2-[rac- (3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 167	WD repeat-containing protein 5				 5.76						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553118	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553118&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607928	469796985							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166879	CN(C)[C@@H]1CCN(C1)c1cc(F)c(cc1NC(=O)c1cc(Cl)cc(Cl)c1)-c1cnc(nc1)N1CCOCC1	InChI=1S/C27H29Cl2FN6O2/c1-34(2)21-3-4-36(16-21)25-13-23(30)22(18-14-31-27(32-15-18)35-5-7-38-8-6-35)12-24(25)33-26(37)17-9-19(28)11-20(29)10-17/h9-15,21H,3-8,16H2,1-2H3,(H,33,37)/t21-/m1/s1	NSHJMTHDTWJICB-OAQYLSRUSA-N	553119	3,5-dichloro-N-[4-fluoro- 5-(2-morpholin-4- ylpyrimidin-5-yl)-2-[rac- (3R)-3-(dimethylamino) pyrrolidin-1-yl]phenyl] benzamide::US11319299, Example 168	WD repeat-containing protein 5				 30.0						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553119	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553119&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			137376768	469796986							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166880	CN(C)[C@@H]1CCN(C1)c1cc(F)c(cc1NC(=O)c1cc(Cl)cc(Cl)c1)-c1ccc(cc1)N1CCOCC1	InChI=1S/C29H31Cl2FN4O2/c1-34(2)24-7-8-36(18-24)28-17-26(32)25(19-3-5-23(6-4-19)35-9-11-38-12-10-35)16-27(28)33-29(37)20-13-21(30)15-22(31)14-20/h3-6,13-17,24H,7-12,18H2,1-2H3,(H,33,37)/t24-/m1/s1	AXJMRSMXXRBOOZ-XMMPIXPASA-N	553120	3,5-dichloro-N-[4-fluoro- 5-(4-morpholin-4- ylphenyl)-2-[rac-(3R)-3- (dimethylamino)pyrrolidin-1- yl]phenyl]benzamide::US11319299, Example 169	WD repeat-containing protein 5				 122						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553120	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553120&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			137376862	469796987							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166881	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cnc(N2CCOCC2)c(c1)C#N			553121	N-[5-(5-cyano-6- morpholin-4-ylpyridin-3- yl)-4-fluoro-2-[rac- (3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 170	WD repeat-containing protein 5				 1.17						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553121	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553121&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607929	469796988							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166882	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cnc(N2CCOCC2)c(C)c1			553122	N-[4-fluoro-5-(5-methyl- 6-morpholin-4-ylpyridin- 3-yl)-2-[rac-(3R,5S)- 3,4,5-trimethylpiperazin- 1-yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 171	WD repeat-containing protein 5				 2.50						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553122	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553122&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607930	469796989							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166883	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cnc2NCCc2c1			553123	N-[5-(2,3-dihydro-1H- pyrrolo[2,3-b]pyridin-5- yl)-4-fluoro-2-[rac- (3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 172	WD repeat-containing protein 5				 10.3						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553123	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553123&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607931	469796990							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166884	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cncc(c1)C(F)(F)F			553124	N-[4-fluoro-2-[rac- (3R,5S)-3,4,5- trimethylpiperazin-1-yl]- 5-[5-(trifluoromethyl)pyridin- 3-yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 173	WD repeat-containing protein 5				 2.78						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553124	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553124&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607932	469796991							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166885	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cncc(c1)C(=O)NC(C)(C)C			553125	N-[5-[5-(tert- butylcarbamoyl)pyridin- 3-yl]-4-fluoro-2-[rac- (3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 174	WD repeat-containing protein 5				 1.53						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553125	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553125&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607933	469796992							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166886	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1cc(Cl)cc(c1)C(F)(F)F)-c1cnc(nc1)N1CCOCC1	InChI=1S/C29H31ClF4N6O2/c1-17-15-40(16-18(2)38(17)3)26-12-24(31)23(20-13-35-28(36-14-20)39-4-6-42-7-5-39)11-25(26)37-27(41)19-8-21(29(32,33)34)10-22(30)9-19/h8-14,17-18H,4-7,15-16H2,1-3H3,(H,37,41)/t17-,18+	VXEIFCUMDIIQDX-HDICACEKSA-N	553126	3-chloro-N-[4-fluoro-5- (2-morpholin-4- ylpyrimidin-5-yl)-2-[rac- (3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-5- (trifluoromethyl) benzamide::US11319299, Example 175	WD repeat-containing protein 5				 20.6						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553126	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553126&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			137376973	469796993							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166887	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1cc(F)cc(c1)C(F)(F)F)-c1cnc(nc1)N1CCOCC1	InChI=1S/C29H31F5N6O2/c1-17-15-40(16-18(2)38(17)3)26-12-24(31)23(20-13-35-28(36-14-20)39-4-6-42-7-5-39)11-25(26)37-27(41)19-8-21(29(32,33)34)10-22(30)9-19/h8-14,17-18H,4-7,15-16H2,1-3H3,(H,37,41)/t17-,18+	LZRCBEUAJJZLNT-HDICACEKSA-N	553127	3-fluoro-N-[4-fluoro-5- (2-morpholin-4- ylpyrimidin-5-yl)-2-[rac- (3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-5- (trifluoromethyl)benzamide::US11319299, Example 176	WD repeat-containing protein 5				 50.9						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553127	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553127&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			137376943	469796994							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166888	CN(C)[C@@H]1CCN(C1)c1cc(F)c(cc1NC(=O)c1cn[nH]c1)-c1ccc(cc1)N1CCOCC1			553128	N-[4-fluoro-5-(4- morpholin-4-ylphenyl)-2- [rac-(3R)-3- (dimethylamino)pyrrolidin-1- yl]phenyl]-1H-pyrazole-4- carboxamide::US11319299, Example 177	WD repeat-containing protein 5				>200						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553128	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553128&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			137377510	469796995							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166889	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cncc(C)c1			553129	N-[4-fluoro-5-(5- methylpyridin-3-yl)-2- [rac-(3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 178	WD repeat-containing protein 5				 6.50						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553129	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553129&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607934	469796996							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166890	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cncc(c1)C(N)=O			553130	N-[5-(5-carbamoylpyridin-3- yl)-4-fluoro-2-[rac-(3R,5S)- 3,4,5-trimethylpiperazin- 1-yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 179	WD repeat-containing protein 5				 11.5						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553130	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553130&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607935	469796997							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166891	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1cn(C)c(=O)cc1C(F)(F)F)-c1cncc(c1)C(F)(F)F	InChI=1S/C27H26F7N5O2/c1-14-11-39(12-15(2)38(14)4)23-8-21(28)18(16-5-17(10-35-9-16)26(29,30)31)6-22(23)36-25(41)19-13-37(3)24(40)7-20(19)27(32,33)34/h5-10,13-15H,11-12H2,1-4H3,(H,36,41)/t14-,15+	NZDCGPATBOYWEA-GASCZTMLSA-N	553131	N-[4-fluoro-2-[rac- (3R,5S)-3,4,5- trimethylpiperazin-1-yl]-5- [5-(trifluoromethyl)pyridin-3- yl]phenyl]-1-methyl-6- oxo-4-(trifluoromethyl) pyridine-3-carboxamide::US11319299, Example 180	WD repeat-containing protein 5				 35.4						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553131	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553131&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138541817	469796998							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166892	C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1nc(C)cs1)-c1cnc(nc1)N1CCOCC1	InChI=1S/C25H30FN7O2S/c1-16-15-36-24(29-16)23(34)30-21-10-19(18-12-27-25(28-13-18)32-6-8-35-9-7-32)20(26)11-22(21)33-5-4-31(3)17(2)14-33/h10-13,15,17H,4-9,14H2,1-3H3,(H,30,34)/t17-/m0/s1	GKEHOVGMOLDKIT-KRWDZBQOSA-N	553132	N-[4-fluoro-5-(2- morpholin-4-ylpyrimidin- 5-yl)-2-[rac-(3R)-3,4- dimethylpiperazin-1- yl]phenyl]-4-methyl-1,3- thiazole-2-carboxamide::US11319299, Example 181	WD repeat-containing protein 5				>200						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553132	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553132&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138551529	469796999							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166893	C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1csc(CN(C)C)n1)-c1cnc(nc1)N1CCOCC1	InChI=1S/C27H35FN8O2S/c1-18-15-36(6-5-34(18)4)24-12-21(28)20(19-13-29-27(30-14-19)35-7-9-38-10-8-35)11-22(24)32-26(37)23-17-39-25(31-23)16-33(2)3/h11-14,17-18H,5-10,15-16H2,1-4H3,(H,32,37)/t18-/m0/s1	WZTJEHAHJNDWAR-SFHVURJKSA-N	553133	2-[(dimethylamino)methyl]- N-[4-fluoro-5-(2- morpholin-4-ylpyrimidin- 5-yl)-2-[rac-(3R)-3,4- dimethylpiperazin-1- yl]phenyl]-1,3-thiazole-4- carboxamide::US11319299, Example 182	WD repeat-containing protein 5				>200						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553133	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553133&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138551382	469797000							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166894	C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1n[nH]cc1Cl)-c1cnc(nc1)N1CCOCC1			553134	4-chloro-N-[4-fluoro-5- (2-morpholin-4- ylpyrimidin-5-yl)-2-[rac- (3R)-3,4-dimethylpiperazin-1- yl]phenyl]-1H-pyrazole- 3-carboxamide::US11319299, Example 183	WD repeat-containing protein 5				 113						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553134	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553134&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138551302	469797001							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166895	CN(C)[C@@H]1CCN(C1)c1cc(F)c(cc1NC(=O)c1cn(C)c(=O)cc1C(F)(F)F)-c1cnc(nc1)N1CCOCC1	InChI=1S/C28H31F4N7O3/c1-36(2)18-4-5-39(15-18)24-12-22(29)19(17-13-33-27(34-14-17)38-6-8-42-9-7-38)10-23(24)35-26(41)20-16-37(3)25(40)11-21(20)28(30,31)32/h10-14,16,18H,4-9,15H2,1-3H3,(H,35,41)/t18-/m1/s1	OZQJEGFKGIVCCF-GOSISDBHSA-N	553135	N-[4-fluoro-5-(2- morpholin-4-ylpyrimidin- 5-yl)-2-[rac-(3R)-3- (dimethylamino)pyrrolidin-1- yl]phenyl]-1-methyl-6-oxo-4- (trifluoromethyl)pyridine- 3-carboxamide::US11319299, Example 184	WD repeat-containing protein 5				 9.80						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553135	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553135&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138541731	469797002							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166896	CN(C)[C@@H]1CCN(C1)c1cc(F)c(cc1NC(=O)c1c[nH]nc1C(F)(F)F)-c1cnc(nc1)N1CCOCC1			553136	N-[4-fluoro-5-(2- morpholin-4-ylpyrimidin- 5-yl)-2-[rac-(3R)-3- (dimethylamino)pyrrolidin-1- yl]phenyl]-3-(trifluoromethyl)- 1H-pyrazole-4-carboxamide::US11319299, Example 185	WD repeat-containing protein 5				 29.8						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553136	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553136&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138541771	469797003							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166897	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1cccc(c1)C(F)(F)F)-c1cnc(nc1)N1CCOCC1	InChI=1S/C29H32F4N6O2/c1-18-16-39(17-19(2)37(18)3)26-13-24(30)23(21-14-34-28(35-15-21)38-7-9-41-10-8-38)12-25(26)36-27(40)20-5-4-6-22(11-20)29(31,32)33/h4-6,11-15,18-19H,7-10,16-17H2,1-3H3,(H,36,40)/t18-,19+	XNGURGUFKUEZJJ-KDURUIRLSA-N	553137	N-[4-fluoro-5-(2- morpholin-4-ylpyrimidin- 5-yl)-2-[rac-(3R,5S)- 3,4,5-trimethylpiperazin- 1-yl]phenyl]-3- (trifluoromethyl)benzamide::US11319299, Example 186	WD repeat-containing protein 5				 40.2						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553137	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553137&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			137376904	469797004							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166898	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1cncnc1C(F)(F)F)-c1cnc(nc1)N1CCOCC1	InChI=1S/C27H30F4N8O2/c1-16-13-39(14-17(2)37(16)3)23-9-21(28)19(18-10-33-26(34-11-18)38-4-6-41-7-5-38)8-22(23)36-25(40)20-12-32-15-35-24(20)27(29,30)31/h8-12,15-17H,4-7,13-14H2,1-3H3,(H,36,40)/t16-,17+	RUPUHLIZROVTGP-CALCHBBNSA-N	553138	N-[4-fluoro-5-(2- morpholin-4-ylpyrimidin- 5-yl)-2-[rac-(3R,5S)- 3,4,5-trimethylpiperazin- 1-yl]phenyl]-4- (trifluoromethyl)pyrimidine- 5-carboxamide::US11319299, Example 187	WD repeat-containing protein 5				 209						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553138	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553138&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			137376844	469797005							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166899	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1scnc1C(F)(F)F)-c1cnc(nc1)N1CCOCC1	InChI=1S/C26H29F4N7O2S/c1-15-12-37(13-16(2)35(15)3)21-9-19(27)18(17-10-31-25(32-11-17)36-4-6-39-7-5-36)8-20(21)34-24(38)22-23(26(28,29)30)33-14-40-22/h8-11,14-16H,4-7,12-13H2,1-3H3,(H,34,38)/t15-,16+	DLWWWOYTMSAGFU-IYBDPMFKSA-N	553139	N-[4-fluoro-5-(2- morpholin-4-ylpyrimidin- 5-yl)-2-[rac-(3R,5S)- 3,4,5-trimethylpiperazin- 1-yl]phenyl]-4- (trifluoromethyl)-1,3- thiazole-5-carboxamide::US11319299, Example 188	WD repeat-containing protein 5				 93.2						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553139	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553139&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138541660	469797006							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166900	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1cc(ccc1F)C(F)(F)F)-c1cnc(nc1)N1CCOCC1	InChI=1S/C29H31F5N6O2/c1-17-15-40(16-18(2)38(17)3)26-12-24(31)21(19-13-35-28(36-14-19)39-6-8-42-9-7-39)11-25(26)37-27(41)22-10-20(29(32,33)34)4-5-23(22)30/h4-5,10-14,17-18H,6-9,15-16H2,1-3H3,(H,37,41)/t17-,18+	MPHUDQGSNSEQPS-HDICACEKSA-N	553140	2-fluoro-N-[4-fluoro-5- (2-morpholin-4- ylpyrimidin-5-yl)-2-[rac- (3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-5- (trifluoromethyl)benzamide::US11319299, Example 189	WD repeat-containing protein 5				 442						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553140	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553140&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			137377146	469797007							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166901	COc1cc(F)cc(c1)C(=O)Nc1cc(c(F)cc1N1C[C@H](C)N(C)[C@H](C)C1)-c1cnc(nc1)N1CCOCC1	InChI=1S/C29H34F2N6O3/c1-18-16-37(17-19(2)35(18)3)27-13-25(31)24(21-14-32-29(33-15-21)36-5-7-40-8-6-36)12-26(27)34-28(38)20-9-22(30)11-23(10-20)39-4/h9-15,18-19H,5-8,16-17H2,1-4H3,(H,34,38)/t18-,19+	PKDFFVKJSBENPK-KDURUIRLSA-N	553141	3-fluoro-N-[4-fluoro-5- (2-morpholin-4- ylpyrimidin-5-yl)-2-[rac- (3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-5- methoxybenzamide::US11319299, Example 190	WD repeat-containing protein 5				 14.7						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553141	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553141&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			137377003	469797008							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166902	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1cc(Cl)cc(Cl)c1)-c1ccc(cc1)N1CCOCC1	InChI=1S/C30H33Cl2FN4O2/c1-19-17-37(18-20(2)35(19)3)29-16-27(33)26(21-4-6-25(7-5-21)36-8-10-39-11-9-36)15-28(29)34-30(38)22-12-23(31)14-24(32)13-22/h4-7,12-16,19-20H,8-11,17-18H2,1-3H3,(H,34,38)/t19-,20+	DDEZEMUMMOZZLK-BGYRXZFFSA-N	553142	3,5-dichloro-N-[4-fluoro- 5-(4-morpholin-4- ylphenyl)-2-[rac-(3R,5S)- 3,4,5-trimethylpiperazin- 1-yl]phenyl]benzamide::US11319299, Example 191	WD repeat-containing protein 5				 21.5						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553142	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553142&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			137376703	469797009							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166903	C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1ccn(C)n1)-c1cnc(nc1)N1CCOCC1	InChI=1S/C25H31FN8O2/c1-17-16-34(7-6-31(17)2)23-13-20(26)19(12-22(23)29-24(35)21-4-5-32(3)30-21)18-14-27-25(28-15-18)33-8-10-36-11-9-33/h4-5,12-15,17H,6-11,16H2,1-3H3,(H,29,35)/t17-/m0/s1	IUCXFCQIQFULIN-KRWDZBQOSA-N	553143	N-[4-fluoro-5-(2- morpholin-4-ylpyrimidin- 5-yl)-2-[rac-(3R)-3,4- dimethylpiperazin-1- yl]phenyl]-1-methylpyrazole-3- carboxamide::US11319299, Example 192	WD repeat-containing protein 5				 1260						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553143	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553143&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138551491	469797010							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166904	C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1cc[nH]n1)-c1cnc(nc1)N1CCOCC1			553144	N-[4-fluoro-5-(2- morpholin-4-ylpyrimidin- 5-yl)-2-[rac-(3R)-3,4- dimethylpiperazin-1- yl]phenyl]-1H-pyrazole- 3-carboxamide::US11319299, Example 193	WD repeat-containing protein 5				 592						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553144	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553144&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138551329	469797011							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166905	C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1csc(C)n1)-c1cnc(nc1)N1CCOCC1	InChI=1S/C25H30FN7O2S/c1-16-14-33(5-4-31(16)3)23-11-20(26)19(10-21(23)30-24(34)22-15-36-17(2)29-22)18-12-27-25(28-13-18)32-6-8-35-9-7-32/h10-13,15-16H,4-9,14H2,1-3H3,(H,30,34)/t16-/m0/s1	YXOSTINZUJCQDD-INIZCTEOSA-N	553145	N-[4-fluoro-5-(2- morpholin-4-ylpyrimidin- 5-yl)-2-[rac-(3R)-3,4- dimethylpiperazin-1- yl]phenyl]-2-methyl-1,3- thiazole-4-carboxamide::US11319299, Example 194	WD repeat-containing protein 5				 113						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553145	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553145&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138551545	469797012							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166906	C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1cnc(C)s1)-c1cnc(nc1)N1CCOCC1	InChI=1S/C25H30FN7O2S/c1-16-15-33(5-4-31(16)3)22-11-20(26)19(10-21(22)30-24(34)23-14-27-17(2)36-23)18-12-28-25(29-13-18)32-6-8-35-9-7-32/h10-14,16H,4-9,15H2,1-3H3,(H,30,34)/t16-/m0/s1	MSXCRBSSIOOQJA-INIZCTEOSA-N	553146	N-[4-fluoro-5-(2- morpholin-4-ylpyrimidin- 5-yl)-2-[rac-(3R)-3,4- dimethylpiperazin-1- yl]phenyl]-2-methyl-1,3- thiazole-5-carboxamide::US11319299, Example 195	WD repeat-containing protein 5				 106						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553146	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553146&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138551326	469797013							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166907	C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(NC(C)=O)nc1			553147	N-[5-(6- acetamidopyridin-3-yl)-4- fluoro-2-[rac-(3R)-3,4- dimethylpiperazin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 196	WD repeat-containing protein 5				 0.240						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553147	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553147&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607936	469797014							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166908	C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cnc(nc1)C#N			553148	N-[5-(2-cyanopyrimidin- 5-yl)-4-fluoro-2-[rac- (3R)-3,4-dimethylpiperazin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 197	WD repeat-containing protein 5				 0.681						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553148	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553148&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607937	469797015							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166909	C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(OCC2CC2)nc1			553149	N-[5-[6- (cyclopropylmethoxy) pyridin-3-yl]-4-fluoro-2-[rac- (3R)-3,4-dimethylpiperazin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 198	WD repeat-containing protein 5				 0.666						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553149	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553149&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607938	469797016							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166910	C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1sc(C)nc1C(F)(F)F)-c1cnc(nc1)N1CCOCC1	InChI=1S/C26H29F4N7O2S/c1-15-14-37(5-4-35(15)3)21-11-19(27)18(17-12-31-25(32-13-17)36-6-8-39-9-7-36)10-20(21)34-24(38)22-23(26(28,29)30)33-16(2)40-22/h10-13,15H,4-9,14H2,1-3H3,(H,34,38)/t15-/m0/s1	JIQDKYPMGHRZCX-HNNXBMFYSA-N	553150	N-[4-fluoro-5-(2- morpholin-4-ylpyrimidin- 5-yl)-2-[rac-(3R)-3,4- dimethylpiperazin-1- yl]phenyl]-2-methyl-4- (trifluoromethyl)-1,3- thiazole-5-carboxamide::US11319299, Example 199	WD repeat-containing protein 5				 23.4						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553150	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553150&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138551434	469797017							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166911	C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1cc(Cl)cc(Cl)c1)-c1cnc(nc1)N1CCOCC1	InChI=1S/C27H29Cl2FN6O2/c1-17-16-36(4-3-34(17)2)25-13-23(30)22(19-14-31-27(32-15-19)35-5-7-38-8-6-35)12-24(25)33-26(37)18-9-20(28)11-21(29)10-18/h9-15,17H,3-8,16H2,1-2H3,(H,33,37)/t17-/m0/s1	JMGCJYGZCRFPOY-KRWDZBQOSA-N	553151	3,5-dichloro-N-[4-fluoro- 5-(2-morpholin-4- ylpyrimidin-5-yl)-2-[rac- (3R)-3,4-dimethylpiperazin-1- yl]phenyl]benzamide::US11319299, Example 200	WD repeat-containing protein 5				 9.70						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553151	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553151&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138551484	469797018							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166912	C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(N2CCOCC2)c(F)c1			553152	N-[4-fluoro-5-(3-fluoro- 4-morpholin-4-ylphenyl)- 2-[rac-(3R)-3,4- dimethylpiperazin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 201	WD repeat-containing protein 5				 0.466						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553152	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553152&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607939	469797019							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166913	C[C@H]1CN(C[C@@H](C)O1)c1ncc(cn1)-c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)(F)F)c(cc1F)N1CCN(C)[C@@H](C)C1			553153	N-[4-fluoro-5-[2-[rac- (2R,6S)-2,6- dimethylmorpholin-4- yl]pyrimidin-5-yl]-2-[rac- (3R)-3,4-dimethylpiperazin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 202	WD repeat-containing protein 5				 0.434						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553153	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553153&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607940	469797020							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166914	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1ccc(F)cc1C(F)(F)F)-c1cnc(nc1)N1CCCN(C)CC1	InChI=1S/C31H36F5N7O/c1-19-17-43(18-20(2)41(19)4)28-14-26(33)24(21-15-37-30(38-16-21)42-9-5-8-40(3)10-11-42)13-27(28)39-29(44)23-7-6-22(32)12-25(23)31(34,35)36/h6-7,12-16,19-20H,5,8-11,17-18H2,1-4H3,(H,39,44)/t19-,20+	ASUJCSXQIRXZER-BGYRXZFFSA-N	553154	4-fluoro-N-[4-fluoro-5-[2- (4-methyl-1,4-diazepan-1- yl)pyrimidin-5-yl]-2-[rac- (3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-2- (trifluoromethyl)benzamide::US11319299, Example 203	WD repeat-containing protein 5				 1.66						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553154	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553154&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138541646	469797021							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166915	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1cn(C)c(=O)cc1C(F)(F)F)-c1ccc(cc1)N1CCOCC1	InChI=1S/C31H35F4N5O3/c1-19-16-40(17-20(2)38(19)4)28-15-26(32)23(21-5-7-22(8-6-21)39-9-11-43-12-10-39)13-27(28)36-30(42)24-18-37(3)29(41)14-25(24)31(33,34)35/h5-8,13-15,18-20H,9-12,16-17H2,1-4H3,(H,36,42)/t19-,20+	RGGQHPLPVBDOKN-BGYRXZFFSA-N	553155	N-[4-fluoro-5-(4- morpholin-4-ylphenyl)-2- [rac-(3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-1-methyl-6- oxo-4-(trifluoromethyl)pyridine- 3-carboxamide::US11319299, Example 204	WD repeat-containing protein 5				 13.8						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553155	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553155&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138541697	469797022							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166916	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cncc(c1)C#N			553156	N-[5-(5-cyanopyridin-3- yl)-4-fluoro-2-[rac- (3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 205	WD repeat-containing protein 5				 8.15						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553156	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553156&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607941	469797023							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166917	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cncc(Cl)c1			553157	N-[5-(5-chloropyridin-3- yl)-4-fluoro-2-[rac- (3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 206	WD repeat-containing protein 5				 3.85						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553157	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553157&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607942	469797024							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166918	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cccnc1OC1CCCCC1			553158	N-[5-(2- cyclohexyloxypyridin-3- yl)-4-fluoro-2-[rac- (3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 207	WD repeat-containing protein 5				 6.69						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553158	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553158&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607943	469797025							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166919	COc1ccc(CC(=O)N2CCC(=CC2)c2cc(NC(=O)c3c[nH]c(=O)cc3C(F)(F)F)c(cc2F)N2C[C@H](C)N(C)[C@H](C)C2)cc1			553159	N-[4-fluoro-5-[1-[2-(4- methoxyphenyl)acetyl]- 3,6-dihydro-2H-pyridin- 4-yl]-2-[rac-(3R,5S)- 3,4,5-trimethylpiperazin- 1-yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 208	WD repeat-containing protein 5				 0.570						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553159	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553159&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607944	469797026							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166920	COCCOc1ccc(cn1)-c1cc(NC(=O)c2cn(C)c(=O)cc2C(F)(F)F)c(cc1F)N1C[C@H](C)N(C)[C@H](C)C1	InChI=1S/C29H33F4N5O4/c1-17-14-38(15-18(2)37(17)4)25-12-23(30)20(19-6-7-26(34-13-19)42-9-8-41-5)10-24(25)35-28(40)21-16-36(3)27(39)11-22(21)29(31,32)33/h6-7,10-13,16-18H,8-9,14-15H2,1-5H3,(H,35,40)/t17-,18+	QZBGZIATYPDSKW-HDICACEKSA-N	553160	N-[4-fluoro-5-[6-(2- methoxyethoxy)pyridin- 3-yl]-2-[rac-(3R,5S)- 3,4,5-trimethylpiperazin- 1-yl]phenyl]-1-methyl-6- oxo-4-(trifluoromethyl)pyridine- 3-carboxamide::US11319299, Example 209	WD repeat-containing protein 5				 9.53						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553160	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553160&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			137376753	469797027							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166921	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1cn(C)c(=O)cc1C(F)(F)F)-c1cnc(nc1)N1CCCC1	InChI=1S/C29H33F4N7O2/c1-17-14-40(15-18(2)38(17)4)25-11-23(30)20(19-12-34-28(35-13-19)39-7-5-6-8-39)9-24(25)36-27(42)21-16-37(3)26(41)10-22(21)29(31,32)33/h9-13,16-18H,5-8,14-15H2,1-4H3,(H,36,42)/t17-,18+	ILEXXYIMBZHJIB-HDICACEKSA-N	553161	N-[4-fluoro-5-(2- pyrrolidin-1-ylpyrimidin- 5-yl)-2-[rac-(3R,5S)- 3,4,5-trimethylpiperazin- 1-yl]phenyl]-1-methyl-6- oxo-4-(trifluoromethyl)pyridine- 3-carboxamide::US11319299, Example 210	WD repeat-containing protein 5				 3.86						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553161	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553161&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138542386	469797028							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166922	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1sccc1C(F)(F)F)-c1cnc(nc1)N1CCOCC1	InChI=1S/C27H30F4N6O2S/c1-16-14-37(15-17(2)35(16)3)23-11-21(28)19(18-12-32-26(33-13-18)36-5-7-39-8-6-36)10-22(23)34-25(38)24-20(4-9-40-24)27(29,30)31/h4,9-13,16-17H,5-8,14-15H2,1-3H3,(H,34,38)/t16-,17+	BTCHLURQMWRZGT-CALCHBBNSA-N	553162	N-[4-fluoro-5-(2- morpholin-4-ylpyrimidin- 5-yl)-2-[rac-(3R,5S)- 3,4,5-trimethylpiperazin- 1-yl]phenyl]-3- (trifluoromethyl)thiophene-2- carboxamide::US11319299, Example 211	WD repeat-containing protein 5				 120						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553162	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553162&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138541910	469797029							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166923	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1cc(Cl)c(F)c(Cl)c1)-c1cnc(nc1)N1CCOCC1	InChI=1S/C28H30Cl2F2N6O2/c1-16-14-38(15-17(2)36(16)3)25-11-23(31)20(19-12-33-28(34-13-19)37-4-6-40-7-5-37)10-24(25)35-27(39)18-8-21(29)26(32)22(30)9-18/h8-13,16-17H,4-7,14-15H2,1-3H3,(H,35,39)/t16-,17+	LNCJRCRMVZXUPY-CALCHBBNSA-N	553163	3,5-dichloro-4-fluoro-N- [4-fluoro-5-(2-morpholin- 4-ylpyrimidin-5-yl)-2- [rac-(3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]benzamide::US11319299, Example 212	WD repeat-containing protein 5				 2.71						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553163	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553163&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			137377324	469797030							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166924	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1cccc(Cl)c1Cl)-c1cnc(nc1)N1CCOCC1	InChI=1S/C28H31Cl2FN6O2/c1-17-15-37(16-18(2)35(17)3)25-12-23(31)21(19-13-32-28(33-14-19)36-7-9-39-10-8-36)11-24(25)34-27(38)20-5-4-6-22(29)26(20)30/h4-6,11-14,17-18H,7-10,15-16H2,1-3H3,(H,34,38)/t17-,18+	RWAPXLQUONTCET-HDICACEKSA-N	553164	2,3-dichloro-N-[4-fluoro- 5-(2-morpholin-4- ylpyrimidin-5-yl)-2-[rac- (3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]benzamide::US11319299, Example 213	WD repeat-containing protein 5				 6.91						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553164	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553164&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			137377409	469797031							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166925	C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cccc(CN(C)C2COC2)c1			553165	N-[4-fluoro-5-[3- [[methyl(oxetan-3- yl)amino]methyl]phenyl]- 2-[rac-(3R)-3,4- dimethylpiperazin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 214	WD repeat-containing protein 5				 2.15						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553165	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553165&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607945	469797032							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166926	CCOc1cncc(c1)-c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)(F)F)c(cc1F)N1C[C@H](C)N(C)[C@H](C)C1			553166	N-[5-(5-ethoxypyridin-3- yl)-4-fluoro-2-[rac- (3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 215	WD repeat-containing protein 5				 5.76						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553166	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553166&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607946	469797033							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166927	C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1cn(C)c(=O)cc1C(F)F)-c1cnc(nc1)N1CCOCC1	InChI=1S/C28H32F3N7O3/c1-17-15-38(5-4-35(17)2)24-12-22(29)19(18-13-32-28(33-14-18)37-6-8-41-9-7-37)10-23(24)34-27(40)21-16-36(3)25(39)11-20(21)26(30)31/h10-14,16-17,26H,4-9,15H2,1-3H3,(H,34,40)/t17-/m0/s1	MAMCQIDNEWXMCJ-KRWDZBQOSA-N	553167	4-(difluoromethyl)-N-[4- fluoro-5-(2-morpholin-4- ylpyrimidin-5-yl)-2-[rac- (3R)-3,4-dimethylpiperazin-1- yl]phenyl]-1-methyl-6- oxopyridine-3-carboxamide::US11319299, Example 216	WD repeat-containing protein 5				 2.71						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553167	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553167&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138542416	469797034							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166928	C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1cn(C)c(=O)cc1C(F)F)-c1ccc(NC(C)=O)nc1	InChI=1S/C27H29F3N6O3/c1-15-13-36(8-7-34(15)3)23-11-21(28)18(17-5-6-24(31-12-17)32-16(2)37)9-22(23)33-27(39)20-14-35(4)25(38)10-19(20)26(29)30/h5-6,9-12,14-15,26H,7-8,13H2,1-4H3,(H,33,39)(H,31,32,37)/t15-/m0/s1	UOYZNLPMXQNDOB-HNNXBMFYSA-N	553168	N-[5-(6- acetamidopyridin-3-yl)-4- fluoro-2-[rac-(3R)-3,4- dimethylpiperazin-1- yl]phenyl]-4- (difluoromethyl)-1- methyl-6-oxopyridine-3- carboxamide::US11319299, Example 217	WD repeat-containing protein 5				 4.32						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553168	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553168&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138551533	469797035							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166929	C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1cn(C)c(=O)cc1C(F)F)-c1cnc(nc1)C#N	InChI=1S/C25H24F3N7O2/c1-14-12-35(5-4-33(14)2)21-8-19(26)16(15-10-30-22(9-29)31-11-15)6-20(21)32-25(37)18-13-34(3)23(36)7-17(18)24(27)28/h6-8,10-11,13-14,24H,4-5,12H2,1-3H3,(H,32,37)/t14-/m0/s1	DJHAAPZISXGUQE-AWEZNQCLSA-N	553169	N-[5-(2-cyanopyrimidin- 5-yl)-4-fluoro-2-[rac- (3R)-3,4-dimethylpiperazin-1- yl]phenyl]-4-(difluoromethyl)- 1-methyl-6-oxopyridine-3- carboxamide::US11319299, Example 218	WD repeat-containing protein 5				 3.18						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553169	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553169&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138551570	469797036							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166930	C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(nc1)N(C)C			553170	N-[5-[6-(dimethylamino) pyridin-3-yl]-4-fluoro-2-[rac- (3R)-3,4-dimethylpiperazin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 219	WD repeat-containing protein 5				 1.40						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553170	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553170&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607947	469797037							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166931	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cnc(N(C)C)c(c1)C#N			553171	N-[5-[5-cyano-6- (dimethylamino)pyridin- 3-yl]-4-fluoro-2-[rac- (3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 220	WD repeat-containing protein 5				 2.25						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553171	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553171&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607948	469797038							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166932	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cnc(N(C)C)c(F)c1			553172	N-[5-[6-(dimethylamino)- 5-fluoropyridin-3-yl]-4- fluoro-2-[rac-(3R,5S)- 3,4,5-trimethylpiperazin- 1-yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 221	WD repeat-containing protein 5				 0.769						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553172	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553172&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607949	469797039							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166933	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cnc(N2CCOCC2)c(Cl)c1			553173	N-[5-(5-chloro-6- morpholin-4-ylpyridin-3- yl)-4-fluoro-2-[rac- (3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 222	WD repeat-containing protein 5				 1.34						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553173	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553173&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607950	469797040							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166934	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cnc2OCCOc2c1			553174	N-[5-(2,3-dihydro- [1,4]dioxino[2,3-b] pyridin-7-yl)-4-fluoro- 2-[rac-(3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 223	WD repeat-containing protein 5				 1.63						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553174	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553174&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607951	469797041							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166935	CN1CCN(CC1(C)C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cnc(nc1)N1CCOCC1	InChI=1S/C28H31F4N7O3/c1-27(2)16-39(5-4-37(27)3)23-12-21(29)18(17-13-34-26(35-14-17)38-6-8-42-9-7-38)10-22(23)36-25(41)19-15-33-24(40)11-20(19)28(30,31)32/h10-15H,4-9,16H2,1-3H3,(H,33,40)(H,36,41)	NAQVVLMOXKGZLS-UHFFFAOYSA-N	553175	N-[4-fluoro-5-(2- morpholin-4-ylpyrimidin- 5-yl)-2-(3,3,4- trimethylpiperazin-1- yl)phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 225	WD repeat-containing protein 5				 3000						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553175	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553175&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607952	469797042							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166936	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1cn(C)c(=O)cc1C(F)(F)F)-c1ccnc(c1)N1CCOCC1	InChI=1S/C30H34F4N6O3/c1-18-15-40(16-19(2)38(18)4)26-14-24(31)21(20-5-6-35-27(11-20)39-7-9-43-10-8-39)12-25(26)36-29(42)22-17-37(3)28(41)13-23(22)30(32,33)34/h5-6,11-14,17-19H,7-10,15-16H2,1-4H3,(H,36,42)/t18-,19+	YFXIMBDAHSTROL-KDURUIRLSA-N	553176	N-[4-fluoro-5-(2- morpholin-4-ylpyridin-4- yl)-2-[rac-(3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-1-methyl-6- oxo-4-(trifluoromethyl)pyridine- 3-carboxamide::US11319299, Example 226	WD repeat-containing protein 5				 7.99						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553176	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553176&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138541773	469797043							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166937	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1cn(C)c(=O)cc1C(F)(F)F)-c1ccc(cc1)N1CCCC1	InChI=1S/C31H35F4N5O2/c1-19-16-40(17-20(2)38(19)4)28-15-26(32)23(21-7-9-22(10-8-21)39-11-5-6-12-39)13-27(28)36-30(42)24-18-37(3)29(41)14-25(24)31(33,34)35/h7-10,13-15,18-20H,5-6,11-12,16-17H2,1-4H3,(H,36,42)/t19-,20+	ZCDKHBWFAXURNQ-BGYRXZFFSA-N	553177	N-[4-fluoro-5-(4- pyrrolidin-1-ylphenyl)-2- [rac-(3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-1-methyl-6- oxo-4-(trifluoromethyl)pyridine- 3-carboxamide::US11319299, Example 227	WD repeat-containing protein 5				 9.14						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553177	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553177&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138541686	469797044							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166938	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1cn(C)c(=O)cc1C(F)(F)F)-c1ccc(OCC2CC2)cc1	InChI=1S/C31H34F4N4O3/c1-18-14-39(15-19(2)38(18)4)28-13-26(32)23(21-7-9-22(10-8-21)42-17-20-5-6-20)11-27(28)36-30(41)24-16-37(3)29(40)12-25(24)31(33,34)35/h7-13,16,18-20H,5-6,14-15,17H2,1-4H3,(H,36,41)/t18-,19+	XUPOVLZXYRJULS-KDURUIRLSA-N	553178	N-[5-[4- (cyclopropylmethoxy)phenyl]- 4-fluoro-2-[rac-(3R,5S)-3,4,5- trimethylpiperazin-1-yl] phenyl]-1-methyl-6-oxo-4- (trifluoromethyl)pyridine- 3-carboxamide::US11319299, Example 228	WD repeat-containing protein 5				 7.26						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553178	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553178&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			137376770	469797045							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166939	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1cccc(F)c1F)-c1cnc(nc1)N1CCOCC1	InChI=1S/C28H31F3N6O2/c1-17-15-37(16-18(2)35(17)3)25-12-23(30)21(19-13-32-28(33-14-19)36-7-9-39-10-8-36)11-24(25)34-27(38)20-5-4-6-22(29)26(20)31/h4-6,11-14,17-18H,7-10,15-16H2,1-3H3,(H,34,38)/t17-,18+	KXCUSVGDGUDLND-HDICACEKSA-N	553179	2,3-difluoro-N-[4-fluoro- 5-(2-morpholin-4- ylpyrimidin-5-yl)-2-[rac- (3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]benzamide::US11319299, Example 229	WD repeat-containing protein 5				 83.0						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553179	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553179&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138541612	469797046							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166940	C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1ccc(F)cc1Cl)-c1cnc(nc1)N1CCOCC1	InChI=1S/C27H29ClF2N6O2/c1-17-16-36(6-5-34(17)2)25-13-23(30)21(18-14-31-27(32-15-18)35-7-9-38-10-8-35)12-24(25)33-26(37)20-4-3-19(29)11-22(20)28/h3-4,11-15,17H,5-10,16H2,1-2H3,(H,33,37)/t17-/m0/s1	GIMWIECNKXXFDO-KRWDZBQOSA-N	553180	2-chloro-4-fluoro-N-[4- fluoro-5-(2-morpholin-4- ylpyrimidin-5-yl)-2-[rac- (3R)-3,4-dimethylpiperazin-1- yl]phenyl]benzamide::US11319299, Example 230	WD repeat-containing protein 5				 8.95						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553180	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553180&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138551553	469797047							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166941	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCN(CC1)C1CCCC1			553181	N-[5-(1-cyclopentyl-3,6- dihydro-2H-pyridin-4-yl)- 4-fluoro-2-[rac-(3R,5S)- 3,4,5-trimethylpiperazin- 1-yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 231	WD repeat-containing protein 5				 2.51						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553181	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553181&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607953	469797048							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166942	COc1ccc(cc1)C(C)N1CCC(=CC1)c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)(F)F)c(cc1F)N1C[C@H](C)N(C)[C@H](C)C1			553182	N-[4-fluoro-5-[1-[1-(4- methoxyphenyl)ethyl]- 3,6-dihydro-2H-pyridin- 4-yl]-2-[rac-(3R,5S)- 3,4,5-trimethylpiperazin- 1-yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 232	WD repeat-containing protein 5				 2.72						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553182	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553182&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607954	469797049							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166943	CCC(C)N1CCC(=CC1)c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)(F)F)c(cc1F)N1C[C@H](C)N(C)[C@H](C)C1			553183	N-[5-(1-butan-2-yl-3,6- dihydro-2H-pyridin-4-yl)- 4-fluoro-2-[rac-(3R,5S)- 3,4,5-trimethylpiperazin- 1-yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 233	WD repeat-containing protein 5				 3.89						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553183	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553183&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607955	469797050							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166944	CN(C)[C@@H]1CCN(C1)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(nc1)N1CCOCC1			553184	N-[4-fluoro-5-(6- morpholin-4-ylpyridin-3- yl)-2-[rac-(3R)-3- (dimethylamino)pyrrolidin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 234	WD repeat-containing protein 5				 1.86						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553184	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553184&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607956	469797051							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166945	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCN(CC1)C1COC1			553185	N-[4-fluoro-5-[1-(oxetan- 3-yl)-3,6-dihydro-2H- pyridin-4-yl]-2-[rac- (3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 235	WD repeat-containing protein 5				 0.943						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553185	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553185&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607957	469797052							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166946	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1CCNCC1			553186	N-[4-fluoro-5-piperidin- 4-yl-2-[rac-(3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 236	WD repeat-containing protein 5				 31.1						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553186	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553186&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607958	469797053							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166947	CN(C)[C@@H]1CCN(C1)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(O)nc1			553187	N-[4-fluoro-5-(6- hydroxypyridin-3-yl)-2- [rac-(3R)-3- (dimethylamino)pyrrolidin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 237	WD repeat-containing protein 5				 9.33						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553187	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553187&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607959	469797054							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166948	CN(C)[C@@H]1CCN(C1)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(OCC2CC2)nc1			553188	N-[5-[6-(cyclopropylmethoxy) pyridin-3-yl]-4-fluoro-2-[rac- (3R)-3-(dimethylamino) pyrrolidin-1-yl]phenyl]-6-oxo- 4-(trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 238	WD repeat-containing protein 5				 5.11						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553188	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553188&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607960	469797055							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166949	C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(nc1)N1CCOCC1			553189	N-[4-fluoro-5-(6- morpholin-4-ylpyridin-3- yl)-2-[rac-(3R)-3,4- dimethylpiperazin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 239	WD repeat-containing protein 5				 1.07						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553189	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553189&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607961	469797056							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166950	CC(C)Oc1ncc(cn1)-c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)(F)F)c(cc1F)N1CCN(C)[C@@H](C)C1			553190	N-[4-fluoro-5-(2-propan- 2-yloxypyrimidin-5-yl)-2- [rac-(3R)-3,4-dimethylpiperazin- 1-yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 240	WD repeat-containing protein 5				 2.23						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553190	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553190&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607962	469797057							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166951	C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cnc2OCCOc2c1			553191	N-[5-(2,3-dihydro- [1,4]dioxino[2,3-b]pyridin-7- yl)-4-fluoro-2-[rac-(3R)-3,4- dimethylpiperazin-1-yl]phenyl]-6- oxo-4-(trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 241	WD repeat-containing protein 5				 2.82						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553191	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553191&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607963	469797058							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166952	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCN(CC1)C1CCN(C)CC1			553192	N-[4-fluoro-5-[1-(1- methylpiperidin-4-yl)- 3,6-dihydro-2H-pyridin- 4-yl]-2-[rac-(3R,5S)- 3,4,5-trimethylpiperazin- 1-yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 242	WD repeat-containing protein 5				 3.49						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553192	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553192&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607964	469797059							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166953	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCN(CC1)C(=O)C(C)(C)C			553193	N-[5-[1-(2,2- dimethylpropanoyl)-3,6- dihydro-2H-pyridin-4-yl]- 4-fluoro-2-[rac-(3R,5S)- 3,4,5-trimethylpiperazin- 1-yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 243	WD repeat-containing protein 5				 2.16						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553193	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553193&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607965	469797060							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166954	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1CCN(CC1)C(=O)C(C)(C)C			553194	N-[5-[1-(2,2- dimethylpropanoyl)piperidin- 4-yl]-4-fluoro-2-[rac-(3R,5S)- 3,4,5-trimethylpiperazin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 244	WD repeat-containing protein 5				 1.97						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553194	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553194&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607966	469797061							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166955	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCN(CC1)c1ncccn1			553195	N-[4-fluoro-5-(1- pyrimidin-2-yl-3,6- dihydro-2H-pyridin-4-yl)- 2-[rac-(3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 245	WD repeat-containing protein 5				 1.39						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553195	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553195&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607967	469797062							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166956	C[C@H]1CN(C[C@@H](C)O1)c1ncc(cn1)-c1cc(NC(=O)c2cn(C)c(=O)cc2C(F)(F)F)c(cc1F)N1C[C@H](C)N(C)[C@H](C)C1	InChI=1S/C31H37F4N7O3/c1-17-12-41(13-18(2)40(17)6)27-9-25(32)22(21-10-36-30(37-11-21)42-14-19(3)45-20(4)15-42)7-26(27)38-29(44)23-16-39(5)28(43)8-24(23)31(33,34)35/h7-11,16-20H,12-15H2,1-6H3,(H,38,44)/t17-,18+,19-,20+	XVAVYLGVIGIDHZ-FGYAAKKASA-N	553196	N-[4-fluoro-5-[2-[rac- (2R,6S)-2,6- dimethylmorpholin- 4-yl]pyrimidin-5-yl]-2- [rac-(3S,5R)-3,4,5- trimethylpiperazin-1- yl]phenyl]-1-methyl-6- oxo-4-(trifluoromethyl) pyridine-3-carboxamide::US11319299, Example 246	WD repeat-containing protein 5				 2.51						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553196	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553196&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138541749	469797063							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166957	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1cn(C)c(=O)cc1C(F)(F)F)-c1ccc(N2CCOCC2)c(F)c1	InChI=1S/C31H34F5N5O3/c1-18-15-41(16-19(2)39(18)4)28-14-24(32)21(20-5-6-27(25(33)11-20)40-7-9-44-10-8-40)12-26(28)37-30(43)22-17-38(3)29(42)13-23(22)31(34,35)36/h5-6,11-14,17-19H,7-10,15-16H2,1-4H3,(H,37,43)/t18-,19+	VQYRENMNLMEHOT-KDURUIRLSA-N	553197	N-[4-fluoro-5-(3-fluoro- 4-morpholin-4-ylphenyl)- 2-[rac-(3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-1-methyl-6- oxo-4-(trifluoromethyl) pyridine-3-carboxamide::US11319299, Example 247	WD repeat-containing protein 5				 5.16						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553197	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553197&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			137377839	469797064							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166958	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1ccc(F)cc1C(F)(F)F)-c1cnc(nc1)N1CCOCC1	InChI=1S/C29H31F5N6O2/c1-17-15-40(16-18(2)38(17)3)26-12-24(31)22(19-13-35-28(36-14-19)39-6-8-42-9-7-39)11-25(26)37-27(41)21-5-4-20(30)10-23(21)29(32,33)34/h4-5,10-14,17-18H,6-9,15-16H2,1-3H3,(H,37,41)/t17-,18+	OVAUTHLIMOXPHS-HDICACEKSA-N	553198	4-fluoro-N-[4-fluoro-5-(2- morpholin-4-ylpyrimidin- 5-yl)-2-[rac-(3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-2-(trifluoromethyl) benzamide::US11319299, Example 248	WD repeat-containing protein 5				 1.33						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553198	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553198&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			137376865	469797065							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166959	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCN(C1)S(C)(=O)=O			553199	N-[4-fluoro-5-(1- methylsulfonyl-2,5- dihydropyrrol-3-yl)-2- [rac-(3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 249	WD repeat-containing protein 5				 0.665						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553199	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553199&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607968	469797066							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166960	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1cc(Cl)cc(Cl)c1)-c1ccc(OCC2CC2)nc1	InChI=1S/C29H31Cl2FN4O2/c1-17-14-36(15-18(2)35(17)3)27-12-25(32)24(20-6-7-28(33-13-20)38-16-19-4-5-19)11-26(27)34-29(37)21-8-22(30)10-23(31)9-21/h6-13,17-19H,4-5,14-16H2,1-3H3,(H,34,37)/t17-,18+	QMZXXQAFWAEJII-HDICACEKSA-N	553200	3,5-dichloro-N-[5-[6- (cyclopropylmethoxy) pyridin-3-yl]-4-fluoro-2- [rac-(3R,5S)-3,4,5- trimethylpiperazin-1-yl] phenyl]benzamide::US11319299, Example 250	WD repeat-containing protein 5				 76.9						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553200	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553200&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			137376882	469797067							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166961	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1ccc(F)cc1Cl)-c1ccc(OCC2CC2)nc1	InChI=1S/C29H31ClF2N4O2/c1-17-14-36(15-18(2)35(17)3)27-12-25(32)23(20-6-9-28(33-13-20)38-16-19-4-5-19)11-26(27)34-29(37)22-8-7-21(31)10-24(22)30/h6-13,17-19H,4-5,14-16H2,1-3H3,(H,34,37)/t17-,18+	MIMHFISDRAEPDG-HDICACEKSA-N	553201	2-chloro-N-[5-[6- (cyclopropylmethoxy) pyridin-3-yl]-4-fluoro-2- [rac-(3R,5S)-3,4,5- trimethylpiperazin-1-yl] phenyl]-4-fluorobenzamide::US11319299, Example 251	WD repeat-containing protein 5				 15.6						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553201	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553201&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			137376846	469797068							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166962	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCN(CC1)C(C)=O			553202	N-[5-(1-acetyl-3,6-dihydro- 2H-pyridin-4-yl)-4-fluoro- 2-[rac-(3R,5S)-3,4,5- trimethylpiperazin- 1-yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 252	WD repeat-containing protein 5				 2.79						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553202	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553202&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607969	469797069							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166963	CCOC(=O)N1CCC(=CC1)c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)(F)F)c(cc1F)N1C[C@H](C)N(C)[C@H](C)C1			553203	US11319299, Example 253::ethyl 4-[2-fluoro-5-[[6- oxo-4-(trifluoromethyl)- 1H-pyridine-3-carbonyl] amino]-4-[rac-(3R,5S)- 3,4,5-trimethylpiperazin-1- yl]phenyl]-3,6-dihydro-2H- pyridine-1-carboxylate	WD repeat-containing protein 5				 3.30						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553203	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553203&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607970	469797070							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166964	CC(C)COC(=O)N1CCC(=CC1)c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)(F)F)c(cc1F)N1C[C@H](C)N(C)[C@H](C)C1			553204	2-methylpropyl 4-[2-fluoro- 5-[[6-oxo-4-(trifluoromethyl)- 1H-pyridine-3-carbonyl] amino]-4-[rac-(3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-3,6-dihydro-2H- pyridine-1-carboxylate::US11319299, Example 254	WD repeat-containing protein 5				 3.34						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553204	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553204&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607971	469797071							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166965	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCN(CC1)C(=O)CC(C)(C)C			553205	N-[5-[1-(3,3- dimethylbutanoyl)-3,6- dihydro-2H-pyridin-4-yl]- 4-fluoro-2-[rac-(3R,5S)- 3,4,5-trimethylpiperazin- 1-yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 255	WD repeat-containing protein 5				 1.98						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553205	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553205&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607972	469797072							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166966	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1CCN(CC1)C(=O)CC(C)(C)C			553206	N-[5-[1-(3,3- dimethylbutanoyl) piperidin-4-yl]-4-fluoro- 2-[rac-(3R,5S)-3,4,5- trimethylpiperazin- 1-yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 256	WD repeat-containing protein 5				 11.8						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553206	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553206&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607973	469797073							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166967	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(F)nc1			553207	N-[4-fluoro-5-(6- fluoropyridin-3-yl)-2- [rac-(3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 257	WD repeat-containing protein 5				 1.70						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553207	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553207&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607974	469797074							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166968	CN(C)C1CCN(CC1)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cnc(nc1)N1CCOCC1	InChI=1S/C28H31F4N7O3/c1-37(2)18-3-5-38(6-4-18)24-13-22(29)19(17-14-34-27(35-15-17)39-7-9-42-10-8-39)11-23(24)36-26(41)20-16-33-25(40)12-21(20)28(30,31)32/h11-16,18H,3-10H2,1-2H3,(H,33,40)(H,36,41)	GGBCIXPYULSFCI-UHFFFAOYSA-N	553208	N-[2-[4-(dimethylamino) piperidin-1-yl]-4-fluoro-5-(2- morpholin-4-ylpyrimidin- 5-yl)phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 258	WD repeat-containing protein 5				 66.1						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553208	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553208&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607975	469797075							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166969	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(nc1)N1CCCC1			553209	N-[4-fluoro-5-(6- pyrrolidin-1-ylpyridin-3- yl)-2-[rac-(3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 261	WD repeat-containing protein 5				 1.64						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553209	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553209&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607976	469797076							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166970	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1ccc(F)c(Cl)c1)-c1cnc(nc1)N1CCOCC1	InChI=1S/C28H31ClF2N6O2/c1-17-15-37(16-18(2)35(17)3)26-12-24(31)21(20-13-32-28(33-14-20)36-6-8-39-9-7-36)11-25(26)34-27(38)19-4-5-23(30)22(29)10-19/h4-5,10-14,17-18H,6-9,15-16H2,1-3H3,(H,34,38)/t17-,18+	NBSSZEPXMIZXLI-HDICACEKSA-N	553210	3-chloro-4-fluoro-N-[4- fluoro-5-(2-morpholin-4- ylpyrimidin-5-yl)-2-[rac- (3R,5S)-3,4,5- trimethylpiperazin-1-yl] phenyl]benzamide::US11319299, Example 264	WD repeat-containing protein 5				 2.94						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553210	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553210&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138541695	469797077							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166971	COc1cc(Cl)cc(c1)C(=O)Nc1cc(c(F)cc1N1C[C@H](C)N(C)[C@H](C)C1)-c1cnc(nc1)N1CCOCC1	InChI=1S/C29H34ClFN6O3/c1-18-16-37(17-19(2)35(18)3)27-13-25(31)24(21-14-32-29(33-15-21)36-5-7-40-8-6-36)12-26(27)34-28(38)20-9-22(30)11-23(10-20)39-4/h9-15,18-19H,5-8,16-17H2,1-4H3,(H,34,38)/t18-,19+	PUAAPKUZSJEOAK-KDURUIRLSA-N	553211	3-chloro-N-[4-fluoro-5- (2-morpholin-4-ylpyrimidin- 5-yl)-2-[rac-(3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-5- methoxybenzamide::US11319299, Example 265	WD repeat-containing protein 5				 28.3						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553211	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553211&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			137376793	469797078							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166972	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1ccc(F)c(Cl)c1F)-c1cnc(nc1)N1CCOCC1	InChI=1S/C28H30ClF3N6O2/c1-16-14-38(15-17(2)36(16)3)24-11-22(31)20(18-12-33-28(34-13-18)37-6-8-40-9-7-37)10-23(24)35-27(39)19-4-5-21(30)25(29)26(19)32/h4-5,10-13,16-17H,6-9,14-15H2,1-3H3,(H,35,39)/t16-,17+	DKZXWCHZCVJVON-CALCHBBNSA-N	553212	3-chloro-2,4-difluoro-N- [4-fluoro-5-(2-morpholin- 4-ylpyrimidin-5-yl)-2- [rac-(3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]benzamide::US11319299, Example 266	WD repeat-containing protein 5				 13.7						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553212	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553212&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			137377249	469797079							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166973	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCN(C)CC1			553213	N-[4-fluoro-5-(1-methyl- 3,6-dihydro-2H-pyridin- 4-yl)-2-[rac-(3R,5S)- 3,4,5-trimethylpiperazin- 1-yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 267	WD repeat-containing protein 5				 10.7						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553213	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553213&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607977	469797080							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166974	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cnc(cc1C)C#N			553214	N-[5-(6-cyano-4- methylpyridin-3-yl)-4- fluoro-2-[rac-(3R,5S)- 3,4,5-trimethylpiperazin- 1-yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 269	WD repeat-containing protein 5				 8.74						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553214	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553214&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607978	469797081							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166975	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCN(CC1)c1ccccn1			553215	N-[4-fluoro-5-(1-pyridin- 2-yl-3,6-dihydro-2H-pyridin- 4-yl)-2-[rac-(3R,5S)-3,4,5- trimethylpiperazin-1-yl] phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 270	WD repeat-containing protein 5				 0.938						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553215	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553215&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607979	469797082							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166976	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCN(CC1)c1ncc(C)cn1			553216	N-[4-fluoro-5-[1-(5- methylpyrimidin-2-yl)- 3,6-dihydro-2H-pyridin- 4-yl]-2-[rac-(3R,5S)- 3,4,5-trimethylpiperazin- 1-yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 271	WD repeat-containing protein 5				 0.499						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553216	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553216&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607980	469797083							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166977	C[C@H]1CN(C[C@@H](C)O1)c1ccc(cn1)-c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)(F)F)c(cc1F)N1C[C@H](C)N(C)[C@H](C)C1			553217	N-[4-fluoro-5-[6-[rac- (2R,6S)-2,6- dimethylmorpholin-4- yl]pyridin-3-yl]-2-[rac- (3S,5R)-3,4,5- trimethylpiperazin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 272	WD repeat-containing protein 5				 0.532						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553217	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553217&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607981	469797084							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166978	C[C@H]1CN(C[C@@H](C)O1)c1ncc(cn1)-c1cc(NC(=O)c2cn(C)c(=O)cc2C(F)(F)F)c(cc1F)N1CCN(C)[C@@H](C)C1	InChI=1S/C30H35F4N7O3/c1-17-13-40(7-6-38(17)4)26-10-24(31)21(20-11-35-29(36-12-20)41-14-18(2)44-19(3)15-41)8-25(26)37-28(43)22-16-39(5)27(42)9-23(22)30(32,33)34/h8-12,16-19H,6-7,13-15H2,1-5H3,(H,37,43)/t17-,18-,19+/m0/s1	VRJIKZBYTFROSJ-GBESFXJTSA-N	553218	N-[4-fluoro-5-[2-[rac- (2R,6S)-2,6- dimethylmorpholin- 4-yl]pyrimidin-5-yl]-2-[rac- (3R)-3,4-dimethylpiperazin- 1-yl]phenyl]-1-methyl-6- oxo-4-(trifluoromethyl) pyridine-3-carboxamide::US11319299, Example 273	WD repeat-containing protein 5				 2.11						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553218	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553218&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138551333	469797085							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166979	COc1cc(ncn1)N1CCC(=CC1)c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)(F)F)c(cc1F)N1C[C@H](C)N(C)[C@H](C)C1			553219	N-[4-fluoro-5-[1-(6- methoxypyrimidin-4-yl)- 3,6-dihydro-2H-pyridin- 4-yl]-2-[rac-(3R,5S)- 3,4,5-trimethylpiperazin- 1-yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 274	WD repeat-containing protein 5				 1.29						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553219	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553219&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607982	469797086							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166980	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCN(CC1)c1ncc(Cl)cn1			553220	N-[5-[1-(5-chloropyrimidin- 2-yl)-3,6-dihydro-2H- pyridin-4-yl]-4-fluoro-2- [rac-(3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 275	WD repeat-containing protein 5				 1.54						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553220	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553220&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607983	469797087							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166981	CCOC(=O)c1ccnc(n1)N1CCC(=CC1)c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)(F)F)c(cc1F)N1C[C@H](C)N(C)[C@H](C)C1			553221	US11319299, Example 276::ethyl 2-[4-[2-fluoro-5- [[6-oxo-4-(trifluoromethyl)- 1H-pyridine-3-carbonyl] amino]-4-[rac-(3R,5S)- 3,4,5-trimethylpiperazin-1- yl]phenyl]-3,6-dihydro-2H- pyridin-1-yl]pyrimidine-4- carboxylate	WD repeat-containing protein 5				 1.67						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553221	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553221&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607984	469797088							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166982	CNC1CCN(C1)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cnc(nc1)N1CCOCC1			553222	N-[4-fluoro-2-[3- (methylamino)pyrrolidin- 1-yl]-5-(2-morpholin-4- ylpyrimidin-5-yl)phenyl]- 6-oxo-4-(trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 277	WD repeat-containing protein 5				 14.9						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553222	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553222&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607985	469797089							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166983	C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1cn(C)c(=O)cc1C(F)(F)F)-c1cnc(nc1)N1CCN(C)CC1	InChI=1S/C29H34F4N8O2/c1-18-16-41(10-7-38(18)3)25-13-23(30)20(19-14-34-28(35-15-19)40-8-5-37(2)6-9-40)11-24(25)36-27(43)21-17-39(4)26(42)12-22(21)29(31,32)33/h11-15,17-18H,5-10,16H2,1-4H3,(H,36,43)/t18-/m0/s1	DQTHXSJKHKMLNF-SFHVURJKSA-N	553223	N-[4-fluoro-5-[2-(4- methylpiperazin-1-yl) pyrimidin-5-yl]-2-[rac- (3R)-3,4-dimethylpiperazin-1- yl]phenyl]-1-methyl-6-oxo-4- (trifluoromethyl)pyridine- 3-carboxamide::US11319299, Example 279	WD repeat-containing protein 5				 2.08						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553223	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553223&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138551544	469797090							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166984	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1cc(O)cc(c1)C(F)(F)F)-c1cnc(nc1)N1CCOCC1	InChI=1S/C29H32F4N6O3/c1-17-15-39(16-18(2)37(17)3)26-12-24(30)23(20-13-34-28(35-14-20)38-4-6-42-7-5-38)11-25(26)36-27(41)19-8-21(29(31,32)33)10-22(40)9-19/h8-14,17-18,40H,4-7,15-16H2,1-3H3,(H,36,41)/t17-,18+	XPEVVCQFBFUDTA-HDICACEKSA-N	553224	N-[4-fluoro-5-(2- morpholin-4-ylpyrimidin- 5-yl)-2-[rac-(3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-3-hydroxy-5- (trifluoromethyl)benzamide::US11319299, Example 280	WD repeat-containing protein 5				 3.12						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553224	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553224&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			137377204	469797091							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166985	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1cccc(O)c1)-c1cnc(nc1)N1CCOCC1	InChI=1S/C28H33FN6O3/c1-18-16-35(17-19(2)33(18)3)26-13-24(29)23(12-25(26)32-27(37)20-5-4-6-22(36)11-20)21-14-30-28(31-15-21)34-7-9-38-10-8-34/h4-6,11-15,18-19,36H,7-10,16-17H2,1-3H3,(H,32,37)/t18-,19+	BBSKAFJIOXPDNK-KDURUIRLSA-N	553225	N-[4-fluoro-5-(2- morpholin-4-ylpyrimidin- 5-yl)-2-[rac-(3R,5S)-3,4,5- trimethylpiperazin-1-yl]phenyl]- 3-hydroxybenzamide::US11319299, Example 281	WD repeat-containing protein 5				 29.1						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553225	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553225&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			137376890	469797092							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166986	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c(O)cnc2ccccc12)-c1cnc(nc1)N1CCOCC1	InChI=1S/C31H34FN7O3/c1-19-17-39(18-20(2)37(19)3)27-13-24(32)23(21-14-34-31(35-15-21)38-8-10-42-11-9-38)12-26(27)36-30(41)29-22-6-4-5-7-25(22)33-16-28(29)40/h4-7,12-16,19-20,40H,8-11,17-18H2,1-3H3,(H,36,41)/t19-,20+	PIEUITOJHWUOLV-BGYRXZFFSA-N	553226	N-[4-fluoro-5-(2-morpholin- 4-ylpyrimidin-5-yl)-2-[rac- (3R,5S)-3,4,5- trimethylpiperazin-1-yl] phenyl]-3-hydroxyquinoline- 4-carboxamide::US11319299, Example 282	WD repeat-containing protein 5				 1.98						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553226	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553226&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138541638	469797093							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166987	CN(C)[C@@H]1CCN(C1)c1cc(F)c(cc1NC(=O)c1cn(C)nc1C(F)(F)F)-c1cnc(nc1)N1CCOCC1	InChI=1S/C26H30F4N8O2/c1-35(2)17-4-5-38(14-17)22-11-20(27)18(16-12-31-25(32-13-16)37-6-8-40-9-7-37)10-21(22)33-24(39)19-15-36(3)34-23(19)26(28,29)30/h10-13,15,17H,4-9,14H2,1-3H3,(H,33,39)/t17-/m1/s1	PFYCWMDTXIYYTR-QGZVFWFLSA-N	553227	N-[4-fluoro-5-(2- morpholin-4-ylpyrimidin- 5-yl)-2-[rac-(3R)-3- (dimethylamino)pyrrolidin-1- yl]phenyl]-1-methyl-3- (trifluoromethyl)pyrazole-4- carboxamide::US11319299, Example 283	WD repeat-containing protein 5				 14.8						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553227	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553227&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138541648	469797094							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166988	C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1cn(C)nc1C(F)(F)F)-c1cnc(nc1)N1CCOCC1	InChI=1S/C26H30F4N8O2/c1-16-14-38(5-4-35(16)2)22-11-20(27)18(17-12-31-25(32-13-17)37-6-8-40-9-7-37)10-21(22)33-24(39)19-15-36(3)34-23(19)26(28,29)30/h10-13,15-16H,4-9,14H2,1-3H3,(H,33,39)/t16-/m0/s1	BRBNCQUKOWCIAU-INIZCTEOSA-N	553228	N-[4-fluoro-5-(2-morpholin-4- ylpyrimidin-5-yl)-2-[rac-(3R)- 3,4-dimethylpiperazin-1- yl]phenyl]-1-methyl-3- (trifluoromethyl)pyrazole-4- carboxamide::US11319299, Example 284	WD repeat-containing protein 5				 8.13						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553228	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553228&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138551465	469797095							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166989	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCN(CC1)C(=O)N(C)C			553229	N-[5-[1-(dimethylcarbamoyl)- 3,6-dihydro-2H-pyridin-4- yl]-4-fluoro-2-[rac-(3R,5S)- 3,4,5-trimethylpiperazin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 285	WD repeat-containing protein 5				 1.01						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553229	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553229&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607986	469797096							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166990	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCN(CC1)C(=O)N1CCCC1			553230	N-[4-fluoro-5-[1- (pyrrolidine-1-carbonyl)- 3,6-dihydro-2H-pyridin- 4-yl]-2-[rac-(3R,5S)- 3,4,5-trimethylpiperazin- 1-yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 286	WD repeat-containing protein 5				 1.18						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553230	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553230&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607987	469797097							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166991	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCN(CC1)C(=O)N1CCN(C)CC1			553231	N-[4-fluoro-5-[1-(4- methylpiperazine-1- carbonyl)-3,6-dihydro- 2H-pyridin-4-yl]-2-[rac- (3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 287	WD repeat-containing protein 5				 1.39						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553231	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553231&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607988	469797098							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166992	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCN(CC1)C(=O)Oc1ccccc1			553232	US11319299, Example 288::phenyl 4-[2-fluoro-5-[[6- oxo-4-(trifluoromethyl)- 1H-pyridine-3- carbonyl]amino]-4-[rac- (3R,5S)-3,4,5- trimethylpiperazin- 1-yl]phenyl]-3,6-dihydro- 2H-pyridine-1-carboxylate	WD repeat-containing protein 5				 1.11						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553232	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553232&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607989	469797099							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166993	C[C@H]1CC(C[C@@H](C)O1)N1CCC(=CC1)c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)(F)F)c(cc1F)N1C[C@H](C)N(C)[C@H](C)C1			553233	N-[4-fluoro-5-[1-[rac- (2R,6S)-2,6-dimethyloxan- 4-yl]-3,6-dihydro-2H- pyridin-4-yl]-2-[rac- (3S,5R)-3,4,5- trimethylpiperazin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 289	WD repeat-containing protein 5				 3.74						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553233	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553233&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607990	469797100							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166994	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1ccc(O)cc1C(F)(F)F)-c1cnc(nc1)N1CCOCC1	InChI=1S/C29H32F4N6O3/c1-17-15-39(16-18(2)37(17)3)26-12-24(30)22(19-13-34-28(35-14-19)38-6-8-42-9-7-38)11-25(26)36-27(41)21-5-4-20(40)10-23(21)29(31,32)33/h4-5,10-14,17-18,40H,6-9,15-16H2,1-3H3,(H,36,41)/t17-,18+	PODUHTRDZORXNJ-HDICACEKSA-N	553234	N-[4-fluoro-5-(2-morpholin- 4-ylpyrimidin-5-yl)-2-[rac- (3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-4-hydroxy-2- (trifluoromethyl)benzamide::US11319299, Example 290	WD repeat-containing protein 5				 8.90						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553234	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553234&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			137377525	469797101							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166995	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1cc(O)cc(F)c1F)-c1cnc(nc1)N1CCOCC1	InChI=1S/C28H31F3N6O3/c1-16-14-37(15-17(2)35(16)3)25-11-22(29)20(18-12-32-28(33-13-18)36-4-6-40-7-5-36)10-24(25)34-27(39)21-8-19(38)9-23(30)26(21)31/h8-13,16-17,38H,4-7,14-15H2,1-3H3,(H,34,39)/t16-,17+	AFEJHDQULKSWMA-CALCHBBNSA-N	553235	2,3-difluoro-N-[4-fluoro- 5-(2-morpholin-4- ylpyrimidin-5-yl)-2-[rac- (3R,5S)-3,4,5- trimethylpiperazin-1-yl] phenyl]-5-hydroxybenzamide::US11319299, Example 291	WD repeat-containing protein 5				 4.21						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553235	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553235&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138542025	469797102							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166996	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccnc(OCC2CCC2)c1			553236	N-[5-[2-(cyclobutylmethoxy) pyridin-4-yl]-4-fluoro-2-[rac- (3R,5S)-3,4,5- trimethylpiperazin-1-yl] phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 292	WD repeat-containing protein 5				 4.32						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553236	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553236&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607991	469797103							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166997	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccnc(OCC(C)(C)C)c1			553237	N-[5-[2-(2,2- dimethylpropoxy)pyridin- 4-yl]-4-fluoro-2-[rac-(3R,5S)- 3,4,5-trimethylpiperazin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 293	WD repeat-containing protein 5				 3.00						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553237	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553237&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607992	469797104							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166998	CCN(CC)c1ncc(cn1)-c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)(F)F)c(cc1F)N1C[C@H](C)N(C)[C@H](C)C1			553238	N-[5-[2-(diethylamino) pyrimidin-5-yl]-4- fluoro-2-[rac-(3R,5S)- 3,4,5-trimethylpiperazin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 294	WD repeat-containing protein 5				 2.24						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553238	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553238&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607993	469797105							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1166999	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1cccc(F)c1C(F)(F)F)-c1cnc(nc1)N1CCOCC1	InChI=1S/C29H31F5N6O2/c1-17-15-40(16-18(2)38(17)3)25-12-23(31)21(19-13-35-28(36-14-19)39-7-9-42-10-8-39)11-24(25)37-27(41)20-5-4-6-22(30)26(20)29(32,33)34/h4-6,11-14,17-18H,7-10,15-16H2,1-3H3,(H,37,41)/t17-,18+	OXFDXLFRAFTCOD-HDICACEKSA-N	553239	3-fluoro-N-[4-fluoro-5-(2- morpholin-4-ylpyrimidin- 5-yl)-2-[rac-(3R,5S)-3,4,5- trimethylpiperazin-1-yl] phenyl]-2-(trifluoromethyl) benzamide::US11319299, Example 295	WD repeat-containing protein 5				 11.1						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553239	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553239&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			137376700	469797106							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167000	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1cc(F)c(F)c(F)c1)-c1cnc(nc1)N1CCOCC1	InChI=1S/C28H30F4N6O2/c1-16-14-38(15-17(2)36(16)3)25-11-21(29)20(19-12-33-28(34-13-19)37-4-6-40-7-5-37)10-24(25)35-27(39)18-8-22(30)26(32)23(31)9-18/h8-13,16-17H,4-7,14-15H2,1-3H3,(H,35,39)/t16-,17+	UNXVTEPFUXMILW-CALCHBBNSA-N	553240	3,4,5-trifluoro-N-[4-fluoro- 5-(2-morpholin-4- ylpyrimidin-5-yl)-2- [rac-(3R,5S)-3,4,5- trimethylpiperazin-1-yl] phenyl]benzamide::US11319299, Example 296	WD repeat-containing protein 5				 21.2						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553240	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553240&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			137376916	469797107							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167001	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c(F)cccc1C(F)(F)F)-c1cnc(nc1)N1CCOCC1	InChI=1S/C29H31F5N6O2/c1-17-15-40(16-18(2)38(17)3)25-12-23(31)20(19-13-35-28(36-14-19)39-7-9-42-10-8-39)11-24(25)37-27(41)26-21(29(32,33)34)5-4-6-22(26)30/h4-6,11-14,17-18H,7-10,15-16H2,1-3H3,(H,37,41)/t17-,18+	GSGOUECYJUQOBF-HDICACEKSA-N	553241	2-fluoro-N-[4-fluoro-5- (2-morpholin-4-ylpyrimidin- 5-yl)-2-[rac-(3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-6- (trifluoromethyl)benzamide::US11319299, Example 297	WD repeat-containing protein 5				 22.9						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553241	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553241&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			137377097	469797108							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167002	C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1ccc(F)cc1C(F)(F)F)-c1cnc(nc1)N1CCOCC1	InChI=1S/C28H29F5N6O2/c1-17-16-39(6-5-37(17)2)25-13-23(30)21(18-14-34-27(35-15-18)38-7-9-41-10-8-38)12-24(25)36-26(40)20-4-3-19(29)11-22(20)28(31,32)33/h3-4,11-15,17H,5-10,16H2,1-2H3,(H,36,40)/t17-/m0/s1	RYOBVJGRASCNFQ-KRWDZBQOSA-N	553242	4-fluoro-N-[4-fluoro-5- (2-morpholin-4-ylpyrimidin- 5-yl)-2-[rac-(3R)-3,4- dimethylpiperazin-1- yl]phenyl]-2- (trifluoromethyl)benzamide::US11319299, Example 298::US11319299, Example 299	WD repeat-containing protein 5				 4.22						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553242	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553242&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138551560	469797109							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167003	C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1ccc(F)cc1C(F)(F)F)-c1cnc(nc1)N1CCOCC1	InChI=1S/C28H29F5N6O2/c1-17-16-39(6-5-37(17)2)25-13-23(30)21(18-14-34-27(35-15-18)38-7-9-41-10-8-38)12-24(25)36-26(40)20-4-3-19(29)11-22(20)28(31,32)33/h3-4,11-15,17H,5-10,16H2,1-2H3,(H,36,40)/t17-/m0/s1	RYOBVJGRASCNFQ-KRWDZBQOSA-N	553242	4-fluoro-N-[4-fluoro-5- (2-morpholin-4-ylpyrimidin- 5-yl)-2-[rac-(3R)-3,4- dimethylpiperazin-1- yl]phenyl]-2- (trifluoromethyl)benzamide::US11319299, Example 298::US11319299, Example 299	WD repeat-containing protein 5				 0.569						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553242	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553242&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138551560	469797109							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167004	C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1cn(C)c(=O)cc1C(F)(F)F)-c1ccc(nc1)N1CCN(C)CC1	InChI=1S/C30H35F4N7O2/c1-19-17-41(12-9-38(19)3)26-15-24(31)21(20-5-6-27(35-16-20)40-10-7-37(2)8-11-40)13-25(26)36-29(43)22-18-39(4)28(42)14-23(22)30(32,33)34/h5-6,13-16,18-19H,7-12,17H2,1-4H3,(H,36,43)/t19-/m0/s1	VWDUQBBEOGKQCJ-IBGZPJMESA-N	553244	N-[4-fluoro-5-[6-(4- methylpiperazin-1- yl)pyridin-3-yl]-2-[rac-(3R)- 3,4-dimethylpiperazin-1- yl]phenyl]-1-methyl-6-oxo- (trifluoromethyl)pyridine- 3-carboxamide::US11319299, Example 301	WD repeat-containing protein 5				 5.26						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553244	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553244&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138551445	469797110							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167005	C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1cn(C)c(=O)cc1C(F)(F)F)-c1ccc(cc1)N1CCN(C)CC1	InChI=1S/C31H36F4N6O2/c1-20-18-41(14-11-38(20)3)28-17-26(32)23(21-5-7-22(8-6-21)40-12-9-37(2)10-13-40)15-27(28)36-30(43)24-19-39(4)29(42)16-25(24)31(33,34)35/h5-8,15-17,19-20H,9-14,18H2,1-4H3,(H,36,43)/t20-/m0/s1	NXDIXYKRMWWSNT-FQEVSTJZSA-N	553245	N-[4-fluoro-5-[4-(4- methylpiperazin-1- yl)phenyl]-2-[rac-(3R)-3,4- dimethylpiperazin-1- yl]phenyl]-1-methyl-6-oxo- 4-(trifluoromethyl)pyridine- 3-carboxamide::US11319299, Example 302	WD repeat-containing protein 5				 5.37						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553245	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553245&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138551452	469797111							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167006	CCCN(C)C1CCN(C1)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cnc(nc1)N1CCOCC1			553246	N-[4-fluoro-2-[3- [methyl(propyl)amino] pyrrolidin-1-yl]-5-(2- morpholin-4-ylpyrimidin- 5-yl)phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 303	WD repeat-containing protein 5				 1.68						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553246	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553246&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607994	469797112							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167007	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCN(CC1)C(=O)CN(C)C			553247	N-[5-[1-[2- (dimethylamino)acetyl]- 3,6-dihydro-2H-pyridin- 4-yl]-4-fluoro-2-[rac- (3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 305	WD repeat-containing protein 5				 2.61						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553247	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553247&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607995	469797113							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167008	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cnc(nc1)N1CCN(CC1)C(=O)CCC(O)=O			553248	4-[4-[5-[2-fluoro-5-[[6- oxo-4-(trifluoromethyl)- 1H-pyridine-3-carbonyl]amino]- 4-[rac-(3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]pyrimidin-2- yl]piperazin-1-yl]-4- oxobutanoic acid::US11319299, Example 306	WD repeat-containing protein 5				 0.789						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553248	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553248&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607996	469797114							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167009	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1cn(C)c(=O)cc1C(F)(F)F)C1=CCN(CC1)C(=O)OC(C)(C)C	InChI=1S/C31H39F4N5O4/c1-18-15-40(16-19(2)38(18)7)26-14-24(32)21(20-8-10-39(11-9-20)29(43)44-30(3,4)5)12-25(26)36-28(42)22-17-37(6)27(41)13-23(22)31(33,34)35/h8,12-14,17-19H,9-11,15-16H2,1-7H3,(H,36,42)/t18-,19+	KNQZMPKRDSEDHL-KDURUIRLSA-N	553249	US11319299, Example 313::tert-butyl 4-[2-fluoro-5- [[1-methyl-6-oxo-4- (trifluoromethyl)pyridine- 3-carbonyl]amino]-4- [rac-(3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-3,6-dihydro- 2H-pyridine-1-carboxylate	WD repeat-containing protein 5				 3.10						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553249	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553249&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			137376754	469797115							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167010	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)F)-c1ccc(OCC2CC2)nc1			553250	N-[5-[6-(cyclopropylmethoxy) pyridin-3-yl]-4-fluoro-2-[rac- (3R,5S)-3,4,5-trimethylpiperazin- 1-yl]phenyl]-4-(difluoromethyl)- 6-oxo-1H-pyridine-3-carboxamide::US11319299, Example 314	WD repeat-containing protein 5				 1.67						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553250	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553250&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607997	469797116							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167011	CCn1cc(C(=O)Nc2cc(c(F)cc2N2C[C@H](C)N(C)[C@H](C)C2)-c2cnc(nc2)N2CCOCC2)c(cc1=O)C(F)(F)F	InChI=1S/C30H35F4N7O3/c1-5-39-17-22(23(11-27(39)42)30(32,33)34)28(43)37-25-10-21(20-13-35-29(36-14-20)40-6-8-44-9-7-40)24(31)12-26(25)41-15-18(2)38(4)19(3)16-41/h10-14,17-19H,5-9,15-16H2,1-4H3,(H,37,43)/t18-,19+	HJYQEVDQXZSVMQ-KDURUIRLSA-N	553251	1-ethyl-N-[4-fluoro-5-(2- morpholin-4-ylpyrimidin- 5-yl)-2-[rac-(3R,5S)- 3,4,5-trimethylpiperazin- 1-yl]phenyl]-6-oxo-4- (trifluoromethyl)pyridine- 3-carboxamide::US11319299, Example 315	WD repeat-containing protein 5				 8.49						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553251	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553251&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138541772	469797117							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167012	C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1ccc(F)cc1C(F)(F)F)-c1cnc(nc1)N1CCN(C)CC1	InChI=1S/C29H32F5N7O/c1-18-17-41(11-8-39(18)3)26-14-24(31)22(19-15-35-28(36-16-19)40-9-6-38(2)7-10-40)13-25(26)37-27(42)21-5-4-20(30)12-23(21)29(32,33)34/h4-5,12-16,18H,6-11,17H2,1-3H3,(H,37,42)/t18-/m0/s1	HVKIUSLOHGSPGV-SFHVURJKSA-N	553252	4-fluoro-N-[4-fluoro-5-[2- (4-methylpiperazin-1- yl)pyrimidin-5-yl]-2-[rac- (3R)-3,4-dimethylpiperazin-1- yl]phenyl]-2-(trifluoromethyl) benzamide::US11319299, Example 316	WD repeat-containing protein 5				 0.989						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553252	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553252&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138542106	469797118							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167013	C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1ccc(F)cc1C(F)(F)F)-c1ccc(nc1)N1CCN(C)CC1	InChI=1S/C30H33F5N6O/c1-19-18-41(13-10-39(19)3)27-16-25(32)23(20-4-7-28(36-17-20)40-11-8-38(2)9-12-40)15-26(27)37-29(42)22-6-5-21(31)14-24(22)30(33,34)35/h4-7,14-17,19H,8-13,18H2,1-3H3,(H,37,42)/t19-/m0/s1	GDQZJYOBXGEDSY-IBGZPJMESA-N	553253	4-fluoro-N-[4-fluoro-5-[6- (4-methylpiperazin-1- yl)pyridin-3-yl]-2-[rac- (3R)-3,4-dimethylpiperazin-1- yl]phenyl]-2-(trifluoromethyl) benzamide::US11319299, Example 317	WD repeat-containing protein 5				 5.54						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553253	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553253&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138551349	469797119							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167014	C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1cccc(Cl)c1Cl)-c1cnc(nc1)N1CCOCC1	InChI=1S/C27H29Cl2FN6O2/c1-17-16-36(7-6-34(17)2)24-13-22(30)20(18-14-31-27(32-15-18)35-8-10-38-11-9-35)12-23(24)33-26(37)19-4-3-5-21(28)25(19)29/h3-5,12-15,17H,6-11,16H2,1-2H3,(H,33,37)/t17-/m0/s1	DXCOFRVCVLVXFQ-KRWDZBQOSA-N	553254	2,3-dichloro-N-[4-fluoro- 5-(2-morpholin-4- ylpyrimidin-5-yl)-2-[rac- (3R)-3,4-dimethylpiperazin-1- yl]phenyl]benzamide::US11319299, Example 318	WD repeat-containing protein 5				 6.68						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553254	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553254&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138551566	469797120							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167015	C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cnc(nc1)N1CC(C)(C)OC(C)(C)C1			553255	N-[4-fluoro-2-[rac-(3R)- 3,4-dimethylpiperazin-1- yl]-5-[2-(2,2,6,6- tetramethylmorpholin-4- yl)pyrimidin-5-yl]phenyl]-6- oxo-4-(trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 319	WD repeat-containing protein 5				 1.61						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553255	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553255&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607998	469797121							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167016	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cnc(nc1)N1CC(C)(C)OC(C)(C)C1			553256	N-[4-fluoro-2-[rac-(3R,5S)-3,4,5- trimethylpiperazin-1-yl]- 5-[2-(2,2,6,6- tetramethylmorpholin-4- yl)pyrimidin-5-yl]phenyl]-6- oxo-4-(trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 320	WD repeat-containing protein 5				 0.722						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553256	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553256&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607999	469797122							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167017	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1cc([nH]n1)C(F)(F)F)-c1cnc(nc1)N1CCOCC1			553257	N-[4-fluoro-5-(2- morpholin-4-ylpyrimidin- 5-yl)-2-[rac-(3R,5S)- 3,4,5-trimethylpiperazin- 1-yl]phenyl]-5-(trifluoromethyl)- 1H-pyrazole-3-carboxamide::US11319299, Example 321	WD repeat-containing protein 5				 63.1						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553257	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553257&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			137377417	469797123							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167018	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCCN(C1)C(=O)OC(C)(C)C			553258	US11319299, Example 322::tert-butyl 5-[2-fluoro-5- [[6-oxo-4-(trifluoromethyl)-1H- pyridine-3-carbonyl]amino]-4- [rac-(3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-3,6-dihydro- 2H-pyridine-1-carboxylate	WD repeat-containing protein 5				 1.36						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553258	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553258&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608000	469797124							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167019	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCN(C1)C(=O)OC(C)(C)C			553259	US11319299, Example 323::tert-butyl 3-[2-fluoro-5- [[6-oxo-4-(trifluoromethyl)-1H- pyridine-3-carbonyl]amino]-4- [rac-(3R,5S)-3,4,5- trimethylpiperazin-1-yl]phenyl]- 2,5-dihydropyrrole-1-carboxylate	WD repeat-containing protein 5				 2.48						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553259	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553259&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608001	469797125							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167020	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CC2CCC(C1)N2C(=O)OC(C)(C)C			553260	US11319299, Example 324::tert-butyl 3-[2-fluoro-5- [[6-oxo-4-(trifluoromethyl)-1H- pyridine-3-carbonyl]amino]-4- [rac-(3R,5S)-3,4,5- trimethylpiperazin-1-yl]phenyl]- 8-azabicyclo[3.2.1]oct-2-ene- 8-carboxylate	WD repeat-containing protein 5				 15.2						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553260	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553260&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608002	469797126							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167021	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1cn(C)c(=O)cc1C(F)(F)F)C1=CCCN(C1)C(=O)OC(C)(C)C	InChI=1S/C31H39F4N5O4/c1-18-14-40(15-19(2)38(18)7)26-13-24(32)21(20-9-8-10-39(16-20)29(43)44-30(3,4)5)11-25(26)36-28(42)22-17-37(6)27(41)12-23(22)31(33,34)35/h9,11-13,17-19H,8,10,14-16H2,1-7H3,(H,36,42)/t18-,19+	ROSJNMMXKDMKTJ-KDURUIRLSA-N	553261	US11319299, Example 325::tert-butyl 5-[2-fluoro-5- [[1-methyl-6-oxo-4- (trifluoromethyl)pyridine- 3-carbonyl]amino]-4- [rac-(3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-3,6-dihydro- 2H-pyridine-1-carboxylate	WD repeat-containing protein 5				 7.30						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553261	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553261&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138541790	469797127							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167022	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1cn(C)c(=O)cc1C(F)(F)F)C1=CCN(C1)C(=O)OC(C)(C)C	InChI=1S/C30H37F4N5O4/c1-17-13-39(14-18(2)37(17)7)25-12-23(31)20(19-8-9-38(15-19)28(42)43-29(3,4)5)10-24(25)35-27(41)21-16-36(6)26(40)11-22(21)30(32,33)34/h8,10-12,16-18H,9,13-15H2,1-7H3,(H,35,41)/t17-,18+	JUAPNWKLPCRPCQ-HDICACEKSA-N	553262	US11319299, Example 326::tert-butyl 3-[2-fluoro-5- [[1-methyl-6-oxo-4- (trifluoromethyl)pyridine- 3-carbonyl]amino]-4- [rac-(3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-2,5-dihydropyrrole- 1-carboxylate	WD repeat-containing protein 5				 3.05						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553262	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553262&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			137376773	469797128							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167023	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1cn(C)c(=O)cc1C(F)(F)F)C1=CC2CCC(C1)N2C(=O)OC(C)(C)C	InChI=1S/C33H41F4N5O4/c1-18-15-41(16-19(2)40(18)7)28-14-26(34)23(20-10-21-8-9-22(11-20)42(21)31(45)46-32(3,4)5)12-27(28)38-30(44)24-17-39(6)29(43)13-25(24)33(35,36)37/h10,12-14,17-19,21-22H,8-9,11,15-16H2,1-7H3,(H,38,44)/t18-,19+,21?,22?	CGAKXNPHSFHSGB-IVCWUUCSSA-N	553263	US11319299, Example 327::tert-butyl 3-[2-fluoro-5- [[1-methyl-6-oxo-4- (trifluoromethyl)pyridine- 3-carbonyl]amino]-4- [rac-(3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-8-azabicyclo[3.2.1] oct-2-ene-8-carboxylate	WD repeat-containing protein 5				 123						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553263	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553263&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			137376743	469797129							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167024	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCCNC1			553264	N-[4-fluoro-2-[rac-(3R,5S)- 3,4,5-trimethylpiperazin-1-yl]- 5-(1,2,3,6-tetrahydropyridin-5- yl)phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 328	WD repeat-containing protein 5				 1.89						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553264	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553264&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608003	469797130							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167025	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCNC1			553265	N-[5-(2,5-dihydro-1H- pyrrol-3-yl)-4-fluoro-2- [rac-(3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 329	WD repeat-containing protein 5				 4.05						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553265	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553265&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608004	469797131							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167026	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CC2CCC(C1)N2			553266	N-[5-(8-azabicyclo[3.2.1]oct-2- en-3-yl)-4-fluoro-2-[rac- (3R,5S)-3,4,5- trimethylpiperazin-1-yl]phenyl]- 6-oxo-4-(trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 330	WD repeat-containing protein 5				 5.74						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553266	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553266&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608005	469797132							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167027	C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)F)-c1ccc(nc1)N1CCOCC1			553267	4-(difluoromethyl)-N-[4- fluoro-5-(6-morpholin-4- ylpyridin-3-yl)-2-[rac-(3R)-3,4- dimethylpiperazin-1-yl]phenyl]- 6-oxo-1H-pyridine-3-carboxamide::US11319299, Example 331	WD repeat-containing protein 5				 2.01						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553267	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553267&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608006	469797133							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167028	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCCN(C1)c1ncccn1			553268	N-[4-fluoro-5-(1-pyrimidin-2- yl-3,6-dihydro-2H-pyridin-5-yl)- 2-[rac-(3R,5S)-3,4,5- trimethylpiperazin-1-yl]phenyl]- 6-oxo-4-(trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 334::US11319299, Example 644	WD repeat-containing protein 5				 0.095						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553268	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553268&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608007	469797134							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167029	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCN(C1)c1ncccn1			553269	N-[4-fluoro-5-(1-pyrimidin-2- yl-2,5-dihydropyrrol-3-yl)-2- [rac-(3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 335	WD repeat-containing protein 5				 2.56						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553269	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553269&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608008	469797135							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167030	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CC2CCC(C1)N2c1ncccn1			553270	N-[4-fluoro-5-(8-pyrimidin-2- yl-8-azabicyclo[3.2.1]oct-2- en-3-yl)-2-[rac-(3R,5S)- 3,4,5-trimethylpiperazin- 1-yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 336	WD repeat-containing protein 5				 12.5						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553270	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553270&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608009	469797136							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167031	C[C@H]1COCCN1c1ncc(cn1)-c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)(F)F)c(cc1F)N1CCN(C)[C@@H](C)C1			553271	N-[4-fluoro-2-[rac-(3R)- 3,4-dimethylpiperazin-1- yl]-5-[2-[rac-(3R)-3- methylmorpholin-4- yl]pyrimidin-5-yl]phenyl]- 6-oxo-4-(trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 337	WD repeat-containing protein 5				 1.16						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553271	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553271&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608010	469797137							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167032	C[C@H]1COCCN1c1ncc(cn1)-c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)(F)F)c(cc1F)N1C[C@H](C)N(C)[C@H](C)C1			553272	N-[4-fluoro-5-[2-[rac- (3R)-3-methylmorpholin- 4-yl]pyrimidin-5-yl]-2- [rac-(3S,5R)-3,4,5- trimethylpiperazin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 338	WD repeat-containing protein 5				 2.08						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553272	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553272&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608011	469797138							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167033	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1CNC(=NC1)N1CCOCC1			553273	N-[4-fluoro-5-(2- morpholin-4-yl-1,4,5,6- tetrahydropyrimidin-5- yl)-2-[rac-(3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 339	WD repeat-containing protein 5				 275						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553273	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553273&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608012	469797139							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167034	C[C@@H]1CN(CCO1)c1ncc(cn1)-c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)(F)F)c(cc1F)N1CCN(C)[C@@H](C)C1			553274	N-[4-fluoro-2-[rac-(3S)-3,4- dimethylpiperazin-1-yl]-5-[2- [rac-(2R)-2-methylmorpholin-4- yl]pyrimidin-5-yl]phenyl]-6-oxo- 4-(trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 340	WD repeat-containing protein 5				 0.551						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553274	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553274&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608013	469797140							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167035	C[C@H]1CN(C[C@@H](C)O1)c1ccc(cn1)-c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)(F)F)c(cc1F)N1CCN(C)[C@@H](C)C1			553275	N-[4-fluoro-5-[6-[rac-(2R,6S)- 2,6-dimethylmorpholin-4- yl]pyridin-3-yl]-2-[rac-(3R)-3,4- dimethylpiperazin-1-yl]phenyl]- 6-oxo-4-(trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 341	WD repeat-containing protein 5				 1.97						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553275	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553275&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608014	469797141							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167036	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1cn(C)c(=O)cc1C(F)F)-c1cnc(nc1)N1CCOCC1	InChI=1S/C29H34F3N7O3/c1-17-14-39(15-18(2)37(17)4)25-11-23(30)20(19-12-33-29(34-13-19)38-5-7-42-8-6-38)9-24(25)35-28(41)22-16-36(3)26(40)10-21(22)27(31)32/h9-13,16-18,27H,5-8,14-15H2,1-4H3,(H,35,41)/t17-,18+	ZQNSTLNTAVMJTL-HDICACEKSA-N	553276	4-(difluoromethyl)-N-[4- fluoro-5-(2-morpholin-4- ylpyrimidin-5-yl)-2-[rac- (3R,5S)-3,4,5-trimethylpiperazin- 1-yl]phenyl]-1-methyl-6- oxopyridine-3-carboxamide::US11319299, Example 342	WD repeat-containing protein 5				 6.87						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553276	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553276&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			137377538	469797142							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167037	CCN(C)[C@@H]1CN(C[C@H]1F)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cnc(nc1)N1CCOCC1			553277	N-[4-fluoro-5-(2-morpholin-4- ylpyrimidin-5-yl)-2-[rac- (3R,4R)-3-[ethyl(methyl) amino]-4-fluoropyrrolidin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 344	WD repeat-containing protein 5				 12.4						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553277	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553277&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608015	469797143							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167038	CCN(C)[C@@H]1CCN(C1)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cnc(nc1)N1CCOCC1			553278	N-[4-fluoro-5-(2-morpholin-4- ylpyrimidin-5-yl)-2-[rac-(3R)-3- [ethyl(methyl)amino]pyrrolidin- 1-yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H-pyridine-3- carboxamide::US11319299, Example 345	WD repeat-containing protein 5				 1.20						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553278	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553278&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608016	469797144							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167039	CC(C)[C@H]1CN(CCO1)c1ncc(cn1)-c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)(F)F)c(cc1F)N1CCN(C)[C@@H](C)C1			553279	N-[4-fluoro-2-[rac-(3R)- 3,4-dimethylpiperazin-1- yl]-5-[2-[rac-(2R)-2- propan-2-ylmorpholin-4- yl]pyrimidin-5-yl]phenyl]-6- oxo-4-(trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 347	WD repeat-containing protein 5				 0.606						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553279	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553279&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608017	469797145							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167040	CC(C)[C@H]1CN(CCO1)c1ncc(cn1)-c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)(F)F)c(cc1F)N1C[C@H](C)N(C)[C@H](C)C1			553280	N-[4-fluoro-5-[2-[rac-(2R)-2- propan-2-ylmorpholin-4- yl]pyrimidin-5-yl]-2-[rac- (3S,5R)-3,4,5-trimethylpiperazin- 1-yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 348	WD repeat-containing protein 5				 2.28						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553280	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553280&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608018	469797146							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167041	C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cnc(nc1)N1CCOC(C)(C)C1			553281	N-[5-[2-(2,2-dimethylmorpholin- 4-yl)pyrimidin-5-yl]-4-fluoro-2- [rac-(3R)-3,4-dimethylpiperazin- 1-yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 349	WD repeat-containing protein 5				 2.35						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553281	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553281&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608019	469797147							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167042	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cnc(nc1)N1CCOC(C)(C)C1			553282	N-[5-[2-(2,2-dimethylmorpholin- 4-yl)pyrimidin-5-yl]-4- fluoro-2-[rac-(3R,5S)- 3,4,5-trimethylpiperazin- 1-yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 350	WD repeat-containing protein 5				 1.42						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553282	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553282&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608020	469797148							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167043	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cnc(nc1)N1C2CCC1CC2			553283	N-[5-[2-(7-azabicyclo[2.2.1] heptan-7-yl)pyrimidin-5-yl]-4- fluoro-2-[rac-(3R,5S)-3,4,5- trimethylpiperazin-1-yl]phenyl]- 6-oxo-4-(trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 352	WD repeat-containing protein 5				 2.73						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553283	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553283&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608021	469797149							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167044	C[C@H]1CN(C[C@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cnc(nc1)N1CCOCC1			553284	N-[4-fluoro-5-(2-morpholin-4- ylpyrimidin-5-yl)-2-[rac-(3R,5R)- 3,4,5-trimethylpiperazin-1-yl] phenyl]-6-oxo-4-(trifluoromethyl)- 1H-pyridine-3-carboxamide::US11319299, Example 355	WD repeat-containing protein 5				 37.9						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553284	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553284&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608022	469797150							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167045	C[C@H]1CN(C[C@@H](C)O1)c1ncc(cn1)-c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)(F)F)c(cc1F)N1C[C@H](C)N(C)[C@@H](C)C1			553285	N-[4-fluoro-5-[2-[rac-(2R,6S)-2,6- dimethylmorpholin-4-yl] pyrimidin-5-yl]-2-[rac-(3R,5R)- 3,4,5-trimethylpiperazin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 356	WD repeat-containing protein 5				 19.9						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553285	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553285&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608023	469797151							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167046	C[C@H]1CN(C[C@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(N2CCOCC2)c(F)c1			553286	N-[4-fluoro-5-(3-fluoro- 4-morpholin-4-ylphenyl)- 2-[rac-(3R,5R)-3,4,5- trimethylpiperazin-1-yl]phenyl]- 6-oxo-4-(trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 357	WD repeat-containing protein 5				 133						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553286	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553286&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608024	469797152							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167047	C[C@H]1CN(C[C@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(OCC2CC2)nc1			553287	N-[5-[6-(cyclopropylmethoxy) pyridin-3-yl]-4-fluoro-2-[rac- (3R,5R)-3,4,5-trimethylpiperazin- 1-yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 361	WD repeat-containing protein 5				 48.3						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553287	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553287&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608025	469797153							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167048	C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cnc(nc1)N(C)[C@H]1CCOC1			553288	N-[4-fluoro-5-[2-[methyl- [rac-(3R)-oxolan-3- yl]amino]pyrimidin-5-yl]- 2-[rac-(3R)-3,4- dimethylpiperazin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 362	WD repeat-containing protein 5				 0.244						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553288	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553288&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608026	469797154							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167049	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cnc(nc1)N(C)[C@H]1CCOC1			553289	N-[4-fluoro-5-[2-[methyl- [rac-(3R)-oxolan-3- yl]amino]pyrimidin-5-yl]- 2-[rac-(3S,5R)-3,4,5- trimethylpiperazin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 363	WD repeat-containing protein 5				 0.634						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553289	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553289&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608027	469797155							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167050	C[C@H]1CN(C[C@@H](C)N1)c1cc(F)c(cc1NC(=O)c1ccc(F)cc1C(F)(F)F)-c1cnc(nc1)N1CCOCC1	InChI=1S/C28H29F5N6O2/c1-16-14-39(15-17(2)36-16)25-11-23(30)21(18-12-34-27(35-13-18)38-5-7-41-8-6-38)10-24(25)37-26(40)20-4-3-19(29)9-22(20)28(31,32)33/h3-4,9-13,16-17,36H,5-8,14-15H2,1-2H3,(H,37,40)/t16-,17+	NBPIUQUGOVWIDG-CALCHBBNSA-N	553290	4-fluoro-N-[4-fluoro-5-(2- morpholin-4-ylpyrimidin- 5-yl)-2-[rac-(3R,5S)-3,5- dimethylpiperazin-1- yl]phenyl]-2-(trifluoromethyl) benzamide::US11319299, Example 364	WD repeat-containing protein 5				 5.87						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553290	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553290&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			137377177	469797156							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167051	COc1cc(ncn1)N1CCC=C(C1)c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)(F)F)c(cc1F)N1C[C@H](C)N(C)[C@H](C)C1			553291	N-[4-fluoro-5-[1-(6- methoxypyrimidin-4-yl)- 3,6-dihydro-2H-pyridin- 5-yl]-2-[rac-(3R,5S)- 3,4,5-trimethylpiperazin- 1-yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 365	WD repeat-containing protein 5				 0.246						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553291	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553291&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608028	469797157							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167052	COc1cnc(nc1)N1CCC(=CC1)c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)(F)F)c(cc1F)N1C[C@H](C)N(C)[C@H](C)C1			553292	N-[4-fluoro-5-[1-(5- methoxypyrimidin-2-yl)- 3,6-dihydro-2H-pyridin- 4-yl]-2-[rac-(3R,5S)- 3,4,5-trimethylpiperazin- 1-yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 366	WD repeat-containing protein 5				 1.76						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553292	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553292&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608029	469797158							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167053	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCN(CC1)c1ncc(F)cn1			553293	N-[4-fluoro-5-[1-(5- fluoropyrimidin-2-yl)- 3,6-dihydro-2H-pyridin- 4-yl]-2-[rac-(3R,5S)- 3,4,5-trimethylpiperazin- 1-yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 367	WD repeat-containing protein 5				 1.04						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553293	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553293&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608030	469797159							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167054	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCN(CC1)c1nc(C)cc(C)n1			553294	N-[5-[1-(4,6- dimethylpyrimidin-2-yl)- 3,6-dihydro-2H-pyridin- 4-yl]-4-fluoro-2-[rac-(3R,5S)- 3,4,5-trimethylpiperazin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 368	WD repeat-containing protein 5				 2.30						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553294	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553294&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608031	469797160							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167055	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCN(CC1)c1ncc(C=O)cn1			553295	N-[4-fluoro-5-[1-(5- formylpyrimidin-2-yl)- 3,6-dihydro-2H-pyridin- 4-yl]-2-[rac-(3R,5S)- 3,4,5-trimethylpiperazin- 1-yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 369	WD repeat-containing protein 5				 0.685						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553295	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553295&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608032	469797161							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167056	C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cnc(nc1)N(C)C1CCOCC1			553296	N-[4-fluoro-5-[2-[methyl(oxan- 4-yl)amino]pyrimidin-5-yl]- 2-[rac-(3R)-3,4-dimethylpiperazin- 1-yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H-pyridine-3- carboxamide::US11319299, Example 370	WD repeat-containing protein 5				 0.866						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553296	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553296&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608033	469797162							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167057	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cnc(nc1)N(C)C1CCOCC1			553297	N-[4-fluoro-5-[2-[methyl(oxan- 4-yl)amino]pyrimidin-5-yl]- 2-[rac-(3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 371	WD repeat-containing protein 5				 0.590						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553297	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553297&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608034	469797163							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167058	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCCN(C1)C(=O)N(C)C			553298	N-[5-[1-(dimethylcarbamoyl)- 3,6-dihydro-2H-pyridin-5-yl]- 4-fluoro-2-[rac-(3R,5S)- 3,4,5-trimethylpiperazin- 1-yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 372	WD repeat-containing protein 5				 1.75						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553298	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553298&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608035	469797164							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167059	CCOC(=O)N1CCC=C(C1)c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)(F)F)c(cc1F)N1C[C@H](C)N(C)[C@H](C)C1			553299	US11319299, Example 373::ethyl 5-[2-fluoro-5-[[6-oxo-4- (trifluoromethyl)-1H-pyridine-3- carbonyl]amino]-4-[rac-(3R,5S)- 3,4,5-trimethylpiperazin-1- yl]phenyl]-3,6-dihydro-2H- pyridine-1-carboxylate	WD repeat-containing protein 5				 0.808						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553299	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553299&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608036	469797165							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167060	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCCN(C1)C(=O)N1CCCC1			553300	N-[4-fluoro-5-[1-pyrrolidine-1- carbonyl)-3,6-dihydro-2H- pyridin-5-yl]-2-[rac-(3R,5S)- 3,4,5-trimethylpiperazin-1-yl] phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 374	WD repeat-containing protein 5				 1.15						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553300	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553300&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608037	469797166							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167061	COc1cnc(nc1)N1CCC=C(C1)c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)(F)F)c(cc1F)N1C[C@H](C)N(C)[C@H](C)C1			553301	N-[4-fluoro-5-[1-(5- methoxypyrimidin-2-yl)- 3,6-dihydro-2H-pyridin- 5-yl]-2-[rac-(3R,5S)-3,4,5- trimethylpiperazin-1-yl]phenyl]- 6-oxo-4-(trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 375	WD repeat-containing protein 5				 0.688						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553301	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553301&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608038	469797167							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167062	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCCN(C1)c1ncc(C)cn1			553302	N-[4-fluoro-5-[1-(5- methylpyrimidin-2-yl)-3,6- dihydro-2H-pyridin-5-yl]-2-[rac- (3R,5S)-3,4,5-trimethylpiperazin- 1-yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H-pyridine-3- carboxamide::US11319299, Example 376	WD repeat-containing protein 5				 0.673						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553302	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553302&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608039	469797168							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167063	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCCN(C1)c1ncc(F)cn1			553303	N-[4-fluoro-5-[1-(5- fluoropyrimidin-2-yl)- 3,6-dihydro-2H-pyridin- 5-yl]-2-[rac-(3R,5S)- 3,4,5-trimethylpiperazin- 1-yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 377	WD repeat-containing protein 5				 1.30						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553303	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553303&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608040	469797169							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167064	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccnc(n1)N1CCOCC1			553304	N-[4-fluoro-5-(2- morpholin-4-ylpyrimidin- 4-yl)-2-[rac-(3R,5S)- 3,4,5-trimethylpiperazin- 1-yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 378	WD repeat-containing protein 5				 0.877						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553304	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553304&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608041	469797170							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167065	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1ccc(F)cc1C(F)(F)F)-c1cnc(nc1)N1CCN(C)CC1	InChI=1S/C30H34F5N7O/c1-18-16-42(17-19(2)40(18)4)27-13-25(32)23(20-14-36-29(37-15-20)41-9-7-39(3)8-10-41)12-26(27)38-28(43)22-6-5-21(31)11-24(22)30(33,34)35/h5-6,11-15,18-19H,7-10,16-17H2,1-4H3,(H,38,43)/t18-,19+	GWAUIRJYZIWNHS-KDURUIRLSA-N	553305	4-fluoro-N-[4-fluoro-5- [2-(4-methylpiperazin-1- yl)pyrimidin-5-yl]-2-[rac- (3R,5S)-3,4,5-trimethylpiperazin- 1-yl]phenyl]-2-(trifluoromethyl) benzamide::US11319299, Example 379	WD repeat-containing protein 5				 0.933						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553305	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553305&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138541789	469797171							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167066	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1ccc(F)cc1C(F)(F)F)-c1cnc(nc1)N(C)C	InChI=1S/C27H29F5N6O/c1-15-13-38(14-16(2)37(15)5)24-10-22(29)20(17-11-33-26(34-12-17)36(3)4)9-23(24)35-25(39)19-7-6-18(28)8-21(19)27(30,31)32/h6-12,15-16H,13-14H2,1-5H3,(H,35,39)/t15-,16+	MAKIKSDYKJDQRG-IYBDPMFKSA-N	553306	N-[5-[2-(dimethylamino) pyrimidin-5-yl]-4-fluoro-2-[rac- (3R,5S)-3,4,5-trimethylpiperazin- 1-yl]phenyl]-4-fluoro-2- (trifluoromethyl)benzamide::US11319299, Example 380	WD repeat-containing protein 5				 1.70						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553306	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553306&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138541622	469797172							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167067	C[C@H]1CN(C[C@@H](C)N1C)c1ncc(cn1)-c1cc(NC(=O)c2ccc(F)cc2C(F)(F)F)c(cc1F)N1C[C@H](C)N(C)[C@H](C)C1	InChI=1S/C32H38F5N7O/c1-18-14-43(15-19(2)41(18)5)29-11-27(34)25(22-12-38-31(39-13-22)44-16-20(3)42(6)21(4)17-44)10-28(29)40-30(45)24-8-7-23(33)9-26(24)32(35,36)37/h7-13,18-21H,14-17H2,1-6H3,(H,40,45)/t18-,19+,20-,21+	DYHKUOKFQBAXGE-FXELSEDVSA-N	553307	4-fluoro-N-[4-fluoro-2- [rac-(3R,5S)-3,4,5- trimethylpiperazin-1-yl]-5- [2-[rac-(3R,5S)-3,4,5- trimethylpiperazin-1- yl]pyrimidin-5-yl]phenyl]- 2-(trifluoromethyl)benzamide::US11319299, Example 381	WD repeat-containing protein 5				 0.310						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553307	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553307&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			137376815	469797173							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167068	C[C@H]1CN(C[C@H](C)N1C)c1cc(F)c(cc1NC(=O)c1ccc(F)cc1C(F)(F)F)-c1cnc(nc1)N1CCN(C)CC1	InChI=1S/C30H34F5N7O/c1-18-16-42(17-19(2)40(18)4)27-13-25(32)23(20-14-36-29(37-15-20)41-9-7-39(3)8-10-41)12-26(27)38-28(43)22-6-5-21(31)11-24(22)30(33,34)35/h5-6,11-15,18-19H,7-10,16-17H2,1-4H3,(H,38,43)/t18-,19-/m0/s1	GWAUIRJYZIWNHS-OALUTQOASA-N	553308	4-fluoro-N-[4-fluoro-5-[2- (4-methylpiperazin-1- yl)pyrimidin-5-yl]-2-[rac- (3R,5R)-3,4,5-trimethylpiperazin- 1-yl]phenyl]-2-(trifluoromethyl) benzamide::US11319299, Example 382	WD repeat-containing protein 5				 117						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553308	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553308&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138551519	469797174							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167069	C[C@H]1CN(C[C@@H](C)O1)c1ncc(cn1)-c1cc(NC(=O)c2cn(C)c(=O)cc2C(F)F)c(cc1F)N1CCN(C)[C@@H](C)C1	InChI=1S/C30H36F3N7O3/c1-17-13-39(7-6-37(17)4)26-10-24(31)21(20-11-34-30(35-12-20)40-14-18(2)43-19(3)15-40)8-25(26)36-29(42)23-16-38(5)27(41)9-22(23)28(32)33/h8-12,16-19,28H,6-7,13-15H2,1-5H3,(H,36,42)/t17-,18-,19+/m0/s1	KDCDWHIXQCFBPT-GBESFXJTSA-N	553309	4-(difluoromethyl)-N-[4- fluoro-5-[2-[rac-(2R,6S)- 2,6-dimethylmorpholin-4- yl]pyrimidin-5-yl]-2-[rac- (3R)-3,4-dimethylpiperazin-1- yl]phenyl]-1-methyl-6- oxopyridine-3-carboxamide::US11319299, Example 383	WD repeat-containing protein 5				 1.19						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553309	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553309&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138551362	469797175							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167070	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(nn1)N1CCOCC1			553310	N-[4-fluoro-5-(6- morpholin-4-ylpyridazin- 3-yl)-2-[rac-(3R,5S)- 3,4,5-trimethylpiperazin- 1-yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 384	WD repeat-containing protein 5				 1.53						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553310	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553310&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608042	469797176							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167071	C[C@H]1CN(C[C@@H](C)O1)c1ncc(cn1)-c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)F)c(cc1F)N1C[C@H](C)N(C)[C@H](C)C1			553311	4-(difluoromethyl)-N-[4- fluoro-5-[2-[rac-(2R,6S)- 2,6-dimethylmorpholin-4- yl]pyrimidin-5-yl]-2-[rac- (3S,5R)-3,4,5- trimethylpiperazin-1- yl]phenyl]-6-oxo-1H- pyridine-3-carboxamide::US11319299, Example 385	WD repeat-containing protein 5				 0.720						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553311	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553311&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608043	469797177							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167072	C[C@@H]1CN(CCO1)c1ncc(cn1)-c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)F)c(cc1F)N1C[C@H](C)N(C)[C@H](C)C1			553312	4-(difluoromethyl)-N-[4- fluoro-5-[2-[rac-(2R)-2- methylmorpholin-4- yl]pyrimidin-5-yl]-2-[rac- (3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-6-oxo-1H- pyridine-3-carboxamide::US11319299, Example 386	WD repeat-containing protein 5				 1.49						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553312	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553312&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608044	469797178							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167073	C[C@H]1CN(C[C@H](C)N1C)c1cc(F)c(cc1NC(=O)c1ccc(F)cc1C(F)(F)F)-c1cnc(nc1)N1CCOCC1	InChI=1S/C29H31F5N6O2/c1-17-15-40(16-18(2)38(17)3)26-12-24(31)22(19-13-35-28(36-14-19)39-6-8-42-9-7-39)11-25(26)37-27(41)21-5-4-20(30)10-23(21)29(32,33)34/h4-5,10-14,17-18H,6-9,15-16H2,1-3H3,(H,37,41)/t17-,18-/m0/s1	OVAUTHLIMOXPHS-ROUUACIJSA-N	553313	4-fluoro-N-[4-fluoro-5-(2- morpholin-4-ylpyrimidin-5- yl)-2-[rac-(3R,5R)-3,4,5- trimethylpiperazin-1- yl]phenyl]-2-(trifluoromethyl) benzamide::US11319299, Example 387	WD repeat-containing protein 5				 83.5						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553313	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553313&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138551461	469797179							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167074	C[C@@H]1CN(CCO1)c1ncc(cn1)-c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)(F)F)c(cc1F)N1C[C@H](C)N(C)[C@H](C)C1			553314	N-[4-fluoro-5-[2-[rac- (2R)-2-methylmorpholin- 4-yl]pyrimidin-5-yl]-2- [rac-(3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 388	WD repeat-containing protein 5				 0.788						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553314	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553314&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608045	469797180							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167075	C[C@H]1CN(CCO1)c1ncc(cn1)-c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)(F)F)c(cc1F)N1CCN(C)[C@@H](C)C1			553315	N-[4-fluoro-2-[rac-(3R)- 3,4-dimethylpiperazin-1- yl]-5-[2-[rac-(2R)-2- methylmorpholin-4- yl]pyrimidin-5-yl]phenyl]-6- oxo-4-(trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 389	WD repeat-containing protein 5				 0.522						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553315	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553315&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608046	469797181							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167076	C[C@H]1CN(CCO1)c1ncc(cn1)-c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)(F)F)c(cc1F)N1C[C@H](C)N(C)[C@H](C)C1			553316	N-[4-fluoro-5-[2-[rac- (2R)-2-methylmorpholin- 4-yl]pyrimidin-5-yl]-2- [rac-(3S,5R)-3,4,5- trimethylpiperazin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 390	WD repeat-containing protein 5				 0.634						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553316	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553316&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608047	469797182							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167077	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1cn(C)c(=O)cc1C(F)(F)F)C1=CCCN(C1)c1ncccn1	InChI=1S/C30H33F4N7O2/c1-18-14-41(15-19(2)39(18)4)26-13-24(31)21(20-7-5-10-40(16-20)29-35-8-6-9-36-29)11-25(26)37-28(43)22-17-38(3)27(42)12-23(22)30(32,33)34/h6-9,11-13,17-19H,5,10,14-16H2,1-4H3,(H,37,43)/t18-,19+	SUYCZVBKROVXCE-KDURUIRLSA-N	553317	N-[4-fluoro-5-(1-pyrimidin-2- yl-3,6-dihydro-2H-pyridin-5- yl)-2-[rac-(3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-1-methyl-6- oxo-4-(trifluoromethyl) pyridine-3-carboxamide::US11319299, Example 391	WD repeat-containing protein 5				 4.27						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553317	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553317&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138541654	469797183							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167078	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)N1CCN(Cc2ccc(F)cc2)CC1			553318	N-[4-fluoro-5-[4-[(4- fluorophenyl)methyl] piperazin-1-yl]-2-[rac- (3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 392	WD repeat-containing protein 5				 8.08						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553318	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553318&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608048	469797184							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167079	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)N1CCN(CC1)c1ncccn1			553319	N-[4-fluoro-5-(4- pyrimidin-2-ylpiperazin- 1-yl)-2-[rac-(3R,5S)- 3,4,5-trimethylpiperazin- 1-yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 393	WD repeat-containing protein 5				 13.3						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553319	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553319&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608049	469797185							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167080	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCN(CC1)c1ncc(CO)cn1			553320	N-[4-fluoro-5-[1-[5- (hydroxymethyl)pyrimidin- 2-yl]-3,6-dihydro-2H- pyridin-4-yl]-2-[rac- (3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 394	WD repeat-containing protein 5				 0.775						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553320	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553320&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608050	469797186							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167081	C[C@H]1CN(C[C@@H](C)O1)c1ncc(cn1)-c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)F)c(cc1F)N1CCN(C)[C@@H](C)C1			553321	4-(difluoromethyl)-N-[4- fluoro-5-[2-[rac-(2R,6S)- 2,6-dimethylmorpholin-4- yl]pyrimidin-5-yl]-2-[rac- (3S)-3,4-dimethylpiperazin-1- yl]phenyl]-6-oxo-1H- pyridine-3-carboxamide::US11319299, Example 395	WD repeat-containing protein 5				 0.152						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553321	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553321&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608051	469797187							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167082	C[C@@H]1CN(CCO1)c1ncc(cn1)-c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)F)c(cc1F)N1CCN(C)[C@@H](C)C1			553322	4-(difluoromethyl)-N-[4- fluoro-2-[rac-(3S)-3,4- dimethylpiperazin-1-yl]- 5-[2-[rac-(2R)-2- methylmorpholin-4- yl]pyrimidin-5-yl]phenyl]- 6-oxo-1H-pyridine-3- carboxamide::US11319299, Example 396	WD repeat-containing protein 5				 0.564						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553322	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553322&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608052	469797188							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167083	C[C@H]1CN(CCO1)c1ncc(cn1)-c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)F)c(cc1F)N1C[C@H](C)N(C)[C@H](C)C1			553323	4-(difluoromethyl)-N-[4- fluoro-5-[2-[rac-(2R)-2- methylmorpholin-4- yl]pyrimidin-5-yl]-2-[rac- (3S,5R)-3,4,5- trimethylpiperazin-1- yl]phenyl]-6-oxo-1H- pyridine-3-carboxamide::US11319299, Example 397	WD repeat-containing protein 5				 0.680						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553323	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553323&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608053	469797189							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167084	C[C@H]1CN(CCO1)c1ncc(cn1)-c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)F)c(cc1F)N1CCN(C)[C@@H](C)C1			553324	4-(difluoromethyl)-N-[4- fluoro-2-[rac-(3R)-3,4- dimethylpiperazin-1-yl]- 5-[2-[rac-(2R)-2- methylmorpholin-4- yl]pyrimidin-5- yl]phenyl]-6-oxo-1H- pyridine-3-carboxamide::US11319299, Example 398	WD repeat-containing protein 5				 0.899						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553324	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553324&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608054	469797190							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167085	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccnc(n1)S(C)(=O)=O			553325	N-[4-fluoro-5-(2- methylsulfonylpyrimidin- 4-yl)-2-[rac-(3R,5S)- 3,4,5-trimethylpiperazin- 1-yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 399	WD repeat-containing protein 5				 4.58						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553325	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553325&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608055	469797191							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167086	C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1ccc(F)cc1C(F)(F)F)-c1cnc(nc1)N1CCCN(C)CC1	InChI=1S/C30H34F5N7O/c1-19-18-42(12-10-40(19)3)27-15-25(32)23(20-16-36-29(37-17-20)41-8-4-7-39(2)9-11-41)14-26(27)38-28(43)22-6-5-21(31)13-24(22)30(33,34)35/h5-6,13-17,19H,4,7-12,18H2,1-3H3,(H,38,43)/t19-/m0/s1	DBNDJZSXBHLXAG-IBGZPJMESA-N	553326	4-fluoro-N-[4-fluoro-5-[2- (4-methyl-1,4-diazepan-1- yl)pyrimidin-5-yl]-2-[rac- (3R)-3,4-dimethylpiperazin-1- yl]phenyl]-2-(trifluoromethyl) benzamide::US11319299, Example 400	WD repeat-containing protein 5				 1.47						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553326	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553326&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138551462	469797192							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167087	C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1ccc(F)cc1C(F)(F)F)-c1cnc(nc1)N1CCNCC1	InChI=1S/C28H30F5N7O/c1-17-16-40(10-9-38(17)2)25-13-23(30)21(18-14-35-27(36-15-18)39-7-5-34-6-8-39)12-24(25)37-26(41)20-4-3-19(29)11-22(20)28(31,32)33/h3-4,11-15,17,34H,5-10,16H2,1-2H3,(H,37,41)/t17-/m0/s1	DQNBTQRQDJILHR-KRWDZBQOSA-N	553327	4-fluoro-N-[4-fluoro-5-(2- piperazin-1-ylpyrimidin-5- yl)-2-[rac-(3R)-3,4- dimethylpiperazin-1- yl]phenyl]-2-(trifluoromethyl) benzamide::US11319299, Example 401	WD repeat-containing protein 5				 1.11						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553327	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553327&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138551593	469797193							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167088	C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1ccc(F)cc1C(F)(F)F)-c1ccc(nc1)N1CCOCC1	InChI=1S/C29H30F5N5O2/c1-18-17-39(8-7-37(18)2)26-15-24(31)22(19-3-6-27(35-16-19)38-9-11-41-12-10-38)14-25(26)36-28(40)21-5-4-20(30)13-23(21)29(32,33)34/h3-6,13-16,18H,7-12,17H2,1-2H3,(H,36,40)/t18-/m0/s1	ZGXSENXXYHGSLU-SFHVURJKSA-N	553328	4-fluoro-N-[4-fluoro-5-(6- morpholin-4-ylpyridin-3- yl)-2-[rac-(3R)-3,4- dimethylpiperazin-1- yl]phenyl]-2-(trifluoromethyl) benzamide::US11319299, Example 402	WD repeat-containing protein 5				 3.70						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553328	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553328&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138551359	469797194							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167089	C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(OC2CCOCC2)nc1			553329	4-(difluoromethyl)-N-[4- fluoro-5-[6-(oxan-4- yloxy)pyridin-3-yl]-2- [rac-(3R)-3,4- dimethylpiperazin-1- yl]phenyl]-6-oxo-1H- pyridine-3-carboxamide::US11319299, Example 403	WD repeat-containing protein 5				 1.16						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553329	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553329&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608056	469797195							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167090	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCN(CC1)c1ncc(cn1)C#N			553330	N-[5-[1-(5-cyanopyrimidin- 2-yl)-3,6-dihydro-2H- pyridin-4-yl]-4-fluoro-2- [rac-(3R,5S)-3,4,5- trimethylpiperazin- 1-yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 404	WD repeat-containing protein 5				 1.000						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553330	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553330&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608057	469797196							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167091	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCN(CC1)c1ncc(CN(C)C)cn1			553331	N-[5-[1-[5-[(dimethylamino) methyl]pyrimidin-2-yl]-3,6- dihydro-2H-pyridin-4-yl]- 4-fluoro-2-[rac-(3R,5S)- 3,4,5-trimethylpiperazin- 1-yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 405	WD repeat-containing protein 5				 0.095						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553331	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553331&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608058	469797197							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167092	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCN(CC1)c1ncc(CN2CCOCC2)cn1			553332	N-[4-fIuoro-5-[1-[5- (morpholin-4-ylmethyl) pyrimidin-2-yl]-3,6-dihydro-2H- pyridin-4-yl]-2-[rac-(3R,5S)- 3,4,5-trimethylpiperazin- 1-yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 406	WD repeat-containing protein 5				 0.457						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553332	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553332&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608059	469797198							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167093	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCN(CC1)c1ncc(CN2CCN(C)CC2)cn1			553333	N-[4-fluoro-5-[1-[5-[(4- methylpiperazin-1-yl)methyl] pyrimidin-2-yl]-3,6-dihydro- 2H-pyridin-4-yl]-2-[rac- (3R,5S)-3,4,5- trimethylpiperazin-1-yl]phenyl]- 6-oxo-4-(trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 407	WD repeat-containing protein 5				 0.231						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553333	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553333&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608060	469797199							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167094	CC(C)COC(=O)N1CCC=C(C1)c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)(F)F)c(cc1F)N1C[C@H](C)N(C)[C@H](C)C1			553334	2-methylpropyl 5-[2-fluoro- 5-[[6-oxo-4-(trifluoromethyl)- 1H-pyridine-3-carbonyl]amino]- 4-[rac-(3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-3,6-dihydro- 2H-pyridine-1-carboxylate::US11319299, Example 408	WD repeat-containing protein 5				 2.75						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553334	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553334&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608061	469797200							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167095	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCCN(C1)c1ncc(C=O)cn1			553335	N-[4-fluoro-5-[1-(5- formylpyrimidin-2-yl)-3,6- dihydro-2H-pyridin-5-yl]-2- [rac-(3R,5S)-3,4,5- trimethylpiperazin- 1-yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 409	WD repeat-containing protein 5				 0.229						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553335	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553335&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608062	469797201							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167096	C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)F)-c1cnc(nc1)N1CCOCC1			553336	4-(difluoromethyl)-N-[4- fluoro-5-(2-morpholin-4- ylpyrimidin-5-yl)-2-[rac- (3R)-3,4-dimethylpiperazin- 1-yl]phenyl]-6-oxo-1H- pyridine-3-carboxamide::US11319299, Example 410	WD repeat-containing protein 5				 0.840						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553336	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553336&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608063	469797202							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167097	C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)F)-c1ccc(OCC2CC2)nc1			553337	N-[5-[6-(cyclopropylmethoxy) pyridin-3-yl]-4-fluoro-2-[rac- (3R)-3,4-dimethylpiperazin-1- yl]phenyl]-4-(difhioromethyl)-6- oxo-1H-pyridine-3-carboxamide::US11319299, Example 411	WD repeat-containing protein 5				 2.29						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553337	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553337&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608064	469797203							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167098	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)F)-c1ccc(nc1)N1CCOCC1			553338	4-(difluoromethyl)-N-[4-fluoro- 5-(6-morpholin-4-ylpyridin-3- yl)-2-[rac-(3R,5S)-3,4,5- trimethylpiperazin-1-yl] phenyl]-6-oxo-1H-pyridine-3- carboxamide::US11319299, Example 412	WD repeat-containing protein 5				 0.962						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553338	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553338&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608065	469797204							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167099	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCCN(C1)c1ncc(CO)cn1			553339	N-[4-fluoro-5-[1-[5- (hydroxymethyl)pyrimidin-2-yl]- 3,6-dihydro-2H-pyridin-5-yl]-2- [rac-(3R,5S)-3,4,5- trimethylpiperazin-1-yl)phenyl]- 6-oxo-4-(trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 413	WD repeat-containing protein 5				 0.302						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553339	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553339&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608066	469797205							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167100	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCCN(C1)c1ncc(CN(C)C)cn1			553340	N-[5-[1-[5-[(dimethylamino) methyl]pyrimidin-2-yl]-3,6- dihydro-2H-pyridin-5-yl]- 4-fluoro-2-[rac-(3R,5S)- 3,4,5-trimethylpiperazin- 1-yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 414	WD repeat-containing protein 5				 0.658						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553340	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553340&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608067	469797206							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167101	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCCN(C1)c1ncc(CN2CCOCC2)cn1			553341	N-[4-fluoro-5-[1-[5- (morpholin-4-ylmethyl) pyrimidin-2-yl]-3,6-dihydro- 2H-pyridin-5-yl]-2-[rac-(3R,5S)- 3,4,5-trimethylpiperazin- 1-yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 415	WD repeat-containing protein 5				 1.10						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553341	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553341&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608068	469797207							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167102	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCCN(C1)c1ncc(CN2CCN(C)CC2)cn1			553342	N-[4-fluoro-5-[1-[5-[(4- methylpiperazin-1- yl)methyl]pyrimidin-2- yl]-3,6-dihydro-2H- pyridin-5-yl]-2-[rac- (3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 416	WD repeat-containing protein 5				 0.108						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553342	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553342&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608069	469797208							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167103	C[C@H]1CN(C[C@@H](C)O1)c1ncc(cn1)-c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)(F)F)c(cc1F)N1CC[C@H](C1)N(C)C			553343	N-[4-fluoro-2-[rac-(3S)- 3-(dimethylamino)pyrrolidin-1- yl]-5-[2-[rac-(2R,6S)- 2,6-dimethylmorpholin-4- yl]pyrimidin-5-yl]phenyl]-6-oxo- 4-(trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 417	WD repeat-containing protein 5				 1.41						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553343	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553343&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608070	469797209							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167104	CCN(C)[C@@H]1CCN(C1)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cnc(nc1)N1C[C@H](C)O[C@H](C)C1			553344	N-[4-fluoro-5-[2-[rac- (2R,6S)-2,6-dimethylmorpholin- 4-yl]pyrimidin-5-yl]-2-[rac- (3S)-3-[ethyl(methyl)amino] pyrrolidin-1-yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H-pyridine-3- carboxamide::US11319299, Example 418	WD repeat-containing protein 5				 1.05						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553344	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553344&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608071	469797210							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167105	CCN(CC)[C@@H]1CCN(C1)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cnc(nc1)N1CCOCC1			553345	N-[4-fluoro-5-(2- morpholin-4-ylpyrimidin- 5-yl)-2-[rac-(3R)-3-(diethylamino) pyrrolidin-1-yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 419	WD repeat-containing protein 5				 5.37						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553345	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553345&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608072	469797211							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167106	CC(C)N(C)[C@@H]1CCN(C1)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cnc(nc1)N1CCOCC1			553346	N-[4-fluoro-5-(2-morpholin-4- ylpyrimidin-5-yl)-2-[rac-(3R)-3- [methyl(propan-2-yl)amino] pyrrolidin-1-yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H-pyridine-3- carboxamide::US11319299, Example 420	WD repeat-containing protein 5				 172						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553346	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553346&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608073	469797212							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167107	C[C@H]1CN(C[C@@H](C)O1)c1ccc(cn1)-c1cc(NC(=O)c2cn(C)c(=O)cc2C(F)(F)F)c(cc1F)N1CCN(C)[C@@H](C)C1	InChI=1S/C31H36F4N6O3/c1-18-14-40(9-8-38(18)4)27-12-25(32)22(21-6-7-28(36-13-21)41-15-19(2)44-20(3)16-41)10-26(27)37-30(43)23-17-39(5)29(42)11-24(23)31(33,34)35/h6-7,10-13,17-20H,8-9,14-16H2,1-5H3,(H,37,43)/t18-,19-,20+/m0/s1	FPUHELKSPQHCAR-SLFFLAALSA-N	553347	N-[4-fluoro-5-[6-[rac-(2R,6S)-2,6- dimethylmorpholin-4-yl]pyridin- 3-yl]-2-[rac-(3R)-3,4- dimethylpiperazin-1-yl]phenyl]-1- methyl-6-oxo-4-(trifluoromethyl) pyridine-3-carboxamide::US11319299, Example 421	WD repeat-containing protein 5				 1.96						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553347	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553347&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138551463	469797213							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167108	C[C@H]1CN(C[C@@H](C)O1)c1ccc(cn1)-c1cc(NC(=O)c2cn(C)c(=O)cc2C(F)(F)F)c(cc1F)N1C[C@H](C)N(C)[C@H](C)C1	InChI=1S/C32H38F4N6O3/c1-18-13-41(14-19(2)40(18)6)28-11-26(33)23(22-7-8-29(37-12-22)42-15-20(3)45-21(4)16-42)9-27(28)38-31(44)24-17-39(5)30(43)10-25(24)32(34,35)36/h7-12,17-21H,13-16H2,1-6H3,(H,38,44)/t18-,19+,20-,21+	UNHOCOGRITXWKY-FXELSEDVSA-N	553348	N-(4-fluoro-5-[6-[rac-(2R,6S)- 2,6-dimethylmorpholin-4- yl]pyridin-3-yl]-2-[rac- (3S,5R)-3,4,5- trimethylpiperazin-1- yl]phenyl]-1-methyl-6-oxo- 4-(trifluoromethyl)pyridine-3- carboxamide::US11319299, Example 422	WD repeat-containing protein 5				 2.43						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553348	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553348&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			137377626	469797214							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167109	C[C@H]1CN(C[C@@H](C)O1)c1ccc(cn1)-c1cc(NC(=O)c2ccc(F)cc2C(F)(F)F)c(cc1F)N1CCN(C)[C@@H](C)C1	InChI=1S/C31H34F5N5O2/c1-18-15-40(10-9-39(18)4)28-13-26(33)24(21-5-8-29(37-14-21)41-16-19(2)43-20(3)17-41)12-27(28)38-30(42)23-7-6-22(32)11-25(23)31(34,35)36/h5-8,11-14,18-20H,9-10,15-17H2,1-4H3,(H,38,42)/t18-,19-,20+/m0/s1	UFGCOUPQDHMESY-SLFFLAALSA-N	553349	4-fluoro-N-[4-fluoro-5-[6-[rac- (2R,6S)-2,6-dimethylmorpholin-4- yl]pyridin-3-yl]-2-[rac-(3R)-3,4- dimethylpiperazin-1-yl]phenyl]-2- (trifluoromethyl)benzamide::US11319299, Example 423::US11319299, Example 432	WD repeat-containing protein 5				 1.93						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553349	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553349&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138551408	469797215							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167110	C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cnc(nc1)N1CCC(C)(O)CC1			553350	N-[4-fluoro-5-[2-(4-hydroxy-4- methylpiperidin-1-yl)pyrimidin- 5-yl]-2-[rac-(3R)-3,4- dimethylpiperazin-1-yl]phenyl]- 6-oxo-4-(trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 424	WD repeat-containing protein 5				 0.609						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553350	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553350&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608074	469797216							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167111	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cnc(nc1)N1CCC(C)(O)CC1			553351	N-[4-fluoro-5-[2-(4-hydroxy-4- methylpiperidin-1-yl)pyrimidin- 5-yl]-2-[rac-(3R,5S)-3,4,5- trimethylpiperazin-1-yl]phenyl]- 6-oxo-4-(trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 425	WD repeat-containing protein 5				 1.06						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553351	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553351&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608075	469797217							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167112	C[C@H]1CN(C[C@@H](C)O1)c1ncc(cn1)-c1cc(NC(=O)c2cn(C)c(=O)cc2C(F)(F)F)c(cc1F)N1CC[C@H](C1)N(C)C	InChI=1S/C30H35F4N7O3/c1-17-13-41(14-18(2)44-17)29-35-11-19(12-36-29)21-8-25(26(10-24(21)31)40-7-6-20(15-40)38(3)4)37-28(43)22-16-39(5)27(42)9-23(22)30(32,33)34/h8-12,16-18,20H,6-7,13-15H2,1-5H3,(H,37,43)/t17-,18+,20-/m1/s1	IYBGGAZGPWXFKR-WSTZPKSXSA-N	553352	N-[4-fluoro-2-[rac-(3S)-3- (dimethylamino)pyrrolidin-1- yl]-5-[2-[rac-(2R,6S)- 2,6-dimethylmorpholin-4- yl]pyrimidin-5-yl]phenyl]-1- methyl-6-oxo-4-(trifluoromethyl) pyridine-3-carboxamide::US11319299, Example 426	WD repeat-containing protein 5				 10.9						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553352	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553352&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138551490	469797218							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167113	CCN(C)[C@@H]1CCN(C1)c1cc(F)c(cc1NC(=O)c1cn(C)c(=O)cc1C(F)(F)F)-c1cnc(nc1)N1C[C@H](C)O[C@H](C)C1	InChI=1S/C31H37F4N7O3/c1-6-39(4)21-7-8-41(16-21)27-11-25(32)22(20-12-36-30(37-13-20)42-14-18(2)45-19(3)15-42)9-26(27)38-29(44)23-17-40(5)28(43)10-24(23)31(33,34)35/h9-13,17-19,21H,6-8,14-16H2,1-5H3,(H,38,44)/t18-,19+,21-/m1/s1	VCDKNSAHIQDQGN-SVFBPWRDSA-N	553353	N-[4-fluoro-5-[2-[rac-(2R,6S)-2,6- dimethylmorpholin-4- yl]pyrimidin-5-yl]-2-[rac- (3S)-3-[ethyl(methyl)amino] pyrrolidin-1-yl]phenyl]-1- methyl-6-oxo-4-(trifluoromethyl) pyridine-3-carboxamide::US11319299, Example 427	WD repeat-containing protein 5				 5.59						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553353	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553353&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138551470	469797219							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167114	CCN(CC)[C@@H]1CCN(C1)c1cc(F)c(cc1NC(=O)c1cn(C)c(=O)cc1C(F)(F)F)-c1cnc(nc1)N1CCOCC1	InChI=1S/C30H35F4N7O3/c1-4-39(5-2)20-6-7-41(17-20)26-14-24(31)21(19-15-35-29(36-16-19)40-8-10-44-11-9-40)12-25(26)37-28(43)22-18-38(3)27(42)13-23(22)30(32,33)34/h12-16,18,20H,4-11,17H2,1-3H3,(H,37,43)/t20-/m1/s1	CTAZSSJAKLEXTN-HXUWFJFHSA-N	553354	N-[4-fluoro-5-(2-morpholin- ylpyrimidin-5-yl)-2-[rac-(3R)-3- (diethylamino)pyrrolidin-1-yl] phenyl]-1-methyl-6-oxo-4- (trifluoromethyl)pyridine- 3-carboxamide::US11319299, Example 428	WD repeat-containing protein 5				 145						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553354	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553354&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			137377000	469797220							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167115	C[C@H]1CN(C[C@@H](C)O1)c1ncc(cn1)-c1cc(NC(=O)c2ccc(F)cc2C(F)(F)F)c(cc1F)N1CCN(C)[C@@H](C)C1	InChI=1S/C30H33F5N6O2/c1-17-14-40(8-7-39(17)4)27-11-25(32)23(20-12-36-29(37-13-20)41-15-18(2)43-19(3)16-41)10-26(27)38-28(42)22-6-5-21(31)9-24(22)30(33,34)35/h5-6,9-13,17-19H,7-8,14-16H2,1-4H3,(H,38,42)/t17-,18-,19+/m0/s1	JNEFXRAXVQTGTB-GBESFXJTSA-N	553355	4-fluoro-N-[4-fluoro-5-[2-[rac- (2R,6S)-2,6-dimethylmorpholin- 4-yl]pyrimidin-5-yl]-2-[rac- (3R)-3,4-dimethylpiperazin-1- yl]phenyl]-2-(trifluoromethyl) benzamide::US11319299, Example 430	WD repeat-containing protein 5				 0.296						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553355	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553355&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138551337	469797221							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167116	C[C@H]1CN(C[C@@H](C)O1)c1ncc(cn1)-c1cc(NC(=O)c2ccc(F)cc2C(F)(F)F)c(cc1F)N1C[C@H](C)N(C)[C@H](C)C1	InChI=1S/C31H35F5N6O2/c1-17-13-41(14-18(2)40(17)5)28-10-26(33)24(21-11-37-30(38-12-21)42-15-19(3)44-20(4)16-42)9-27(28)39-29(43)23-7-6-22(32)8-25(23)31(34,35)36/h6-12,17-20H,13-16H2,1-5H3,(H,39,43)/t17-,18+,19-,20+	JSSGHMCWUFZLLD-FGYAAKKASA-N	553356	4-fluoro-N-[4-fluoro-5- [2-[rac-(2R,6S)-2,6- dimethylmorpholin-4- yl]pyrimidin-5-yl]-2-[rac- (3S,5R)-3,4,5-trimethylpiperazin- 1-yl]phenyl]-2-(trifluoromethyl) benzamide::US11319299, Example 431	WD repeat-containing protein 5				 0.649						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553356	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553356&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138541973	469797222							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167117	C[C@H]1CN(C[C@@H](C)O1)c1ccc(cn1)-c1cc(NC(=O)c2ccc(F)cc2C(F)(F)F)c(cc1F)N1CCN(C)[C@@H](C)C1	InChI=1S/C31H34F5N5O2/c1-18-15-40(10-9-39(18)4)28-13-26(33)24(21-5-8-29(37-14-21)41-16-19(2)43-20(3)17-41)12-27(28)38-30(42)23-7-6-22(32)11-25(23)31(34,35)36/h5-8,11-14,18-20H,9-10,15-17H2,1-4H3,(H,38,42)/t18-,19-,20+/m0/s1	UFGCOUPQDHMESY-SLFFLAALSA-N	553349	4-fluoro-N-[4-fluoro-5-[6-[rac- (2R,6S)-2,6-dimethylmorpholin-4- yl]pyridin-3-yl]-2-[rac-(3R)-3,4- dimethylpiperazin-1-yl]phenyl]-2- (trifluoromethyl)benzamide::US11319299, Example 423::US11319299, Example 432	WD repeat-containing protein 5				 2.31						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553349	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553349&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138551408	469797215							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167118	C[C@H]1CN(CCO1)c1ccc(cn1)-c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)(F)F)c(cc1F)N1CCN(C)[C@@H](C)C1			553358	N-[4-fluoro-2-[rac-(3R)-3,4- dimethylpiperazin-1-yl]-5-[6- [rac-(2R)-2-methylmorpholin-4- yl]pyridin-3-yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H-pyridine-3- carboxamide::US11319299, Example 433	WD repeat-containing protein 5				 2.84						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553358	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553358&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608076	469797223							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167119	C[C@H]1CN(CCO1)c1ccc(cn1)-c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)(F)F)c(cc1F)N1C[C@H](C)N(C)[C@H](C)C1			553359	N-[4-fluoro-5-[6-[rac-(2R)-2- methylmorpholin-4-yl]pyndin-3- yl]-2-[rac-(3S,5R)-3,4,5- trimethylpiperazin-1-yl]phenyl]- 6-oxo-4-(trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 434	WD repeat-containing protein 5				 0.617						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553359	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553359&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608077	469797224							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167120	C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1ccc(F)cc1C(F)(F)F)-c1cnc(nc1)N1CCN(CC1)C1CC1	InChI=1S/C31H34F5N7O/c1-19-18-43(8-7-40(19)2)28-15-26(33)24(14-27(28)39-29(44)23-6-3-21(32)13-25(23)31(34,35)36)20-16-37-30(38-17-20)42-11-9-41(10-12-42)22-4-5-22/h3,6,13-17,19,22H,4-5,7-12,18H2,1-2H3,(H,39,44)/t19-/m0/s1	JAYSDHKFQZMPHP-IBGZPJMESA-N	553360	N-[5-[2-(4-cyclopropylpiperazin- 1-yl)pyrimidin-5-yl]-4-fluoro-2- [rac-(3R)-3,4-dimethylpiperazin- 1-yl]phenyl]-4-fluoro-2- (trifluoromethyl)benzamide::US11319299, Example 435	WD repeat-containing protein 5				 1.47						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553360	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553360&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138551419	469797225							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167121	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)F)-c1ccc(N2CCOCC2)c(F)c1			553361	4-(difluoromethyl)-N-[4-fluoro- 5-(3-fluoro-4-morpholin-4- ylphenyl)-2-[rac-(3R,5S)-3,4,5- trimethylpiperazin-1-yl]phenyl]- 6-oxo-1H-pyridine-3- carboxamide::US11319299, Example 436	WD repeat-containing protein 5				 1.39						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553361	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553361&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608078	469797226							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167122	COc1cnc(nc1)N1CC=C(C1)c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)(F)F)c(cc1F)N1C[C@H](C)N(C)[C@H](C)C1			553362	N-[4-fluoro-5-[1-(5- methoxypyrimidin- 2-yl)-2,5-dihydropyrrol-3-yl]- 2-[rac-(3R,5S)-3,4,5- trimethylpiperazin-1-yl] phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 437	WD repeat-containing protein 5				 0.721						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553362	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553362&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608079	469797227							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167123	COc1cc(ncn1)N1CC=C(C1)c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)(F)F)c(cc1F)N1C[C@H](C)N(C)[C@H](C)C1			553363	N-[4-fluoro-5-[1-(6- methoxypyrimidin-4-yl)- 2,5-dihydropyrrol-3-yl]-2-[rac- (3R,5S)-3,4,5- trimethylpiperazin- 1-yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 438	WD repeat-containing protein 5				 1.99						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553363	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553363&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608080	469797228							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167124	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCN(C1)c1ncc(C)cn1			553364	N-[4-fluoro-5-[1-(5- methylpyrimidin-2-yl)- 2,5-dihydropyrrol-3-yl]- 2-[rac-(3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 439	WD repeat-containing protein 5				 2.45						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553364	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553364&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608081	469797229							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167125	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCN(C1)c1ncc(F)cn1			553365	N-[4-fluoro-5-[1-(5- fluoropyrimidin-2-yl)- 2,5-dihydropyrrol-3-yl]- 2-[rac-(3R,5S)-3,4,5- trimethylpiperazin-1- yl)phenyl]-6-oxo-4- (trifluoromethyl)-1H-pyridine- 3-carboxamide::US11319299, Example 440	WD repeat-containing protein 5				 2.88						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553365	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553365&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608082	469797230							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167126	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCN(C1)C(=O)N1CCCC1			553366	N-[4-fluoro-5-[1- (pyrrolidine-1-carbonyl)- 2,5-dihydropyrrol-3-yl]- 2-[rac-(3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 441	WD repeat-containing protein 5				 1.91						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553366	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553366&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608083	469797231							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167127	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCN(C1)C(=O)c1cnccn1			553367	N-[4-fluoro-5-[1-(pyrazine-2- carbonyl)-2,5-dihydropyrrol-3- yl]-2-[rac-(3R,5S)-3,4,5- trimethylpiperazin-1- yl)phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 442	WD repeat-containing protein 5				 3.67						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553367	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553367&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608084	469797232							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167128	CC(C)COC(=O)N1CC=C(C1)c1cc(NC(=O)c2c[nH]c(=O)cc2C(F)(F)F)c(cc1F)N1C[C@H](C)N(C)[C@H](C)C1			553368	2-methylpropyl 3-[2- fluoro-5-[[6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carbonyl]amino]-4- [rac-(3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-2,5- dihydropyrrole-1-carboxylate::US11319299, Example 443	WD repeat-containing protein 5				 2.37						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553368	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553368&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608085	469797233							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167129	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCN(C1)c1ncc(C=O)cn1			553369	N-[4-fluoro-5-[1-(5- formylpyrimidin-2-yl)- 2,5-dihydropyrrol-3-yl]- 2-[rac-(3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 444	WD repeat-containing protein 5				 2.96						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553369	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553369&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608086	469797234							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167130	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CN(C)[S]=C1			553370	N-[4-fluoro-5-(1- methylpyrazol-4-yl)-2- [rac-(3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 445	WD repeat-containing protein 5				 1.95						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553370	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553370&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164885349	469797235							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167131	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1nc(cs1)C#N			553371	N-[5-(4-cyano-1,3- thiazol-2-yl)-4-fluoro-2- [rac-(3R,5S)-3,4,5- trimethylpiperazin-1- yl)phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 446	WD repeat-containing protein 5				 2.94						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553371	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553371&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608087	469797236							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167132	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ncc(s1)C#N			553372	N-[5-(5-cyano-1,3- thiazol-2-yl)-4-fluoro-2- [rac-(3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 447	WD repeat-containing protein 5				 2.88						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553372	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553372&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608088	469797237							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167133	C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)F)-c1ccc(N2CCOCC2)c(F)c1			553373	4-(difluoromethyl)-N-[4- fluoro-5-(3-fluoro-4- morpholin-4-ylphenyl)-2- [rac-(3R)-3,4- dimethylpiperazin- 1-yl]phenyl]-6-oxo-1H- pyridine-3-carboxamide::US11319299, Example 448	WD repeat-containing protein 5				 1.01						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553373	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553373&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608089	469797238							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167134	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1cn(C)c(=O)cc1C(F)F)-c1ccc(N2CCOCC2)c(F)c1	InChI=1S/C31H35F4N5O3/c1-18-15-40(16-19(2)38(18)4)28-14-24(32)21(20-5-6-27(25(33)11-20)39-7-9-43-10-8-39)12-26(28)36-31(42)23-17-37(3)29(41)13-22(23)30(34)35/h5-6,11-14,17-19,30H,7-10,15-16H2,1-4H3,(H,36,42)/t18-,19+	IIVBFEPYECYNRM-KDURUIRLSA-N	553374	4-(difluoromethyl)-N-[4- fluoro-5-(3-fluoro-4- morpholin-4-ylphenyl)-2- [rac-(3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-1-methyl-6- oxopyridine-3-carboxamide::US11319299, Example 449	WD repeat-containing protein 5				 9.03						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553374	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553374&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			137377124	469797239							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167135	C[C@H]1CN(CCO1)c1ncc(cn1)-c1cc(NC(=O)c2cn(C)c(=O)cc2C(F)(F)F)c(cc1F)N1CCN(C)[C@@H](C)C1	InChI=1S/C29H33F4N7O3/c1-17-14-39(6-5-37(17)3)25-11-23(30)20(19-12-34-28(35-13-19)40-7-8-43-18(2)15-40)9-24(25)36-27(42)21-16-38(4)26(41)10-22(21)29(31,32)33/h9-13,16-18H,5-8,14-15H2,1-4H3,(H,36,42)/t17-,18-/m0/s1	UQOLIVLMQOQTBL-ROUUACIJSA-N	553375	N-[4-fluoro-2-[rac-(3R)- 3,4-dimethylpiperazin-1- yl]-5-[2-[rac-(2R)-2- methylmorpholin-4- yl]pyrimidin-5-yl]phenyl]- 1-methyl-6-oxo-4- (trifluoromethyl)pyridine- 3-carboxamide::US11319299, Example 450	WD repeat-containing protein 5				 1.02						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553375	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553375&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138551493	469797240							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167136	C[C@H]1CN(CCO1)c1ncc(cn1)-c1cc(NC(=O)c2cn(C)c(=O)cc2C(F)(F)F)c(cc1F)N1C[C@H](C)N(C)[C@H](C)C1	InChI=1S/C30H35F4N7O3/c1-17-13-41(14-18(2)39(17)5)26-10-24(31)21(20-11-35-29(36-12-20)40-6-7-44-19(3)15-40)8-25(26)37-28(43)22-16-38(4)27(42)9-23(22)30(32,33)34/h8-12,16-19H,6-7,13-15H2,1-5H3,(H,37,43)/t17-,18+,19-/m0/s1	LGIULJQHFBTTOT-OTWHNJEPSA-N	553376	N-[4-fluoro-5-[2-[rac- (2R)-2-methylmorpholin- 4-yl]pyrimidin-5-yl]-2- [rac-(3S,5R)-3,4,5- trimethylpiperazin-1- yl]phenyl]-1-methyl-6- oxo-4-(trifluoromethyl) pyridine-3-carboxamide::US11319299, Example 451	WD repeat-containing protein 5				 1.72						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553376	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553376&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138551338	469797241							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167137	C[C@H]1CN(CCO1)c1ncc(cn1)-c1cc(NC(=O)c2ccc(F)cc2C(F)(F)F)c(cc1F)N1CCN(C)[C@@H](C)C1	InChI=1S/C29H31F5N6O2/c1-17-15-39(7-6-38(17)3)26-12-24(31)22(19-13-35-28(36-14-19)40-8-9-42-18(2)16-40)11-25(26)37-27(41)21-5-4-20(30)10-23(21)29(32,33)34/h4-5,10-14,17-18H,6-9,15-16H2,1-3H3,(H,37,41)/t17-,18-/m0/s1	ICWHVNWEWUCKRA-ROUUACIJSA-N	553377	4-fluoro-N-[4-fluoro-2- [rac-(3R)-3,4- dimethylpiperazin- 1-yl]-5-[2-[rac-(2R)-2- methylmorpholin-4- yl]pyrimidin-5-yl]phenyl]- 2-(trifluoromethyl)benzamide::US11319299, Example 452	WD repeat-containing protein 5				 0.493						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553377	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553377&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138551336	469797242							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167138	C[C@H]1CN(CCO1)c1ncc(cn1)-c1cc(NC(=O)c2ccc(F)cc2C(F)(F)F)c(cc1F)N1C[C@H](C)N(C)[C@H](C)C1	InChI=1S/C30H33F5N6O2/c1-17-14-41(15-18(2)39(17)4)27-11-25(32)23(20-12-36-29(37-13-20)40-7-8-43-19(3)16-40)10-26(27)38-28(42)22-6-5-21(31)9-24(22)30(33,34)35/h5-6,9-13,17-19H,7-8,14-16H2,1-4H3,(H,38,42)/t17-,18+,19-/m0/s1	YHRUDJMQAFXZEQ-OTWHNJEPSA-N	553378	4-fluoro-N-[4-fluoro-5- [2-[rac-(2R)-2- methylmorpholin-4- yl]pyrimidin-5-yl]-2-[rac- (3S,5R)-3,4,5- trimethylpiperazin- 1-yl]phenyl]-2- (trifluoromethyl)benzamide::US11319299, Example 453	WD repeat-containing protein 5				 0.822						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553378	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553378&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138551579	469797243							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167139	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1ccc(F)cc1C(F)(F)F)-c1cnc(nc1)N1CCN(CC1)C1CC1	InChI=1S/C32H36F5N7O/c1-19-17-44(18-20(2)41(19)3)29-14-27(34)25(13-28(29)40-30(45)24-7-4-22(33)12-26(24)32(35,36)37)21-15-38-31(39-16-21)43-10-8-42(9-11-43)23-5-6-23/h4,7,12-16,19-20,23H,5-6,8-11,17-18H2,1-3H3,(H,40,45)/t19-,20+	COTJDORAMZYNMT-BGYRXZFFSA-N	553379	N-[5-[2-(4- cyclopropylpiperazin- 1-yl)pyrimidin-5-yl]-4- fluoro-2-[rac-(3R,5S)- 3,4,5-trimethylpiperazin-1- yl]phenyl]-4-fluoro-2- (trifluoromethyl)benzamide::US11319299, Example 454	WD repeat-containing protein 5				 4.05						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553379	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553379&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			137376839	469797244							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167140	C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1cn(C)c(=O)cc1C(F)(F)F)-c1cnc(nc1)N1CCN(CC1)C1CC1	InChI=1S/C31H36F4N8O2/c1-19-17-43(7-6-39(19)2)27-14-25(32)22(20-15-36-30(37-16-20)42-10-8-41(9-11-42)21-4-5-21)12-26(27)38-29(45)23-18-40(3)28(44)13-24(23)31(33,34)35/h12-16,18-19,21H,4-11,17H2,1-3H3,(H,38,45)/t19-/m0/s1	LBKYZVYBTXXVCT-IBGZPJMESA-N	553380	N-[5-[2-(4- cyclopropylpiperazin- 1-yl)pyrimidin-5-yl]-4- fluoro-2-[rac-(3R)-3,4- dimethylpiperazin-1- yl]phenyl]-1-methyl-6- oxo-4-(trifluoromethyl) pyridine-3-carboxamide::US11319299, Example 455	WD repeat-containing protein 5				 1.98						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553380	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553380&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			138551423	469797245							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167141	C[C@@H]1CN(CCO1)c1ncc(cn1)-c1cc(NC(=O)c2ccc(F)cc2C(F)(F)F)c(cc1F)N1CCN(C)[C@@H](C)C1	InChI=1S/C29H31F5N6O2/c1-17-15-39(7-6-38(17)3)26-12-24(31)22(19-13-35-28(36-14-19)40-8-9-42-18(2)16-40)11-25(26)37-27(41)21-5-4-20(30)10-23(21)29(32,33)34/h4-5,10-14,17-18H,6-9,15-16H2,1-3H3,(H,37,41)/t17-,18+/m0/s1	ICWHVNWEWUCKRA-ZWKOTPCHSA-N	553381	4-fluoro-N-[4-fluoro-2- [rac-(3S)-3,4- dimethylpiperazin- 1-yl]-5-[2-[rac-(2R)-2- methylmorpholin-4- yl]pyrimidin-5-yl]phenyl]- 2-(trifluoromethyl)benzamide::US11319299, Example 456	WD repeat-containing protein 5				 1.08						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553381	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553381&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			137376763	469797246							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
1167142	C[C@H]1CN(C[C@@H](C)N1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)C1=CCN(C1)c1ncc(CN(C)C)cn1			553382	N-[5-[1-[5- [(dimethylamino)methyl] pyrimidin-2-yl]-2,5- dihydropyrrol-3-yl]-4- fluoro-2-[rac-(3R,5S)- 3,4,5-trimethylpiperazin- 1-yl]phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 457	WD repeat-containing protein 5				 2.57						US Patent		10.7270/Q27W6GD6		aid1806515	US11319299	Al-Awar, R; Zepeda-Velazquez, CA; Poda, G; Isaac, M; Uehling, D; Wilson, B; Joseph, B; Liu, Y; Subramanian, P; Mamai, A; Prakesch, M; Stille, JK	Propellon Therapeutics Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=553382	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=553382&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164608090	469797247							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51422338	CN1CCN(CC1)c1ccc(cc1NC(=O)c1cc(N)c(F)c(C)c1Cl)C#CCNC(=O)C1CCOCC1	InChI=1S/C28H33ClFN5O3/c1-18-25(29)21(17-22(31)26(18)30)28(37)33-23-16-19(5-6-24(23)35-12-10-34(2)11-13-35)4-3-9-32-27(36)20-7-14-38-15-8-20/h5-6,16-17,20H,7-15,31H2,1-2H3,(H,32,36)(H,33,37)	DQKAXADDLDHJAJ-UHFFFAOYSA-N	50574657	CHEMBL4857312	WD repeat-containing protein 5			 95							ChEMBL	10.1016/j.ejmech.2021.113677	10.7270/Q2J38XCR	34225179			Chen, W; Chen, X; Li, D; Wang, X; Long, G; Jiang, Z; You, Q; Guo, X	China Pharmaceutical University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50574657	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50574657&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164616338	471064802							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51422339	CN1CCN(CC1)c1ccc(cc1NC(=O)c1cc(N)c(F)c(C)c1Cl)C#CCN	InChI=1S/C22H25ClFN5O/c1-14-20(23)16(13-17(26)21(14)24)22(30)27-18-12-15(4-3-7-25)5-6-19(18)29-10-8-28(2)9-11-29/h5-6,12-13H,7-11,25-26H2,1-2H3,(H,27,30)	WNDVATIEYUOHIZ-UHFFFAOYSA-N	50574658	CHEMBL4853161	WD repeat-containing protein 5			 444							ChEMBL	10.1016/j.ejmech.2021.113677	10.7270/Q2J38XCR	34225179			Chen, W; Chen, X; Li, D; Wang, X; Long, G; Jiang, Z; You, Q; Guo, X	China Pharmaceutical University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50574658	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50574658&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164612895	471064803							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51422340	CN1CCN(CC1)c1ccc(cc1NC(=O)c1cc(N)c(F)c(C)c1Cl)-c1ccc(NC(=O)CCCN)cc1	InChI=1S/C29H34ClFN6O2/c1-18-27(30)22(17-23(33)28(18)31)29(39)35-24-16-20(7-10-25(24)37-14-12-36(2)13-15-37)19-5-8-21(9-6-19)34-26(38)4-3-11-32/h5-10,16-17H,3-4,11-15,32-33H2,1-2H3,(H,34,38)(H,35,39)	PVXYYWORFYROCX-UHFFFAOYSA-N	50208354	CHEMBL3884329	WD repeat-containing protein 5			 7.6							ChEMBL	10.1016/j.ejmech.2021.113677	10.7270/Q2J38XCR	34225179			Chen, W; Chen, X; Li, D; Wang, X; Long, G; Jiang, Z; You, Q; Guo, X	China Pharmaceutical University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50208354	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50208354&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			134130757	375982008		CHEMBL3884329					1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51422341	CN1CCC(CC1)C(=O)NCC#Cc1ccc(N2CCN(C)CC2)c(NC(=O)c2cc(N)c(F)c(C)c2Cl)c1	InChI=1S/C29H36ClFN6O2/c1-19-26(30)22(18-23(32)27(19)31)29(39)34-24-17-20(6-7-25(24)37-15-13-36(3)14-16-37)5-4-10-33-28(38)21-8-11-35(2)12-9-21/h6-7,17-18,21H,8-16,32H2,1-3H3,(H,33,38)(H,34,39)	GKKMASWBFXJDID-UHFFFAOYSA-N	50574659	CHEMBL4847340	WD repeat-containing protein 5			 94							ChEMBL	10.1016/j.ejmech.2021.113677	10.7270/Q2J38XCR	34225179			Chen, W; Chen, X; Li, D; Wang, X; Long, G; Jiang, Z; You, Q; Guo, X	China Pharmaceutical University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50574659	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50574659&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164617680	471064804							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51422342	CN1CCN(CC1)c1ccc(cc1NC(=O)c1cc(N)c(F)c(C)c1Cl)C#CCNC(=O)C1CCC(O)CC1	InChI=1S/C29H35ClFN5O3/c1-18-26(30)22(17-23(32)27(18)31)29(39)34-24-16-19(5-10-25(24)36-14-12-35(2)13-15-36)4-3-11-33-28(38)20-6-8-21(37)9-7-20/h5,10,16-17,20-21,37H,6-9,11-15,32H2,1-2H3,(H,33,38)(H,34,39)	QDIHXTGBZAYDNY-UHFFFAOYSA-N	50574660	CHEMBL4877455	WD repeat-containing protein 5			 125							ChEMBL	10.1016/j.ejmech.2021.113677	10.7270/Q2J38XCR	34225179			Chen, W; Chen, X; Li, D; Wang, X; Long, G; Jiang, Z; You, Q; Guo, X	China Pharmaceutical University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50574660	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50574660&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164627738	471064805							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51422343	CN1CCN(CC1)c1ccc(cc1NC(=O)c1cc(N)c(F)c(C)c1Cl)C#CCNC(=O)CC1CCOCC1	InChI=1S/C29H35ClFN5O3/c1-19-27(30)22(18-23(32)28(19)31)29(38)34-24-16-20(5-6-25(24)36-12-10-35(2)11-13-36)4-3-9-33-26(37)17-21-7-14-39-15-8-21/h5-6,16,18,21H,7-15,17,32H2,1-2H3,(H,33,37)(H,34,38)	LVLAVFWECSPOMI-UHFFFAOYSA-N	50574661	CHEMBL4859991	WD repeat-containing protein 5			 179							ChEMBL	10.1016/j.ejmech.2021.113677	10.7270/Q2J38XCR	34225179			Chen, W; Chen, X; Li, D; Wang, X; Long, G; Jiang, Z; You, Q; Guo, X	China Pharmaceutical University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50574661	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50574661&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164618030	471064806							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51422344	CN1CCN(CC1)c1ccc(cc1NC(=O)c1cc(N)c(F)c(C)c1Cl)C#CCNC(=O)CCCCO	InChI=1S/C27H33ClFN5O3/c1-18-25(28)20(17-21(30)26(18)29)27(37)32-22-16-19(6-5-10-31-24(36)7-3-4-15-35)8-9-23(22)34-13-11-33(2)12-14-34/h8-9,16-17,35H,3-4,7,10-15,30H2,1-2H3,(H,31,36)(H,32,37)	NAVJRMICJNPOSB-UHFFFAOYSA-N	50574662	CHEMBL4852501	WD repeat-containing protein 5			 148							ChEMBL	10.1016/j.ejmech.2021.113677	10.7270/Q2J38XCR	34225179			Chen, W; Chen, X; Li, D; Wang, X; Long, G; Jiang, Z; You, Q; Guo, X	China Pharmaceutical University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50574662	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50574662&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164611232	471064807							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51422345	CC(C)C(N)C(=O)NCC#Cc1ccc(N2CCN(C)CC2)c(NC(=O)c2cc(N)c(F)c(C)c2Cl)c1	InChI=1S/C27H34ClFN6O2/c1-16(2)25(31)27(37)32-9-5-6-18-7-8-22(35-12-10-34(4)11-13-35)21(14-18)33-26(36)19-15-20(30)24(29)17(3)23(19)28/h7-8,14-16,25H,9-13,30-31H2,1-4H3,(H,32,37)(H,33,36)	FTPFJGRCKOYJBW-UHFFFAOYSA-N	50574663	CHEMBL4846292	WD repeat-containing protein 5			 390							ChEMBL	10.1016/j.ejmech.2021.113677	10.7270/Q2J38XCR	34225179			Chen, W; Chen, X; Li, D; Wang, X; Long, G; Jiang, Z; You, Q; Guo, X	China Pharmaceutical University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50574663	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50574663&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164609212	471064808							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51422346	CN(C)C(=O)c1ccc(cc1)C(=O)NCC#Cc1ccc(N2CCN(C)CC2)c(NC(=O)c2cc(N)c(F)c(C)c2Cl)c1	InChI=1S/C32H34ClFN6O3/c1-20-28(33)24(19-25(35)29(20)34)31(42)37-26-18-21(7-12-27(26)40-16-14-39(4)15-17-40)6-5-13-36-30(41)22-8-10-23(11-9-22)32(43)38(2)3/h7-12,18-19H,13-17,35H2,1-4H3,(H,36,41)(H,37,42)	USSJDXKXMPIJJT-UHFFFAOYSA-N	50574664	CHEMBL4868412	WD repeat-containing protein 5			 60							ChEMBL	10.1016/j.ejmech.2021.113677	10.7270/Q2J38XCR	34225179			Chen, W; Chen, X; Li, D; Wang, X; Long, G; Jiang, Z; You, Q; Guo, X	China Pharmaceutical University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50574664	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50574664&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164623801	471064809							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51422347	CN1CCN(CC1)c1ccc(cc1NC(=O)c1cc(N)c(F)c(C)c1Cl)C#CCNC(=O)c1ccc(cc1)C(=O)N1CCOCC1	InChI=1S/C34H36ClFN6O4/c1-22-30(35)26(21-27(37)31(22)36)33(44)39-28-20-23(5-10-29(28)41-14-12-40(2)13-15-41)4-3-11-38-32(43)24-6-8-25(9-7-24)34(45)42-16-18-46-19-17-42/h5-10,20-21H,11-19,37H2,1-2H3,(H,38,43)(H,39,44)	OKASGPAJFIOSGT-UHFFFAOYSA-N	50574665	CHEMBL4864032	WD repeat-containing protein 5			 41							ChEMBL	10.1016/j.ejmech.2021.113677	10.7270/Q2J38XCR	34225179			Chen, W; Chen, X; Li, D; Wang, X; Long, G; Jiang, Z; You, Q; Guo, X	China Pharmaceutical University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50574665	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50574665&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164621331	471064810							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51422348	COC(=O)c1cn(nn1)-c1ccc(N2CCN(C)CC2)c(NC(=O)c2cc(N)c(F)c(C)c2Cl)c1	InChI=1S/C23H25ClFN7O3/c1-13-20(24)15(11-16(26)21(13)25)22(33)27-17-10-14(32-12-18(28-29-32)23(34)35-3)4-5-19(17)31-8-6-30(2)7-9-31/h4-5,10-12H,6-9,26H2,1-3H3,(H,27,33)	SKNBJKQSMQVYLP-UHFFFAOYSA-N	50574666	CHEMBL4868706	WD repeat-containing protein 5			 68							ChEMBL	10.1016/j.ejmech.2021.113677	10.7270/Q2J38XCR	34225179			Chen, W; Chen, X; Li, D; Wang, X; Long, G; Jiang, Z; You, Q; Guo, X	China Pharmaceutical University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50574666	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50574666&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			141725708	471064811							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51422349	CN1CCN(CC1)c1ccc(cc1NC(=O)c1cc(N)c(F)c(C)c1Cl)-n1cc(nn1)C(O)=O	InChI=1S/C22H23ClFN7O3/c1-12-19(23)14(10-15(25)20(12)24)21(32)26-16-9-13(31-11-17(22(33)34)27-28-31)3-4-18(16)30-7-5-29(2)6-8-30/h3-4,9-11H,5-8,25H2,1-2H3,(H,26,32)(H,33,34)	ULYZOXPTGWTZKW-UHFFFAOYSA-N	50574667	CHEMBL4866458	WD repeat-containing protein 5			 1036							ChEMBL	10.1016/j.ejmech.2021.113677	10.7270/Q2J38XCR	34225179			Chen, W; Chen, X; Li, D; Wang, X; Long, G; Jiang, Z; You, Q; Guo, X	China Pharmaceutical University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50574667	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50574667&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			141725705	471064812							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51422350	CN(C)C(=O)c1cn(nn1)-c1ccc(N2CCN(C)CC2)c(NC(=O)c2cc(N)c(F)c(C)c2Cl)c1	InChI=1S/C24H28ClFN8O2/c1-14-21(25)16(12-17(27)22(14)26)23(35)28-18-11-15(34-13-19(29-30-34)24(36)31(2)3)5-6-20(18)33-9-7-32(4)8-10-33/h5-6,11-13H,7-10,27H2,1-4H3,(H,28,35)	YVYDEUSEBPMHIF-UHFFFAOYSA-N	50574668	CHEMBL4850959	WD repeat-containing protein 5			 34							ChEMBL	10.1016/j.ejmech.2021.113677	10.7270/Q2J38XCR	34225179			Chen, W; Chen, X; Li, D; Wang, X; Long, G; Jiang, Z; You, Q; Guo, X	China Pharmaceutical University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50574668	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50574668&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			141725707	471064813							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51422351	CN1CCN(CC1)c1ccc(cc1NC(=O)c1cc(N)c(F)c(C)c1Cl)-n1cc(nn1)C(=O)N1CCOCC1	InChI=1S/C26H30ClFN8O3/c1-16-23(27)18(14-19(29)24(16)28)25(37)30-20-13-17(3-4-22(20)34-7-5-33(2)6-8-34)36-15-21(31-32-36)26(38)35-9-11-39-12-10-35/h3-4,13-15H,5-12,29H2,1-2H3,(H,30,37)	PBPMDBKPPQYRLH-UHFFFAOYSA-N	50574669	CHEMBL4852951	WD repeat-containing protein 5			 11							ChEMBL	10.1016/j.ejmech.2021.113677	10.7270/Q2J38XCR	34225179			Chen, W; Chen, X; Li, D; Wang, X; Long, G; Jiang, Z; You, Q; Guo, X	China Pharmaceutical University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50574669	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50574669&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			141725700	471064814							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51422352	CN1CCN(CC1)c1ccc(cc1NC(=O)c1cc(N)c(F)c(C)c1Cl)-n1cc(nn1)C(=O)NC1CCOCC1	InChI=1S/C27H32ClFN8O3/c1-16-24(28)19(14-20(30)25(16)29)26(38)32-21-13-18(3-4-23(21)36-9-7-35(2)8-10-36)37-15-22(33-34-37)27(39)31-17-5-11-40-12-6-17/h3-4,13-15,17H,5-12,30H2,1-2H3,(H,31,39)(H,32,38)	WKDPERRTFWPQQI-UHFFFAOYSA-N	50574670	CHEMBL4863061	WD repeat-containing protein 5			 16							ChEMBL	10.1016/j.ejmech.2021.113677	10.7270/Q2J38XCR	34225179			Chen, W; Chen, X; Li, D; Wang, X; Long, G; Jiang, Z; You, Q; Guo, X	China Pharmaceutical University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50574670	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50574670&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			141725706	471064815							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51422353	CN1CCC(CC1)NC(=O)c1cn(nn1)-c1ccc(N2CCN(C)CC2)c(NC(=O)c2cc(N)c(F)c(C)c2Cl)c1	InChI=1S/C28H35ClFN9O2/c1-17-25(29)20(15-21(31)26(17)30)27(40)33-22-14-19(4-5-24(22)38-12-10-37(3)11-13-38)39-16-23(34-35-39)28(41)32-18-6-8-36(2)9-7-18/h4-5,14-16,18H,6-13,31H2,1-3H3,(H,32,41)(H,33,40)	AQQCBBDWEBSYPT-UHFFFAOYSA-N	50574671	CHEMBL4869658	WD repeat-containing protein 5			 8.9							ChEMBL	10.1016/j.ejmech.2021.113677	10.7270/Q2J38XCR	34225179			Chen, W; Chen, X; Li, D; Wang, X; Long, G; Jiang, Z; You, Q; Guo, X	China Pharmaceutical University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50574671	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50574671&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			141725709	471064816							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51422354	CN1CCN(CC1)c1ccc(cc1NC(=O)c1cc(N)c(F)c(C)c1Cl)-n1cc(nn1)C(=O)NCCCN1CCOCC1	InChI=1S/C29H37ClFN9O3/c1-19-26(30)21(17-22(32)27(19)31)28(41)34-23-16-20(4-5-25(23)39-10-8-37(2)9-11-39)40-18-24(35-36-40)29(42)33-6-3-7-38-12-14-43-15-13-38/h4-5,16-18H,3,6-15,32H2,1-2H3,(H,33,42)(H,34,41)	MPTAUAHHFUFKAG-UHFFFAOYSA-N	50574672	CHEMBL4861912	WD repeat-containing protein 5			 8.6							ChEMBL	10.1016/j.ejmech.2021.113677	10.7270/Q2J38XCR	34225179			Chen, W; Chen, X; Li, D; Wang, X; Long, G; Jiang, Z; You, Q; Guo, X	China Pharmaceutical University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50574672	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50574672&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			156112343	471064817							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51422355	CN1CCN(CC1)C(=O)c1cn(nn1)-c1ccc(N2CCN(C)CC2)c(NC(=O)c2cc(N)c(F)c(C)c2Cl)c1	InChI=1S/C27H33ClFN9O2/c1-17-24(28)19(15-20(30)25(17)29)26(39)31-21-14-18(4-5-23(21)36-10-6-34(2)7-11-36)38-16-22(32-33-38)27(40)37-12-8-35(3)9-13-37/h4-5,14-16H,6-13,30H2,1-3H3,(H,31,39)	ODAHPVIJSAJSJC-UHFFFAOYSA-N	50574673	CHEMBL4851969	WD repeat-containing protein 5			 9.0							ChEMBL	10.1016/j.ejmech.2021.113677	10.7270/Q2J38XCR	34225179			Chen, W; Chen, X; Li, D; Wang, X; Long, G; Jiang, Z; You, Q; Guo, X	China Pharmaceutical University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50574673	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50574673&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			156112338	471064818							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51422356	CN1CCN(CC1)c1ccc(cc1NC(=O)c1cc(N)c(F)c(C)c1Cl)-n1cc(nn1)C(=O)NCCN1CCOCC1	InChI=1S/C28H35ClFN9O3/c1-18-25(29)20(16-21(31)26(18)30)27(40)33-22-15-19(3-4-24(22)38-9-7-36(2)8-10-38)39-17-23(34-35-39)28(41)32-5-6-37-11-13-42-14-12-37/h3-4,15-17H,5-14,31H2,1-2H3,(H,32,41)(H,33,40)	GVBIZPYPVRMOAF-UHFFFAOYSA-N	50574674	CHEMBL4852196	WD repeat-containing protein 5			 20							ChEMBL	10.1016/j.ejmech.2021.113677	10.7270/Q2J38XCR	34225179			Chen, W; Chen, X; Li, D; Wang, X; Long, G; Jiang, Z; You, Q; Guo, X	China Pharmaceutical University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50574674	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50574674&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			156112342	471064819							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51422357	COC(=O)c1ccc(cc1)-c1ccc(N2CCN(C)CC2)c(NC(=O)c2cc(N)c(F)c(C)c2Cl)c1	InChI=1S/C27H28ClFN4O3/c1-16-24(28)20(15-21(30)25(16)29)26(34)31-22-14-19(17-4-6-18(7-5-17)27(35)36-3)8-9-23(22)33-12-10-32(2)11-13-33/h4-9,14-15H,10-13,30H2,1-3H3,(H,31,34)	ADXWUOCLGQOCFF-UHFFFAOYSA-N	50208384	CHEMBL3884212	WD repeat-containing protein 5			 70							ChEMBL	10.1016/j.ejmech.2021.113677	10.7270/Q2J38XCR	34225179			Chen, W; Chen, X; Li, D; Wang, X; Long, G; Jiang, Z; You, Q; Guo, X	China Pharmaceutical University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50208384	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50208384&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			134131548	375982032		CHEMBL3884212					1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51422358	CN1CCN(CC1)c1ccc(cc1NC(=O)c1cc(N)c(F)c(C)c1Cl)-c1ccc(cc1)C(O)=O	InChI=1S/C26H26ClFN4O3/c1-15-23(27)19(14-20(29)24(15)28)25(33)30-21-13-18(16-3-5-17(6-4-16)26(34)35)7-8-22(21)32-11-9-31(2)10-12-32/h3-8,13-14H,9-12,29H2,1-2H3,(H,30,33)(H,34,35)	FMVQTQJEPRFHFC-UHFFFAOYSA-N	50574675	CHEMBL4878567	WD repeat-containing protein 5			 99							ChEMBL	10.1016/j.ejmech.2021.113677	10.7270/Q2J38XCR	34225179			Chen, W; Chen, X; Li, D; Wang, X; Long, G; Jiang, Z; You, Q; Guo, X	China Pharmaceutical University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50574675	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50574675&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164626399	471064820							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51422359	CN(C)C(=O)c1ccc(cc1)-c1ccc(N2CCN(C)CC2)c(NC(=O)c2cc(N)c(F)c(C)c2Cl)c1	InChI=1S/C28H31ClFN5O2/c1-17-25(29)21(16-22(31)26(17)30)27(36)32-23-15-20(9-10-24(23)35-13-11-34(4)12-14-35)18-5-7-19(8-6-18)28(37)33(2)3/h5-10,15-16H,11-14,31H2,1-4H3,(H,32,36)	TYHLFPRXEUVIDJ-UHFFFAOYSA-N	50574676	CHEMBL4868755	WD repeat-containing protein 5			 73							ChEMBL	10.1016/j.ejmech.2021.113677	10.7270/Q2J38XCR	34225179			Chen, W; Chen, X; Li, D; Wang, X; Long, G; Jiang, Z; You, Q; Guo, X	China Pharmaceutical University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50574676	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50574676&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			156357381	471064821							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51422360	CN1CCN(CC1)c1ccc(cc1NC(=O)c1cc(N)c(F)c(C)c1Cl)-c1ccc(cc1)C(=O)N1CCOCC1	InChI=1S/C30H33ClFN5O3/c1-19-27(31)23(18-24(33)28(19)32)29(38)34-25-17-22(7-8-26(25)36-11-9-35(2)10-12-36)20-3-5-21(6-4-20)30(39)37-13-15-40-16-14-37/h3-8,17-18H,9-16,33H2,1-2H3,(H,34,38)	GQCCHJGHPVLGRW-UHFFFAOYSA-N	50574677	CHEMBL4847277	WD repeat-containing protein 5			 56							ChEMBL	10.1016/j.ejmech.2021.113677	10.7270/Q2J38XCR	34225179			Chen, W; Chen, X; Li, D; Wang, X; Long, G; Jiang, Z; You, Q; Guo, X	China Pharmaceutical University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50574677	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50574677&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			156357408	471064822							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51422361	CN1CCC(CC1)C(=O)Nc1ccc(cc1)-c1ccc(N2CCN(C)CC2)c(NC(=O)c2cc(N)c(F)c(C)c2Cl)c1	InChI=1S/C32H38ClFN6O2/c1-20-29(33)25(19-26(35)30(20)34)32(42)37-27-18-23(6-9-28(27)40-16-14-39(3)15-17-40)21-4-7-24(8-5-21)36-31(41)22-10-12-38(2)13-11-22/h4-9,18-19,22H,10-17,35H2,1-3H3,(H,36,41)(H,37,42)	SLXSSKXBCOHTGP-UHFFFAOYSA-N	50574678	CHEMBL4852048	WD repeat-containing protein 5			 16							ChEMBL	10.1016/j.ejmech.2021.113677	10.7270/Q2J38XCR	34225179			Chen, W; Chen, X; Li, D; Wang, X; Long, G; Jiang, Z; You, Q; Guo, X	China Pharmaceutical University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50574678	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50574678&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			156357252	471064823							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51422362	CN1CCN(CC1)c1ccc(cc1NC(=O)c1cc(N)c(F)c(C)c1Cl)-c1ccc(NC(=O)C2CCOCC2)cc1	InChI=1S/C31H35ClFN5O3/c1-19-28(32)24(18-25(34)29(19)33)31(40)36-26-17-22(5-8-27(26)38-13-11-37(2)12-14-38)20-3-6-23(7-4-20)35-30(39)21-9-15-41-16-10-21/h3-8,17-18,21H,9-16,34H2,1-2H3,(H,35,39)(H,36,40)	ISZJFLIDMRJLNB-UHFFFAOYSA-N	50574679	CHEMBL4845887	WD repeat-containing protein 5			 6.5							ChEMBL	10.1016/j.ejmech.2021.113677	10.7270/Q2J38XCR	34225179			Chen, W; Chen, X; Li, D; Wang, X; Long, G; Jiang, Z; You, Q; Guo, X	China Pharmaceutical University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50574679	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50574679&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164609003	471064824							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51422363	CN1CCN(CC1)c1ccc(cc1NC(=O)c1cc(N)c(F)c(C)c1Cl)-n1cc(nn1)C(=O)NCCCN1CCOCC1	InChI=1S/C29H37ClFN9O3/c1-19-26(30)21(17-22(32)27(19)31)28(41)34-23-16-20(4-5-25(23)39-10-8-37(2)9-11-39)40-18-24(35-36-40)29(42)33-6-3-7-38-12-14-43-15-13-38/h4-5,16-18H,3,6-15,32H2,1-2H3,(H,33,42)(H,34,41)	MPTAUAHHFUFKAG-UHFFFAOYSA-N	50574672	CHEMBL4861912	WD repeat-containing protein 5				 12						ChEMBL	10.1016/j.ejmech.2021.113677	10.7270/Q2J38XCR	34225179			Chen, W; Chen, X; Li, D; Wang, X; Long, G; Jiang, Z; You, Q; Guo, X	China Pharmaceutical University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50574672	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50574672&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			156112343	471064817							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51422371	CCC(CC)(NC(=O)C(C)C)C(=O)N[C@@H](CCCNC(N)=N)C(=O)NC1(CCCC1)C(=O)NC(c1ccc(F)cc1)c1ccc(F)cc1	InChI=1S/C35H49F2N7O4/c1-5-34(6-2,43-29(45)22(3)4)31(47)41-27(10-9-21-40-33(38)39)30(46)44-35(19-7-8-20-35)32(48)42-28(23-11-15-25(36)16-12-23)24-13-17-26(37)18-14-24/h11-18,22,27-28H,5-10,19-21H2,1-4H3,(H,41,47)(H,42,48)(H,43,45)(H,44,46)(H4,38,39,40)/t27-/m0/s1	RZKSQRIPRKWVBU-MHZLTWQESA-N	200723	US9233086, 10L	WD repeat-containing protein 5			 2.4							ChEMBL	10.1016/j.ejmech.2021.113677	10.7270/Q2J38XCR	34225179			Chen, W; Chen, X; Li, D; Wang, X; Long, G; Jiang, Z; You, Q; Guo, X	China Pharmaceutical University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=200723	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=200723&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			54766613	318834336							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51422372	CN1CCN(CC1)c1ccc(cc1NC(=O)c1ccccc1Cl)[N+]([O-])=O	InChI=1S/C18H19ClN4O3/c1-21-8-10-22(11-9-21)17-7-6-13(23(25)26)12-16(17)20-18(24)14-4-2-3-5-15(14)19/h2-7,12H,8-11H2,1H3,(H,20,24)	WOGZFCMBPXJNFI-UHFFFAOYSA-N	50428254	CHEMBL1609857	WD repeat-containing protein 5				 12000						ChEMBL	10.1016/j.ejmech.2021.113677	10.7270/Q2J38XCR	34225179			Chen, W; Chen, X; Li, D; Wang, X; Long, G; Jiang, Z; You, Q; Guo, X	China Pharmaceutical University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50428254	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50428254&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	NP7	3SMR	2965974	164157129		CHEMBL1609857				ZINC05049228	1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51438468	CN(C)C(=O)c1ccc(cc1)-c1cc(Nc2ncnc(Cl)c2N)c(cc1F)N1CCN(C)CC1	InChI=1S/C24H27ClFN7O/c1-31(2)24(34)16-6-4-15(5-7-16)17-12-19(30-23-21(27)22(25)28-14-29-23)20(13-18(17)26)33-10-8-32(3)9-11-33/h4-7,12-14H,8-11,27H2,1-3H3,(H,28,29,30)	LXONEMNSYOAQJT-UHFFFAOYSA-N	50581147	CHEMBL5094242	WD repeat-containing protein 5				 73						ChEMBL	10.1021/acs.jmedchem.1c00091	10.7270/Q22B92X1	34105966			Chen, W; Chen, X; Li, D; Zhou, J; Jiang, Z; You, Q; Guo, X	China Pharmaceutical University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50581147	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50581147&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			145926792	476026152							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51438474	CN1CCN(CC1)c1ccc(cc1NC(=O)c1ccccc1Cl)[N+]([O-])=O	InChI=1S/C18H19ClN4O3/c1-21-8-10-22(11-9-21)17-7-6-13(23(25)26)12-16(17)20-18(24)14-4-2-3-5-15(14)19/h2-7,12H,8-11H2,1H3,(H,20,24)	WOGZFCMBPXJNFI-UHFFFAOYSA-N	50428254	CHEMBL1609857	WD repeat-containing protein 5				 7000						ChEMBL	10.1021/acs.jmedchem.1c00091	10.7270/Q22B92X1	34105966			Chen, W; Chen, X; Li, D; Zhou, J; Jiang, Z; You, Q; Guo, X	China Pharmaceutical University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50428254	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50428254&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	NP7	3SMR	2965974	164157129		CHEMBL1609857				ZINC05049228	1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51493601	C[C@H]1CN(CCN1C)c1cc(F)c(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cnc(nc1)N1CCOCC1			552952	N-[2-[(3S)-3,4- dimethylpiperazin-1-yl]- 4-fluoro-5-(2-morpholin- 4-ylpyrimidin-5- yl)phenyl]-6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carboxamide::US11319299, Example 7	WD repeat-containing protein 5				 0.060000						ChEMBL		10.7270/Q2B85D61	34283608			Chen, X; Xu, J; Wang, X; Long, G; You, Q; Guo, X	China Pharmaceutical University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=552952	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=552952&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			164607808	469796821							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51493602	CC[C@@H]1NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@@H](CCCCNC(=O)[C@H](NC1=O)c1ccccc1)NC(=O)C(C)C	InChI=1S/C28H44N8O5/c1-4-19-24(38)36-22(18-11-6-5-7-12-18)27(41)31-15-9-8-13-20(34-23(37)17(2)3)26(40)35-21(25(39)33-19)14-10-16-32-28(29)30/h5-7,11-12,17,19-22H,4,8-10,13-16H2,1-3H3,(H,31,41)(H,33,39)(H,34,37)(H,35,40)(H,36,38)(H4,29,30,32)/t19-,20+,21-,22+/m0/s1	PYARBFPEJRKODC-LNRXMEIDSA-N	50601691	CHEMBL4116915	WD repeat-containing protein 5			 0.900000							ChEMBL		10.7270/Q2B85D61	34283608			Chen, X; Xu, J; Wang, X; Long, G; You, Q; Guo, X	China Pharmaceutical University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50601691	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50601691&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			137630583	482612542							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51493603	CCC(CC)(NC(=O)C(C)C)C(=O)N[C@@H](CCCNC(N)=N)C(=O)NC1(CCCC1)C(=O)NC(c1ccc(F)cc1)c1ccc(F)cc1	InChI=1S/C35H49F2N7O4/c1-5-34(6-2,43-29(45)22(3)4)31(47)41-27(10-9-21-40-33(38)39)30(46)44-35(19-7-8-20-35)32(48)42-28(23-11-15-25(36)16-12-23)24-13-17-26(37)18-14-24/h11-18,22,27-28H,5-10,19-21H2,1-4H3,(H,41,47)(H,42,48)(H,43,45)(H,44,46)(H4,38,39,40)/t27-/m0/s1	RZKSQRIPRKWVBU-MHZLTWQESA-N	200723	US9233086, 10L	WD repeat-containing protein 5			 2.4							ChEMBL		10.7270/Q2B85D61	34283608			Chen, X; Xu, J; Wang, X; Long, G; You, Q; Guo, X	China Pharmaceutical University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=200723	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=200723&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			54766613	318834336							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51493604	CCC(CC)(NC(=O)C(C)C)C(=O)N[C@@H](CCCNC(N)=N)C(=O)NC1(CCCC1)C(=O)NC(c1ccccc1)c1ccccc1	InChI=1S/C35H51N7O4/c1-5-34(6-2,41-29(43)24(3)4)31(45)39-27(20-15-23-38-33(36)37)30(44)42-35(21-13-14-22-35)32(46)40-28(25-16-9-7-10-17-25)26-18-11-8-12-19-26/h7-12,16-19,24,27-28H,5-6,13-15,20-23H2,1-4H3,(H,39,45)(H,40,46)(H,41,43)(H,42,44)(H4,36,37,38)/t27-/m0/s1	BCIPILGGOSCOMC-MHZLTWQESA-N	200712	US9233086, 10A	WD repeat-containing protein 5			 2.9							ChEMBL		10.7270/Q2B85D61	34283608			Chen, X; Xu, J; Wang, X; Long, G; You, Q; Guo, X	China Pharmaceutical University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=200712	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=200712&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			53356803	318834325							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51493605	CN1CCN(CC1)c1ccc(cc1NC(=O)c1cc(N)c(F)c(C)c1Cl)-c1ccc(cc1)C(=O)NCCCN	InChI=1S/C29H34ClFN6O2/c1-18-26(30)22(17-23(33)27(18)31)29(39)35-24-16-21(8-9-25(24)37-14-12-36(2)13-15-37)19-4-6-20(7-5-19)28(38)34-11-3-10-32/h4-9,16-17H,3,10-15,32-33H2,1-2H3,(H,34,38)(H,35,39)	OGLREAITVXTJOM-UHFFFAOYSA-N	50601692	CHEMBL5172154	WD repeat-containing protein 5			 7.4							ChEMBL		10.7270/Q2B85D61	34283608			Chen, X; Xu, J; Wang, X; Long, G; You, Q; Guo, X	China Pharmaceutical University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50601692	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50601692&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			168269940	482612543							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51493606	CN(C)C(=O)c1ccc(cc1)-c1cc(Nc2ncnc(Cl)c2N)c(cc1F)N1CCN(C)CC1	InChI=1S/C24H27ClFN7O/c1-31(2)24(34)16-6-4-15(5-7-16)17-12-19(30-23-21(27)22(25)28-14-29-23)20(13-18(17)26)33-10-8-32(3)9-11-33/h4-7,12-14H,8-11,27H2,1-3H3,(H,28,29,30)	LXONEMNSYOAQJT-UHFFFAOYSA-N	50581147	CHEMBL5094242	WD repeat-containing protein 5			 29							ChEMBL		10.7270/Q2B85D61	34283608			Chen, X; Xu, J; Wang, X; Long, G; You, Q; Guo, X	China Pharmaceutical University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50581147	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50581147&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			145926792	476026152							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51493607	CN1CCN(CC1)c1ccc(cc1NC(=O)c1cc(N)c(F)c(C)c1Cl)-n1cc(nn1)C(=O)NCCCN1CCOCC1	InChI=1S/C29H37ClFN9O3/c1-19-26(30)21(17-22(32)27(19)31)28(41)34-23-16-20(4-5-25(23)39-10-8-37(2)9-11-39)40-18-24(35-36-40)29(42)33-6-3-7-38-12-14-43-15-13-38/h4-5,16-18H,3,6-15,32H2,1-2H3,(H,33,42)(H,34,41)	MPTAUAHHFUFKAG-UHFFFAOYSA-N	50574672	CHEMBL4861912	WD repeat-containing protein 5			<10.0							ChEMBL		10.7270/Q2B85D61	34283608			Chen, X; Xu, J; Wang, X; Long, G; You, Q; Guo, X	China Pharmaceutical University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50574672	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50574672&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			156112343	471064817							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51492472	CN1CCN(CC1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(cc1)C(=O)NCCCCCC(=O)N[C@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)NCc1ccc(cc1)-c1scnc1C)C(C)(C)C	InChI=1S/C53H62F3N9O7S/c1-32-46(73-31-60-32)35-12-10-33(11-13-35)28-59-50(71)43-26-38(66)30-65(43)51(72)47(52(2,3)4)62-44(67)9-7-6-8-20-57-48(69)36-16-14-34(15-17-36)37-18-19-42(64-23-21-63(5)22-24-64)41(25-37)61-49(70)39-29-58-45(68)27-40(39)53(54,55)56/h10-19,25,27,29,31,38,43,47,66H,6-9,20-24,26,28,30H2,1-5H3,(H,57,69)(H,58,68)(H,59,71)(H,61,70)(H,62,67)/t38-,43+,47-/m1/s1	UPLJFUHLGRAYID-MXPJCAPISA-N	50601522	CHEMBL5186307	WD repeat-containing protein 5				 12000						ChEMBL		10.7270/Q20Z77B9	33980013			Dölle, A; Adhikari, B; Krämer, A; Weckesser, J; Berner, N; Berger, LM; Diebold, M; Szewczyk, MM; Barsyte-Lovejoy, D; Arrowsmith, CH; Gebel, J; Löhr, F; Dötsch, V; Eilers, M; Heinzlmeir, S; Kuster, B; Sotriffer, C; Wolf, E; Knapp, S	Goethe University Frankfurt am Main	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50601522	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50601522&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			168279616	482612374							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51492473	CN1CCN(CC1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(cc1)C(=O)NCCCCCCC(=O)N[C@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)NCc1ccc(cc1)-c1scnc1C)C(C)(C)C	InChI=1S/C54H64F3N9O7S/c1-33-47(74-32-61-33)36-13-11-34(12-14-36)29-60-51(72)44-27-39(67)31-66(44)52(73)48(53(2,3)4)63-45(68)10-8-6-7-9-21-58-49(70)37-17-15-35(16-18-37)38-19-20-43(65-24-22-64(5)23-25-65)42(26-38)62-50(71)40-30-59-46(69)28-41(40)54(55,56)57/h11-20,26,28,30,32,39,44,48,67H,6-10,21-25,27,29,31H2,1-5H3,(H,58,70)(H,59,69)(H,60,72)(H,62,71)(H,63,68)/t39-,44+,48-/m1/s1	BXKFHYMDHAHJSX-UOHLUGTHSA-N	50601523	CHEMBL5180413	WD repeat-containing protein 5				 11000						ChEMBL		10.7270/Q20Z77B9	33980013			Dölle, A; Adhikari, B; Krämer, A; Weckesser, J; Berner, N; Berger, LM; Diebold, M; Szewczyk, MM; Barsyte-Lovejoy, D; Arrowsmith, CH; Gebel, J; Löhr, F; Dötsch, V; Eilers, M; Heinzlmeir, S; Kuster, B; Sotriffer, C; Wolf, E; Knapp, S	Goethe University Frankfurt am Main	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50601523	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50601523&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			168276743	482612375							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51492474	CN1CCN(CC1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(cc1)C(=O)NCc1ccc(CC(=O)N[C@H](C(=O)N2C[C@H](O)C[C@H]2C(=O)NCc2ccc(cc2)-c2scnc2C)C(C)(C)C)cc1	InChI=1S/C56H60F3N9O7S/c1-33-49(76-32-63-33)38-12-10-36(11-13-38)29-62-53(74)46-26-41(69)31-68(46)54(75)50(55(2,3)4)65-48(71)24-34-6-8-35(9-7-34)28-61-51(72)39-16-14-37(15-17-39)40-18-19-45(67-22-20-66(5)21-23-67)44(25-40)64-52(73)42-30-60-47(70)27-43(42)56(57,58)59/h6-19,25,27,30,32,41,46,50,69H,20-24,26,28-29,31H2,1-5H3,(H,60,70)(H,61,72)(H,62,74)(H,64,73)(H,65,71)/t41-,46+,50-/m1/s1	PJYZWCPLYVFKHH-PNWJTEEHSA-N	50601524	CHEMBL5201006	WD repeat-containing protein 5				 33000						ChEMBL		10.7270/Q20Z77B9	33980013			Dölle, A; Adhikari, B; Krämer, A; Weckesser, J; Berner, N; Berger, LM; Diebold, M; Szewczyk, MM; Barsyte-Lovejoy, D; Arrowsmith, CH; Gebel, J; Löhr, F; Dötsch, V; Eilers, M; Heinzlmeir, S; Kuster, B; Sotriffer, C; Wolf, E; Knapp, S	Goethe University Frankfurt am Main	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50601524	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50601524&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			165416424	482612376							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51492475	COc1ccc(cc1CNC(=O)Cc1ccc(Cl)c(Cl)c1)-c1cn2CCCc2n1	InChI=1S/C22H21Cl2N3O2/c1-29-20-7-5-15(19-13-27-8-2-3-21(27)26-19)11-16(20)12-25-22(28)10-14-4-6-17(23)18(24)9-14/h4-7,9,11,13H,2-3,8,10,12H2,1H3,(H,25,28)	VZEIIDRXHZLNCH-UHFFFAOYSA-N	50601525	CHEMBL5186473	WD repeat-containing protein 5				 125000						ChEMBL		10.7270/Q20Z77B9	33980013			Dölle, A; Adhikari, B; Krämer, A; Weckesser, J; Berner, N; Berger, LM; Diebold, M; Szewczyk, MM; Barsyte-Lovejoy, D; Arrowsmith, CH; Gebel, J; Löhr, F; Dötsch, V; Eilers, M; Heinzlmeir, S; Kuster, B; Sotriffer, C; Wolf, E; Knapp, S	Goethe University Frankfurt am Main	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50601525	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50601525&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			168278610	482612377							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51492476	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCOCCOCCOc2ccc(cc2CNC(=O)Cc2ccc(Cl)c(Cl)c2)-c2cn3CCCc3n2)C(C)(C)C)cc1	InChI=1S/C50H59Cl2N7O8S/c1-31-46(68-30-55-31)34-10-7-32(8-11-34)26-54-48(63)41-25-37(60)28-59(41)49(64)47(50(2,3)4)57-44(61)15-17-65-18-19-66-20-21-67-42-14-12-35(40-29-58-16-5-6-43(58)56-40)24-36(42)27-53-45(62)23-33-9-13-38(51)39(52)22-33/h7-14,22,24,29-30,37,41,47,60H,5-6,15-21,23,25-28H2,1-4H3,(H,53,62)(H,54,63)(H,57,61)/t37-,41+,47-/m1/s1	KUOHKJIOVPXKOP-AWWHSMTCSA-N	50601526	CHEMBL5193707	WD repeat-containing protein 5				 97000						ChEMBL		10.7270/Q20Z77B9	33980013			Dölle, A; Adhikari, B; Krämer, A; Weckesser, J; Berner, N; Berger, LM; Diebold, M; Szewczyk, MM; Barsyte-Lovejoy, D; Arrowsmith, CH; Gebel, J; Löhr, F; Dötsch, V; Eilers, M; Heinzlmeir, S; Kuster, B; Sotriffer, C; Wolf, E; Knapp, S	Goethe University Frankfurt am Main	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50601526	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50601526&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			168288801	482612378							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51492477	CN1CCN(CC1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(CN2CCOCC2)cc1	InChI=1S/C29H32F3N5O3/c1-35-8-10-37(11-9-35)26-7-6-22(21-4-2-20(3-5-21)19-36-12-14-40-15-13-36)16-25(26)34-28(39)23-18-33-27(38)17-24(23)29(30,31)32/h2-7,16-18H,8-15,19H2,1H3,(H,33,38)(H,34,39)	GQTXDUXACYMXPD-UHFFFAOYSA-N	50601515	CHEMBL5194499	WD repeat-containing protein 5			 310							ChEMBL		10.7270/Q20Z77B9	33980013			Dölle, A; Adhikari, B; Krämer, A; Weckesser, J; Berner, N; Berger, LM; Diebold, M; Szewczyk, MM; Barsyte-Lovejoy, D; Arrowsmith, CH; Gebel, J; Löhr, F; Dötsch, V; Eilers, M; Heinzlmeir, S; Kuster, B; Sotriffer, C; Wolf, E; Knapp, S	Goethe University Frankfurt am Main	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50601515	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50601515&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			168289697	482612367							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51492478	CN1CCN(CC1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(cc1)C(=O)OC(C)(C)C	InChI=1S/C29H31F3N4O4/c1-28(2,3)40-27(39)19-7-5-18(6-8-19)20-9-10-24(36-13-11-35(4)12-14-36)23(15-20)34-26(38)21-17-33-25(37)16-22(21)29(30,31)32/h5-10,15-17H,11-14H2,1-4H3,(H,33,37)(H,34,38)	HATZDQFMULXBFB-UHFFFAOYSA-N	50601516	CHEMBL5181586	WD repeat-containing protein 5			 140							ChEMBL		10.7270/Q20Z77B9	33980013			Dölle, A; Adhikari, B; Krämer, A; Weckesser, J; Berner, N; Berger, LM; Diebold, M; Szewczyk, MM; Barsyte-Lovejoy, D; Arrowsmith, CH; Gebel, J; Löhr, F; Dötsch, V; Eilers, M; Heinzlmeir, S; Kuster, B; Sotriffer, C; Wolf, E; Knapp, S	Goethe University Frankfurt am Main	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50601516	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50601516&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			168277961	482612368							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51492479	CN1CCN(CC1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(cc1)C(=O)NCCOCCNc1cccc2C(=O)N(C3CCC(=O)NC3=O)C(=O)c12	InChI=1S/C42H41F3N8O8/c1-51-15-17-52(18-16-51)32-10-9-26(21-31(32)49-38(57)28-23-48-35(55)22-29(28)42(43,44)45)24-5-7-25(8-6-24)37(56)47-14-20-61-19-13-46-30-4-2-3-27-36(30)41(60)53(40(27)59)33-11-12-34(54)50-39(33)58/h2-10,21-23,33,46H,11-20H2,1H3,(H,47,56)(H,48,55)(H,49,57)(H,50,54,58)	CCAKBASGLWLWPO-UHFFFAOYSA-N	50601517	CHEMBL5181611	WD repeat-containing protein 5			 4300							ChEMBL		10.7270/Q20Z77B9	33980013			Dölle, A; Adhikari, B; Krämer, A; Weckesser, J; Berner, N; Berger, LM; Diebold, M; Szewczyk, MM; Barsyte-Lovejoy, D; Arrowsmith, CH; Gebel, J; Löhr, F; Dötsch, V; Eilers, M; Heinzlmeir, S; Kuster, B; Sotriffer, C; Wolf, E; Knapp, S	Goethe University Frankfurt am Main	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50601517	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50601517&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			168272844	482612369							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51492480	CN1CCN(CC1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(cc1)C(=O)NCCOCCOCCOCCNc1cccc2C(=O)N(C3CCC(=O)NC3=O)C(=O)c12	InChI=1S/C46H49F3N8O10/c1-55-15-17-56(18-16-55)36-10-9-30(25-35(36)53-42(61)32-27-52-39(59)26-33(32)46(47,48)49)28-5-7-29(8-6-28)41(60)51-14-20-66-22-24-67-23-21-65-19-13-50-34-4-2-3-31-40(34)45(64)57(44(31)63)37-11-12-38(58)54-43(37)62/h2-10,25-27,37,50H,11-24H2,1H3,(H,51,60)(H,52,59)(H,53,61)(H,54,58,62)	MPVUSWCQRFACNA-UHFFFAOYSA-N	50601527	CHEMBL5178796	WD repeat-containing protein 5			 4180							ChEMBL		10.7270/Q20Z77B9	33980013			Dölle, A; Adhikari, B; Krämer, A; Weckesser, J; Berner, N; Berger, LM; Diebold, M; Szewczyk, MM; Barsyte-Lovejoy, D; Arrowsmith, CH; Gebel, J; Löhr, F; Dötsch, V; Eilers, M; Heinzlmeir, S; Kuster, B; Sotriffer, C; Wolf, E; Knapp, S	Goethe University Frankfurt am Main	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50601527	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50601527&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			168274224	482612379							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51492481	CN1CCN(CC1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(cc1)C(=O)NCCOCCOCCOCCOCCOCCNc1cccc2C(=O)N(C3CCC(=O)NC3=O)C(=O)c12	InChI=1S/C50H57F3N8O12/c1-59-15-17-60(18-16-59)40-10-9-34(29-39(40)57-46(65)36-31-56-43(63)30-37(36)50(51,52)53)32-5-7-33(8-6-32)45(64)55-14-20-70-22-24-72-26-28-73-27-25-71-23-21-69-19-13-54-38-4-2-3-35-44(38)49(68)61(48(35)67)41-11-12-42(62)58-47(41)66/h2-10,29-31,41,54H,11-28H2,1H3,(H,55,64)(H,56,63)(H,57,65)(H,58,62,66)	DHDXVQJEEHRETI-UHFFFAOYSA-N	50601528	CHEMBL5176119	WD repeat-containing protein 5			 14100							ChEMBL		10.7270/Q20Z77B9	33980013			Dölle, A; Adhikari, B; Krämer, A; Weckesser, J; Berner, N; Berger, LM; Diebold, M; Szewczyk, MM; Barsyte-Lovejoy, D; Arrowsmith, CH; Gebel, J; Löhr, F; Dötsch, V; Eilers, M; Heinzlmeir, S; Kuster, B; Sotriffer, C; Wolf, E; Knapp, S	Goethe University Frankfurt am Main	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50601528	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50601528&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			168276134	482612380							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51492482	CN1CCN(CC1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(cc1)C(=O)NCCOCCOCCOCCOCCOCCOCCOCCNc1cccc2C(=O)N(C3CCC(=O)NC3=O)C(=O)c12	InChI=1S/C54H65F3N8O14/c1-63-15-17-64(18-16-63)44-10-9-38(33-43(44)61-50(69)40-35-60-47(67)34-41(40)54(55,56)57)36-5-7-37(8-6-36)49(68)59-14-20-74-22-24-76-26-28-78-30-32-79-31-29-77-27-25-75-23-21-73-19-13-58-42-4-2-3-39-48(42)53(72)65(52(39)71)45-11-12-46(66)62-51(45)70/h2-10,33-35,45,58H,11-32H2,1H3,(H,59,68)(H,60,67)(H,61,69)(H,62,66,70)	OPZUCPBYLOKUIE-UHFFFAOYSA-N	50601529	CHEMBL5176431	WD repeat-containing protein 5			 4920							ChEMBL		10.7270/Q20Z77B9	33980013			Dölle, A; Adhikari, B; Krämer, A; Weckesser, J; Berner, N; Berger, LM; Diebold, M; Szewczyk, MM; Barsyte-Lovejoy, D; Arrowsmith, CH; Gebel, J; Löhr, F; Dötsch, V; Eilers, M; Heinzlmeir, S; Kuster, B; Sotriffer, C; Wolf, E; Knapp, S	Goethe University Frankfurt am Main	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50601529	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50601529&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			168273097	482612381							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51492483	CN1CCN(CC1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(cc1)C(=O)NCc1ccc(CNc2ccc3C(=O)N(C4CCC(=O)NC4=O)C(=O)c3c2)cc1	InChI=1S/C46H41F3N8O7/c1-55-16-18-56(19-17-55)37-13-10-30(20-36(37)53-42(61)34-25-51-40(59)22-35(34)46(47,48)49)28-6-8-29(9-7-28)41(60)52-24-27-4-2-26(3-5-27)23-50-31-11-12-32-33(21-31)45(64)57(44(32)63)38-14-15-39(58)54-43(38)62/h2-13,20-22,25,38,50H,14-19,23-24H2,1H3,(H,51,59)(H,52,60)(H,53,61)(H,54,58,62)	PXGLQUOVJRNPQL-UHFFFAOYSA-N	50601530	CHEMBL5203844	WD repeat-containing protein 5			 1180							ChEMBL		10.7270/Q20Z77B9	33980013			Dölle, A; Adhikari, B; Krämer, A; Weckesser, J; Berner, N; Berger, LM; Diebold, M; Szewczyk, MM; Barsyte-Lovejoy, D; Arrowsmith, CH; Gebel, J; Löhr, F; Dötsch, V; Eilers, M; Heinzlmeir, S; Kuster, B; Sotriffer, C; Wolf, E; Knapp, S	Goethe University Frankfurt am Main	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50601530	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50601530&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			168293470	482612382							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51492484	CN1CCN(CC1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(cc1)C(=O)NCCOCCC(=O)N[C@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)NCc1ccc(cc1)-c1scnc1C)C(C)(C)C	InChI=1S/C52H60F3N9O8S/c1-31-45(73-30-59-31)34-8-6-32(7-9-34)27-58-49(70)42-25-37(65)29-64(42)50(71)46(51(2,3)4)61-43(66)16-22-72-23-17-56-47(68)35-12-10-33(11-13-35)36-14-15-41(63-20-18-62(5)19-21-63)40(24-36)60-48(69)38-28-57-44(67)26-39(38)52(53,54)55/h6-15,24,26,28,30,37,42,46,65H,16-23,25,27,29H2,1-5H3,(H,56,68)(H,57,67)(H,58,70)(H,60,69)(H,61,66)/t37-,42+,46-/m1/s1	WZJUOFSNOKPRHG-BQGOKDIQSA-N	50601518	CHEMBL5173110	WD repeat-containing protein 5			 8650							ChEMBL		10.7270/Q20Z77B9	33980013			Dölle, A; Adhikari, B; Krämer, A; Weckesser, J; Berner, N; Berger, LM; Diebold, M; Szewczyk, MM; Barsyte-Lovejoy, D; Arrowsmith, CH; Gebel, J; Löhr, F; Dötsch, V; Eilers, M; Heinzlmeir, S; Kuster, B; Sotriffer, C; Wolf, E; Knapp, S	Goethe University Frankfurt am Main	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50601518	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50601518&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			168274409	482612370							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51492485	CN1CCN(CC1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)c1ccc(cc1)-c1ccc(cc1)C(=O)NCCOCCOCCOCCOCCC(=O)N[C@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)NCc1ccc(cc1)-c1scnc1C)C(C)(C)C	InChI=1S/C58H72F3N9O11S/c1-37-51(82-36-65-37)41-8-6-38(7-9-41)32-64-55(76)47-30-44(71)34-70(47)56(77)52(57(2,3)4)67-49(72)18-22-78-24-26-80-28-29-81-27-25-79-23-19-62-53(74)42-12-10-39(11-13-42)40-14-16-43(17-15-40)69-21-20-68(5)48(35-69)66-54(75)45-33-63-50(73)31-46(45)58(59,60)61/h6-17,31,33,36,44,47-48,52,71H,18-30,32,34-35H2,1-5H3,(H,62,74)(H,63,73)(H,64,76)(H,66,75)(H,67,72)/t44-,47+,48?,52-/m1/s1	ACMVOJXLOLDHDX-XTVHMVLRSA-N	50601531	CHEMBL5184488	WD repeat-containing protein 5			 12500							ChEMBL		10.7270/Q20Z77B9	33980013			Dölle, A; Adhikari, B; Krämer, A; Weckesser, J; Berner, N; Berger, LM; Diebold, M; Szewczyk, MM; Barsyte-Lovejoy, D; Arrowsmith, CH; Gebel, J; Löhr, F; Dötsch, V; Eilers, M; Heinzlmeir, S; Kuster, B; Sotriffer, C; Wolf, E; Knapp, S	Goethe University Frankfurt am Main	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50601531	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50601531&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			168282158	482612383							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51492486	CN1CCN(CC1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(cc1)C(=O)N[C@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)NCc1ccc(cc1)-c1scnc1C)C(C)(C)C	InChI=1S/C47H51F3N8O6S/c1-27-40(65-26-53-27)30-8-6-28(7-9-30)23-52-44(63)38-21-33(59)25-58(38)45(64)41(46(2,3)4)55-42(61)31-12-10-29(11-13-31)32-14-15-37(57-18-16-56(5)17-19-57)36(20-32)54-43(62)34-24-51-39(60)22-35(34)47(48,49)50/h6-15,20,22,24,26,33,38,41,59H,16-19,21,23,25H2,1-5H3,(H,51,60)(H,52,63)(H,54,62)(H,55,61)/t33-,38+,41-/m1/s1	QAANVDJLUGLPQA-OEFLFKSQSA-N	50601532	CHEMBL5186486	WD repeat-containing protein 5			 1590							ChEMBL		10.7270/Q20Z77B9	33980013			Dölle, A; Adhikari, B; Krämer, A; Weckesser, J; Berner, N; Berger, LM; Diebold, M; Szewczyk, MM; Barsyte-Lovejoy, D; Arrowsmith, CH; Gebel, J; Löhr, F; Dötsch, V; Eilers, M; Heinzlmeir, S; Kuster, B; Sotriffer, C; Wolf, E; Knapp, S	Goethe University Frankfurt am Main	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50601532	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50601532&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			168279254	482612384							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51492487	CN1CCN(CC1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(cc1)C(=O)NCCCCC(=O)N[C@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)NCc1ccc(cc1)-c1scnc1C)C(C)(C)C	InChI=1S/C52H60F3N9O7S/c1-31-45(72-30-59-31)34-11-9-32(10-12-34)27-58-49(70)42-25-37(65)29-64(42)50(71)46(51(2,3)4)61-43(66)8-6-7-19-56-47(68)35-15-13-33(14-16-35)36-17-18-41(63-22-20-62(5)21-23-63)40(24-36)60-48(69)38-28-57-44(67)26-39(38)52(53,54)55/h9-18,24,26,28,30,37,42,46,65H,6-8,19-23,25,27,29H2,1-5H3,(H,56,68)(H,57,67)(H,58,70)(H,60,69)(H,61,66)/t37-,42+,46-/m1/s1	OFNZESNEBSQKSE-BQGOKDIQSA-N	50601521	CHEMBL5092273	WD repeat-containing protein 5			 13600							ChEMBL		10.7270/Q20Z77B9	33980013			Dölle, A; Adhikari, B; Krämer, A; Weckesser, J; Berner, N; Berger, LM; Diebold, M; Szewczyk, MM; Barsyte-Lovejoy, D; Arrowsmith, CH; Gebel, J; Löhr, F; Dötsch, V; Eilers, M; Heinzlmeir, S; Kuster, B; Sotriffer, C; Wolf, E; Knapp, S	Goethe University Frankfurt am Main	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50601521	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50601521&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	8KH		157049306	482612373							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51492488	CN1CCN(CC1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(cc1)C(=O)NCc1ccc(CC(=O)N[C@H](C(=O)N2C[C@H](O)C[C@H]2C(=O)NCc2ccc(cc2)-c2scnc2C)C(C)(C)C)cc1	InChI=1S/C56H60F3N9O7S/c1-33-49(76-32-63-33)38-12-10-36(11-13-38)29-62-53(74)46-26-41(69)31-68(46)54(75)50(55(2,3)4)65-48(71)24-34-6-8-35(9-7-34)28-61-51(72)39-16-14-37(15-17-39)40-18-19-45(67-22-20-66(5)21-23-67)44(25-40)64-52(73)42-30-60-47(70)27-43(42)56(57,58)59/h6-19,25,27,30,32,41,46,50,69H,20-24,26,28-29,31H2,1-5H3,(H,60,70)(H,61,72)(H,62,74)(H,64,73)(H,65,71)/t41-,46+,50-/m1/s1	PJYZWCPLYVFKHH-PNWJTEEHSA-N	50601524	CHEMBL5201006	WD repeat-containing protein 5			 15800							ChEMBL		10.7270/Q20Z77B9	33980013			Dölle, A; Adhikari, B; Krämer, A; Weckesser, J; Berner, N; Berger, LM; Diebold, M; Szewczyk, MM; Barsyte-Lovejoy, D; Arrowsmith, CH; Gebel, J; Löhr, F; Dötsch, V; Eilers, M; Heinzlmeir, S; Kuster, B; Sotriffer, C; Wolf, E; Knapp, S	Goethe University Frankfurt am Main	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50601524	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50601524&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			165416424	482612376							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51492489	CN1CCN(CC1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(CN2CCOCC2)cc1	InChI=1S/C29H32F3N5O3/c1-35-8-10-37(11-9-35)26-7-6-22(21-4-2-20(3-5-21)19-36-12-14-40-15-13-36)16-25(26)34-28(39)23-18-33-27(38)17-24(23)29(30,31)32/h2-7,16-18H,8-15,19H2,1H3,(H,33,38)(H,34,39)	GQTXDUXACYMXPD-UHFFFAOYSA-N	50601515	CHEMBL5194499	WD repeat-containing protein 5			 1850							ChEMBL		10.7270/Q20Z77B9	33980013			Dölle, A; Adhikari, B; Krämer, A; Weckesser, J; Berner, N; Berger, LM; Diebold, M; Szewczyk, MM; Barsyte-Lovejoy, D; Arrowsmith, CH; Gebel, J; Löhr, F; Dötsch, V; Eilers, M; Heinzlmeir, S; Kuster, B; Sotriffer, C; Wolf, E; Knapp, S	Goethe University Frankfurt am Main	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50601515	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50601515&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			168289697	482612367							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51492490	CN1CCN(CC1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(cc1)C(=O)OC(C)(C)C	InChI=1S/C29H31F3N4O4/c1-28(2,3)40-27(39)19-7-5-18(6-8-19)20-9-10-24(36-13-11-35(4)12-14-36)23(15-20)34-26(38)21-17-33-25(37)16-22(21)29(30,31)32/h5-10,15-17H,11-14H2,1-4H3,(H,33,37)(H,34,38)	HATZDQFMULXBFB-UHFFFAOYSA-N	50601516	CHEMBL5181586	WD repeat-containing protein 5			 80							ChEMBL		10.7270/Q20Z77B9	33980013			Dölle, A; Adhikari, B; Krämer, A; Weckesser, J; Berner, N; Berger, LM; Diebold, M; Szewczyk, MM; Barsyte-Lovejoy, D; Arrowsmith, CH; Gebel, J; Löhr, F; Dötsch, V; Eilers, M; Heinzlmeir, S; Kuster, B; Sotriffer, C; Wolf, E; Knapp, S	Goethe University Frankfurt am Main	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50601516	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50601516&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			168277961	482612368							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51492491	CN1CCN(CC1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(cc1)C(=O)NCCOCCNc1cccc2C(=O)N(C3CCC(=O)NC3=O)C(=O)c12	InChI=1S/C42H41F3N8O8/c1-51-15-17-52(18-16-51)32-10-9-26(21-31(32)49-38(57)28-23-48-35(55)22-29(28)42(43,44)45)24-5-7-25(8-6-24)37(56)47-14-20-61-19-13-46-30-4-2-3-27-36(30)41(60)53(40(27)59)33-11-12-34(54)50-39(33)58/h2-10,21-23,33,46H,11-20H2,1H3,(H,47,56)(H,48,55)(H,49,57)(H,50,54,58)	CCAKBASGLWLWPO-UHFFFAOYSA-N	50601517	CHEMBL5181611	WD repeat-containing protein 5			 990							ChEMBL		10.7270/Q20Z77B9	33980013			Dölle, A; Adhikari, B; Krämer, A; Weckesser, J; Berner, N; Berger, LM; Diebold, M; Szewczyk, MM; Barsyte-Lovejoy, D; Arrowsmith, CH; Gebel, J; Löhr, F; Dötsch, V; Eilers, M; Heinzlmeir, S; Kuster, B; Sotriffer, C; Wolf, E; Knapp, S	Goethe University Frankfurt am Main	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50601517	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50601517&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			168272844	482612369							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51492492	CN1CCN(CC1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(cc1)C(=O)NCCOCCOCCOCCNc1cccc2C(=O)N(C3CCC(=O)NC3=O)C(=O)c12	InChI=1S/C46H49F3N8O10/c1-55-15-17-56(18-16-55)36-10-9-30(25-35(36)53-42(61)32-27-52-39(59)26-33(32)46(47,48)49)28-5-7-29(8-6-28)41(60)51-14-20-66-22-24-67-23-21-65-19-13-50-34-4-2-3-31-40(34)45(64)57(44(31)63)37-11-12-38(58)54-43(37)62/h2-10,25-27,37,50H,11-24H2,1H3,(H,51,60)(H,52,59)(H,53,61)(H,54,58,62)	MPVUSWCQRFACNA-UHFFFAOYSA-N	50601527	CHEMBL5178796	WD repeat-containing protein 5			 1220							ChEMBL		10.7270/Q20Z77B9	33980013			Dölle, A; Adhikari, B; Krämer, A; Weckesser, J; Berner, N; Berger, LM; Diebold, M; Szewczyk, MM; Barsyte-Lovejoy, D; Arrowsmith, CH; Gebel, J; Löhr, F; Dötsch, V; Eilers, M; Heinzlmeir, S; Kuster, B; Sotriffer, C; Wolf, E; Knapp, S	Goethe University Frankfurt am Main	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50601527	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50601527&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			168274224	482612379							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51492493	CN1CCN(CC1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(cc1)C(=O)NCCOCCOCCOCCOCCOCCNc1cccc2C(=O)N(C3CCC(=O)NC3=O)C(=O)c12	InChI=1S/C50H57F3N8O12/c1-59-15-17-60(18-16-59)40-10-9-34(29-39(40)57-46(65)36-31-56-43(63)30-37(36)50(51,52)53)32-5-7-33(8-6-32)45(64)55-14-20-70-22-24-72-26-28-73-27-25-71-23-21-69-19-13-54-38-4-2-3-35-44(38)49(68)61(48(35)67)41-11-12-42(62)58-47(41)66/h2-10,29-31,41,54H,11-28H2,1H3,(H,55,64)(H,56,63)(H,57,65)(H,58,62,66)	DHDXVQJEEHRETI-UHFFFAOYSA-N	50601528	CHEMBL5176119	WD repeat-containing protein 5			 2870							ChEMBL		10.7270/Q20Z77B9	33980013			Dölle, A; Adhikari, B; Krämer, A; Weckesser, J; Berner, N; Berger, LM; Diebold, M; Szewczyk, MM; Barsyte-Lovejoy, D; Arrowsmith, CH; Gebel, J; Löhr, F; Dötsch, V; Eilers, M; Heinzlmeir, S; Kuster, B; Sotriffer, C; Wolf, E; Knapp, S	Goethe University Frankfurt am Main	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50601528	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50601528&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			168276134	482612380							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51492494	CN1CCN(CC1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(cc1)C(=O)NCCOCCOCCOCCOCCOCCOCCOCCNc1cccc2C(=O)N(C3CCC(=O)NC3=O)C(=O)c12	InChI=1S/C54H65F3N8O14/c1-63-15-17-64(18-16-63)44-10-9-38(33-43(44)61-50(69)40-35-60-47(67)34-41(40)54(55,56)57)36-5-7-37(8-6-36)49(68)59-14-20-74-22-24-76-26-28-78-30-32-79-31-29-77-27-25-75-23-21-73-19-13-58-42-4-2-3-39-48(42)53(72)65(52(39)71)45-11-12-46(66)62-51(45)70/h2-10,33-35,45,58H,11-32H2,1H3,(H,59,68)(H,60,67)(H,61,69)(H,62,66,70)	OPZUCPBYLOKUIE-UHFFFAOYSA-N	50601529	CHEMBL5176431	WD repeat-containing protein 5			 1050							ChEMBL		10.7270/Q20Z77B9	33980013			Dölle, A; Adhikari, B; Krämer, A; Weckesser, J; Berner, N; Berger, LM; Diebold, M; Szewczyk, MM; Barsyte-Lovejoy, D; Arrowsmith, CH; Gebel, J; Löhr, F; Dötsch, V; Eilers, M; Heinzlmeir, S; Kuster, B; Sotriffer, C; Wolf, E; Knapp, S	Goethe University Frankfurt am Main	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50601529	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50601529&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			168273097	482612381							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51492495	CN1CCN(CC1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(cc1)C(=O)NCc1ccc(CNc2ccc3C(=O)N(C4CCC(=O)NC4=O)C(=O)c3c2)cc1	InChI=1S/C46H41F3N8O7/c1-55-16-18-56(19-17-55)37-13-10-30(20-36(37)53-42(61)34-25-51-40(59)22-35(34)46(47,48)49)28-6-8-29(9-7-28)41(60)52-24-27-4-2-26(3-5-27)23-50-31-11-12-32-33(21-31)45(64)57(44(32)63)38-14-15-39(58)54-43(38)62/h2-13,20-22,25,38,50H,14-19,23-24H2,1H3,(H,51,59)(H,52,60)(H,53,61)(H,54,58,62)	PXGLQUOVJRNPQL-UHFFFAOYSA-N	50601530	CHEMBL5203844	WD repeat-containing protein 5			 850							ChEMBL		10.7270/Q20Z77B9	33980013			Dölle, A; Adhikari, B; Krämer, A; Weckesser, J; Berner, N; Berger, LM; Diebold, M; Szewczyk, MM; Barsyte-Lovejoy, D; Arrowsmith, CH; Gebel, J; Löhr, F; Dötsch, V; Eilers, M; Heinzlmeir, S; Kuster, B; Sotriffer, C; Wolf, E; Knapp, S	Goethe University Frankfurt am Main	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50601530	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50601530&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			168293470	482612382							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51492496	CN1CCN(CC1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(cc1)C(=O)NCCOCCC(=O)N[C@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)NCc1ccc(cc1)-c1scnc1C)C(C)(C)C	InChI=1S/C52H60F3N9O8S/c1-31-45(73-30-59-31)34-8-6-32(7-9-34)27-58-49(70)42-25-37(65)29-64(42)50(71)46(51(2,3)4)61-43(66)16-22-72-23-17-56-47(68)35-12-10-33(11-13-35)36-14-15-41(63-20-18-62(5)19-21-63)40(24-36)60-48(69)38-28-57-44(67)26-39(38)52(53,54)55/h6-15,24,26,28,30,37,42,46,65H,16-23,25,27,29H2,1-5H3,(H,56,68)(H,57,67)(H,58,70)(H,60,69)(H,61,66)/t37-,42+,46-/m1/s1	WZJUOFSNOKPRHG-BQGOKDIQSA-N	50601518	CHEMBL5173110	WD repeat-containing protein 5			 740							ChEMBL		10.7270/Q20Z77B9	33980013			Dölle, A; Adhikari, B; Krämer, A; Weckesser, J; Berner, N; Berger, LM; Diebold, M; Szewczyk, MM; Barsyte-Lovejoy, D; Arrowsmith, CH; Gebel, J; Löhr, F; Dötsch, V; Eilers, M; Heinzlmeir, S; Kuster, B; Sotriffer, C; Wolf, E; Knapp, S	Goethe University Frankfurt am Main	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50601518	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50601518&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			168274409	482612370							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51492497	CN1CCN(CC1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(cc1)C(=O)NCCOCCOCCC(=O)N[C@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)NCc1ccc(cc1)-c1scnc1C)C(C)(C)C	InChI=1S/C54H64F3N9O9S/c1-33-47(76-32-61-33)36-8-6-34(7-9-36)29-60-51(72)44-27-39(67)31-66(44)52(73)48(53(2,3)4)63-45(68)16-22-74-24-25-75-23-17-58-49(70)37-12-10-35(11-13-37)38-14-15-43(65-20-18-64(5)19-21-65)42(26-38)62-50(71)40-30-59-46(69)28-41(40)54(55,56)57/h6-15,26,28,30,32,39,44,48,67H,16-25,27,29,31H2,1-5H3,(H,58,70)(H,59,69)(H,60,72)(H,62,71)(H,63,68)/t39-,44+,48-/m1/s1	CTQDFWAQIJZIMB-UOHLUGTHSA-N	50601533	CHEMBL5171029	WD repeat-containing protein 5			 5210							ChEMBL		10.7270/Q20Z77B9	33980013			Dölle, A; Adhikari, B; Krämer, A; Weckesser, J; Berner, N; Berger, LM; Diebold, M; Szewczyk, MM; Barsyte-Lovejoy, D; Arrowsmith, CH; Gebel, J; Löhr, F; Dötsch, V; Eilers, M; Heinzlmeir, S; Kuster, B; Sotriffer, C; Wolf, E; Knapp, S	Goethe University Frankfurt am Main	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50601533	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50601533&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			168269703	482612385							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51492498	CN1CCN(CC1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)c1ccc(cc1)-c1ccc(cc1)C(=O)NCCOCCOCCOCCOCCC(=O)N[C@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)NCc1ccc(cc1)-c1scnc1C)C(C)(C)C	InChI=1S/C58H72F3N9O11S/c1-37-51(82-36-65-37)41-8-6-38(7-9-41)32-64-55(76)47-30-44(71)34-70(47)56(77)52(57(2,3)4)67-49(72)18-22-78-24-26-80-28-29-81-27-25-79-23-19-62-53(74)42-12-10-39(11-13-42)40-14-16-43(17-15-40)69-21-20-68(5)48(35-69)66-54(75)45-33-63-50(73)31-46(45)58(59,60)61/h6-17,31,33,36,44,47-48,52,71H,18-30,32,34-35H2,1-5H3,(H,62,74)(H,63,73)(H,64,76)(H,66,75)(H,67,72)/t44-,47+,48?,52-/m1/s1	ACMVOJXLOLDHDX-XTVHMVLRSA-N	50601531	CHEMBL5184488	WD repeat-containing protein 5			 1540							ChEMBL		10.7270/Q20Z77B9	33980013			Dölle, A; Adhikari, B; Krämer, A; Weckesser, J; Berner, N; Berger, LM; Diebold, M; Szewczyk, MM; Barsyte-Lovejoy, D; Arrowsmith, CH; Gebel, J; Löhr, F; Dötsch, V; Eilers, M; Heinzlmeir, S; Kuster, B; Sotriffer, C; Wolf, E; Knapp, S	Goethe University Frankfurt am Main	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50601531	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50601531&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			168282158	482612383							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51492499	CN1CCN(CC1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(cc1)C(=O)N[C@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)NCc1ccc(cc1)-c1scnc1C)C(C)(C)C	InChI=1S/C47H51F3N8O6S/c1-27-40(65-26-53-27)30-8-6-28(7-9-30)23-52-44(63)38-21-33(59)25-58(38)45(64)41(46(2,3)4)55-42(61)31-12-10-29(11-13-31)32-14-15-37(57-18-16-56(5)17-19-57)36(20-32)54-43(62)34-24-51-39(60)22-35(34)47(48,49)50/h6-15,20,22,24,26,33,38,41,59H,16-19,21,23,25H2,1-5H3,(H,51,60)(H,52,63)(H,54,62)(H,55,61)/t33-,38+,41-/m1/s1	QAANVDJLUGLPQA-OEFLFKSQSA-N	50601532	CHEMBL5186486	WD repeat-containing protein 5			 990							ChEMBL		10.7270/Q20Z77B9	33980013			Dölle, A; Adhikari, B; Krämer, A; Weckesser, J; Berner, N; Berger, LM; Diebold, M; Szewczyk, MM; Barsyte-Lovejoy, D; Arrowsmith, CH; Gebel, J; Löhr, F; Dötsch, V; Eilers, M; Heinzlmeir, S; Kuster, B; Sotriffer, C; Wolf, E; Knapp, S	Goethe University Frankfurt am Main	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50601532	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50601532&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			168279254	482612384							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51492500	CN1CCN(CC1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(cc1)C(=O)NCCC(=O)N[C@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)NCc1ccc(cc1)-c1scnc1C)C(C)(C)C	InChI=1S/C50H56F3N9O7S/c1-29-43(70-28-57-29)32-8-6-30(7-9-32)25-56-47(68)40-23-35(63)27-62(40)48(69)44(49(2,3)4)59-41(64)16-17-54-45(66)33-12-10-31(11-13-33)34-14-15-39(61-20-18-60(5)19-21-61)38(22-34)58-46(67)36-26-55-42(65)24-37(36)50(51,52)53/h6-15,22,24,26,28,35,40,44,63H,16-21,23,25,27H2,1-5H3,(H,54,66)(H,55,65)(H,56,68)(H,58,67)(H,59,64)/t35-,40+,44-/m1/s1	YOILXXMNXUOXLA-HOPMZIQWSA-N	50601519	CHEMBL5191015	WD repeat-containing protein 5			 3930							ChEMBL		10.7270/Q20Z77B9	33980013			Dölle, A; Adhikari, B; Krämer, A; Weckesser, J; Berner, N; Berger, LM; Diebold, M; Szewczyk, MM; Barsyte-Lovejoy, D; Arrowsmith, CH; Gebel, J; Löhr, F; Dötsch, V; Eilers, M; Heinzlmeir, S; Kuster, B; Sotriffer, C; Wolf, E; Knapp, S	Goethe University Frankfurt am Main	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50601519	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50601519&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			168285686	482612371							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51492501	CN1CCN(CC1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(cc1)C(=O)NCCCC(=O)N[C@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)NCc1ccc(cc1)-c1scnc1C)C(C)(C)C	InChI=1S/C51H58F3N9O7S/c1-30-44(71-29-58-30)33-10-8-31(9-11-33)26-57-48(69)41-24-36(64)28-63(41)49(70)45(50(2,3)4)60-42(65)7-6-18-55-46(67)34-14-12-32(13-15-34)35-16-17-40(62-21-19-61(5)20-22-62)39(23-35)59-47(68)37-27-56-43(66)25-38(37)51(52,53)54/h8-17,23,25,27,29,36,41,45,64H,6-7,18-22,24,26,28H2,1-5H3,(H,55,67)(H,56,66)(H,57,69)(H,59,68)(H,60,65)/t36-,41+,45-/m1/s1	KFCLTULBYCCZBG-LTJJNQLXSA-N	50601520	CHEMBL5185035	WD repeat-containing protein 5			 3290							ChEMBL		10.7270/Q20Z77B9	33980013			Dölle, A; Adhikari, B; Krämer, A; Weckesser, J; Berner, N; Berger, LM; Diebold, M; Szewczyk, MM; Barsyte-Lovejoy, D; Arrowsmith, CH; Gebel, J; Löhr, F; Dötsch, V; Eilers, M; Heinzlmeir, S; Kuster, B; Sotriffer, C; Wolf, E; Knapp, S	Goethe University Frankfurt am Main	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50601520	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50601520&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			165416423	482612372							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51492502	CN1CCN(CC1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(cc1)C(=O)NCCCCC(=O)N[C@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)NCc1ccc(cc1)-c1scnc1C)C(C)(C)C	InChI=1S/C52H60F3N9O7S/c1-31-45(72-30-59-31)34-11-9-32(10-12-34)27-58-49(70)42-25-37(65)29-64(42)50(71)46(51(2,3)4)61-43(66)8-6-7-19-56-47(68)35-15-13-33(14-16-35)36-17-18-41(63-22-20-62(5)21-23-63)40(24-36)60-48(69)38-28-57-44(67)26-39(38)52(53,54)55/h9-18,24,26,28,30,37,42,46,65H,6-8,19-23,25,27,29H2,1-5H3,(H,56,68)(H,57,67)(H,58,70)(H,60,69)(H,61,66)/t37-,42+,46-/m1/s1	OFNZESNEBSQKSE-BQGOKDIQSA-N	50601521	CHEMBL5092273	WD repeat-containing protein 5			 2150							ChEMBL		10.7270/Q20Z77B9	33980013			Dölle, A; Adhikari, B; Krämer, A; Weckesser, J; Berner, N; Berger, LM; Diebold, M; Szewczyk, MM; Barsyte-Lovejoy, D; Arrowsmith, CH; Gebel, J; Löhr, F; Dötsch, V; Eilers, M; Heinzlmeir, S; Kuster, B; Sotriffer, C; Wolf, E; Knapp, S	Goethe University Frankfurt am Main	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50601521	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50601521&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	8KH		157049306	482612373							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51492503	CN1CCN(CC1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(cc1)C(=O)NCCCCCC(=O)N[C@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)NCc1ccc(cc1)-c1scnc1C)C(C)(C)C	InChI=1S/C53H62F3N9O7S/c1-32-46(73-31-60-32)35-12-10-33(11-13-35)28-59-50(71)43-26-38(66)30-65(43)51(72)47(52(2,3)4)62-44(67)9-7-6-8-20-57-48(69)36-16-14-34(15-17-36)37-18-19-42(64-23-21-63(5)22-24-64)41(25-37)61-49(70)39-29-58-45(68)27-40(39)53(54,55)56/h10-19,25,27,29,31,38,43,47,66H,6-9,20-24,26,28,30H2,1-5H3,(H,57,69)(H,58,68)(H,59,71)(H,61,70)(H,62,67)/t38-,43+,47-/m1/s1	UPLJFUHLGRAYID-MXPJCAPISA-N	50601522	CHEMBL5186307	WD repeat-containing protein 5			 4950							ChEMBL		10.7270/Q20Z77B9	33980013			Dölle, A; Adhikari, B; Krämer, A; Weckesser, J; Berner, N; Berger, LM; Diebold, M; Szewczyk, MM; Barsyte-Lovejoy, D; Arrowsmith, CH; Gebel, J; Löhr, F; Dötsch, V; Eilers, M; Heinzlmeir, S; Kuster, B; Sotriffer, C; Wolf, E; Knapp, S	Goethe University Frankfurt am Main	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50601522	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50601522&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			168279616	482612374							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51492504	CN1CCN(CC1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(cc1)C(=O)NCCCCCCC(=O)N[C@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)NCc1ccc(cc1)-c1scnc1C)C(C)(C)C	InChI=1S/C54H64F3N9O7S/c1-33-47(74-32-61-33)36-13-11-34(12-14-36)29-60-51(72)44-27-39(67)31-66(44)52(73)48(53(2,3)4)63-45(68)10-8-6-7-9-21-58-49(70)37-17-15-35(16-18-37)38-19-20-43(65-24-22-64(5)23-25-65)42(26-38)62-50(71)40-30-59-46(69)28-41(40)54(55,56)57/h11-20,26,28,30,32,39,44,48,67H,6-10,21-25,27,29,31H2,1-5H3,(H,58,70)(H,59,69)(H,60,72)(H,62,71)(H,63,68)/t39-,44+,48-/m1/s1	BXKFHYMDHAHJSX-UOHLUGTHSA-N	50601523	CHEMBL5180413	WD repeat-containing protein 5			 15800							ChEMBL		10.7270/Q20Z77B9	33980013			Dölle, A; Adhikari, B; Krämer, A; Weckesser, J; Berner, N; Berger, LM; Diebold, M; Szewczyk, MM; Barsyte-Lovejoy, D; Arrowsmith, CH; Gebel, J; Löhr, F; Dötsch, V; Eilers, M; Heinzlmeir, S; Kuster, B; Sotriffer, C; Wolf, E; Knapp, S	Goethe University Frankfurt am Main	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50601523	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50601523&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			168276743	482612375							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51492505	CN1CCN(CC1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(cc1)C(=O)NCc1ccc(CC(=O)N[C@H](C(=O)N2C[C@H](O)C[C@H]2C(=O)NCc2ccc(cc2)-c2scnc2C)C(C)(C)C)cc1	InChI=1S/C56H60F3N9O7S/c1-33-49(76-32-63-33)38-12-10-36(11-13-38)29-62-53(74)46-26-41(69)31-68(46)54(75)50(55(2,3)4)65-48(71)24-34-6-8-35(9-7-34)28-61-51(72)39-16-14-37(15-17-39)40-18-19-45(67-22-20-66(5)21-23-67)44(25-40)64-52(73)42-30-60-47(70)27-43(42)56(57,58)59/h6-19,25,27,30,32,41,46,50,69H,20-24,26,28-29,31H2,1-5H3,(H,60,70)(H,61,72)(H,62,74)(H,64,73)(H,65,71)/t41-,46+,50-/m1/s1	PJYZWCPLYVFKHH-PNWJTEEHSA-N	50601524	CHEMBL5201006	WD repeat-containing protein 5			 2990							ChEMBL		10.7270/Q20Z77B9	33980013			Dölle, A; Adhikari, B; Krämer, A; Weckesser, J; Berner, N; Berger, LM; Diebold, M; Szewczyk, MM; Barsyte-Lovejoy, D; Arrowsmith, CH; Gebel, J; Löhr, F; Dötsch, V; Eilers, M; Heinzlmeir, S; Kuster, B; Sotriffer, C; Wolf, E; Knapp, S	Goethe University Frankfurt am Main	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50601524	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50601524&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			165416424	482612376							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51492465	CN1CCN(CC1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(CN2CCOCC2)cc1	InChI=1S/C29H32F3N5O3/c1-35-8-10-37(11-9-35)26-7-6-22(21-4-2-20(3-5-21)19-36-12-14-40-15-13-36)16-25(26)34-28(39)23-18-33-27(38)17-24(23)29(30,31)32/h2-7,16-18H,8-15,19H2,1H3,(H,33,38)(H,34,39)	GQTXDUXACYMXPD-UHFFFAOYSA-N	50601515	CHEMBL5194499	WD repeat-containing protein 5				 98000						ChEMBL		10.7270/Q20Z77B9	33980013			Dölle, A; Adhikari, B; Krämer, A; Weckesser, J; Berner, N; Berger, LM; Diebold, M; Szewczyk, MM; Barsyte-Lovejoy, D; Arrowsmith, CH; Gebel, J; Löhr, F; Dötsch, V; Eilers, M; Heinzlmeir, S; Kuster, B; Sotriffer, C; Wolf, E; Knapp, S	Goethe University Frankfurt am Main	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50601515	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50601515&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			168289697	482612367							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51492466	CN1CCN(CC1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(cc1)C(=O)OC(C)(C)C	InChI=1S/C29H31F3N4O4/c1-28(2,3)40-27(39)19-7-5-18(6-8-19)20-9-10-24(36-13-11-35(4)12-14-36)23(15-20)34-26(38)21-17-33-25(37)16-22(21)29(30,31)32/h5-10,15-17H,11-14H2,1-4H3,(H,33,37)(H,34,38)	HATZDQFMULXBFB-UHFFFAOYSA-N	50601516	CHEMBL5181586	WD repeat-containing protein 5				 25000						ChEMBL		10.7270/Q20Z77B9	33980013			Dölle, A; Adhikari, B; Krämer, A; Weckesser, J; Berner, N; Berger, LM; Diebold, M; Szewczyk, MM; Barsyte-Lovejoy, D; Arrowsmith, CH; Gebel, J; Löhr, F; Dötsch, V; Eilers, M; Heinzlmeir, S; Kuster, B; Sotriffer, C; Wolf, E; Knapp, S	Goethe University Frankfurt am Main	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50601516	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50601516&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			168277961	482612368							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51492467	CN1CCN(CC1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(cc1)C(=O)NCCOCCNc1cccc2C(=O)N(C3CCC(=O)NC3=O)C(=O)c12	InChI=1S/C42H41F3N8O8/c1-51-15-17-52(18-16-51)32-10-9-26(21-31(32)49-38(57)28-23-48-35(55)22-29(28)42(43,44)45)24-5-7-25(8-6-24)37(56)47-14-20-61-19-13-46-30-4-2-3-27-36(30)41(60)53(40(27)59)33-11-12-34(54)50-39(33)58/h2-10,21-23,33,46H,11-20H2,1H3,(H,47,56)(H,48,55)(H,49,57)(H,50,54,58)	CCAKBASGLWLWPO-UHFFFAOYSA-N	50601517	CHEMBL5181611	WD repeat-containing protein 5				 12000						ChEMBL		10.7270/Q20Z77B9	33980013			Dölle, A; Adhikari, B; Krämer, A; Weckesser, J; Berner, N; Berger, LM; Diebold, M; Szewczyk, MM; Barsyte-Lovejoy, D; Arrowsmith, CH; Gebel, J; Löhr, F; Dötsch, V; Eilers, M; Heinzlmeir, S; Kuster, B; Sotriffer, C; Wolf, E; Knapp, S	Goethe University Frankfurt am Main	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50601517	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50601517&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			168272844	482612369							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51492468	CN1CCN(CC1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(cc1)C(=O)NCCOCCC(=O)N[C@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)NCc1ccc(cc1)-c1scnc1C)C(C)(C)C	InChI=1S/C52H60F3N9O8S/c1-31-45(73-30-59-31)34-8-6-32(7-9-34)27-58-49(70)42-25-37(65)29-64(42)50(71)46(51(2,3)4)61-43(66)16-22-72-23-17-56-47(68)35-12-10-33(11-13-35)36-14-15-41(63-20-18-62(5)19-21-63)40(24-36)60-48(69)38-28-57-44(67)26-39(38)52(53,54)55/h6-15,24,26,28,30,37,42,46,65H,16-23,25,27,29H2,1-5H3,(H,56,68)(H,57,67)(H,58,70)(H,60,69)(H,61,66)/t37-,42+,46-/m1/s1	WZJUOFSNOKPRHG-BQGOKDIQSA-N	50601518	CHEMBL5173110	WD repeat-containing protein 5				 41000						ChEMBL		10.7270/Q20Z77B9	33980013			Dölle, A; Adhikari, B; Krämer, A; Weckesser, J; Berner, N; Berger, LM; Diebold, M; Szewczyk, MM; Barsyte-Lovejoy, D; Arrowsmith, CH; Gebel, J; Löhr, F; Dötsch, V; Eilers, M; Heinzlmeir, S; Kuster, B; Sotriffer, C; Wolf, E; Knapp, S	Goethe University Frankfurt am Main	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50601518	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50601518&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			168274409	482612370							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51492469	CN1CCN(CC1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(cc1)C(=O)NCCC(=O)N[C@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)NCc1ccc(cc1)-c1scnc1C)C(C)(C)C	InChI=1S/C50H56F3N9O7S/c1-29-43(70-28-57-29)32-8-6-30(7-9-32)25-56-47(68)40-23-35(63)27-62(40)48(69)44(49(2,3)4)59-41(64)16-17-54-45(66)33-12-10-31(11-13-33)34-14-15-39(61-20-18-60(5)19-21-61)38(22-34)58-46(67)36-26-55-42(65)24-37(36)50(51,52)53/h6-15,22,24,26,28,35,40,44,63H,16-21,23,25,27H2,1-5H3,(H,54,66)(H,55,65)(H,56,68)(H,58,67)(H,59,64)/t35-,40+,44-/m1/s1	YOILXXMNXUOXLA-HOPMZIQWSA-N	50601519	CHEMBL5191015	WD repeat-containing protein 5				 9000						ChEMBL		10.7270/Q20Z77B9	33980013			Dölle, A; Adhikari, B; Krämer, A; Weckesser, J; Berner, N; Berger, LM; Diebold, M; Szewczyk, MM; Barsyte-Lovejoy, D; Arrowsmith, CH; Gebel, J; Löhr, F; Dötsch, V; Eilers, M; Heinzlmeir, S; Kuster, B; Sotriffer, C; Wolf, E; Knapp, S	Goethe University Frankfurt am Main	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50601519	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50601519&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			168285686	482612371							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51492470	CN1CCN(CC1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(cc1)C(=O)NCCCC(=O)N[C@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)NCc1ccc(cc1)-c1scnc1C)C(C)(C)C	InChI=1S/C51H58F3N9O7S/c1-30-44(71-29-58-30)33-10-8-31(9-11-33)26-57-48(69)41-24-36(64)28-63(41)49(70)45(50(2,3)4)60-42(65)7-6-18-55-46(67)34-14-12-32(13-15-34)35-16-17-40(62-21-19-61(5)20-22-62)39(23-35)59-47(68)37-27-56-43(66)25-38(37)51(52,53)54/h8-17,23,25,27,29,36,41,45,64H,6-7,18-22,24,26,28H2,1-5H3,(H,55,67)(H,56,66)(H,57,69)(H,59,68)(H,60,65)/t36-,41+,45-/m1/s1	KFCLTULBYCCZBG-LTJJNQLXSA-N	50601520	CHEMBL5185035	WD repeat-containing protein 5				 6000						ChEMBL		10.7270/Q20Z77B9	33980013			Dölle, A; Adhikari, B; Krämer, A; Weckesser, J; Berner, N; Berger, LM; Diebold, M; Szewczyk, MM; Barsyte-Lovejoy, D; Arrowsmith, CH; Gebel, J; Löhr, F; Dötsch, V; Eilers, M; Heinzlmeir, S; Kuster, B; Sotriffer, C; Wolf, E; Knapp, S	Goethe University Frankfurt am Main	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50601520	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50601520&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			165416423	482612372							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51492471	CN1CCN(CC1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1ccc(cc1)C(=O)NCCCCC(=O)N[C@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)NCc1ccc(cc1)-c1scnc1C)C(C)(C)C	InChI=1S/C52H60F3N9O7S/c1-31-45(72-30-59-31)34-11-9-32(10-12-34)27-58-49(70)42-25-37(65)29-64(42)50(71)46(51(2,3)4)61-43(66)8-6-7-19-56-47(68)35-15-13-33(14-16-35)36-17-18-41(63-22-20-62(5)21-23-63)40(24-36)60-48(69)38-28-57-44(67)26-39(38)52(53,54)55/h9-18,24,26,28,30,37,42,46,65H,6-8,19-23,25,27,29H2,1-5H3,(H,56,68)(H,57,67)(H,58,70)(H,60,69)(H,61,66)/t37-,42+,46-/m1/s1	OFNZESNEBSQKSE-BQGOKDIQSA-N	50601521	CHEMBL5092273	WD repeat-containing protein 5				 18000						ChEMBL		10.7270/Q20Z77B9	33980013			Dölle, A; Adhikari, B; Krämer, A; Weckesser, J; Berner, N; Berger, LM; Diebold, M; Szewczyk, MM; Barsyte-Lovejoy, D; Arrowsmith, CH; Gebel, J; Löhr, F; Dötsch, V; Eilers, M; Heinzlmeir, S; Kuster, B; Sotriffer, C; Wolf, E; Knapp, S	Goethe University Frankfurt am Main	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50601521	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50601521&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	8KH		157049306	482612373							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51474526	OC(=O)c1ccc2n(cnc2c1)C1CCCCC1	InChI=1S/C14H16N2O2/c17-14(18)10-6-7-13-12(8-10)15-9-16(13)11-4-2-1-3-5-11/h6-9,11H,1-5H2,(H,17,18)	VDTQDVBTYFQIPB-UHFFFAOYSA-N	50137497	1-Cyclohexyl-1H-benzoimidazole-5-carboxylic acid::CHEMBL177122	WD repeat-containing protein 5				>20000000						ChEMBL		10.7270/Q2KD22XQ	34928151			de Esch, IJP; Erlanson, DA; Jahnke, W; Johnson, CN; Walsh, L	Vrije Universiteit Amsterdam	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50137497	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50137497&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	Q8G	6UHY	513903	104027663		CHEMBL177122				ZINC04638824	1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51474527	CS(=O)(=O)c1nc(NS(=O)(=O)c2cc(Br)cc(Cl)c2O)cn1C1CCCC1	InChI=1S/C15H17BrClN3O5S2/c1-26(22,23)15-18-13(8-20(15)10-4-2-3-5-10)19-27(24,25)12-7-9(16)6-11(17)14(12)21/h6-8,10,19,21H,2-5H2,1H3	ZBIVDOJYQHNICX-UHFFFAOYSA-N	50538305	CHEMBL4645862	WD repeat-containing protein 5				 100						ChEMBL		10.7270/Q2KD22XQ	34928151			de Esch, IJP; Erlanson, DA; Jahnke, W; Johnson, CN; Walsh, L	Vrije Universiteit Amsterdam	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50538305	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50538305&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	QF1	6UOZ	146019259	442139868							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51493608	CN(C(=O)c1cc(N)c(F)c(C)c1Cl)c1cc(ccc1N1CCN(C)CC1)C(=O)Oc1ccccc1	InChI=1S/C27H28ClFN4O3/c1-17-24(28)20(16-21(30)25(17)29)26(34)32(3)23-15-18(27(35)36-19-7-5-4-6-8-19)9-10-22(23)33-13-11-31(2)12-14-33/h4-10,15-16H,11-14,30H2,1-3H3	YVIIFQWVNDENNM-UHFFFAOYSA-N	50601693	CHEMBL5198658	WD repeat-containing protein 5			 26							ChEMBL		10.7270/Q2B85D61	34283608			Chen, X; Xu, J; Wang, X; Long, G; You, Q; Guo, X	China Pharmaceutical University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50601693	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50601693&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			168289079	482612544							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51493609	CN1CCN(CC1)c1ccc(cc1NC(=O)c1ccccc1Cl)[N+]([O-])=O	InChI=1S/C18H19ClN4O3/c1-21-8-10-22(11-9-21)17-7-6-13(23(25)26)12-16(17)20-18(24)14-4-2-3-5-15(14)19/h2-7,12H,8-11H2,1H3,(H,20,24)	WOGZFCMBPXJNFI-UHFFFAOYSA-N	50428254	CHEMBL1609857	WD repeat-containing protein 5				 4000						ChEMBL		10.7270/Q2B85D61	34283608			Chen, X; Xu, J; Wang, X; Long, G; You, Q; Guo, X	China Pharmaceutical University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50428254	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50428254&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	NP7	3SMR	2965974	164157129		CHEMBL1609857				ZINC05049228	1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51493610	CN1CCN(CC1)c1ccc(cc1NC(=O)c1cc(N)c(F)c(C)c1Cl)-c1ccc(cc1)C(=O)NCCCN	InChI=1S/C29H34ClFN6O2/c1-18-26(30)22(17-23(33)27(18)31)29(39)35-24-16-21(8-9-25(24)37-14-12-36(2)13-15-37)19-4-6-20(7-5-19)28(38)34-11-3-10-32/h4-9,16-17H,3,10-15,32-33H2,1-2H3,(H,34,38)(H,35,39)	OGLREAITVXTJOM-UHFFFAOYSA-N	50601692	CHEMBL5172154	WD repeat-containing protein 5				 14						ChEMBL		10.7270/Q2B85D61	34283608			Chen, X; Xu, J; Wang, X; Long, G; You, Q; Guo, X	China Pharmaceutical University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50601692	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50601692&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			168269940	482612543							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51493613	CN1CCN(CC1)c1ccc(cc1NC(=O)c1cc(N)c(F)c(C)c1Cl)-c1ccc(NC(=O)CCCCCNC(=O)CCCC[C@@H]2SC[C@@H]3NC(=O)N[C@H]23)cc1	InChI=1S/C41H52ClFN8O4S/c1-25-37(42)29(23-30(44)38(25)43)40(54)47-31-22-27(13-16-33(31)51-20-18-50(2)19-21-51)26-11-14-28(15-12-26)46-36(53)10-4-3-7-17-45-35(52)9-6-5-8-34-39-32(24-56-34)48-41(55)49-39/h11-16,22-23,32,34,39H,3-10,17-21,24,44H2,1-2H3,(H,45,52)(H,46,53)(H,47,54)(H2,48,49,55)/t32-,34-,39-/m0/s1	VPTAKNRDGAVVAF-WQLQHLIKSA-N	50601695	CHEMBL5179283	WD repeat-containing protein 5			 17							ChEMBL		10.7270/Q2B85D61	34283608			Chen, X; Xu, J; Wang, X; Long, G; You, Q; Guo, X	China Pharmaceutical University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50601695	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50601695&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			168272259	482612546							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51502272	CC[C@@H]1NC(=O)[C@H](CCCNC(=N)NC)NC(=O)[C@@](C)(CCNC(=O)[C@H](NC1=O)c1ccccc1)NC(=O)C(C)C	InChI=1S/C28H44N8O5/c1-6-19-23(38)35-21(18-11-8-7-9-12-18)25(40)31-16-14-28(4,36-22(37)17(2)3)26(41)34-20(24(39)33-19)13-10-15-32-27(29)30-5/h7-9,11-12,17,19-21H,6,10,13-16H2,1-5H3,(H,31,40)(H,33,39)(H,34,41)(H,35,38)(H,36,37)(H3,29,30,32)/t19-,20-,21+,28+/m0/s1	ZAIPJVQTYUSDTG-LDFBIXNTSA-N	50605317	CHEMBL4116919	WD repeat-containing protein 5		<1.000000								ChEMBL		10.7270/Q2JQ153M	35436124			Teuscher, KB; Meyers, KM; Wei, Q; Mills, JJ; Tian, J; Alvarado, J; Sai, J; Van Meveren, M; South, TM; Rietz, TA; Zhao, B; Moore, WJ; Stott, GM; Tansey, WP; Lee, T; Fesik, SW	Frederick National Laboratory for Cancer Research	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50605317	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50605317&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	9BA		129010138	482616168							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51502273	CN1CCN(CC1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cccc(CN2CCOCC2)c1	InChI=1S/C29H32F3N5O3/c1-35-7-9-37(10-8-35)26-6-5-22(21-4-2-3-20(15-21)19-36-11-13-40-14-12-36)16-25(26)34-28(39)23-18-33-27(38)17-24(23)29(30,31)32/h2-6,15-18H,7-14,19H2,1H3,(H,33,38)(H,34,39)	DJOVLOYCGXNVPI-UHFFFAOYSA-N	50164794	CHEMBL3798846::US11174250, Example Table4.1.1::US11319299, Comp. No. 57	WD repeat-containing protein 5				 30						ChEMBL		10.7270/Q2JQ153M	35436124			Teuscher, KB; Meyers, KM; Wei, Q; Mills, JJ; Tian, J; Alvarado, J; Sai, J; Van Meveren, M; South, TM; Rietz, TA; Zhao, B; Moore, WJ; Stott, GM; Tansey, WP; Lee, T; Fesik, SW	Frederick National Laboratory for Cancer Research	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50164794	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50164794&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	35Q	4QL1	91623360	341097539		CHEMBL3798846					1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51502274	CN1CCN(CC1)c1ccc(cc1NC(=O)c1cc(N)c(F)c(C)c1Cl)-n1cc(nn1)C(=O)NCCCN1CCOCC1	InChI=1S/C29H37ClFN9O3/c1-19-26(30)21(17-22(32)27(19)31)28(41)34-23-16-20(4-5-25(23)39-10-8-37(2)9-11-39)40-18-24(35-36-40)29(42)33-6-3-7-38-12-14-43-15-13-38/h4-5,16-18H,3,6-15,32H2,1-2H3,(H,33,42)(H,34,41)	MPTAUAHHFUFKAG-UHFFFAOYSA-N	50574672	CHEMBL4861912	WD repeat-containing protein 5			<10.0							ChEMBL		10.7270/Q2JQ153M	35436124			Teuscher, KB; Meyers, KM; Wei, Q; Mills, JJ; Tian, J; Alvarado, J; Sai, J; Van Meveren, M; South, TM; Rietz, TA; Zhao, B; Moore, WJ; Stott, GM; Tansey, WP; Lee, T; Fesik, SW	Frederick National Laboratory for Cancer Research	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50574672	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50574672&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			156112343	471064817							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51502275	COc1cc(CN2CCc3c(cc(Cn4ccn(C)c4=N)cc3-c3ccc(F)cc3C)C2=O)cc(OC)c1	InChI=1S/C30H31FN4O3/c1-19-11-22(31)5-6-25(19)27-14-21(18-35-10-9-33(2)30(35)32)15-28-26(27)7-8-34(29(28)36)17-20-12-23(37-3)16-24(13-20)38-4/h5-6,9-16,32H,7-8,17-18H2,1-4H3	PKONCIPMLLIAIL-UHFFFAOYSA-N	50520131	CHEMBL4588661	WD repeat-containing protein 5		<0.020000								ChEMBL		10.7270/Q2JQ153M	35436124			Teuscher, KB; Meyers, KM; Wei, Q; Mills, JJ; Tian, J; Alvarado, J; Sai, J; Van Meveren, M; South, TM; Rietz, TA; Zhao, B; Moore, WJ; Stott, GM; Tansey, WP; Lee, T; Fesik, SW	Frederick National Laboratory for Cancer Research	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50520131	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50520131&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146014479	440728713							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51502276	COc1cc(CN2CCc3c(cc(Cn4ccn(C)c4=N)cc3-c3ccc(F)cc3OC)C2=O)cc(OC)c1	InChI=1S/C30H31FN4O4/c1-33-9-10-35(30(33)32)18-20-13-26(25-6-5-21(31)15-28(25)39-4)24-7-8-34(29(36)27(24)14-20)17-19-11-22(37-2)16-23(12-19)38-3/h5-6,9-16,32H,7-8,17-18H2,1-4H3	DVRXVJVTWZDGSC-UHFFFAOYSA-N	50605318	CHEMBL5171315	WD repeat-containing protein 5		 0.033000								ChEMBL		10.7270/Q2JQ153M	35436124			Teuscher, KB; Meyers, KM; Wei, Q; Mills, JJ; Tian, J; Alvarado, J; Sai, J; Van Meveren, M; South, TM; Rietz, TA; Zhao, B; Moore, WJ; Stott, GM; Tansey, WP; Lee, T; Fesik, SW	Frederick National Laboratory for Cancer Research	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50605318	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50605318&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			168269455	482616169							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51502277	COc1cc(CN2CCc3c(cc(Cn4ccn(C)c4=N)cc3-c3ccc(F)cc3O)C2=O)cc(OC)c1	InChI=1S/C29H29FN4O4/c1-32-8-9-34(29(32)31)17-19-12-25(24-5-4-20(30)14-27(24)35)23-6-7-33(28(36)26(23)13-19)16-18-10-21(37-2)15-22(11-18)38-3/h4-5,8-15,31,35H,6-7,16-17H2,1-3H3	FOTQAEWSOCFZJP-UHFFFAOYSA-N	50605319	CHEMBL5171953	WD repeat-containing protein 5		 0.035000								ChEMBL		10.7270/Q2JQ153M	35436124			Teuscher, KB; Meyers, KM; Wei, Q; Mills, JJ; Tian, J; Alvarado, J; Sai, J; Van Meveren, M; South, TM; Rietz, TA; Zhao, B; Moore, WJ; Stott, GM; Tansey, WP; Lee, T; Fesik, SW	Frederick National Laboratory for Cancer Research	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50605319	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50605319&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			168270643	482616170							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51502278	COc1cc(CN2CCc3c(cc(Cn4ccn(C)c4=N)cc3-c3cccnc3C)C2=O)cc(OC)c1	InChI=1S/C29H31N5O3/c1-19-24(6-5-8-31-19)26-14-21(18-34-11-10-32(2)29(34)30)15-27-25(26)7-9-33(28(27)35)17-20-12-22(36-3)16-23(13-20)37-4/h5-6,8,10-16,30H,7,9,17-18H2,1-4H3	ISDXSXRXQJIJGT-UHFFFAOYSA-N	50605320	CHEMBL5202878	WD repeat-containing protein 5		 0.036000								ChEMBL		10.7270/Q2JQ153M	35436124			Teuscher, KB; Meyers, KM; Wei, Q; Mills, JJ; Tian, J; Alvarado, J; Sai, J; Van Meveren, M; South, TM; Rietz, TA; Zhao, B; Moore, WJ; Stott, GM; Tansey, WP; Lee, T; Fesik, SW	Frederick National Laboratory for Cancer Research	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50605320	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50605320&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			168293846	482616171							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51502279	COc1cc(CN2CCc3c(cc(Cn4ccn(C)c4=N)cc3-c3cccnc3OC)C2=O)cc(OC)c1	InChI=1S/C29H31N5O4/c1-32-10-11-34(29(32)30)18-20-14-25(24-6-5-8-31-27(24)38-4)23-7-9-33(28(35)26(23)15-20)17-19-12-21(36-2)16-22(13-19)37-3/h5-6,8,10-16,30H,7,9,17-18H2,1-4H3	SCAVCMXGKQTZFE-UHFFFAOYSA-N	50605321	CHEMBL5182077	WD repeat-containing protein 5		 0.055000								ChEMBL		10.7270/Q2JQ153M	35436124			Teuscher, KB; Meyers, KM; Wei, Q; Mills, JJ; Tian, J; Alvarado, J; Sai, J; Van Meveren, M; South, TM; Rietz, TA; Zhao, B; Moore, WJ; Stott, GM; Tansey, WP; Lee, T; Fesik, SW	Frederick National Laboratory for Cancer Research	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50605321	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50605321&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			168273867	482616172							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51502280	COc1cc(CN2CCc3c(cc(Cn4ccn(C)c4=N)cc3-c3cc(C)cnc3C)C2=O)cc(OC)c1	InChI=1S/C30H33N5O3/c1-19-10-26(20(2)32-16-19)27-13-22(18-35-9-8-33(3)30(35)31)14-28-25(27)6-7-34(29(28)36)17-21-11-23(37-4)15-24(12-21)38-5/h8-16,31H,6-7,17-18H2,1-5H3	OABHMYNMKKCFRT-UHFFFAOYSA-N	50605322	CHEMBL5169425	WD repeat-containing protein 5		 0.022000								ChEMBL		10.7270/Q2JQ153M	35436124			Teuscher, KB; Meyers, KM; Wei, Q; Mills, JJ; Tian, J; Alvarado, J; Sai, J; Van Meveren, M; South, TM; Rietz, TA; Zhao, B; Moore, WJ; Stott, GM; Tansey, WP; Lee, T; Fesik, SW	Frederick National Laboratory for Cancer Research	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50605322	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50605322&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			168270681	482616173							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51502281	COc1cc(CN2CCc3c(cc(Cn4ccn(C)c4=N)cc3-c3cccnc3C(F)(F)F)C2=O)cc(OC)c1	InChI=1S/C29H28F3N5O3/c1-35-9-10-37(28(35)33)17-19-13-24(23-5-4-7-34-26(23)29(30,31)32)22-6-8-36(27(38)25(22)14-19)16-18-11-20(39-2)15-21(12-18)40-3/h4-5,7,9-15,33H,6,8,16-17H2,1-3H3	NYVNNSYIUNCYFG-UHFFFAOYSA-N	50605323	CHEMBL5174357	WD repeat-containing protein 5		<0.020000								ChEMBL		10.7270/Q2JQ153M	35436124			Teuscher, KB; Meyers, KM; Wei, Q; Mills, JJ; Tian, J; Alvarado, J; Sai, J; Van Meveren, M; South, TM; Rietz, TA; Zhao, B; Moore, WJ; Stott, GM; Tansey, WP; Lee, T; Fesik, SW	Frederick National Laboratory for Cancer Research	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50605323	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50605323&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			153572423	482616174							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51502282	COc1cc(CN2CCc3c(cc(Cn4ccn(C)c4=N)cc3-c3ccncc3C)C2=O)cc(OC)c1	InChI=1S/C29H31N5O3/c1-19-16-31-7-5-24(19)26-13-21(18-34-10-9-32(2)29(34)30)14-27-25(26)6-8-33(28(27)35)17-20-11-22(36-3)15-23(12-20)37-4/h5,7,9-16,30H,6,8,17-18H2,1-4H3	LQPXGTDDZRBHBY-UHFFFAOYSA-N	50605324	CHEMBL5182982	WD repeat-containing protein 5		 0.029000								ChEMBL		10.7270/Q2JQ153M	35436124			Teuscher, KB; Meyers, KM; Wei, Q; Mills, JJ; Tian, J; Alvarado, J; Sai, J; Van Meveren, M; South, TM; Rietz, TA; Zhao, B; Moore, WJ; Stott, GM; Tansey, WP; Lee, T; Fesik, SW	Frederick National Laboratory for Cancer Research	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50605324	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50605324&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			168281685	482616175							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51502283	COc1cc(CN2CCc3c(cc(Cn4ccn(C)c4=N)cc3-c3cc(C)ncc3C)C2=O)cc(OC)c1	InChI=1S/C30H33N5O3/c1-19-16-32-20(2)10-26(19)27-13-22(18-35-9-8-33(3)30(35)31)14-28-25(27)6-7-34(29(28)36)17-21-11-23(37-4)15-24(12-21)38-5/h8-16,31H,6-7,17-18H2,1-5H3	YANGZQLKLWLJSK-UHFFFAOYSA-N	50605325	CHEMBL5199203	WD repeat-containing protein 5		<0.020000								ChEMBL		10.7270/Q2JQ153M	35436124			Teuscher, KB; Meyers, KM; Wei, Q; Mills, JJ; Tian, J; Alvarado, J; Sai, J; Van Meveren, M; South, TM; Rietz, TA; Zhao, B; Moore, WJ; Stott, GM; Tansey, WP; Lee, T; Fesik, SW	Frederick National Laboratory for Cancer Research	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50605325	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50605325&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			168291826	482616176							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51502284	COc1cc(CN2CCc3c(cc(Cn4ccn(C)c4=N)cc3C2=O)-c2conc2C)cc(OC)c1	InChI=1S/C27H29N5O4/c1-17-25(16-36-29-17)23-11-19(15-32-8-7-30(2)27(32)28)12-24-22(23)5-6-31(26(24)33)14-18-9-20(34-3)13-21(10-18)35-4/h7-13,16,28H,5-6,14-15H2,1-4H3	YFBKQFHRTNARGY-UHFFFAOYSA-N	50605326	CHEMBL5206455	WD repeat-containing protein 5		 0.046000								ChEMBL		10.7270/Q2JQ153M	35436124			Teuscher, KB; Meyers, KM; Wei, Q; Mills, JJ; Tian, J; Alvarado, J; Sai, J; Van Meveren, M; South, TM; Rietz, TA; Zhao, B; Moore, WJ; Stott, GM; Tansey, WP; Lee, T; Fesik, SW	Frederick National Laboratory for Cancer Research	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50605326	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50605326&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			168294577	482616177							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51502285	COc1cc(CN2CCc3c(cc(Cn4ccn(C)c4=N)cc3C2=O)-c2cn(C)nc2C)cc(OC)c1	InChI=1S/C28H32N6O3/c1-18-26(17-32(3)30-18)24-12-20(16-34-9-8-31(2)28(34)29)13-25-23(24)6-7-33(27(25)35)15-19-10-21(36-4)14-22(11-19)37-5/h8-14,17,29H,6-7,15-16H2,1-5H3	RSZACBCSSWKYIC-UHFFFAOYSA-N	50605327	CHEMBL5181314	WD repeat-containing protein 5		 0.023000								ChEMBL		10.7270/Q2JQ153M	35436124			Teuscher, KB; Meyers, KM; Wei, Q; Mills, JJ; Tian, J; Alvarado, J; Sai, J; Van Meveren, M; South, TM; Rietz, TA; Zhao, B; Moore, WJ; Stott, GM; Tansey, WP; Lee, T; Fesik, SW	Frederick National Laboratory for Cancer Research	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50605327	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50605327&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			153572276	482616178							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51502286	COc1cc(CN2CCc3c(cc(Cn4ccn(C)c4=N)cc3C2=O)-c2c(C)nn(C)c2C)cc(OC)c1	InChI=1S/C29H34N6O3/c1-18-27(19(2)33(4)31-18)25-13-21(17-35-10-9-32(3)29(35)30)14-26-24(25)7-8-34(28(26)36)16-20-11-22(37-5)15-23(12-20)38-6/h9-15,30H,7-8,16-17H2,1-6H3	YJBFAEKIPXLKCN-UHFFFAOYSA-N	50605328	CHEMBL5199310	WD repeat-containing protein 5		 0.210000								ChEMBL		10.7270/Q2JQ153M	35436124			Teuscher, KB; Meyers, KM; Wei, Q; Mills, JJ; Tian, J; Alvarado, J; Sai, J; Van Meveren, M; South, TM; Rietz, TA; Zhao, B; Moore, WJ; Stott, GM; Tansey, WP; Lee, T; Fesik, SW	Frederick National Laboratory for Cancer Research	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50605328	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50605328&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			153572559	482616179							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51502287	COc1cc(CN2CCc3c(cc(Cn4ccn(C)c4=N)cc3C2=O)-c2cc(C)nn2C)cc(OC)c1	InChI=1S/C28H32N6O3/c1-18-10-26(32(3)30-18)24-13-20(17-34-9-8-31(2)28(34)29)14-25-23(24)6-7-33(27(25)35)16-19-11-21(36-4)15-22(12-19)37-5/h8-15,29H,6-7,16-17H2,1-5H3	GSPVNRNVCGLYPV-UHFFFAOYSA-N	50605329	CHEMBL5186072	WD repeat-containing protein 5		 0.025000								ChEMBL		10.7270/Q2JQ153M	35436124			Teuscher, KB; Meyers, KM; Wei, Q; Mills, JJ; Tian, J; Alvarado, J; Sai, J; Van Meveren, M; South, TM; Rietz, TA; Zhao, B; Moore, WJ; Stott, GM; Tansey, WP; Lee, T; Fesik, SW	Frederick National Laboratory for Cancer Research	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50605329	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50605329&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			168281439	482616180							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51502288	COc1cc(CN2CCc3c(cc(Cn4ccn(C)c4=N)cc3C2=O)-c2cn(C)nc2C(F)(F)F)cc(OC)c1	InChI=1S/C28H29F3N6O3/c1-34-7-8-37(27(34)32)15-18-11-22(24-16-35(2)33-25(24)28(29,30)31)21-5-6-36(26(38)23(21)12-18)14-17-9-19(39-3)13-20(10-17)40-4/h7-13,16,32H,5-6,14-15H2,1-4H3	RHEVHQUBLKDXBF-UHFFFAOYSA-N	50605330	CHEMBL5201192	WD repeat-containing protein 5		<0.020000								ChEMBL		10.7270/Q2JQ153M	35436124			Teuscher, KB; Meyers, KM; Wei, Q; Mills, JJ; Tian, J; Alvarado, J; Sai, J; Van Meveren, M; South, TM; Rietz, TA; Zhao, B; Moore, WJ; Stott, GM; Tansey, WP; Lee, T; Fesik, SW	Frederick National Laboratory for Cancer Research	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50605330	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50605330&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			153572427	482616181							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51502289	CCn1cc(c(n1)C(F)(F)F)-c1cc(Cn2ccn(C)c2=N)cc2C(=O)N(Cc3cc(OC)cc(OC)c3)CCc12	InChI=1S/C29H31F3N6O3/c1-5-38-17-25(26(34-38)29(30,31)32)23-12-19(16-37-9-8-35(2)28(37)33)13-24-22(23)6-7-36(27(24)39)15-18-10-20(40-3)14-21(11-18)41-4/h8-14,17,33H,5-7,15-16H2,1-4H3	XQKWUJVZVJKWFS-UHFFFAOYSA-N	50605331	CHEMBL5190578	WD repeat-containing protein 5		<0.020000								ChEMBL		10.7270/Q2JQ153M	35436124			Teuscher, KB; Meyers, KM; Wei, Q; Mills, JJ; Tian, J; Alvarado, J; Sai, J; Van Meveren, M; South, TM; Rietz, TA; Zhao, B; Moore, WJ; Stott, GM; Tansey, WP; Lee, T; Fesik, SW	Frederick National Laboratory for Cancer Research	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50605331	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50605331&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			168281603	482616182							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51502290	COc1cc(CN2CCc3c(cc(Cn4ccnc4)cc3C2=O)-c2cn(C)nc2C(F)(F)F)cc(OC)c1	InChI=1S/C27H26F3N5O3/c1-33-15-24(25(32-33)27(28,29)30)22-10-18(13-34-7-5-31-16-34)11-23-21(22)4-6-35(26(23)36)14-17-8-19(37-2)12-20(9-17)38-3/h5,7-12,15-16H,4,6,13-14H2,1-3H3	KDFFNVCQAAKSPX-UHFFFAOYSA-N	50605332	CHEMBL5195031	WD repeat-containing protein 5		<0.020000								ChEMBL		10.7270/Q2JQ153M	35436124			Teuscher, KB; Meyers, KM; Wei, Q; Mills, JJ; Tian, J; Alvarado, J; Sai, J; Van Meveren, M; South, TM; Rietz, TA; Zhao, B; Moore, WJ; Stott, GM; Tansey, WP; Lee, T; Fesik, SW	Frederick National Laboratory for Cancer Research	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50605332	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50605332&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			168285855	482616183							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51502291	COc1cc(CN2CCc3c(cc(Cn4cccn4)cc3C2=O)-c2cn(C)nc2C(F)(F)F)cc(OC)c1	InChI=1S/C27H26F3N5O3/c1-33-16-24(25(32-33)27(28,29)30)22-11-18(15-35-7-4-6-31-35)12-23-21(22)5-8-34(26(23)36)14-17-9-19(37-2)13-20(10-17)38-3/h4,6-7,9-13,16H,5,8,14-15H2,1-3H3	BBJZSIAMRDBCHT-UHFFFAOYSA-N	50605333	CHEMBL5184980	WD repeat-containing protein 5		>6.7								ChEMBL		10.7270/Q2JQ153M	35436124			Teuscher, KB; Meyers, KM; Wei, Q; Mills, JJ; Tian, J; Alvarado, J; Sai, J; Van Meveren, M; South, TM; Rietz, TA; Zhao, B; Moore, WJ; Stott, GM; Tansey, WP; Lee, T; Fesik, SW	Frederick National Laboratory for Cancer Research	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50605333	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50605333&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			168283797	482616184							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51502292	COc1cc(CN2CCc3c(cc(Cn4cccc4)cc3C2=O)-c2cn(C)nc2C(F)(F)F)cc(OC)c1	InChI=1S/C28H27F3N4O3/c1-33-17-25(26(32-33)28(29,30)31)23-12-19(15-34-7-4-5-8-34)13-24-22(23)6-9-35(27(24)36)16-18-10-20(37-2)14-21(11-18)38-3/h4-5,7-8,10-14,17H,6,9,15-16H2,1-3H3	OINVJVRDEFGPHI-UHFFFAOYSA-N	50605334	CHEMBL5201482	WD repeat-containing protein 5		>6.7								ChEMBL		10.7270/Q2JQ153M	35436124			Teuscher, KB; Meyers, KM; Wei, Q; Mills, JJ; Tian, J; Alvarado, J; Sai, J; Van Meveren, M; South, TM; Rietz, TA; Zhao, B; Moore, WJ; Stott, GM; Tansey, WP; Lee, T; Fesik, SW	Frederick National Laboratory for Cancer Research	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50605334	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50605334&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			168291877	482616185							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51502293	COc1cc(CN2CCc3c(cc(Cn4cnnc4)cc3C2=O)-c2cn(C)nc2C(F)(F)F)cc(OC)c1	InChI=1S/C26H25F3N6O3/c1-33-13-23(24(32-33)26(27,28)29)21-8-17(11-34-14-30-31-15-34)9-22-20(21)4-5-35(25(22)36)12-16-6-18(37-2)10-19(7-16)38-3/h6-10,13-15H,4-5,11-12H2,1-3H3	JTNDJAJCJJIOTQ-UHFFFAOYSA-N	50605335	CHEMBL5190488	WD repeat-containing protein 5		 6.5								ChEMBL		10.7270/Q2JQ153M	35436124			Teuscher, KB; Meyers, KM; Wei, Q; Mills, JJ; Tian, J; Alvarado, J; Sai, J; Van Meveren, M; South, TM; Rietz, TA; Zhao, B; Moore, WJ; Stott, GM; Tansey, WP; Lee, T; Fesik, SW	Frederick National Laboratory for Cancer Research	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50605335	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50605335&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			168280112	482616186							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51502294	COc1cc(CN2CCc3c(cc(Cn4ccnc4C)cc3C2=O)-c2cn(C)nc2C(F)(F)F)cc(OC)c1	InChI=1S/C28H28F3N5O3/c1-17-32-6-8-35(17)14-19-11-23(25-16-34(2)33-26(25)28(29,30)31)22-5-7-36(27(37)24(22)12-19)15-18-9-20(38-3)13-21(10-18)39-4/h6,8-13,16H,5,7,14-15H2,1-4H3	IJUGJEQXAKUEAB-UHFFFAOYSA-N	50605336	CHEMBL5202831	WD repeat-containing protein 5		<0.020000								ChEMBL		10.7270/Q2JQ153M	35436124			Teuscher, KB; Meyers, KM; Wei, Q; Mills, JJ; Tian, J; Alvarado, J; Sai, J; Van Meveren, M; South, TM; Rietz, TA; Zhao, B; Moore, WJ; Stott, GM; Tansey, WP; Lee, T; Fesik, SW	Frederick National Laboratory for Cancer Research	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50605336	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50605336&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	4U 		153572432	482616187							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51502295	CCc1nccn1Cc1cc(-c2cn(C)nc2C(F)(F)F)c2CCN(Cc3cc(OC)cc(OC)c3)C(=O)c2c1	InChI=1S/C29H30F3N5O3/c1-5-26-33-7-9-36(26)15-19-12-23(25-17-35(2)34-27(25)29(30,31)32)22-6-8-37(28(38)24(22)13-19)16-18-10-20(39-3)14-21(11-18)40-4/h7,9-14,17H,5-6,8,15-16H2,1-4H3	RFAXXFXKTBIANZ-UHFFFAOYSA-N	50605337	CHEMBL5192283	WD repeat-containing protein 5		 0.028000								ChEMBL		10.7270/Q2JQ153M	35436124			Teuscher, KB; Meyers, KM; Wei, Q; Mills, JJ; Tian, J; Alvarado, J; Sai, J; Van Meveren, M; South, TM; Rietz, TA; Zhao, B; Moore, WJ; Stott, GM; Tansey, WP; Lee, T; Fesik, SW	Frederick National Laboratory for Cancer Research	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50605337	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50605337&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			168287350	482616188							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51502296	COc1cc(CN2CCc3c(cc(Cn4ccnc4C(C)C)cc3C2=O)-c2cn(C)nc2C(F)(F)F)cc(OC)c1	InChI=1S/C30H32F3N5O3/c1-18(2)28-34-7-9-37(28)15-20-12-24(26-17-36(3)35-27(26)30(31,32)33)23-6-8-38(29(39)25(23)13-20)16-19-10-21(40-4)14-22(11-19)41-5/h7,9-14,17-18H,6,8,15-16H2,1-5H3	JKTKUPSGMFKLLQ-UHFFFAOYSA-N	50605338	CHEMBL5202465	WD repeat-containing protein 5		 3.4								ChEMBL		10.7270/Q2JQ153M	35436124			Teuscher, KB; Meyers, KM; Wei, Q; Mills, JJ; Tian, J; Alvarado, J; Sai, J; Van Meveren, M; South, TM; Rietz, TA; Zhao, B; Moore, WJ; Stott, GM; Tansey, WP; Lee, T; Fesik, SW	Frederick National Laboratory for Cancer Research	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50605338	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50605338&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			168292688	482616189							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51502297	COc1cc(CN2CCc3c(cc(Cn4ccnc4C4CC4)cc3C2=O)-c2cn(C)nc2C(F)(F)F)cc(OC)c1	InChI=1S/C30H30F3N5O3/c1-36-17-26(27(35-36)30(31,32)33)24-12-19(15-37-9-7-34-28(37)20-4-5-20)13-25-23(24)6-8-38(29(25)39)16-18-10-21(40-2)14-22(11-18)41-3/h7,9-14,17,20H,4-6,8,15-16H2,1-3H3	LWBGSZQHGTUROL-UHFFFAOYSA-N	50605339	CHEMBL5171051	WD repeat-containing protein 5		 0.028000								ChEMBL		10.7270/Q2JQ153M	35436124			Teuscher, KB; Meyers, KM; Wei, Q; Mills, JJ; Tian, J; Alvarado, J; Sai, J; Van Meveren, M; South, TM; Rietz, TA; Zhao, B; Moore, WJ; Stott, GM; Tansey, WP; Lee, T; Fesik, SW	Frederick National Laboratory for Cancer Research	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50605339	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50605339&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			168269871	482616190							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51502298	COc1cc(CN2CCc3c(cc(Cn4ccnc4C(F)F)cc3C2=O)-c2cn(C)nc2C(F)(F)F)cc(OC)c1	InChI=1S/C28H26F5N5O3/c1-36-15-23(24(35-36)28(31,32)33)21-10-17(13-37-7-5-34-26(37)25(29)30)11-22-20(21)4-6-38(27(22)39)14-16-8-18(40-2)12-19(9-16)41-3/h5,7-12,15,25H,4,6,13-14H2,1-3H3	NPPUETMCSMKHAQ-UHFFFAOYSA-N	50605340	CHEMBL5174099	WD repeat-containing protein 5		>6.7								ChEMBL		10.7270/Q2JQ153M	35436124			Teuscher, KB; Meyers, KM; Wei, Q; Mills, JJ; Tian, J; Alvarado, J; Sai, J; Van Meveren, M; South, TM; Rietz, TA; Zhao, B; Moore, WJ; Stott, GM; Tansey, WP; Lee, T; Fesik, SW	Frederick National Laboratory for Cancer Research	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50605340	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50605340&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			168275293	482616191							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51502299	Cc1nccn1Cc1cc(-c2cn(C)nc2C(F)(F)F)c2CCN(Cc3ccccn3)C(=O)c2c1	InChI=1S/C25H23F3N6O/c1-16-29-8-10-33(16)13-17-11-20(22-15-32(2)31-23(22)25(26,27)28)19-6-9-34(24(35)21(19)12-17)14-18-5-3-4-7-30-18/h3-5,7-8,10-12,15H,6,9,13-14H2,1-2H3	WRAJXTAYFDNAPQ-UHFFFAOYSA-N	50605341	CHEMBL5208340	WD repeat-containing protein 5		 0.230000								ChEMBL		10.7270/Q2JQ153M	35436124			Teuscher, KB; Meyers, KM; Wei, Q; Mills, JJ; Tian, J; Alvarado, J; Sai, J; Van Meveren, M; South, TM; Rietz, TA; Zhao, B; Moore, WJ; Stott, GM; Tansey, WP; Lee, T; Fesik, SW	Frederick National Laboratory for Cancer Research	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50605341	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50605341&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			153238800	482616192							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51502300	Cc1nccn1Cc1cc(-c2cn(C)nc2C(F)(F)F)c2CCN(Cc3cccc(C)n3)C(=O)c2c1	InChI=1S/C26H25F3N6O/c1-16-5-4-6-19(31-16)14-35-9-7-20-21(23-15-33(3)32-24(23)26(27,28)29)11-18(12-22(20)25(35)36)13-34-10-8-30-17(34)2/h4-6,8,10-12,15H,7,9,13-14H2,1-3H3	FGSKGLJDKCYMOK-UHFFFAOYSA-N	50605342	CHEMBL5194215	WD repeat-containing protein 5		 0.039000								ChEMBL		10.7270/Q2JQ153M	35436124			Teuscher, KB; Meyers, KM; Wei, Q; Mills, JJ; Tian, J; Alvarado, J; Sai, J; Van Meveren, M; South, TM; Rietz, TA; Zhao, B; Moore, WJ; Stott, GM; Tansey, WP; Lee, T; Fesik, SW	Frederick National Laboratory for Cancer Research	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50605342	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50605342&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			153572508	482616193							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51502301	Cc1nccn1Cc1cc(-c2cn(C)nc2C(F)(F)F)c2CCN(Cc3cc(C)ccn3)C(=O)c2c1	InChI=1S/C26H25F3N6O/c1-16-4-6-31-19(10-16)14-35-8-5-20-21(23-15-33(3)32-24(23)26(27,28)29)11-18(12-22(20)25(35)36)13-34-9-7-30-17(34)2/h4,6-7,9-12,15H,5,8,13-14H2,1-3H3	NQLMHXRNQWPCBA-UHFFFAOYSA-N	50605343	CHEMBL5190556	WD repeat-containing protein 5		 0.020000								ChEMBL		10.7270/Q2JQ153M	35436124			Teuscher, KB; Meyers, KM; Wei, Q; Mills, JJ; Tian, J; Alvarado, J; Sai, J; Van Meveren, M; South, TM; Rietz, TA; Zhao, B; Moore, WJ; Stott, GM; Tansey, WP; Lee, T; Fesik, SW	Frederick National Laboratory for Cancer Research	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50605343	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50605343&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			153572325	482616194							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51502302	Cc1nccn1Cc1cc(-c2cn(C)nc2C(F)(F)F)c2CCN(Cc3ncccc3C)C(=O)c2c1	InChI=1S/C26H25F3N6O/c1-16-5-4-7-31-23(16)15-35-9-6-19-20(22-14-33(3)32-24(22)26(27,28)29)11-18(12-21(19)25(35)36)13-34-10-8-30-17(34)2/h4-5,7-8,10-12,14H,6,9,13,15H2,1-3H3	AZNSVNKRAUMUJR-UHFFFAOYSA-N	50605344	CHEMBL5171801	WD repeat-containing protein 5		 0.590000								ChEMBL		10.7270/Q2JQ153M	35436124			Teuscher, KB; Meyers, KM; Wei, Q; Mills, JJ; Tian, J; Alvarado, J; Sai, J; Van Meveren, M; South, TM; Rietz, TA; Zhao, B; Moore, WJ; Stott, GM; Tansey, WP; Lee, T; Fesik, SW	Frederick National Laboratory for Cancer Research	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50605344	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50605344&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			153572565	482616195							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51502303	Cc1nccn1Cc1cc(-c2cn(C)nc2C(F)(F)F)c2CCN(Cc3ccnc(C)c3)C(=O)c2c1	InChI=1S/C26H25F3N6O/c1-16-10-18(4-6-30-16)13-35-8-5-20-21(23-15-33(3)32-24(23)26(27,28)29)11-19(12-22(20)25(35)36)14-34-9-7-31-17(34)2/h4,6-7,9-12,15H,5,8,13-14H2,1-3H3	IKOSBIPAJNHXGY-UHFFFAOYSA-N	50605345	CHEMBL5190202	WD repeat-containing protein 5		 0.064000								ChEMBL		10.7270/Q2JQ153M	35436124			Teuscher, KB; Meyers, KM; Wei, Q; Mills, JJ; Tian, J; Alvarado, J; Sai, J; Van Meveren, M; South, TM; Rietz, TA; Zhao, B; Moore, WJ; Stott, GM; Tansey, WP; Lee, T; Fesik, SW	Frederick National Laboratory for Cancer Research	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50605345	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50605345&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			147934765	482616196							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51502304	COc1ccnc(CN2CCc3c(cc(Cn4ccnc4C)cc3C2=O)-c2cn(C)nc2C(F)(F)F)c1	InChI=1S/C26H25F3N6O2/c1-16-30-7-9-34(16)13-17-10-21(23-15-33(2)32-24(23)26(27,28)29)20-5-8-35(25(36)22(20)11-17)14-18-12-19(37-3)4-6-31-18/h4,6-7,9-12,15H,5,8,13-14H2,1-3H3	YGNFBQUKKVHYGI-UHFFFAOYSA-N	50605346	CHEMBL5177738	WD repeat-containing protein 5		<0.020000								ChEMBL		10.7270/Q2JQ153M	35436124			Teuscher, KB; Meyers, KM; Wei, Q; Mills, JJ; Tian, J; Alvarado, J; Sai, J; Van Meveren, M; South, TM; Rietz, TA; Zhao, B; Moore, WJ; Stott, GM; Tansey, WP; Lee, T; Fesik, SW	Frederick National Laboratory for Cancer Research	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50605346	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50605346&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			153572459	482616197							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51502305	CCc1ccnc(CN2CCc3c(cc(Cn4ccnc4C)cc3C2=O)-c2cn(C)nc2C(F)(F)F)c1	InChI=1S/C27H27F3N6O/c1-4-18-5-7-32-20(11-18)15-36-9-6-21-22(24-16-34(3)33-25(24)27(28,29)30)12-19(13-23(21)26(36)37)14-35-10-8-31-17(35)2/h5,7-8,10-13,16H,4,6,9,14-15H2,1-3H3	IEGWXZPIWMLBRP-UHFFFAOYSA-N	50605347	CHEMBL5174178	WD repeat-containing protein 5		<0.020000								ChEMBL		10.7270/Q2JQ153M	35436124			Teuscher, KB; Meyers, KM; Wei, Q; Mills, JJ; Tian, J; Alvarado, J; Sai, J; Van Meveren, M; South, TM; Rietz, TA; Zhao, B; Moore, WJ; Stott, GM; Tansey, WP; Lee, T; Fesik, SW	Frederick National Laboratory for Cancer Research	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50605347	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50605347&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			168271568	482616198							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51502306	CCn1cc(c(n1)C(F)(F)F)-c1cc(Cn2ccnc2C)cc2C(=O)N(Cc3cc(OC)ccn3)CCc12	InChI=1S/C27H27F3N6O2/c1-4-36-16-24(25(33-36)27(28,29)30)22-11-18(14-34-10-8-31-17(34)2)12-23-21(22)6-9-35(26(23)37)15-19-13-20(38-3)5-7-32-19/h5,7-8,10-13,16H,4,6,9,14-15H2,1-3H3	GLOSEPKLMDGBBB-UHFFFAOYSA-N	50605348	CHEMBL5183319	WD repeat-containing protein 5		<0.020000								ChEMBL		10.7270/Q2JQ153M	35436124			Teuscher, KB; Meyers, KM; Wei, Q; Mills, JJ; Tian, J; Alvarado, J; Sai, J; Van Meveren, M; South, TM; Rietz, TA; Zhao, B; Moore, WJ; Stott, GM; Tansey, WP; Lee, T; Fesik, SW	Frederick National Laboratory for Cancer Research	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50605348	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50605348&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			168283719	482616199							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51502307	CCc1ccnc(CN2CCc3c(cc(Cn4ccnc4C)cc3C2=O)-c2cn(CC)nc2C(F)(F)F)c1	InChI=1S/C28H29F3N6O/c1-4-19-6-8-33-21(12-19)16-36-10-7-22-23(25-17-37(5-2)34-26(25)28(29,30)31)13-20(14-24(22)27(36)38)15-35-11-9-32-18(35)3/h6,8-9,11-14,17H,4-5,7,10,15-16H2,1-3H3	GFJWQGWZIAQBFB-UHFFFAOYSA-N	50605349	CHEMBL5191181	WD repeat-containing protein 5		<0.020000								ChEMBL		10.7270/Q2JQ153M	35436124			Teuscher, KB; Meyers, KM; Wei, Q; Mills, JJ; Tian, J; Alvarado, J; Sai, J; Van Meveren, M; South, TM; Rietz, TA; Zhao, B; Moore, WJ; Stott, GM; Tansey, WP; Lee, T; Fesik, SW	Frederick National Laboratory for Cancer Research	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50605349	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50605349&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			153572297	482616200							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51502308	CCn1cc(c(n1)C(F)(F)F)-c1cc(Cn2ccnc2C)cc2C(=O)N(CCc12)[C@@H](C)c1cc(OC)ccn1	InChI=1S/C28H29F3N6O2/c1-5-36-16-24(26(34-36)28(29,30)31)22-12-19(15-35-11-9-32-18(35)3)13-23-21(22)7-10-37(27(23)38)17(2)25-14-20(39-4)6-8-33-25/h6,8-9,11-14,16-17H,5,7,10,15H2,1-4H3/t17-/m0/s1	ZHJGXPCMCSZPPK-KRWDZBQOSA-N	50605350	CHEMBL5177656	WD repeat-containing protein 5		<0.020000								ChEMBL		10.7270/Q2JQ153M	35436124			Teuscher, KB; Meyers, KM; Wei, Q; Mills, JJ; Tian, J; Alvarado, J; Sai, J; Van Meveren, M; South, TM; Rietz, TA; Zhao, B; Moore, WJ; Stott, GM; Tansey, WP; Lee, T; Fesik, SW	Frederick National Laboratory for Cancer Research	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50605350	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50605350&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			149503094	482616201							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51502309	CCn1cc(c(n1)C(F)(F)F)-c1cc(Cn2ccnc2C)cc2C(=O)N(CCc12)[C@H](C)c1cc(OC)ccn1	InChI=1S/C28H29F3N6O2/c1-5-36-16-24(26(34-36)28(29,30)31)22-12-19(15-35-11-9-32-18(35)3)13-23-21(22)7-10-37(27(23)38)17(2)25-14-20(39-4)6-8-33-25/h6,8-9,11-14,16-17H,5,7,10,15H2,1-4H3/t17-/m1/s1	ZHJGXPCMCSZPPK-QGZVFWFLSA-N	50605351	CHEMBL5180435	WD repeat-containing protein 5		 0.029000								ChEMBL		10.7270/Q2JQ153M	35436124			Teuscher, KB; Meyers, KM; Wei, Q; Mills, JJ; Tian, J; Alvarado, J; Sai, J; Van Meveren, M; South, TM; Rietz, TA; Zhao, B; Moore, WJ; Stott, GM; Tansey, WP; Lee, T; Fesik, SW	Frederick National Laboratory for Cancer Research	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50605351	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50605351&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			168277456	482616202							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51502310	CCn1cc(c(n1)C(F)(F)F)-c1cc(Cn2ccnc2C)cc2C(=O)N(CCc12)[C@H](C1CC1)c1cc(OC)ccn1	InChI=1S/C30H31F3N6O2/c1-4-38-17-25(28(36-38)30(31,32)33)23-13-19(16-37-12-10-34-18(37)2)14-24-22(23)8-11-39(29(24)40)27(20-5-6-20)26-15-21(41-3)7-9-35-26/h7,9-10,12-15,17,20,27H,4-6,8,11,16H2,1-3H3/t27-/m1/s1	YCIMDILXHOWXJJ-HHHXNRCGSA-N	50605352	CHEMBL5198319	WD repeat-containing protein 5		<0.020000								ChEMBL		10.7270/Q2JQ153M	35436124			Teuscher, KB; Meyers, KM; Wei, Q; Mills, JJ; Tian, J; Alvarado, J; Sai, J; Van Meveren, M; South, TM; Rietz, TA; Zhao, B; Moore, WJ; Stott, GM; Tansey, WP; Lee, T; Fesik, SW	Frederick National Laboratory for Cancer Research	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50605352	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50605352&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			168285249	482616203							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51502311	CCn1cc(c(n1)C(F)(F)F)-c1cc(Cn2ccnc2C)cc2C(=O)N(CCc12)[C@@H](C1CC1)c1cc(C)ccn1	InChI=1S/C30H31F3N6O/c1-4-38-17-25(28(36-38)30(31,32)33)23-14-20(16-37-12-10-34-19(37)3)15-24-22(23)8-11-39(29(24)40)27(21-5-6-21)26-13-18(2)7-9-35-26/h7,9-10,12-15,17,21,27H,4-6,8,11,16H2,1-3H3/t27-/m0/s1	URNMGEJXPZLHRK-MHZLTWQESA-N	50605353	CHEMBL5190717	WD repeat-containing protein 5		<0.020000								ChEMBL		10.7270/Q2JQ153M	35436124			Teuscher, KB; Meyers, KM; Wei, Q; Mills, JJ; Tian, J; Alvarado, J; Sai, J; Van Meveren, M; South, TM; Rietz, TA; Zhao, B; Moore, WJ; Stott, GM; Tansey, WP; Lee, T; Fesik, SW	Frederick National Laboratory for Cancer Research	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50605353	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50605353&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	BU 		153572417	482616204							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51502312	CCn1cc(c(n1)C(F)(F)F)-c1cc(Cn2ccnc2C)cc2C(=O)N(CCc12)[C@@H](C)c1cc(OC)ccn1	InChI=1S/C28H29F3N6O2/c1-5-36-16-24(26(34-36)28(29,30)31)22-12-19(15-35-11-9-32-18(35)3)13-23-21(22)7-10-37(27(23)38)17(2)25-14-20(39-4)6-8-33-25/h6,8-9,11-14,16-17H,5,7,10,15H2,1-4H3/t17-/m0/s1	ZHJGXPCMCSZPPK-KRWDZBQOSA-N	50605350	CHEMBL5177656	WD repeat-containing protein 5		<0.020000								ChEMBL		10.7270/Q2JQ153M	35436124			Teuscher, KB; Meyers, KM; Wei, Q; Mills, JJ; Tian, J; Alvarado, J; Sai, J; Van Meveren, M; South, TM; Rietz, TA; Zhao, B; Moore, WJ; Stott, GM; Tansey, WP; Lee, T; Fesik, SW	Frederick National Laboratory for Cancer Research	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50605350	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50605350&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			149503094	482616201							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51502313	CCn1cc(c(n1)C(F)(F)F)-c1cc(Cn2ccnc2)cc2C(=O)N(CCc12)[C@H](C)c1cc(OC)ccn1	InChI=1S/C27H27F3N6O2/c1-4-35-15-23(25(33-35)27(28,29)30)21-11-18(14-34-10-8-31-16-34)12-22-20(21)6-9-36(26(22)37)17(2)24-13-19(38-3)5-7-32-24/h5,7-8,10-13,15-17H,4,6,9,14H2,1-3H3/t17-/m1/s1	WBTTWUZIOAJQRP-QGZVFWFLSA-N	50605354	CHEMBL5179388	WD repeat-containing protein 5		 0.028000								ChEMBL		10.7270/Q2JQ153M	35436124			Teuscher, KB; Meyers, KM; Wei, Q; Mills, JJ; Tian, J; Alvarado, J; Sai, J; Van Meveren, M; South, TM; Rietz, TA; Zhao, B; Moore, WJ; Stott, GM; Tansey, WP; Lee, T; Fesik, SW	Frederick National Laboratory for Cancer Research	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50605354	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50605354&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			168276711	482616205							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51502314	CCn1cc(c(n1)C(F)(F)F)-c1cc(Cn2ccnc2)cc2C(=O)N(CCc12)[C@@H](C1CC1)c1cc(OC)ccn1	InChI=1S/C29H29F3N6O2/c1-3-37-16-24(27(35-37)29(30,31)32)22-12-18(15-36-11-9-33-17-36)13-23-21(22)7-10-38(28(23)39)26(19-4-5-19)25-14-20(40-2)6-8-34-25/h6,8-9,11-14,16-17,19,26H,3-5,7,10,15H2,1-2H3/t26-/m0/s1	IRXFPIASUFJVNS-SANMLTNESA-N	50605355	CHEMBL5170717	WD repeat-containing protein 5		<0.020000								ChEMBL		10.7270/Q2JQ153M	35436124			Teuscher, KB; Meyers, KM; Wei, Q; Mills, JJ; Tian, J; Alvarado, J; Sai, J; Van Meveren, M; South, TM; Rietz, TA; Zhao, B; Moore, WJ; Stott, GM; Tansey, WP; Lee, T; Fesik, SW	Frederick National Laboratory for Cancer Research	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50605355	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50605355&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			153572492	482616206							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51502315	CCn1cc(c(n1)C(F)(F)F)-c1cc(Cn2ccnc2)cc2C(=O)N(CCc12)[C@H](C1CC1)c1cc(OC)ccn1	InChI=1S/C29H29F3N6O2/c1-3-37-16-24(27(35-37)29(30,31)32)22-12-18(15-36-11-9-33-17-36)13-23-21(22)7-10-38(28(23)39)26(19-4-5-19)25-14-20(40-2)6-8-34-25/h6,8-9,11-14,16-17,19,26H,3-5,7,10,15H2,1-2H3/t26-/m1/s1	IRXFPIASUFJVNS-AREMUKBSSA-N	50605356	CHEMBL5170071	WD repeat-containing protein 5		<0.020000								ChEMBL		10.7270/Q2JQ153M	35436124			Teuscher, KB; Meyers, KM; Wei, Q; Mills, JJ; Tian, J; Alvarado, J; Sai, J; Van Meveren, M; South, TM; Rietz, TA; Zhao, B; Moore, WJ; Stott, GM; Tansey, WP; Lee, T; Fesik, SW	Frederick National Laboratory for Cancer Research	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50605356	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50605356&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			168268943	482616207							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51510435	Clc1ccc(OCCCNC2=NCCN2)c(Cl)c1	InChI=1S/C12H15Cl2N3O/c13-9-2-3-11(10(14)8-9)18-7-1-4-15-12-16-5-6-17-12/h2-3,8H,1,4-7H2,(H2,15,16,17)	XIKGAVKOOOYGIY-UHFFFAOYSA-N	50608083	CHEMBL5205374	WD repeat-containing protein 5				 66000						ChEMBL		10.7270/Q2HQ444G	34591474			n/a	n/a	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50608083	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50608083&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			53593645	494497831							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E,8HMX,8Q1N	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51510436	CC(NC(=O)c1cccc(CNC2=NCCN2)c1)c1cccc(Cl)c1	InChI=1S/C19H21ClN4O/c1-13(15-5-3-7-17(20)11-15)24-18(25)16-6-2-4-14(10-16)12-23-19-21-8-9-22-19/h2-7,10-11,13H,8-9,12H2,1H3,(H,24,25)(H2,21,22,23)	ZHGJIKXLESXIHK-UHFFFAOYSA-N	468872	US10807959, Example B5	WD repeat-containing protein 5				 22						ChEMBL		10.7270/Q2HQ444G	34591474			n/a	n/a	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468872	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468872&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	HLM	6E1Y	146370875	441570973							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E,8HMX,8Q1N	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51510437	COc1cc(CNC(=O)c2ccc(F)c(CNC3=NCCN3)c2)cc(OC)c1	InChI=1S/C20H23FN4O3/c1-27-16-7-13(8-17(10-16)28-2)11-24-19(26)14-3-4-18(21)15(9-14)12-25-20-22-5-6-23-20/h3-4,7-10H,5-6,11-12H2,1-2H3,(H,24,26)(H2,22,23,25)	VDAMWMOTTUWVPR-UHFFFAOYSA-N	468882	US10807959, Example B15	WD repeat-containing protein 5				 1.3						ChEMBL		10.7270/Q2HQ444G	34591474			n/a	n/a	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=468882	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=468882&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	HLS	6E22	138753248	441570983							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	2G99,2G9A,2GNQ,2H13,2H14,2H68,2H6K,2H6N,2H6Q,2XL2,2XL3,3EG6,3EMH,3MXX,3N0D,3N0E,3P4F,3PSL,3UVK,3UVL,3UVM,3UVN,3UVO,4A7J,4CY1,4CY2,4ERQ,4ERY,4ERZ,4ES0,4ESG,4EWR,4GM3,4GM8,4GM9,4GMB,4Y7R,5SXM,5VFC,6BYN,6D9X,6DAI,6DAK,6DAR,6DAS,6DY7,6DYA,6E1Y,6E1Z,6E22,6E23,6IAM,6KIU,6KIV,6KIW,6KIX,6KIZ,6OFZ,6OI0,6OI1,6OI2,6OI3,6PG3,6PG4,6PG5,6PG6,6PG7,6PG8,6PG9,6PGA,6PGB,6PGC,6PGD,6PGE,6PGF,6PWV,6PWW,6U5M,6U5Y,6U6W,6U80,6U8B,6U8L,6U8O,6UCS,6UHY,6UHZ,6UIF,6UIK,6UJ4,6UJH,6UJJ,6UJL,6UOZ,6W5I,6W5M,6W5N,6WJQ,7AXP,7AXQ,7AXS,7AXU,7AXX,7BCY,7BED,7CFP,7CFQ,7DNO,7JTO,7JTP,7MBM,7MBN,7U9Y,7UAS,7UD5,7WVK,8BB2,8BB3,8BB4,8BB5,8DU4,8E9F,8F1G,8F93,8G3C,8G3E,8HMX,8Q1N	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51570930	CC[C@H](C)[C@H](NC(=O)[C@H](CCC(O)=O)NC(=O)[C@H](CCC(O)=O)NC(=O)[C@H](CCC(O)=O)NC(=O)[C@H](CC(O)=O)NC(=O)COCCOCCNC(=S)Nc1ccc(c(c1)C(O)=O)-c1c2ccc(O)cc2oc2cc(=O)ccc12)C(=O)N[C@H]1CC(=O)NCC[C@H](NC(=O)[C@@H](NC(=O)[C@@H](NC1=O)C(C)C)C(C)C)C(=O)N[C@@H](C(C)C)C(=O)N[C@@H](CCC(O)=O)C(N)=O	InChI=1S/C80H107N15O30S/c1-9-39(8)67(78(120)91-52-33-56(98)82-25-24-51(90-76(118)65(37(4)5)94-77(119)66(38(6)7)93-74(52)116)72(114)92-64(36(2)3)75(117)86-47(68(81)110)16-20-58(100)101)95-71(113)50(19-23-61(106)107)88-69(111)48(17-21-59(102)103)87-70(112)49(18-22-60(104)105)89-73(115)53(34-62(108)109)85-57(99)35-124-29-28-123-27-26-83-80(126)84-40-10-13-43(46(30-40)79(121)122)63-44-14-11-41(96)31-54(44)125-55-32-42(97)12-15-45(55)63/h10-15,30-32,36-39,47-53,64-67,96H,9,16-29,33-35H2,1-8H3,(H2,81,110)(H,82,98)(H,85,99)(H,86,117)(H,87,112)(H,88,111)(H,89,115)(H,90,118)(H,91,120)(H,92,114)(H,93,116)(H,94,119)(H,95,113)(H,100,101)(H,102,103)(H,104,105)(H,106,107)(H,108,109)(H,121,122)(H2,83,84,126)/t39-,47-,48-,49-,50-,51-,52-,53-,64-,65-,66-,67-/m0/s1	PSZBBHQYVVVGDN-LNKBOCRRSA-N	50631812	CHEMBL5440056	WD repeat-containing protein 5	Homo sapiens			 347						ChEMBL	10.1039/d3md00605k	10.7270/Q2833XH5	38389889			n/a	n/a	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50631812	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50631812&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search											1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	8X3R,7CFQ,7CFP,7BED,7AXX,7AXU,7AXS,7AXQ,7AXP,6KIZ,6KIX,6KIW,6KIV,6KIU,2XL3,2XL2,2GNQ,8DU4,7UD5,8X3S,3UVO,3UVN,3UVM,3UVL,3UVK,3PSL,8OKF,4A7J,8G3E,8F93,8F1G,8G3C,7WVK,7UAS,7MBN,7MBM,6WJQ,6W5N,6W5M,6W5I,6UJL,6UJJ,6UJH,6UCS,6PWW,6PWV,6PG9,6PG8,6PG6,6PG3,6OI3,6OI2,6OI1,6OI0,6OFZ,6E23,6E22,6E1Z,6E1Y,6DAS,6DAR,6DAK,6DAI,6D9X,4Y7R,4GMB,4GM9,4GM8,4GM3,3P4F,2H14,2H13,8Q1N,5SXM,4CY2,4CY1,4EWR,4ESG,4ES0,4ERZ,4ERY,4ERQ,3EG6,2H6Q,2H6N,2H6K,2H68,7DNO,6U8B,6U80,6U6W,5VFC,3EMH,7BCY,2G99,6IAM,8E9F,7U9Y,6DYA,2G9A,8HMX,6UOZ,6UJ4,6UIK,6UIF,6UHZ,6UHY,6U8O,6U8L,6U5Y,6U5M,6DY7,7JTP,7JTO,6BYN,3MXX,3N0E,6PGF,6PGE,6PGD,6PGC,6PGB,6PGA,6PG7,6PG5,6PG4,3N0D,8BB5,8BB4,8BB3,8BB2	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51570931	CC(C)C[C@H](NC(=O)[C@H](Cc1cnc[nH]1)NC(=O)[C@@H](NC(=O)[C@H](CCC(O)=O)NC(=O)[C@@H](NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@H](C)NC(C)=O)[C@@H](C)O)C(C)C)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CO)C(=O)NCCCCCC(=O)NCCCCCC(=O)N[C@@H](CCCCNC(=O)c1ccc(c(c1)C(O)=O)-c1c2ccc(O)cc2oc2cc(=O)ccc12)C(N)=O	InChI=1S/C91H136N24O24/c1-48(2)40-66(111-86(134)67(42-54-45-98-47-104-54)112-87(135)75(49(3)4)114-84(132)65(32-33-73(123)124)110-88(136)76(51(6)117)115-83(131)64(23-19-39-103-91(96)97)107-78(126)50(5)105-52(7)118)85(133)109-63(22-18-38-102-90(94)95)81(129)108-62(21-12-14-34-92)82(130)113-68(46-116)80(128)101-36-16-8-10-24-71(121)99-35-15-9-11-25-72(122)106-61(77(93)125)20-13-17-37-100-79(127)53-26-29-57(60(41-53)89(137)138)74-58-30-27-55(119)43-69(58)139-70-44-56(120)28-31-59(70)74/h26-31,41,43-45,47-51,61-68,75-76,116-117,119H,8-25,32-40,42,46,92H2,1-7H3,(H2,93,125)(H,98,104)(H,99,121)(H,100,127)(H,101,128)(H,105,118)(H,106,122)(H,107,126)(H,108,129)(H,109,133)(H,110,136)(H,111,134)(H,112,135)(H,113,130)(H,114,132)(H,115,131)(H,123,124)(H,137,138)(H4,94,95,102)(H4,96,97,103)/t50-,51+,61-,62-,63-,64-,65-,66-,67-,68-,75-,76-/m0/s1	LVHMEOMYGFPCIV-CLNRVIFCSA-N	50631811	CHEMBL5417280	WD repeat-containing protein 5	Homo sapiens			 78						ChEMBL	10.1039/d3md00605k	10.7270/Q2833XH5	38389889			n/a	n/a	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50631811	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50631811&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search											1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	8X3R,7CFQ,7CFP,7BED,7AXX,7AXU,7AXS,7AXQ,7AXP,6KIZ,6KIX,6KIW,6KIV,6KIU,2XL3,2XL2,2GNQ,8DU4,7UD5,8X3S,3UVO,3UVN,3UVM,3UVL,3UVK,3PSL,8OKF,4A7J,8G3E,8F93,8F1G,8G3C,7WVK,7UAS,7MBN,7MBM,6WJQ,6W5N,6W5M,6W5I,6UJL,6UJJ,6UJH,6UCS,6PWW,6PWV,6PG9,6PG8,6PG6,6PG3,6OI3,6OI2,6OI1,6OI0,6OFZ,6E23,6E22,6E1Z,6E1Y,6DAS,6DAR,6DAK,6DAI,6D9X,4Y7R,4GMB,4GM9,4GM8,4GM3,3P4F,2H14,2H13,8Q1N,5SXM,4CY2,4CY1,4EWR,4ESG,4ES0,4ERZ,4ERY,4ERQ,3EG6,2H6Q,2H6N,2H6K,2H68,7DNO,6U8B,6U80,6U6W,5VFC,3EMH,7BCY,2G99,6IAM,8E9F,7U9Y,6DYA,2G9A,8HMX,6UOZ,6UJ4,6UIK,6UIF,6UHZ,6UHY,6U8O,6U8L,6U5Y,6U5M,6DY7,7JTP,7JTO,6BYN,3MXX,3N0E,6PGF,6PGE,6PGD,6PGC,6PGB,6PGA,6PG7,6PG5,6PG4,3N0D,8BB5,8BB4,8BB3,8BB2	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51570932	CC[C@H](C)[C@H](NC(=O)[C@H](CCC(O)=O)NC(=O)[C@H](CCC(O)=O)NC(=O)[C@H](CCC(O)=O)NC(=O)[C@H](CC(O)=O)NC(=O)COCCOCCNC(=S)Nc1ccc(c(c1)C(O)=O)-c1c2ccc(O)cc2oc2cc(=O)ccc12)C(=O)N[C@H]1CC(=O)NCC[C@H](NC(=O)[C@@H](NC(=O)[C@@H](NC1=O)C(C)C)C(C)C)C(=O)N[C@@H](C(C)C)C(=O)N[C@@H](CCC(O)=O)C(N)=O	InChI=1S/C80H107N15O30S/c1-9-39(8)67(78(120)91-52-33-56(98)82-25-24-51(90-76(118)65(37(4)5)94-77(119)66(38(6)7)93-74(52)116)72(114)92-64(36(2)3)75(117)86-47(68(81)110)16-20-58(100)101)95-71(113)50(19-23-61(106)107)88-69(111)48(17-21-59(102)103)87-70(112)49(18-22-60(104)105)89-73(115)53(34-62(108)109)85-57(99)35-124-29-28-123-27-26-83-80(126)84-40-10-13-43(46(30-40)79(121)122)63-44-14-11-41(96)31-54(44)125-55-32-42(97)12-15-45(55)63/h10-15,30-32,36-39,47-53,64-67,96H,9,16-29,33-35H2,1-8H3,(H2,81,110)(H,82,98)(H,85,99)(H,86,117)(H,87,112)(H,88,111)(H,89,115)(H,90,118)(H,91,120)(H,92,114)(H,93,116)(H,94,119)(H,95,113)(H,100,101)(H,102,103)(H,104,105)(H,106,107)(H,108,109)(H,121,122)(H2,83,84,126)/t39-,47-,48-,49-,50-,51-,52-,53-,64-,65-,66-,67-/m0/s1	PSZBBHQYVVVGDN-LNKBOCRRSA-N	50631812	CHEMBL5440056	WD repeat-containing protein 5	Homo sapiens			 11200						ChEMBL	10.1039/d3md00605k	10.7270/Q2833XH5	38389889			n/a	n/a	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50631812	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50631812&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search											1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	8X3R,7CFQ,7CFP,7BED,7AXX,7AXU,7AXS,7AXQ,7AXP,6KIZ,6KIX,6KIW,6KIV,6KIU,2XL3,2XL2,2GNQ,8DU4,7UD5,8X3S,3UVO,3UVN,3UVM,3UVL,3UVK,3PSL,8OKF,4A7J,8G3E,8F93,8F1G,8G3C,7WVK,7UAS,7MBN,7MBM,6WJQ,6W5N,6W5M,6W5I,6UJL,6UJJ,6UJH,6UCS,6PWW,6PWV,6PG9,6PG8,6PG6,6PG3,6OI3,6OI2,6OI1,6OI0,6OFZ,6E23,6E22,6E1Z,6E1Y,6DAS,6DAR,6DAK,6DAI,6D9X,4Y7R,4GMB,4GM9,4GM8,4GM3,3P4F,2H14,2H13,8Q1N,5SXM,4CY2,4CY1,4EWR,4ESG,4ES0,4ERZ,4ERY,4ERQ,3EG6,2H6Q,2H6N,2H6K,2H68,7DNO,6U8B,6U80,6U6W,5VFC,3EMH,7BCY,2G99,6IAM,8E9F,7U9Y,6DYA,2G9A,8HMX,6UOZ,6UJ4,6UIK,6UIF,6UHZ,6UHY,6U8O,6U8L,6U5Y,6U5M,6DY7,7JTP,7JTO,6BYN,3MXX,3N0E,6PGF,6PGE,6PGD,6PGC,6PGB,6PGA,6PG7,6PG5,6PG4,3N0D,8BB5,8BB4,8BB3,8BB2	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51570933	CN1CCN(CC1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cccc(CN2CCOCC2)c1	InChI=1S/C29H32F3N5O3/c1-35-7-9-37(10-8-35)26-6-5-22(21-4-2-3-20(15-21)19-36-11-13-40-14-12-36)16-25(26)34-28(39)23-18-33-27(38)17-24(23)29(30,31)32/h2-6,15-18H,7-14,19H2,1H3,(H,33,38)(H,34,39)	DJOVLOYCGXNVPI-UHFFFAOYSA-N	50164794	CHEMBL3798846::US11174250, Example Table4.1.1::US11319299, Comp. No. 57	WD repeat-containing protein 5	Homo sapiens	 1.2								ChEMBL	10.1039/d3md00605k	10.7270/Q2833XH5	38389889			n/a	n/a	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50164794	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50164794&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	35Q    	4QL1	91623360	341097539		CHEMBL3798846					1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	8X3R,7CFQ,7CFP,7BED,7AXX,7AXU,7AXS,7AXQ,7AXP,6KIZ,6KIX,6KIW,6KIV,6KIU,2XL3,2XL2,2GNQ,8DU4,7UD5,8X3S,3UVO,3UVN,3UVM,3UVL,3UVK,3PSL,8OKF,4A7J,8G3E,8F93,8F1G,8G3C,7WVK,7UAS,7MBN,7MBM,6WJQ,6W5N,6W5M,6W5I,6UJL,6UJJ,6UJH,6UCS,6PWW,6PWV,6PG9,6PG8,6PG6,6PG3,6OI3,6OI2,6OI1,6OI0,6OFZ,6E23,6E22,6E1Z,6E1Y,6DAS,6DAR,6DAK,6DAI,6D9X,4Y7R,4GMB,4GM9,4GM8,4GM3,3P4F,2H14,2H13,8Q1N,5SXM,4CY2,4CY1,4EWR,4ESG,4ES0,4ERZ,4ERY,4ERQ,3EG6,2H6Q,2H6N,2H6K,2H68,7DNO,6U8B,6U80,6U6W,5VFC,3EMH,7BCY,2G99,6IAM,8E9F,7U9Y,6DYA,2G9A,8HMX,6UOZ,6UJ4,6UIK,6UIF,6UHZ,6UHY,6U8O,6U8L,6U5Y,6U5M,6DY7,7JTP,7JTO,6BYN,3MXX,3N0E,6PGF,6PGE,6PGD,6PGC,6PGB,6PGA,6PG7,6PG5,6PG4,3N0D,8BB5,8BB4,8BB3,8BB2	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51570934	CNC(=O)c1cc(cc(NS(=O)(=O)c2cc(Br)cc(Cl)c2O)c1O)C1(CCC1)C#N	InChI=1S/C19H17BrClN3O5S/c1-23-18(27)12-5-10(19(9-22)3-2-4-19)6-14(16(12)25)24-30(28,29)15-8-11(20)7-13(21)17(15)26/h5-8,24-26H,2-4H2,1H3,(H,23,27)	COYGYHFILXAMSQ-UHFFFAOYSA-N	50531074	CHEMBL4472649	WD repeat-containing protein 5	Homo sapiens	>40000								ChEMBL	10.1039/d3md00605k	10.7270/Q2833XH5	38389889			n/a	n/a	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50531074	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50531074&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	Q0M    	6U5Y	145704698	440739656							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	8X3R,7CFQ,7CFP,7BED,7AXX,7AXU,7AXS,7AXQ,7AXP,6KIZ,6KIX,6KIW,6KIV,6KIU,2XL3,2XL2,2GNQ,8DU4,7UD5,8X3S,3UVO,3UVN,3UVM,3UVL,3UVK,3PSL,8OKF,4A7J,8G3E,8F93,8F1G,8G3C,7WVK,7UAS,7MBN,7MBM,6WJQ,6W5N,6W5M,6W5I,6UJL,6UJJ,6UJH,6UCS,6PWW,6PWV,6PG9,6PG8,6PG6,6PG3,6OI3,6OI2,6OI1,6OI0,6OFZ,6E23,6E22,6E1Z,6E1Y,6DAS,6DAR,6DAK,6DAI,6D9X,4Y7R,4GMB,4GM9,4GM8,4GM3,3P4F,2H14,2H13,8Q1N,5SXM,4CY2,4CY1,4EWR,4ESG,4ES0,4ERZ,4ERY,4ERQ,3EG6,2H6Q,2H6N,2H6K,2H68,7DNO,6U8B,6U80,6U6W,5VFC,3EMH,7BCY,2G99,6IAM,8E9F,7U9Y,6DYA,2G9A,8HMX,6UOZ,6UJ4,6UIK,6UIF,6UHZ,6UHY,6U8O,6U8L,6U5Y,6U5M,6DY7,7JTP,7JTO,6BYN,3MXX,3N0E,6PGF,6PGE,6PGD,6PGC,6PGB,6PGA,6PG7,6PG5,6PG4,3N0D,8BB5,8BB4,8BB3,8BB2	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51570935	CC(C)C[C@H](NC(=O)[C@H](Cc1cnc[nH]1)NC(=O)[C@@H](NC(=O)[C@H](CCC(O)=O)NC(=O)[C@@H](NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@H](C)NC(C)=O)[C@@H](C)O)C(C)C)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CO)C(N)=O	InChI=1S/C52H92N20O15/c1-25(2)20-35(47(84)66-32(13-10-18-60-51(55)56)43(80)65-31(12-8-9-17-53)44(81)70-37(23-73)41(54)78)68-48(85)36(21-30-22-59-24-62-30)69-49(86)39(26(3)4)71-46(83)34(15-16-38(76)77)67-50(87)40(28(6)74)72-45(82)33(14-11-19-61-52(57)58)64-42(79)27(5)63-29(7)75/h22,24-28,31-37,39-40,73-74H,8-21,23,53H2,1-7H3,(H2,54,78)(H,59,62)(H,63,75)(H,64,79)(H,65,80)(H,66,84)(H,67,87)(H,68,85)(H,69,86)(H,70,81)(H,71,83)(H,72,82)(H,76,77)(H4,55,56,60)(H4,57,58,61)/t27-,28+,31-,32-,33-,34-,35-,36-,37-,39-,40-/m0/s1	YABWHPOODAWVRU-RETQXLQUSA-N	50631813	CHEMBL5434345	WD repeat-containing protein 5	Homo sapiens	 0.270000								ChEMBL	10.1039/d3md00605k	10.7270/Q2833XH5	38389889			n/a	n/a	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50631813	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50631813&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search											1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	8X3R,7CFQ,7CFP,7BED,7AXX,7AXU,7AXS,7AXQ,7AXP,6KIZ,6KIX,6KIW,6KIV,6KIU,2XL3,2XL2,2GNQ,8DU4,7UD5,8X3S,3UVO,3UVN,3UVM,3UVL,3UVK,3PSL,8OKF,4A7J,8G3E,8F93,8F1G,8G3C,7WVK,7UAS,7MBN,7MBM,6WJQ,6W5N,6W5M,6W5I,6UJL,6UJJ,6UJH,6UCS,6PWW,6PWV,6PG9,6PG8,6PG6,6PG3,6OI3,6OI2,6OI1,6OI0,6OFZ,6E23,6E22,6E1Z,6E1Y,6DAS,6DAR,6DAK,6DAI,6D9X,4Y7R,4GMB,4GM9,4GM8,4GM3,3P4F,2H14,2H13,8Q1N,5SXM,4CY2,4CY1,4EWR,4ESG,4ES0,4ERZ,4ERY,4ERQ,3EG6,2H6Q,2H6N,2H6K,2H68,7DNO,6U8B,6U80,6U6W,5VFC,3EMH,7BCY,2G99,6IAM,8E9F,7U9Y,6DYA,2G9A,8HMX,6UOZ,6UJ4,6UIK,6UIF,6UHZ,6UHY,6U8O,6U8L,6U5Y,6U5M,6DY7,7JTP,7JTO,6BYN,3MXX,3N0E,6PGF,6PGE,6PGD,6PGC,6PGB,6PGA,6PG7,6PG5,6PG4,3N0D,8BB5,8BB4,8BB3,8BB2	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51570936	CC[C@H](C)[C@H](NC(=O)[C@H](CCC(O)=O)NC(=O)[C@H](CCC(O)=O)NC(=O)[C@H](CCC(O)=O)NC(=O)[C@H](CC(O)=O)NC(C)=O)C(=O)N[C@H]1CC(=O)NCC[C@H](NC(=O)[C@@H](NC(=O)[C@@H](NC1=O)C(C)C)C(C)C)C(=O)N[C@@H](C(C)C)C(=O)N[C@@H](CCC(O)=O)C(N)=O	InChI=1S/C55H87N13O23/c1-10-26(8)44(68-48(84)31(14-18-39(77)78)61-46(82)29(12-16-37(73)74)60-47(83)30(13-17-38(75)76)62-50(86)34(22-40(79)80)58-27(9)69)55(91)64-33-21-35(70)57-20-19-32(63-53(89)42(24(4)5)67-54(90)43(25(6)7)66-51(33)87)49(85)65-41(23(2)3)52(88)59-28(45(56)81)11-15-36(71)72/h23-26,28-34,41-44H,10-22H2,1-9H3,(H2,56,81)(H,57,70)(H,58,69)(H,59,88)(H,60,83)(H,61,82)(H,62,86)(H,63,89)(H,64,91)(H,65,85)(H,66,87)(H,67,90)(H,68,84)(H,71,72)(H,73,74)(H,75,76)(H,77,78)(H,79,80)/t26-,28-,29-,30-,31-,32-,33-,34-,41-,42-,43-,44-/m0/s1	CYWWYCJTGSTQEL-XWYYWFNKSA-N	50631814	CHEMBL5435898	WD repeat-containing protein 5	Homo sapiens	>40000								ChEMBL	10.1039/d3md00605k	10.7270/Q2833XH5	38389889			n/a	n/a	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50631814	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50631814&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search											1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	8X3R,7CFQ,7CFP,7BED,7AXX,7AXU,7AXS,7AXQ,7AXP,6KIZ,6KIX,6KIW,6KIV,6KIU,2XL3,2XL2,2GNQ,8DU4,7UD5,8X3S,3UVO,3UVN,3UVM,3UVL,3UVK,3PSL,8OKF,4A7J,8G3E,8F93,8F1G,8G3C,7WVK,7UAS,7MBN,7MBM,6WJQ,6W5N,6W5M,6W5I,6UJL,6UJJ,6UJH,6UCS,6PWW,6PWV,6PG9,6PG8,6PG6,6PG3,6OI3,6OI2,6OI1,6OI0,6OFZ,6E23,6E22,6E1Z,6E1Y,6DAS,6DAR,6DAK,6DAI,6D9X,4Y7R,4GMB,4GM9,4GM8,4GM3,3P4F,2H14,2H13,8Q1N,5SXM,4CY2,4CY1,4EWR,4ESG,4ES0,4ERZ,4ERY,4ERQ,3EG6,2H6Q,2H6N,2H6K,2H68,7DNO,6U8B,6U80,6U6W,5VFC,3EMH,7BCY,2G99,6IAM,8E9F,7U9Y,6DYA,2G9A,8HMX,6UOZ,6UJ4,6UIK,6UIF,6UHZ,6UHY,6U8O,6U8L,6U5Y,6U5M,6DY7,7JTP,7JTO,6BYN,3MXX,3N0E,6PGF,6PGE,6PGD,6PGC,6PGB,6PGA,6PG7,6PG5,6PG4,3N0D,8BB5,8BB4,8BB3,8BB2	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51570937	CN1CCN(CC1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cccc(CN2CCOCC2)c1	InChI=1S/C29H32F3N5O3/c1-35-7-9-37(10-8-35)26-6-5-22(21-4-2-3-20(15-21)19-36-11-13-40-14-12-36)16-25(26)34-28(39)23-18-33-27(38)17-24(23)29(30,31)32/h2-6,15-18H,7-14,19H2,1H3,(H,33,38)(H,34,39)	DJOVLOYCGXNVPI-UHFFFAOYSA-N	50164794	CHEMBL3798846::US11174250, Example Table4.1.1::US11319299, Comp. No. 57	WD repeat-containing protein 5	Homo sapiens	>40000								ChEMBL	10.1039/d3md00605k	10.7270/Q2833XH5	38389889			n/a	n/a	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50164794	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50164794&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	35Q    	4QL1	91623360	341097539		CHEMBL3798846					1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	8X3R,7CFQ,7CFP,7BED,7AXX,7AXU,7AXS,7AXQ,7AXP,6KIZ,6KIX,6KIW,6KIV,6KIU,2XL3,2XL2,2GNQ,8DU4,7UD5,8X3S,3UVO,3UVN,3UVM,3UVL,3UVK,3PSL,8OKF,4A7J,8G3E,8F93,8F1G,8G3C,7WVK,7UAS,7MBN,7MBM,6WJQ,6W5N,6W5M,6W5I,6UJL,6UJJ,6UJH,6UCS,6PWW,6PWV,6PG9,6PG8,6PG6,6PG3,6OI3,6OI2,6OI1,6OI0,6OFZ,6E23,6E22,6E1Z,6E1Y,6DAS,6DAR,6DAK,6DAI,6D9X,4Y7R,4GMB,4GM9,4GM8,4GM3,3P4F,2H14,2H13,8Q1N,5SXM,4CY2,4CY1,4EWR,4ESG,4ES0,4ERZ,4ERY,4ERQ,3EG6,2H6Q,2H6N,2H6K,2H68,7DNO,6U8B,6U80,6U6W,5VFC,3EMH,7BCY,2G99,6IAM,8E9F,7U9Y,6DYA,2G9A,8HMX,6UOZ,6UJ4,6UIK,6UIF,6UHZ,6UHY,6U8O,6U8L,6U5Y,6U5M,6DY7,7JTP,7JTO,6BYN,3MXX,3N0E,6PGF,6PGE,6PGD,6PGC,6PGB,6PGA,6PG7,6PG5,6PG4,3N0D,8BB5,8BB4,8BB3,8BB2	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51570938	CNC(=O)c1cc(cc(NS(=O)(=O)c2cc(Br)cc(Cl)c2O)c1O)C1(CCC1)C#N	InChI=1S/C19H17BrClN3O5S/c1-23-18(27)12-5-10(19(9-22)3-2-4-19)6-14(16(12)25)24-30(28,29)15-8-11(20)7-13(21)17(15)26/h5-8,24-26H,2-4H2,1H3,(H,23,27)	COYGYHFILXAMSQ-UHFFFAOYSA-N	50531074	CHEMBL4472649	WD repeat-containing protein 5	Homo sapiens	 107								ChEMBL	10.1039/d3md00605k	10.7270/Q2833XH5	38389889			n/a	n/a	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50531074	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50531074&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	Q0M    	6U5Y	145704698	440739656							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	8X3R,7CFQ,7CFP,7BED,7AXX,7AXU,7AXS,7AXQ,7AXP,6KIZ,6KIX,6KIW,6KIV,6KIU,2XL3,2XL2,2GNQ,8DU4,7UD5,8X3S,3UVO,3UVN,3UVM,3UVL,3UVK,3PSL,8OKF,4A7J,8G3E,8F93,8F1G,8G3C,7WVK,7UAS,7MBN,7MBM,6WJQ,6W5N,6W5M,6W5I,6UJL,6UJJ,6UJH,6UCS,6PWW,6PWV,6PG9,6PG8,6PG6,6PG3,6OI3,6OI2,6OI1,6OI0,6OFZ,6E23,6E22,6E1Z,6E1Y,6DAS,6DAR,6DAK,6DAI,6D9X,4Y7R,4GMB,4GM9,4GM8,4GM3,3P4F,2H14,2H13,8Q1N,5SXM,4CY2,4CY1,4EWR,4ESG,4ES0,4ERZ,4ERY,4ERQ,3EG6,2H6Q,2H6N,2H6K,2H68,7DNO,6U8B,6U80,6U6W,5VFC,3EMH,7BCY,2G99,6IAM,8E9F,7U9Y,6DYA,2G9A,8HMX,6UOZ,6UJ4,6UIK,6UIF,6UHZ,6UHY,6U8O,6U8L,6U5Y,6U5M,6DY7,7JTP,7JTO,6BYN,3MXX,3N0E,6PGF,6PGE,6PGD,6PGC,6PGB,6PGA,6PG7,6PG5,6PG4,3N0D,8BB5,8BB4,8BB3,8BB2	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51570939	CC(C)C[C@H](NC(=O)[C@H](Cc1cnc[nH]1)NC(=O)[C@@H](NC(=O)[C@H](CCC(O)=O)NC(=O)[C@@H](NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@H](C)NC(C)=O)[C@@H](C)O)C(C)C)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CO)C(N)=O	InChI=1S/C52H92N20O15/c1-25(2)20-35(47(84)66-32(13-10-18-60-51(55)56)43(80)65-31(12-8-9-17-53)44(81)70-37(23-73)41(54)78)68-48(85)36(21-30-22-59-24-62-30)69-49(86)39(26(3)4)71-46(83)34(15-16-38(76)77)67-50(87)40(28(6)74)72-45(82)33(14-11-19-61-52(57)58)64-42(79)27(5)63-29(7)75/h22,24-28,31-37,39-40,73-74H,8-21,23,53H2,1-7H3,(H2,54,78)(H,59,62)(H,63,75)(H,64,79)(H,65,80)(H,66,84)(H,67,87)(H,68,85)(H,69,86)(H,70,81)(H,71,83)(H,72,82)(H,76,77)(H4,55,56,60)(H4,57,58,61)/t27-,28+,31-,32-,33-,34-,35-,36-,37-,39-,40-/m0/s1	YABWHPOODAWVRU-RETQXLQUSA-N	50631813	CHEMBL5434345	WD repeat-containing protein 5	Homo sapiens	>40000								ChEMBL	10.1039/d3md00605k	10.7270/Q2833XH5	38389889			n/a	n/a	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50631813	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50631813&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search											1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	8X3R,7CFQ,7CFP,7BED,7AXX,7AXU,7AXS,7AXQ,7AXP,6KIZ,6KIX,6KIW,6KIV,6KIU,2XL3,2XL2,2GNQ,8DU4,7UD5,8X3S,3UVO,3UVN,3UVM,3UVL,3UVK,3PSL,8OKF,4A7J,8G3E,8F93,8F1G,8G3C,7WVK,7UAS,7MBN,7MBM,6WJQ,6W5N,6W5M,6W5I,6UJL,6UJJ,6UJH,6UCS,6PWW,6PWV,6PG9,6PG8,6PG6,6PG3,6OI3,6OI2,6OI1,6OI0,6OFZ,6E23,6E22,6E1Z,6E1Y,6DAS,6DAR,6DAK,6DAI,6D9X,4Y7R,4GMB,4GM9,4GM8,4GM3,3P4F,2H14,2H13,8Q1N,5SXM,4CY2,4CY1,4EWR,4ESG,4ES0,4ERZ,4ERY,4ERQ,3EG6,2H6Q,2H6N,2H6K,2H68,7DNO,6U8B,6U80,6U6W,5VFC,3EMH,7BCY,2G99,6IAM,8E9F,7U9Y,6DYA,2G9A,8HMX,6UOZ,6UJ4,6UIK,6UIF,6UHZ,6UHY,6U8O,6U8L,6U5Y,6U5M,6DY7,7JTP,7JTO,6BYN,3MXX,3N0E,6PGF,6PGE,6PGD,6PGC,6PGB,6PGA,6PG7,6PG5,6PG4,3N0D,8BB5,8BB4,8BB3,8BB2	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51570940	CC[C@H](C)[C@H](NC(=O)[C@H](CCC(O)=O)NC(=O)[C@H](CCC(O)=O)NC(=O)[C@H](CCC(O)=O)NC(=O)[C@H](CC(O)=O)NC(C)=O)C(=O)N[C@H]1CC(=O)NCC[C@H](NC(=O)[C@@H](NC(=O)[C@@H](NC1=O)C(C)C)C(C)C)C(=O)N[C@@H](C(C)C)C(=O)N[C@@H](CCC(O)=O)C(N)=O	InChI=1S/C55H87N13O23/c1-10-26(8)44(68-48(84)31(14-18-39(77)78)61-46(82)29(12-16-37(73)74)60-47(83)30(13-17-38(75)76)62-50(86)34(22-40(79)80)58-27(9)69)55(91)64-33-21-35(70)57-20-19-32(63-53(89)42(24(4)5)67-54(90)43(25(6)7)66-51(33)87)49(85)65-41(23(2)3)52(88)59-28(45(56)81)11-15-36(71)72/h23-26,28-34,41-44H,10-22H2,1-9H3,(H2,56,81)(H,57,70)(H,58,69)(H,59,88)(H,60,83)(H,61,82)(H,62,86)(H,63,89)(H,64,91)(H,65,85)(H,66,87)(H,67,90)(H,68,84)(H,71,72)(H,73,74)(H,75,76)(H,77,78)(H,79,80)/t26-,28-,29-,30-,31-,32-,33-,34-,41-,42-,43-,44-/m0/s1	CYWWYCJTGSTQEL-XWYYWFNKSA-N	50631814	CHEMBL5435898	WD repeat-containing protein 5	Homo sapiens	 387								ChEMBL	10.1039/d3md00605k	10.7270/Q2833XH5	38389889			n/a	n/a	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50631814	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50631814&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search											1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	8X3R,7CFQ,7CFP,7BED,7AXX,7AXU,7AXS,7AXQ,7AXP,6KIZ,6KIX,6KIW,6KIV,6KIU,2XL3,2XL2,2GNQ,8DU4,7UD5,8X3S,3UVO,3UVN,3UVM,3UVL,3UVK,3PSL,8OKF,4A7J,8G3E,8F93,8F1G,8G3C,7WVK,7UAS,7MBN,7MBM,6WJQ,6W5N,6W5M,6W5I,6UJL,6UJJ,6UJH,6UCS,6PWW,6PWV,6PG9,6PG8,6PG6,6PG3,6OI3,6OI2,6OI1,6OI0,6OFZ,6E23,6E22,6E1Z,6E1Y,6DAS,6DAR,6DAK,6DAI,6D9X,4Y7R,4GMB,4GM9,4GM8,4GM3,3P4F,2H14,2H13,8Q1N,5SXM,4CY2,4CY1,4EWR,4ESG,4ES0,4ERZ,4ERY,4ERQ,3EG6,2H6Q,2H6N,2H6K,2H68,7DNO,6U8B,6U80,6U6W,5VFC,3EMH,7BCY,2G99,6IAM,8E9F,7U9Y,6DYA,2G9A,8HMX,6UOZ,6UJ4,6UIK,6UIF,6UHZ,6UHY,6U8O,6U8L,6U5Y,6U5M,6DY7,7JTP,7JTO,6BYN,3MXX,3N0E,6PGF,6PGE,6PGD,6PGC,6PGB,6PGA,6PG7,6PG5,6PG4,3N0D,8BB5,8BB4,8BB3,8BB2	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51570288	CN1CCN(CC1)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cccc(CN2CCOCC2)c1	InChI=1S/C29H32F3N5O3/c1-35-7-9-37(10-8-35)26-6-5-22(21-4-2-3-20(15-21)19-36-11-13-40-14-12-36)16-25(26)34-28(39)23-18-33-27(38)17-24(23)29(30,31)32/h2-6,15-18H,7-14,19H2,1H3,(H,33,38)(H,34,39)	DJOVLOYCGXNVPI-UHFFFAOYSA-N	50164794	CHEMBL3798846::US11174250, Example Table4.1.1::US11319299, Comp. No. 57	WD repeat-containing protein 5	Homo sapiens	 30								ChEMBL	10.1021/acs.jmedchem.3c01529	10.7270/Q2KH0SSW	38085679			n/a	n/a	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50164794	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50164794&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	35Q    	4QL1	91623360	341097539		CHEMBL3798846					1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	8X3R,7CFQ,7CFP,7BED,7AXX,7AXU,7AXS,7AXQ,7AXP,6KIZ,6KIX,6KIW,6KIV,6KIU,2XL3,2XL2,2GNQ,8DU4,7UD5,8X3S,3UVO,3UVN,3UVM,3UVL,3UVK,3PSL,8OKF,4A7J,8G3E,8F93,8F1G,8G3C,7WVK,7UAS,7MBN,7MBM,6WJQ,6W5N,6W5M,6W5I,6UJL,6UJJ,6UJH,6UCS,6PWW,6PWV,6PG9,6PG8,6PG6,6PG3,6OI3,6OI2,6OI1,6OI0,6OFZ,6E23,6E22,6E1Z,6E1Y,6DAS,6DAR,6DAK,6DAI,6D9X,4Y7R,4GMB,4GM9,4GM8,4GM3,3P4F,2H14,2H13,8Q1N,5SXM,4CY2,4CY1,4EWR,4ESG,4ES0,4ERZ,4ERY,4ERQ,3EG6,2H6Q,2H6N,2H6K,2H68,7DNO,6U8B,6U80,6U6W,5VFC,3EMH,7BCY,2G99,6IAM,8E9F,7U9Y,6DYA,2G9A,8HMX,6UOZ,6UJ4,6UIK,6UIF,6UHZ,6UHY,6U8O,6U8L,6U5Y,6U5M,6DY7,7JTP,7JTO,6BYN,3MXX,3N0E,6PGF,6PGE,6PGD,6PGC,6PGB,6PGA,6PG7,6PG5,6PG4,3N0D,8BB5,8BB4,8BB3,8BB2	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51570289	C[C@H](NC(=O)[C@@H]1C[C@@H](O)CN1C(=O)[C@@H](NC(=O)CNC(=O)c1ccc(F)c(c1)-c1ccc(N2C[C@H](C)N(C)[C@H](C)C2)c(NC(=O)c2c[nH]c(=O)cc2C(F)(F)F)c1)C(C)(C)C)c1ccc(cc1)-c1scnc1C	InChI=1S/C52H59F4N9O7S/c1-27-23-64(24-28(2)63(27)8)41-16-14-33(18-40(41)61-48(70)37-21-57-43(67)20-38(37)52(54,55)56)36-17-34(13-15-39(36)53)47(69)58-22-44(68)62-46(51(5,6)7)50(72)65-25-35(66)19-42(65)49(71)60-29(3)31-9-11-32(12-10-31)45-30(4)59-26-73-45/h9-18,20-21,26-29,35,42,46,66H,19,22-25H2,1-8H3,(H,57,67)(H,58,69)(H,60,71)(H,61,70)(H,62,68)/t27-,28+,29-,35+,42-,46+/m0/s1	HBHSDSLZXDASLT-FLKKWHKHSA-N	50631529	CHEMBL5415680	WD repeat-containing protein 5	Homo sapiens				 4.0					ChEMBL	10.1021/acs.jmedchem.3c01529	10.7270/Q2KH0SSW	38085679			n/a	n/a	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50631529	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50631529&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	X6M    	7JTP									1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	8X3R,7CFQ,7CFP,7BED,7AXX,7AXU,7AXS,7AXQ,7AXP,6KIZ,6KIX,6KIW,6KIV,6KIU,2XL3,2XL2,2GNQ,8DU4,7UD5,8X3S,3UVO,3UVN,3UVM,3UVL,3UVK,3PSL,8OKF,4A7J,8G3E,8F93,8F1G,8G3C,7WVK,7UAS,7MBN,7MBM,6WJQ,6W5N,6W5M,6W5I,6UJL,6UJJ,6UJH,6UCS,6PWW,6PWV,6PG9,6PG8,6PG6,6PG3,6OI3,6OI2,6OI1,6OI0,6OFZ,6E23,6E22,6E1Z,6E1Y,6DAS,6DAR,6DAK,6DAI,6D9X,4Y7R,4GMB,4GM9,4GM8,4GM3,3P4F,2H14,2H13,8Q1N,5SXM,4CY2,4CY1,4EWR,4ESG,4ES0,4ERZ,4ERY,4ERQ,3EG6,2H6Q,2H6N,2H6K,2H68,7DNO,6U8B,6U80,6U6W,5VFC,3EMH,7BCY,2G99,6IAM,8E9F,7U9Y,6DYA,2G9A,8HMX,6UOZ,6UJ4,6UIK,6UIF,6UHZ,6UHY,6U8O,6U8L,6U5Y,6U5M,6DY7,7JTP,7JTO,6BYN,3MXX,3N0E,6PGF,6PGE,6PGD,6PGC,6PGB,6PGA,6PG7,6PG5,6PG4,3N0D,8BB5,8BB4,8BB3,8BB2	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51570290	COc1cc(CNC(=O)c2cc(Cn3ccn(C)c3=N)cc(c2)-c2ccc(F)cc2C)cc(OC)c1	InChI=1S/C28H29FN4O3/c1-18-9-23(29)5-6-26(18)21-10-20(17-33-8-7-32(2)28(33)30)11-22(14-21)27(34)31-16-19-12-24(35-3)15-25(13-19)36-4/h5-15,30H,16-17H2,1-4H3,(H,31,34)	PSABMKXBOJUOBD-UHFFFAOYSA-N	50520130	CHEMBL4435250	WD repeat-containing protein 5	Homo sapiens	 0.049000								ChEMBL	10.1021/acs.jmedchem.3c01529	10.7270/Q2KH0SSW	38085679			n/a	n/a	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50520130	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50520130&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	Q6S    	6UFX	145946119	440728712							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	8X3R,7CFQ,7CFP,7BED,7AXX,7AXU,7AXS,7AXQ,7AXP,6KIZ,6KIX,6KIW,6KIV,6KIU,2XL3,2XL2,2GNQ,8DU4,7UD5,8X3S,3UVO,3UVN,3UVM,3UVL,3UVK,3PSL,8OKF,4A7J,8G3E,8F93,8F1G,8G3C,7WVK,7UAS,7MBN,7MBM,6WJQ,6W5N,6W5M,6W5I,6UJL,6UJJ,6UJH,6UCS,6PWW,6PWV,6PG9,6PG8,6PG6,6PG3,6OI3,6OI2,6OI1,6OI0,6OFZ,6E23,6E22,6E1Z,6E1Y,6DAS,6DAR,6DAK,6DAI,6D9X,4Y7R,4GMB,4GM9,4GM8,4GM3,3P4F,2H14,2H13,8Q1N,5SXM,4CY2,4CY1,4EWR,4ESG,4ES0,4ERZ,4ERY,4ERQ,3EG6,2H6Q,2H6N,2H6K,2H68,7DNO,6U8B,6U80,6U6W,5VFC,3EMH,7BCY,2G99,6IAM,8E9F,7U9Y,6DYA,2G9A,8HMX,6UOZ,6UJ4,6UIK,6UIF,6UHZ,6UHY,6U8O,6U8L,6U5Y,6U5M,6DY7,7JTP,7JTO,6BYN,3MXX,3N0E,6PGF,6PGE,6PGD,6PGC,6PGB,6PGA,6PG7,6PG5,6PG4,3N0D,8BB5,8BB4,8BB3,8BB2	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51569346	C[C@H]1CN(C[C@@H](C)N1C)c1ccc(cc1NC(=O)c1c[nH]c(=O)cc1C(F)(F)F)-c1cc(ccc1F)C(=O)NCC(=O)N[C@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)NCc1ccc(cc1)-c1scnc1C)C(C)(C)C	InChI=1S/C51H57F4N9O7S/c1-27-23-63(24-28(2)62(27)7)40-15-13-32(17-39(40)60-47(69)36-21-56-42(66)19-37(36)51(53,54)55)35-16-33(12-14-38(35)52)46(68)58-22-43(67)61-45(50(4,5)6)49(71)64-25-34(65)18-41(64)48(70)57-20-30-8-10-31(11-9-30)44-29(3)59-26-72-44/h8-17,19,21,26-28,34,41,45,65H,18,20,22-25H2,1-7H3,(H,56,66)(H,57,70)(H,58,68)(H,60,69)(H,61,67)/t27-,28+,34-,41+,45-/m1/s1	OJCYPKZNPSJLGY-KQNJQULYSA-N	50631212	CHEMBL5417352	WD repeat-containing protein 5	Homo sapiens			 122						ChEMBL	10.1021/acs.jmedchem.3c01521	10.7270/Q2HQ44CM	38019706			n/a	n/a	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50631212	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50631212&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search											1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	8X3R,7CFQ,7CFP,7BED,7AXX,7AXU,7AXS,7AXQ,7AXP,6KIZ,6KIX,6KIW,6KIV,6KIU,2XL3,2XL2,2GNQ,8DU4,7UD5,8X3S,3UVO,3UVN,3UVM,3UVL,3UVK,3PSL,8OKF,4A7J,8G3E,8F93,8F1G,8G3C,7WVK,7UAS,7MBN,7MBM,6WJQ,6W5N,6W5M,6W5I,6UJL,6UJJ,6UJH,6UCS,6PWW,6PWV,6PG9,6PG8,6PG6,6PG3,6OI3,6OI2,6OI1,6OI0,6OFZ,6E23,6E22,6E1Z,6E1Y,6DAS,6DAR,6DAK,6DAI,6D9X,4Y7R,4GMB,4GM9,4GM8,4GM3,3P4F,2H14,2H13,8Q1N,5SXM,4CY2,4CY1,4EWR,4ESG,4ES0,4ERZ,4ERY,4ERQ,3EG6,2H6Q,2H6N,2H6K,2H68,7DNO,6U8B,6U80,6U6W,5VFC,3EMH,7BCY,2G99,6IAM,8E9F,7U9Y,6DYA,2G9A,8HMX,6UOZ,6UJ4,6UIK,6UIF,6UHZ,6UHY,6U8O,6U8L,6U5Y,6U5M,6DY7,7JTP,7JTO,6BYN,3MXX,3N0E,6PGF,6PGE,6PGD,6PGC,6PGB,6PGA,6PG7,6PG5,6PG4,3N0D,8BB5,8BB4,8BB3,8BB2	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51570291	COc1cc(CN2Cc3c(cc(Cn4ccn(C)c4=N)cc3-c3ccc(F)cc3C)C2=O)cc(OC)c1	InChI=1S/C29H29FN4O3/c1-18-9-21(30)5-6-24(18)25-12-20(15-33-8-7-32(2)29(33)31)13-26-27(25)17-34(28(26)35)16-19-10-22(36-3)14-23(11-19)37-4/h5-14,31H,15-17H2,1-4H3	GTGSQXJNKTZDSD-UHFFFAOYSA-N	50631530	CHEMBL5440410	WD repeat-containing protein 5	Homo sapiens	 0.570000								ChEMBL	10.1021/acs.jmedchem.3c01529	10.7270/Q2KH0SSW	38085679			n/a	n/a	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50631530	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50631530&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search											1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	8X3R,7CFQ,7CFP,7BED,7AXX,7AXU,7AXS,7AXQ,7AXP,6KIZ,6KIX,6KIW,6KIV,6KIU,2XL3,2XL2,2GNQ,8DU4,7UD5,8X3S,3UVO,3UVN,3UVM,3UVL,3UVK,3PSL,8OKF,4A7J,8G3E,8F93,8F1G,8G3C,7WVK,7UAS,7MBN,7MBM,6WJQ,6W5N,6W5M,6W5I,6UJL,6UJJ,6UJH,6UCS,6PWW,6PWV,6PG9,6PG8,6PG6,6PG3,6OI3,6OI2,6OI1,6OI0,6OFZ,6E23,6E22,6E1Z,6E1Y,6DAS,6DAR,6DAK,6DAI,6D9X,4Y7R,4GMB,4GM9,4GM8,4GM3,3P4F,2H14,2H13,8Q1N,5SXM,4CY2,4CY1,4EWR,4ESG,4ES0,4ERZ,4ERY,4ERQ,3EG6,2H6Q,2H6N,2H6K,2H68,7DNO,6U8B,6U80,6U6W,5VFC,3EMH,7BCY,2G99,6IAM,8E9F,7U9Y,6DYA,2G9A,8HMX,6UOZ,6UJ4,6UIK,6UIF,6UHZ,6UHY,6U8O,6U8L,6U5Y,6U5M,6DY7,7JTP,7JTO,6BYN,3MXX,3N0E,6PGF,6PGE,6PGD,6PGC,6PGB,6PGA,6PG7,6PG5,6PG4,3N0D,8BB5,8BB4,8BB3,8BB2	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51570292	COc1cc(CN2CCc3c(cc(Cn4ccn(C)c4=N)cc3-c3ccc(F)cc3C)C2=O)cc(OC)c1	InChI=1S/C30H31FN4O3/c1-19-11-22(31)5-6-25(19)27-14-21(18-35-10-9-33(2)30(35)32)15-28-26(27)7-8-34(29(28)36)17-20-12-23(37-3)16-24(13-20)38-4/h5-6,9-16,32H,7-8,17-18H2,1-4H3	PKONCIPMLLIAIL-UHFFFAOYSA-N	50520131	CHEMBL4588661	WD repeat-containing protein 5	Homo sapiens	<0.020000								ChEMBL	10.1021/acs.jmedchem.3c01529	10.7270/Q2KH0SSW	38085679			n/a	n/a	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50520131	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50520131&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			146014479	440728713							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	8X3R,7CFQ,7CFP,7BED,7AXX,7AXU,7AXS,7AXQ,7AXP,6KIZ,6KIX,6KIW,6KIV,6KIU,2XL3,2XL2,2GNQ,8DU4,7UD5,8X3S,3UVO,3UVN,3UVM,3UVL,3UVK,3PSL,8OKF,4A7J,8G3E,8F93,8F1G,8G3C,7WVK,7UAS,7MBN,7MBM,6WJQ,6W5N,6W5M,6W5I,6UJL,6UJJ,6UJH,6UCS,6PWW,6PWV,6PG9,6PG8,6PG6,6PG3,6OI3,6OI2,6OI1,6OI0,6OFZ,6E23,6E22,6E1Z,6E1Y,6DAS,6DAR,6DAK,6DAI,6D9X,4Y7R,4GMB,4GM9,4GM8,4GM3,3P4F,2H14,2H13,8Q1N,5SXM,4CY2,4CY1,4EWR,4ESG,4ES0,4ERZ,4ERY,4ERQ,3EG6,2H6Q,2H6N,2H6K,2H68,7DNO,6U8B,6U80,6U6W,5VFC,3EMH,7BCY,2G99,6IAM,8E9F,7U9Y,6DYA,2G9A,8HMX,6UOZ,6UJ4,6UIK,6UIF,6UHZ,6UHY,6U8O,6U8L,6U5Y,6U5M,6DY7,7JTP,7JTO,6BYN,3MXX,3N0E,6PGF,6PGE,6PGD,6PGC,6PGB,6PGA,6PG7,6PG5,6PG4,3N0D,8BB5,8BB4,8BB3,8BB2	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51570293	COc1cc(CN2CCCc3c(cc(Cn4ccn(C)c4=N)cc3C2=O)-c2ccc(F)cc2C)cc(OC)c1	InChI=1S/C31H33FN4O3/c1-20-12-23(32)7-8-26(20)28-15-22(19-36-11-10-34(2)31(36)33)16-29-27(28)6-5-9-35(30(29)37)18-21-13-24(38-3)17-25(14-21)39-4/h7-8,10-17,33H,5-6,9,18-19H2,1-4H3	FVAXSVKVQVTTEZ-UHFFFAOYSA-N	50631531	CHEMBL5431390	WD repeat-containing protein 5	Homo sapiens	 0.037000								ChEMBL	10.1021/acs.jmedchem.3c01529	10.7270/Q2KH0SSW	38085679			n/a	n/a	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50631531	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50631531&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search											1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	8X3R,7CFQ,7CFP,7BED,7AXX,7AXU,7AXS,7AXQ,7AXP,6KIZ,6KIX,6KIW,6KIV,6KIU,2XL3,2XL2,2GNQ,8DU4,7UD5,8X3S,3UVO,3UVN,3UVM,3UVL,3UVK,3PSL,8OKF,4A7J,8G3E,8F93,8F1G,8G3C,7WVK,7UAS,7MBN,7MBM,6WJQ,6W5N,6W5M,6W5I,6UJL,6UJJ,6UJH,6UCS,6PWW,6PWV,6PG9,6PG8,6PG6,6PG3,6OI3,6OI2,6OI1,6OI0,6OFZ,6E23,6E22,6E1Z,6E1Y,6DAS,6DAR,6DAK,6DAI,6D9X,4Y7R,4GMB,4GM9,4GM8,4GM3,3P4F,2H14,2H13,8Q1N,5SXM,4CY2,4CY1,4EWR,4ESG,4ES0,4ERZ,4ERY,4ERQ,3EG6,2H6Q,2H6N,2H6K,2H68,7DNO,6U8B,6U80,6U6W,5VFC,3EMH,7BCY,2G99,6IAM,8E9F,7U9Y,6DYA,2G9A,8HMX,6UOZ,6UJ4,6UIK,6UIF,6UHZ,6UHY,6U8O,6U8L,6U5Y,6U5M,6DY7,7JTP,7JTO,6BYN,3MXX,3N0E,6PGF,6PGE,6PGD,6PGC,6PGB,6PGA,6PG7,6PG5,6PG4,3N0D,8BB5,8BB4,8BB3,8BB2	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51570294	COc1cc(CN2COc3c(cc(Cn4ccn(C)c4=N)cc3-c3ccc(F)cc3C)C2=O)cc(OC)c1	InChI=1S/C29H29FN4O4/c1-18-9-21(30)5-6-24(18)25-12-20(15-33-8-7-32(2)29(33)31)13-26-27(25)38-17-34(28(26)35)16-19-10-22(36-3)14-23(11-19)37-4/h5-14,31H,15-17H2,1-4H3	ORUSYCGZISHLQU-UHFFFAOYSA-N	50631532	CHEMBL5401714	WD repeat-containing protein 5	Homo sapiens	 0.051000								ChEMBL	10.1021/acs.jmedchem.3c01529	10.7270/Q2KH0SSW	38085679			n/a	n/a	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50631532	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50631532&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search											1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	8X3R,7CFQ,7CFP,7BED,7AXX,7AXU,7AXS,7AXQ,7AXP,6KIZ,6KIX,6KIW,6KIV,6KIU,2XL3,2XL2,2GNQ,8DU4,7UD5,8X3S,3UVO,3UVN,3UVM,3UVL,3UVK,3PSL,8OKF,4A7J,8G3E,8F93,8F1G,8G3C,7WVK,7UAS,7MBN,7MBM,6WJQ,6W5N,6W5M,6W5I,6UJL,6UJJ,6UJH,6UCS,6PWW,6PWV,6PG9,6PG8,6PG6,6PG3,6OI3,6OI2,6OI1,6OI0,6OFZ,6E23,6E22,6E1Z,6E1Y,6DAS,6DAR,6DAK,6DAI,6D9X,4Y7R,4GMB,4GM9,4GM8,4GM3,3P4F,2H14,2H13,8Q1N,5SXM,4CY2,4CY1,4EWR,4ESG,4ES0,4ERZ,4ERY,4ERQ,3EG6,2H6Q,2H6N,2H6K,2H68,7DNO,6U8B,6U80,6U6W,5VFC,3EMH,7BCY,2G99,6IAM,8E9F,7U9Y,6DYA,2G9A,8HMX,6UOZ,6UJ4,6UIK,6UIF,6UHZ,6UHY,6U8O,6U8L,6U5Y,6U5M,6DY7,7JTP,7JTO,6BYN,3MXX,3N0E,6PGF,6PGE,6PGD,6PGC,6PGB,6PGA,6PG7,6PG5,6PG4,3N0D,8BB5,8BB4,8BB3,8BB2	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51570295	COc1cc(Cn2cnc3c(cc(Cn4ccn(C)c4=N)cc3c2=O)-c2ccc(F)cc2C)cc(OC)c1	InChI=1S/C29H28FN5O3/c1-18-9-21(30)5-6-24(18)25-12-20(15-34-8-7-33(2)29(34)31)13-26-27(25)32-17-35(28(26)36)16-19-10-22(37-3)14-23(11-19)38-4/h5-14,17,31H,15-16H2,1-4H3	XUJQZQBHCJAMSU-UHFFFAOYSA-N	50631533	CHEMBL5434280	WD repeat-containing protein 5	Homo sapiens	 0.079000								ChEMBL	10.1021/acs.jmedchem.3c01529	10.7270/Q2KH0SSW	38085679			n/a	n/a	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50631533	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50631533&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search											1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	8X3R,7CFQ,7CFP,7BED,7AXX,7AXU,7AXS,7AXQ,7AXP,6KIZ,6KIX,6KIW,6KIV,6KIU,2XL3,2XL2,2GNQ,8DU4,7UD5,8X3S,3UVO,3UVN,3UVM,3UVL,3UVK,3PSL,8OKF,4A7J,8G3E,8F93,8F1G,8G3C,7WVK,7UAS,7MBN,7MBM,6WJQ,6W5N,6W5M,6W5I,6UJL,6UJJ,6UJH,6UCS,6PWW,6PWV,6PG9,6PG8,6PG6,6PG3,6OI3,6OI2,6OI1,6OI0,6OFZ,6E23,6E22,6E1Z,6E1Y,6DAS,6DAR,6DAK,6DAI,6D9X,4Y7R,4GMB,4GM9,4GM8,4GM3,3P4F,2H14,2H13,8Q1N,5SXM,4CY2,4CY1,4EWR,4ESG,4ES0,4ERZ,4ERY,4ERQ,3EG6,2H6Q,2H6N,2H6K,2H68,7DNO,6U8B,6U80,6U6W,5VFC,3EMH,7BCY,2G99,6IAM,8E9F,7U9Y,6DYA,2G9A,8HMX,6UOZ,6UJ4,6UIK,6UIF,6UHZ,6UHY,6U8O,6U8L,6U5Y,6U5M,6DY7,7JTP,7JTO,6BYN,3MXX,3N0E,6PGF,6PGE,6PGD,6PGC,6PGB,6PGA,6PG7,6PG5,6PG4,3N0D,8BB5,8BB4,8BB3,8BB2	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51570296	COc1cc(CN2CNc3c(cc(Cn4ccn(C)c4=N)cc3-c3ccc(F)cc3C)C2=O)cc(OC)c1	InChI=1S/C29H30FN5O3/c1-18-9-21(30)5-6-24(18)25-12-20(15-34-8-7-33(2)29(34)31)13-26-27(25)32-17-35(28(26)36)16-19-10-22(37-3)14-23(11-19)38-4/h5-14,31-32H,15-17H2,1-4H3	BKDGXFQGTYBNAT-UHFFFAOYSA-N	50631534	CHEMBL5398302	WD repeat-containing protein 5	Homo sapiens	 0.026000								ChEMBL	10.1021/acs.jmedchem.3c01529	10.7270/Q2KH0SSW	38085679			n/a	n/a	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50631534	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50631534&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search											1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	8X3R,7CFQ,7CFP,7BED,7AXX,7AXU,7AXS,7AXQ,7AXP,6KIZ,6KIX,6KIW,6KIV,6KIU,2XL3,2XL2,2GNQ,8DU4,7UD5,8X3S,3UVO,3UVN,3UVM,3UVL,3UVK,3PSL,8OKF,4A7J,8G3E,8F93,8F1G,8G3C,7WVK,7UAS,7MBN,7MBM,6WJQ,6W5N,6W5M,6W5I,6UJL,6UJJ,6UJH,6UCS,6PWW,6PWV,6PG9,6PG8,6PG6,6PG3,6OI3,6OI2,6OI1,6OI0,6OFZ,6E23,6E22,6E1Z,6E1Y,6DAS,6DAR,6DAK,6DAI,6D9X,4Y7R,4GMB,4GM9,4GM8,4GM3,3P4F,2H14,2H13,8Q1N,5SXM,4CY2,4CY1,4EWR,4ESG,4ES0,4ERZ,4ERY,4ERQ,3EG6,2H6Q,2H6N,2H6K,2H68,7DNO,6U8B,6U80,6U6W,5VFC,3EMH,7BCY,2G99,6IAM,8E9F,7U9Y,6DYA,2G9A,8HMX,6UOZ,6UJ4,6UIK,6UIF,6UHZ,6UHY,6U8O,6U8L,6U5Y,6U5M,6DY7,7JTP,7JTO,6BYN,3MXX,3N0E,6PGF,6PGE,6PGD,6PGC,6PGB,6PGA,6PG7,6PG5,6PG4,3N0D,8BB5,8BB4,8BB3,8BB2	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51570297	COc1cc(CN2CCOc3c(cc(Cn4ccn(C)c4=N)cc3C2=O)-c2ccc(F)cc2C)cc(OC)c1	InChI=1S/C30H31FN4O4/c1-19-11-22(31)5-6-25(19)26-14-21(18-35-8-7-33(2)30(35)32)15-27-28(26)39-10-9-34(29(27)36)17-20-12-23(37-3)16-24(13-20)38-4/h5-8,11-16,32H,9-10,17-18H2,1-4H3	KLFBZLMEAVVEOS-UHFFFAOYSA-N	50631535	CHEMBL5398730	WD repeat-containing protein 5	Homo sapiens	 0.023000								ChEMBL	10.1021/acs.jmedchem.3c01529	10.7270/Q2KH0SSW	38085679			n/a	n/a	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50631535	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50631535&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	VV3    	8UJY									1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	8X3R,7CFQ,7CFP,7BED,7AXX,7AXU,7AXS,7AXQ,7AXP,6KIZ,6KIX,6KIW,6KIV,6KIU,2XL3,2XL2,2GNQ,8DU4,7UD5,8X3S,3UVO,3UVN,3UVM,3UVL,3UVK,3PSL,8OKF,4A7J,8G3E,8F93,8F1G,8G3C,7WVK,7UAS,7MBN,7MBM,6WJQ,6W5N,6W5M,6W5I,6UJL,6UJJ,6UJH,6UCS,6PWW,6PWV,6PG9,6PG8,6PG6,6PG3,6OI3,6OI2,6OI1,6OI0,6OFZ,6E23,6E22,6E1Z,6E1Y,6DAS,6DAR,6DAK,6DAI,6D9X,4Y7R,4GMB,4GM9,4GM8,4GM3,3P4F,2H14,2H13,8Q1N,5SXM,4CY2,4CY1,4EWR,4ESG,4ES0,4ERZ,4ERY,4ERQ,3EG6,2H6Q,2H6N,2H6K,2H68,7DNO,6U8B,6U80,6U6W,5VFC,3EMH,7BCY,2G99,6IAM,8E9F,7U9Y,6DYA,2G9A,8HMX,6UOZ,6UJ4,6UIK,6UIF,6UHZ,6UHY,6U8O,6U8L,6U5Y,6U5M,6DY7,7JTP,7JTO,6BYN,3MXX,3N0E,6PGF,6PGE,6PGD,6PGC,6PGB,6PGA,6PG7,6PG5,6PG4,3N0D,8BB5,8BB4,8BB3,8BB2	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51570298	COc1cc(CN2CC(=O)Nc3c(cc(Cn4ccn(C)c4=N)cc3C2=O)-c2ccc(F)cc2C)cc(OC)c1	InChI=1S/C30H30FN5O4/c1-18-9-21(31)5-6-24(18)25-12-20(15-35-8-7-34(2)30(35)32)13-26-28(25)33-27(37)17-36(29(26)38)16-19-10-22(39-3)14-23(11-19)40-4/h5-14,32H,15-17H2,1-4H3,(H,33,37)	LYDQZWAZFFPXAQ-UHFFFAOYSA-N	50631536	CHEMBL5404726	WD repeat-containing protein 5	Homo sapiens	 0.100000								ChEMBL	10.1021/acs.jmedchem.3c01529	10.7270/Q2KH0SSW	38085679			n/a	n/a	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50631536	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50631536&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search											1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	8X3R,7CFQ,7CFP,7BED,7AXX,7AXU,7AXS,7AXQ,7AXP,6KIZ,6KIX,6KIW,6KIV,6KIU,2XL3,2XL2,2GNQ,8DU4,7UD5,8X3S,3UVO,3UVN,3UVM,3UVL,3UVK,3PSL,8OKF,4A7J,8G3E,8F93,8F1G,8G3C,7WVK,7UAS,7MBN,7MBM,6WJQ,6W5N,6W5M,6W5I,6UJL,6UJJ,6UJH,6UCS,6PWW,6PWV,6PG9,6PG8,6PG6,6PG3,6OI3,6OI2,6OI1,6OI0,6OFZ,6E23,6E22,6E1Z,6E1Y,6DAS,6DAR,6DAK,6DAI,6D9X,4Y7R,4GMB,4GM9,4GM8,4GM3,3P4F,2H14,2H13,8Q1N,5SXM,4CY2,4CY1,4EWR,4ESG,4ES0,4ERZ,4ERY,4ERQ,3EG6,2H6Q,2H6N,2H6K,2H68,7DNO,6U8B,6U80,6U6W,5VFC,3EMH,7BCY,2G99,6IAM,8E9F,7U9Y,6DYA,2G9A,8HMX,6UOZ,6UJ4,6UIK,6UIF,6UHZ,6UHY,6U8O,6U8L,6U5Y,6U5M,6DY7,7JTP,7JTO,6BYN,3MXX,3N0E,6PGF,6PGE,6PGD,6PGC,6PGB,6PGA,6PG7,6PG5,6PG4,3N0D,8BB5,8BB4,8BB3,8BB2	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51570299	COc1cc(CN2CCNc3c(cc(Cn4ccn(C)c4=N)cc3C2=O)-c2ccc(F)cc2C)cc(OC)c1	InChI=1S/C30H32FN5O3/c1-19-11-22(31)5-6-25(19)26-14-21(18-36-10-9-34(2)30(36)32)15-27-28(26)33-7-8-35(29(27)37)17-20-12-23(38-3)16-24(13-20)39-4/h5-6,9-16,32-33H,7-8,17-18H2,1-4H3	LHOMSBUTZVALQI-UHFFFAOYSA-N	50631537	CHEMBL5425914	WD repeat-containing protein 5	Homo sapiens	 0.047000								ChEMBL	10.1021/acs.jmedchem.3c01529	10.7270/Q2KH0SSW	38085679			n/a	n/a	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50631537	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50631537&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search											1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	8X3R,7CFQ,7CFP,7BED,7AXX,7AXU,7AXS,7AXQ,7AXP,6KIZ,6KIX,6KIW,6KIV,6KIU,2XL3,2XL2,2GNQ,8DU4,7UD5,8X3S,3UVO,3UVN,3UVM,3UVL,3UVK,3PSL,8OKF,4A7J,8G3E,8F93,8F1G,8G3C,7WVK,7UAS,7MBN,7MBM,6WJQ,6W5N,6W5M,6W5I,6UJL,6UJJ,6UJH,6UCS,6PWW,6PWV,6PG9,6PG8,6PG6,6PG3,6OI3,6OI2,6OI1,6OI0,6OFZ,6E23,6E22,6E1Z,6E1Y,6DAS,6DAR,6DAK,6DAI,6D9X,4Y7R,4GMB,4GM9,4GM8,4GM3,3P4F,2H14,2H13,8Q1N,5SXM,4CY2,4CY1,4EWR,4ESG,4ES0,4ERZ,4ERY,4ERQ,3EG6,2H6Q,2H6N,2H6K,2H68,7DNO,6U8B,6U80,6U6W,5VFC,3EMH,7BCY,2G99,6IAM,8E9F,7U9Y,6DYA,2G9A,8HMX,6UOZ,6UJ4,6UIK,6UIF,6UHZ,6UHY,6U8O,6U8L,6U5Y,6U5M,6DY7,7JTP,7JTO,6BYN,3MXX,3N0E,6PGF,6PGE,6PGD,6PGC,6PGB,6PGA,6PG7,6PG5,6PG4,3N0D,8BB5,8BB4,8BB3,8BB2	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51570300	CCn1cc(c(n1)C(F)(F)F)-c1cc(Cn2ccnc2)cc2C(=O)N(CCc12)[C@@H](C1CC1)c1cc(OC)ccn1	InChI=1S/C29H29F3N6O2/c1-3-37-16-24(27(35-37)29(30,31)32)22-12-18(15-36-11-9-33-17-36)13-23-21(22)7-10-38(28(23)39)26(19-4-5-19)25-14-20(40-2)6-8-34-25/h6,8-9,11-14,16-17,19,26H,3-5,7,10,15H2,1-2H3/t26-/m0/s1	IRXFPIASUFJVNS-SANMLTNESA-N	50605355	CHEMBL5170717	WD repeat-containing protein 5	Homo sapiens	<0.020000								ChEMBL	10.1021/acs.jmedchem.3c01529	10.7270/Q2KH0SSW	38085679			n/a	n/a	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50605355	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50605355&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search			153572492	482616206							1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	8X3R,7CFQ,7CFP,7BED,7AXX,7AXU,7AXS,7AXQ,7AXP,6KIZ,6KIX,6KIW,6KIV,6KIU,2XL3,2XL2,2GNQ,8DU4,7UD5,8X3S,3UVO,3UVN,3UVM,3UVL,3UVK,3PSL,8OKF,4A7J,8G3E,8F93,8F1G,8G3C,7WVK,7UAS,7MBN,7MBM,6WJQ,6W5N,6W5M,6W5I,6UJL,6UJJ,6UJH,6UCS,6PWW,6PWV,6PG9,6PG8,6PG6,6PG3,6OI3,6OI2,6OI1,6OI0,6OFZ,6E23,6E22,6E1Z,6E1Y,6DAS,6DAR,6DAK,6DAI,6D9X,4Y7R,4GMB,4GM9,4GM8,4GM3,3P4F,2H14,2H13,8Q1N,5SXM,4CY2,4CY1,4EWR,4ESG,4ES0,4ERZ,4ERY,4ERQ,3EG6,2H6Q,2H6N,2H6K,2H68,7DNO,6U8B,6U80,6U6W,5VFC,3EMH,7BCY,2G99,6IAM,8E9F,7U9Y,6DYA,2G9A,8HMX,6UOZ,6UJ4,6UIK,6UIF,6UHZ,6UHY,6U8O,6U8L,6U5Y,6U5M,6DY7,7JTP,7JTO,6BYN,3MXX,3N0E,6PGF,6PGE,6PGD,6PGC,6PGB,6PGA,6PG7,6PG5,6PG4,3N0D,8BB5,8BB4,8BB3,8BB2	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51570301	CCn1cc(c(n1)C(F)(F)F)-c1cc(Cn2ccnc2)cc2c1OCCN([C@@H](C1CC1)c1cc(OC)ccn1)C2=O	InChI=1S/C29H29F3N6O3/c1-3-37-16-23(27(35-37)29(30,31)32)21-12-18(15-36-9-8-33-17-36)13-22-26(21)41-11-10-38(28(22)39)25(19-4-5-19)24-14-20(40-2)6-7-34-24/h6-9,12-14,16-17,19,25H,3-5,10-11,15H2,1-2H3/t25-/m0/s1	CWWDKVDXNLGSHY-VWLOTQADSA-N	50631538	CHEMBL5409903	WD repeat-containing protein 5	Homo sapiens	<0.020000								ChEMBL	10.1021/acs.jmedchem.3c01529	10.7270/Q2KH0SSW	38085679			n/a	n/a	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50631538	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50631538&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search											1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	8X3R,7CFQ,7CFP,7BED,7AXX,7AXU,7AXS,7AXQ,7AXP,6KIZ,6KIX,6KIW,6KIV,6KIU,2XL3,2XL2,2GNQ,8DU4,7UD5,8X3S,3UVO,3UVN,3UVM,3UVL,3UVK,3PSL,8OKF,4A7J,8G3E,8F93,8F1G,8G3C,7WVK,7UAS,7MBN,7MBM,6WJQ,6W5N,6W5M,6W5I,6UJL,6UJJ,6UJH,6UCS,6PWW,6PWV,6PG9,6PG8,6PG6,6PG3,6OI3,6OI2,6OI1,6OI0,6OFZ,6E23,6E22,6E1Z,6E1Y,6DAS,6DAR,6DAK,6DAI,6D9X,4Y7R,4GMB,4GM9,4GM8,4GM3,3P4F,2H14,2H13,8Q1N,5SXM,4CY2,4CY1,4EWR,4ESG,4ES0,4ERZ,4ERY,4ERQ,3EG6,2H6Q,2H6N,2H6K,2H68,7DNO,6U8B,6U80,6U6W,5VFC,3EMH,7BCY,2G99,6IAM,8E9F,7U9Y,6DYA,2G9A,8HMX,6UOZ,6UJ4,6UIK,6UIF,6UHZ,6UHY,6U8O,6U8L,6U5Y,6U5M,6DY7,7JTP,7JTO,6BYN,3MXX,3N0E,6PGF,6PGE,6PGD,6PGC,6PGB,6PGA,6PG7,6PG5,6PG4,3N0D,8BB5,8BB4,8BB3,8BB2	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51570302	CCn1cc(c(n1)C(F)(F)F)-c1cc(Cn2ccnc2)cc2C(=O)N(CNc12)[C@@H](C1CC1)c1cc(OC)ccn1	InChI=1S/C28H28F3N7O2/c1-3-37-14-22(26(35-37)28(29,30)31)20-10-17(13-36-9-8-32-15-36)11-21-24(20)34-16-38(27(21)39)25(18-4-5-18)23-12-19(40-2)6-7-33-23/h6-12,14-15,18,25,34H,3-5,13,16H2,1-2H3/t25-/m0/s1	GFMPRGZTLIKKFV-VWLOTQADSA-N	50631539	CHEMBL5417425	WD repeat-containing protein 5	Homo sapiens	<0.020000								ChEMBL	10.1021/acs.jmedchem.3c01529	10.7270/Q2KH0SSW	38085679			n/a	n/a	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50631539	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50631539&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search											1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	8X3R,7CFQ,7CFP,7BED,7AXX,7AXU,7AXS,7AXQ,7AXP,6KIZ,6KIX,6KIW,6KIV,6KIU,2XL3,2XL2,2GNQ,8DU4,7UD5,8X3S,3UVO,3UVN,3UVM,3UVL,3UVK,3PSL,8OKF,4A7J,8G3E,8F93,8F1G,8G3C,7WVK,7UAS,7MBN,7MBM,6WJQ,6W5N,6W5M,6W5I,6UJL,6UJJ,6UJH,6UCS,6PWW,6PWV,6PG9,6PG8,6PG6,6PG3,6OI3,6OI2,6OI1,6OI0,6OFZ,6E23,6E22,6E1Z,6E1Y,6DAS,6DAR,6DAK,6DAI,6D9X,4Y7R,4GMB,4GM9,4GM8,4GM3,3P4F,2H14,2H13,8Q1N,5SXM,4CY2,4CY1,4EWR,4ESG,4ES0,4ERZ,4ERY,4ERQ,3EG6,2H6Q,2H6N,2H6K,2H68,7DNO,6U8B,6U80,6U6W,5VFC,3EMH,7BCY,2G99,6IAM,8E9F,7U9Y,6DYA,2G9A,8HMX,6UOZ,6UJ4,6UIK,6UIF,6UHZ,6UHY,6U8O,6U8L,6U5Y,6U5M,6DY7,7JTP,7JTO,6BYN,3MXX,3N0E,6PGF,6PGE,6PGD,6PGC,6PGB,6PGA,6PG7,6PG5,6PG4,3N0D,8BB5,8BB4,8BB3,8BB2	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51570303	COc1cnc2cccc(N3CCc4c(cc(Cn5ccnc5)cc4C3=O)-c3cn(C)nc3C(F)(F)F)c2c1	InChI=1S/C28H23F3N6O2/c1-35-15-23(26(34-35)28(29,30)31)20-10-17(14-36-9-7-32-16-36)11-21-19(20)6-8-37(27(21)38)25-5-3-4-24-22(25)12-18(39-2)13-33-24/h3-5,7,9-13,15-16H,6,8,14H2,1-2H3	OHQJCMRWBTXWPF-UHFFFAOYSA-N	50631540	CHEMBL5422217	WD repeat-containing protein 5	Homo sapiens	 0.020000								ChEMBL	10.1021/acs.jmedchem.3c01529	10.7270/Q2KH0SSW	38085679			n/a	n/a	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50631540	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50631540&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search											1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	8X3R,7CFQ,7CFP,7BED,7AXX,7AXU,7AXS,7AXQ,7AXP,6KIZ,6KIX,6KIW,6KIV,6KIU,2XL3,2XL2,2GNQ,8DU4,7UD5,8X3S,3UVO,3UVN,3UVM,3UVL,3UVK,3PSL,8OKF,4A7J,8G3E,8F93,8F1G,8G3C,7WVK,7UAS,7MBN,7MBM,6WJQ,6W5N,6W5M,6W5I,6UJL,6UJJ,6UJH,6UCS,6PWW,6PWV,6PG9,6PG8,6PG6,6PG3,6OI3,6OI2,6OI1,6OI0,6OFZ,6E23,6E22,6E1Z,6E1Y,6DAS,6DAR,6DAK,6DAI,6D9X,4Y7R,4GMB,4GM9,4GM8,4GM3,3P4F,2H14,2H13,8Q1N,5SXM,4CY2,4CY1,4EWR,4ESG,4ES0,4ERZ,4ERY,4ERQ,3EG6,2H6Q,2H6N,2H6K,2H68,7DNO,6U8B,6U80,6U6W,5VFC,3EMH,7BCY,2G99,6IAM,8E9F,7U9Y,6DYA,2G9A,8HMX,6UOZ,6UJ4,6UIK,6UIF,6UHZ,6UHY,6U8O,6U8L,6U5Y,6U5M,6DY7,7JTP,7JTO,6BYN,3MXX,3N0E,6PGF,6PGE,6PGD,6PGC,6PGB,6PGA,6PG7,6PG5,6PG4,3N0D,8BB5,8BB4,8BB3,8BB2	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51570304	CCc1cc(OC)c2nccc(N3CCc4c(cc(Cn5ccnc5)cc4C3=O)-c3cn(C)nc3C(F)(F)F)c2c1	InChI=1S/C30H27F3N6O2/c1-4-18-11-23-25(5-7-35-27(23)26(14-18)41-3)39-9-6-20-21(24-16-37(2)36-28(24)30(31,32)33)12-19(13-22(20)29(39)40)15-38-10-8-34-17-38/h5,7-8,10-14,16-17H,4,6,9,15H2,1-3H3	GKMOABIBMOIMEJ-UHFFFAOYSA-N	50631541	CHEMBL5412813	WD repeat-containing protein 5	Homo sapiens	<0.020000								ChEMBL	10.1021/acs.jmedchem.3c01529	10.7270/Q2KH0SSW	38085679			n/a	n/a	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50631541	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50631541&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search											1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	8X3R,7CFQ,7CFP,7BED,7AXX,7AXU,7AXS,7AXQ,7AXP,6KIZ,6KIX,6KIW,6KIV,6KIU,2XL3,2XL2,2GNQ,8DU4,7UD5,8X3S,3UVO,3UVN,3UVM,3UVL,3UVK,3PSL,8OKF,4A7J,8G3E,8F93,8F1G,8G3C,7WVK,7UAS,7MBN,7MBM,6WJQ,6W5N,6W5M,6W5I,6UJL,6UJJ,6UJH,6UCS,6PWW,6PWV,6PG9,6PG8,6PG6,6PG3,6OI3,6OI2,6OI1,6OI0,6OFZ,6E23,6E22,6E1Z,6E1Y,6DAS,6DAR,6DAK,6DAI,6D9X,4Y7R,4GMB,4GM9,4GM8,4GM3,3P4F,2H14,2H13,8Q1N,5SXM,4CY2,4CY1,4EWR,4ESG,4ES0,4ERZ,4ERY,4ERQ,3EG6,2H6Q,2H6N,2H6K,2H68,7DNO,6U8B,6U80,6U6W,5VFC,3EMH,7BCY,2G99,6IAM,8E9F,7U9Y,6DYA,2G9A,8HMX,6UOZ,6UJ4,6UIK,6UIF,6UHZ,6UHY,6U8O,6U8L,6U5Y,6U5M,6DY7,7JTP,7JTO,6BYN,3MXX,3N0E,6PGF,6PGE,6PGD,6PGC,6PGB,6PGA,6PG7,6PG5,6PG4,3N0D,8BB5,8BB4,8BB3,8BB2	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51570305	COc1cnc2cccc(N3CCOc4c(cc(Cn5ccnc5)cc4C3=O)-c3cn(C)nc3C(F)(F)F)c2c1	InChI=1S/C28H23F3N6O3/c1-35-15-22(26(34-35)28(29,30)31)19-10-17(14-36-7-6-32-16-36)11-21-25(19)40-9-8-37(27(21)38)24-5-3-4-23-20(24)12-18(39-2)13-33-23/h3-7,10-13,15-16H,8-9,14H2,1-2H3	FKSTZJVXESJFRS-UHFFFAOYSA-N	50631542	CHEMBL5401138	WD repeat-containing protein 5	Homo sapiens	 0.033000								ChEMBL	10.1021/acs.jmedchem.3c01529	10.7270/Q2KH0SSW	38085679			n/a	n/a	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50631542	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50631542&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search											1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	8X3R,7CFQ,7CFP,7BED,7AXX,7AXU,7AXS,7AXQ,7AXP,6KIZ,6KIX,6KIW,6KIV,6KIU,2XL3,2XL2,2GNQ,8DU4,7UD5,8X3S,3UVO,3UVN,3UVM,3UVL,3UVK,3PSL,8OKF,4A7J,8G3E,8F93,8F1G,8G3C,7WVK,7UAS,7MBN,7MBM,6WJQ,6W5N,6W5M,6W5I,6UJL,6UJJ,6UJH,6UCS,6PWW,6PWV,6PG9,6PG8,6PG6,6PG3,6OI3,6OI2,6OI1,6OI0,6OFZ,6E23,6E22,6E1Z,6E1Y,6DAS,6DAR,6DAK,6DAI,6D9X,4Y7R,4GMB,4GM9,4GM8,4GM3,3P4F,2H14,2H13,8Q1N,5SXM,4CY2,4CY1,4EWR,4ESG,4ES0,4ERZ,4ERY,4ERQ,3EG6,2H6Q,2H6N,2H6K,2H68,7DNO,6U8B,6U80,6U6W,5VFC,3EMH,7BCY,2G99,6IAM,8E9F,7U9Y,6DYA,2G9A,8HMX,6UOZ,6UJ4,6UIK,6UIF,6UHZ,6UHY,6U8O,6U8L,6U5Y,6U5M,6DY7,7JTP,7JTO,6BYN,3MXX,3N0E,6PGF,6PGE,6PGD,6PGC,6PGB,6PGA,6PG7,6PG5,6PG4,3N0D,8BB5,8BB4,8BB3,8BB2	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51570306	CCc1cc(OC)c2nccc(N3CCOc4c(cc(Cn5ccnc5)cc4C3=O)-c3cn(C)nc3C(F)(F)F)c2c1	InChI=1S/C30H27F3N6O3/c1-4-18-11-21-24(5-6-35-26(21)25(14-18)41-3)39-9-10-42-27-20(23-16-37(2)36-28(23)30(31,32)33)12-19(13-22(27)29(39)40)15-38-8-7-34-17-38/h5-8,11-14,16-17H,4,9-10,15H2,1-3H3	FRYNOSFCEFAFOX-UHFFFAOYSA-N	50631543	CHEMBL5440128	WD repeat-containing protein 5	Homo sapiens	 0.039000								ChEMBL	10.1021/acs.jmedchem.3c01529	10.7270/Q2KH0SSW	38085679			n/a	n/a	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50631543	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50631543&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search											1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	8X3R,7CFQ,7CFP,7BED,7AXX,7AXU,7AXS,7AXQ,7AXP,6KIZ,6KIX,6KIW,6KIV,6KIU,2XL3,2XL2,2GNQ,8DU4,7UD5,8X3S,3UVO,3UVN,3UVM,3UVL,3UVK,3PSL,8OKF,4A7J,8G3E,8F93,8F1G,8G3C,7WVK,7UAS,7MBN,7MBM,6WJQ,6W5N,6W5M,6W5I,6UJL,6UJJ,6UJH,6UCS,6PWW,6PWV,6PG9,6PG8,6PG6,6PG3,6OI3,6OI2,6OI1,6OI0,6OFZ,6E23,6E22,6E1Z,6E1Y,6DAS,6DAR,6DAK,6DAI,6D9X,4Y7R,4GMB,4GM9,4GM8,4GM3,3P4F,2H14,2H13,8Q1N,5SXM,4CY2,4CY1,4EWR,4ESG,4ES0,4ERZ,4ERY,4ERQ,3EG6,2H6Q,2H6N,2H6K,2H68,7DNO,6U8B,6U80,6U6W,5VFC,3EMH,7BCY,2G99,6IAM,8E9F,7U9Y,6DYA,2G9A,8HMX,6UOZ,6UJ4,6UIK,6UIF,6UHZ,6UHY,6U8O,6U8L,6U5Y,6U5M,6DY7,7JTP,7JTO,6BYN,3MXX,3N0E,6PGF,6PGE,6PGD,6PGC,6PGB,6PGA,6PG7,6PG5,6PG4,3N0D,8BB5,8BB4,8BB3,8BB2	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51570307	CCc1cc(OC)c2nccc(N3COc4c(cc(Cn5ccnc5)cc4C3=O)-c3cn(C)nc3C(F)(F)F)c2c1	InChI=1S/C29H25F3N6O3/c1-4-17-9-20-23(5-6-34-25(20)24(12-17)40-3)38-16-41-26-19(22-14-36(2)35-27(22)29(30,31)32)10-18(11-21(26)28(38)39)13-37-8-7-33-15-37/h5-12,14-15H,4,13,16H2,1-3H3	HXBMBWNJVZICES-UHFFFAOYSA-N	50631544	CHEMBL5405792	WD repeat-containing protein 5	Homo sapiens	 0.027000								ChEMBL	10.1021/acs.jmedchem.3c01529	10.7270/Q2KH0SSW	38085679			n/a	n/a	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50631544	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50631544&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search											1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	8X3R,7CFQ,7CFP,7BED,7AXX,7AXU,7AXS,7AXQ,7AXP,6KIZ,6KIX,6KIW,6KIV,6KIU,2XL3,2XL2,2GNQ,8DU4,7UD5,8X3S,3UVO,3UVN,3UVM,3UVL,3UVK,3PSL,8OKF,4A7J,8G3E,8F93,8F1G,8G3C,7WVK,7UAS,7MBN,7MBM,6WJQ,6W5N,6W5M,6W5I,6UJL,6UJJ,6UJH,6UCS,6PWW,6PWV,6PG9,6PG8,6PG6,6PG3,6OI3,6OI2,6OI1,6OI0,6OFZ,6E23,6E22,6E1Z,6E1Y,6DAS,6DAR,6DAK,6DAI,6D9X,4Y7R,4GMB,4GM9,4GM8,4GM3,3P4F,2H14,2H13,8Q1N,5SXM,4CY2,4CY1,4EWR,4ESG,4ES0,4ERZ,4ERY,4ERQ,3EG6,2H6Q,2H6N,2H6K,2H68,7DNO,6U8B,6U80,6U6W,5VFC,3EMH,7BCY,2G99,6IAM,8E9F,7U9Y,6DYA,2G9A,8HMX,6UOZ,6UJ4,6UIK,6UIF,6UHZ,6UHY,6U8O,6U8L,6U5Y,6U5M,6DY7,7JTP,7JTO,6BYN,3MXX,3N0E,6PGF,6PGE,6PGD,6PGC,6PGB,6PGA,6PG7,6PG5,6PG4,3N0D,8BB5,8BB4,8BB3,8BB2	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51570308	COc1ccc2CCCC(N3CCOc4c(cc(Cn5ccnc5C)cc4C3=O)-c3cn(C)nc3C(F)(F)F)c2c1	InChI=1S/C30H30F3N5O3/c1-18-34-9-10-37(18)16-19-13-23(25-17-36(2)35-28(25)30(31,32)33)27-24(14-19)29(39)38(11-12-41-27)26-6-4-5-20-7-8-21(40-3)15-22(20)26/h7-10,13-15,17,26H,4-6,11-12,16H2,1-3H3	IGAOEWLHZMAHFW-UHFFFAOYSA-N	50631545	CHEMBL5414839	WD repeat-containing protein 5	Homo sapiens	 0.020000								ChEMBL	10.1021/acs.jmedchem.3c01529	10.7270/Q2KH0SSW	38085679			n/a	n/a	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50631545	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50631545&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search											1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	8X3R,7CFQ,7CFP,7BED,7AXX,7AXU,7AXS,7AXQ,7AXP,6KIZ,6KIX,6KIW,6KIV,6KIU,2XL3,2XL2,2GNQ,8DU4,7UD5,8X3S,3UVO,3UVN,3UVM,3UVL,3UVK,3PSL,8OKF,4A7J,8G3E,8F93,8F1G,8G3C,7WVK,7UAS,7MBN,7MBM,6WJQ,6W5N,6W5M,6W5I,6UJL,6UJJ,6UJH,6UCS,6PWW,6PWV,6PG9,6PG8,6PG6,6PG3,6OI3,6OI2,6OI1,6OI0,6OFZ,6E23,6E22,6E1Z,6E1Y,6DAS,6DAR,6DAK,6DAI,6D9X,4Y7R,4GMB,4GM9,4GM8,4GM3,3P4F,2H14,2H13,8Q1N,5SXM,4CY2,4CY1,4EWR,4ESG,4ES0,4ERZ,4ERY,4ERQ,3EG6,2H6Q,2H6N,2H6K,2H68,7DNO,6U8B,6U80,6U6W,5VFC,3EMH,7BCY,2G99,6IAM,8E9F,7U9Y,6DYA,2G9A,8HMX,6UOZ,6UJ4,6UIK,6UIF,6UHZ,6UHY,6U8O,6U8L,6U5Y,6U5M,6DY7,7JTP,7JTO,6BYN,3MXX,3N0E,6PGF,6PGE,6PGD,6PGC,6PGB,6PGA,6PG7,6PG5,6PG4,3N0D,8BB5,8BB4,8BB3,8BB2	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51570309	CCn1cc(c(n1)C(F)(F)F)-c1cc(Cn2ccnc2C)cc2c1OCCN([C@H]1CCOc3ccc(OC)cc13)C2=O	InChI=1S/C30H30F3N5O4/c1-4-37-17-24(28(35-37)30(31,32)33)21-13-19(16-36-9-8-34-18(36)2)14-23-27(21)42-12-10-38(29(23)39)25-7-11-41-26-6-5-20(40-3)15-22(25)26/h5-6,8-9,13-15,17,25H,4,7,10-12,16H2,1-3H3/t25-/m0/s1	FDCJPULEHRJDGT-VWLOTQADSA-N	50631546	CHEMBL5411289	WD repeat-containing protein 5	Homo sapiens	<0.020000								ChEMBL	10.1021/acs.jmedchem.3c01529	10.7270/Q2KH0SSW	38085679			n/a	n/a	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50631546	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50631546&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search											1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	8X3R,7CFQ,7CFP,7BED,7AXX,7AXU,7AXS,7AXQ,7AXP,6KIZ,6KIX,6KIW,6KIV,6KIU,2XL3,2XL2,2GNQ,8DU4,7UD5,8X3S,3UVO,3UVN,3UVM,3UVL,3UVK,3PSL,8OKF,4A7J,8G3E,8F93,8F1G,8G3C,7WVK,7UAS,7MBN,7MBM,6WJQ,6W5N,6W5M,6W5I,6UJL,6UJJ,6UJH,6UCS,6PWW,6PWV,6PG9,6PG8,6PG6,6PG3,6OI3,6OI2,6OI1,6OI0,6OFZ,6E23,6E22,6E1Z,6E1Y,6DAS,6DAR,6DAK,6DAI,6D9X,4Y7R,4GMB,4GM9,4GM8,4GM3,3P4F,2H14,2H13,8Q1N,5SXM,4CY2,4CY1,4EWR,4ESG,4ES0,4ERZ,4ERY,4ERQ,3EG6,2H6Q,2H6N,2H6K,2H68,7DNO,6U8B,6U80,6U6W,5VFC,3EMH,7BCY,2G99,6IAM,8E9F,7U9Y,6DYA,2G9A,8HMX,6UOZ,6UJ4,6UIK,6UIF,6UHZ,6UHY,6U8O,6U8L,6U5Y,6U5M,6DY7,7JTP,7JTO,6BYN,3MXX,3N0E,6PGF,6PGE,6PGD,6PGC,6PGB,6PGA,6PG7,6PG5,6PG4,3N0D,8BB5,8BB4,8BB3,8BB2	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51570310	CCn1cc(c(n1)C(F)(F)F)-c1cc(Cn2ccnc2)cc2c1OCCN([C@H]1CCOc3ccc(OC)cc13)C2=O	InChI=1S/C29H28F3N5O4/c1-3-36-16-23(27(34-36)29(30,31)32)20-12-18(15-35-8-7-33-17-35)13-22-26(20)41-11-9-37(28(22)38)24-6-10-40-25-5-4-19(39-2)14-21(24)25/h4-5,7-8,12-14,16-17,24H,3,6,9-11,15H2,1-2H3/t24-/m0/s1	GOVJZVCNGLOGNS-DEOSSOPVSA-N	50631547	CHEMBL5418460	WD repeat-containing protein 5	Homo sapiens	<0.020000								ChEMBL	10.1021/acs.jmedchem.3c01529	10.7270/Q2KH0SSW	38085679			n/a	n/a	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50631547	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50631547&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search											1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	8X3R,7CFQ,7CFP,7BED,7AXX,7AXU,7AXS,7AXQ,7AXP,6KIZ,6KIX,6KIW,6KIV,6KIU,2XL3,2XL2,2GNQ,8DU4,7UD5,8X3S,3UVO,3UVN,3UVM,3UVL,3UVK,3PSL,8OKF,4A7J,8G3E,8F93,8F1G,8G3C,7WVK,7UAS,7MBN,7MBM,6WJQ,6W5N,6W5M,6W5I,6UJL,6UJJ,6UJH,6UCS,6PWW,6PWV,6PG9,6PG8,6PG6,6PG3,6OI3,6OI2,6OI1,6OI0,6OFZ,6E23,6E22,6E1Z,6E1Y,6DAS,6DAR,6DAK,6DAI,6D9X,4Y7R,4GMB,4GM9,4GM8,4GM3,3P4F,2H14,2H13,8Q1N,5SXM,4CY2,4CY1,4EWR,4ESG,4ES0,4ERZ,4ERY,4ERQ,3EG6,2H6Q,2H6N,2H6K,2H68,7DNO,6U8B,6U80,6U6W,5VFC,3EMH,7BCY,2G99,6IAM,8E9F,7U9Y,6DYA,2G9A,8HMX,6UOZ,6UJ4,6UIK,6UIF,6UHZ,6UHY,6U8O,6U8L,6U5Y,6U5M,6DY7,7JTP,7JTO,6BYN,3MXX,3N0E,6PGF,6PGE,6PGD,6PGC,6PGB,6PGA,6PG7,6PG5,6PG4,3N0D,8BB5,8BB4,8BB3,8BB2	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51570311	COc1cnc2CCC[C@H](N3CCOc4c(cc(Cn5ccnc5)cc4C3=O)-c3cn(C)nc3C(F)(F)F)c2c1	InChI=1S/C28H27F3N6O3/c1-35-15-22(26(34-35)28(29,30)31)19-10-17(14-36-7-6-32-16-36)11-21-25(19)40-9-8-37(27(21)38)24-5-3-4-23-20(24)12-18(39-2)13-33-23/h6-7,10-13,15-16,24H,3-5,8-9,14H2,1-2H3/t24-/m0/s1	OTVQRTLMBVTANG-DEOSSOPVSA-N	50631548	CHEMBL5418271	WD repeat-containing protein 5	Homo sapiens	<0.020000								ChEMBL	10.1021/acs.jmedchem.3c01529	10.7270/Q2KH0SSW	38085679			n/a	n/a	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50631548	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50631548&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search											1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	8X3R,7CFQ,7CFP,7BED,7AXX,7AXU,7AXS,7AXQ,7AXP,6KIZ,6KIX,6KIW,6KIV,6KIU,2XL3,2XL2,2GNQ,8DU4,7UD5,8X3S,3UVO,3UVN,3UVM,3UVL,3UVK,3PSL,8OKF,4A7J,8G3E,8F93,8F1G,8G3C,7WVK,7UAS,7MBN,7MBM,6WJQ,6W5N,6W5M,6W5I,6UJL,6UJJ,6UJH,6UCS,6PWW,6PWV,6PG9,6PG8,6PG6,6PG3,6OI3,6OI2,6OI1,6OI0,6OFZ,6E23,6E22,6E1Z,6E1Y,6DAS,6DAR,6DAK,6DAI,6D9X,4Y7R,4GMB,4GM9,4GM8,4GM3,3P4F,2H14,2H13,8Q1N,5SXM,4CY2,4CY1,4EWR,4ESG,4ES0,4ERZ,4ERY,4ERQ,3EG6,2H6Q,2H6N,2H6K,2H68,7DNO,6U8B,6U80,6U6W,5VFC,3EMH,7BCY,2G99,6IAM,8E9F,7U9Y,6DYA,2G9A,8HMX,6UOZ,6UJ4,6UIK,6UIF,6UHZ,6UHY,6U8O,6U8L,6U5Y,6U5M,6DY7,7JTP,7JTO,6BYN,3MXX,3N0E,6PGF,6PGE,6PGD,6PGC,6PGB,6PGA,6PG7,6PG5,6PG4,3N0D,8BB5,8BB4,8BB3,8BB2	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51570312	CCc1cnc2CCC[C@H](N3CCOc4c(cc(Cn5ccnc5)cc4C3=O)-c3cn(C)nc3C(F)(F)F)c2c1	InChI=1S/C29H29F3N6O2/c1-3-18-11-21-24(34-14-18)5-4-6-25(21)38-9-10-40-26-20(23-16-36(2)35-27(23)29(30,31)32)12-19(13-22(26)28(38)39)15-37-8-7-33-17-37/h7-8,11-14,16-17,25H,3-6,9-10,15H2,1-2H3/t25-/m0/s1	UNJHUGGXCYVFOK-VWLOTQADSA-N	50631549	CHEMBL5432148	WD repeat-containing protein 5	Homo sapiens	<0.020000								ChEMBL	10.1021/acs.jmedchem.3c01529	10.7270/Q2KH0SSW	38085679			n/a	n/a	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50631549	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50631549&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search											1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	8X3R,7CFQ,7CFP,7BED,7AXX,7AXU,7AXS,7AXQ,7AXP,6KIZ,6KIX,6KIW,6KIV,6KIU,2XL3,2XL2,2GNQ,8DU4,7UD5,8X3S,3UVO,3UVN,3UVM,3UVL,3UVK,3PSL,8OKF,4A7J,8G3E,8F93,8F1G,8G3C,7WVK,7UAS,7MBN,7MBM,6WJQ,6W5N,6W5M,6W5I,6UJL,6UJJ,6UJH,6UCS,6PWW,6PWV,6PG9,6PG8,6PG6,6PG3,6OI3,6OI2,6OI1,6OI0,6OFZ,6E23,6E22,6E1Z,6E1Y,6DAS,6DAR,6DAK,6DAI,6D9X,4Y7R,4GMB,4GM9,4GM8,4GM3,3P4F,2H14,2H13,8Q1N,5SXM,4CY2,4CY1,4EWR,4ESG,4ES0,4ERZ,4ERY,4ERQ,3EG6,2H6Q,2H6N,2H6K,2H68,7DNO,6U8B,6U80,6U6W,5VFC,3EMH,7BCY,2G99,6IAM,8E9F,7U9Y,6DYA,2G9A,8HMX,6UOZ,6UJ4,6UIK,6UIF,6UHZ,6UHY,6U8O,6U8L,6U5Y,6U5M,6DY7,7JTP,7JTO,6BYN,3MXX,3N0E,6PGF,6PGE,6PGD,6PGC,6PGB,6PGA,6PG7,6PG5,6PG4,3N0D,8BB5,8BB4,8BB3,8BB2	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51570313	CCc1cc(C(=O)NC)c2nccc(N3CCc4c(cc(Cn5ccnc5)cc4C3=O)-c3cn(C)nc3C(F)(F)F)c2c1	InChI=1S/C31H28F3N7O2/c1-4-18-11-23-26(5-7-37-27(23)24(12-18)29(42)35-2)41-9-6-20-21(25-16-39(3)38-28(25)31(32,33)34)13-19(14-22(20)30(41)43)15-40-10-8-36-17-40/h5,7-8,10-14,16-17H,4,6,9,15H2,1-3H3,(H,35,42)	SHGMSJNVTCKQHS-UHFFFAOYSA-N	50631550	CHEMBL5421916	WD repeat-containing protein 5	Homo sapiens	<0.020000								ChEMBL	10.1021/acs.jmedchem.3c01529	10.7270/Q2KH0SSW	38085679			n/a	n/a	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50631550	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50631550&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	UY9    	8E9F									1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	8X3R,7CFQ,7CFP,7BED,7AXX,7AXU,7AXS,7AXQ,7AXP,6KIZ,6KIX,6KIW,6KIV,6KIU,2XL3,2XL2,2GNQ,8DU4,7UD5,8X3S,3UVO,3UVN,3UVM,3UVL,3UVK,3PSL,8OKF,4A7J,8G3E,8F93,8F1G,8G3C,7WVK,7UAS,7MBN,7MBM,6WJQ,6W5N,6W5M,6W5I,6UJL,6UJJ,6UJH,6UCS,6PWW,6PWV,6PG9,6PG8,6PG6,6PG3,6OI3,6OI2,6OI1,6OI0,6OFZ,6E23,6E22,6E1Z,6E1Y,6DAS,6DAR,6DAK,6DAI,6D9X,4Y7R,4GMB,4GM9,4GM8,4GM3,3P4F,2H14,2H13,8Q1N,5SXM,4CY2,4CY1,4EWR,4ESG,4ES0,4ERZ,4ERY,4ERQ,3EG6,2H6Q,2H6N,2H6K,2H68,7DNO,6U8B,6U80,6U6W,5VFC,3EMH,7BCY,2G99,6IAM,8E9F,7U9Y,6DYA,2G9A,8HMX,6UOZ,6UJ4,6UIK,6UIF,6UHZ,6UHY,6U8O,6U8L,6U5Y,6U5M,6DY7,7JTP,7JTO,6BYN,3MXX,3N0E,6PGF,6PGE,6PGD,6PGC,6PGB,6PGA,6PG7,6PG5,6PG4,3N0D,8BB5,8BB4,8BB3,8BB2	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51570929	CC(C)C[C@H](NC(=O)[C@H](Cc1cnc[nH]1)NC(=O)[C@@H](NC(=O)[C@H](CCC(O)=O)NC(=O)[C@@H](NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@H](C)NC(C)=O)[C@@H](C)O)C(C)C)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CO)C(=O)NCCCCCC(=O)NCCCCCC(=O)N[C@@H](CCCCNC(=O)c1ccc(c(c1)C(O)=O)-c1c2ccc(O)cc2oc2cc(=O)ccc12)C(N)=O	InChI=1S/C91H136N24O24/c1-48(2)40-66(111-86(134)67(42-54-45-98-47-104-54)112-87(135)75(49(3)4)114-84(132)65(32-33-73(123)124)110-88(136)76(51(6)117)115-83(131)64(23-19-39-103-91(96)97)107-78(126)50(5)105-52(7)118)85(133)109-63(22-18-38-102-90(94)95)81(129)108-62(21-12-14-34-92)82(130)113-68(46-116)80(128)101-36-16-8-10-24-71(121)99-35-15-9-11-25-72(122)106-61(77(93)125)20-13-17-37-100-79(127)53-26-29-57(60(41-53)89(137)138)74-58-30-27-55(119)43-69(58)139-70-44-56(120)28-31-59(70)74/h26-31,41,43-45,47-51,61-68,75-76,116-117,119H,8-25,32-40,42,46,92H2,1-7H3,(H2,93,125)(H,98,104)(H,99,121)(H,100,127)(H,101,128)(H,105,118)(H,106,122)(H,107,126)(H,108,129)(H,109,133)(H,110,136)(H,111,134)(H,112,135)(H,113,130)(H,114,132)(H,115,131)(H,123,124)(H,137,138)(H4,94,95,102)(H4,96,97,103)/t50-,51+,61-,62-,63-,64-,65-,66-,67-,68-,75-,76-/m0/s1	LVHMEOMYGFPCIV-CLNRVIFCSA-N	50631811	CHEMBL5417280	WD repeat-containing protein 5	Homo sapiens			 0.840000						ChEMBL	10.1039/d3md00605k	10.7270/Q2833XH5	38389889			n/a	n/a	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50631811	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50631811&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search											1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	8X3R,7CFQ,7CFP,7BED,7AXX,7AXU,7AXS,7AXQ,7AXP,6KIZ,6KIX,6KIW,6KIV,6KIU,2XL3,2XL2,2GNQ,8DU4,7UD5,8X3S,3UVO,3UVN,3UVM,3UVL,3UVK,3PSL,8OKF,4A7J,8G3E,8F93,8F1G,8G3C,7WVK,7UAS,7MBN,7MBM,6WJQ,6W5N,6W5M,6W5I,6UJL,6UJJ,6UJH,6UCS,6PWW,6PWV,6PG9,6PG8,6PG6,6PG3,6OI3,6OI2,6OI1,6OI0,6OFZ,6E23,6E22,6E1Z,6E1Y,6DAS,6DAR,6DAK,6DAI,6D9X,4Y7R,4GMB,4GM9,4GM8,4GM3,3P4F,2H14,2H13,8Q1N,5SXM,4CY2,4CY1,4EWR,4ESG,4ES0,4ERZ,4ERY,4ERQ,3EG6,2H6Q,2H6N,2H6K,2H68,7DNO,6U8B,6U80,6U6W,5VFC,3EMH,7BCY,2G99,6IAM,8E9F,7U9Y,6DYA,2G9A,8HMX,6UOZ,6UJ4,6UIK,6UIF,6UHZ,6UHY,6U8O,6U8L,6U5Y,6U5M,6DY7,7JTP,7JTO,6BYN,3MXX,3N0E,6PGF,6PGE,6PGD,6PGC,6PGB,6PGA,6PG7,6PG5,6PG4,3N0D,8BB5,8BB4,8BB3,8BB2	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51554764	Cc1cc(=O)c(nn1-c1ccccc1)C(=O)NCc1c(F)cc(cc1F)-c1cccc(c1)S(F)(=O)=O	InChI=1S/C25H18F3N3O4S/c1-15-10-23(32)24(30-31(15)18-7-3-2-4-8-18)25(33)29-14-20-21(26)12-17(13-22(20)27)16-6-5-9-19(11-16)36(28,34)35/h2-13H,14H2,1H3,(H,29,33)	KCMSIHHWMOTDFN-UHFFFAOYSA-N	50625549	CHEMBL5410251	WD repeat-containing protein 5	Homo sapiens		 2090							ChEMBL	10.1021/acs.jmedchem.3c00787	10.7270/Q26D5ZDG	37307526			n/a	n/a	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50625549	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50625549&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search											1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	8X3R,7CFQ,7CFP,7BED,7AXX,7AXU,7AXS,7AXQ,7AXP,6KIZ,6KIX,6KIW,6KIV,6KIU,2XL3,2XL2,2GNQ,8DU4,7UD5,8X3S,3UVO,3UVN,3UVM,3UVL,3UVK,3PSL,8OKF,4A7J,8G3E,8F93,8F1G,8G3C,7WVK,7UAS,7MBN,7MBM,6WJQ,6W5N,6W5M,6W5I,6UJL,6UJJ,6UJH,6UCS,6PWW,6PWV,6PG9,6PG8,6PG6,6PG3,6OI3,6OI2,6OI1,6OI0,6OFZ,6E23,6E22,6E1Z,6E1Y,6DAS,6DAR,6DAK,6DAI,6D9X,4Y7R,4GMB,4GM9,4GM8,4GM3,3P4F,2H14,2H13,8Q1N,5SXM,4CY2,4CY1,4EWR,4ESG,4ES0,4ERZ,4ERY,4ERQ,3EG6,2H6Q,2H6N,2H6K,2H68,7DNO,6U8B,6U80,6U6W,5VFC,3EMH,7BCY,2G99,6IAM,8E9F,7U9Y,6DYA,2G9A,8HMX,6UOZ,6UJ4,6UIK,6UIF,6UHZ,6UHY,6U8O,6U8L,6U5Y,6U5M,6DY7,7JTP,7JTO,6BYN,3MXX,3N0E,6PGF,6PGE,6PGD,6PGC,6PGB,6PGA,6PG7,6PG5,6PG4,3N0D,8BB5,8BB4,8BB3,8BB2	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51554765	Cc1cc(=O)c(nn1-c1ccccc1)C(=O)NCc1c(F)cc(cc1F)-c1cccc(c1)S(F)(=O)=O	InChI=1S/C25H18F3N3O4S/c1-15-10-23(32)24(30-31(15)18-7-3-2-4-8-18)25(33)29-14-20-21(26)12-17(13-22(20)27)16-6-5-9-19(11-16)36(28,34)35/h2-13H,14H2,1H3,(H,29,33)	KCMSIHHWMOTDFN-UHFFFAOYSA-N	50625549	CHEMBL5410251	WD repeat-containing protein 5	Homo sapiens		 790							ChEMBL	10.1021/acs.jmedchem.3c00787	10.7270/Q26D5ZDG	37307526			n/a	n/a	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50625549	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50625549&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search											1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	8X3R,7CFQ,7CFP,7BED,7AXX,7AXU,7AXS,7AXQ,7AXP,6KIZ,6KIX,6KIW,6KIV,6KIU,2XL3,2XL2,2GNQ,8DU4,7UD5,8X3S,3UVO,3UVN,3UVM,3UVL,3UVK,3PSL,8OKF,4A7J,8G3E,8F93,8F1G,8G3C,7WVK,7UAS,7MBN,7MBM,6WJQ,6W5N,6W5M,6W5I,6UJL,6UJJ,6UJH,6UCS,6PWW,6PWV,6PG9,6PG8,6PG6,6PG3,6OI3,6OI2,6OI1,6OI0,6OFZ,6E23,6E22,6E1Z,6E1Y,6DAS,6DAR,6DAK,6DAI,6D9X,4Y7R,4GMB,4GM9,4GM8,4GM3,3P4F,2H14,2H13,8Q1N,5SXM,4CY2,4CY1,4EWR,4ESG,4ES0,4ERZ,4ERY,4ERQ,3EG6,2H6Q,2H6N,2H6K,2H68,7DNO,6U8B,6U80,6U6W,5VFC,3EMH,7BCY,2G99,6IAM,8E9F,7U9Y,6DYA,2G9A,8HMX,6UOZ,6UJ4,6UIK,6UIF,6UHZ,6UHY,6U8O,6U8L,6U5Y,6U5M,6DY7,7JTP,7JTO,6BYN,3MXX,3N0E,6PGF,6PGE,6PGD,6PGC,6PGB,6PGA,6PG7,6PG5,6PG4,3N0D,8BB5,8BB4,8BB3,8BB2	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51554766	Cc1cc(=O)c(nn1-c1ccccc1)C(=O)NCc1c(F)cc(cc1F)-c1cccc(c1)S(F)(=O)=O	InChI=1S/C25H18F3N3O4S/c1-15-10-23(32)24(30-31(15)18-7-3-2-4-8-18)25(33)29-14-20-21(26)12-17(13-22(20)27)16-6-5-9-19(11-16)36(28,34)35/h2-13H,14H2,1H3,(H,29,33)	KCMSIHHWMOTDFN-UHFFFAOYSA-N	50625549	CHEMBL5410251	WD repeat-containing protein 5	Homo sapiens		 300							ChEMBL	10.1021/acs.jmedchem.3c00787	10.7270/Q26D5ZDG	37307526			n/a	n/a	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50625549	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50625549&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search											1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	8X3R,7CFQ,7CFP,7BED,7AXX,7AXU,7AXS,7AXQ,7AXP,6KIZ,6KIX,6KIW,6KIV,6KIU,2XL3,2XL2,2GNQ,8DU4,7UD5,8X3S,3UVO,3UVN,3UVM,3UVL,3UVK,3PSL,8OKF,4A7J,8G3E,8F93,8F1G,8G3C,7WVK,7UAS,7MBN,7MBM,6WJQ,6W5N,6W5M,6W5I,6UJL,6UJJ,6UJH,6UCS,6PWW,6PWV,6PG9,6PG8,6PG6,6PG3,6OI3,6OI2,6OI1,6OI0,6OFZ,6E23,6E22,6E1Z,6E1Y,6DAS,6DAR,6DAK,6DAI,6D9X,4Y7R,4GMB,4GM9,4GM8,4GM3,3P4F,2H14,2H13,8Q1N,5SXM,4CY2,4CY1,4EWR,4ESG,4ES0,4ERZ,4ERY,4ERQ,3EG6,2H6Q,2H6N,2H6K,2H68,7DNO,6U8B,6U80,6U6W,5VFC,3EMH,7BCY,2G99,6IAM,8E9F,7U9Y,6DYA,2G9A,8HMX,6UOZ,6UJ4,6UIK,6UIF,6UHZ,6UHY,6U8O,6U8L,6U5Y,6U5M,6DY7,7JTP,7JTO,6BYN,3MXX,3N0E,6PGF,6PGE,6PGD,6PGC,6PGB,6PGA,6PG7,6PG5,6PG4,3N0D,8BB5,8BB4,8BB3,8BB2	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51554767	Cc1cc(=O)c(nn1-c1ccccc1)C(=O)NCc1c(F)cc(cc1F)-c1cccc(c1)S(F)(=O)=O	InChI=1S/C25H18F3N3O4S/c1-15-10-23(32)24(30-31(15)18-7-3-2-4-8-18)25(33)29-14-20-21(26)12-17(13-22(20)27)16-6-5-9-19(11-16)36(28,34)35/h2-13H,14H2,1H3,(H,29,33)	KCMSIHHWMOTDFN-UHFFFAOYSA-N	50625549	CHEMBL5410251	WD repeat-containing protein 5	Homo sapiens		 170							ChEMBL	10.1021/acs.jmedchem.3c00787	10.7270/Q26D5ZDG	37307526			n/a	n/a	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50625549	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50625549&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search											1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	8X3R,7CFQ,7CFP,7BED,7AXX,7AXU,7AXS,7AXQ,7AXP,6KIZ,6KIX,6KIW,6KIV,6KIU,2XL3,2XL2,2GNQ,8DU4,7UD5,8X3S,3UVO,3UVN,3UVM,3UVL,3UVK,3PSL,8OKF,4A7J,8G3E,8F93,8F1G,8G3C,7WVK,7UAS,7MBN,7MBM,6WJQ,6W5N,6W5M,6W5I,6UJL,6UJJ,6UJH,6UCS,6PWW,6PWV,6PG9,6PG8,6PG6,6PG3,6OI3,6OI2,6OI1,6OI0,6OFZ,6E23,6E22,6E1Z,6E1Y,6DAS,6DAR,6DAK,6DAI,6D9X,4Y7R,4GMB,4GM9,4GM8,4GM3,3P4F,2H14,2H13,8Q1N,5SXM,4CY2,4CY1,4EWR,4ESG,4ES0,4ERZ,4ERY,4ERQ,3EG6,2H6Q,2H6N,2H6K,2H68,7DNO,6U8B,6U80,6U6W,5VFC,3EMH,7BCY,2G99,6IAM,8E9F,7U9Y,6DYA,2G9A,8HMX,6UOZ,6UJ4,6UIK,6UIF,6UHZ,6UHY,6U8O,6U8L,6U5Y,6U5M,6DY7,7JTP,7JTO,6BYN,3MXX,3N0E,6PGF,6PGE,6PGD,6PGC,6PGB,6PGA,6PG7,6PG5,6PG4,3N0D,8BB5,8BB4,8BB3,8BB2	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51554768	Cc1cc(=O)c(nn1-c1ccccc1)C(=O)NCc1c(F)cc(cc1F)-c1cccc(c1)S(F)(=O)=O	InChI=1S/C25H18F3N3O4S/c1-15-10-23(32)24(30-31(15)18-7-3-2-4-8-18)25(33)29-14-20-21(26)12-17(13-22(20)27)16-6-5-9-19(11-16)36(28,34)35/h2-13H,14H2,1H3,(H,29,33)	KCMSIHHWMOTDFN-UHFFFAOYSA-N	50625549	CHEMBL5410251	WD repeat-containing protein 5	Homo sapiens		 100							ChEMBL	10.1021/acs.jmedchem.3c00787	10.7270/Q26D5ZDG	37307526			n/a	n/a	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50625549	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50625549&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search											1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	8X3R,7CFQ,7CFP,7BED,7AXX,7AXU,7AXS,7AXQ,7AXP,6KIZ,6KIX,6KIW,6KIV,6KIU,2XL3,2XL2,2GNQ,8DU4,7UD5,8X3S,3UVO,3UVN,3UVM,3UVL,3UVK,3PSL,8OKF,4A7J,8G3E,8F93,8F1G,8G3C,7WVK,7UAS,7MBN,7MBM,6WJQ,6W5N,6W5M,6W5I,6UJL,6UJJ,6UJH,6UCS,6PWW,6PWV,6PG9,6PG8,6PG6,6PG3,6OI3,6OI2,6OI1,6OI0,6OFZ,6E23,6E22,6E1Z,6E1Y,6DAS,6DAR,6DAK,6DAI,6D9X,4Y7R,4GMB,4GM9,4GM8,4GM3,3P4F,2H14,2H13,8Q1N,5SXM,4CY2,4CY1,4EWR,4ESG,4ES0,4ERZ,4ERY,4ERQ,3EG6,2H6Q,2H6N,2H6K,2H68,7DNO,6U8B,6U80,6U6W,5VFC,3EMH,7BCY,2G99,6IAM,8E9F,7U9Y,6DYA,2G9A,8HMX,6UOZ,6UJ4,6UIK,6UIF,6UHZ,6UHY,6U8O,6U8L,6U5Y,6U5M,6DY7,7JTP,7JTO,6BYN,3MXX,3N0E,6PGF,6PGE,6PGD,6PGC,6PGB,6PGA,6PG7,6PG5,6PG4,3N0D,8BB5,8BB4,8BB3,8BB2	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51540010	CC(C)C[C@H](NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)[C@H](CC(N)=O)NC(=O)[C@@H](NC(=O)[C@H](CC(O)=O)NC(=O)[C@H](C)NC(=O)[C@@H](N)CS)[C@@H](C)O)C(=O)N[C@@H](C(C)C)C(=O)N[C@@H](CS)C(O)=O	InChI=1S/C43H65N11O14S2/c1-18(2)11-26(39(63)53-33(19(3)4)41(65)52-30(17-70)43(67)68)49-37(61)27(12-22-15-46-25-10-8-7-9-23(22)25)50-38(62)28(13-31(45)56)51-42(66)34(21(6)55)54-40(64)29(14-32(57)58)48-35(59)20(5)47-36(60)24(44)16-69/h7-10,15,18-21,24,26-30,33-34,46,55,69-70H,11-14,16-17,44H2,1-6H3,(H2,45,56)(H,47,60)(H,48,59)(H,49,61)(H,50,62)(H,51,66)(H,52,65)(H,53,63)(H,54,64)(H,57,58)(H,67,68)/t20-,21+,24-,26-,27-,28-,29-,30-,33-,34-/m0/s1	XMQGQQKVXNXJGV-QBYIZTRCSA-N	50619319	CHEMBL5437580	WD repeat-containing protein 5	Homo sapiens		 65000							ChEMBL	10.1039/d3md00288h	10.7270/Q20Z77NB	37859722			n/a	n/a	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50619319	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50619319&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search											1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	8X3R,7CFQ,7CFP,7BED,7AXX,7AXU,7AXS,7AXQ,7AXP,6KIZ,6KIX,6KIW,6KIV,6KIU,2XL3,2XL2,2GNQ,8DU4,7UD5,8X3S,3UVO,3UVN,3UVM,3UVL,3UVK,3PSL,8OKF,4A7J,8G3E,8F93,8F1G,8G3C,7WVK,7UAS,7MBN,7MBM,6WJQ,6W5N,6W5M,6W5I,6UJL,6UJJ,6UJH,6UCS,6PWW,6PWV,6PG9,6PG8,6PG6,6PG3,6OI3,6OI2,6OI1,6OI0,6OFZ,6E23,6E22,6E1Z,6E1Y,6DAS,6DAR,6DAK,6DAI,6D9X,4Y7R,4GMB,4GM9,4GM8,4GM3,3P4F,2H14,2H13,8Q1N,5SXM,4CY2,4CY1,4EWR,4ESG,4ES0,4ERZ,4ERY,4ERQ,3EG6,2H6Q,2H6N,2H6K,2H68,7DNO,6U8B,6U80,6U6W,5VFC,3EMH,7BCY,2G99,6IAM,8E9F,7U9Y,6DYA,2G9A,8HMX,6UOZ,6UJ4,6UIK,6UIF,6UHZ,6UHY,6U8O,6U8L,6U5Y,6U5M,6DY7,7JTP,7JTO,6BYN,3MXX,3N0E,6PGF,6PGE,6PGD,6PGC,6PGB,6PGA,6PG7,6PG5,6PG4,3N0D,8BB5,8BB4,8BB3,8BB2	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51540011	NCCCC[C@H](NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](CC(N)=O)NC(=O)[C@@H]1CCCN1C(=O)[C@H](N)CS)C(=O)N[C@@H](CO)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CS)C(O)=O	InChI=1S/C49H69N13O14S2/c50-16-4-3-8-31(41(67)60-36(22-63)46(72)57-33(18-25-10-12-27(64)13-11-25)43(69)61-37(24-78)49(75)76)55-44(70)34(19-26-21-54-30-7-2-1-6-28(26)30)58-42(68)32(14-15-39(52)65)56-45(71)35(20-40(53)66)59-47(73)38-9-5-17-62(38)48(74)29(51)23-77/h1-2,6-7,10-13,21,29,31-38,54,63-64,77-78H,3-5,8-9,14-20,22-24,50-51H2,(H2,52,65)(H2,53,66)(H,55,70)(H,56,71)(H,57,72)(H,58,68)(H,59,73)(H,60,67)(H,61,69)(H,75,76)/t29-,31+,32+,33+,34+,35+,36+,37+,38+/m1/s1	FPTXXNDEEQKCCT-UHGYHLOUSA-N	50619320	CHEMBL5396034	WD repeat-containing protein 5	Homo sapiens		>100000							ChEMBL	10.1039/d3md00288h	10.7270/Q20Z77NB	37859722			n/a	n/a	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50619320	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50619320&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search											1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	8X3R,7CFQ,7CFP,7BED,7AXX,7AXU,7AXS,7AXQ,7AXP,6KIZ,6KIX,6KIW,6KIV,6KIU,2XL3,2XL2,2GNQ,8DU4,7UD5,8X3S,3UVO,3UVN,3UVM,3UVL,3UVK,3PSL,8OKF,4A7J,8G3E,8F93,8F1G,8G3C,7WVK,7UAS,7MBN,7MBM,6WJQ,6W5N,6W5M,6W5I,6UJL,6UJJ,6UJH,6UCS,6PWW,6PWV,6PG9,6PG8,6PG6,6PG3,6OI3,6OI2,6OI1,6OI0,6OFZ,6E23,6E22,6E1Z,6E1Y,6DAS,6DAR,6DAK,6DAI,6D9X,4Y7R,4GMB,4GM9,4GM8,4GM3,3P4F,2H14,2H13,8Q1N,5SXM,4CY2,4CY1,4EWR,4ESG,4ES0,4ERZ,4ERY,4ERQ,3EG6,2H6Q,2H6N,2H6K,2H68,7DNO,6U8B,6U80,6U6W,5VFC,3EMH,7BCY,2G99,6IAM,8E9F,7U9Y,6DYA,2G9A,8HMX,6UOZ,6UJ4,6UIK,6UIF,6UHZ,6UHY,6U8O,6U8L,6U5Y,6U5M,6DY7,7JTP,7JTO,6BYN,3MXX,3N0E,6PGF,6PGE,6PGD,6PGC,6PGB,6PGA,6PG7,6PG5,6PG4,3N0D,8BB5,8BB4,8BB3,8BB2	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51540012	C[C@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](CO)NC(=O)[C@@H](N)CS)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CS)C(O)=O	InChI=1S/C53H67N13O14S2/c1-26(59-47(73)36(14-16-43(55)69)61-52(78)41(23-67)65-46(72)33(54)24-81)45(71)62-39(19-28-21-57-34-8-4-2-6-31(28)34)50(76)64-40(20-29-22-58-35-9-5-3-7-32(29)35)51(77)63-38(18-27-10-12-30(68)13-11-27)49(75)60-37(15-17-44(56)70)48(74)66-42(25-82)53(79)80/h2-13,21-22,26,33,36-42,57-58,67-68,81-82H,14-20,23-25,54H2,1H3,(H2,55,69)(H2,56,70)(H,59,73)(H,60,75)(H,61,78)(H,62,71)(H,63,77)(H,64,76)(H,65,72)(H,66,74)(H,79,80)/t26-,33-,36-,37-,38-,39-,40-,41-,42-/m0/s1	KKQCPHPNRCSZHS-DXTHKOOBSA-N	50619321	CHEMBL5397601	WD repeat-containing protein 5	Homo sapiens		 30000							ChEMBL	10.1039/d3md00288h	10.7270/Q20Z77NB	37859722			n/a	n/a	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50619321	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50619321&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search											1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	8X3R,7CFQ,7CFP,7BED,7AXX,7AXU,7AXS,7AXQ,7AXP,6KIZ,6KIX,6KIW,6KIV,6KIU,2XL3,2XL2,2GNQ,8DU4,7UD5,8X3S,3UVO,3UVN,3UVM,3UVL,3UVK,3PSL,8OKF,4A7J,8G3E,8F93,8F1G,8G3C,7WVK,7UAS,7MBN,7MBM,6WJQ,6W5N,6W5M,6W5I,6UJL,6UJJ,6UJH,6UCS,6PWW,6PWV,6PG9,6PG8,6PG6,6PG3,6OI3,6OI2,6OI1,6OI0,6OFZ,6E23,6E22,6E1Z,6E1Y,6DAS,6DAR,6DAK,6DAI,6D9X,4Y7R,4GMB,4GM9,4GM8,4GM3,3P4F,2H14,2H13,8Q1N,5SXM,4CY2,4CY1,4EWR,4ESG,4ES0,4ERZ,4ERY,4ERQ,3EG6,2H6Q,2H6N,2H6K,2H68,7DNO,6U8B,6U80,6U6W,5VFC,3EMH,7BCY,2G99,6IAM,8E9F,7U9Y,6DYA,2G9A,8HMX,6UOZ,6UJ4,6UIK,6UIF,6UHZ,6UHY,6U8O,6U8L,6U5Y,6U5M,6DY7,7JTP,7JTO,6BYN,3MXX,3N0E,6PGF,6PGE,6PGD,6PGC,6PGB,6PGA,6PG7,6PG5,6PG4,3N0D,8BB5,8BB4,8BB3,8BB2	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51540013	CC(C)C[C@H](NC(=O)[C@H](Cc1ccccc1)NC(=O)[C@@H](N)CS)C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](C(C)C)C(=O)N[C@@H](CO)C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](C)C(=O)N[C@@H](CS)C(O)=O	InChI=1S/C40H63N11O13S2/c1-18(2)11-23(46-36(59)24(45-33(56)22(41)16-65)12-21-9-7-6-8-10-21)35(58)47-26(14-30(43)54)37(60)51-31(19(3)4)39(62)49-27(15-52)38(61)48-25(13-29(42)53)34(57)44-20(5)32(55)50-28(17-66)40(63)64/h6-10,18-20,22-28,31,52,65-66H,11-17,41H2,1-5H3,(H2,42,53)(H2,43,54)(H,44,57)(H,45,56)(H,46,59)(H,47,58)(H,48,61)(H,49,62)(H,50,55)(H,51,60)(H,63,64)/t20-,22-,23-,24-,25-,26-,27-,28-,31-/m0/s1	VQMJAXSLFJIPAT-MURBELKFSA-N	50619322	CHEMBL5441098	WD repeat-containing protein 5	Homo sapiens		>100000							ChEMBL	10.1039/d3md00288h	10.7270/Q20Z77NB	37859722			n/a	n/a	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50619322	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50619322&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search											1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	8X3R,7CFQ,7CFP,7BED,7AXX,7AXU,7AXS,7AXQ,7AXP,6KIZ,6KIX,6KIW,6KIV,6KIU,2XL3,2XL2,2GNQ,8DU4,7UD5,8X3S,3UVO,3UVN,3UVM,3UVL,3UVK,3PSL,8OKF,4A7J,8G3E,8F93,8F1G,8G3C,7WVK,7UAS,7MBN,7MBM,6WJQ,6W5N,6W5M,6W5I,6UJL,6UJJ,6UJH,6UCS,6PWW,6PWV,6PG9,6PG8,6PG6,6PG3,6OI3,6OI2,6OI1,6OI0,6OFZ,6E23,6E22,6E1Z,6E1Y,6DAS,6DAR,6DAK,6DAI,6D9X,4Y7R,4GMB,4GM9,4GM8,4GM3,3P4F,2H14,2H13,8Q1N,5SXM,4CY2,4CY1,4EWR,4ESG,4ES0,4ERZ,4ERY,4ERQ,3EG6,2H6Q,2H6N,2H6K,2H68,7DNO,6U8B,6U80,6U6W,5VFC,3EMH,7BCY,2G99,6IAM,8E9F,7U9Y,6DYA,2G9A,8HMX,6UOZ,6UJ4,6UIK,6UIF,6UHZ,6UHY,6U8O,6U8L,6U5Y,6U5M,6DY7,7JTP,7JTO,6BYN,3MXX,3N0E,6PGF,6PGE,6PGD,6PGC,6PGB,6PGA,6PG7,6PG5,6PG4,3N0D,8BB5,8BB4,8BB3,8BB2	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51540014	CC(C)C[C@H](NC(=O)[C@H](CO)NC(=O)CNC(=O)[C@@H](N)CS)C(=O)N[C@@H](CC(O)=O)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N1CCC[C@H]1C(=O)N[C@@H](Cc1c[nH]cn1)C(=O)N[C@@H](CS)C(O)=O	InChI=1S/C43H60N12O13S2/c1-21(2)10-27(50-40(64)31(17-56)49-34(57)16-47-36(60)25(44)18-69)37(61)51-29(13-35(58)59)39(63)53-30(11-22-14-46-26-7-4-3-6-24(22)26)42(66)55-9-5-8-33(55)41(65)52-28(12-23-15-45-20-48-23)38(62)54-32(19-70)43(67)68/h3-4,6-7,14-15,20-21,25,27-33,46,56,69-70H,5,8-13,16-19,44H2,1-2H3,(H,45,48)(H,47,60)(H,49,57)(H,50,64)(H,51,61)(H,52,65)(H,53,63)(H,54,62)(H,58,59)(H,67,68)/t25-,27-,28-,29-,30-,31-,32-,33-/m0/s1	XSVYHGUITLPVEA-XSTSSERXSA-N	50619323	CHEMBL5421163	WD repeat-containing protein 5	Homo sapiens		 25000							ChEMBL	10.1039/d3md00288h	10.7270/Q20Z77NB	37859722			n/a	n/a	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50619323	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50619323&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search											1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	8X3R,7CFQ,7CFP,7BED,7AXX,7AXU,7AXS,7AXQ,7AXP,6KIZ,6KIX,6KIW,6KIV,6KIU,2XL3,2XL2,2GNQ,8DU4,7UD5,8X3S,3UVO,3UVN,3UVM,3UVL,3UVK,3PSL,8OKF,4A7J,8G3E,8F93,8F1G,8G3C,7WVK,7UAS,7MBN,7MBM,6WJQ,6W5N,6W5M,6W5I,6UJL,6UJJ,6UJH,6UCS,6PWW,6PWV,6PG9,6PG8,6PG6,6PG3,6OI3,6OI2,6OI1,6OI0,6OFZ,6E23,6E22,6E1Z,6E1Y,6DAS,6DAR,6DAK,6DAI,6D9X,4Y7R,4GMB,4GM9,4GM8,4GM3,3P4F,2H14,2H13,8Q1N,5SXM,4CY2,4CY1,4EWR,4ESG,4ES0,4ERZ,4ERY,4ERQ,3EG6,2H6Q,2H6N,2H6K,2H68,7DNO,6U8B,6U80,6U6W,5VFC,3EMH,7BCY,2G99,6IAM,8E9F,7U9Y,6DYA,2G9A,8HMX,6UOZ,6UJ4,6UIK,6UIF,6UHZ,6UHY,6U8O,6U8L,6U5Y,6U5M,6DY7,7JTP,7JTO,6BYN,3MXX,3N0E,6PGF,6PGE,6PGD,6PGC,6PGB,6PGA,6PG7,6PG5,6PG4,3N0D,8BB5,8BB4,8BB3,8BB2	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51540015	CC(C)C[C@H](NC(=O)[C@H](CO)NC(=O)[C@H](CC(N)=O)NC(=O)[C@@H](N)CS)C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CS)C(O)=O	InChI=1S/C54H69N13O13S2/c1-27(2)16-36(61-53(78)42(24-68)66-52(77)40(20-44(56)69)60-46(71)33(55)25-81)47(72)65-41(21-45(57)70)51(76)64-38(18-29-22-58-34-14-8-6-12-31(29)34)49(74)62-37(17-28-10-4-3-5-11-28)48(73)63-39(50(75)67-43(26-82)54(79)80)19-30-23-59-35-15-9-7-13-32(30)35/h3-15,22-23,27,33,36-43,58-59,68,81-82H,16-21,24-26,55H2,1-2H3,(H2,56,69)(H2,57,70)(H,60,71)(H,61,78)(H,62,74)(H,63,73)(H,64,76)(H,65,72)(H,66,77)(H,67,75)(H,79,80)/t33-,36-,37-,38-,39-,40-,41-,42-,43-/m0/s1	ZKOYDBJZZCCWCY-WXGDXGANSA-N	50619324	CHEMBL5428912	WD repeat-containing protein 5	Homo sapiens		 2200							ChEMBL	10.1039/d3md00288h	10.7270/Q20Z77NB	37859722			n/a	n/a	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50619324	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50619324&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search											1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	8X3R,7CFQ,7CFP,7BED,7AXX,7AXU,7AXS,7AXQ,7AXP,6KIZ,6KIX,6KIW,6KIV,6KIU,2XL3,2XL2,2GNQ,8DU4,7UD5,8X3S,3UVO,3UVN,3UVM,3UVL,3UVK,3PSL,8OKF,4A7J,8G3E,8F93,8F1G,8G3C,7WVK,7UAS,7MBN,7MBM,6WJQ,6W5N,6W5M,6W5I,6UJL,6UJJ,6UJH,6UCS,6PWW,6PWV,6PG9,6PG8,6PG6,6PG3,6OI3,6OI2,6OI1,6OI0,6OFZ,6E23,6E22,6E1Z,6E1Y,6DAS,6DAR,6DAK,6DAI,6D9X,4Y7R,4GMB,4GM9,4GM8,4GM3,3P4F,2H14,2H13,8Q1N,5SXM,4CY2,4CY1,4EWR,4ESG,4ES0,4ERZ,4ERY,4ERQ,3EG6,2H6Q,2H6N,2H6K,2H68,7DNO,6U8B,6U80,6U6W,5VFC,3EMH,7BCY,2G99,6IAM,8E9F,7U9Y,6DYA,2G9A,8HMX,6UOZ,6UJ4,6UIK,6UIF,6UHZ,6UHY,6U8O,6U8L,6U5Y,6U5M,6DY7,7JTP,7JTO,6BYN,3MXX,3N0E,6PGF,6PGE,6PGD,6PGC,6PGB,6PGA,6PG7,6PG5,6PG4,3N0D,8BB5,8BB4,8BB3,8BB2	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51540016	CC(C)[C@H](NC(=O)[C@H](CC(O)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCC(O)=O)NC(=O)CNC(=O)[C@H](CCC(O)=O)NC(=O)CNC(=O)[C@@H](N)CS)C(=O)N[C@@H](CS)C(O)=O	InChI=1S/C32H51N9O16S2/c1-13(2)25(31(55)40-19(12-59)32(56)57)41-30(54)18(8-24(48)49)39-26(50)14(3)36-29(53)17(5-7-23(46)47)38-21(43)10-35-28(52)16(4-6-22(44)45)37-20(42)9-34-27(51)15(33)11-58/h13-19,25,58-59H,4-12,33H2,1-3H3,(H,34,51)(H,35,52)(H,36,53)(H,37,42)(H,38,43)(H,39,50)(H,40,55)(H,41,54)(H,44,45)(H,46,47)(H,48,49)(H,56,57)/t14-,15-,16-,17-,18-,19-,25-/m0/s1	PFQHBUJIAIYXPD-WDVQKFPESA-N	50619325	CHEMBL5394572	WD repeat-containing protein 5	Homo sapiens		>100000							ChEMBL	10.1039/d3md00288h	10.7270/Q20Z77NB	37859722			n/a	n/a	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50619325	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50619325&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search											1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	8X3R,7CFQ,7CFP,7BED,7AXX,7AXU,7AXS,7AXQ,7AXP,6KIZ,6KIX,6KIW,6KIV,6KIU,2XL3,2XL2,2GNQ,8DU4,7UD5,8X3S,3UVO,3UVN,3UVM,3UVL,3UVK,3PSL,8OKF,4A7J,8G3E,8F93,8F1G,8G3C,7WVK,7UAS,7MBN,7MBM,6WJQ,6W5N,6W5M,6W5I,6UJL,6UJJ,6UJH,6UCS,6PWW,6PWV,6PG9,6PG8,6PG6,6PG3,6OI3,6OI2,6OI1,6OI0,6OFZ,6E23,6E22,6E1Z,6E1Y,6DAS,6DAR,6DAK,6DAI,6D9X,4Y7R,4GMB,4GM9,4GM8,4GM3,3P4F,2H14,2H13,8Q1N,5SXM,4CY2,4CY1,4EWR,4ESG,4ES0,4ERZ,4ERY,4ERQ,3EG6,2H6Q,2H6N,2H6K,2H68,7DNO,6U8B,6U80,6U6W,5VFC,3EMH,7BCY,2G99,6IAM,8E9F,7U9Y,6DYA,2G9A,8HMX,6UOZ,6UJ4,6UIK,6UIF,6UHZ,6UHY,6U8O,6U8L,6U5Y,6U5M,6DY7,7JTP,7JTO,6BYN,3MXX,3N0E,6PGF,6PGE,6PGD,6PGC,6PGB,6PGA,6PG7,6PG5,6PG4,3N0D,8BB5,8BB4,8BB3,8BB2	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51540017	CC(C)C[C@@H]1NC(=O)[C@H](CO)NC(=O)[C@H](CC(N)=O)NC(=O)[C@@H](N)CSCc2ccc(CSC[C@H](NC(=O)[C@H](Cc3c[nH]c4ccccc34)NC(=O)[C@H](Cc3ccccc3)NC(=O)[C@H](Cc3c[nH]c4ccccc34)NC(=O)[C@H](CC(N)=O)NC1=O)C(O)=O)cc2	InChI=1S/C62H75N13O13S2/c1-33(2)20-44-55(80)73-49(25-53(65)78)59(84)72-46(22-37-26-66-42-14-8-6-12-39(37)42)57(82)70-45(21-34-10-4-3-5-11-34)56(81)71-47(23-38-27-67-43-15-9-7-13-40(38)43)58(83)75-51(62(87)88)32-90-30-36-18-16-35(17-19-36)29-89-31-41(63)54(79)68-48(24-52(64)77)60(85)74-50(28-76)61(86)69-44/h3-19,26-27,33,41,44-51,66-67,76H,20-25,28-32,63H2,1-2H3,(H2,64,77)(H2,65,78)(H,68,79)(H,69,86)(H,70,82)(H,71,81)(H,72,84)(H,73,80)(H,74,85)(H,75,83)(H,87,88)/t41-,44-,45-,46-,47-,48-,49-,50-,51-/m0/s1	VULIIDBOQCEVCZ-ACPIDWHBSA-N	50619326	CHEMBL5428456	WD repeat-containing protein 5	Homo sapiens		 8100							ChEMBL	10.1039/d3md00288h	10.7270/Q20Z77NB	37859722			n/a	n/a	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50619326	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50619326&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search											1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	8X3R,7CFQ,7CFP,7BED,7AXX,7AXU,7AXS,7AXQ,7AXP,6KIZ,6KIX,6KIW,6KIV,6KIU,2XL3,2XL2,2GNQ,8DU4,7UD5,8X3S,3UVO,3UVN,3UVM,3UVL,3UVK,3PSL,8OKF,4A7J,8G3E,8F93,8F1G,8G3C,7WVK,7UAS,7MBN,7MBM,6WJQ,6W5N,6W5M,6W5I,6UJL,6UJJ,6UJH,6UCS,6PWW,6PWV,6PG9,6PG8,6PG6,6PG3,6OI3,6OI2,6OI1,6OI0,6OFZ,6E23,6E22,6E1Z,6E1Y,6DAS,6DAR,6DAK,6DAI,6D9X,4Y7R,4GMB,4GM9,4GM8,4GM3,3P4F,2H14,2H13,8Q1N,5SXM,4CY2,4CY1,4EWR,4ESG,4ES0,4ERZ,4ERY,4ERQ,3EG6,2H6Q,2H6N,2H6K,2H68,7DNO,6U8B,6U80,6U6W,5VFC,3EMH,7BCY,2G99,6IAM,8E9F,7U9Y,6DYA,2G9A,8HMX,6UOZ,6UJ4,6UIK,6UIF,6UHZ,6UHY,6U8O,6U8L,6U5Y,6U5M,6DY7,7JTP,7JTO,6BYN,3MXX,3N0E,6PGF,6PGE,6PGD,6PGC,6PGB,6PGA,6PG7,6PG5,6PG4,3N0D,8BB5,8BB4,8BB3,8BB2	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51540018	CC(C)C[C@@H]1NC(=O)[C@H](CO)NC(=O)[C@H](CC(N)=O)NC(=O)[C@@H](N)CSC\C=C/CSC[C@H](NC(=O)[C@H](Cc2c[nH]c3ccccc23)NC(=O)[C@H](Cc2ccccc2)NC(=O)[C@H](Cc2c[nH]c3ccccc23)NC(=O)[C@H](CC(N)=O)NC1=O)C(O)=O	InChI=1S/C58H73N13O13S2/c1-31(2)20-40-51(76)69-45(25-49(61)74)55(80)68-42(22-33-26-62-38-16-8-6-14-35(33)38)53(78)66-41(21-32-12-4-3-5-13-32)52(77)67-43(23-34-27-63-39-17-9-7-15-36(34)39)54(79)71-47(58(83)84)30-86-19-11-10-18-85-29-37(59)50(75)64-44(24-48(60)73)56(81)70-46(28-72)57(82)65-40/h3-17,26-27,31,37,40-47,62-63,72H,18-25,28-30,59H2,1-2H3,(H2,60,73)(H2,61,74)(H,64,75)(H,65,82)(H,66,78)(H,67,77)(H,68,80)(H,69,76)(H,70,81)(H,71,79)(H,83,84)/b11-10-/t37-,40-,41-,42-,43-,44-,45-,46-,47-/m0/s1	IEZRFWNDHMFKDL-DVLONYMRSA-N	50619327	CHEMBL5440089	WD repeat-containing protein 5	Homo sapiens		 10900							ChEMBL	10.1039/d3md00288h	10.7270/Q20Z77NB	37859722			n/a	n/a	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50619327	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50619327&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search											1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	8X3R,7CFQ,7CFP,7BED,7AXX,7AXU,7AXS,7AXQ,7AXP,6KIZ,6KIX,6KIW,6KIV,6KIU,2XL3,2XL2,2GNQ,8DU4,7UD5,8X3S,3UVO,3UVN,3UVM,3UVL,3UVK,3PSL,8OKF,4A7J,8G3E,8F93,8F1G,8G3C,7WVK,7UAS,7MBN,7MBM,6WJQ,6W5N,6W5M,6W5I,6UJL,6UJJ,6UJH,6UCS,6PWW,6PWV,6PG9,6PG8,6PG6,6PG3,6OI3,6OI2,6OI1,6OI0,6OFZ,6E23,6E22,6E1Z,6E1Y,6DAS,6DAR,6DAK,6DAI,6D9X,4Y7R,4GMB,4GM9,4GM8,4GM3,3P4F,2H14,2H13,8Q1N,5SXM,4CY2,4CY1,4EWR,4ESG,4ES0,4ERZ,4ERY,4ERQ,3EG6,2H6Q,2H6N,2H6K,2H68,7DNO,6U8B,6U80,6U6W,5VFC,3EMH,7BCY,2G99,6IAM,8E9F,7U9Y,6DYA,2G9A,8HMX,6UOZ,6UJ4,6UIK,6UIF,6UHZ,6UHY,6U8O,6U8L,6U5Y,6U5M,6DY7,7JTP,7JTO,6BYN,3MXX,3N0E,6PGF,6PGE,6PGD,6PGC,6PGB,6PGA,6PG7,6PG5,6PG4,3N0D,8BB5,8BB4,8BB3,8BB2	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51540019	CC(C)C[C@@H]1NC(=O)[C@H](CO)NC(=O)[C@H](CC(N)=O)NC(=O)[C@@H](N)CSCc2cccc(CSC[C@H](NC(=O)[C@H](Cc3c[nH]c4ccccc34)NC(=O)[C@H](Cc3ccccc3)NC(=O)[C@H](Cc3c[nH]c4ccccc34)NC(=O)[C@H](CC(N)=O)NC1=O)C(O)=O)n2	InChI=1S/C61H74N14O13S2/c1-32(2)19-43-54(80)73-48(24-52(64)78)58(84)72-45(21-34-25-65-41-17-8-6-15-38(34)41)56(82)70-44(20-33-11-4-3-5-12-33)55(81)71-46(22-35-26-66-42-18-9-7-16-39(35)42)57(83)75-50(61(87)88)31-90-29-37-14-10-13-36(67-37)28-89-30-40(62)53(79)68-47(23-51(63)77)59(85)74-49(27-76)60(86)69-43/h3-18,25-26,32,40,43-50,65-66,76H,19-24,27-31,62H2,1-2H3,(H2,63,77)(H2,64,78)(H,68,79)(H,69,86)(H,70,82)(H,71,81)(H,72,84)(H,73,80)(H,74,85)(H,75,83)(H,87,88)/t40-,43-,44-,45-,46-,47-,48-,49-,50-/m0/s1	AEMVGSPCLOHJOG-GBPBLIGGSA-N	50619328	CHEMBL5432299	WD repeat-containing protein 5	Homo sapiens		 8700							ChEMBL	10.1039/d3md00288h	10.7270/Q20Z77NB	37859722			n/a	n/a	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50619328	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50619328&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search											1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	8X3R,7CFQ,7CFP,7BED,7AXX,7AXU,7AXS,7AXQ,7AXP,6KIZ,6KIX,6KIW,6KIV,6KIU,2XL3,2XL2,2GNQ,8DU4,7UD5,8X3S,3UVO,3UVN,3UVM,3UVL,3UVK,3PSL,8OKF,4A7J,8G3E,8F93,8F1G,8G3C,7WVK,7UAS,7MBN,7MBM,6WJQ,6W5N,6W5M,6W5I,6UJL,6UJJ,6UJH,6UCS,6PWW,6PWV,6PG9,6PG8,6PG6,6PG3,6OI3,6OI2,6OI1,6OI0,6OFZ,6E23,6E22,6E1Z,6E1Y,6DAS,6DAR,6DAK,6DAI,6D9X,4Y7R,4GMB,4GM9,4GM8,4GM3,3P4F,2H14,2H13,8Q1N,5SXM,4CY2,4CY1,4EWR,4ESG,4ES0,4ERZ,4ERY,4ERQ,3EG6,2H6Q,2H6N,2H6K,2H68,7DNO,6U8B,6U80,6U6W,5VFC,3EMH,7BCY,2G99,6IAM,8E9F,7U9Y,6DYA,2G9A,8HMX,6UOZ,6UJ4,6UIK,6UIF,6UHZ,6UHY,6U8O,6U8L,6U5Y,6U5M,6DY7,7JTP,7JTO,6BYN,3MXX,3N0E,6PGF,6PGE,6PGD,6PGC,6PGB,6PGA,6PG7,6PG5,6PG4,3N0D,8BB5,8BB4,8BB3,8BB2	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51540020	CC[C@H](C)[C@H](NC(=O)[C@H](CCC(O)=O)NC(=O)[C@H](CCC(O)=O)NC(=O)[C@H](CCC(O)=O)NC(=O)[C@@H](N)CO)C(=O)N[C@@H](CC(O)=O)C(=O)N[C@@H](C(C)C)C(=O)N[C@@H](C(C)C)C(=O)N[C@@H](CO)C(=O)N[C@@H](C(C)C)C(O)=O	InChI=1S/C46H76N10O21/c1-9-22(8)36(56-40(70)26(12-15-31(63)64)50-39(69)25(11-14-30(61)62)49-38(68)24(10-13-29(59)60)48-37(67)23(47)17-57)45(75)51-27(16-32(65)66)41(71)53-34(20(4)5)44(74)54-33(19(2)3)43(73)52-28(18-58)42(72)55-35(21(6)7)46(76)77/h19-28,33-36,57-58H,9-18,47H2,1-8H3,(H,48,67)(H,49,68)(H,50,69)(H,51,75)(H,52,73)(H,53,71)(H,54,74)(H,55,72)(H,56,70)(H,59,60)(H,61,62)(H,63,64)(H,65,66)(H,76,77)/t22-,23-,24-,25-,26-,27-,28-,33-,34-,35-,36-/m0/s1	BQHGWSAVMQWHGI-RDAIJIBISA-N	50619329	CHEMBL5407534	WD repeat-containing protein 5	Homo sapiens		 1600							ChEMBL	10.1039/d3md00288h	10.7270/Q20Z77NB	37859722			n/a	n/a	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50619329	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50619329&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search											1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	8X3R,7CFQ,7CFP,7BED,7AXX,7AXU,7AXS,7AXQ,7AXP,6KIZ,6KIX,6KIW,6KIV,6KIU,2XL3,2XL2,2GNQ,8DU4,7UD5,8X3S,3UVO,3UVN,3UVM,3UVL,3UVK,3PSL,8OKF,4A7J,8G3E,8F93,8F1G,8G3C,7WVK,7UAS,7MBN,7MBM,6WJQ,6W5N,6W5M,6W5I,6UJL,6UJJ,6UJH,6UCS,6PWW,6PWV,6PG9,6PG8,6PG6,6PG3,6OI3,6OI2,6OI1,6OI0,6OFZ,6E23,6E22,6E1Z,6E1Y,6DAS,6DAR,6DAK,6DAI,6D9X,4Y7R,4GMB,4GM9,4GM8,4GM3,3P4F,2H14,2H13,8Q1N,5SXM,4CY2,4CY1,4EWR,4ESG,4ES0,4ERZ,4ERY,4ERQ,3EG6,2H6Q,2H6N,2H6K,2H68,7DNO,6U8B,6U80,6U6W,5VFC,3EMH,7BCY,2G99,6IAM,8E9F,7U9Y,6DYA,2G9A,8HMX,6UOZ,6UJ4,6UIK,6UIF,6UHZ,6UHY,6U8O,6U8L,6U5Y,6U5M,6DY7,7JTP,7JTO,6BYN,3MXX,3N0E,6PGF,6PGE,6PGD,6PGC,6PGB,6PGA,6PG7,6PG5,6PG4,3N0D,8BB5,8BB4,8BB3,8BB2	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
51540021	CC[C@H](C)[C@H](NC(=O)[C@H](CCC(O)=O)NC(=O)[C@H](CCC(O)=O)NC(=O)[C@H](CCC(O)=O)NC(=O)[C@@H](N)CO)C(=O)N[C@@H](CC(O)=O)C(=O)N[C@@H](C(C)C)C(=O)N[C@@H](C(C)C)C(=O)N[C@@H](CO)C(=O)N[C@@H](C(C)C)C(O)=O	InChI=1S/C46H76N10O21/c1-9-22(8)36(56-40(70)26(12-15-31(63)64)50-39(69)25(11-14-30(61)62)49-38(68)24(10-13-29(59)60)48-37(67)23(47)17-57)45(75)51-27(16-32(65)66)41(71)53-34(20(4)5)44(74)54-33(19(2)3)43(73)52-28(18-58)42(72)55-35(21(6)7)46(76)77/h19-28,33-36,57-58H,9-18,47H2,1-8H3,(H,48,67)(H,49,68)(H,50,69)(H,51,75)(H,52,73)(H,53,71)(H,54,74)(H,55,72)(H,56,70)(H,59,60)(H,61,62)(H,63,64)(H,65,66)(H,76,77)/t22-,23-,24-,25-,26-,27-,28-,33-,34-,35-,36-/m0/s1	BQHGWSAVMQWHGI-RDAIJIBISA-N	50619329	CHEMBL5407534	WD repeat-containing protein 5	Homo sapiens			 9300						ChEMBL	10.1039/d3md00288h	10.7270/Q20Z77NB	37859722			n/a	n/a	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50619329	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=8469&target=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50619329&enzyme=WD+repeat-containing+protein+5&column=ki&startPg=0&Increment=50&submit=Search											1	MATEEKKPETEAARAQPTPSSSATQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC	8X3R,7CFQ,7CFP,7BED,7AXX,7AXU,7AXS,7AXQ,7AXP,6KIZ,6KIX,6KIW,6KIV,6KIU,2XL3,2XL2,2GNQ,8DU4,7UD5,8X3S,3UVO,3UVN,3UVM,3UVL,3UVK,3PSL,8OKF,4A7J,8G3E,8F93,8F1G,8G3C,7WVK,7UAS,7MBN,7MBM,6WJQ,6W5N,6W5M,6W5I,6UJL,6UJJ,6UJH,6UCS,6PWW,6PWV,6PG9,6PG8,6PG6,6PG3,6OI3,6OI2,6OI1,6OI0,6OFZ,6E23,6E22,6E1Z,6E1Y,6DAS,6DAR,6DAK,6DAI,6D9X,4Y7R,4GMB,4GM9,4GM8,4GM3,3P4F,2H14,2H13,8Q1N,5SXM,4CY2,4CY1,4EWR,4ESG,4ES0,4ERZ,4ERY,4ERQ,3EG6,2H6Q,2H6N,2H6K,2H68,7DNO,6U8B,6U80,6U6W,5VFC,3EMH,7BCY,2G99,6IAM,8E9F,7U9Y,6DYA,2G9A,8HMX,6UOZ,6UJ4,6UIK,6UIF,6UHZ,6UHY,6U8O,6U8L,6U5Y,6U5M,6DY7,7JTP,7JTO,6BYN,3MXX,3N0E,6PGF,6PGE,6PGD,6PGC,6PGB,6PGA,6PG7,6PG5,6PG4,3N0D,8BB5,8BB4,8BB3,8BB2	WD repeat-containing protein 5	WDR5_HUMAN	P61964	Q91VA5 Q9NWX7 Q9UGP9						
