BindingDB Reactant_set_id	Ligand SMILES	Ligand InChI	Ligand InChI Key	BindingDB MonomerID	BindingDB Ligand Name	Target Name	Target Source Organism According to Curator or DataSource	Ki (nM)	IC50 (nM)	Kd (nM)	EC50 (nM)	kon (M-1-s-1)	koff (s-1)	pH	Temp (C)	Curation/DataSource	Article DOI	BindingDB Entry DOI	PMID	PubChem AID	Patent Number	Authors	Institution	Link to Ligand in BindingDB	Link to Target in BindingDB	Link to Ligand-Target Pair in BindingDB	Ligand HET ID in PDB	PDB ID(s) for Ligand-Target Complex	PubChem CID of Ligand	PubChem SID of Ligand	ChEBI ID of Ligand	ChEMBL ID of Ligand	DrugBank ID of Ligand	IUPHAR_GRAC ID of Ligand	KEGG ID of Ligand	ZINC ID of Ligand	Number of Protein Chains in Target (>1 implies a multichain complex)	BindingDB Target Chain Sequence	PDB ID(s) of Target Chain	UniProt (SwissProt) Recommended Name of Target Chain	UniProt (SwissProt) Entry Name of Target Chain	UniProt (SwissProt) Primary ID of Target Chain	UniProt (SwissProt) Secondary ID(s) of Target Chain	UniProt (SwissProt) Alternative ID(s) of Target Chain	UniProt (TrEMBL) Submitted Name of Target Chain	UniProt (TrEMBL) Entry Name of Target Chain	UniProt (TrEMBL) Primary ID of Target Chain	UniProt (TrEMBL) Secondary ID(s) of Target Chain	UniProt (TrEMBL) Alternative ID(s) of Target Chain
1210908	Nc1nc2n(cnc2c(=O)[nH]1)[C@@H]1O[C@@H]2COP(O)(=O)O[C@H]3C[C@@H](O[C@@H]3COP(O)(=O)O[C@@H]1[C@@H]2O)n1cnc2c(N)ncnc12	InChI=1S/C20H24N10O12P2/c21-15-11-16(24-4-23-15)29(5-25-11)10-1-7-8(39-10)2-37-44(35,36)42-14-13(31)9(3-38-43(33,34)41-7)40-19(14)30-6-26-12-17(30)27-20(22)28-18(12)32/h4-10,13-14,19,31H,1-3H2,(H,33,34)(H,35,36)(H2,21,23,24)(H3,22,27,28,32)/t7-,8+,9+,10+,13+,14+,19+/m0/s1	RFDHWTXDKIGDJD-BEAYCLROSA-N	50509412	CHEMBL4474321::US11453697, Example 1	Stimulator of interferon genes protein [H232R]					 3.50					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50509412	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50509412&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			137102579	440717997							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1210909	Nc1nc2n(cnc2c(=O)[nH]1)[C@@H]1O[C@@H]2COP(O)(=O)OC3[C@@H](COP(O)(=O)O[C@H]1C2O)O[C@H]([C@H]3F)n1cnc2c(N)ncnc12			573838	(5R,7R,8R,12aR,14R,15R,15aR,16R)-7-(2- amino-6-oxo-1,6-dihydro-9H-purin-9-yl)-14-(6- amino-9H-purin-9-yl)-15-fluoro-16- hydroxyoctahydro-12H-5,8-methanofuro[3,2-l] [1,3,6,9,11,2,10]pentaoxadiphosphacyclotetradecine- 2,10-diolate 2,10-dioxide::US11453697, Example 2::US11453697, Example 7	Stimulator of interferon genes protein [H232R]					 0.700					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=573838	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=573838&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177454	474496201							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1210910	Nc1nc2n(cnc2c(=O)[nH]1)[C@@H]1O[C@@H]2COP(O)(=O)OC3C[C@@H](O[C@@H]3COP(O)(=O)O[C@H]1C2O)n1cnc2c(N)ncnc12			573839	(5R,7R,8R,12aR,14R,15aS,16R)-7,14-bis(6- amino-9H-purin-9-yl)-16-hydroxyoctahydro- 12H-5,8-methanofuro[3,2-l] [1,3,6,9,11,2,10]pentaoxadiphosphacyclotetradecine- 2,10-diolate 2,10-dioxide::US11453697, Example 3	Stimulator of interferon genes protein [H232R]					 574					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=573839	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=573839&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177455	474496202							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1210911	Nc1ncnc2n(cnc12)[C@@H]1O[C@@H]2COP(O)(=O)O[C@H]3C(O)[C@@H](COP(O)(=O)OC2[C@@H]1F)O[C@H]3n1cnc2c(N)ncnc12	InChI=1S/C20H23FN10O11P2/c21-9-13-8(40-19(9)30-5-28-10-15(22)24-3-26-17(10)30)2-38-44(35,36)42-14-12(32)7(1-37-43(33,34)41-13)39-20(14)31-6-29-11-16(23)25-4-27-18(11)31/h3-9,12-14,19-20,32H,1-2H2,(H,33,34)(H,35,36)(H2,22,24,26)(H2,23,25,27)/t7-,8-,9+,12?,13?,14+,19-,20-/m1/s1	AKJJTMOTMKBURB-QMCVZGSNSA-N	573840	(5R,7R,8R,12aR,14R,15R,15aR,16R)-7,14-bis(6- amino-9H-purin-9-yl)-15-fluoro-16- hydroxyoctahydro-12H-5,8-methanofuro[3,2-l] [1,3,6,9,11,2,10]pentaoxadiphosphacyclotetradecine- 2,10-diolate 2,10-dioxide::US11453697, Example 4	Stimulator of interferon genes protein [H232R]					 43.5					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=573840	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=573840&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			140899397	474496203							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1210912	Nc1nc2n(cnc2c(=O)[nH]1)[C@@H]1O[C@@H]2COP(O)(=O)OC3[C@@H](COP(O)(=O)O[C@H]1C2F)O[C@H]([C@H]3O)n1cnc2c(N)ncnc12			573841	(5R,7R,8S,12aR,14R,15R,15aS,16R)-7-(2- amino-6-oxo-1,6-dihydro-9H-purin-9-yl)-14-(6- amino-9H-purin-9-yl)-16-fluoro-15- hydroxyoctahydro-12H-5,8-methanofuro[3,2-l] [1,3,6,9,11,2,10]pentaoxadiphosphacyclotetradecine- 2,10-diolate 2,10-dioxide::US11453697, Example 5	Stimulator of interferon genes protein [H232R]					 1.50					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=573841	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=573841&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177456	474496204							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1210913	Nc1nc2n(cnc2c(=O)[nH]1)[C@@H]1O[C@@H]2COP(O)(=O)OC3[C@@H]4OC[C@]3(COP(O)(=O)O[C@H]1C2O)O[C@H]4n1cnc2c(N)ncnc12			573842	(5R,7R,8R,12aR,14R,15R,15aS,18R)-7-(2-amino- 6-oxo-1,6-dihydro-9H-purin-9-yl)-14-(6-amino- 9H-purin-9-yl)-18-hydroxyhexahydro-14H- 15,12a-(epoxymethano)-5,8-methanofuro[3,2-l] [1,3,6,9,11,2,10]pentaoxadiphosphacyclotetradecine- 2,10(12H)-diolate 2,10-dioxide::US11453697, Example 6	Stimulator of interferon genes protein [H232R]					 2.90					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=573842	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=573842&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177457	474496205							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1210914	Nc1nc2n(cnc2c(=O)[nH]1)[C@@H]1O[C@@H]2COP(O)(=O)OC3[C@@H](COP(O)(=O)O[C@H]1C2O)O[C@H]([C@H]3F)n1cnc2c(N)ncnc12			573838	(5R,7R,8R,12aR,14R,15R,15aR,16R)-7-(2- amino-6-oxo-1,6-dihydro-9H-purin-9-yl)-14-(6- amino-9H-purin-9-yl)-15-fluoro-16- hydroxyoctahydro-12H-5,8-methanofuro[3,2-l] [1,3,6,9,11,2,10]pentaoxadiphosphacyclotetradecine- 2,10-diolate 2,10-dioxide::US11453697, Example 2::US11453697, Example 7	Stimulator of interferon genes protein [H232R]					<1.000					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=573838	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=573838&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177454	474496201							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1210915	Nc1nc2n(cnc2c(=O)[nH]1)[C@@H]1O[C@@H]2COP(O)(=O)OC3C[C@@H](O[C@@H]3COP(O)(=O)O[C@H]1C2O)n1cnc2c1nc[nH]c2=O			573844	(5R,7R,8R,12aR,14R,15aS,16R)-7-(2-amino-6- oxo-1,6-dihydro-9H-purin-9-yl)-16-hydroxy-14- (6-oxo-1,6-dihydro-9H-purin-9-yl)octahydro- 12H-5,8-methanofuro[3,2-l][1,3,6,9,11,2,10] pentaoxadiphosphacyclotetradecine-2,10-diolate 2,10-dioxide::US11453697, Example 8	Stimulator of interferon genes protein [H232R]					 81.4					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=573844	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=573844&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177458	474496206							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1210916	Nc1nc2n(cnc2c(=O)[nH]1)[C@@H]1O[C@@H]2COP(O)(=O)OC3[C@@H](COP(O)(=O)O[C@H]1C2O)O[C@H]([C@H]3O)n1ccc2c(N)ncnc12			573845	(5R,7R,8R,12aR,14R,15R,15aS,16R)-7-(2-amino- 6-oxo-1,6-dihydro-9H-purin-9-yl)-14-(4-amino- 7H-pyrrolo[2,3-d]pyrimidin-7-yl)-15,16- dihydroxyoctahydro-12H-5,8-methanofuro[3,2-l] [1,3,6,9,11,2,10]pentaoxadiphosphacyclotetradecine- 2,10-diolate 2,10-dioxide::US11453697, Example 9	Stimulator of interferon genes protein [H232R]					 12.4					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=573845	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=573845&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177459	474496207							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1210917	Nc1nc2n(cnc2c(=O)[nH]1)[C@@H]1O[C@@H]2COP(O)(=O)OC3C[C@@H](O[C@@H]3COP(O)(=O)O[C@H]1C2O)n1ccc2c(N)ncnc12			573846	(5R,7R,8R,12aR,14R,15aS,16R)-7-(2-amino-6- oxo-1,6-dihydro-9H-purin-9-yl)-14-(4-amino- 7H-pyrrolo[2,3-d]pyrimidin-7-yl)-16- hydroxyoctahydro-12H-5,8-methanofuro[3,2-l] [1,3,6,9,11,2,10] pentaoxadiphosphacyclotetradecine- 2,10-diolate 2,10-dioxide::US11453697, Example 10	Stimulator of interferon genes protein [H232R]					 23.2					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=573846	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=573846&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177460	474496208							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1210918	CO[C@@H]1[C@H]2COP(O)(=O)O[C@@H]3[C@@H](COP(O)(=O)O[C@H]1[C@@H](O2)n1cnc2c1nc(N)[nH]c2=O)O[C@H]([C@@H]3O)n1cnc2c(N)ncnc12			573849	2-amino-9- [(5R,7R,8R,12aR,14R,15R,15aS,16R)-14-(6- amino-9H-purin-9-yl)-2,10,15-trihydroxy-16- methoxy-2,10-dioxidooctahydro-12H-5,8- methanofuro[3,2-l][1,3,6,9,11,2,10] pentaoxadiphosphacyclotetradecin-7-yl]-1,9- dihydro-6H-purin-6-one::US11453697, Example 13	Stimulator of interferon genes protein [H232R]					 0.700					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=573849	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=573849&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177463	474496211							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1210919	Nc1nc2n(cnc2c(=O)[nH]1)[C@@H]1O[C@@H]2COP(O)(=O)O[C@@H]3[C@@H](COP(O)(=O)O[C@@H]1[C@@H]2N=[N+]=[N-])O[C@H]([C@@H]3O)n1cnc2c(N)ncnc12			573850	2-amino-9- [(5S,7R,8R,12aR,14R,15R,15aS,16R)-14-(6- amino-9H-purin-9-yl)-16-azido-2,10,15- trihydroxy-2,10-dioxidooctahydro-12H-5,8- methanofuro[3,2-l][1,3,6,9,11,2,10] pentaoxadiphosphacyclotetradecin-7-yl]-1,9- dihydro-6H-purin-6-one::US11453697, Example 14	Stimulator of interferon genes protein [H232R]					 1.40					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=573850	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=573850&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177464	474496212							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1210920	Nc1nc2n(cnc2c(=O)[nH]1)[C@@H]1O[C@@H]2COP(O)(=O)O[C@H]3[C@H]4OC[C@]3(COP(O)(=O)O[C@@H]1[C@@H]2F)O[C@H]4n1cnc2c(N)ncnc12			573856	US11453697, Example 20	Stimulator of interferon genes protein [H232R]					 1.40					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=573856	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=573856&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177470	474496218							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1210921	NC1NC(N)=Nc2c1ncn2[C@@H]1O[C@H]2C[C@@H]1OP(O)(=O)OC[C@H]1O[C@H]([C@@H](F)C1OP(O)(=O)OC2)n1cnc2c(N)ncnc12	InChI=1S/C20H26FN11O10P2/c21-10-13-9(40-19(10)31-5-27-11-14(22)25-4-26-16(11)31)3-38-43(33,34)41-8-1-7(2-37-44(35,36)42-13)39-18(8)32-6-28-12-15(23)29-20(24)30-17(12)32/h4-10,13,15,18-19H,1-3,23H2,(H,33,34)(H,35,36)(H2,22,25,26)(H3,24,29,30)/t7-,8-,9+,10-,13?,15?,18+,19+/m0/s1	NMFBAATXPJARJT-WUFZOPORSA-N	573857	2-amino-9-[(5S,7R,8R,12aR,14R,15R,15aR)-14- (6-amino-9H-purin-9-yl)-15-fluoro-2,10- dihydroxy-2,10-dioxidooctahydro-12H-5,8- methanofuro[3,2-l][1,3,6,9,11,2,10] pentaoxadiphosphacyclotetradecin-7-yl]-1,9- dihydro-6H-purin-6-one::US11453697, Example 21	Stimulator of interferon genes protein [H232R]					 1.40					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=573857	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=573857&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			140902707	474496219							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1210922	Nc1nc2n(cnc2c(=O)[nH]1)[C@@H]1O[C@H]2C[C@@H]1OP(O)(=O)OC[C@H]1O[C@H]([C@@H](F)C1OP(O)(=O)OC2)n1cnc2c(N)ncnc12			573861	2-amino-9-[(5S,7R,8R,12aR,14R,15S,15aR)-14- (6-amino-9H-purin-9-yl)-15-fluoro-2,10- dihydroxy-2,10-dioxidooctahydro-12H-5,8- methanofuro[3,2-l][1,3,6,9,11,2,10] pentaoxadiphosphacyclotetradecin-7-yl]-1,9- dihydro-6H-purin-6-one::US11453697, Example 25	Stimulator of interferon genes protein [H232R]					 16.1					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=573861	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=573861&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177474	474496223							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1210923	Nc1nc2n(cnc2c(=O)[nH]1)[C@@H]1O[C@@H]2COP(O)(=O)OC3[C@@H](COP(O)(=O)O[C@H]1C2F)O[C@H]([C@H]3F)n1cnc2c(N)ncnc12			573859	2-amino-9- [(5R,7R,8S,12aR,14R,15R,15aR,16R)-14-(6- amino-9H-purin-9-yl)-15,16-difluoro-2,10- dihydroxy-2,10-dioxidooctahydro-12H-5,8- methanofuro[3,2-l][1,3,6,9,11,2,10] pentaoxadiphosphacyclotetradecin-7-yl]-1,9- dihydro-6H-purin-6-one::US11453697, Example 23::US11453697, Example 26	Stimulator of interferon genes protein [H232R]					 3.70					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=573859	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=573859&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177472	474496221							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1210924	Nc1nc2n(cnc2c(=O)[nH]1)[C@@H]1O[C@H]2C[C@H]1OP(O)(=O)OC[C@H]1O[C@H](C[C@@H]1OP(O)(=O)OC2)n1cnc2c(N)ncnc12	InChI=1S/C20H24N10O11P2/c21-15-13-16(24-5-23-15)29(6-25-13)12-2-9-11(39-12)4-37-43(34,35)41-10-1-8(3-36-42(32,33)40-9)38-19(10)30-7-26-14-17(30)27-20(22)28-18(14)31/h5-12,19H,1-4H2,(H,32,33)(H,34,35)(H2,21,23,24)(H3,22,27,28,31)/t8-,9-,10+,11+,12+,19+/m0/s1	QZIXPPJOQTVBNB-MFRTWQQUSA-N	50509425	CHEMBL4566174::US11453697, Example 27	Stimulator of interferon genes protein [H232R]					 10.00					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50509425	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50509425&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			137102549	440718010							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1210925	C[C@@H]1[C@@H]2OP(O)(=O)OC[C@@H]3C[C@@H](OP(O)(=O)OC[C@H]2O[C@H]1n1cnc2c(N)ncnc12)[C@@H](O3)n1cnc2c1nc(N)[nH]c2=O			573864	2-amino-9-[(5S,7R,8R,12aR,14R,15R,15aS)-14- (6-amino-9H-purin-9-yl)-2,10-dihydroxy-15- methyl-2,10-dioxidooctahydro-12H-5,8- methanofuro[3,2-l][1,3,6,9,11,2,10] pentaoxadiphosphacyclotetradecin-7-yl]-1,9- dihydro-6H-purin-6-one::US11453697, Example 28	Stimulator of interferon genes protein [H232R]					 265					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=573864	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=573864&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177475	474496225							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1210926	C[C@]1(F)[C@@H]2OP(O)(=O)OC[C@@H]3C[C@@H](OP(O)(=O)OC[C@H]2OC1n1cnc2c(N)ncnc12)C(O3)n1cnc2c1nc(N)[nH]c2=O			574007	2-amino-9-[(5S,8R,12aR,15S,15aR)-14-(6- amino-9H-purin-9-yl)-15-fluoro-2,10-dihydroxy- 15-methyl-2,10-dioxidooctahydro-12H-5,8- methanofuro[3,2-l][1,3,6,9,11,2,10] pentaoxadiphosphacyclotetradecin-7-yl]-1,9- dihydro-6H-purin-6-one::US11453697, Example 29	Stimulator of interferon genes protein [H232R]					 5835					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574007	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574007&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177567	474496330							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1210927	Nc1nc2n(cnc2c(=O)[nH]1)[C@@H]1O[C@@H]2COP(O)(=O)O[C@@H]3[C@@H](COP(O)(=O)O[C@@H]1[C@@H]2O)O[C@H]([C@@H]3O)n1cnc2c(Cl)ncnc12			573867	2-amino-9- [(5R,7R,8R,12aR,14R,15R,15aS,16R)-14- (6-chloro-9H-purin-9-yl)-2,10,15,16- tetrahydroxy-2,10-dioxidooctahydro-12H- 5,8-methanofuro[3,2-l][1,3,6,9,11,2,10] pentaoxadiphosphacyclotetradecin-7-yl]- 1,9-dihydro-6H-purin-6-one::US11453697, Example 32	Stimulator of interferon genes protein [H232R]					 25.0					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=573867	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=573867&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177477	474496228							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1210928	NC1NC(N)=Nc2c1ncn2[C@@H]1O[C@@H]2COP(O)(=S)O[C@@H]3[C@@H](COP(O)(=O)O[C@@H]1[C@@H]2O)O[C@H]([C@@H]3O)n1cnc2c(N)ncnc12	InChI=1S/C20H27N11O11P2S/c21-14-8-16(25-3-24-14)30(4-26-8)18-11(33)12-7(40-18)2-37-43(34,35)41-13-10(32)6(1-38-44(36,45)42-12)39-19(13)31-5-27-9-15(22)28-20(23)29-17(9)31/h3-7,10-13,15,18-19,32-33H,1-2,22H2,(H,34,35)(H,36,45)(H2,21,24,25)(H3,23,28,29)/t6-,7-,10-,11-,12-,13-,15?,18-,19-,44?/m1/s1	RWIPJGKLHFTWQC-GIOTYLNYSA-N	573873	2-amino-9- [(5R,7R,8R,12aR,14R,15R,15aS,16R)-14- (6-amino-9H-purin-9-yl)-2,10,15,16- tetrahydroxy-10-oxido-2-sulfidooctahydro- 12H-5,8-methanofuro[3,2- l][1,3,6,9,11,2,10] pentaoxadiphosphacyclotetradecin-7-yl]- 1,9-dihydro-6H-purin-6-one::US11453697, Example 38	Stimulator of interferon genes protein [H232R]					 24.9					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=573873	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=573873&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			140902706	474496234							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1210929	Nc1nc2n(cnc2c(=O)[nH]1)[C@@H]1O[C@@H]2COP(O)(=O)O[C@@H]3[C@@H](COP(O)(=O)O[C@@H]1[C@@H]2O)O[C@H]([C@@H]3O)c1ccc2c(N)ncnn12			573882	2-amino-9- [(5R,7R,8R,12aR,14S,15S,15aS,16R)-14- (4-aminopyrrolo[2,1-f][1,2,4]triazin-7-yl)- 2,10,15,16-tetrahydroxy-2,10- dioxidooctahydro-12H-5,8- methanofuro[3,2-l][1,3,6,9,11,2,10] pentaoxadiphosphacyclotetradecin-7-yl]- 1,9-dihydro-6H-purin-6-one::US11453697, Example 41	Stimulator of interferon genes protein [H232R]					 506					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=573882	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=573882&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177491	474496243							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1210930	Nc1nc(N)c2ncn([C@@H]3O[C@@H]4COP(O)(=O)O[C@@H]5[C@H](O)[C@@H](COP(O)(=O)O[C@H]4[C@H]3O)O[C@H]5n3cnc4c3nc(N)[nH]c4=O)c2n1			573883	2-amino-9- [(5R,7R,8R,12aR,14R,15R,15aS,16R)-14- (2,6-diamino-9H-purin-9-yl)-2,10,15,16- tetrahydroxy-2,10-dioxidooctahydro-12H- 5,8-methanofuro[3,2-l][1,3,6,9,11,2,10] pentaoxadiphosphacyclotetradecin-7-yl]- 1,9-dihydro-6H-purin-6-one::US11453697, Example 42	Stimulator of interferon genes protein [H232R]					 219					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=573883	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=573883&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177492	474496244							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1210931	Nc1nc2n(cnc2c(=O)[nH]1)[C@@H]1O[C@@H]2COP(O)(=O)O[C@@H]3[C@@H](COP(O)(=O)O[C@@H]1[C@@H]2O)O[C@H]([C@@H]3O)n1ccc2c(N)ncnc12	InChI=1S/C21H25N9O13P2/c22-15-7-1-2-29(16(7)25-5-24-15)19-12(32)13-9(41-19)4-39-45(36,37)43-14-11(31)8(3-38-44(34,35)42-13)40-20(14)30-6-26-10-17(30)27-21(23)28-18(10)33/h1-2,5-6,8-9,11-14,19-20,31-32H,3-4H2,(H,34,35)(H,36,37)(H2,22,24,25)(H3,23,27,28,33)/t8-,9-,11-,12-,13-,14-,19-,20-/m1/s1	UTYHBKZTJXGVRM-NFASUMMFSA-N	50509409	CHEMBL4578839::US11453697, Example 43	Stimulator of interferon genes protein [H232R]					 1015					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50509409	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50509409&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	KT2	6S26	137102595	440717994							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1210932	Nc1ncnc2n(cnc12)[C@@H]1O[C@@H]2COP(O)(=O)O[C@@H]3[C@H](O)[C@@H](COP(O)(=O)O[C@H]2[C@H]1O)O[C@H]3n1cnc2c1[nH]c(=O)[nH]c2=O			573885	9-[(5R,7R,8R,12aR,14R,15R,15aS,16R)- 14-(6-amino-9H-purin-9-yl)-2,10,15,16- tetrahydroxy-2,10-dioxidooctahydro-12H- 5,8-methanofuro[3,2-l][1,3,6,9,11,2,10] pentaoxadiphosphacyclotetradecin-7-yl]- 3,9-dihydro-1H-purine-2,6-dione::US11453697, Example 44	Stimulator of interferon genes protein [H232R]					 1363					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=573885	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=573885&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177493	474496246							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1210933	Nc1nc2n(cnc2c(=O)[nH]1)[C@@H]1O[C@H]2C[C@H]1OP(O)(=O)OC[C@H]1O[C@H]([C@H](O)[C@@H]1OP(O)(=O)OC2)n1ccc2c(N)ncnc12			573886	2-amino-9- [(5S,7R,8R,12aR,14R,15R,15aS)-14-(4- amino-7H-pyrrolo[2,3-d]pyrimidin-7-yl)- 2,10,15-trihydroxy-2,10-dioxidooctahydro- 12H-5,8-methanofuro[3,2- l][1,3,6,9,11,2,10] pentaoxadiphosphacyclotetradecin-7-yl]- 1,9-dihydro-6H-purin-6-one::US11453697, Example 45	Stimulator of interferon genes protein [H232R]					 105					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=573886	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=573886&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177494	474496247							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1210934	Nc1nc2n(cnc2c(=O)[nH]1)[C@@H]1O[C@]2(F)COP(O)(=O)O[C@@H]3[C@@H](COP(O)(=O)O[C@@H]1[C@@H]2O)O[C@H]([C@@H]3O)n1cnc2c(N)ncnc12			573887	2-amino-9- [(5S,7R,8R,12aR,14R,15R,15aS,16S)-14- (6-amino-9H-purin-9-yl)-5-fluoro- 2,10,15,16-tetrahydroxy-2,10- dioxidooctahydro-12H-5,8- methanofuro[3,2-l][1,3,6,9,11,2,10] pentaoxadiphosphacyclotetradecin-7-yl]- 1,9-dihydro-6H-purin-6-one::US11453697, Example 46	Stimulator of interferon genes protein [H232R]					 337					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=573887	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=573887&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177495	474496248							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1210935	Nc1nc(N)c2ncn([C@@H]3O[C@@H]4COP(O)(=O)O[C@@H]5[C@H](O)[C@@H](COP(O)(=O)O[C@H]4[C@H]3O)O[C@H]5n3cnc4c3nc[nH]c4=O)c2n1			573888	9-[(5R,7R,8R,12aR,14R,15R,15aS,16R)- 14-(2,6-diamino-9H-purin-9-yl)-2,10,15,16- tetrahydroxy-2,10-dioxidooctahydro-12H- 5,8-methanofuro[3,2-l][1,3,6,9,11,2,10] pentaoxadiphosphacyclotetradecin-7-yl]- 1,9-dihydro-6H-purin-6-one::US11453697, Example 47	Stimulator of interferon genes protein [H232R]					 444					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=573888	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=573888&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177496	474496249							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1210936	Nc1nc2n(cnc2c(=O)[nH]1)[C@@H]1O[C@@H]2COP(O)(=O)O[C@@H]3[C@@H](COP(O)(=O)O[C@@H]1[C@@H]2O)O[C@H]([C@@H]3O)n1cnc2c(N)nccc12			573892	2-amino-9- [(5R,7R,8R,12aR,14R,15R,15aS,16R)-14- (4-amino-1H-imidazo[4,5-c]pyridin-1-yl)- 2,10,15,16-tetrahydroxy-2,10- dioxidooctahydro-12H-5,8- methanofuro[3,2-l][1,3,6,9,11,2,10] pentaoxadiphosphacyclotetradecin-7-yl]- 1,9-dihydro-6H-purin-6-one::US11453697, Example 51	Stimulator of interferon genes protein [H232R]					 996					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=573892	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=573892&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177499	474496253							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1210937	Nc1ncnc2n(ccc12)[C@@H]1O[C@@H]2COP(O)(=O)O[C@@H]3[C@H](O)[C@@H](COP(O)(=O)O[C@H]2[C@H]1O)O[C@H]3n1cnc2c1cc[nH]c2=O			573902	1-[(5R,7R,8R,12aR,14R,15R,15aS,16R)- 14-(4-amino-7H-pyrrolo[2,3-d]pyrimidin-7- yl)-2,10,15,16-tetrahydroxy-2,10- dioxidooctahydro-12H-5,8- methanofuro[3,2-l][1,3,6,9,11,2,10] pentaoxadiphosphacyclotetradecin-7-yl]- 1,5-dihydro-4H-imidazo[4,5-c]pyridin-4- one::US11453697, Example 61	Stimulator of interferon genes protein [H232R]					 379					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=573902	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=573902&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177507	474496263							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1210938	Nc1nc2n(cnc2c(=O)[nH]1)[C@@H]1O[C@@H]2COP(O)(=O)O[C@@H]3[C@@H](COP(O)(=O)O[C@@H]1C2=C)O[C@H]([C@@H]3O)n1cnc2c(N)ncnc12			574008	2-amino-9- [(5S,7R,8R,12aR,14R,15R,15aS)-14-(6- amino-9H-purin-9-yl)-2,10,15-trihydroxy- 16-methylidene-2,10-dioxidooctahydro- 12H-5,8-methanofuro[3,2- l][1,3,6,9,11,2,10]/ pentaoxadiphosphacyclotetradecin-7-yl]- 1,9-dihydro-6H-purin-6-one::US11453697, Example 62	Stimulator of interferon genes protein [H232R]					 2.60					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574008	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574008&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177568	474496331							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1210939	Nc1ncnc2n(cnc12)[C@@H]1O[C@@H]2COP(O)(=O)O[C@@H]3[C@@H](COP(O)(=O)O[C@@H]1[C@@H]2O)O[C@H]([C@@H]3O)n1cnc2c1nn[nH]c2=O			574009	7-[(5R,7R,8R,12aR,14R,15R,15aS,16R)-7- (6-amino-9H-purin-9-yl)-2,10,15,16- tetrahydroxy-2,10-dioxidooctahydro-12H- 5,8-methanofuro[3,2-l][1,3,6,9,11,2,10] pentaoxadiphosphacyclotetradecin-14-yl]- 3,7-dihydro-4H-imidazo[4,5- d][1,2,3]triazin-4-one::US11453697, Example 63	Stimulator of interferon genes protein [H232R]					 68.8					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574009	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574009&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177569	474496332							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1210940	Nc1ccnc2n(cnc12)[C@@H]1O[C@@H]2COP(O)(=O)O[C@@H]3[C@H](O)[C@@H](COP(O)(=O)O[C@H]2[C@H]1O)O[C@H]3n1cnc2c1nc(N)[nH]c2=O			574010	2-amino-9- [(5R,7R,8R,12aR,14R,15R,15aS,16R)-14- (7-amino-3H-imidazo[4,5-b]pyridin-3-yl)- 2,10,15,16-tetrahydroxy-2,10- dioxidooctahydro-12H-5,8- methanofuro[3,2-l][1,3,6,9,11,2,10] pentaoxadiphosphacyclotetradecin-7-yl]- 1,9-dihydro-6H-purin-6-one::US11453697, Example 64	Stimulator of interferon genes protein [H232R]					 61.6					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574010	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574010&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177570	474496333							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1210941	Nc1ncnc2n(cnc12)[C@@H]1O[C@@H]2COP(O)(=O)O[C@@H]3[C@H](O)[C@@H](COP(O)(=O)O[C@H]2[C@H]1O)O[C@H]3n1cnc2c1cn[nH]c2=O			574011	1-[(5R,7R,8R,12aR,14R,15R,15aS,16R)- 14-(6-amino-9H-purin-9-yl)-2,10,15,16- tetrahydroxy-2,10-dioxidooctahydro-12H- 5,8-methanofuro[3,2-l][1,3,6,9,11,2,10] pentaoxadiphosphacyclotetradecin-7-yl]- 1,5-dihydro-4H-imidazo[4,5-d]pyridazin-4- one::US11453697, Example 65	Stimulator of interferon genes protein [H232R]					 250					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574011	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574011&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177571	474496334							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1210942	Cc1ncnc2n(cnc12)[C@@H]1O[C@@H]2COP(O)(=O)O[C@@H]3[C@H](O)[C@@H](COP(O)(=O)O[C@H]2[C@H]1O)O[C@H]3n1cnc2c1nc(N)[nH]c2=O			573875	2-amino-9- [(5R,7R,8R,12aR,14R,15R,15aS,16R)- 2,10,15,16-tetrahydroxy-14-(6-methyl-9H- purin-9-yl)-2,10-dioxidooctahydro-12H-5,8- methanofuro[3,2-l][1,3,6,9,11,2,10] pentaoxadiphosphacyclotetradecin-7-yl]- 1,9-dihydro-6H-purin-6-one::US11453697, Example 70	Stimulator of interferon genes protein [H232R]					 19.4					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=573875	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=573875&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177484	474496236							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1210943	Nc1nc2n(cnc2c(=O)[nH]1)[C@@H]1O[C@@H]2COP(O)(=O)O[C@@H]3[C@@H](COP(O)(=O)O[C@@H]1[C@@H]2O)O[C@H]([C@@H]3O)n1ccc2c(Cl)ncnc12			573876	2-amino-9- [(5R,7R,8R,12aR,14R,15R,15aS,16R)-14- (4-chloro-7H-pyrrolo[2,3-d]pyrimidin-7- yl)-2,10,15,16-tetrahydroxy-2,10- dioxidooctahydro-12H-5,8- methanofuro[3,2-l][1,3,6,9,11,2,10] pentaoxadiphosphacyclotetradecin-7-yl]- 1,9-dihydro-6H-purin-6-one::US11453697, Example 71	Stimulator of interferon genes protein [H232R]					 4.40					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=573876	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=573876&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177485	474496237							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1210944	Nc1nc2n(cnc2c(=O)[nH]1)[C@@H]1O[C@@H]2COP(O)(=O)O[C@@H]3[C@@H](COP(O)(=O)O[C@@H]1[C@@H]2O)O[C@H]([C@@H]3O)n1cnc2cncnc12			573877	2-amino-9- [(5R,7R,8R,12aR,14R,15R,15aS,16R)- 2,10,15,16-tetrahydroxy-2,10-dioxido-14- (9H-purin-9-yl)octahydro-12H-5,8- methanofuro[3,2-l][1,3,6,9,11,2,10] pentaoxadiphosphacyclotetradecin-7-yl]- 1,9-dihydro-6H-purin-6-one::US11453697, Example 72	Stimulator of interferon genes protein [H232R]					<1.000					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=573877	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=573877&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177486	474496238							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1210945	Nc1nc2n(cnc2c(=O)[nH]1)[C@@H]1O[C@@H]2COP(S)(=O)OC3[C@@H](COP(S)(=O)O[C@H]1C2O)O[C@H]([C@H]3F)n1cnc2c(N)ncnc12			573912	US11453697, Example 81::US11453697, Example 82::US11453697, Example 83::US11453697, Example 90::US11453697, Example 91::US11453697, Example 92	Stimulator of interferon genes protein [H232R]					 3.10					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=573912	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=573912&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177514	474496271							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1210946	Nc1nc2n(cnc2c(=O)[nH]1)[C@@H]1O[C@@H]2COP(S)(=O)OC3[C@@H](COP(S)(=O)O[C@H]1C2O)O[C@H]([C@H]3F)n1cnc2c(N)ncnc12			573912	US11453697, Example 81::US11453697, Example 82::US11453697, Example 83::US11453697, Example 90::US11453697, Example 91::US11453697, Example 92	Stimulator of interferon genes protein [H232R]					 14.6					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=573912	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=573912&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177514	474496271							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1210947	Nc1nc2n(cnc2c(=O)[nH]1)[C@@H]1O[C@@H]2COP(S)(=O)OC3C[C@@H](O[C@@H]3COP(S)(=O)O[C@H]1C2O)n1cnc2c(N)ncnc12			573915	2-amino-9-[(5R,7R,8R,12aR,14R,15aS,16R)-14- (6-amino-9H-purin-9-yl)-2,10,16-trihydroxy- 2,10-disulfidooctahydro-12H-5,8- methanofuro[3,2-l][1,3,6,9,11,2,10] pentaoxadiphosphacyclotetradecin-7-yl]-1,9- dihydro-6H-purin-6-one (Diastereomer 2)::US11453697, Example 84::US11453697, Example 85	Stimulator of interferon genes protein [H232R]					 6.30					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=573915	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=573915&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177515	474496272							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1210948	Nc1nc2n(cnc2c(=O)[nH]1)[C@@H]1O[C@H]2C[C@@H]1O[P@@](S)(=O)OC[C@H]1O[C@H]([C@@H](O)C1O[P@@](S)(=O)OC2)n1cnc2c(N)ncnc12			573916	2-amino-9-[(2R,5S,7R,8R,10R, 12aR,14R,15R,15aS)-14-(6-amino-9H-purin-9- yl)-2,10,15-trihydroxy-2,10-disulfidooctahydro- 12H-5,8-methanofuro[3,2-1][1,3,6,9,11,2,10] pentaoxadiphosphacyclotetradecin-7-yl]-1,9- dihydro-6H-purin-6-one (Diastereomer 1)::US11453697, Example 86	Stimulator of interferon genes protein [H232R]					 2.00					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=573916	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=573916&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177516	474496273							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1210949	Nc1nc2n(cnc2c(=O)[nH]1)[C@@H]1O[C@@H]2CO[P@](S)(=O)OC3[C@@H](CO[P@](S)(=O)O[C@H]1C2O)O[C@H]([C@H]3F)n1cnc2c(N)ncnc12			573919	2-amino-9-[(2R,5R,7R,8R,10,R, 12aR,14R,15S,15aR,16R)-14-(6-amino-9H- purin-9-yl)-15-fluoro-2,10,16-trihydroxy-2,10- disulfidooctahydro-12H-5,8- methanofuro[3,2-l][1,3,6,9,11,2,10] pentaoxadiphosphacyclotetradecin-7-yl]-1,9- dihydro-6H-purin-6-one (Diastereomer 1)::US11453697, Example 89	Stimulator of interferon genes protein [H232R]					<1.000					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=573919	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=573919&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177517	474496275							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1210950	Nc1nc2n(cnc2c(=O)[nH]1)[C@@H]1O[C@@H]2COP(S)(=O)OC3[C@@H](COP(S)(=O)O[C@H]1C2O)O[C@H]([C@H]3F)n1cnc2c(N)ncnc12			573912	US11453697, Example 81::US11453697, Example 82::US11453697, Example 83::US11453697, Example 90::US11453697, Example 91::US11453697, Example 92	Stimulator of interferon genes protein [H232R]					 4.40					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=573912	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=573912&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177514	474496271							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1210951	Nc1nc2n(cnc2c(=O)[nH]1)[C@@H]1O[C@@H]2COP(S)(=O)OC3[C@@H]4OC[C@]3(COP(S)(=O)O[C@H]1C2O)O[C@H]4n1cnc2c(N)ncnc12			573923	2-amino-9- [(5R,7R,8R,12aR,14R,15R,15aS,18R)-14-(6- amino-9H-purin-9-yl)-2,10,18-trihydroxy-2,10- disulfidohexahydro-14H-15,12a- (epoxymethano)-5,8-methanofuro [3,2-l][1,3,6,9,11,2,10] pentaoxadiphosphacyclotetradecin-7(12H)-yl]- 1,9-dihydro-6H-purin-6-one (Diastereomer 1)::US11453697, Example 93::US11453697, Example 94::US11453697, Example 95	Stimulator of interferon genes protein [H232R]					 1.90					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=573923	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=573923&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177518	474496276							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1210952	Nc1nc2n(cnc2c(=O)[nH]1)[C@@H]1O[C@@H]2COP(S)(=O)OC3[C@@H]4OC[C@]3(COP(S)(=O)O[C@H]1C2O)O[C@H]4n1cnc2c(N)ncnc12			573923	2-amino-9- [(5R,7R,8R,12aR,14R,15R,15aS,18R)-14-(6- amino-9H-purin-9-yl)-2,10,18-trihydroxy-2,10- disulfidohexahydro-14H-15,12a- (epoxymethano)-5,8-methanofuro [3,2-l][1,3,6,9,11,2,10] pentaoxadiphosphacyclotetradecin-7(12H)-yl]- 1,9-dihydro-6H-purin-6-one (Diastereomer 1)::US11453697, Example 93::US11453697, Example 94::US11453697, Example 95	Stimulator of interferon genes protein [H232R]					 524					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=573923	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=573923&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177518	474496276							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1210953	Nc1nc2n(cnc2c(=O)[nH]1)[C@@H]1O[C@@H]2COP(S)(=O)OC3[C@@H]4OC[C@]3(COP(S)(=O)O[C@H]1C2O)O[C@H]4n1cnc2c(N)ncnc12			573923	2-amino-9- [(5R,7R,8R,12aR,14R,15R,15aS,18R)-14-(6- amino-9H-purin-9-yl)-2,10,18-trihydroxy-2,10- disulfidohexahydro-14H-15,12a- (epoxymethano)-5,8-methanofuro [3,2-l][1,3,6,9,11,2,10] pentaoxadiphosphacyclotetradecin-7(12H)-yl]- 1,9-dihydro-6H-purin-6-one (Diastereomer 1)::US11453697, Example 93::US11453697, Example 94::US11453697, Example 95	Stimulator of interferon genes protein [H232R]					 64.0					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=573923	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=573923&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177518	474496276							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1210954	Nc1nc2n(cnc2c(=O)[nH]1)[C@@H]1S[C@@H]2COP(S)(=O)O[C@@H]3[C@@H](COP(S)(=O)O[C@@H]1[C@@H]2O)O[C@H]([C@H]3F)n1cnc2c(N)ncnc12			573926	2-amino-9- [(5R,7R,8R,12aR,14R,15S,15aR,16S)-14-(6- amino-9H-purin-9-yl)-15-fluoro-16-hydroxy- 2,10-dioxido-2,10-disulfanyloctahydro-12H-5,8- methanofuro[3,2-l][1,3,9,11,6,2,10] tetraoxathiadiphosphacyclotetradecin-7-yl]-1,9- dihydro-6H-purin-6-one (Diastereomer 1)::US11453697, Example 96::US11453697, Example 98::US11453697, Example 99	Stimulator of interferon genes protein [H232R]					 57.8					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=573926	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=573926&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177519	474496277							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1210955	Nc1nc2n(cnc2c(=O)[nH]1)[C@@H]1S[C@@H]2CO[P@](S)(=O)O[C@@H]3[C@@H](CO[P@](S)(=O)O[C@@H]1[C@@H]2O)O[C@H]([C@H]3F)n1cnc2c(N)ncnc12			573927	2-amino-9-[(2R,5R,7R,8R,10R, 12aR,14R,15S,15aR,16S)-14-(6-amino-9H- purin-9-yl)-15-fluoro-16-hydroxy-2,10-dioxido- 2,10-disulfanyloctahydro-12H-5,8- methanofuro[3,2-l][1,3,9,11,6,2,10] tetraoxathiadiphosphacyclotetradecin-7-yl]-1,9- dihydro-6H-purin-6-one (Diastereomer 2)::US11453697, Example 97	Stimulator of interferon genes protein [H232R]					 0.400					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=573927	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=573927&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177519	474496278							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1210956	Nc1nc2n(cnc2c(=O)[nH]1)[C@@H]1S[C@@H]2COP(S)(=O)O[C@@H]3[C@@H](COP(S)(=O)O[C@@H]1[C@@H]2O)O[C@H]([C@H]3F)n1cnc2c(N)ncnc12			573926	2-amino-9- [(5R,7R,8R,12aR,14R,15S,15aR,16S)-14-(6- amino-9H-purin-9-yl)-15-fluoro-16-hydroxy- 2,10-dioxido-2,10-disulfanyloctahydro-12H-5,8- methanofuro[3,2-l][1,3,9,11,6,2,10] tetraoxathiadiphosphacyclotetradecin-7-yl]-1,9- dihydro-6H-purin-6-one (Diastereomer 1)::US11453697, Example 96::US11453697, Example 98::US11453697, Example 99	Stimulator of interferon genes protein [H232R]					 152					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=573926	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=573926&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177519	474496277							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1210957	Nc1nc2n(cnc2c(=O)[nH]1)[C@@H]1S[C@@H]2COP(S)(=O)O[C@@H]3[C@@H](COP(S)(=O)O[C@@H]1[C@@H]2O)O[C@H]([C@H]3F)n1cnc2c(N)ncnc12			573926	2-amino-9- [(5R,7R,8R,12aR,14R,15S,15aR,16S)-14-(6- amino-9H-purin-9-yl)-15-fluoro-16-hydroxy- 2,10-dioxido-2,10-disulfanyloctahydro-12H-5,8- methanofuro[3,2-l][1,3,9,11,6,2,10] tetraoxathiadiphosphacyclotetradecin-7-yl]-1,9- dihydro-6H-purin-6-one (Diastereomer 1)::US11453697, Example 96::US11453697, Example 98::US11453697, Example 99	Stimulator of interferon genes protein [H232R]					 1.80					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=573926	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=573926&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177519	474496277							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1210958	Nc1nc2n(cnc2c(=O)[nH]1)[C@@H]1S[C@@H]2COP(O)(=S)O[C@H]3[C@H]4OC[C@]3(COP(O)(=S)O[C@@H]1[C@@H]2O)O[C@H]4n1cnc2c(N)ncnc12			573930	2-amino-9- [(5R,7R,8R,12aR,14R,15R,15aS,18S)-14-(6- amino-9H-purin-9-yl)-2,10,18-trihydroxy-2,10- disulfidohexahydro-14H-15,12a- (epoxymethano)-5,8-methanofuro[3,2- l][1,3,9,11,6,2,10] tetraoxathiadiphosphacyclotetradecin- 7(12H)-yl]-1,9-dihydro-6H-purin-6-one (Diastereomer 1)::US11453697, Example 100::US11453697, Example 101::US11453697, Example 102	Stimulator of interferon genes protein [H232R]					 552					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=573930	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=573930&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177520	474496279							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1210959	Nc1nc2n(cnc2c(=O)[nH]1)[C@@H]1S[C@@H]2COP(O)(=S)O[C@H]3[C@H]4OC[C@]3(COP(O)(=S)O[C@@H]1[C@@H]2O)O[C@H]4n1cnc2c(N)ncnc12			573930	2-amino-9- [(5R,7R,8R,12aR,14R,15R,15aS,18S)-14-(6- amino-9H-purin-9-yl)-2,10,18-trihydroxy-2,10- disulfidohexahydro-14H-15,12a- (epoxymethano)-5,8-methanofuro[3,2- l][1,3,9,11,6,2,10] tetraoxathiadiphosphacyclotetradecin- 7(12H)-yl]-1,9-dihydro-6H-purin-6-one (Diastereomer 1)::US11453697, Example 100::US11453697, Example 101::US11453697, Example 102	Stimulator of interferon genes protein [H232R]					 74.4					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=573930	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=573930&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177520	474496279							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1210960	Nc1nc2n(cnc2c(=O)[nH]1)[C@@H]1O[C@@H]2COP(S)(=O)OC3C[C@@H](O[C@@H]3COP(S)(=O)O[C@H]1C2O)n1cnc2c(N)ncnc12			573915	2-amino-9-[(5R,7R,8R,12aR,14R,15aS,16R)-14- (6-amino-9H-purin-9-yl)-2,10,16-trihydroxy- 2,10-disulfidooctahydro-12H-5,8- methanofuro[3,2-l][1,3,6,9,11,2,10] pentaoxadiphosphacyclotetradecin-7-yl]-1,9- dihydro-6H-purin-6-one (Diastereomer 2)::US11453697, Example 84::US11453697, Example 85	Stimulator of interferon genes protein [H232R]					 6.30					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=573915	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=573915&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177515	474496272							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1210961	Nc1nc2n(cnc2c(=O)[nH]1)[C@@H]1O[C@H]2C[C@@H]1O[P@@](S)(=O)OC[C@H]1O[C@H]([C@@H](O)C1O[P@@](S)(=O)OC2)n1cnc2c(N)ncnc12			573916	2-amino-9-[(2R,5S,7R,8R,10R, 12aR,14R,15R,15aS)-14-(6-amino-9H-purin-9- yl)-2,10,15-trihydroxy-2,10-disulfidooctahydro- 12H-5,8-methanofuro[3,2-1][1,3,6,9,11,2,10] pentaoxadiphosphacyclotetradecin-7-yl]-1,9- dihydro-6H-purin-6-one (Diastereomer 1)::US11453697, Example 86	Stimulator of interferon genes protein [H232R]					 2.00					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=573916	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=573916&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177516	474496273							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1210962	Nc1nc2n(cnc2c(=O)[nH]1)[C@@H]1S[C@@H]2COP(O)(=S)O[C@H]3[C@H]4OC[C@]3(COP(O)(=S)O[C@@H]1[C@@H]2O)O[C@H]4n1cnc2c(N)ncnc12			573930	2-amino-9- [(5R,7R,8R,12aR,14R,15R,15aS,18S)-14-(6- amino-9H-purin-9-yl)-2,10,18-trihydroxy-2,10- disulfidohexahydro-14H-15,12a- (epoxymethano)-5,8-methanofuro[3,2- l][1,3,9,11,6,2,10] tetraoxathiadiphosphacyclotetradecin- 7(12H)-yl]-1,9-dihydro-6H-purin-6-one (Diastereomer 1)::US11453697, Example 100::US11453697, Example 101::US11453697, Example 102	Stimulator of interferon genes protein [H232R]					 1.000					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=573930	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=573930&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177520	474496279							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1210963	Nc1nc2n(cnc2c(=O)[nH]1)[C@@H]1O[C@@H]2COP(O)(=S)O[C@H]3[C@@H](O)[C@@H](O[C@@]3(COP(O)(=S)O[C@@H]1[C@H]2F)C#C)n1cnc2c(N)ncnc12			574013	2-amino-9- [(5R,7R,8S,12aR,14R,15R,15aS,16S)-14-(6- amino-9H-purin-9-yl)-12a-ethynyl-16-fluoro- 2,10,15-trihydroxy-2,10-disulfidooctahydro-12H- 5,8-methanofuro[3,2-l][1,3,6,9,11,2,10] pentaoxadiphosphacyclotetradecin-7-yl]-1,9- dihydro-6H-purin-6-one (Diastereomer 1)::US11453697, Example 103::US11453697, Example 104::US11453697, Example 105	Stimulator of interferon genes protein [H232R]					<1.000					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574013	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574013&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177572	474496335							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1210964	Nc1nc2n(cnc2c(=O)[nH]1)[C@@H]1O[C@@H]2COP(O)(=S)O[C@H]3[C@@H](O)[C@@H](O[C@@]3(COP(O)(=S)O[C@@H]1[C@H]2F)C#C)n1cnc2c(N)ncnc12			574013	2-amino-9- [(5R,7R,8S,12aR,14R,15R,15aS,16S)-14-(6- amino-9H-purin-9-yl)-12a-ethynyl-16-fluoro- 2,10,15-trihydroxy-2,10-disulfidooctahydro-12H- 5,8-methanofuro[3,2-l][1,3,6,9,11,2,10] pentaoxadiphosphacyclotetradecin-7-yl]-1,9- dihydro-6H-purin-6-one (Diastereomer 1)::US11453697, Example 103::US11453697, Example 104::US11453697, Example 105	Stimulator of interferon genes protein [H232R]					 11.6					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574013	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574013&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177572	474496335							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1210965	Nc1nc2n(cnc2c(=O)[nH]1)[C@@H]1O[C@@H]2COP(O)(=S)O[C@H]3[C@@H](O)[C@@H](O[C@@]3(COP(O)(=S)O[C@@H]1[C@H]2F)C#C)n1cnc2c(N)ncnc12			574013	2-amino-9- [(5R,7R,8S,12aR,14R,15R,15aS,16S)-14-(6- amino-9H-purin-9-yl)-12a-ethynyl-16-fluoro- 2,10,15-trihydroxy-2,10-disulfidooctahydro-12H- 5,8-methanofuro[3,2-l][1,3,6,9,11,2,10] pentaoxadiphosphacyclotetradecin-7-yl]-1,9- dihydro-6H-purin-6-one (Diastereomer 1)::US11453697, Example 103::US11453697, Example 104::US11453697, Example 105	Stimulator of interferon genes protein [H232R]					 3.90					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574013	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574013&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177572	474496335							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1210966	Nc1nc2n(cnc2c(=O)[nH]1)[C@@H]1O[C@@H]2COP(O)(=S)O[C@H]3[C@@H](O)[C@@H](O[C@@]3(COP(O)(=S)O[C@@H]1[C@@H]2F)C#C)n1cnc2c(N)ncnc12			574016	2-amino-9- [(5R,7R,8S,12aR,14R,15R,15aS,16R)-14-(6- amino-9H-purin-9-yl)-12a-ethynyl-16-fluoro- 2,10,15-trihydroxy-2,10-disulfidooctahydro-12H- 5,8-methanofuro[3,2-l][1,3,6,9,11,2,10] pentaoxadiphosphacyclotetradecin-7-yl]-1,9- dihydro-6H-purin-6-one (Diastereomer 1)::US11453697, Example 106::US11453697, Example 107	Stimulator of interferon genes protein [H232R]					<1.000					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574016	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574016&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177573	474496336							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1210967	Nc1nc2n(cnc2c(=O)[nH]1)[C@@H]1O[C@@H]2COP(O)(=S)O[C@H]3[C@@H](O)[C@@H](O[C@@]3(COP(O)(=S)O[C@@H]1[C@@H]2F)C#C)n1cnc2c(N)ncnc12			574016	2-amino-9- [(5R,7R,8S,12aR,14R,15R,15aS,16R)-14-(6- amino-9H-purin-9-yl)-12a-ethynyl-16-fluoro- 2,10,15-trihydroxy-2,10-disulfidooctahydro-12H- 5,8-methanofuro[3,2-l][1,3,6,9,11,2,10] pentaoxadiphosphacyclotetradecin-7-yl]-1,9- dihydro-6H-purin-6-one (Diastereomer 1)::US11453697, Example 106::US11453697, Example 107	Stimulator of interferon genes protein [H232R]					 17.9					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574016	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574016&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177573	474496336							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1210968	Nc1nc2n(nnc2c(=O)[nH]1)[C@@H]1S[C@@H]2COP(S)(=O)O[C@H]3C[C@@H](O[C@@H]3COP(S)(=O)O[C@@H]1[C@@H]2O)c1cnn2c(N)ncnc12			574018	5-amino-3-[(5R,7R,8R,12aR,14R,15aS,16S)-14- (4-aminopyrazolo[1,5-a][1,3,5]triazin-8-yl)-16- hydroxy-2,10-dioxido-2,10-disulfanyloctahydro- 12H-5,8-methanofuro[3,2-l][1,3,9,11,6,2,10] tetraoxathiadiphosphacyclotetradecin-7-yl]-3,6- dihydro-7H-[1,2,3]triazolo[4,5-d]pyrimidin-7- one (Diastereomer 1)::US11453697, Example 108::US11453697, Example 109::US11453697, Example 110	Stimulator of interferon genes protein [H232R]					 1784					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574018	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574018&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177574	474496337							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1210969	Nc1nc2n(nnc2c(=O)[nH]1)[C@@H]1S[C@@H]2COP(S)(=O)O[C@H]3C[C@@H](O[C@@H]3COP(S)(=O)O[C@@H]1[C@@H]2O)c1cnn2c(N)ncnc12			574018	5-amino-3-[(5R,7R,8R,12aR,14R,15aS,16S)-14- (4-aminopyrazolo[1,5-a][1,3,5]triazin-8-yl)-16- hydroxy-2,10-dioxido-2,10-disulfanyloctahydro- 12H-5,8-methanofuro[3,2-l][1,3,9,11,6,2,10] tetraoxathiadiphosphacyclotetradecin-7-yl]-3,6- dihydro-7H-[1,2,3]triazolo[4,5-d]pyrimidin-7- one (Diastereomer 1)::US11453697, Example 108::US11453697, Example 109::US11453697, Example 110	Stimulator of interferon genes protein [H232R]					 1393					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574018	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574018&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177574	474496337							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1210970	Nc1nc2n(nnc2c(=O)[nH]1)[C@@H]1S[C@@H]2COP(S)(=O)O[C@H]3C[C@@H](O[C@@H]3COP(S)(=O)O[C@@H]1[C@@H]2O)c1cnn2c(N)ncnc12			574018	5-amino-3-[(5R,7R,8R,12aR,14R,15aS,16S)-14- (4-aminopyrazolo[1,5-a][1,3,5]triazin-8-yl)-16- hydroxy-2,10-dioxido-2,10-disulfanyloctahydro- 12H-5,8-methanofuro[3,2-l][1,3,9,11,6,2,10] tetraoxathiadiphosphacyclotetradecin-7-yl]-3,6- dihydro-7H-[1,2,3]triazolo[4,5-d]pyrimidin-7- one (Diastereomer 1)::US11453697, Example 108::US11453697, Example 109::US11453697, Example 110	Stimulator of interferon genes protein [H232R]					 141					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574018	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574018&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177574	474496337							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1210971	Nc1nc2n(nnc2c(=O)[nH]1)[C@@H]1S[C@@H]2COP(S)(=O)O[C@H]3C[C@@H](O[C@@H]3COP(S)(=O)O[C@@H]1[C@@H]2O)c1cnc2c(N)ncnn12			574021	5-amino-3-[(5R,7R,8R,12aR,14R,15aS,16S)-14- (4-aminoimidazo[2,1-f][1,2,4]triazin-7-yl)-16- hydroxy-2,10-dioxido-2,10-disulfanyloctahydro- 12H-5,8-methanofuro[3,2-l][1,3,9,11,6,2,10] tetraoxathiadiphosphacyclotetradecin-7-yl]-3,6- dihydro-7H-[1,2,3]triazolo[4,5-d] pyrimidin-7-one (Diastereomer 1)::US11453697, Example 111::US11453697, Example 112::US11453697, Example 113::US11453697, Example 114	Stimulator of interferon genes protein [H232R]					 155					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574021	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574021&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177575	474496338							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1210972	Nc1nc2n(nnc2c(=O)[nH]1)[C@@H]1S[C@@H]2COP(S)(=O)O[C@H]3C[C@@H](O[C@@H]3COP(S)(=O)O[C@@H]1[C@@H]2O)c1cnc2c(N)ncnn12			574021	5-amino-3-[(5R,7R,8R,12aR,14R,15aS,16S)-14- (4-aminoimidazo[2,1-f][1,2,4]triazin-7-yl)-16- hydroxy-2,10-dioxido-2,10-disulfanyloctahydro- 12H-5,8-methanofuro[3,2-l][1,3,9,11,6,2,10] tetraoxathiadiphosphacyclotetradecin-7-yl]-3,6- dihydro-7H-[1,2,3]triazolo[4,5-d] pyrimidin-7-one (Diastereomer 1)::US11453697, Example 111::US11453697, Example 112::US11453697, Example 113::US11453697, Example 114	Stimulator of interferon genes protein [H232R]					 1279					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574021	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574021&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177575	474496338							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1210973	Nc1nc2n(nnc2c(=O)[nH]1)[C@@H]1S[C@@H]2COP(S)(=O)O[C@H]3C[C@@H](O[C@@H]3COP(S)(=O)O[C@@H]1[C@@H]2O)c1cnc2c(N)ncnn12			574021	5-amino-3-[(5R,7R,8R,12aR,14R,15aS,16S)-14- (4-aminoimidazo[2,1-f][1,2,4]triazin-7-yl)-16- hydroxy-2,10-dioxido-2,10-disulfanyloctahydro- 12H-5,8-methanofuro[3,2-l][1,3,9,11,6,2,10] tetraoxathiadiphosphacyclotetradecin-7-yl]-3,6- dihydro-7H-[1,2,3]triazolo[4,5-d] pyrimidin-7-one (Diastereomer 1)::US11453697, Example 111::US11453697, Example 112::US11453697, Example 113::US11453697, Example 114	Stimulator of interferon genes protein [H232R]					 44.2					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574021	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574021&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177575	474496338							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1210974	Nc1nc2n(nnc2c(=O)[nH]1)[C@@H]1S[C@@H]2COP(S)(=O)O[C@H]3C[C@@H](O[C@@H]3COP(S)(=O)O[C@@H]1[C@@H]2O)c1cnc2c(N)ncnn12			574021	5-amino-3-[(5R,7R,8R,12aR,14R,15aS,16S)-14- (4-aminoimidazo[2,1-f][1,2,4]triazin-7-yl)-16- hydroxy-2,10-dioxido-2,10-disulfanyloctahydro- 12H-5,8-methanofuro[3,2-l][1,3,9,11,6,2,10] tetraoxathiadiphosphacyclotetradecin-7-yl]-3,6- dihydro-7H-[1,2,3]triazolo[4,5-d] pyrimidin-7-one (Diastereomer 1)::US11453697, Example 111::US11453697, Example 112::US11453697, Example 113::US11453697, Example 114	Stimulator of interferon genes protein [H232R]					 3.30					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574021	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574021&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177575	474496338							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1210975	Nc1nc2n(nnc2c(=O)[nH]1)[C@@H]1S[C@@H]2COP(S)(=O)O[C@@H]3[C@@H](COP(S)(=O)O[C@@H]1[C@@H]2O)O[C@H]([C@H]3F)n1nnc2c(N)ncnc12			574025	5-amino-3- [(5R,7R,8R,12aR,14R,15S,15aR,16S)-14-(7- amino-3H-[1,2,3]triazolo[4,5-d]pyrimidin-3-yl)- 15-fluoro-16-hydroxy-2,10-dioxido-2,10- disulfanyloctahydro-12H-5,8-methanofuro[3,2- l][1,3,9,11,6,2,10] tetraoxathiadiphosphacyclotetradecin- 7-yl]-3,6-dihydro-7H-[1,2,3] triazolo[4,5-d]pyrimidin-7-one (Diastereomer 1)::US11453697, Example 115::US11453697, Example 116	Stimulator of interferon genes protein [H232R]					 67.9					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574025	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574025&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177576	474496339							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1210976	Nc1nc2n(nnc2c(=O)[nH]1)[C@@H]1S[C@@H]2COP(S)(=O)O[C@@H]3[C@@H](COP(S)(=O)O[C@@H]1[C@@H]2O)O[C@H]([C@H]3F)n1nnc2c(N)ncnc12			574025	5-amino-3- [(5R,7R,8R,12aR,14R,15S,15aR,16S)-14-(7- amino-3H-[1,2,3]triazolo[4,5-d]pyrimidin-3-yl)- 15-fluoro-16-hydroxy-2,10-dioxido-2,10- disulfanyloctahydro-12H-5,8-methanofuro[3,2- l][1,3,9,11,6,2,10] tetraoxathiadiphosphacyclotetradecin- 7-yl]-3,6-dihydro-7H-[1,2,3] triazolo[4,5-d]pyrimidin-7-one (Diastereomer 1)::US11453697, Example 115::US11453697, Example 116	Stimulator of interferon genes protein [H232R]					 1624					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574025	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574025&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177576	474496339							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1210977	Nc1nc2n(cnc2c(=O)[nH]1)[C@@H]1O[C@@H]2COP(S)(=O)O[C@H]3C[C@@H](O[C@@H]3COP(S)(=O)O[C@@H]1[C@@H]2F)n1cnc2c(N)ncnc12			573933	2-amino-9-[(2R,5R,7R,8S,10R,12aR,14R,15aS,16R)-14-(6-amino-9H-purin-9-yl)-16-fluoro-2,10-dihydroxy-2,10-disulfidooctahydro-12H-5,8-methanofuro [3,2-l][1,3,6,9,11,2,10]pentaoxadiphosphacyclotetradecin-7-yl]-1,9-dihydro-6H-purin-6-one (Diastereomer 1) and 2-amino-9-[(5R,7R,8S,12aR,14R,15aS,16R)-14-(6-amino-91H-purin-9-yl)-16-fluoro-2,10-dihydroxy-2,10-disulfidooctahydro-12H-5,8-methanofuro[3,2-l][1,3,6,9,11,2,10]pentaoxadiphosphacyclotetradecin-7-yl]-1,9-dihydro-6H-purin-6-one (Diastereomer 2)::US11453697, Example 117::US11453697, Example 118::US11453697, Example 119::US11453697, Example 120	Stimulator of interferon genes protein [H232R]					 1.70					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=573933	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=573933&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177521	474496280							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1210978	Nc1nc2n(cnc2c(=O)[nH]1)[C@@H]1O[C@@H]2COP(S)(=O)O[C@H]3C[C@@H](O[C@@H]3COP(S)(=O)O[C@@H]1[C@@H]2F)n1cnc2c(N)ncnc12			573933	2-amino-9-[(2R,5R,7R,8S,10R,12aR,14R,15aS,16R)-14-(6-amino-9H-purin-9-yl)-16-fluoro-2,10-dihydroxy-2,10-disulfidooctahydro-12H-5,8-methanofuro [3,2-l][1,3,6,9,11,2,10]pentaoxadiphosphacyclotetradecin-7-yl]-1,9-dihydro-6H-purin-6-one (Diastereomer 1) and 2-amino-9-[(5R,7R,8S,12aR,14R,15aS,16R)-14-(6-amino-91H-purin-9-yl)-16-fluoro-2,10-dihydroxy-2,10-disulfidooctahydro-12H-5,8-methanofuro[3,2-l][1,3,6,9,11,2,10]pentaoxadiphosphacyclotetradecin-7-yl]-1,9-dihydro-6H-purin-6-one (Diastereomer 2)::US11453697, Example 117::US11453697, Example 118::US11453697, Example 119::US11453697, Example 120	Stimulator of interferon genes protein [H232R]					 1.60					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=573933	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=573933&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177521	474496280							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1210979	Nc1nc2n(cnc2c(=O)[nH]1)[C@@H]1O[C@@H]2COP(S)(=O)O[C@H]3C[C@@H](O[C@@H]3COP(S)(=O)O[C@@H]1[C@@H]2F)n1cnc2c(N)ncnc12			573933	2-amino-9-[(2R,5R,7R,8S,10R,12aR,14R,15aS,16R)-14-(6-amino-9H-purin-9-yl)-16-fluoro-2,10-dihydroxy-2,10-disulfidooctahydro-12H-5,8-methanofuro [3,2-l][1,3,6,9,11,2,10]pentaoxadiphosphacyclotetradecin-7-yl]-1,9-dihydro-6H-purin-6-one (Diastereomer 1) and 2-amino-9-[(5R,7R,8S,12aR,14R,15aS,16R)-14-(6-amino-91H-purin-9-yl)-16-fluoro-2,10-dihydroxy-2,10-disulfidooctahydro-12H-5,8-methanofuro[3,2-l][1,3,6,9,11,2,10]pentaoxadiphosphacyclotetradecin-7-yl]-1,9-dihydro-6H-purin-6-one (Diastereomer 2)::US11453697, Example 117::US11453697, Example 118::US11453697, Example 119::US11453697, Example 120	Stimulator of interferon genes protein [H232R]					 40.0					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=573933	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=573933&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177521	474496280							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1210980	Nc1nc2n(cnc2c(=O)[nH]1)[C@@H]1O[C@@H]2COP(S)(=O)O[C@H]3C[C@@H](O[C@@H]3COP(S)(=O)O[C@@H]1[C@@H]2F)n1cnc2c(N)ncnc12			573933	2-amino-9-[(2R,5R,7R,8S,10R,12aR,14R,15aS,16R)-14-(6-amino-9H-purin-9-yl)-16-fluoro-2,10-dihydroxy-2,10-disulfidooctahydro-12H-5,8-methanofuro [3,2-l][1,3,6,9,11,2,10]pentaoxadiphosphacyclotetradecin-7-yl]-1,9-dihydro-6H-purin-6-one (Diastereomer 1) and 2-amino-9-[(5R,7R,8S,12aR,14R,15aS,16R)-14-(6-amino-91H-purin-9-yl)-16-fluoro-2,10-dihydroxy-2,10-disulfidooctahydro-12H-5,8-methanofuro[3,2-l][1,3,6,9,11,2,10]pentaoxadiphosphacyclotetradecin-7-yl]-1,9-dihydro-6H-purin-6-one (Diastereomer 2)::US11453697, Example 117::US11453697, Example 118::US11453697, Example 119::US11453697, Example 120	Stimulator of interferon genes protein [H232R]					 394					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=573933	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=573933&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177521	474496280							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1210981	Nc1nc2n(cnc2c(=O)[nH]1)[C@@H]1O[C@H]2C[C@H]1OP(S)(=O)OCC1O[C@H](C[C@@H]1OP(S)(=O)OC2)n1ccc2c(N)[nH]cnc12			574027	US11453697, Example 122	Stimulator of interferon genes protein [H232R]					 179					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574027	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574027&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177577	474496340							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1210982	Nc1nc2n(cnc2c(=O)[nH]1)[C@@H]1O[C@@H]2COP(O)(=S)O[C@H]3[C@H]4OC[C@]3(COP(O)(=S)O[C@@H]1[C@H]2F)O[C@H]4n1cnc2c(N)[nH]cnc12			573939	US11453697, Example 124	Stimulator of interferon genes protein [H232R]					 4.00					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=573939	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=573939&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177523	474496282							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1210983	Nc1nc2n(cnc2c(=O)[nH]1)[C@@H]1O[C@@H]2COP(O)(=S)O[C@H]3[C@H]4OC[C@]3(COP(O)(=S)O[C@@H]1[C@H]2F)O[C@H]4n1cnc2c(N)ncnc12			573941	US11453697, Example 126	Stimulator of interferon genes protein [H232R]					 447					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=573941	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=573941&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177524	474496284							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1210984	Nc1nc2n(cnc2c(=O)[nH]1)[C@@H]1O[C@@H]2COP(O)(=S)O[C@@H]3[C@@H](COP(O)(=S)O[C@@H]1[C@@H]2F)O[C@H]([C@H]3F)n1nnc2c(N)ncnc12			573942	2-amino-9-[(5R,7R,8S,12aR,14R,15S,15aR,16R)-14-(7-amino-3H-[1,2,3]triazolo[4,5-d]pyrimidin-3-yl)-15,16-difluoro-2,10-dihydroxy-2,10-disulfidooctahydro-12H-5,8-methanofuro[3,2-l][1,3,6,9,11,2,10]pentaoxadiphosphacyclotetradecin-7-yl]-1,9-dihydro-6H-purin-6-one (Diastereomer 1)::US11453697, Example 127::US11453697, Example 128	Stimulator of interferon genes protein [H232R]					 19.5					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=573942	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=573942&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177525	474496285							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1210985	Nc1nc2n(cnc2c(=O)[nH]1)[C@@H]1O[C@@H]2COP(S)(=O)O[C@@H]3[C@@H](COP(S)(=O)O[C@@H]1[C@@H]2F)O[C@H]([C@H]3F)n1nnc2c(N)ncnc12			573944	2-amino-9- [(5R,7R,8S,12aR,14R,15S,15aR,16R)-14-(7- amino-3H-[1,2,3]triazolo[4,5-d]pyrimidin-3-yl)- 15,16-difluoro-2,10-dioxido-2,10- disulfanyloctahydro-12H-5,8-methanofuro[3,2-l] [1,3,6,9,11,2,10]pentaoxadiphosphacyclotetra- decin-7-yl]-1,9-dihydro-6H-purin-6-one (Diastereomer 3)::US11453697, Example 129	Stimulator of interferon genes protein [H232R]					 973					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=573944	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=573944&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177526	474496286							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1210986	Nc1nc2n(cnc2c(=O)[nH]1)[C@@H]1O[C@H]2C[C@H]1OP(S)(=O)OCC13CO[C@@H]([C@@H](O1)n1cnc4c(N)ncnc14)[C@@H]3OP(S)(=O)OC2			573954	2-amino-9-[(5S,7R,8R,12aR,14R,15R,15aS)-14- (6-amino-9H-purin-9-yl)-2,10-dioxido-2,10- disulfanylhexahydro-14H-15,12a- (epoxymethano)-5,8-methanofuro[3,2-l] [1,3,6,9,11,2,10]pentaoxadiphosphacyclotetra- decin-7(12H)-yl]-1,9-dihydro-6H-purin-6-one (Diastereomer 1)::US11453697, Example 139::US11453697, Example 140::US11453697, Example 141::US11453697, Example 142	Stimulator of interferon genes protein [H232R]					 1.20					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=573954	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=573954&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177531	474496292							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1210987	Nc1nc2n(cnc2c(=O)[nH]1)[C@@H]1O[C@H]2C[C@H]1OP(S)(=O)OCC13CO[C@@H]([C@@H](O1)n1cnc4c(N)ncnc14)[C@@H]3OP(S)(=O)OC2			573954	2-amino-9-[(5S,7R,8R,12aR,14R,15R,15aS)-14- (6-amino-9H-purin-9-yl)-2,10-dioxido-2,10- disulfanylhexahydro-14H-15,12a- (epoxymethano)-5,8-methanofuro[3,2-l] [1,3,6,9,11,2,10]pentaoxadiphosphacyclotetra- decin-7(12H)-yl]-1,9-dihydro-6H-purin-6-one (Diastereomer 1)::US11453697, Example 139::US11453697, Example 140::US11453697, Example 141::US11453697, Example 142	Stimulator of interferon genes protein [H232R]					<1.000					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=573954	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=573954&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177531	474496292							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1210988	Nc1nc2n(cnc2c(=O)[nH]1)[C@@H]1O[C@H]2C[C@H]1OP(S)(=O)OCC13CO[C@@H]([C@@H](O1)n1cnc4c(N)ncnc14)[C@@H]3OP(S)(=O)OC2			573954	2-amino-9-[(5S,7R,8R,12aR,14R,15R,15aS)-14- (6-amino-9H-purin-9-yl)-2,10-dioxido-2,10- disulfanylhexahydro-14H-15,12a- (epoxymethano)-5,8-methanofuro[3,2-l] [1,3,6,9,11,2,10]pentaoxadiphosphacyclotetra- decin-7(12H)-yl]-1,9-dihydro-6H-purin-6-one (Diastereomer 1)::US11453697, Example 139::US11453697, Example 140::US11453697, Example 141::US11453697, Example 142	Stimulator of interferon genes protein [H232R]					 175					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=573954	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=573954&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177531	474496292							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1210989	Nc1nc2n(cnc2c(=O)[nH]1)[C@@H]1O[C@@H]2CO[P@](S)(=O)O[C@@H]3[C@@H](CO[P@](S)(=O)O[C@@H]1[C@H]2F)O[C@H]([C@H]3F)n1cnc2c(N)ncnc12			573959	2-amino-9- [(2R,5R,7R,8S,10R,12aR,14R,15S,15aR,16S)- 14-(6-amino-9H-purin-9-yl)-15,16-difluoro- 2,10-dioxido-2,10-disulfanyloctahydro-12H-5,8- methanofuro[3,2-l][1,3,6,9,11,2,10] pentaoxadiphosphacyclotetradecin-7-yl]-1,9- dihydro-6H-purin-6-one (Diastereomer 1)::US11453697, Example 144	Stimulator of interferon genes protein [H232R]					 4.60					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=573959	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=573959&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177533	474496294							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1210990	Nc1nc2n(cnc2c(=O)[nH]1)[C@@H]1O[C@@H]2COP(S)(=O)O[C@@H]3[C@@H](COP(S)(=O)O[C@@H]1[C@H]2F)O[C@H]([C@H]3F)n1cnc2c(N)ncnc12			573960	2-amino-9- [(5R,7R,8S,12aR,14R,15S,15aR,16S)-14-(6- amino-9H-purin-9-yl)-15,16-difluoro-2,10- dioxido-2,10-disulfanyloctahydro-12H-5,8- methanofuro[3,2-l][1,3,6,9,11,2,10] pentaoxadiphosphacyclotetradecin-7-yl]-1,9- dihydro-6H-purin-6-one (Diastereomer 2)::US11453697, Example 145::US11453697, Example 146	Stimulator of interferon genes protein [H232R]					 14.0					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=573960	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=573960&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177533	474496295							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1210991	Nc1nc2n(cnc2c(=O)[nH]1)[C@@H]1O[C@@H]2COP(S)(=O)O[C@@H]3[C@@H](COP(S)(=O)O[C@@H]1[C@H]2F)O[C@H]([C@H]3F)n1nnc2c(N)ncnc12			573962	2-amino-9-[(5R,7R,8S,12aR,14R,15S,15aR,16S)-14-(7- amino-3H-[1,2,3]triazolo[4,5-d]pyrimidin-3-yl)- 15,16-difluoro-2,10-dioxido-2,10- disulfanyloctahydro-12H-5,8-methanofuro[3,2-l] [1,3,6,9,11,2,10]pentaoxadiphosphacyclotetra- decin-7-yl]-1,9-dihydro-6H-purin-6-one (Diastereomer 1)::US11453697, Example 147::US11453697, Example 148	Stimulator of interferon genes protein [H232R]					 1932					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=573962	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=573962&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177534	474496296							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1210992	Nc1nc2n(cnc2c(=O)[nH]1)[C@@H]1O[C@H]2C[C@H]1OP(S)(=O)OC[C@H]1O[C@H](C[C@@H]1OP(S)(=O)OC2)c1cnc2c(N)ncnn12			573964	2-amino-9-[(5S,7R,8R,12aR,14R,15aS)-14-(4- aminoimidazo[2,1-f][1,2,4]triazin-7-yl)-2,10- dioxido-2,10-disulfanyloctahydro-12H-5,8- methanofuro[3,2-l][1,3,6,9,11,2,10] pentaoxadiphosphacyclotetradecin-7-yl]-1,9- dihydro-6H-purin-6-one (Diastereomer 1)::US11453697, Example 149::US11453697, Example 150::US11453697, Example 152	Stimulator of interferon genes protein [H232R]					 111					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=573964	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=573964&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177535	474496297							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1210993	Nc1nc2n(cnc2c(=O)[nH]1)[C@@H]1O[C@H]2C[C@H]1OP(S)(=O)OC[C@H]1O[C@H](C[C@@H]1OP(S)(=O)OC2)c1cnc2c(N)ncnn12			573964	2-amino-9-[(5S,7R,8R,12aR,14R,15aS)-14-(4- aminoimidazo[2,1-f][1,2,4]triazin-7-yl)-2,10- dioxido-2,10-disulfanyloctahydro-12H-5,8- methanofuro[3,2-l][1,3,6,9,11,2,10] pentaoxadiphosphacyclotetradecin-7-yl]-1,9- dihydro-6H-purin-6-one (Diastereomer 1)::US11453697, Example 149::US11453697, Example 150::US11453697, Example 152	Stimulator of interferon genes protein [H232R]					 5.70					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=573964	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=573964&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177535	474496297							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1210994	Nc1nc2n(cnc2c(=O)[nH]1)[C@@H]1S[C@@H]2COP(S)(=O)O[C@@H]3[C@@H](COP(S)(=O)O[C@@H]1[C@H]2F)O[C@H]([C@H]3F)n1cnc2c(N)ncnc12			574028	(5R,7R,8R,12aR,14R,15S,15aR,16R)-7-(2- amino-6-oxo-1,6-dihydro-9H-purin-9-yl)-14-(6- amino-9H-purin-9-yl)-15,16-difluorooctahydro- 12H-5,8-methanofuro[3,2- l][1,3,9,11,6,2,10]tetraoxathiadiphosphacyclotetra- decine-2,10-bis(thiolate) 2,10-dioxide (Diastereomer 1)::US11453697, Example 153::US11453697, Example 154	Stimulator of interferon genes protein [H232R]					 6.50					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574028	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574028&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177578	474496341							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1210995	Nc1nc2n(cnc2c(=O)[nH]1)[C@@H]1S[C@@H]2COP(S)(=O)O[C@@H]3[C@@H](COP(S)(=O)O[C@@H]1[C@H]2F)O[C@H]([C@H]3F)n1cnc2c(N)ncnc12			574028	(5R,7R,8R,12aR,14R,15S,15aR,16R)-7-(2- amino-6-oxo-1,6-dihydro-9H-purin-9-yl)-14-(6- amino-9H-purin-9-yl)-15,16-difluorooctahydro- 12H-5,8-methanofuro[3,2- l][1,3,9,11,6,2,10]tetraoxathiadiphosphacyclotetra- decine-2,10-bis(thiolate) 2,10-dioxide (Diastereomer 1)::US11453697, Example 153::US11453697, Example 154	Stimulator of interferon genes protein [H232R]					 60.0					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574028	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574028&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177578	474496341							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1210996	Nc1nc2n(cnc2c(=O)[nH]1)[C@@H]1O[C@@H]2COP(O)(=S)O[C@@H]3[C@@H](COP(O)(=S)O[C@@H]1C2(F)F)O[C@H]([C@H]3F)n1cnc2c(N)ncnc12			574030	2-amino-9-[(5R,7R,8S,12aR,14R,15S,15aR)-14- (6-amino-9H-purin-9-yl)-15,16,16-trifluoro- 2,10-dihydroxy-2,10-disulfidooctahydro-12H- 5,8-methanofuro[3,2- l][1,3,6,9,11,2,10]pentaoxadiphosphacyclotetra- decin-7-yl]-1,9-dihydro-6H-purin-6-one (Diastereomer 1)::US11453697, Example 155::US11453697, Example 156	Stimulator of interferon genes protein [H232R]					<1.000					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574030	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574030&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177579	474496342							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1210997	Nc1nc2n(cnc2c(=O)[nH]1)[C@@H]1O[C@@H]2COP(O)(=S)O[C@@H]3[C@@H](COP(O)(=S)O[C@@H]1C2(F)F)O[C@H]([C@H]3F)n1cnc2c(N)ncnc12			574030	2-amino-9-[(5R,7R,8S,12aR,14R,15S,15aR)-14- (6-amino-9H-purin-9-yl)-15,16,16-trifluoro- 2,10-dihydroxy-2,10-disulfidooctahydro-12H- 5,8-methanofuro[3,2- l][1,3,6,9,11,2,10]pentaoxadiphosphacyclotetra- decin-7-yl]-1,9-dihydro-6H-purin-6-one (Diastereomer 1)::US11453697, Example 155::US11453697, Example 156	Stimulator of interferon genes protein [H232R]					<1.000					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574030	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574030&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177579	474496342							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1210998	Nc1nc2n(cnc2c(=O)[nH]1)[C@@H]1O[C@@H]2COP(O)(=S)O[C@H]3[C@H]4OCC3(COP(O)(=S)O[C@@H]1C2(F)F)O[C@H]4n1cnc2c(N)ncnc12			574032	2-amino-9-[(5R,7R,8S,12aR,14R,15R,15aS)-14- (6-amino-9H-purin-9-yl)-18,18-difluoro-2,10- dihydroxy-2,10-disulfidohexahydro-14H-15,12a- (epoxymethano)-5,8-methanofuro[3,2- l][1,3,6,9,11,2,10] pentaoxadiphosphacyclotetra- decin-7(12H)-yl]-1,9-dihydro-6H-purin-6-one (Diastereomer 1)::US11453697, Example 157::US11453697, Example 159::US11453697, Example 160	Stimulator of interferon genes protein [H232R]					<1.000					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574032	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574032&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177580	474496343							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1210999	Nc1nc(O)c2ncn([C@@H]3O[C@@H]4COP(O)(=S)O[C@H]5[C@H]6OCC5(COP(O)(=S)O[C@@H]3C4(F)F)O[C@H]6n3cnc4c(N)ncnc34)c2n1	InChI=1S/C21H22F2N10O10P2S2/c22-21(23)7-1-38-44(35,46)42-11-10-17(32-5-28-8-13(24)26-4-27-14(8)32)41-20(11,2-37-10)3-39-45(36,47)43-12(21)18(40-7)33-6-29-9-15(33)30-19(25)31-16(9)34/h4-7,10-12,17-18H,1-3H2,(H,35,46)(H,36,47)(H2,24,26,27)(H3,25,30,31,34)/t7-,10-,11+,12+,17-,18-,20?,44?,45?/m1/s1	FAPHJTDZMJNZHV-BSQGMMHLSA-N	574033	2-amino-9-[(5R,7R,8S,12aR,14R,15R,15aS)-14- (6-amino-9H-purin-9-yl)-18,18-difluoro-2,10- dihydroxy-2,10-disulfidohexahydro-14H-15,12a- (epoxymethano)-5,8-methanofuro[3,2- l][1,3,6,9,11,2,10]pentaoxadiphosphacyclotetra- decin-7(12H)-yl]-1,9-dihydro-6H-purin-6-one (Diastereomer 2)::US11453697, Example 158	Stimulator of interferon genes protein [H232R]					 40.0					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574033	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574033&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177581	474496344							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1211000	Nc1nc2n(cnc2c(=O)[nH]1)[C@@H]1O[C@@H]2COP(O)(=S)O[C@H]3[C@H]4OCC3(COP(O)(=S)O[C@@H]1C2(F)F)O[C@H]4n1cnc2c(N)ncnc12			574032	2-amino-9-[(5R,7R,8S,12aR,14R,15R,15aS)-14- (6-amino-9H-purin-9-yl)-18,18-difluoro-2,10- dihydroxy-2,10-disulfidohexahydro-14H-15,12a- (epoxymethano)-5,8-methanofuro[3,2- l][1,3,6,9,11,2,10] pentaoxadiphosphacyclotetra- decin-7(12H)-yl]-1,9-dihydro-6H-purin-6-one (Diastereomer 1)::US11453697, Example 157::US11453697, Example 159::US11453697, Example 160	Stimulator of interferon genes protein [H232R]					 7.10					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574032	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574032&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177580	474496343							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1211001	Nc1nc2n(cnc2c(=O)[nH]1)[C@@H]1O[C@@H]2COP(O)(=S)O[C@H]3[C@H]4OCC3(COP(O)(=S)O[C@@H]1C2(F)F)O[C@H]4n1cnc2c(N)ncnc12			574032	2-amino-9-[(5R,7R,8S,12aR,14R,15R,15aS)-14- (6-amino-9H-purin-9-yl)-18,18-difluoro-2,10- dihydroxy-2,10-disulfidohexahydro-14H-15,12a- (epoxymethano)-5,8-methanofuro[3,2- l][1,3,6,9,11,2,10] pentaoxadiphosphacyclotetra- decin-7(12H)-yl]-1,9-dihydro-6H-purin-6-one (Diastereomer 1)::US11453697, Example 157::US11453697, Example 159::US11453697, Example 160	Stimulator of interferon genes protein [H232R]					 10.3					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574032	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574032&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177580	474496343							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1211002	Nc1nc2n(cnc2c(=O)[nH]1)[C@@H]1O[C@@H]2COP(O)(=S)O[C@H]3C[C@@H](O[C@@H]3COP(O)(=S)O[C@@H]1[C@@H]2F)n1ccc2c(N)ncnc12			574036	2-amino-9-[(5R,7R,8S,12aR,14R,15aS,16R)-14- (4-amino-7H-pyrrolo[2,3-d]pyrimidin-7-yl)-16- fluoro-2,10-dihydroxy-2,10-disulfidooctahydro- 12H-5,8-methanofuro[3,2- l][1,3,6, 9,11,2,10]pentaoxadiphosphacyclotetra- decin-7-yl]-1,9-dihydro-6H-purin-6-one (Diastereomer 1)::US11453697, Example 161::US11453697, Example 162::US11453697, Example 163::US11453697, Example 164	Stimulator of interferon genes protein [H232R]					 6.20					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574036	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574036&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177582	474496345							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1211003	Nc1nc2n(cnc2c(=O)[nH]1)[C@@H]1O[C@@H]2COP(O)(=S)O[C@H]3C[C@@H](O[C@@H]3COP(O)(=S)O[C@@H]1[C@@H]2F)n1ccc2c(N)ncnc12			574036	2-amino-9-[(5R,7R,8S,12aR,14R,15aS,16R)-14- (4-amino-7H-pyrrolo[2,3-d]pyrimidin-7-yl)-16- fluoro-2,10-dihydroxy-2,10-disulfidooctahydro- 12H-5,8-methanofuro[3,2- l][1,3,6, 9,11,2,10]pentaoxadiphosphacyclotetra- decin-7-yl]-1,9-dihydro-6H-purin-6-one (Diastereomer 1)::US11453697, Example 161::US11453697, Example 162::US11453697, Example 163::US11453697, Example 164	Stimulator of interferon genes protein [H232R]					 101					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574036	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574036&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177582	474496345							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1211004	Nc1nc2n(cnc2c(=O)[nH]1)[C@@H]1O[C@@H]2COP(O)(=S)O[C@H]3C[C@@H](O[C@@H]3COP(O)(=S)O[C@@H]1[C@@H]2F)n1ccc2c(N)ncnc12			574036	2-amino-9-[(5R,7R,8S,12aR,14R,15aS,16R)-14- (4-amino-7H-pyrrolo[2,3-d]pyrimidin-7-yl)-16- fluoro-2,10-dihydroxy-2,10-disulfidooctahydro- 12H-5,8-methanofuro[3,2- l][1,3,6, 9,11,2,10]pentaoxadiphosphacyclotetra- decin-7-yl]-1,9-dihydro-6H-purin-6-one (Diastereomer 1)::US11453697, Example 161::US11453697, Example 162::US11453697, Example 163::US11453697, Example 164	Stimulator of interferon genes protein [H232R]					 14.3					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574036	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574036&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177582	474496345							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1211005	Nc1nc2n(cnc2c(=O)[nH]1)[C@@H]1O[C@@H]2COP(O)(=S)O[C@H]3C[C@@H](O[C@@H]3COP(O)(=S)O[C@@H]1[C@@H]2F)n1ccc2c(N)ncnc12			574036	2-amino-9-[(5R,7R,8S,12aR,14R,15aS,16R)-14- (4-amino-7H-pyrrolo[2,3-d]pyrimidin-7-yl)-16- fluoro-2,10-dihydroxy-2,10-disulfidooctahydro- 12H-5,8-methanofuro[3,2- l][1,3,6, 9,11,2,10]pentaoxadiphosphacyclotetra- decin-7-yl]-1,9-dihydro-6H-purin-6-one (Diastereomer 1)::US11453697, Example 161::US11453697, Example 162::US11453697, Example 163::US11453697, Example 164	Stimulator of interferon genes protein [H232R]					 312					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574036	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574036&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177582	474496345							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1211006	Nc1nc2n(cnc2c(=O)[nH]1)[C@@H]1O[C@@H]2COP(O)(=S)O[C@@H]3[C@@H](COP(O)(=S)O[C@@H]1[C@@H]2F)O[C@@H](n1nnc2c(N)ncnc12)C3(F)F			574040	2-amino-9-[(5R,7R,8S,12aR,14R,15aR,16R)-14- (7-amino-3H-[1,2,3]triazolo[4,5-d]pyrimidin-3- yl)-15,15,16-trifluoro-2,10-dihydroxy-2,10- disulfidooctahydro-12H-5,8-methanofuro[3,2- l][1,3,6,9,11,2,10]pentaoxadiphosphacyclotetra- decin-7-yl]-1,9-dihydro-6H-purin-6-one (Diastereomer 1)::US11453697, Example 165::US11453697, Example 166::US11453697, Example 167	Stimulator of interferon genes protein [H232R]					 2.90					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574040	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574040&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177583	474496346							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1211007	Nc1nc2n(cnc2c(=O)[nH]1)[C@@H]1O[C@@H]2COP(O)(=S)O[C@@H]3[C@@H](COP(O)(=S)O[C@@H]1[C@@H]2F)O[C@@H](n1nnc2c(N)ncnc12)C3(F)F			574040	2-amino-9-[(5R,7R,8S,12aR,14R,15aR,16R)-14- (7-amino-3H-[1,2,3]triazolo[4,5-d]pyrimidin-3- yl)-15,15,16-trifluoro-2,10-dihydroxy-2,10- disulfidooctahydro-12H-5,8-methanofuro[3,2- l][1,3,6,9,11,2,10]pentaoxadiphosphacyclotetra- decin-7-yl]-1,9-dihydro-6H-purin-6-one (Diastereomer 1)::US11453697, Example 165::US11453697, Example 166::US11453697, Example 167	Stimulator of interferon genes protein [H232R]					 463					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574040	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574040&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177583	474496346							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1211008	Nc1nc2n(cnc2c(=O)[nH]1)[C@@H]1O[C@@H]2COP(O)(=S)O[C@@H]3[C@@H](COP(O)(=S)O[C@@H]1[C@@H]2F)O[C@@H](n1nnc2c(N)ncnc12)C3(F)F			574040	2-amino-9-[(5R,7R,8S,12aR,14R,15aR,16R)-14- (7-amino-3H-[1,2,3]triazolo[4,5-d]pyrimidin-3- yl)-15,15,16-trifluoro-2,10-dihydroxy-2,10- disulfidooctahydro-12H-5,8-methanofuro[3,2- l][1,3,6,9,11,2,10]pentaoxadiphosphacyclotetra- decin-7-yl]-1,9-dihydro-6H-purin-6-one (Diastereomer 1)::US11453697, Example 165::US11453697, Example 166::US11453697, Example 167	Stimulator of interferon genes protein [H232R]					 87.7					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574040	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574040&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177583	474496346							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1211009	Nc1nc2n(cnc2c(=O)[nH]1)[C@@H]1O[C@@H]2COP(O)(=S)O[C@@H]3[C@@H](COP(O)(=S)O[C@@H]1[C@@H]2F)O[C@H]([C@H]3F)n1ccc2c(N)ncnc12			574043	2-amino-9- [(5R,7R,8S,12aR,14R,15S,15aR,16R)-14-(4- amino-7H-pyrrolo[2,3-d]pyrimidin-7-yl)-15,16- difluoro-2,10-dihydroxy-2,10- disulfidooctahydro-12H-5,8-methanofuro[3,2- l][1,3,6,9,11,2,10]pentaoxadiphosphacyclotetra- decin-7-yl]-1,9-dihydro-6H-purin-6-one (Diastereomer 1)::US11453697, Example 168::US11453697, Example 169::US11453697, Example 170	Stimulator of interferon genes protein [H232R]					 8.60					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574043	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574043&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177584	474496347							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1211010	Nc1nc2n(cnc2c(=O)[nH]1)[C@@H]1O[C@@H]2COP(O)(=S)O[C@@H]3[C@@H](COP(O)(=S)O[C@@H]1[C@@H]2F)O[C@H]([C@H]3F)n1ccc2c(N)ncnc12			574043	2-amino-9- [(5R,7R,8S,12aR,14R,15S,15aR,16R)-14-(4- amino-7H-pyrrolo[2,3-d]pyrimidin-7-yl)-15,16- difluoro-2,10-dihydroxy-2,10- disulfidooctahydro-12H-5,8-methanofuro[3,2- l][1,3,6,9,11,2,10]pentaoxadiphosphacyclotetra- decin-7-yl]-1,9-dihydro-6H-purin-6-one (Diastereomer 1)::US11453697, Example 168::US11453697, Example 169::US11453697, Example 170	Stimulator of interferon genes protein [H232R]					 187					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574043	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574043&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177584	474496347							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1211011	Nc1nc2n(cnc2c(=O)[nH]1)[C@@H]1O[C@@H]2COP(O)(=S)O[C@@H]3[C@@H](COP(O)(=S)O[C@@H]1[C@@H]2F)O[C@H]([C@H]3F)n1ccc2c(N)ncnc12			574043	2-amino-9- [(5R,7R,8S,12aR,14R,15S,15aR,16R)-14-(4- amino-7H-pyrrolo[2,3-d]pyrimidin-7-yl)-15,16- difluoro-2,10-dihydroxy-2,10- disulfidooctahydro-12H-5,8-methanofuro[3,2- l][1,3,6,9,11,2,10]pentaoxadiphosphacyclotetra- decin-7-yl]-1,9-dihydro-6H-purin-6-one (Diastereomer 1)::US11453697, Example 168::US11453697, Example 169::US11453697, Example 170	Stimulator of interferon genes protein [H232R]					 25.5					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574043	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574043&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177584	474496347							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1211012	Nc1nc2n(cnc2c(=O)[nH]1)[C@@H]1O[C@H]2C[C@H]1O[P@@](S)(=O)OC[C@H]1O[C@H]([C@@H](F)[C@@H]1O[P@@](S)(=O)OC2)n1ccc2c(N)ncnc12			574046	2-amino-9-[(2R,5S,7R,8R,10R, 12aR,14R,15S,15aR)-14-(4-amino-7H- pyrrolo[2,3-d]pyrimidin-7-yl)-15-fluoro-2,10- dihydroxy-2,10-disulfidooctahydro-12H-5,8- methanofuro[3,2- l][1,3,6,9,11,2,10]pentaoxadiphosphacyclotetra- decin-7-yl]-1,9-dihydro-6H-purin-6-one (Diastereomer 1)::US11453697, Example 171	Stimulator of interferon genes protein [H232R]					 18.7					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574046	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574046&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177585	474496348							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1211013	Nc1nc2n(cnc2c(=O)[nH]1)[C@@H]1O[C@H]2C[C@H]1OP(O)(=S)OC[C@H]1O[C@H]([C@@H](F)[C@@H]1OP(O)(=S)OC2)n1ccc2c(N)ncnc12			574047	2-amino-9-[(5S,7R,8R,12aR,14R,15S,15aR)-14- (4-amino-7H-pyrrolo[2,3-d]pyrimidin-7-yl)-15- fluoro-2,10-dihydroxy-2,10-disulfidooctahydro- 12H-5,8-methanofuro[3,2- l][1,3,6,9,11,2,10]pentaoxadiphosphacyclotetra- decin-7-yl]-1,9-dihydro-6H-purin-6-one (Diastereomer 2)::US11453697, Example 172	Stimulator of interferon genes protein [H232R]					 106					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574047	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574047&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177586	474496349							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1211014	Nc1nc2n(nnc2c(=O)[nH]1)[C@@H]1O[C@H]2C[C@H]1OP(O)(=S)OC[C@H]1O[C@H]([C@@H](F)[C@@H]1OP(O)(=S)OC2)n1cnc2c(N)ncnc12			574048	5-amino-3-[(5S,7R,8R,12aR,14R,15S,15aR)-14- (6-amino-9H-purin-9-yl)-15-fluoro-2,10- dihydroxy-2,10-disulfidooctahydro-12H-5,8- methanofuro[3,2- l][1,3,6,9,11,2,10]pentaoxadiphosphacyclotetra- decin-7-yl]-3,6-dihydro-7H-[1,2,3]triazolo[4,5- d]pyrimidin-7-one (Diastereomer 2)::US11453697, Example 176	Stimulator of interferon genes protein [H232R]					 16.2					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574048	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574048&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177587	474496350							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1211015	Nc1nc2n(nnc2c(=O)[nH]1)[C@@H]1O[C@@H]2COP(O)(=S)O[C@@H]3[C@@H](COP(O)(=S)O[C@@H]1[C@H]2F)O[C@H]([C@H]3F)n1cnc2c(N)ncnc12			574049	5-amino-3- [(5R,7R,8S,12aR,14R,15S,15aR,16S)-14-(6- amino-9H-purin-9-yl)-15,16-difluoro-2,10- dihydroxy-2,10-disulfidooctahydro-12H-5,8- methanofuro[3,2- l][1,3,6,9,11,2,10]pentaoxadiphosphacyclotetra- decin-7-yl]-3,6-dihydro-7H-[1,2,3]triazolo[4,5- d]pyrimidin-7-one (Diastereomer 1)::US11453697, Example 177::US11453697, Example 178::US11453697, Example 179	Stimulator of interferon genes protein [H232R]					 7.90					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574049	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574049&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177588	474496351							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1211016	Nc1nc2n(nnc2c(=O)[nH]1)[C@@H]1O[C@@H]2COP(O)(=S)O[C@@H]3[C@@H](COP(O)(=S)O[C@@H]1[C@H]2F)O[C@H]([C@H]3F)n1cnc2c(N)ncnc12			574049	5-amino-3- [(5R,7R,8S,12aR,14R,15S,15aR,16S)-14-(6- amino-9H-purin-9-yl)-15,16-difluoro-2,10- dihydroxy-2,10-disulfidooctahydro-12H-5,8- methanofuro[3,2- l][1,3,6,9,11,2,10]pentaoxadiphosphacyclotetra- decin-7-yl]-3,6-dihydro-7H-[1,2,3]triazolo[4,5- d]pyrimidin-7-one (Diastereomer 1)::US11453697, Example 177::US11453697, Example 178::US11453697, Example 179	Stimulator of interferon genes protein [H232R]					 37.4					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574049	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574049&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177588	474496351							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1211017	Nc1nc2n(nnc2c(=O)[nH]1)[C@@H]1O[C@@H]2COP(O)(=S)O[C@@H]3[C@@H](COP(O)(=S)O[C@@H]1[C@H]2F)O[C@H]([C@H]3F)n1cnc2c(N)ncnc12			574049	5-amino-3- [(5R,7R,8S,12aR,14R,15S,15aR,16S)-14-(6- amino-9H-purin-9-yl)-15,16-difluoro-2,10- dihydroxy-2,10-disulfidooctahydro-12H-5,8- methanofuro[3,2- l][1,3,6,9,11,2,10]pentaoxadiphosphacyclotetra- decin-7-yl]-3,6-dihydro-7H-[1,2,3]triazolo[4,5- d]pyrimidin-7-one (Diastereomer 1)::US11453697, Example 177::US11453697, Example 178::US11453697, Example 179	Stimulator of interferon genes protein [H232R]					 112					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574049	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574049&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177588	474496351							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1211018	Nc1ncnc2n(cnc12)[C@@H]1O[C@@H]2COP(O)(=S)O[C@@H]3[C@@H](F)[C@@H](COP(O)(=S)O[C@H]2[C@@H]1F)O[C@H]3n1cnc2c1cc[nH]c2=O			574052	1-[(5R,7R,8S,12aR,14R,15S,15aR,16S)-14-(6- amino-9H-purin-9-yl)-15,16-difluoro-2,10- dihydroxy-2,10-disulfidooctahydro-12H-5,8- methanofuro[3,2- l][1,3,6,9,11,2,10]pentaoxadiphosphacyclotetra- decin-7-yl]-1,5-dihydro-4H-imidazo[4,5- c]pyridin-4-one::US11453697, Example 180	Stimulator of interferon genes protein [H232R]					 832					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574052	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574052&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177589	474496352							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1211019	Nc1nc2n(nnc2c(=O)[nH]1)[C@@H]1O[C@H]2C[C@H]1OP(O)(=S)OC[C@H]1O[C@H]([C@@H](F)[C@@H]1OP(O)(=S)OC2)n1nnc2c(N)ncnc12			574053	5-amino-3-[(5S,7R,8R,12aR,14R,15S,15aR)-14- (7-amino-3H-[1,2,3]triazolo[4,5-d]pyrimidin-3- yl)-15-fluoro-2,10-dihydroxy-2,10- disulfidooctahydro-12H-5,8-methanofuro[3,2- l][1,3,6,9,11,2,10]pentaoxadiphosphacyclotetra- decin-7-yl]-3,6-dihydro-7H-[1,2,3]triazolo[4,5- d]pyrimidin-7-one (Diastereomer 1)::US11453697, Example 181::US11453697, Example 182::US11453697, Example 183	Stimulator of interferon genes protein [H232R]					 459					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574053	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574053&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177590	474496353							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1211020	Nc1nc2n(nnc2c(=O)[nH]1)[C@@H]1O[C@H]2C[C@H]1OP(O)(=S)OC[C@H]1O[C@H]([C@@H](F)[C@@H]1OP(O)(=S)OC2)n1nnc2c(N)ncnc12			574053	5-amino-3-[(5S,7R,8R,12aR,14R,15S,15aR)-14- (7-amino-3H-[1,2,3]triazolo[4,5-d]pyrimidin-3- yl)-15-fluoro-2,10-dihydroxy-2,10- disulfidooctahydro-12H-5,8-methanofuro[3,2- l][1,3,6,9,11,2,10]pentaoxadiphosphacyclotetra- decin-7-yl]-3,6-dihydro-7H-[1,2,3]triazolo[4,5- d]pyrimidin-7-one (Diastereomer 1)::US11453697, Example 181::US11453697, Example 182::US11453697, Example 183	Stimulator of interferon genes protein [H232R]					 3276					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574053	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574053&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177590	474496353							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1211021	Nc1nc2n(nnc2c(=O)[nH]1)[C@@H]1O[C@H]2C[C@H]1OP(O)(=S)OC[C@H]1O[C@H]([C@@H](F)[C@@H]1OP(O)(=S)OC2)n1nnc2c(N)ncnc12			574053	5-amino-3-[(5S,7R,8R,12aR,14R,15S,15aR)-14- (7-amino-3H-[1,2,3]triazolo[4,5-d]pyrimidin-3- yl)-15-fluoro-2,10-dihydroxy-2,10- disulfidooctahydro-12H-5,8-methanofuro[3,2- l][1,3,6,9,11,2,10]pentaoxadiphosphacyclotetra- decin-7-yl]-3,6-dihydro-7H-[1,2,3]triazolo[4,5- d]pyrimidin-7-one (Diastereomer 1)::US11453697, Example 181::US11453697, Example 182::US11453697, Example 183	Stimulator of interferon genes protein [H232R]					 3180					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574053	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574053&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177590	474496353							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1211022	Nc1nc2n(nnc2c(=O)[nH]1)[C@@H]1O[C@H]2C[C@H]1OP(O)(=S)OC[C@@]13CO[C@@H]([C@@H](O1)n1cnc4c(N)ncnc14)[C@@H]3OP(O)(=S)OC2			574056	5-amino-3-[(5S,7R,8R,12aR,14R,15R,15aS)-14- (6-amino-9H-purin-9-yl)-2,10-dihydroxy-2,10- disulfidohexahydro-14H-15,12a- (epoxymethano)-5,8-methanofuro[3,2- l][1,3,6,9,11,2,10]pentaoxadiphosphacyclotetra- decin-7(12H)-yl]-3,6-dihydro-7H- [1,2,3]triazolo[4,5-d]pyrimidin-7-one (Diastereomer 1)::US11453697, Example 184::US11453697, Example 185::US11453697, Example 186::US11453697, Example 187	Stimulator of interferon genes protein [H232R]					<1.000					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574056	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574056&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177591	474496354							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1211023	Nc1nc2n(nnc2c(=O)[nH]1)[C@@H]1O[C@H]2C[C@H]1OP(O)(=S)OC[C@@]13CO[C@@H]([C@@H](O1)n1cnc4c(N)ncnc14)[C@@H]3OP(O)(=S)OC2			574056	5-amino-3-[(5S,7R,8R,12aR,14R,15R,15aS)-14- (6-amino-9H-purin-9-yl)-2,10-dihydroxy-2,10- disulfidohexahydro-14H-15,12a- (epoxymethano)-5,8-methanofuro[3,2- l][1,3,6,9,11,2,10]pentaoxadiphosphacyclotetra- decin-7(12H)-yl]-3,6-dihydro-7H- [1,2,3]triazolo[4,5-d]pyrimidin-7-one (Diastereomer 1)::US11453697, Example 184::US11453697, Example 185::US11453697, Example 186::US11453697, Example 187	Stimulator of interferon genes protein [H232R]					 201					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574056	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574056&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177591	474496354							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1211024	Nc1nc2n(nnc2c(=O)[nH]1)[C@@H]1O[C@H]2C[C@H]1OP(O)(=S)OC[C@@]13CO[C@@H]([C@@H](O1)n1cnc4c(N)ncnc14)[C@@H]3OP(O)(=S)OC2			574056	5-amino-3-[(5S,7R,8R,12aR,14R,15R,15aS)-14- (6-amino-9H-purin-9-yl)-2,10-dihydroxy-2,10- disulfidohexahydro-14H-15,12a- (epoxymethano)-5,8-methanofuro[3,2- l][1,3,6,9,11,2,10]pentaoxadiphosphacyclotetra- decin-7(12H)-yl]-3,6-dihydro-7H- [1,2,3]triazolo[4,5-d]pyrimidin-7-one (Diastereomer 1)::US11453697, Example 184::US11453697, Example 185::US11453697, Example 186::US11453697, Example 187	Stimulator of interferon genes protein [H232R]					 30.2					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574056	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574056&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177591	474496354							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1211025	Nc1nc2n(nnc2c(=O)[nH]1)[C@@H]1O[C@H]2C[C@H]1OP(O)(=S)OC[C@@]13CO[C@@H]([C@@H](O1)n1cnc4c(N)ncnc14)[C@@H]3OP(O)(=S)OC2			574056	5-amino-3-[(5S,7R,8R,12aR,14R,15R,15aS)-14- (6-amino-9H-purin-9-yl)-2,10-dihydroxy-2,10- disulfidohexahydro-14H-15,12a- (epoxymethano)-5,8-methanofuro[3,2- l][1,3,6,9,11,2,10]pentaoxadiphosphacyclotetra- decin-7(12H)-yl]-3,6-dihydro-7H- [1,2,3]triazolo[4,5-d]pyrimidin-7-one (Diastereomer 1)::US11453697, Example 184::US11453697, Example 185::US11453697, Example 186::US11453697, Example 187	Stimulator of interferon genes protein [H232R]					 6.50					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574056	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574056&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177591	474496354							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1211026	Nc1nc2n(nnc2c(=O)[nH]1)[C@@H]1O[C@H]2C[C@H]1OP(O)(=S)OC[C@H]1O[C@H](C[C@@H]1OP(O)(=S)OC2)n1ccc2c(N)ncnc12			574060	5-amino-3-[(5S,7R,8R,12aR,14R,15aS)-14-(4- amino-7H-pyrrolo[2,3-d]pyrimidin-7-yl)-2,10- dihydroxy-2,10-disulfidooctahydro-12H-5,8- methanofuro[3,2- l][1,3,6,9,11,2,10]pentaoxadiphosphacyclotetra- decin-7-yl]-3,6-dihydro-7H-[1,2,3]triazolo[4,5- d]pyrimidin-7-one (Diastereomer 1)::US11453697, Example 188::US11453697, Example 189::US11453697, Example 190	Stimulator of interferon genes protein [H232R]					 47.6					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574060	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574060&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177592	474496355							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1211027	Nc1nc2n(nnc2c(=O)[nH]1)[C@@H]1O[C@H]2C[C@H]1OP(O)(=S)OC[C@H]1O[C@H](C[C@@H]1OP(O)(=S)OC2)n1ccc2c(N)ncnc12			574060	5-amino-3-[(5S,7R,8R,12aR,14R,15aS)-14-(4- amino-7H-pyrrolo[2,3-d]pyrimidin-7-yl)-2,10- dihydroxy-2,10-disulfidooctahydro-12H-5,8- methanofuro[3,2- l][1,3,6,9,11,2,10]pentaoxadiphosphacyclotetra- decin-7-yl]-3,6-dihydro-7H-[1,2,3]triazolo[4,5- d]pyrimidin-7-one (Diastereomer 1)::US11453697, Example 188::US11453697, Example 189::US11453697, Example 190	Stimulator of interferon genes protein [H232R]					 424					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574060	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574060&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177592	474496355							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1211028	Nc1nc2n(nnc2c(=O)[nH]1)[C@@H]1O[C@H]2C[C@H]1OP(O)(=S)OC[C@H]1O[C@H](C[C@@H]1OP(O)(=S)OC2)n1ccc2c(N)ncnc12			574060	5-amino-3-[(5S,7R,8R,12aR,14R,15aS)-14-(4- amino-7H-pyrrolo[2,3-d]pyrimidin-7-yl)-2,10- dihydroxy-2,10-disulfidooctahydro-12H-5,8- methanofuro[3,2- l][1,3,6,9,11,2,10]pentaoxadiphosphacyclotetra- decin-7-yl]-3,6-dihydro-7H-[1,2,3]triazolo[4,5- d]pyrimidin-7-one (Diastereomer 1)::US11453697, Example 188::US11453697, Example 189::US11453697, Example 190	Stimulator of interferon genes protein [H232R]					 409					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574060	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574060&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177592	474496355							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1211029	Nc1nc2n(cnc2c(=O)[nH]1)[C@@H]1S[C@H]2C[C@H]1OP(O)(=S)OC[C@H]1O[C@H]([C@@H](F)[C@@H]1OP(O)(=S)OC2)n1nnc2c(N)ncnc12			574063	2-amino-9-[(5S,7R,8R,12aR,14R,15S,15aR)-14- (7-amino-3H-[1,2,3]triazolo[4,5-d]pyrimidin-3- yl)-15-fluoro-2,10-dihydroxy-2,10- disulfidooctahydro-12H-5,8-methanofuro[3,2- l][1,3,9,11,6,2,10]tetraoxathiadiphosphacyclotetra- decin-7-yl]-1,9-dihydro-6H-purin-6-one (Diastereomer 1)::US11453697, Example 191::US11453697, Example 192	Stimulator of interferon genes protein [H232R]					 281					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574063	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574063&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177593	474496356							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1211030	Nc1nc2n(cnc2c(=O)[nH]1)[C@@H]1S[C@H]2C[C@H]1OP(O)(=S)OC[C@H]1O[C@H]([C@@H](F)[C@@H]1OP(O)(=S)OC2)n1nnc2c(N)ncnc12			574063	2-amino-9-[(5S,7R,8R,12aR,14R,15S,15aR)-14- (7-amino-3H-[1,2,3]triazolo[4,5-d]pyrimidin-3- yl)-15-fluoro-2,10-dihydroxy-2,10- disulfidooctahydro-12H-5,8-methanofuro[3,2- l][1,3,9,11,6,2,10]tetraoxathiadiphosphacyclotetra- decin-7-yl]-1,9-dihydro-6H-purin-6-one (Diastereomer 1)::US11453697, Example 191::US11453697, Example 192	Stimulator of interferon genes protein [H232R]					 3867					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574063	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574063&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177593	474496356							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1211031	Nc1nc2n(cnc2c(=O)[nH]1)[C@@H]1S[C@H]2C[C@H]1OP(O)(=S)OC[C@H]1O[C@H]([C@@H](F)[C@@H]1OP(O)(=S)OC2)n1ccc2c(N)ncnc12			574065	2-amino-9-[(5S,7R,8R,12aR,14R,15S,15aR)-14- (4-amino-7H-pyrrolo[2,3-d]pyrimidin-7-yl)-15- fluoro-2,10-dihydroxy-2,10-disulfidooctahydro- 12H-5,8-methanofuro[3,2- l][1,3,9,11,6,2,10]tetraoxathiadiphosphacyclotetra- decin-7-yl]-1,9-dihydro-6H-purin-6-one::US11453697, Example 193	Stimulator of interferon genes protein [H232R]					 190					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574065	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574065&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177594	474496357							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1211032	Nc1nc2n(nnc2c(=O)[nH]1)[C@@H]1O[C@H]2C[C@H]1OP(O)(=S)OC[C@H]1O[C@H]([C@@H](F)[C@@H]1OP(O)(=S)OC2)n1ccc2c(N)ncnc12			574066	5-amino-3-[(5S,7R,8R,12aR,14R,15S,15aR)-14- (4-amino-7H-pyrrolo[2,3-d]pyrimidin-7-yl)-15- fluoro-2,10-dihydroxy-2,10-disulfidooctahydro- 12H-5,8-methanofuro[3,2- l][1,3,6,9,11,2,10]pentaoxadiphosphacyclotetra- decin-7-yl]-3,6-dihydro-7H-[1,2,3]triazolo[4,5- d]pyrimidin-7-one (Diastereomer 1)::US11453697, Example 194::US11453697, Example 195::US11453697, Example 196	Stimulator of interferon genes protein [H232R]					 159					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574066	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574066&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177595	474496358							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1211033	Nc1nc2n(nnc2c(=O)[nH]1)[C@@H]1O[C@H]2C[C@H]1OP(O)(=S)OC[C@H]1O[C@H]([C@@H](F)[C@@H]1OP(O)(=S)OC2)n1ccc2c(N)ncnc12			574066	5-amino-3-[(5S,7R,8R,12aR,14R,15S,15aR)-14- (4-amino-7H-pyrrolo[2,3-d]pyrimidin-7-yl)-15- fluoro-2,10-dihydroxy-2,10-disulfidooctahydro- 12H-5,8-methanofuro[3,2- l][1,3,6,9,11,2,10]pentaoxadiphosphacyclotetra- decin-7-yl]-3,6-dihydro-7H-[1,2,3]triazolo[4,5- d]pyrimidin-7-one (Diastereomer 1)::US11453697, Example 194::US11453697, Example 195::US11453697, Example 196	Stimulator of interferon genes protein [H232R]					 1855					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574066	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574066&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177595	474496358							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1211034	Nc1nc2n(nnc2c(=O)[nH]1)[C@@H]1O[C@H]2C[C@H]1OP(O)(=S)OC[C@H]1O[C@H]([C@@H](F)[C@@H]1OP(O)(=S)OC2)n1ccc2c(N)ncnc12			574066	5-amino-3-[(5S,7R,8R,12aR,14R,15S,15aR)-14- (4-amino-7H-pyrrolo[2,3-d]pyrimidin-7-yl)-15- fluoro-2,10-dihydroxy-2,10-disulfidooctahydro- 12H-5,8-methanofuro[3,2- l][1,3,6,9,11,2,10]pentaoxadiphosphacyclotetra- decin-7-yl]-3,6-dihydro-7H-[1,2,3]triazolo[4,5- d]pyrimidin-7-one (Diastereomer 1)::US11453697, Example 194::US11453697, Example 195::US11453697, Example 196	Stimulator of interferon genes protein [H232R]					 1033					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574066	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574066&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177595	474496358							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1211035	Nc1nc2n(nnc2c(=O)[nH]1)[C@@H]1O[C@@H]2COP(O)(=S)O[C@@H]3[C@@H](COP(O)(=S)O[C@@H]1[C@@H]2F)O[C@H]([C@H]3F)n1cnc2c(N)ncnc12			574069	5-amino-3- [(5R,7R,8S,12aR,14R,15S,15aR,16R)-14-(6- amino-9H-purin-9-yl)-15,16-difluoro-2,10- dihydroxy-2,10-disulfidooctahydro-12H-5,8- methanofuro[3,2- l][1,3,6,9,11,2,10]pentaoxadiphosphacyclotetra- decin-7-yl]-3,6-dihydro-7H-[1,2,3]triazolo[4,5- d]pyrimidin-7-one (Diastereomer 1)::US11453697, Example 197::US11453697, Example 198::US11453697, Example 199	Stimulator of interferon genes protein [H232R]					 1.20					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574069	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574069&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177596	474496359							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1211036	Nc1nc2n(nnc2c(=O)[nH]1)[C@@H]1O[C@@H]2COP(O)(=S)O[C@@H]3[C@@H](COP(O)(=S)O[C@@H]1[C@@H]2F)O[C@H]([C@H]3F)n1cnc2c(N)ncnc12			574069	5-amino-3- [(5R,7R,8S,12aR,14R,15S,15aR,16R)-14-(6- amino-9H-purin-9-yl)-15,16-difluoro-2,10- dihydroxy-2,10-disulfidooctahydro-12H-5,8- methanofuro[3,2- l][1,3,6,9,11,2,10]pentaoxadiphosphacyclotetra- decin-7-yl]-3,6-dihydro-7H-[1,2,3]triazolo[4,5- d]pyrimidin-7-one (Diastereomer 1)::US11453697, Example 197::US11453697, Example 198::US11453697, Example 199	Stimulator of interferon genes protein [H232R]					 19.1					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574069	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574069&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177596	474496359							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1211037	Nc1nc2n(nnc2c(=O)[nH]1)[C@@H]1O[C@@H]2COP(O)(=S)O[C@@H]3[C@@H](COP(O)(=S)O[C@@H]1[C@@H]2F)O[C@H]([C@H]3F)n1cnc2c(N)ncnc12			574069	5-amino-3- [(5R,7R,8S,12aR,14R,15S,15aR,16R)-14-(6- amino-9H-purin-9-yl)-15,16-difluoro-2,10- dihydroxy-2,10-disulfidooctahydro-12H-5,8- methanofuro[3,2- l][1,3,6,9,11,2,10]pentaoxadiphosphacyclotetra- decin-7-yl]-3,6-dihydro-7H-[1,2,3]triazolo[4,5- d]pyrimidin-7-one (Diastereomer 1)::US11453697, Example 197::US11453697, Example 198::US11453697, Example 199	Stimulator of interferon genes protein [H232R]					 72.0					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574069	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574069&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177596	474496359							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1211038	Nc1nc2n(nnc2c(=O)[nH]1)[C@@H]1O[C@@H]2COP(O)(=S)O[C@@H]3[C@@H](COP(O)(=S)O[C@@H]1[C@@H]2F)O[C@H]([C@H]3F)n1nnc2c(N)ncnc12			574072	5-amino-3- [(5R,7R,8S,12aR,14R,15S,15aR,16R)-14-(7- amino-3H-[1,2,3]triazolo[4,5-d]pyrimidin-3-yl)- 15,16-difluoro-2,10-dihydroxy-2,10- disulfidooctahydro-12H-5,8-methanofuro[3,2- l][1,3,6,9,11,2,10]pentaoxadiphosphacyclotetra- decin-7-yl]-3,6-dihydro-7H-[1,2,3]triazolo[4,5- d]pyrimidin-7-one (Diastereomer 1)::US11453697, Example 200::US11453697, Example 201	Stimulator of interferon genes protein [H232R]					 15.0					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574072	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574072&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177597	474496360							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1211039	Nc1nc2n(nnc2c(=O)[nH]1)[C@@H]1O[C@@H]2COP(O)(=S)O[C@@H]3[C@@H](COP(O)(=S)O[C@@H]1[C@@H]2F)O[C@H]([C@H]3F)n1nnc2c(N)ncnc12			574072	5-amino-3- [(5R,7R,8S,12aR,14R,15S,15aR,16R)-14-(7- amino-3H-[1,2,3]triazolo[4,5-d]pyrimidin-3-yl)- 15,16-difluoro-2,10-dihydroxy-2,10- disulfidooctahydro-12H-5,8-methanofuro[3,2- l][1,3,6,9,11,2,10]pentaoxadiphosphacyclotetra- decin-7-yl]-3,6-dihydro-7H-[1,2,3]triazolo[4,5- d]pyrimidin-7-one (Diastereomer 1)::US11453697, Example 200::US11453697, Example 201	Stimulator of interferon genes protein [H232R]					 650					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574072	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574072&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177597	474496360							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1211040	Nc1nc2n(nnc2c(=O)[nH]1)[C@@H]1O[C@@H]2COP(O)(=S)O[C@@H]3[C@@H](COP(O)(=S)O[C@@H]1[C@H]2F)O[C@H]([C@H]3F)n1nnc2c(N)ncnc12			574074	5-amino-3- [(5R,7R,8S,12aR,14R,15S,15aR,16S)-14-(7- amino-3H-[1,2,3]triazolo[4,5-d]pyrimidin-3-yl)- 15,16-difluoro-2,10-dihydroxy-2,10- disulfidooctahydro-12H-5,8-methanofuro[3,2- l][1,3,6,9,11,2,10]pentaoxadiphosphacyclotetra- decin-7-yl]-3,6-dihydro-7H-[1,2,3]triazolo[4,5- d]pyrimidin-7-one::US11453697, Example 202	Stimulator of interferon genes protein [H232R]					 814					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574074	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574074&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177598	474496361							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1211041	Nc1nc2n(nnc2c(=O)[nH]1)[C@@H]1O[C@@H]2COP(S)(=O)O[C@H]3[C@H]4OCC3(COP(S)(=O)O[C@@H]1[C@H]2F)O[C@H]4n1cnc2c(N)ncnc12			574075	5-amino-3- [(5R,7R,8S,12aR,14R,15R,15aS,18S)-14-(6- amino-9H-purin-9-yl)-18-fluoro-2,10-dioxido- 2,10-disulfanylhexahydro-14H-15,12a- (epoxymethano)-5,8-methanofuro[3,2- l][1,3,6,9,11,2,10]pentaoxadiphosphacyclotetra- decin-7(12H)-yl]-3,6-dihydro-7H- [1,2,3]triazolo[4,5-d]pyrimidin-7-one (Diastereomer 1)::US11453697, Example 203::US11453697, Example 204::US11453697, Example 205	Stimulator of interferon genes protein [H232R]					 7.30					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574075	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574075&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177599	474496362							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1211042	Nc1nc2n(nnc2c(=O)[nH]1)[C@@H]1O[C@@H]2COP(S)(=O)O[C@H]3[C@H]4OCC3(COP(S)(=O)O[C@@H]1[C@H]2F)O[C@H]4n1cnc2c(N)ncnc12			574075	5-amino-3- [(5R,7R,8S,12aR,14R,15R,15aS,18S)-14-(6- amino-9H-purin-9-yl)-18-fluoro-2,10-dioxido- 2,10-disulfanylhexahydro-14H-15,12a- (epoxymethano)-5,8-methanofuro[3,2- l][1,3,6,9,11,2,10]pentaoxadiphosphacyclotetra- decin-7(12H)-yl]-3,6-dihydro-7H- [1,2,3]triazolo[4,5-d]pyrimidin-7-one (Diastereomer 1)::US11453697, Example 203::US11453697, Example 204::US11453697, Example 205	Stimulator of interferon genes protein [H232R]					 1233					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574075	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574075&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177599	474496362							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1211043	Nc1nc2n(nnc2c(=O)[nH]1)[C@@H]1O[C@@H]2COP(S)(=O)O[C@H]3[C@H]4OCC3(COP(S)(=O)O[C@@H]1[C@H]2F)O[C@H]4n1cnc2c(N)ncnc12			574075	5-amino-3- [(5R,7R,8S,12aR,14R,15R,15aS,18S)-14-(6- amino-9H-purin-9-yl)-18-fluoro-2,10-dioxido- 2,10-disulfanylhexahydro-14H-15,12a- (epoxymethano)-5,8-methanofuro[3,2- l][1,3,6,9,11,2,10]pentaoxadiphosphacyclotetra- decin-7(12H)-yl]-3,6-dihydro-7H- [1,2,3]triazolo[4,5-d]pyrimidin-7-one (Diastereomer 1)::US11453697, Example 203::US11453697, Example 204::US11453697, Example 205	Stimulator of interferon genes protein [H232R]					 42.7					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574075	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574075&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177599	474496362							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1211044	Nc1nc2n(nnc2c(=O)[nH]1)[C@@H]1O[C@@H]2COP([S-])(=O)O[C@@H]3[C@@H](COP([S-])(=O)O[C@@H]1[C@H]2F)O[C@H]([C@H]3F)n1ccc2c(N)ncnc12			574078	5-amino-3- [(5R,7R,8S,12aR,14R,15S,15aR,16S)-14-(4- amino-7H-pyrrolo[2,3-d]pyrimidin-7-yl)-15,16- difluoro-2,10-dioxido-2,10-disulfanyloctahydro- 12H-5,8-methanofuro[3,2- l][1,3,6,9,11,2,10]pentaoxadiphosphacyclotetra- decin-7-yl]-3,6-dihydro-7H-[1,2,3]triazolo[4,5- d]pyrimidin-7-one::US11453697, Example 206	Stimulator of interferon genes protein [H232R]					 260					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574078	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574078&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177600	474496363							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1211045	Nc1nc2n(nnc2c(=O)[nH]1)[C@@H]1O[C@@H]2COP(S)(=O)O[C@H]3C[C@@H](O[C@@]3(COP(S)(=O)O[C@@H]1[C@H]2F)C#C)n1cnc2c(N)ncnc12			574079	5-amino-3-[(5R,7R,8S,112aR,14R,15aS,16S)- 14-(6-amino-9H-purin-9-yl)-12a-ethynyl-16- fluoro-2,10-dioxido-2,10-disulfanyloctahydro- 12H-5,8-methanofuro[3,2- l][1,3,6,9,11,2,10]pentaoxadiphosphacyclotetra- decin-7-yl]-3,6-dihydro-7H-[1,2,3]triazolo[4,5- d]pyrimidin-7-one (Diastereomer 1)::US11453697, Example 207::US11453697, Example 208::US11453697, Example 209	Stimulator of interferon genes protein [H232R]					 1.40					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574079	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574079&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177602	474496364							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1211046	Nc1nc2n(nnc2c(=O)[nH]1)[C@@H]1O[C@@H]2COP(S)(=O)O[C@H]3C[C@@H](O[C@@]3(COP(S)(=O)O[C@@H]1[C@H]2F)C#C)n1cnc2c(N)ncnc12			574079	5-amino-3-[(5R,7R,8S,112aR,14R,15aS,16S)- 14-(6-amino-9H-purin-9-yl)-12a-ethynyl-16- fluoro-2,10-dioxido-2,10-disulfanyloctahydro- 12H-5,8-methanofuro[3,2- l][1,3,6,9,11,2,10]pentaoxadiphosphacyclotetra- decin-7-yl]-3,6-dihydro-7H-[1,2,3]triazolo[4,5- d]pyrimidin-7-one (Diastereomer 1)::US11453697, Example 207::US11453697, Example 208::US11453697, Example 209	Stimulator of interferon genes protein [H232R]					 23.3					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574079	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574079&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177602	474496364							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1211047	Nc1nc2n(nnc2c(=O)[nH]1)[C@@H]1O[C@@H]2COP(S)(=O)O[C@H]3C[C@@H](O[C@@]3(COP(S)(=O)O[C@@H]1[C@H]2F)C#C)n1cnc2c(N)ncnc12			574079	5-amino-3-[(5R,7R,8S,112aR,14R,15aS,16S)- 14-(6-amino-9H-purin-9-yl)-12a-ethynyl-16- fluoro-2,10-dioxido-2,10-disulfanyloctahydro- 12H-5,8-methanofuro[3,2- l][1,3,6,9,11,2,10]pentaoxadiphosphacyclotetra- decin-7-yl]-3,6-dihydro-7H-[1,2,3]triazolo[4,5- d]pyrimidin-7-one (Diastereomer 1)::US11453697, Example 207::US11453697, Example 208::US11453697, Example 209	Stimulator of interferon genes protein [H232R]					 9.50					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574079	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574079&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177602	474496364							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1211048	Nc1nc2n(nnc2c(=O)[nH]1)[C@@H]1O[C@@H]2COP(S)(=O)O[C@H]3C[C@@H](O[C@@H]3COP(S)(=O)O[C@@H]1[C@H]2F)c1cnn2c(N)ncnc12			574082	5-amino-3-[(5R,7R,8S,12aR,14R,15aS,16S)-14- (4-aminopyrazolo[1,5-a][1,3,5]triazin-8-yl)-16- fluoro-2,10-dioxido-2,10-disulfanyloctahydro- 12H-5,8-methanofuro[3,2- l][1,3,6,9,11,2,10]pentaoxadiphosphacyclotetra- decin-7-yl]-3,6-dihydro-7H-[1,2,3]triazolo[4,5- d]pyrimidin-7-one (Diastereomer 1)::US11453697, Example 210::US11453697, Example 211	Stimulator of interferon genes protein [H232R]					 28.5					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574082	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574082&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177603	474496365							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1211049	Nc1nc2n(nnc2c(=O)[nH]1)[C@@H]1O[C@@H]2COP(S)(=O)O[C@H]3C[C@@H](O[C@@H]3COP(S)(=O)O[C@@H]1[C@H]2F)c1cnn2c(N)ncnc12			574082	5-amino-3-[(5R,7R,8S,12aR,14R,15aS,16S)-14- (4-aminopyrazolo[1,5-a][1,3,5]triazin-8-yl)-16- fluoro-2,10-dioxido-2,10-disulfanyloctahydro- 12H-5,8-methanofuro[3,2- l][1,3,6,9,11,2,10]pentaoxadiphosphacyclotetra- decin-7-yl]-3,6-dihydro-7H-[1,2,3]triazolo[4,5- d]pyrimidin-7-one (Diastereomer 1)::US11453697, Example 210::US11453697, Example 211	Stimulator of interferon genes protein [H232R]					 1045					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574082	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574082&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177603	474496365							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1211050	Nc1nc2n(nnc2c(=O)[nH]1)[C@@H]1O[C@@H]2COP(O)(=S)O[C@H]3C[C@@H](O[C@@H]3COP(O)(=S)O[C@@H]1[C@H]2F)c1cnc2c(N)ncnn12			574084	5-amino-3-[(5R,7R,8S,12aR,14R,15aS,16S)-14- (4-aminoimidazo[2,1-f][1,2,4]triazin-7-yl)-16- fluoro-2,10-dihydroxy-2,10-disulfidooctahydro- 12H-5,8-methanofuro[3,2- l][1,3,6,9,11,2,10]pentaoxadiphosphacyclotetra- decin-7-yl]-3,6-dihydro-7H-[1,2,3]triazolo[4,5- d]pyrimidin-7-one (Diastereomer 1)::US11453697, Example 212::US11453697, Example 213	Stimulator of interferon genes protein [H232R]					 11.8					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574084	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574084&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177604	474496366							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1211051	Nc1nc2n(nnc2c(=O)[nH]1)[C@@H]1O[C@@H]2COP(O)(=S)O[C@H]3C[C@@H](O[C@@H]3COP(O)(=S)O[C@@H]1[C@H]2F)c1cnc2c(N)ncnn12			574084	5-amino-3-[(5R,7R,8S,12aR,14R,15aS,16S)-14- (4-aminoimidazo[2,1-f][1,2,4]triazin-7-yl)-16- fluoro-2,10-dihydroxy-2,10-disulfidooctahydro- 12H-5,8-methanofuro[3,2- l][1,3,6,9,11,2,10]pentaoxadiphosphacyclotetra- decin-7-yl]-3,6-dihydro-7H-[1,2,3]triazolo[4,5- d]pyrimidin-7-one (Diastereomer 1)::US11453697, Example 212::US11453697, Example 213	Stimulator of interferon genes protein [H232R]					 135					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574084	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574084&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177604	474496366							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1211052	Nc1nc2n(cnc2c(=O)[nH]1)[C@@H]1S[C@@H]2COP(S)(=O)O[C@@H]3[C@@H](COP(S)(=O)O[C@@H]1[C@@H]2F)O[C@H]([C@H]3F)n1cnc2c(N)ncnc12			574086	2-amino-9- [(5R,7R,8R,12aR,14R,15S,15aR,16S)- 14-(6-amino-9H-purin-9-yl)-15,16-difluoro-2,10- dioxido-2,10-disulfanyloctahydro- 12H-5,8-methanofuro[3,2- l][1,3,6,9,11,2,10]tetraoxathiadiphosphacyclo- tetradecin-7-yl]-1,9-dihydro-6H-purin-6-one (Diastereomer 1)::US11453697, Example 214::US11453697, Example 215::US11453697, Example 216::US11453697, Example 217	Stimulator of interferon genes protein [H232R]					 2.10					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574086	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574086&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177605	474496367							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1211053	Nc1nc2n(cnc2c(=O)[nH]1)[C@@H]1S[C@@H]2COP(S)(=O)O[C@@H]3[C@@H](COP(S)(=O)O[C@@H]1[C@@H]2F)O[C@H]([C@H]3F)n1cnc2c(N)ncnc12			574086	2-amino-9- [(5R,7R,8R,12aR,14R,15S,15aR,16S)- 14-(6-amino-9H-purin-9-yl)-15,16-difluoro-2,10- dioxido-2,10-disulfanyloctahydro- 12H-5,8-methanofuro[3,2- l][1,3,6,9,11,2,10]tetraoxathiadiphosphacyclo- tetradecin-7-yl]-1,9-dihydro-6H-purin-6-one (Diastereomer 1)::US11453697, Example 214::US11453697, Example 215::US11453697, Example 216::US11453697, Example 217	Stimulator of interferon genes protein [H232R]					 33.1					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574086	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574086&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177605	474496367							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1211054	Nc1nc2n(cnc2c(=O)[nH]1)[C@@H]1S[C@@H]2COP(S)(=O)O[C@@H]3[C@@H](COP(S)(=O)O[C@@H]1[C@@H]2F)O[C@H]([C@H]3F)n1cnc2c(N)ncnc12			574086	2-amino-9- [(5R,7R,8R,12aR,14R,15S,15aR,16S)- 14-(6-amino-9H-purin-9-yl)-15,16-difluoro-2,10- dioxido-2,10-disulfanyloctahydro- 12H-5,8-methanofuro[3,2- l][1,3,6,9,11,2,10]tetraoxathiadiphosphacyclo- tetradecin-7-yl]-1,9-dihydro-6H-purin-6-one (Diastereomer 1)::US11453697, Example 214::US11453697, Example 215::US11453697, Example 216::US11453697, Example 217	Stimulator of interferon genes protein [H232R]					 3.40					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574086	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574086&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177605	474496367							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1211055	Nc1nc2n(cnc2c(=O)[nH]1)[C@@H]1S[C@@H]2COP(S)(=O)O[C@@H]3[C@@H](COP(S)(=O)O[C@@H]1[C@@H]2F)O[C@H]([C@H]3F)n1cnc2c(N)ncnc12			574086	2-amino-9- [(5R,7R,8R,12aR,14R,15S,15aR,16S)- 14-(6-amino-9H-purin-9-yl)-15,16-difluoro-2,10- dioxido-2,10-disulfanyloctahydro- 12H-5,8-methanofuro[3,2- l][1,3,6,9,11,2,10]tetraoxathiadiphosphacyclo- tetradecin-7-yl]-1,9-dihydro-6H-purin-6-one (Diastereomer 1)::US11453697, Example 214::US11453697, Example 215::US11453697, Example 216::US11453697, Example 217	Stimulator of interferon genes protein [H232R]					 66.2					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574086	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574086&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177605	474496367							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1211056	Nc1nc2n(cnc2c(=O)[nH]1)[C@@H]1S[C@@H]2COP(S)(=O)O[C@@H]3[C@@H](COP(S)(=O)O[C@@H]1[C@@H]2F)O[C@H]([C@H]3F)n1nnc2c(N)ncnc12			574090	2-amino-9- [(5R,7R,8R,12aR,14R,15S,15aR,16S)-14-(7- amino-3H-[1,2,3]triazolo[4,5-d]pyrimidin-3-yl)- 15,16-difluoro-2,10-dioxido-2,10- disulfanyloctahydro-12H-5,8-methanofuro[3,2- l][1,3,9,11,6,2,10]tetraoxathiadiphosphacyclotetra- decin-7-yl]-1,9-dihydro-6H-purin-6-one (Diastereomer 1)::US11453697, Example 218::US11453697, Example 219	Stimulator of interferon genes protein [H232R]					 13.8					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574090	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574090&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177606	474496368							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1211057	Nc1nc2n(cnc2c(=O)[nH]1)[C@@H]1S[C@@H]2COP(S)(=O)O[C@@H]3[C@@H](COP(S)(=O)O[C@@H]1[C@@H]2F)O[C@H]([C@H]3F)n1nnc2c(N)ncnc12			574090	2-amino-9- [(5R,7R,8R,12aR,14R,15S,15aR,16S)-14-(7- amino-3H-[1,2,3]triazolo[4,5-d]pyrimidin-3-yl)- 15,16-difluoro-2,10-dioxido-2,10- disulfanyloctahydro-12H-5,8-methanofuro[3,2- l][1,3,9,11,6,2,10]tetraoxathiadiphosphacyclotetra- decin-7-yl]-1,9-dihydro-6H-purin-6-one (Diastereomer 1)::US11453697, Example 218::US11453697, Example 219	Stimulator of interferon genes protein [H232R]					 530					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574090	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574090&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177606	474496368							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1211058	Nc1nc2n(nnc2c(=O)[nH]1)[C@@H]1O[C@@H]2COP(O)(=S)O[C@@H]3[C@@H](COP(O)(=S)O[C@@H]1[C@H]2F)O[C@@H](n1ccc2c(N)ncnc12)C3(F)F			574092	5-amino-3-[(5R,7R,8S,12aR,14R,15aR,16S)-14- (4-amino-7H-pyrrolo[2,3-d]pyrimidin-7-yl)- 15,15,16-trifluoro-2,10-dihydroxy-2,10- disulfidooctahydro-12H-5,8-methanofuro[3,2- l][1,3,6,9,11,2,10]pentaoxadiphosphacyclotetra- decin-7-yl]-3,6-dihydro-7H-[1,2,3]triazolo[4,5- d]pyrimidin-7-one::US11453697, Example 220	Stimulator of interferon genes protein [H232R]					 29.0					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574092	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574092&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177607	474496369							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1211059	Nc1nc2n(nnc2c(=O)[nH]1)[C@@H]1S[C@@H]2COP(O)(=S)O[C@@H]3[C@@H](COP(O)(=S)O[C@@H]1[C@@H]2F)O[C@H]([C@H]3F)n1cnc2c(N)ncnc12			574093	5-amino-3- [(5R,7R,8R,12aR,14R,15S,15aR,16S)-14-(6- amino-9H-purin-9-yl)-15,16-difluoro-2,10- dihydroxy-2,10-disulfidooctahydro-12H-5,8- methanofuro[3,2- l][1,3,9,11,6,2,10]tetraoxathiadiphosphacyclotetra- decin-7-yl]-3,6-dihydro-7H41,2,3]triazolo[4,5- d]pyrimidin-7-one (Diastereomer 1)::US11453697, Example 221::US11453697, Example 222::US11453697, Example 223	Stimulator of interferon genes protein [H232R]					<1.000					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574093	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574093&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177608	474496370							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1211060	Nc1nc2n(nnc2c(=O)[nH]1)[C@@H]1S[C@@H]2COP(O)(=S)O[C@@H]3[C@@H](COP(O)(=S)O[C@@H]1[C@@H]2F)O[C@H]([C@H]3F)n1cnc2c(N)ncnc12			574093	5-amino-3- [(5R,7R,8R,12aR,14R,15S,15aR,16S)-14-(6- amino-9H-purin-9-yl)-15,16-difluoro-2,10- dihydroxy-2,10-disulfidooctahydro-12H-5,8- methanofuro[3,2- l][1,3,9,11,6,2,10]tetraoxathiadiphosphacyclotetra- decin-7-yl]-3,6-dihydro-7H41,2,3]triazolo[4,5- d]pyrimidin-7-one (Diastereomer 1)::US11453697, Example 221::US11453697, Example 222::US11453697, Example 223	Stimulator of interferon genes protein [H232R]					 60.0					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574093	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574093&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177608	474496370							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1211061	Nc1nc2n(nnc2c(=O)[nH]1)[C@@H]1S[C@@H]2COP(O)(=S)O[C@@H]3[C@@H](COP(O)(=S)O[C@@H]1[C@@H]2F)O[C@H]([C@H]3F)n1cnc2c(N)ncnc12			574093	5-amino-3- [(5R,7R,8R,12aR,14R,15S,15aR,16S)-14-(6- amino-9H-purin-9-yl)-15,16-difluoro-2,10- dihydroxy-2,10-disulfidooctahydro-12H-5,8- methanofuro[3,2- l][1,3,9,11,6,2,10]tetraoxathiadiphosphacyclotetra- decin-7-yl]-3,6-dihydro-7H41,2,3]triazolo[4,5- d]pyrimidin-7-one (Diastereomer 1)::US11453697, Example 221::US11453697, Example 222::US11453697, Example 223	Stimulator of interferon genes protein [H232R]					 302					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574093	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574093&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177608	474496370							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1211062	Nc1nc2n(nnc2c(=O)[nH]1)[C@@H]1S[C@@H]2COP(S)(=O)O[C@@H]3[C@@H](COP(S)(=O)O[C@@H]1[C@@H]2F)O[C@H]([C@H]3F)n1nnc2c(N)ncnc12			574096	5-amino-3- [(5R,7R,8R,12aR,14R,15S,15aR,16S)-14-(7- amino-3H-[1,2,3]triazolo[4,5-d]pyrimidin-3-yl)- 15,16-difluoro-2,10-dioxido-2,10- disulfanyloctahydro-12H-5,8-methanofuro[3,2- l][1,3,9,11,6,2,10]tetraoxathi adiphosphacyclotetra- decin-7-yl]-3,6-dihydro-7H-[1,2,3]triazolo[4,5- d]pyrimidin-7-one (Diastereomer 1)::US11453697, Example 224::US11453697, Example 225	Stimulator of interferon genes protein [H232R]					 37.4					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574096	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574096&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177609	474496371							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1211063	Nc1nc2n(nnc2c(=O)[nH]1)[C@@H]1S[C@@H]2COP(S)(=O)O[C@@H]3[C@@H](COP(S)(=O)O[C@@H]1[C@@H]2F)O[C@H]([C@H]3F)n1nnc2c(N)ncnc12			574096	5-amino-3- [(5R,7R,8R,12aR,14R,15S,15aR,16S)-14-(7- amino-3H-[1,2,3]triazolo[4,5-d]pyrimidin-3-yl)- 15,16-difluoro-2,10-dioxido-2,10- disulfanyloctahydro-12H-5,8-methanofuro[3,2- l][1,3,9,11,6,2,10]tetraoxathi adiphosphacyclotetra- decin-7-yl]-3,6-dihydro-7H-[1,2,3]triazolo[4,5- d]pyrimidin-7-one (Diastereomer 1)::US11453697, Example 224::US11453697, Example 225	Stimulator of interferon genes protein [H232R]					 779					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574096	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574096&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177609	474496371							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1211064	Nc1nc2n(nnc2c(=O)[nH]1)[C@@H]1S[C@@H]2COP(S)(=O)O[C@@H]3[C@@H](COP(S)(=O)O[C@@H]1[C@@H]2F)O[C@H]([C@H]3F)n1ccc2c(N)ncnc12			574098	5-amino-3- [(5R,7R,8R,12aR,14R,15S,15aR,16S)-14-(4- amino-7H-pyrrolo[2,3-d]pyrimidin-7-yl)-15,16- difluoro-2,10-dioxido-2,10-disulfanyloctahydro- 12H-5,8-methanofuro[3,2- l][1,3,9,11,6,2,10]tetraoxathiadiphosphacyclotetra- decin-7-yl]-3,6-dihydro-7H-[1,2,3]triazolo[4,5- d]pyrimidin-7-one (Diastereomer 1)::US11453697, Example 226::US11453697, Example 227	Stimulator of interferon genes protein [H232R]					 27.8					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574098	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574098&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177610	474496372							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1211065	Nc1nc2n(nnc2c(=O)[nH]1)[C@@H]1S[C@@H]2COP(S)(=O)O[C@@H]3[C@@H](COP(S)(=O)O[C@@H]1[C@@H]2F)O[C@H]([C@H]3F)n1ccc2c(N)ncnc12			574098	5-amino-3- [(5R,7R,8R,12aR,14R,15S,15aR,16S)-14-(4- amino-7H-pyrrolo[2,3-d]pyrimidin-7-yl)-15,16- difluoro-2,10-dioxido-2,10-disulfanyloctahydro- 12H-5,8-methanofuro[3,2- l][1,3,9,11,6,2,10]tetraoxathiadiphosphacyclotetra- decin-7-yl]-3,6-dihydro-7H-[1,2,3]triazolo[4,5- d]pyrimidin-7-one (Diastereomer 1)::US11453697, Example 226::US11453697, Example 227	Stimulator of interferon genes protein [H232R]					 261					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574098	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574098&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177610	474496372							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1211066	Nc1ncnc2n(ccc12)[C@@H]1O[C@@H]2COP(S)(=O)O[C@@H]3C[C@@H](COP(S)(=O)O[C@H]2[C@@H]1F)O[C@H]3n1cnc2c1cc[nH]c2=O			574100	1-[(5S,7R,8R,12aR,14R,15S,15aR)-14-(4- amino-7H-pyrrolo[2,3-d]pyrimidin-7-yl)-15- fluoro-2,10-dioxido-2,10-disulfanyloctahydro- 12H-5,8-methanofuro[3,2- l][1,3,6,9,11,2,10]pentaoxadiphosphacyclotetra- decin-7-yl]-1,5-dihydro-4H-imidazo[4,5- c]pyridin-4-one::US11453697, Example 228	Stimulator of interferon genes protein [H232R]					 1005					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574100	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574100&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177611	474496373							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1211067	Nc1cc2n(cnc2c(=O)[nH]1)[C@@H]1O[C@@H]2COP(S)(=O)O[C@@H]3[C@@H](COP(S)(=O)O[C@@H]1[C@@H]2F)O[C@H]([C@H]3F)n1ccc2c(N)ncnc12			574101	6-amino-1- [(5R,7R,8S,12aR,14R,15S,15aR,16R)-14-(4- amino-7H-pyrrolo[2,3-d]pyrimidin-7-yl)-15,16- difluoro-2,10-dioxido-2,10-disulfanyloctahydro- 12H-5,8-methanofuro[3,2- l][1,3,6,9,11,2,10]pentaoxadiphosphacyclotetra- decin-7-yl]-1,5-dihydro-4H-imidazo[4,5- c]pyridin-4-one (Diastereomer 1)::US11453697, Example 229::US11453697, Example 230	Stimulator of interferon genes protein [H232R]					 20000					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574101	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574101&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177612	474496374							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1211068	Nc1cc2n(cnc2c(=O)[nH]1)[C@@H]1O[C@@H]2COP(S)(=O)O[C@@H]3[C@@H](COP(S)(=O)O[C@@H]1[C@@H]2F)O[C@H]([C@H]3F)n1ccc2c(N)ncnc12			574101	6-amino-1- [(5R,7R,8S,12aR,14R,15S,15aR,16R)-14-(4- amino-7H-pyrrolo[2,3-d]pyrimidin-7-yl)-15,16- difluoro-2,10-dioxido-2,10-disulfanyloctahydro- 12H-5,8-methanofuro[3,2- l][1,3,6,9,11,2,10]pentaoxadiphosphacyclotetra- decin-7-yl]-1,5-dihydro-4H-imidazo[4,5- c]pyridin-4-one (Diastereomer 1)::US11453697, Example 229::US11453697, Example 230	Stimulator of interferon genes protein [H232R]					 382					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574101	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574101&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177612	474496374							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1211069	Nc1nc2n(cnc2c(=O)[nH]1)[C@@H]1S[C@@H]2COP(S)(=O)O[C@@H]3[C@@H](COP(S)(=O)O[C@@H]1[C@H]2F)O[C@H]([C@H]3F)n1nnc2c(N)ncnc12			574103	2-amino-9- [(5R,7R,8R,12aR,14R,15S,15aR,16R)-14-(7- amino-3H-[1,2,3]triazolo[4,5-d]pyrimidin-3-yl)- 15,16-difluoro-2,10-dioxido-2,10- disulfanyloctahydro-12H-5,8-methanofuro[3,2- l][1,3,9,11,6,2,10]tetraoxathiadiphosphacyclotetra- decin-7-yl]-1,9-dihydro-6H-purin-6-one (Diastereomer 1)::US11453697, Example 231::US11453697, Example 232::US11453697, Example 233	Stimulator of interferon genes protein [H232R]					 540					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574103	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574103&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177613	474496375							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1211070	Nc1nc2n(cnc2c(=O)[nH]1)[C@@H]1S[C@@H]2COP(S)(=O)O[C@@H]3[C@@H](COP(S)(=O)O[C@@H]1[C@H]2F)O[C@H]([C@H]3F)n1nnc2c(N)ncnc12			574103	2-amino-9- [(5R,7R,8R,12aR,14R,15S,15aR,16R)-14-(7- amino-3H-[1,2,3]triazolo[4,5-d]pyrimidin-3-yl)- 15,16-difluoro-2,10-dioxido-2,10- disulfanyloctahydro-12H-5,8-methanofuro[3,2- l][1,3,9,11,6,2,10]tetraoxathiadiphosphacyclotetra- decin-7-yl]-1,9-dihydro-6H-purin-6-one (Diastereomer 1)::US11453697, Example 231::US11453697, Example 232::US11453697, Example 233	Stimulator of interferon genes protein [H232R]					 3283					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574103	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574103&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177613	474496375							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1211071	Nc1nc2n(cnc2c(=O)[nH]1)[C@@H]1S[C@@H]2COP(S)(=O)O[C@@H]3[C@@H](COP(S)(=O)O[C@@H]1[C@H]2F)O[C@H]([C@H]3F)n1nnc2c(N)ncnc12			574103	2-amino-9- [(5R,7R,8R,12aR,14R,15S,15aR,16R)-14-(7- amino-3H-[1,2,3]triazolo[4,5-d]pyrimidin-3-yl)- 15,16-difluoro-2,10-dioxido-2,10- disulfanyloctahydro-12H-5,8-methanofuro[3,2- l][1,3,9,11,6,2,10]tetraoxathiadiphosphacyclotetra- decin-7-yl]-1,9-dihydro-6H-purin-6-one (Diastereomer 1)::US11453697, Example 231::US11453697, Example 232::US11453697, Example 233	Stimulator of interferon genes protein [H232R]					 33.8					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574103	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574103&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177613	474496375							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1211072	Nc1nc2n(cnc2c(=O)[nH]1)[C@@H]1S[C@H]2C[C@H]1OP(S)(=O)OC[C@H]1O[C@H]([C@@H](F)[C@@H]1OP(S)(=O)OC2)n1ccc2c(N)ncnc12			574106	2-amino-9-[(5S,7R,8R,12aR,14R,15S,15aR)-14- (4-amino-7H-pyrrolo[2,3-d]pyrimidin-7-yl)-15- fluoro-2,10-dioxido-2,10-disulfanyloctahydro- 12H-5,8-methanofuro[3,2- l][1,3,9,11,6,2,10]tetraoxathiadiphosphacyclotetra- decin-7-yl]-1,9-dihydro-6H-purin-6-one::US11453697, Example 234	Stimulator of interferon genes protein [H232R]					 275					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574106	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574106&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177614	474496376							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1211073	Nc1nc2n(nnc2c(=O)[nH]1)[C@@H]1S[C@@H]2COP(S)(=O)O[C@@H]3[C@@H](COP(S)(=O)O[C@@H]1[C@@H]2F)O[C@H]([C@H]3F)n1cnc2c(N)ncnc12			574107	5-amino-3- [(5R,7R,8R,12aR,14R,15S,15aR,16S)-14-(6- amino-9H-purin-9-yl)-15,16-difluoro-2,10- dioxido-2,10-disulfanyloctahydro-12H-5,8- methanofuro[3,2- l][1,3,9,11,6,2,10]tetraoxathiadiphosphacyclo- decin-7-yl]-3,6-dihydro-7H-[1,2,3]triazolo[4,5- d]pyrimidin-7-one::US11453697, Example 235	Stimulator of interferon genes protein [H232R]					 14.9					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574107	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574107&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177615	474496377							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1211074	Nc1nc2n(cnc2c(=O)[nH]1)[C@@H]1S[C@@H]2COP(S)(=O)O[C@@H]3[C@@H](COP(S)(=O)O[C@@H]1[C@H]2F)O[C@@H](n1nnc2c(N)ncnc12)C3(F)F			574108	2-amino-9-[(5R,7R,8R,12aR,14R,15aR,16R)-14- (7-amino-3H-[1,2,3]triazolo[4,5-d]pyrimidin-3- yl)-15,15,16-trifluoro-2,10-dioxido-2,10- disulfanyloctahydro-12H-5,8-methanofuro[3,2- l][1,3,9,11,6,2,10]tetraoxathiadiphosphacyclotetra- decin-7-yl]-1,9-dihydro-6H-purin-6-one (Diastereomer 1)::US11453697, Example 236::US11453697, Example 237::US11453697, Example 238::US11453697, Example 239	Stimulator of interferon genes protein [H232R]					 6963					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574108	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574108&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177616	474496378							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1211075	Nc1nc2n(cnc2c(=O)[nH]1)[C@@H]1S[C@@H]2COP(S)(=O)O[C@@H]3[C@@H](COP(S)(=O)O[C@@H]1[C@H]2F)O[C@@H](n1nnc2c(N)ncnc12)C3(F)F			574108	2-amino-9-[(5R,7R,8R,12aR,14R,15aR,16R)-14- (7-amino-3H-[1,2,3]triazolo[4,5-d]pyrimidin-3- yl)-15,15,16-trifluoro-2,10-dioxido-2,10- disulfanyloctahydro-12H-5,8-methanofuro[3,2- l][1,3,9,11,6,2,10]tetraoxathiadiphosphacyclotetra- decin-7-yl]-1,9-dihydro-6H-purin-6-one (Diastereomer 1)::US11453697, Example 236::US11453697, Example 237::US11453697, Example 238::US11453697, Example 239	Stimulator of interferon genes protein [H232R]					 307					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574108	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574108&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177616	474496378							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1211076	Nc1nc2n(cnc2c(=O)[nH]1)[C@@H]1S[C@@H]2COP(S)(=O)O[C@@H]3[C@@H](COP(S)(=O)O[C@@H]1[C@H]2F)O[C@@H](n1nnc2c(N)ncnc12)C3(F)F			574108	2-amino-9-[(5R,7R,8R,12aR,14R,15aR,16R)-14- (7-amino-3H-[1,2,3]triazolo[4,5-d]pyrimidin-3- yl)-15,15,16-trifluoro-2,10-dioxido-2,10- disulfanyloctahydro-12H-5,8-methanofuro[3,2- l][1,3,9,11,6,2,10]tetraoxathiadiphosphacyclotetra- decin-7-yl]-1,9-dihydro-6H-purin-6-one (Diastereomer 1)::US11453697, Example 236::US11453697, Example 237::US11453697, Example 238::US11453697, Example 239	Stimulator of interferon genes protein [H232R]					 66.3					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574108	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574108&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177616	474496378							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1211077	Nc1nc2n(cnc2c(=O)[nH]1)[C@@H]1S[C@@H]2COP(S)(=O)O[C@@H]3[C@@H](COP(S)(=O)O[C@@H]1[C@H]2F)O[C@@H](n1nnc2c(N)ncnc12)C3(F)F			574108	2-amino-9-[(5R,7R,8R,12aR,14R,15aR,16R)-14- (7-amino-3H-[1,2,3]triazolo[4,5-d]pyrimidin-3- yl)-15,15,16-trifluoro-2,10-dioxido-2,10- disulfanyloctahydro-12H-5,8-methanofuro[3,2- l][1,3,9,11,6,2,10]tetraoxathiadiphosphacyclotetra- decin-7-yl]-1,9-dihydro-6H-purin-6-one (Diastereomer 1)::US11453697, Example 236::US11453697, Example 237::US11453697, Example 238::US11453697, Example 239	Stimulator of interferon genes protein [H232R]					 3.20					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574108	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574108&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177616	474496378							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1211078	Nc1nc2n(cnc2c(=O)[nH]1)[C@@H]1S[C@@H]2COP(S)(=O)O[C@H]3[C@H]4OCC3(COP(S)(=O)O[C@@H]1[C@H]2F)O[C@H]4n1cnc2c(N)ncnc12			574112	2-amino-9- [(5R,7R,8R,12aR,14R,15R,15aS,18R)-14-(6- amino-9H-purin-9-yl)-18-fluoro-2,10-dioxido- 2,10-disulfanylhexahydro-14H-15,12a- (epoxymethano)-5,8-methanofuro[3,2- l][1,3,9,11,6,2,10]tetraoxathiadiphosphacyclotetra- decin-7(12H)-yl]-1,9-dihydro-6H-purin-6-one (Diastereomer 1)::US11453697, Example 240::US11453697, Example 241::US11453697, Example 242	Stimulator of interferon genes protein [H232R]					 73.6					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574112	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574112&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177617	474496379							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1211079	Nc1nc2n(cnc2c(=O)[nH]1)[C@@H]1S[C@@H]2COP(S)(=O)O[C@H]3[C@H]4OCC3(COP(S)(=O)O[C@@H]1[C@H]2F)O[C@H]4n1cnc2c(N)ncnc12			574112	2-amino-9- [(5R,7R,8R,12aR,14R,15R,15aS,18R)-14-(6- amino-9H-purin-9-yl)-18-fluoro-2,10-dioxido- 2,10-disulfanylhexahydro-14H-15,12a- (epoxymethano)-5,8-methanofuro[3,2- l][1,3,9,11,6,2,10]tetraoxathiadiphosphacyclotetra- decin-7(12H)-yl]-1,9-dihydro-6H-purin-6-one (Diastereomer 1)::US11453697, Example 240::US11453697, Example 241::US11453697, Example 242	Stimulator of interferon genes protein [H232R]					 472					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574112	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574112&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177617	474496379							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1211080	Nc1nc2n(cnc2c(=O)[nH]1)[C@@H]1S[C@@H]2COP(S)(=O)O[C@H]3[C@H]4OCC3(COP(S)(=O)O[C@@H]1[C@H]2F)O[C@H]4n1cnc2c(N)ncnc12			574112	2-amino-9- [(5R,7R,8R,12aR,14R,15R,15aS,18R)-14-(6- amino-9H-purin-9-yl)-18-fluoro-2,10-dioxido- 2,10-disulfanylhexahydro-14H-15,12a- (epoxymethano)-5,8-methanofuro[3,2- l][1,3,9,11,6,2,10]tetraoxathiadiphosphacyclotetra- decin-7(12H)-yl]-1,9-dihydro-6H-purin-6-one (Diastereomer 1)::US11453697, Example 240::US11453697, Example 241::US11453697, Example 242	Stimulator of interferon genes protein [H232R]					 1.10					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574112	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574112&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177617	474496379							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1211081	Nc1nc2n(cnc2c(=O)[nH]1)[C@@H]1S[C@@H]2COP(S)(=O)O[C@@H]3[C@@H](COP(S)(=O)O[C@@H]1[C@H]2F)O[C@H]([C@H]3F)n1cnc2c(N)ccnc12			574115	2-amino-9- [(5R,7R,8R,12aR,14R,15S,15aR,16R)-14-(7- amino-3H-imidazo[4,5-b]pyridin-3-yl)-15,16- difluoro-2,10-dioxido-2,10-disulfanyloctahydro- 12H-5,8-methanofuro[3,2- l][1,3,9,11,6,2,10]tetraoxathiadiphosphacyclotetra- decin-7-yl]-1,9-dihydro-6H-purin-6-one::US11453697, Example 243	Stimulator of interferon genes protein [H232R]					 26.3					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574115	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574115&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177618	474496380							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1211082	Nc1nc2n(cnc2c(=O)[nH]1)[C@@H]1O[C@@H]2CO[P@](S)(=O)O[C@@H]3[C@@H](CO[P@](S)(=O)O[C@@H]1[C@@H]2F)O[C@H]([C@H]3F)n1cnc2c(N)ncnc12			573971	US11453697, Example 247	Stimulator of interferon genes protein [H232R]					 1.10					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=573971	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=573971&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177537	474496300							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1211083	Nc1nc2n(cnc2c(=O)[nH]1)[C@@H]1O[C@@H]2COP(S)(=O)O[C@H]3C[C@@H](O[C@@H]3COP(S)(=O)O[C@@H]1[C@@H]2F)c1cnc2c(N)ncnn12			574116	2-amino-9-[(5R,7R,8S,12aR,14R,15aS,16R)-14- (4-aminoimidazo[2,1-f][1,2,4]triazin-7-yl)-16- fluoro-2,10-dioxido-2,10-disulfanyloctahydro- 12H-5,8-methanofuro[3,2- 1][1,3,6,9,11,2,10]pentaoxadiphosphacyclotetra- decin-7-yl]-1,9-dihydro-6H-purin-6-one (Diastereomer 1)::US11453697, Example 248::US11453697, Example 249::US11453697, Example 250::US11453697, Example 251	Stimulator of interferon genes protein [H232R]					 31.7					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574116	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574116&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177619	474496381							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1211084	Nc1nc2n(cnc2c(=O)[nH]1)[C@@H]1O[C@@H]2COP(S)(=O)O[C@H]3C[C@@H](O[C@@H]3COP(S)(=O)O[C@@H]1[C@@H]2F)c1cnc2c(N)ncnn12			574116	2-amino-9-[(5R,7R,8S,12aR,14R,15aS,16R)-14- (4-aminoimidazo[2,1-f][1,2,4]triazin-7-yl)-16- fluoro-2,10-dioxido-2,10-disulfanyloctahydro- 12H-5,8-methanofuro[3,2- 1][1,3,6,9,11,2,10]pentaoxadiphosphacyclotetra- decin-7-yl]-1,9-dihydro-6H-purin-6-one (Diastereomer 1)::US11453697, Example 248::US11453697, Example 249::US11453697, Example 250::US11453697, Example 251	Stimulator of interferon genes protein [H232R]					<1.000					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574116	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574116&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177619	474496381							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1211085	Nc1nc2n(cnc2c(=O)[nH]1)[C@@H]1O[C@@H]2COP(S)(=O)O[C@H]3C[C@@H](O[C@@H]3COP(S)(=O)O[C@@H]1[C@@H]2F)c1cnc2c(N)ncnn12			574116	2-amino-9-[(5R,7R,8S,12aR,14R,15aS,16R)-14- (4-aminoimidazo[2,1-f][1,2,4]triazin-7-yl)-16- fluoro-2,10-dioxido-2,10-disulfanyloctahydro- 12H-5,8-methanofuro[3,2- 1][1,3,6,9,11,2,10]pentaoxadiphosphacyclotetra- decin-7-yl]-1,9-dihydro-6H-purin-6-one (Diastereomer 1)::US11453697, Example 248::US11453697, Example 249::US11453697, Example 250::US11453697, Example 251	Stimulator of interferon genes protein [H232R]					 17.3					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574116	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574116&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177619	474496381							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1211086	Nc1nc2n(cnc2c(=O)[nH]1)[C@@H]1O[C@@H]2COP(S)(=O)O[C@H]3C[C@@H](O[C@@H]3COP(S)(=O)O[C@@H]1[C@@H]2F)c1cnc2c(N)ncnn12			574116	2-amino-9-[(5R,7R,8S,12aR,14R,15aS,16R)-14- (4-aminoimidazo[2,1-f][1,2,4]triazin-7-yl)-16- fluoro-2,10-dioxido-2,10-disulfanyloctahydro- 12H-5,8-methanofuro[3,2- 1][1,3,6,9,11,2,10]pentaoxadiphosphacyclotetra- decin-7-yl]-1,9-dihydro-6H-purin-6-one (Diastereomer 1)::US11453697, Example 248::US11453697, Example 249::US11453697, Example 250::US11453697, Example 251	Stimulator of interferon genes protein [H232R]					<1.000					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574116	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574116&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177619	474496381							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1211087	Nc1nc2n(cnc2c(=O)[nH]1)[C@@H]1O[C@@H]2COP(S)(=O)O[C@H]3C[C@@H](O[C@@H]3COP(S)(=O)O[C@@H]1[C@@H]2F)n1cc(F)c2c(N)ncnc12			574120	2-amino-9-[(5R,7R,8S,12aR,14R,15aS,16R)-14- (4-amino-5-fluoro-7H-pyrrolo[2,3-d]pyrimidin- 7-yl)-16-fluoro-2,10-dioxido-2,10- disulfanyloctahydro-12H-5,8-methanofuro[3,2- 1][1,3,6,9,11,2,10]pentaoxadiphosphacyclotetra- decin-7-yl]-1,9-dihydro-6H-purin-6-one (Diastereomer 1)::US11453697, Example 252::US11453697, Example 253::US11453697, Example 254::US11453697, Example 255::US11453697, Example 256	Stimulator of interferon genes protein [H232R]					 768					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574120	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574120&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177620	474496382							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1211088	Nc1nc2n(cnc2c(=O)[nH]1)[C@@H]1O[C@@H]2COP(S)(=O)O[C@H]3C[C@@H](O[C@@H]3COP(S)(=O)O[C@@H]1[C@@H]2F)n1cc(F)c2c(N)ncnc12			574120	2-amino-9-[(5R,7R,8S,12aR,14R,15aS,16R)-14- (4-amino-5-fluoro-7H-pyrrolo[2,3-d]pyrimidin- 7-yl)-16-fluoro-2,10-dioxido-2,10- disulfanyloctahydro-12H-5,8-methanofuro[3,2- 1][1,3,6,9,11,2,10]pentaoxadiphosphacyclotetra- decin-7-yl]-1,9-dihydro-6H-purin-6-one (Diastereomer 1)::US11453697, Example 252::US11453697, Example 253::US11453697, Example 254::US11453697, Example 255::US11453697, Example 256	Stimulator of interferon genes protein [H232R]					 54.5					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574120	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574120&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177620	474496382							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1211089	Nc1nc2n(cnc2c(=O)[nH]1)[C@@H]1O[C@@H]2COP(S)(=O)O[C@H]3C[C@@H](O[C@@H]3COP(S)(=O)O[C@@H]1[C@@H]2F)n1cc(F)c2c(N)ncnc12			574120	2-amino-9-[(5R,7R,8S,12aR,14R,15aS,16R)-14- (4-amino-5-fluoro-7H-pyrrolo[2,3-d]pyrimidin- 7-yl)-16-fluoro-2,10-dioxido-2,10- disulfanyloctahydro-12H-5,8-methanofuro[3,2- 1][1,3,6,9,11,2,10]pentaoxadiphosphacyclotetra- decin-7-yl]-1,9-dihydro-6H-purin-6-one (Diastereomer 1)::US11453697, Example 252::US11453697, Example 253::US11453697, Example 254::US11453697, Example 255::US11453697, Example 256	Stimulator of interferon genes protein [H232R]					 39.7					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574120	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574120&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177620	474496382							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1211090	Nc1nc2n(cnc2c(=O)[nH]1)[C@@H]1O[C@@H]2COP(S)(=O)O[C@H]3C[C@@H](O[C@@H]3COP(S)(=O)O[C@@H]1[C@@H]2F)n1cc(F)c2c(N)ncnc12			574120	2-amino-9-[(5R,7R,8S,12aR,14R,15aS,16R)-14- (4-amino-5-fluoro-7H-pyrrolo[2,3-d]pyrimidin- 7-yl)-16-fluoro-2,10-dioxido-2,10- disulfanyloctahydro-12H-5,8-methanofuro[3,2- 1][1,3,6,9,11,2,10]pentaoxadiphosphacyclotetra- decin-7-yl]-1,9-dihydro-6H-purin-6-one (Diastereomer 1)::US11453697, Example 252::US11453697, Example 253::US11453697, Example 254::US11453697, Example 255::US11453697, Example 256	Stimulator of interferon genes protein [H232R]					 302					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574120	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574120&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177620	474496382							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1211091	Nc1nc2n(cnc2c(=O)[nH]1)[C@@H]1O[C@@H]2COP(S)(=O)O[C@H]3C[C@@H](O[C@@H]3COP(S)(=O)O[C@@H]1[C@@H]2F)n1cc(F)c2c(N)ncnc12			574120	2-amino-9-[(5R,7R,8S,12aR,14R,15aS,16R)-14- (4-amino-5-fluoro-7H-pyrrolo[2,3-d]pyrimidin- 7-yl)-16-fluoro-2,10-dioxido-2,10- disulfanyloctahydro-12H-5,8-methanofuro[3,2- 1][1,3,6,9,11,2,10]pentaoxadiphosphacyclotetra- decin-7-yl]-1,9-dihydro-6H-purin-6-one (Diastereomer 1)::US11453697, Example 252::US11453697, Example 253::US11453697, Example 254::US11453697, Example 255::US11453697, Example 256	Stimulator of interferon genes protein [H232R]					 93.5					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574120	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574120&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177620	474496382							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1211092	Nc1nc2n(cnc2c(=O)[nH]1)[C@@H]1O[C@@H]2COP(S)(=O)O[C@H]3C[C@@H](O[C@@H]3COP(S)(=O)O[C@@H]1[C@@H]2F)c1cnn2c(N)ncnc12			574125	2-amino-9-[(5R,7R,8S,12aR,14R,15aS,16R)-14- (4-aminopyrazolo[1,5-a][1,3,5]triazin-8-yl)-16- fluoro-2,10-dihydroxy-2,10-disulfidooctahydro- 12H-5,8-methanofuro[3,2- 1][1,3,6,9,11,2,10]pentaoxadiphosphacyclotetra- decin-7-yl]-1,9-dihydro-6H-purin-6-one (Diastereomer 1)::US11453697, Example 257::US11453697, Example 258::US11453697, Example 259	Stimulator of interferon genes protein [H232R]					 136					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574125	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574125&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177621	474496383							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1211093	Nc1nc2n(cnc2c(=O)[nH]1)[C@@H]1O[C@@H]2COP(S)(=O)O[C@H]3C[C@@H](O[C@@H]3COP(S)(=O)O[C@@H]1[C@@H]2F)c1cnn2c(N)ncnc12			574125	2-amino-9-[(5R,7R,8S,12aR,14R,15aS,16R)-14- (4-aminopyrazolo[1,5-a][1,3,5]triazin-8-yl)-16- fluoro-2,10-dihydroxy-2,10-disulfidooctahydro- 12H-5,8-methanofuro[3,2- 1][1,3,6,9,11,2,10]pentaoxadiphosphacyclotetra- decin-7-yl]-1,9-dihydro-6H-purin-6-one (Diastereomer 1)::US11453697, Example 257::US11453697, Example 258::US11453697, Example 259	Stimulator of interferon genes protein [H232R]					 5.00					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574125	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574125&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177621	474496383							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1211094	Nc1nc2n(cnc2c(=O)[nH]1)[C@@H]1O[C@@H]2COP(S)(=O)O[C@H]3C[C@@H](O[C@@H]3COP(S)(=O)O[C@@H]1[C@@H]2F)c1cnn2c(N)ncnc12			574125	2-amino-9-[(5R,7R,8S,12aR,14R,15aS,16R)-14- (4-aminopyrazolo[1,5-a][1,3,5]triazin-8-yl)-16- fluoro-2,10-dihydroxy-2,10-disulfidooctahydro- 12H-5,8-methanofuro[3,2- 1][1,3,6,9,11,2,10]pentaoxadiphosphacyclotetra- decin-7-yl]-1,9-dihydro-6H-purin-6-one (Diastereomer 1)::US11453697, Example 257::US11453697, Example 258::US11453697, Example 259	Stimulator of interferon genes protein [H232R]					 1.50					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574125	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574125&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177621	474496383							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1211095	Nc1nc2n(cnc2c(=O)[nH]1)[C@@H]1O[C@@H]2COP(O)(=S)O[C@@H]3[C@@H](COP(O)(=S)O[C@@H]1[C@@H]2F)O[C@H]([C@@H]3F)n1cnc2c(N)ncnc12			574128	US11453697, Example 260	Stimulator of interferon genes protein [H232R]					 7.20					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574128	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574128&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177622	474496384							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1211096	Nc1nc2n(cnc2c(=O)[nH]1)[C@@H]1O[C@@H]2COP(O)(=S)O[C@H]3C[C@@H](O[C@@]3(COP(O)(=S)O[C@@H]1[C@@H]2F)C#C)n1cc(F)c2c(N)[nH]cnc12			574129	US11453697, Example 261::US11453697, Example 262	Stimulator of interferon genes protein [H232R]					 21.8					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574129	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574129&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177623	474496385							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1211097	Nc1nc2n(cnc2c(=O)[nH]1)[C@@H]1O[C@@H]2COP(O)(=S)O[C@H]3C[C@@H](O[C@@]3(COP(O)(=S)O[C@@H]1[C@@H]2F)C#C)n1cc(F)c2c(N)[nH]cnc12			574129	US11453697, Example 261::US11453697, Example 262	Stimulator of interferon genes protein [H232R]					 57.3					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574129	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574129&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177623	474496385							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1211098	Nc1nc2n(cnc2c(=O)[nH]1)[C@@H]1O[C@@H]2COP(O)(=S)O[C@H]3C[C@@H](O[C@@]3(COP(O)(=S)O[C@@H]1[C@@H]2F)C#C)n1cc(F)c2c(N)ncnc12			574131	US11453697, Example 263	Stimulator of interferon genes protein [H232R]					 4.80					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574131	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574131&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177624	474496386							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1211099	Nc1nc2n(cnc2c(=O)[nH]1)[C@@H]1S[C@@H]2COP(O)(=O)O[C@H]3[C@H]4OCC3(COP(O)(=S)O[C@@H]1[C@@H]2O)O[C@H]4n1cnc2c(N)ncnc12			574132	2-amino-9-[(5R,7R,8R,12aR,14R,15R,15aS,18S)-14-(6-amino-9H-purin-9-yl)-2,10,18-trihydroxy-2-oxido-10-sulfidohexahydro-14H-15,12a-(epoxymethano)-5,8-methanofuro[3,2-l][1,3,9,11,6,2,10]tetraoxathiadiphosphacyclotetradecin-7(12H)-yl]-1,9-dihydro-6H-purin-6-one (Diastereomer 1)::US11453697, Example 264::US11453697, Example 265	Stimulator of interferon genes protein [H232R]					 178					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574132	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574132&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177625	474496387							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1211100	Nc1nc2n(cnc2c(=O)[nH]1)[C@@H]1S[C@@H]2COP(O)(=O)O[C@H]3[C@H]4OCC3(COP(O)(=S)O[C@@H]1[C@@H]2O)O[C@H]4n1cnc2c(N)ncnc12			574132	2-amino-9-[(5R,7R,8R,12aR,14R,15R,15aS,18S)-14-(6-amino-9H-purin-9-yl)-2,10,18-trihydroxy-2-oxido-10-sulfidohexahydro-14H-15,12a-(epoxymethano)-5,8-methanofuro[3,2-l][1,3,9,11,6,2,10]tetraoxathiadiphosphacyclotetradecin-7(12H)-yl]-1,9-dihydro-6H-purin-6-one (Diastereomer 1)::US11453697, Example 264::US11453697, Example 265	Stimulator of interferon genes protein [H232R]					 5473					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574132	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574132&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177625	474496387							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1211101	Nc1nc2n(cnc2c(=O)[nH]1)[C@@H]1S[C@@H]2COP(O)(=O)O[C@@H]3[C@@H](COP(O)(=S)O[C@@H]1[C@@H]2O)O[C@H]([C@H]3F)n1cnc2c(N)ncnc12			574134	2-amino-9-[(5R,7R,8R,12aR,14R,15S,15aR,16S)- 14-(6-amino-9H-purin-9-yl)-15-fluoro-2,10,16- trihydroxy-2-oxido-10-sulfidooctahydro-12H-5,8- methanofuro[3,2- 1][1,3,9,11,6,2,10]tetraoxathiadiphosphacyclo- tetradecin-7-yl]-1,9-dihydro-6H-purin-6-one::US11453697, Example 266	Stimulator of interferon genes protein [H232R]					 1.90					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574134	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574134&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177626	474496388							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1211102	Nc1nc2n(nnc2c(=O)[nH]1)[C@@H]1S[C@@H]2COP(O)(=O)O[C@H]3C[C@@H](O[C@@H]3COP(S)(=O)O[C@@H]1[C@@H]2O)c1cnn2c(N)ncnc12			574135	5-amino-3-[(5R,7R,8R,12aR,14R,15aS,16S)-14- (4-aminopyrazolo[1,5-a][1,3,5]triazin-8-yl)-2,16- dihydroxy-2,10-dioxido-10-sulfanyloctahydro- 12H-5,8-methanofuro[3,2- 1][1,3,9,11,6,2,10]tetraoxathiadiphosphacyclo- tetradecin-7-yl]-3,6-dihydro-7H-[1,2,3]triazolo [4,5-d]pyrimidin-7-one (Diastereomer 1)::US11453697, Example 267::US11453697, Example 268	Stimulator of interferon genes protein [H232R]					 6267					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574135	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574135&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177627	474496389							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1211103	Nc1nc2n(nnc2c(=O)[nH]1)[C@@H]1S[C@@H]2COP(O)(=O)O[C@H]3C[C@@H](O[C@@H]3COP(S)(=O)O[C@@H]1[C@@H]2O)c1cnn2c(N)ncnc12			574135	5-amino-3-[(5R,7R,8R,12aR,14R,15aS,16S)-14- (4-aminopyrazolo[1,5-a][1,3,5]triazin-8-yl)-2,16- dihydroxy-2,10-dioxido-10-sulfanyloctahydro- 12H-5,8-methanofuro[3,2- 1][1,3,9,11,6,2,10]tetraoxathiadiphosphacyclo- tetradecin-7-yl]-3,6-dihydro-7H-[1,2,3]triazolo [4,5-d]pyrimidin-7-one (Diastereomer 1)::US11453697, Example 267::US11453697, Example 268	Stimulator of interferon genes protein [H232R]					 77.0					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574135	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574135&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177627	474496389							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1211104	Nc1nc2n(nnc2c(=O)[nH]1)[C@@H]1S[C@@H]2COP(O)(=O)O[C@@H]3[C@@H](COP(S)(=O)O[C@@H]1[C@@H]2O)O[C@H]([C@H]3F)n1nnc2c(N)ncnc12			574137	5-amino-3-[(5R,7R,8R,12aR,14R,15S,15aR,16S)- 14-(7-amino-3H-[1,2,3]triazolo[4,5-d]pyrimidin- 3-yl)-15-fluoro-2,16-dihydroxy-2,10-dioxido-10- sulfanyloctahydro-12H-5,8-methanofuro[3,2- 1][1,3,9,11,6,2,10]tetraoxathiadiphosphacyclo- tetradecin-7-yl]-3,6-dihydro-7H-[1,2,3]triazolo [4,5-d]pyrimidin-7-one (Diastereomer 1)::US11453697, Example 269::US11453697, Example 270	Stimulator of interferon genes protein [H232R]					 4837					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574137	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574137&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177628	474496390							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1211105	Nc1nc2n(nnc2c(=O)[nH]1)[C@@H]1S[C@@H]2COP(O)(=O)O[C@@H]3[C@@H](COP(S)(=O)O[C@@H]1[C@@H]2O)O[C@H]([C@H]3F)n1nnc2c(N)ncnc12			574137	5-amino-3-[(5R,7R,8R,12aR,14R,15S,15aR,16S)- 14-(7-amino-3H-[1,2,3]triazolo[4,5-d]pyrimidin- 3-yl)-15-fluoro-2,16-dihydroxy-2,10-dioxido-10- sulfanyloctahydro-12H-5,8-methanofuro[3,2- 1][1,3,9,11,6,2,10]tetraoxathiadiphosphacyclo- tetradecin-7-yl]-3,6-dihydro-7H-[1,2,3]triazolo [4,5-d]pyrimidin-7-one (Diastereomer 1)::US11453697, Example 269::US11453697, Example 270	Stimulator of interferon genes protein [H232R]					 4383					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574137	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574137&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177628	474496390							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1211106	Nc1nc2n(nnc2c(=O)[nH]1)[C@@H]1S[C@@H]2COP(O)(=O)O[C@H]3C[C@@H](O[C@@H]3COP(S)(=O)O[C@@H]1[C@@H]2O)c1cnc2c(N)ncnn12			574139	5-amino-3-[(5R,7R,8R,12aR,14R,15aS,16S)-14- (4-aminoimidazo[2,1-f][1,2,4]triazin-7-yl)-2,16- dihydroxy-2,10-dioxido-10-sulfanyloctahydro- 12H-5,8-methanofuro[3,2- 1][1,3,9,11,6,2,10]tetraoxathiadiphosphacyclo- tetradecin-7-yl]-3,6-dihydro-7H-[1,2,3]triazolo [4,5-d]pyrimidin-7-one (Diastereomer 1)::US11453697, Example 271::US11453697, Example 272	Stimulator of interferon genes protein [H232R]					 12.8					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574139	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574139&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177629	474496391							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1211107	Nc1nc2n(nnc2c(=O)[nH]1)[C@@H]1S[C@@H]2COP(O)(=O)O[C@H]3C[C@@H](O[C@@H]3COP(S)(=O)O[C@@H]1[C@@H]2O)c1cnc2c(N)ncnn12			574139	5-amino-3-[(5R,7R,8R,12aR,14R,15aS,16S)-14- (4-aminoimidazo[2,1-f][1,2,4]triazin-7-yl)-2,16- dihydroxy-2,10-dioxido-10-sulfanyloctahydro- 12H-5,8-methanofuro[3,2- 1][1,3,9,11,6,2,10]tetraoxathiadiphosphacyclo- tetradecin-7-yl]-3,6-dihydro-7H-[1,2,3]triazolo [4,5-d]pyrimidin-7-one (Diastereomer 1)::US11453697, Example 271::US11453697, Example 272	Stimulator of interferon genes protein [H232R]					 750					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574139	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574139&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177629	474496391							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1211108	Nc1nc2n(cnc2c(=O)[nH]1)[C@@H]1O[C@@H]2COP(O)(=O)O[C@@H]3[C@@H](COP(O)(=S)O[C@@H]1[C@@H]2F)O[C@H]([C@H]3F)n1cnc2c(N)ncnc12			574141	2-amino-9-[(5R,7R,8S,12aR,14R,15S,15aR,16R)-14-(6-amino-9H-purin-9-yl)-15,16-difluoro-2,10-dihydroxy-2-oxido-10-sulfidooctahydro-12H-5,8-methanofuro[3,2-l][1,3,6,9,11,2,10]pentaoxadiphosphacyclotetradecin-7-yl]-1,9-dihydro-6-purin-6-one (Diastereomer 1)::US11453697, Example 273::US11453697, Example 274	Stimulator of interferon genes protein [H232R]					 216					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574141	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574141&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177630	474496392							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1211109	Nc1nc2n(cnc2c(=O)[nH]1)[C@@H]1O[C@@H]2COP(O)(=O)O[C@@H]3[C@@H](COP(O)(=S)O[C@@H]1[C@@H]2F)O[C@H]([C@H]3F)n1cnc2c(N)ncnc12			574141	2-amino-9-[(5R,7R,8S,12aR,14R,15S,15aR,16R)-14-(6-amino-9H-purin-9-yl)-15,16-difluoro-2,10-dihydroxy-2-oxido-10-sulfidooctahydro-12H-5,8-methanofuro[3,2-l][1,3,6,9,11,2,10]pentaoxadiphosphacyclotetradecin-7-yl]-1,9-dihydro-6-purin-6-one (Diastereomer 1)::US11453697, Example 273::US11453697, Example 274	Stimulator of interferon genes protein [H232R]					 2.30					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574141	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574141&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177630	474496392							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1211110	Nc1nc2n(cnc2c(=O)[nH]1)[C@@H]1O[C@H]2C[C@H]1OP(O)(=S)OC[C@H]1O[C@H](C[C@@H]1OP(O)(=O)OC2)n1ccc2c(N)ncnc12			574143	2-amino-9-[(5S,7R,8R,12aR,14R,15aS)-14-(4- amino-7H-pyrrolo[2,3-d]pyrimidin-7-yl)-2,10- dihydroxy-2-oxido-10-sulfidooctahydro-12H-5,8- methanofuro[3,2-l][1,3,6,9,11,2,10] pentaoxadiphosphacyclotetradecin-7-yl]-1,9- dihydro-6H-purin-6-one (Diastereomer 1)::US11453697, Example 275::US11453697, Example 276	Stimulator of interferon genes protein [H232R]					 21.8					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574143	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574143&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177631	474496393							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1211111	Nc1nc2n(cnc2c(=O)[nH]1)[C@@H]1O[C@H]2C[C@H]1OP(O)(=S)OC[C@H]1O[C@H](C[C@@H]1OP(O)(=O)OC2)n1ccc2c(N)ncnc12			574143	2-amino-9-[(5S,7R,8R,12aR,14R,15aS)-14-(4- amino-7H-pyrrolo[2,3-d]pyrimidin-7-yl)-2,10- dihydroxy-2-oxido-10-sulfidooctahydro-12H-5,8- methanofuro[3,2-l][1,3,6,9,11,2,10] pentaoxadiphosphacyclotetradecin-7-yl]-1,9- dihydro-6H-purin-6-one (Diastereomer 1)::US11453697, Example 275::US11453697, Example 276	Stimulator of interferon genes protein [H232R]					 322					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574143	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574143&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177631	474496393							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1211112	Nc1nc2n(cnc2c(=O)[nH]1)[C@@H]1O[C@@H]2COP(O)(=O)O[C@H]3[C@H]4OC[C@]3(COP(O)(=S)O[C@@H]1[C@H]2F)O[C@H]4n1cnc2c(N)ncnc12			574145	2-amino-9-[(5R,7R,8S,12aR,14R,15R,15aS,18S)- 14-(6-amino-9H-purin-9-yl)-18-fluoro-2,10- dihydroxy-2-oxido-10-sulfindohexahydro-14H- 15,12a-(epoxymethano)-5,8-methanofuro[3,2- l][1,3,6,9,11,2,10]pentaoxadiphosphacyclotetra- decin-7(12H)-yl]-1,9-dihydro-6H-purin-6-one (Diastereomer 1)::US11453697, Example 277::US11453697, Example 278	Stimulator of interferon genes protein [H232R]					 28.7					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574145	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574145&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177632	474496394							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1211113	Nc1nc2n(cnc2c(=O)[nH]1)[C@@H]1O[C@@H]2COP(O)(=O)O[C@H]3[C@H]4OC[C@]3(COP(O)(=S)O[C@@H]1[C@H]2F)O[C@H]4n1cnc2c(N)ncnc12			574145	2-amino-9-[(5R,7R,8S,12aR,14R,15R,15aS,18S)- 14-(6-amino-9H-purin-9-yl)-18-fluoro-2,10- dihydroxy-2-oxido-10-sulfindohexahydro-14H- 15,12a-(epoxymethano)-5,8-methanofuro[3,2- l][1,3,6,9,11,2,10]pentaoxadiphosphacyclotetra- decin-7(12H)-yl]-1,9-dihydro-6H-purin-6-one (Diastereomer 1)::US11453697, Example 277::US11453697, Example 278	Stimulator of interferon genes protein [H232R]					 478					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574145	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574145&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177632	474496394							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1211114	Nc1nc2n(cnc2c(=O)[nH]1)[C@@H]1O[C@@H]2COP(O)(=O)O[C@@H]3[C@@H](COP(O)(=S)O[C@@H]1[C@@H]2F)O[C@H]([C@H]3F)n1nnc2c(N)ncnc12			574147	2-amino-9-[(5R,7R,8S,12aR,14R,15S,15aR,16R)- 14-(7-amino-3H-[1,2,3]triazolo[4,5-d]pyrimidin- 3-yl)-15,16-difluoro-2,10-dihydroxy-2-oxido-10- sulfidooctahydro-12H-5,8-methanofuro[3,2- l][1,3,6,9,11,2,10]pentaoxadiphosphacyclotetra- decin-7-yl]-1,9-dihydro-6H-purin-6-one (Diastereomer 1)::US11453697, Example 279::US11453697, Example 280	Stimulator of interferon genes protein [H232R]					 1235					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574147	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574147&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177633	474496395							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1211115	Nc1nc2n(cnc2c(=O)[nH]1)[C@@H]1O[C@@H]2COP(O)(=O)O[C@@H]3[C@@H](COP(O)(=S)O[C@@H]1[C@@H]2F)O[C@H]([C@H]3F)n1nnc2c(N)ncnc12			574147	2-amino-9-[(5R,7R,8S,12aR,14R,15S,15aR,16R)- 14-(7-amino-3H-[1,2,3]triazolo[4,5-d]pyrimidin- 3-yl)-15,16-difluoro-2,10-dihydroxy-2-oxido-10- sulfidooctahydro-12H-5,8-methanofuro[3,2- l][1,3,6,9,11,2,10]pentaoxadiphosphacyclotetra- decin-7-yl]-1,9-dihydro-6H-purin-6-one (Diastereomer 1)::US11453697, Example 279::US11453697, Example 280	Stimulator of interferon genes protein [H232R]					 1186					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574147	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574147&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177633	474496395							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1211116	Nc1nc2n(nnc2c(=O)[nH]1)[C@@H]1O[C@H]2C[C@H]1OP(O)(=S)OC[C@H]1O[C@H]([C@@H](F)[C@@H]1OP(O)(=O)OC2)n1ccc2c(N)ncnc12			574149	5-amino-3-[(5S,7R,8R,12aR,14R,15S,15aR)-14- (4-amino-7H-pyrrolo[2,3-d]pyrimidin-7-yl)-15- fluoro-2,10-dihydroxy-2-oxido-10- sulfidooctahydro-12H-5,8-methanofuro[3,2- l][1,3,6,9,11,2,10]pentaoxadiphosphacyclotetra- decin-7-yl]-3,6-dihydro-7H-[1,2,3]triazolo[4,5- d]pyrimidin-7-one::US11453697, Example 281	Stimulator of interferon genes protein [H232R]					 2485					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574149	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574149&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177634	474496396							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1211117	Nc1nc2n(nnc2c(=O)[nH]1)[C@@H]1O[C@@H]2COP(O)(=O)O[C@@H]3[C@@H](COP(O)(=S)O[C@@H]1[C@H]2F)O[C@H]([C@H]3F)n1nnc2c(N)ncnc12			574150	5-amino-3-[(5R,7R,8S,12aR,14R,15S,15aR,16S)- 14-(7-amino-3H-[1,2,3]triazolo[4,5-d]pyrimidin- 3-yl)-15,16-difluoro-2,10-dihydroxy-2-oxido-10- sulfidooctahydro-12H-5,8-methanofuro[3,2- l][1,3,6,9,11,2,10]pentaoxadiphosphacyclotetra- decin-7-yl]-3,6-dihydro-7H-[1,2,3]triazolo[4,5- d]pyrimidin-7-one::US11453697, Example 282	Stimulator of interferon genes protein [H232R]					 12190					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574150	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574150&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177635	474496397							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1211118	Nc1nc2n(cnc2c(=O)[nH]1)[C@@H]1O[C@H]2C[C@H]1OP(S)(=O)OC[C@H]1O[C@H](C[C@@H]1OP(O)(=O)OC2)c1cnc2c(N)ncnn12			574151	2-amino-9-[(5S,7R,8R,12aR,14R,15aS)-14-(4- aminoimidazo[2,1-f][1,2,4]triazin-7-yl)-2- hydroxy-2,10-dioxido-10-sulfanyloctahydro-12H- 5,8-methanofuro[3,2-1][1,3,6,9,11,2,10] pentaoxadiphosphacyclotetradecin-7-yl]-1,9- dihydro-6H-purin-6-one::US11453697, Example 283	Stimulator of interferon genes protein [H232R]					 17.2					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574151	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574151&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177636	474496398							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1211119	Nc1nc2n(cnc2c(=O)[nH]1)[C@@H]1S[C@@H]2COP(O)(=O)O[C@H]3[C@H]4OC[C@]3(COP(O)(=S)O[C@@H]1[C@H]2F)O[C@H]4n1cnc2c(N)ncnc12			574152	2-amino-9-[(5R,7R,8R,12aR,14R,15R,15aS,18R)- 14-(6-amino-9H-purin-9-yl)-18-fluoro-2,10- dihydroxy-2-oxido-10-sulfidohexahydro-14H- 15,12a-(epoxymethano)-5,8-methanofuro[3,2- l][1,3,9,11,6,2,10]tetraoxathiadiphosphacyclo- tetradecin-7(12H)-yl]-1,9-dihydro-6H-purin-6- one::US11453697, Example 284	Stimulator of interferon genes protein [H232R]					 128					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574152	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574152&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177637	474496399							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1211120	Nc1nc2n(cnc2c(=O)[nH]1)[C@@H]1S[C@@H]2COP(O)(=O)O[C@@H]3[C@@H](COP(S)(=O)O[C@@H]1[C@H]2F)O[C@H]([C@H]3F)n1nnc2c(N)ncnc12			574153	2-amino-9-[(5R,7R,8R,12aR,14R,15S,15aR,16R)- 14-(7-amino-3H-[1,2,3]triazolo[4,5-d]pyrimidin- 3-yl)-15,16-difluoro-2-hydroxy-2,10-dioxido-10- sulfanyloctahydro-12H-5,8-methanofuro[3,2- l][1,3,9,11,6,2,10]tetraoxathiadiphosphacyclo- tetradecin-7-yl]-1,9-dihydro-6H-purin-6-one::US11453697, Example 285	Stimulator of interferon genes protein [H232R]					 277					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574153	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574153&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177638	474496400							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1211121	Nc1nc2n(cnc2c(=O)[nH]1)[C@@H]1S[C@@H]2COP(O)(=O)O[C@@H]3[C@@H](COP(S)(=O)O[C@@H]1[C@H]2F)O[C@H]([C@H]3F)n1cnc2c(N)ccnc12			574154	2-amino-9-[(5R,7R,8R,12aR,14R,15S,15aR,16R)- 14-(7-amino-3H-imidazo[4,5-b]pyridin-3-yl)- 15,16-difluoro-2-hydroxy-2,10-dioxido-10- sulfanyloctahydro-12H-5,8-methanofuro[3,2- l][1,3,9,11,6,2,10]tetraoxathiadiphosphacyclo- tetradecin-7-yl]-1,9-dihydro-6H-purin-6-one (Diastereomer 1)::US11453697, Example 286::US11453697, Example 287	Stimulator of interferon genes protein [H232R]					 4010					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574154	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574154&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177639	474496401							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1211122	Nc1nc2n(cnc2c(=O)[nH]1)[C@@H]1S[C@@H]2COP(O)(=O)O[C@@H]3[C@@H](COP(S)(=O)O[C@@H]1[C@H]2F)O[C@H]([C@H]3F)n1cnc2c(N)ccnc12			574154	2-amino-9-[(5R,7R,8R,12aR,14R,15S,15aR,16R)- 14-(7-amino-3H-imidazo[4,5-b]pyridin-3-yl)- 15,16-difluoro-2-hydroxy-2,10-dioxido-10- sulfanyloctahydro-12H-5,8-methanofuro[3,2- l][1,3,9,11,6,2,10]tetraoxathiadiphosphacyclo- tetradecin-7-yl]-1,9-dihydro-6H-purin-6-one (Diastereomer 1)::US11453697, Example 286::US11453697, Example 287	Stimulator of interferon genes protein [H232R]					 80.2					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574154	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574154&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177639	474496401							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1211123	Nc1nc2n(cnc2c(=O)[nH]1)[C@@H]1S[C@@H]2COP(O)(=O)O[C@@H]3[C@@H](COP(S)(=O)O[C@@H]1[C@H]2F)O[C@@H](n1nnc2c(N)ncnc12)C3(F)F			574156	2-amino-9-[(5R,7R,8R,12aR,14R,15aR,16R)-14- (7-amino-3H-[1,2,3]triazolo[4,5-d]pyrimidin-3- yl)-15,15,16-trifluoro-2-hydroxy-2,10-dioxido- 10-sulfanyloctahydro-12H-5,8-methanofuro[3,2- l][1,3,9,11,6,2,10]tetraoxathiadiphosphacyclo- tetradecin-7-yl]-1,9-dihydro-6H-purin-6-one::US11453697, Example 288	Stimulator of interferon genes protein [H232R]					 24.9					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574156	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574156&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177640	474496402							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1211124	Nc1nc2n(cnc2c(=O)[nH]1)[C@@H]1O[C@@H]2COP(O)(=O)O[C@@H]3[C@@H](COP(O)(=S)O[C@@H]1[C@@H]2F)O[C@H]([C@@H]3F)n1cnc2c(N)ncnc12			574157	US11453697, Example 289	Stimulator of interferon genes protein [H232R]					 5.30					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574157	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574157&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177641	474496403							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1211125	Nc1nc2n(cnc2c(=O)[nH]1)[C@@H]1O[C@@H]2CO[P@](S)(=O)O[C@@H]3[C@@H](CO[P@](S)(=O)O[C@@H]1[C@@H]2F)O[C@H]([C@H]3F)n1cnc2c1nc[nH]c2=O			573990	2-amino-9-[(2R,5R,7R,8S,10R, 12aR,14R,15S,15aR,16R)-15,16-difluoro- 2,10-dihydroxy-14-(6-oxo-1,6-dihydro- 9H-purin-9-yl)-2,10-disulfidooctahydro- 12H-5,8-methanofuro[3,2- l][1,3,6,9,11,2,10] pentaoxadiphosphacyclotetradecin-7-yl]- 1,9-dihydro-6H-purin-6-one (Diastereomer 1)::US11453697, Example 308	Stimulator of interferon genes protein [H232R]					 3.30					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=573990	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=573990&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177553	474496316							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1211126	Nc1nc2n(cnc2c(=O)[nH]1)[C@@H]1S[C@@H]2CO[P@](S)(=O)O[C@@H]3[C@@H](CO[P@](S)(=O)O[C@@H]1[C@@H]2O)O[C@H]([C@H]3F)n1cnc2c1nc[nH]c2=O			574158	2-amino-9-[(2R,5R,7R,8R,10R, 12aR,14R,15S,15aR,16S)-15-fluoro-16- hydroxy-2,10-dioxido-14-(6-oxo-1,6- dihydro-9H-purin-9-yl)-2,10- disulfanyloctahydro-12H-5,8- methanofuro[3,2-l][1,3,9,11,6,2,10] tetraoxathiadiphosphacyclotetradecin-7- yl]-1,9-dihydro-6H-purin-6-one (Diastereomer 1)::US11453697, Example 323	Stimulator of interferon genes protein [H232R]					 3.70					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574158	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574158&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177642	474496404							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1211127	Nc1nc2n(cnc2c(=O)[nH]1)[C@@H]1S[C@@H]2COP(S)(=O)O[C@@H]3[C@@H](COP(S)(=O)O[C@@H]1[C@@H]2O)O[C@H]([C@H]3F)n1cnc2c1nc[nH]c2=O			574159	2-amino-9-[(5R,7R,8R,12aR,14R,15S, 15aR,16S)-15-fluoro-16-hydroxy-2,10- dioxido-14-(6-oxo-1,6-dihydro-9H-purin- 9-yl)-2,10-disulfanyloctahydro-12H-5,8- methanofuro[3,2-l][1,3,9,11,6,2,10] tetraoxathiadiphosphacyclotetradecin-7- yl]-1,9-dihydro-6H-purin-6-one (Diastereomer 2)::US11453697, Example 324::US11453697, Example 325	Stimulator of interferon genes protein [H232R]					 10.7					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574159	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574159&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177642	474496405							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1211128	Nc1nc2n(cnc2c(=O)[nH]1)[C@@H]1S[C@@H]2COP(S)(=O)O[C@@H]3[C@@H](COP(S)(=O)O[C@@H]1[C@@H]2O)O[C@H]([C@H]3F)n1cnc2c1nc[nH]c2=O			574159	2-amino-9-[(5R,7R,8R,12aR,14R,15S, 15aR,16S)-15-fluoro-16-hydroxy-2,10- dioxido-14-(6-oxo-1,6-dihydro-9H-purin- 9-yl)-2,10-disulfanyloctahydro-12H-5,8- methanofuro[3,2-l][1,3,9,11,6,2,10] tetraoxathiadiphosphacyclotetradecin-7- yl]-1,9-dihydro-6H-purin-6-one (Diastereomer 2)::US11453697, Example 324::US11453697, Example 325	Stimulator of interferon genes protein [H232R]					 866					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574159	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574159&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177642	474496405							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1211129	Nc1nc2n(cnc2c(=O)[nH]1)[C@@H]1O[C@@H]2COP(S)(=O)O[C@@H]3[C@@H](COP(S)(=O)O[C@@H]1[C@@H]2O)O[C@H]([C@H]3F)n1nnc2c1nc[nH]c2=O			574161	3-[(5R,7R,8S,12aR,14R,15S,15aR,16R)- 7-(2-amino-6-oxo-1,6-dihydro-9H-purin- 9-yl)-15,16-difluoro-2,10-dioxido-2,10- disulfanyloctahydro-12H-5,8- methanofuro[3,2-l][1,3,6,9,11,2,10] pentaoxadiphosphacyclotetradecin-14-yl]- 3,6-dihydro-7H-[1,2,3]triazolo[4,5- d]pyrimidin-7-one (Diastereomer 1)::US11453697, Example 326	Stimulator of interferon genes protein [H232R]					 89.7					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574161	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574161&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177643	474496406							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1211130	Nc1nc2n(cnc2c(=O)[nH]1)[C@@H]1O[C@@H]2COP(S)(=O)O[C@@H]3[C@@H](COP(S)(=O)O[C@@H]1[C@@H]2F)O[C@H]([C@H]3F)n1nnc2c1nc[nH]c2=O			574162	3-[(5R,7R,8S,12aR,14R,15S,15aR,16R)- 7-(2-amino-6-oxo-1,6-dihydro-9H-purin- 9-yl)-15,16-difluoro-2,10-dioxido-2,10- disulfanyloctahydro-12H-5,8- methanofuro[3,2-l][1,3,6,9,11,2,10] pentaoxadiphosphacyclotetradecin-14-yl]- 3,6-dihydro-7H-[1,2,3]triazolo[4,5- d]pyrimidin-7-one (Diastereomer 2)::US11453697, Example 327::US11453697, Example 328	Stimulator of interferon genes protein [H232R]					 14.0					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574162	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574162&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177644	474496407							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1211131	Nc1nc2n(cnc2c(=O)[nH]1)[C@@H]1O[C@@H]2COP(S)(=O)O[C@@H]3[C@@H](COP(S)(=O)O[C@@H]1[C@@H]2F)O[C@H]([C@H]3F)n1nnc2c1nc[nH]c2=O			574162	3-[(5R,7R,8S,12aR,14R,15S,15aR,16R)- 7-(2-amino-6-oxo-1,6-dihydro-9H-purin- 9-yl)-15,16-difluoro-2,10-dioxido-2,10- disulfanyloctahydro-12H-5,8- methanofuro[3,2-l][1,3,6,9,11,2,10] pentaoxadiphosphacyclotetradecin-14-yl]- 3,6-dihydro-7H-[1,2,3]triazolo[4,5- d]pyrimidin-7-one (Diastereomer 2)::US11453697, Example 327::US11453697, Example 328	Stimulator of interferon genes protein [H232R]					 74.4					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574162	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574162&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177644	474496407							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1211132	Nc1nc2n(cnc2c(=O)[nH]1)[C@@H]1O[C@@H]2CO[P@](S)(=O)O[C@@H]3[C@@H](CO[P@](S)(=O)O[C@@H]1[C@H]2F)O[C@H]([C@H]3F)n1cnc2c1nc[nH]c2=O			574164	2-amino-9-[(2R,5R,7R,8S,10R, 12aR,14R,15S,15aR,16S)-15,16-difluoro- 2,10-dioxido-14-(6-oxo-1,6-dihydro-9H- purin-9-yl)-2,10-disulfanyloctahydro- 12H-5,8-methanofuro[3,2- l][1,3,6,9,11,2,10] pentaoxadiphosphacyclotetradecin-7-yl]- 1,9-dihydro-6H-purin-6-one (Diastereomer 1)::US11453697, Example 329	Stimulator of interferon genes protein [H232R]					 31.7					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574164	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574164&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177645	474496408							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1211133	Nc1nc2n(cnc2c(=O)[nH]1)[C@@H]1O[C@@H]2COP(S)(=O)O[C@@H]3[C@@H](COP(S)(=O)O[C@@H]1[C@H]2F)O[C@H]([C@H]3F)n1cnc2c1nc[nH]c2=O			574165	2-amino-9-[(5R,7R,8S,12aR,14R,15S, 15aR,16S)-15,16-difluoro-2,10-dioxido- 14-(6-oxo-1,6-dihydro-9H-purin-9-yl)- 2,10-disulfanyloctahydro-12H-5,8- methanofuro[3,2-l][1,3,6,9,11,2,10] pentaoxadiphosphacyclotetradecin-7-yl]- 1,9-dihydro-6H-purin-6-one (Diastereomer 2)::US11453697, Example 330	Stimulator of interferon genes protein [H232R]					 204					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574165	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574165&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177645	474496409							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1211134	Nc1nc2n(cnc2c(=O)[nH]1)[C@@H]1O[C@@H]2COP(S)(=O)O[C@@H]3[C@@H](COP(S)(=O)O[C@@H]1[C@H]2F)O[C@H]([C@H]3F)n1nnc2c1nc[nH]c2=O			574166	3-[(5R,7R,8S,12aR,14R,15S,15aR,16S)- 7-(2-amino-6-oxo-1,6-dihydro-9H-purin- 9-yl)-15,16-difluoro-2,10-dioxido-2,10- disulfanyloctahydro-12H-5,8- methanofuro[3,2-l][1,3,6,9,11,2,10] pentaoxadiphosphacyclotetradecin-14-yl]- 3,6-dihydro-7H-[1,2,3]triazolo[4,5- d]pyrimidin-7-one::US11453697, Example 331	Stimulator of interferon genes protein [H232R]					 183					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574166	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574166&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177646	474496410							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1211135	Nc1nc2n(cnc2c(=O)[nH]1)[C@@H]1O[C@@H]2COP(S)(=O)O[C@@H]3[C@@H](COP([O-])(=O)O[C@@H]1[C@@H]2O)O[C@H]([C@@H]3O)n1cnc2c1nc[nH]c2=O			574167	2-amino-9- [(5R,7R,8R,12ar,14R,15R,15aS,16R)- 10,15,16-trihydroxy-2,10-dioxido-14-(6- oxo-1,6-dihydro-9H-purin-9-yl)-2- sulfanyloctahydro-12H-5,8- methanofuro[3,2-l][1,3,6,9,11,2,10] pentaoxadiphosphacyclotetradecin-7-yl]- 1,9-dihydro-6H-purin-6-one::US11453697, Example 334	Stimulator of interferon genes protein [H232R]					 110					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574167	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574167&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177647	474496411							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1211136	Nc1nc2n(cnc2c(=O)[nH]1)[C@@H]1O[C@@H]2COP(S)(=O)O[C@@H]3[C@@H](COP(S)(=O)O[C@@H]1[C@@H]2F)O[C@H]([C@@H]3F)n1cnc2c1nc[nH]c2=O			574168	2-amino-9- [(5R,7R,8S,12aR,14R,15R,15aR,16R)- 15,16-difluoro-2,10-dioxido-14-(6-oxo- 1,6-dihydro-9H-purin-9-yl)-2,10- disulfanyloctahydro-12H-5,8- methanofuro[3,2-l][1,3,6,9,11,2,10] pentaoxadiphosphacyclotetradecin-7-yl]- 1,9-dihydro-6H-purin-6-one::US11453697, Example 335	Stimulator of interferon genes protein [H232R]					 5.20					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574168	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574168&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177649	474496412							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1211137	Nc1nc2n(cnc2c(=O)[nH]1)[C@@H]1O[C@@H]2COP(S)(=O)O[C@H]3C[C@@H](O[C@@H]3COP(O)(=O)O[C@@H]1[C@@H]2F)c1cnc2n1nc[nH]c2=O			574169	7-[(5R,7R,8S,12aR,14R,15aS,16R)-7-(2- amino-6-oxo-1,6-dihydro-9H-purin-9-yl)- 16-fluoro-2,10-dioxido-2,10- disulfanyloctahydro-12H-5,8- methanofuro[3,2-l][1,3,6,9,11,2,10] pentaoxadiphosphacyclotetradecin-14- yl]imidazo[2,1-f][1,2,4]triazin-4(3H)-one (Diastereomer 1)::US11453697, Example 336	Stimulator of interferon genes protein [H232R]					 422					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574169	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574169&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177650	474496413							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1211138	Nc1nc2n(cnc2c(=O)[nH]1)[C@@H]1O[C@@H]2COP(S)(=O)O[C@@H]3[C@@H](COP(S)(=O)O[C@@H]1[C@@H]2F)O[C@@H](n1nnc2c1nc[nH]c2=O)C3(F)F			574170	3-[5R,7R,8S,12aR,14R,15aR,16R)-7-(2- amino-6-oxo-1,6-dihydro-9H-purin-9-yl)- 15,15,16-trifluoro-2,10-dioxido-2,10- disulfanyloctahydro-12H-5,8- methanofuro[3,2-l][1,3,6,9,11,2,10] pentaoxadiphosphacyclotetradecin-14-yl]- 3,6-dihydro-7H-[1,2,3]triazolo[4,5- d]pyrimidin-7-one (Diastereomer 1)::US11453697, Example 337::US11453697, Example 338	Stimulator of interferon genes protein [H232R]					 29.2					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574170	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574170&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177651	474496414							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1211139	Nc1nc2n(cnc2c(=O)[nH]1)[C@@H]1O[C@@H]2COP(S)(=O)O[C@@H]3[C@@H](COP(S)(=O)O[C@@H]1[C@@H]2F)O[C@@H](n1nnc2c1nc[nH]c2=O)C3(F)F			574170	3-[5R,7R,8S,12aR,14R,15aR,16R)-7-(2- amino-6-oxo-1,6-dihydro-9H-purin-9-yl)- 15,15,16-trifluoro-2,10-dioxido-2,10- disulfanyloctahydro-12H-5,8- methanofuro[3,2-l][1,3,6,9,11,2,10] pentaoxadiphosphacyclotetradecin-14-yl]- 3,6-dihydro-7H-[1,2,3]triazolo[4,5- d]pyrimidin-7-one (Diastereomer 1)::US11453697, Example 337::US11453697, Example 338	Stimulator of interferon genes protein [H232R]					 442					US Patent		10.7270/Q29G5R24			US11453697	Altman, MD; Andresen, B; Chang, W; Cumming, JN; Otte, RD; Trotter, BW	Merck Sharp & Dohme LLC	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574170	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574170&enzyme=Stimulator+of+interferon+genes+protein+%5BH232R%5D&column=ki&startPg=0&Increment=50&submit=Search			166177651	474496414							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1211937	CN1CCN(CC1)c1ccc(c(NC(c2ccccc2)c2ccccc2)c1)[N+]([O-])=O	InChI=1S/C24H26N4O2/c1-26-14-16-27(17-15-26)21-12-13-23(28(29)30)22(18-21)25-24(19-8-4-2-5-9-19)20-10-6-3-7-11-20/h2-13,18,24-25H,14-17H2,1H3	RHCKSABVOKGXBN-UHFFFAOYSA-N	50223308	CHEMBL398481::N-benzhydryl-5-(4-methylpiperazin-1-yl)-2-nitrobenzenamine::US11459308, Compound PPZ-1	Envelope glycoprotein			 2300							US Patent		10.7270/Q28G8PXB		aid1806861	US11459308	Bowlin, TL; Moir, DT; Chandran, K; Dye, Jr., JM; Williams, JD; Aron, ZD; Barbor, JP; Lively, KN; Nash, PJ; Mills, DM; Basu, A	Microbiotix, Inc.; Albert Einstein College of Medicine; The Government of the United States as Represented by the Secretary of the Army	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50223308	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Envelope+glycoprotein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50223308&enzyme=Envelope+glycoprotein&column=ki&startPg=0&Increment=50&submit=Search			5206725	104095403		CHEMBL398481				ZINC04687377	1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1211939	CCN1CCN(CC1)c1ccc(c(NC(c2ccccc2)c2ccccc2)c1)[N+]([O-])=O	InChI=1S/C25H28N4O2/c1-2-27-15-17-28(18-16-27)22-13-14-24(29(30)31)23(19-22)26-25(20-9-5-3-6-10-20)21-11-7-4-8-12-21/h3-14,19,25-26H,2,15-18H2,1H3	VIERHBZALJXRHK-UHFFFAOYSA-N	574746	US11459308, Compound 3556	Envelope glycoprotein			 1100							US Patent		10.7270/Q28G8PXB		aid1806861	US11459308	Bowlin, TL; Moir, DT; Chandran, K; Dye, Jr., JM; Williams, JD; Aron, ZD; Barbor, JP; Lively, KN; Nash, PJ; Mills, DM; Basu, A	Microbiotix, Inc.; Albert Einstein College of Medicine; The Government of the United States as Represented by the Secretary of the Army	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574746	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Envelope+glycoprotein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574746&enzyme=Envelope+glycoprotein&column=ki&startPg=0&Increment=50&submit=Search			134589372	474496975							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1211941	[O-][N+](=O)c1ccc(cc1NC(c1ccccc1)c1ccccc1)N1CCN(Cc2ccccn2)CC1	InChI=1S/C29H29N5O2/c35-34(36)28-15-14-26(33-19-17-32(18-20-33)22-25-13-7-8-16-30-25)21-27(28)31-29(23-9-3-1-4-10-23)24-11-5-2-6-12-24/h1-16,21,29,31H,17-20,22H2	VTHOXIMMPRLARD-UHFFFAOYSA-N	574747	US11459308, Compound 3557	Envelope glycoprotein			 1900							US Patent		10.7270/Q28G8PXB		aid1806861	US11459308	Bowlin, TL; Moir, DT; Chandran, K; Dye, Jr., JM; Williams, JD; Aron, ZD; Barbor, JP; Lively, KN; Nash, PJ; Mills, DM; Basu, A	Microbiotix, Inc.; Albert Einstein College of Medicine; The Government of the United States as Represented by the Secretary of the Army	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574747	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Envelope+glycoprotein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574747&enzyme=Envelope+glycoprotein&column=ki&startPg=0&Increment=50&submit=Search			134589550	474496976							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1211943	CN1CCN(CC1)c1cccc(NC(c2ccccc2)c2ccccc2)c1	InChI=1S/C24H27N3/c1-26-15-17-27(18-16-26)23-14-8-13-22(19-23)25-24(20-9-4-2-5-10-20)21-11-6-3-7-12-21/h2-14,19,24-25H,15-18H2,1H3	NTBJJPBUCDLXTC-UHFFFAOYSA-N	574748	US11459308, Compound 3566::US11459308, Compound 3567	Envelope glycoprotein			 1600							US Patent		10.7270/Q28G8PXB		aid1806861	US11459308	Bowlin, TL; Moir, DT; Chandran, K; Dye, Jr., JM; Williams, JD; Aron, ZD; Barbor, JP; Lively, KN; Nash, PJ; Mills, DM; Basu, A	Microbiotix, Inc.; Albert Einstein College of Medicine; The Government of the United States as Represented by the Secretary of the Army	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574748	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Envelope+glycoprotein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574748&enzyme=Envelope+glycoprotein&column=ki&startPg=0&Increment=50&submit=Search			134589427	474496977							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1211945	[O-][N+](=O)c1ccc(cc1NC(c1ccccc1)c1ccccc1)N1CCN(Cc2ccncc2)CC1	InChI=1S/C29H29N5O2/c35-34(36)28-12-11-26(33-19-17-32(18-20-33)22-23-13-15-30-16-14-23)21-27(28)31-29(24-7-3-1-4-8-24)25-9-5-2-6-10-25/h1-16,21,29,31H,17-20,22H2	FHLGAQISFMBCSG-UHFFFAOYSA-N	574749	US11459308, Compound 3561	Envelope glycoprotein			 1700							US Patent		10.7270/Q28G8PXB		aid1806861	US11459308	Bowlin, TL; Moir, DT; Chandran, K; Dye, Jr., JM; Williams, JD; Aron, ZD; Barbor, JP; Lively, KN; Nash, PJ; Mills, DM; Basu, A	Microbiotix, Inc.; Albert Einstein College of Medicine; The Government of the United States as Represented by the Secretary of the Army	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574749	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Envelope+glycoprotein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574749&enzyme=Envelope+glycoprotein&column=ki&startPg=0&Increment=50&submit=Search			134589580	474496978							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1211947	C\C=C\CN1CCN(CC1)c1ccc(c(NC(c2ccccc2)c2ccccc2)c1)[N+]([O-])=O	InChI=1S/C27H30N4O2/c1-2-3-16-29-17-19-30(20-18-29)24-14-15-26(31(32)33)25(21-24)28-27(22-10-6-4-7-11-22)23-12-8-5-9-13-23/h2-15,21,27-28H,16-20H2,1H3/b3-2+	MSQGMYALMIGNTR-NSCUHMNNSA-N	574750	US11459308, Compound 3559	Envelope glycoprotein			 1700							US Patent		10.7270/Q28G8PXB		aid1806861	US11459308	Bowlin, TL; Moir, DT; Chandran, K; Dye, Jr., JM; Williams, JD; Aron, ZD; Barbor, JP; Lively, KN; Nash, PJ; Mills, DM; Basu, A	Microbiotix, Inc.; Albert Einstein College of Medicine; The Government of the United States as Represented by the Secretary of the Army	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574750	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Envelope+glycoprotein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574750&enzyme=Envelope+glycoprotein&column=ki&startPg=0&Increment=50&submit=Search			134589044	474496979							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1211949	CN1CCN(CC1)c1ccc(c(NC(c2ccccc2)c2ccccc2C)c1)[N+]([O-])=O	InChI=1S/C25H28N4O2/c1-19-8-6-7-11-22(19)25(20-9-4-3-5-10-20)26-23-18-21(12-13-24(23)29(30)31)28-16-14-27(2)15-17-28/h3-13,18,25-26H,14-17H2,1-2H3	XXEPDKCWDKKNHY-UHFFFAOYSA-N	574751	US11459308, Compound 3625	Envelope glycoprotein			 780							US Patent		10.7270/Q28G8PXB		aid1806861	US11459308	Bowlin, TL; Moir, DT; Chandran, K; Dye, Jr., JM; Williams, JD; Aron, ZD; Barbor, JP; Lively, KN; Nash, PJ; Mills, DM; Basu, A	Microbiotix, Inc.; Albert Einstein College of Medicine; The Government of the United States as Represented by the Secretary of the Army	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574751	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Envelope+glycoprotein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574751&enzyme=Envelope+glycoprotein&column=ki&startPg=0&Increment=50&submit=Search			134589581	474496980							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1211951	[O-][N+](=O)c1ccc(cc1NC(c1ccccc1)c1ccccc1)N1CCN(CC1)C1Cc2ccccc2C1	InChI=1S/C32H32N4O2/c37-36(38)31-16-15-28(34-17-19-35(20-18-34)29-21-26-13-7-8-14-27(26)22-29)23-30(31)33-32(24-9-3-1-4-10-24)25-11-5-2-6-12-25/h1-16,23,29,32-33H,17-22H2	ARABTHWZDHPVJF-UHFFFAOYSA-N	574752	US11459308, Compound 3589	Envelope glycoprotein			 8000							US Patent		10.7270/Q28G8PXB		aid1806861	US11459308	Bowlin, TL; Moir, DT; Chandran, K; Dye, Jr., JM; Williams, JD; Aron, ZD; Barbor, JP; Lively, KN; Nash, PJ; Mills, DM; Basu, A	Microbiotix, Inc.; Albert Einstein College of Medicine; The Government of the United States as Represented by the Secretary of the Army	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574752	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Envelope+glycoprotein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574752&enzyme=Envelope+glycoprotein&column=ki&startPg=0&Increment=50&submit=Search			134589623	474496981							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1211953	CN1CCN(CC1)c1ccnc(NC(c2ccccc2)c2ccccc2)c1	InChI=1S/C23H26N4/c1-26-14-16-27(17-15-26)21-12-13-24-22(18-21)25-23(19-8-4-2-5-9-19)20-10-6-3-7-11-20/h2-13,18,23H,14-17H2,1H3,(H,24,25)	TYXYYADCDOAZFU-UHFFFAOYSA-N	574753	US11459308, Compound 3580::US11459308, Compound 3586	Envelope glycoprotein			 2700							US Patent		10.7270/Q28G8PXB		aid1806861	US11459308	Bowlin, TL; Moir, DT; Chandran, K; Dye, Jr., JM; Williams, JD; Aron, ZD; Barbor, JP; Lively, KN; Nash, PJ; Mills, DM; Basu, A	Microbiotix, Inc.; Albert Einstein College of Medicine; The Government of the United States as Represented by the Secretary of the Army	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574753	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Envelope+glycoprotein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574753&enzyme=Envelope+glycoprotein&column=ki&startPg=0&Increment=50&submit=Search			134588755	474496982							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1211955	[O-][N+](=O)c1ccc(cc1NC(c1ccccc1)c1ccccc1)N1CCN(CC1)C1CCC1	InChI=1S/C27H30N4O2/c32-31(33)26-15-14-24(30-18-16-29(17-19-30)23-12-7-13-23)20-25(26)28-27(21-8-3-1-4-9-21)22-10-5-2-6-11-22/h1-6,8-11,14-15,20,23,27-28H,7,12-13,16-19H2	LHSCAJJYNBJTRS-UHFFFAOYSA-N	574754	US11459308, Compound 3588	Envelope glycoprotein			 730							US Patent		10.7270/Q28G8PXB		aid1806861	US11459308	Bowlin, TL; Moir, DT; Chandran, K; Dye, Jr., JM; Williams, JD; Aron, ZD; Barbor, JP; Lively, KN; Nash, PJ; Mills, DM; Basu, A	Microbiotix, Inc.; Albert Einstein College of Medicine; The Government of the United States as Represented by the Secretary of the Army	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574754	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Envelope+glycoprotein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574754&enzyme=Envelope+glycoprotein&column=ki&startPg=0&Increment=50&submit=Search			134588727	474496983							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1211957	[O-][N+](=O)c1ccc(cc1NC(c1ccccc1)c1ccccc1)N1CCN(Cc2ccc(cc2)N=[N+]=[N-])CC1	InChI=1S/C30H29N7O2/c31-34-33-26-13-11-23(12-14-26)22-35-17-19-36(20-18-35)27-15-16-29(37(38)39)28(21-27)32-30(24-7-3-1-4-8-24)25-9-5-2-6-10-25/h1-16,21,30,32H,17-20,22H2	INXTXEGJKWLMSE-UHFFFAOYSA-N	574755	US11459308, Compound 3610	Envelope glycoprotein			 600							US Patent		10.7270/Q28G8PXB		aid1806861	US11459308	Bowlin, TL; Moir, DT; Chandran, K; Dye, Jr., JM; Williams, JD; Aron, ZD; Barbor, JP; Lively, KN; Nash, PJ; Mills, DM; Basu, A	Microbiotix, Inc.; Albert Einstein College of Medicine; The Government of the United States as Represented by the Secretary of the Army	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574755	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Envelope+glycoprotein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574755&enzyme=Envelope+glycoprotein&column=ki&startPg=0&Increment=50&submit=Search			134588889	474496984							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1211959	[O-][N+](=O)c1ccc(cc1NC(c1ccccc1)c1ccccc1)N1CCN(CC1)C1CCc2ccccc2C1	InChI=1S/C33H34N4O2/c38-37(39)32-18-17-30(24-31(32)34-33(26-10-3-1-4-11-26)27-12-5-2-6-13-27)36-21-19-35(20-22-36)29-16-15-25-9-7-8-14-28(25)23-29/h1-14,17-18,24,29,33-34H,15-16,19-23H2	JSFNEBZREBTIBG-UHFFFAOYSA-N	574756	US11459308, Compound 3591	Envelope glycoprotein			 1400							US Patent		10.7270/Q28G8PXB		aid1806861	US11459308	Bowlin, TL; Moir, DT; Chandran, K; Dye, Jr., JM; Williams, JD; Aron, ZD; Barbor, JP; Lively, KN; Nash, PJ; Mills, DM; Basu, A	Microbiotix, Inc.; Albert Einstein College of Medicine; The Government of the United States as Represented by the Secretary of the Army	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574756	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Envelope+glycoprotein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574756&enzyme=Envelope+glycoprotein&column=ki&startPg=0&Increment=50&submit=Search			134589124	474496985							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1211961	[O-][N+](=O)c1ccc(cc1NC(c1ccccc1)c1ccccc1)N1CCN(CC2CC2)CC1	InChI=1S/C27H30N4O2/c32-31(33)26-14-13-24(30-17-15-29(16-18-30)20-21-11-12-21)19-25(26)28-27(22-7-3-1-4-8-22)23-9-5-2-6-10-23/h1-10,13-14,19,21,27-28H,11-12,15-18,20H2	CECABLDBCWYYBO-UHFFFAOYSA-N	574757	US11459308, Compound 3612	Envelope glycoprotein			<600							US Patent		10.7270/Q28G8PXB		aid1806861	US11459308	Bowlin, TL; Moir, DT; Chandran, K; Dye, Jr., JM; Williams, JD; Aron, ZD; Barbor, JP; Lively, KN; Nash, PJ; Mills, DM; Basu, A	Microbiotix, Inc.; Albert Einstein College of Medicine; The Government of the United States as Represented by the Secretary of the Army	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574757	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Envelope+glycoprotein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574757&enzyme=Envelope+glycoprotein&column=ki&startPg=0&Increment=50&submit=Search			134588886	474496986							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1211965	CN1CCN(CC1)c1ccc(c(NC(c2ccccc2)c2ccccc2)c1)[N+]([O-])=O	InChI=1S/C24H26N4O2/c1-26-14-16-27(17-15-26)21-12-13-23(28(29)30)22(18-21)25-24(19-8-4-2-5-9-19)20-10-6-3-7-11-20/h2-13,18,24-25H,14-17H2,1H3	RHCKSABVOKGXBN-UHFFFAOYSA-N	50223308	CHEMBL398481::N-benzhydryl-5-(4-methylpiperazin-1-yl)-2-nitrobenzenamine::US11459308, Compound PPZ-1	Envelope glycoprotein			 2300							US Patent		10.7270/Q28G8PXB		aid1806861	US11459308	Bowlin, TL; Moir, DT; Chandran, K; Dye, Jr., JM; Williams, JD; Aron, ZD; Barbor, JP; Lively, KN; Nash, PJ; Mills, DM; Basu, A	Microbiotix, Inc.; Albert Einstein College of Medicine; The Government of the United States as Represented by the Secretary of the Army	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50223308	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Envelope+glycoprotein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50223308&enzyme=Envelope+glycoprotein&column=ki&startPg=0&Increment=50&submit=Search			5206725	104095403		CHEMBL398481				ZINC04687377	1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1211968	[O-][N+](=O)c1ccc(cc1NC(c1ccccc1)c1ccccc1)N1CCN(Cc2ccoc2)CC1	InChI=1S/C28H28N4O3/c33-32(34)27-12-11-25(31-16-14-30(15-17-31)20-22-13-18-35-21-22)19-26(27)29-28(23-7-3-1-4-8-23)24-9-5-2-6-10-24/h1-13,18-19,21,28-29H,14-17,20H2	OXFOYPGTILYVLX-UHFFFAOYSA-N	574762	US11459308, Compound 3569	Envelope glycoprotein			>20000							US Patent		10.7270/Q28G8PXB		aid1806861	US11459308	Bowlin, TL; Moir, DT; Chandran, K; Dye, Jr., JM; Williams, JD; Aron, ZD; Barbor, JP; Lively, KN; Nash, PJ; Mills, DM; Basu, A	Microbiotix, Inc.; Albert Einstein College of Medicine; The Government of the United States as Represented by the Secretary of the Army	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574762	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Envelope+glycoprotein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574762&enzyme=Envelope+glycoprotein&column=ki&startPg=0&Increment=50&submit=Search			134589683	474496991							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1211971	CCCCN1CCN(CC1)c1ccc(c(NC(c2ccccc2)c2ccccc2)c1)[N+]([O-])=O	InChI=1S/C27H32N4O2/c1-2-3-16-29-17-19-30(20-18-29)24-14-15-26(31(32)33)25(21-24)28-27(22-10-6-4-7-11-22)23-12-8-5-9-13-23/h4-15,21,27-28H,2-3,16-20H2,1H3	NAWCTRPJTBASRP-UHFFFAOYSA-N	574764	US11459308, Compound 3558	Envelope glycoprotein			 2800							US Patent		10.7270/Q28G8PXB		aid1806861	US11459308	Bowlin, TL; Moir, DT; Chandran, K; Dye, Jr., JM; Williams, JD; Aron, ZD; Barbor, JP; Lively, KN; Nash, PJ; Mills, DM; Basu, A	Microbiotix, Inc.; Albert Einstein College of Medicine; The Government of the United States as Represented by the Secretary of the Army	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574764	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Envelope+glycoprotein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574764&enzyme=Envelope+glycoprotein&column=ki&startPg=0&Increment=50&submit=Search			134588867	474496993							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1211973	[O-][N+](=O)c1ccc(cc1NC(c1ccccc1)c1ccccc1)N1CCN(Cc2ccccc2)CC1	InChI=1S/C30H30N4O2/c35-34(36)29-17-16-27(33-20-18-32(19-21-33)23-24-10-4-1-5-11-24)22-28(29)31-30(25-12-6-2-7-13-25)26-14-8-3-9-15-26/h1-17,22,30-31H,18-21,23H2	JBNMUYMPSIGDKH-UHFFFAOYSA-N	574765	US11459308, Compound 3568	Envelope glycoprotein			 4500							US Patent		10.7270/Q28G8PXB		aid1806861	US11459308	Bowlin, TL; Moir, DT; Chandran, K; Dye, Jr., JM; Williams, JD; Aron, ZD; Barbor, JP; Lively, KN; Nash, PJ; Mills, DM; Basu, A	Microbiotix, Inc.; Albert Einstein College of Medicine; The Government of the United States as Represented by the Secretary of the Army	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574765	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Envelope+glycoprotein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574765&enzyme=Envelope+glycoprotein&column=ki&startPg=0&Increment=50&submit=Search			2915525	474496994							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1211975	CN1CCN(CC1)c1cc(NC(c2ccccc2)c2ccccc2)cc(OC(F)(F)F)c1	InChI=1S/C25H26F3N3O/c1-30-12-14-31(15-13-30)22-16-21(17-23(18-22)32-25(26,27)28)29-24(19-8-4-2-5-9-19)20-10-6-3-7-11-20/h2-11,16-18,24,29H,12-15H2,1H3	WOPSQSIBWONVHZ-UHFFFAOYSA-N	574766	US11459308, Compound 3562	Envelope glycoprotein			 3100							US Patent		10.7270/Q28G8PXB		aid1806861	US11459308	Bowlin, TL; Moir, DT; Chandran, K; Dye, Jr., JM; Williams, JD; Aron, ZD; Barbor, JP; Lively, KN; Nash, PJ; Mills, DM; Basu, A	Microbiotix, Inc.; Albert Einstein College of Medicine; The Government of the United States as Represented by the Secretary of the Army	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574766	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Envelope+glycoprotein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574766&enzyme=Envelope+glycoprotein&column=ki&startPg=0&Increment=50&submit=Search			134590051	474496995							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1211977	[O-][N+](=O)c1ccc(cc1NC(c1ccccc1)c1ccccc1)N1CCN(Cc2cccs2)CC1	InChI=1S/C28H28N4O2S/c33-32(34)27-14-13-24(31-17-15-30(16-18-31)21-25-12-7-19-35-25)20-26(27)29-28(22-8-3-1-4-9-22)23-10-5-2-6-11-23/h1-14,19-20,28-29H,15-18,21H2	BQUQJHYNARRJEX-UHFFFAOYSA-N	574768	US11459308, Compound 3575	Envelope glycoprotein			>20000							US Patent		10.7270/Q28G8PXB		aid1806861	US11459308	Bowlin, TL; Moir, DT; Chandran, K; Dye, Jr., JM; Williams, JD; Aron, ZD; Barbor, JP; Lively, KN; Nash, PJ; Mills, DM; Basu, A	Microbiotix, Inc.; Albert Einstein College of Medicine; The Government of the United States as Represented by the Secretary of the Army	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574768	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Envelope+glycoprotein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574768&enzyme=Envelope+glycoprotein&column=ki&startPg=0&Increment=50&submit=Search			134589618	474496997							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1211979	[O-][N+](=O)c1ccc(cc1NC(c1ccccc1)c1ccccc1)N1CCN(Cc2ccco2)CC1	InChI=1S/C28H28N4O3/c33-32(34)27-14-13-24(31-17-15-30(16-18-31)21-25-12-7-19-35-25)20-26(27)29-28(22-8-3-1-4-9-22)23-10-5-2-6-11-23/h1-14,19-20,28-29H,15-18,21H2	XGEJSJJZDFBEKL-UHFFFAOYSA-N	574769	US11459308, Compound 3574	Envelope glycoprotein			 1200							US Patent		10.7270/Q28G8PXB		aid1806861	US11459308	Bowlin, TL; Moir, DT; Chandran, K; Dye, Jr., JM; Williams, JD; Aron, ZD; Barbor, JP; Lively, KN; Nash, PJ; Mills, DM; Basu, A	Microbiotix, Inc.; Albert Einstein College of Medicine; The Government of the United States as Represented by the Secretary of the Army	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574769	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Envelope+glycoprotein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574769&enzyme=Envelope+glycoprotein&column=ki&startPg=0&Increment=50&submit=Search			134589317	474496998							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1211981	[O-][N+](=O)c1ccc(cc1NC(c1ccccc1)c1ccccc1)N1CCN(Cc2ccsc2)CC1	InChI=1S/C28H28N4O2S/c33-32(34)27-12-11-25(31-16-14-30(15-17-31)20-22-13-18-35-21-22)19-26(27)29-28(23-7-3-1-4-8-23)24-9-5-2-6-10-24/h1-13,18-19,21,28-29H,14-17,20H2	ZZGAHWPFJMYWLN-UHFFFAOYSA-N	574770	US11459308, Compound 3576	Envelope glycoprotein			>20000							US Patent		10.7270/Q28G8PXB		aid1806861	US11459308	Bowlin, TL; Moir, DT; Chandran, K; Dye, Jr., JM; Williams, JD; Aron, ZD; Barbor, JP; Lively, KN; Nash, PJ; Mills, DM; Basu, A	Microbiotix, Inc.; Albert Einstein College of Medicine; The Government of the United States as Represented by the Secretary of the Army	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574770	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Envelope+glycoprotein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574770&enzyme=Envelope+glycoprotein&column=ki&startPg=0&Increment=50&submit=Search			134589341	474496999							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1211983	CN1CCC(CC1)N1CCN(CC1)c1ccc(c(NC(c2ccccc2)c2ccccc2)c1)[N+]([O-])=O	InChI=1S/C29H35N5O2/c1-31-16-14-25(15-17-31)32-18-20-33(21-19-32)26-12-13-28(34(35)36)27(22-26)30-29(23-8-4-2-5-9-23)24-10-6-3-7-11-24/h2-13,22,25,29-30H,14-21H2,1H3	SPDWVTOEAKIXOG-UHFFFAOYSA-N	574771	US11459308, Compound 3577	Envelope glycoprotein			>20000							US Patent		10.7270/Q28G8PXB		aid1806861	US11459308	Bowlin, TL; Moir, DT; Chandran, K; Dye, Jr., JM; Williams, JD; Aron, ZD; Barbor, JP; Lively, KN; Nash, PJ; Mills, DM; Basu, A	Microbiotix, Inc.; Albert Einstein College of Medicine; The Government of the United States as Represented by the Secretary of the Army	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574771	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Envelope+glycoprotein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574771&enzyme=Envelope+glycoprotein&column=ki&startPg=0&Increment=50&submit=Search			134589582	474497000							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1211985	CN1CCN(CC1)c1ccc(c(NC(c2ccccc2)c2ccccc2)c1)[N+]([O-])=O	InChI=1S/C24H26N4O2/c1-26-14-16-27(17-15-26)21-12-13-23(28(29)30)22(18-21)25-24(19-8-4-2-5-9-19)20-10-6-3-7-11-20/h2-13,18,24-25H,14-17H2,1H3	RHCKSABVOKGXBN-UHFFFAOYSA-N	50223308	CHEMBL398481::N-benzhydryl-5-(4-methylpiperazin-1-yl)-2-nitrobenzenamine::US11459308, Compound PPZ-1	Envelope glycoprotein			 2300							US Patent		10.7270/Q28G8PXB		aid1806861	US11459308	Bowlin, TL; Moir, DT; Chandran, K; Dye, Jr., JM; Williams, JD; Aron, ZD; Barbor, JP; Lively, KN; Nash, PJ; Mills, DM; Basu, A	Microbiotix, Inc.; Albert Einstein College of Medicine; The Government of the United States as Represented by the Secretary of the Army	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50223308	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Envelope+glycoprotein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50223308&enzyme=Envelope+glycoprotein&column=ki&startPg=0&Increment=50&submit=Search			5206725	104095403		CHEMBL398481				ZINC04687377	1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1211992	CN(C)C1CCN(CC1)c1ccc(c(NC(c2ccccc2)c2ccccc2)c1)[N+]([O-])=O	InChI=1S/C26H30N4O2/c1-28(2)22-15-17-29(18-16-22)23-13-14-25(30(31)32)24(19-23)27-26(20-9-5-3-6-10-20)21-11-7-4-8-12-21/h3-14,19,22,26-27H,15-18H2,1-2H3	SOJISHUHDYZOCG-UHFFFAOYSA-N	574777	US11459308, Compound 3748	Envelope glycoprotein			 700							US Patent		10.7270/Q28G8PXB		aid1806861	US11459308	Bowlin, TL; Moir, DT; Chandran, K; Dye, Jr., JM; Williams, JD; Aron, ZD; Barbor, JP; Lively, KN; Nash, PJ; Mills, DM; Basu, A	Microbiotix, Inc.; Albert Einstein College of Medicine; The Government of the United States as Represented by the Secretary of the Army	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574777	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Envelope+glycoprotein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574777&enzyme=Envelope+glycoprotein&column=ki&startPg=0&Increment=50&submit=Search			134588698	474497006							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1211996	CN1CCN(CC1)c1cc(NC(c2ccccc2)c2ccccc2)c(cc1C)[N+]([O-])=O	InChI=1S/C25H28N4O2/c1-19-17-24(29(30)31)22(18-23(19)28-15-13-27(2)14-16-28)26-25(20-9-5-3-6-10-20)21-11-7-4-8-12-21/h3-12,17-18,25-26H,13-16H2,1-2H3	VYDARSYGTDDXOZ-UHFFFAOYSA-N	574780	US11459308, Compound 3729	Envelope glycoprotein			 1300							US Patent		10.7270/Q28G8PXB		aid1806861	US11459308	Bowlin, TL; Moir, DT; Chandran, K; Dye, Jr., JM; Williams, JD; Aron, ZD; Barbor, JP; Lively, KN; Nash, PJ; Mills, DM; Basu, A	Microbiotix, Inc.; Albert Einstein College of Medicine; The Government of the United States as Represented by the Secretary of the Army	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574780	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Envelope+glycoprotein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574780&enzyme=Envelope+glycoprotein&column=ki&startPg=0&Increment=50&submit=Search			134588733	474497009							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1212000	CN(C)CCNc1ccc(c(NC(c2ccccc2)c2ccccc2)c1)[N+]([O-])=O	InChI=1S/C23H26N4O2/c1-26(2)16-15-24-20-13-14-22(27(28)29)21(17-20)25-23(18-9-5-3-6-10-18)19-11-7-4-8-12-19/h3-14,17,23-25H,15-16H2,1-2H3	DUFXRMWFIDZJBZ-UHFFFAOYSA-N	574784	US11459308, Compound 4329::US11459308, Compound 4334	Envelope glycoprotein			 820							US Patent		10.7270/Q28G8PXB		aid1806861	US11459308	Bowlin, TL; Moir, DT; Chandran, K; Dye, Jr., JM; Williams, JD; Aron, ZD; Barbor, JP; Lively, KN; Nash, PJ; Mills, DM; Basu, A	Microbiotix, Inc.; Albert Einstein College of Medicine; The Government of the United States as Represented by the Secretary of the Army	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574784	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Envelope+glycoprotein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574784&enzyme=Envelope+glycoprotein&column=ki&startPg=0&Increment=50&submit=Search			134605174	474497013							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1212002	CN(C)CCCNc1ccc(c(NC(c2ccccc2)c2ccccc2)c1)[N+]([O-])=O	InChI=1S/C24H28N4O2/c1-27(2)17-9-16-25-21-14-15-23(28(29)30)22(18-21)26-24(19-10-5-3-6-11-19)20-12-7-4-8-13-20/h3-8,10-15,18,24-26H,9,16-17H2,1-2H3	CNFVYFRVJNFAGE-UHFFFAOYSA-N	574785	US11459308, Compound 4335	Envelope glycoprotein			 480							US Patent		10.7270/Q28G8PXB		aid1806861	US11459308	Bowlin, TL; Moir, DT; Chandran, K; Dye, Jr., JM; Williams, JD; Aron, ZD; Barbor, JP; Lively, KN; Nash, PJ; Mills, DM; Basu, A	Microbiotix, Inc.; Albert Einstein College of Medicine; The Government of the United States as Represented by the Secretary of the Army	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574785	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Envelope+glycoprotein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574785&enzyme=Envelope+glycoprotein&column=ki&startPg=0&Increment=50&submit=Search			139518604	474497014							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1212004	CC(C)N(CCNc1ccc(c(NC(c2ccccc2)c2ccccc2)c1)[N+]([O-])=O)C(C)C	InChI=1S/C27H34N4O2/c1-20(2)30(21(3)4)18-17-28-24-15-16-26(31(32)33)25(19-24)29-27(22-11-7-5-8-12-22)23-13-9-6-10-14-23/h5-16,19-21,27-29H,17-18H2,1-4H3	KDOPFMPKHSSSHS-UHFFFAOYSA-N	574786	US11459308, Compound 4336	Envelope glycoprotein			 560							US Patent		10.7270/Q28G8PXB		aid1806861	US11459308	Bowlin, TL; Moir, DT; Chandran, K; Dye, Jr., JM; Williams, JD; Aron, ZD; Barbor, JP; Lively, KN; Nash, PJ; Mills, DM; Basu, A	Microbiotix, Inc.; Albert Einstein College of Medicine; The Government of the United States as Represented by the Secretary of the Army	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574786	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Envelope+glycoprotein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574786&enzyme=Envelope+glycoprotein&column=ki&startPg=0&Increment=50&submit=Search			134605371	474497015							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1212008	CN1CCN(CC1)c1ccc(c(NC(c2ccccc2)c2ccccc2)c1)[N+]([O-])=O	InChI=1S/C24H26N4O2/c1-26-14-16-27(17-15-26)21-12-13-23(28(29)30)22(18-21)25-24(19-8-4-2-5-9-19)20-10-6-3-7-11-20/h2-13,18,24-25H,14-17H2,1H3	RHCKSABVOKGXBN-UHFFFAOYSA-N	50223308	CHEMBL398481::N-benzhydryl-5-(4-methylpiperazin-1-yl)-2-nitrobenzenamine::US11459308, Compound PPZ-1	Envelope glycoprotein			 2300							US Patent		10.7270/Q28G8PXB		aid1806861	US11459308	Bowlin, TL; Moir, DT; Chandran, K; Dye, Jr., JM; Williams, JD; Aron, ZD; Barbor, JP; Lively, KN; Nash, PJ; Mills, DM; Basu, A	Microbiotix, Inc.; Albert Einstein College of Medicine; The Government of the United States as Represented by the Secretary of the Army	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50223308	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Envelope+glycoprotein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50223308&enzyme=Envelope+glycoprotein&column=ki&startPg=0&Increment=50&submit=Search			5206725	104095403		CHEMBL398481				ZINC04687377	1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1212010	CN1CCN(CC1)c1cccc(NC(c2ccccc2)c2ccccc2)c1	InChI=1S/C24H27N3/c1-26-15-17-27(18-16-26)23-14-8-13-22(19-23)25-24(20-9-4-2-5-10-20)21-11-6-3-7-12-21/h2-14,19,24-25H,15-18H2,1H3	NTBJJPBUCDLXTC-UHFFFAOYSA-N	574748	US11459308, Compound 3566::US11459308, Compound 3567	Envelope glycoprotein			 4100							US Patent		10.7270/Q28G8PXB		aid1806861	US11459308	Bowlin, TL; Moir, DT; Chandran, K; Dye, Jr., JM; Williams, JD; Aron, ZD; Barbor, JP; Lively, KN; Nash, PJ; Mills, DM; Basu, A	Microbiotix, Inc.; Albert Einstein College of Medicine; The Government of the United States as Represented by the Secretary of the Army	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574748	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Envelope+glycoprotein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574748&enzyme=Envelope+glycoprotein&column=ki&startPg=0&Increment=50&submit=Search			134589427	474496977							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1212012	CN1CCN(CC1)c1ccnc(NC(c2ccccc2)c2ccccc2)c1	InChI=1S/C23H26N4/c1-26-14-16-27(17-15-26)21-12-13-24-22(18-21)25-23(19-8-4-2-5-9-19)20-10-6-3-7-11-20/h2-13,18,23H,14-17H2,1H3,(H,24,25)	TYXYYADCDOAZFU-UHFFFAOYSA-N	574753	US11459308, Compound 3580::US11459308, Compound 3586	Envelope glycoprotein			 2600							US Patent		10.7270/Q28G8PXB		aid1806861	US11459308	Bowlin, TL; Moir, DT; Chandran, K; Dye, Jr., JM; Williams, JD; Aron, ZD; Barbor, JP; Lively, KN; Nash, PJ; Mills, DM; Basu, A	Microbiotix, Inc.; Albert Einstein College of Medicine; The Government of the United States as Represented by the Secretary of the Army	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574753	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Envelope+glycoprotein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574753&enzyme=Envelope+glycoprotein&column=ki&startPg=0&Increment=50&submit=Search			134588755	474496982							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1212014	CN1CCN(CC1)c1ccc2[nH]c(=O)n(C(c3ccccc3)c3ccccc3)c2c1	InChI=1S/C25H26N4O/c1-27-14-16-28(17-15-27)21-12-13-22-23(18-21)29(25(30)26-22)24(19-8-4-2-5-9-19)20-10-6-3-7-11-20/h2-13,18,24H,14-17H2,1H3,(H,26,30)	HLTOTMADBCSVSU-UHFFFAOYSA-N	574792	US11459308, Compound 3525	Envelope glycoprotein			>20000							US Patent		10.7270/Q28G8PXB		aid1806861	US11459308	Bowlin, TL; Moir, DT; Chandran, K; Dye, Jr., JM; Williams, JD; Aron, ZD; Barbor, JP; Lively, KN; Nash, PJ; Mills, DM; Basu, A	Microbiotix, Inc.; Albert Einstein College of Medicine; The Government of the United States as Represented by the Secretary of the Army	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574792	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Envelope+glycoprotein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574792&enzyme=Envelope+glycoprotein&column=ki&startPg=0&Increment=50&submit=Search			134589501	474497019							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1212016	CN1CCN(CC1)c1ccc(NS(C)(=O)=O)c(NC(c2ccccc2)c2ccccc2)c1	InChI=1S/C25H30N4O2S/c1-28-15-17-29(18-16-28)22-13-14-23(27-32(2,30)31)24(19-22)26-25(20-9-5-3-6-10-20)21-11-7-4-8-12-21/h3-14,19,25-27H,15-18H2,1-2H3	LUBVMRQXYXXBTA-UHFFFAOYSA-N	574793	US11459308, Compound 3536	Envelope glycoprotein			 3100							US Patent		10.7270/Q28G8PXB		aid1806861	US11459308	Bowlin, TL; Moir, DT; Chandran, K; Dye, Jr., JM; Williams, JD; Aron, ZD; Barbor, JP; Lively, KN; Nash, PJ; Mills, DM; Basu, A	Microbiotix, Inc.; Albert Einstein College of Medicine; The Government of the United States as Represented by the Secretary of the Army	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574793	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Envelope+glycoprotein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574793&enzyme=Envelope+glycoprotein&column=ki&startPg=0&Increment=50&submit=Search			134588766	474497020							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1212018	CC(=O)N1CCN(CC1)c1ccc(c(NC(c2ccccc2)c2ccccc2)c1)[N+]([O-])=O	InChI=1S/C25H26N4O3/c1-19(30)27-14-16-28(17-15-27)22-12-13-24(29(31)32)23(18-22)26-25(20-8-4-2-5-9-20)21-10-6-3-7-11-21/h2-13,18,25-26H,14-17H2,1H3	JJWWLFJONCHDJL-UHFFFAOYSA-N	574794	US11459308, Compound 3743	Envelope glycoprotein			 2000							US Patent		10.7270/Q28G8PXB		aid1806861	US11459308	Bowlin, TL; Moir, DT; Chandran, K; Dye, Jr., JM; Williams, JD; Aron, ZD; Barbor, JP; Lively, KN; Nash, PJ; Mills, DM; Basu, A	Microbiotix, Inc.; Albert Einstein College of Medicine; The Government of the United States as Represented by the Secretary of the Army	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574794	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Envelope+glycoprotein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574794&enzyme=Envelope+glycoprotein&column=ki&startPg=0&Increment=50&submit=Search			134588792	474497021							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1212020	CN1CCN(CC1)c1ccc(c(NC(c2ccccc2)c2ccccc2)c1)[N+]([O-])=O	InChI=1S/C24H26N4O2/c1-26-14-16-27(17-15-26)21-12-13-23(28(29)30)22(18-21)25-24(19-8-4-2-5-9-19)20-10-6-3-7-11-20/h2-13,18,24-25H,14-17H2,1H3	RHCKSABVOKGXBN-UHFFFAOYSA-N	50223308	CHEMBL398481::N-benzhydryl-5-(4-methylpiperazin-1-yl)-2-nitrobenzenamine::US11459308, Compound PPZ-1	Envelope glycoprotein			 2300							US Patent		10.7270/Q28G8PXB		aid1806861	US11459308	Bowlin, TL; Moir, DT; Chandran, K; Dye, Jr., JM; Williams, JD; Aron, ZD; Barbor, JP; Lively, KN; Nash, PJ; Mills, DM; Basu, A	Microbiotix, Inc.; Albert Einstein College of Medicine; The Government of the United States as Represented by the Secretary of the Army	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50223308	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Envelope+glycoprotein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50223308&enzyme=Envelope+glycoprotein&column=ki&startPg=0&Increment=50&submit=Search			5206725	104095403		CHEMBL398481				ZINC04687377	1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1212022	CN1CCN(CC1)c1cc(NC(c2ccccc2)c2ccccc2)cc(c1)C(F)(F)F	InChI=1S/C25H26F3N3/c1-30-12-14-31(15-13-30)23-17-21(25(26,27)28)16-22(18-23)29-24(19-8-4-2-5-9-19)20-10-6-3-7-11-20/h2-11,16-18,24,29H,12-15H2,1H3	KMGNRABFDLMYEY-UHFFFAOYSA-N	574795	US11459308, Compound 3540	Envelope glycoprotein			 900							US Patent		10.7270/Q28G8PXB		aid1806861	US11459308	Bowlin, TL; Moir, DT; Chandran, K; Dye, Jr., JM; Williams, JD; Aron, ZD; Barbor, JP; Lively, KN; Nash, PJ; Mills, DM; Basu, A	Microbiotix, Inc.; Albert Einstein College of Medicine; The Government of the United States as Represented by the Secretary of the Army	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574795	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Envelope+glycoprotein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574795&enzyme=Envelope+glycoprotein&column=ki&startPg=0&Increment=50&submit=Search			134589340	474497022							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1212024	CN1CCN(CC1)c1ccc2ncn(C(c3ccccc3)c3ccccc3)c2c1	InChI=1S/C25H26N4/c1-27-14-16-28(17-15-27)22-12-13-23-24(18-22)29(19-26-23)25(20-8-4-2-5-9-20)21-10-6-3-7-11-21/h2-13,18-19,25H,14-17H2,1H3	SLHWFGGHOSQHOS-UHFFFAOYSA-N	574796	US11459308, Compound 3539	Envelope glycoprotein			>20000							US Patent		10.7270/Q28G8PXB		aid1806861	US11459308	Bowlin, TL; Moir, DT; Chandran, K; Dye, Jr., JM; Williams, JD; Aron, ZD; Barbor, JP; Lively, KN; Nash, PJ; Mills, DM; Basu, A	Microbiotix, Inc.; Albert Einstein College of Medicine; The Government of the United States as Represented by the Secretary of the Army	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574796	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Envelope+glycoprotein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574796&enzyme=Envelope+glycoprotein&column=ki&startPg=0&Increment=50&submit=Search			134589008	474497023							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1212029	C1CN(CCN1)c1ccc2ncn(C(c3ccccc3)c3ccccc3)c2c1	InChI=1S/C24H24N4/c1-3-7-19(8-4-1)24(20-9-5-2-6-10-20)28-18-26-22-12-11-21(17-23(22)28)27-15-13-25-14-16-27/h1-12,17-18,24-25H,13-16H2	UMTFHPGVVOECMN-UHFFFAOYSA-N	574799	US11459308, Compound 3587	Envelope glycoprotein			 2200							US Patent		10.7270/Q28G8PXB		aid1806861	US11459308	Bowlin, TL; Moir, DT; Chandran, K; Dye, Jr., JM; Williams, JD; Aron, ZD; Barbor, JP; Lively, KN; Nash, PJ; Mills, DM; Basu, A	Microbiotix, Inc.; Albert Einstein College of Medicine; The Government of the United States as Represented by the Secretary of the Army	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574799	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Envelope+glycoprotein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574799&enzyme=Envelope+glycoprotein&column=ki&startPg=0&Increment=50&submit=Search			139507979	474497026							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1212027	CN1CCN(CC1)c1ccc2nnn(C(c3ccccc3)c3ccccc3)c2c1	InChI=1S/C24H25N5/c1-27-14-16-28(17-15-27)21-12-13-22-23(18-21)29(26-25-22)24(19-8-4-2-5-9-19)20-10-6-3-7-11-20/h2-13,18,24H,14-17H2,1H3	ZFJJIBCWYCAQJP-UHFFFAOYSA-N	574798	US11459308, Compound 3537	Envelope glycoprotein			 2300							US Patent		10.7270/Q28G8PXB		aid1806861	US11459308	Bowlin, TL; Moir, DT; Chandran, K; Dye, Jr., JM; Williams, JD; Aron, ZD; Barbor, JP; Lively, KN; Nash, PJ; Mills, DM; Basu, A	Microbiotix, Inc.; Albert Einstein College of Medicine; The Government of the United States as Represented by the Secretary of the Army	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574798	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Envelope+glycoprotein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574798&enzyme=Envelope+glycoprotein&column=ki&startPg=0&Increment=50&submit=Search			134605160	474497025							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1212031	CN1CCN(CC1)c1ccc(c(NC(c2ccccc2)c2ccccc2)c1)C(F)(F)F	InChI=1S/C25H26F3N3/c1-30-14-16-31(17-15-30)21-12-13-22(25(26,27)28)23(18-21)29-24(19-8-4-2-5-9-19)20-10-6-3-7-11-20/h2-13,18,24,29H,14-17H2,1H3	BCSMPZXKRMFVNE-UHFFFAOYSA-N	574800	US11459308, Compound 3673	Envelope glycoprotein			 2500							US Patent		10.7270/Q28G8PXB		aid1806861	US11459308	Bowlin, TL; Moir, DT; Chandran, K; Dye, Jr., JM; Williams, JD; Aron, ZD; Barbor, JP; Lively, KN; Nash, PJ; Mills, DM; Basu, A	Microbiotix, Inc.; Albert Einstein College of Medicine; The Government of the United States as Represented by the Secretary of the Army	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574800	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Envelope+glycoprotein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574800&enzyme=Envelope+glycoprotein&column=ki&startPg=0&Increment=50&submit=Search			134589158	474497027							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1212033	CN1CCN(CC1)c1ccc(c(NC(c2ccccc2)c2ccccc2)c1)[N+]([O-])=O	InChI=1S/C24H26N4O2/c1-26-14-16-27(17-15-26)21-12-13-23(28(29)30)22(18-21)25-24(19-8-4-2-5-9-19)20-10-6-3-7-11-20/h2-13,18,24-25H,14-17H2,1H3	RHCKSABVOKGXBN-UHFFFAOYSA-N	50223308	CHEMBL398481::N-benzhydryl-5-(4-methylpiperazin-1-yl)-2-nitrobenzenamine::US11459308, Compound PPZ-1	Envelope glycoprotein			 2300							US Patent		10.7270/Q28G8PXB		aid1806861	US11459308	Bowlin, TL; Moir, DT; Chandran, K; Dye, Jr., JM; Williams, JD; Aron, ZD; Barbor, JP; Lively, KN; Nash, PJ; Mills, DM; Basu, A	Microbiotix, Inc.; Albert Einstein College of Medicine; The Government of the United States as Represented by the Secretary of the Army	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50223308	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Envelope+glycoprotein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50223308&enzyme=Envelope+glycoprotein&column=ki&startPg=0&Increment=50&submit=Search			5206725	104095403		CHEMBL398481				ZINC04687377	1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1212035	CN1CCN(CC1)c1ccc(c(NCc2ccccc2)c1)[N+]([O-])=O	InChI=1S/C18H22N4O2/c1-20-9-11-21(12-10-20)16-7-8-18(22(23)24)17(13-16)19-14-15-5-3-2-4-6-15/h2-8,13,19H,9-12,14H2,1H3	LPOIGVZLNWEGJG-UHFFFAOYSA-N	50544038	CHEMBL249033::US11459308, Compound 3514	Envelope glycoprotein			 15000							US Patent		10.7270/Q28G8PXB		aid1806861	US11459308	Bowlin, TL; Moir, DT; Chandran, K; Dye, Jr., JM; Williams, JD; Aron, ZD; Barbor, JP; Lively, KN; Nash, PJ; Mills, DM; Basu, A	Microbiotix, Inc.; Albert Einstein College of Medicine; The Government of the United States as Represented by the Secretary of the Army	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50544038	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Envelope+glycoprotein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50544038&enzyme=Envelope+glycoprotein&column=ki&startPg=0&Increment=50&submit=Search			2866378	442145601							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1212037	CN1CCN(CC1)c1ccc(c(NC(c2ccccc2)c2cccc(C)c2)c1)[N+]([O-])=O	InChI=1S/C25H28N4O2/c1-19-7-6-10-21(17-19)25(20-8-4-3-5-9-20)26-23-18-22(11-12-24(23)29(30)31)28-15-13-27(2)14-16-28/h3-12,17-18,25-26H,13-16H2,1-2H3	FRBQKWPSHZJJMD-UHFFFAOYSA-N	574802	US11459308, Compound 3633	Envelope glycoprotein			 1300							US Patent		10.7270/Q28G8PXB		aid1806861	US11459308	Bowlin, TL; Moir, DT; Chandran, K; Dye, Jr., JM; Williams, JD; Aron, ZD; Barbor, JP; Lively, KN; Nash, PJ; Mills, DM; Basu, A	Microbiotix, Inc.; Albert Einstein College of Medicine; The Government of the United States as Represented by the Secretary of the Army	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574802	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Envelope+glycoprotein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574802&enzyme=Envelope+glycoprotein&column=ki&startPg=0&Increment=50&submit=Search			134605269	474497029							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1212039	COc1ccccc1C(Nc1cc(ccc1[N+]([O-])=O)N1CCN(C)CC1)c1ccccc1	InChI=1S/C25H28N4O3/c1-27-14-16-28(17-15-27)20-12-13-23(29(30)31)22(18-20)26-25(19-8-4-3-5-9-19)21-10-6-7-11-24(21)32-2/h3-13,18,25-26H,14-17H2,1-2H3	YLFYVZYAGLADPW-UHFFFAOYSA-N	574803	US11459308, Compound 3634	Envelope glycoprotein			 3000							US Patent		10.7270/Q28G8PXB		aid1806861	US11459308	Bowlin, TL; Moir, DT; Chandran, K; Dye, Jr., JM; Williams, JD; Aron, ZD; Barbor, JP; Lively, KN; Nash, PJ; Mills, DM; Basu, A	Microbiotix, Inc.; Albert Einstein College of Medicine; The Government of the United States as Represented by the Secretary of the Army	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574803	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Envelope+glycoprotein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574803&enzyme=Envelope+glycoprotein&column=ki&startPg=0&Increment=50&submit=Search			134589228	474497030							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1212042	CN1CCN(CC1)c1ccc(c(NC(c2ccccc2)c2ccc(Cl)cc2)c1)[N+]([O-])=O	InChI=1S/C24H25ClN4O2/c1-27-13-15-28(16-14-27)21-11-12-23(29(30)31)22(17-21)26-24(18-5-3-2-4-6-18)19-7-9-20(25)10-8-19/h2-12,17,24,26H,13-16H2,1H3	SMMKLFYZDDHVIB-UHFFFAOYSA-N	574807	US11459308, Compound 3643	Envelope glycoprotein			>20000							US Patent		10.7270/Q28G8PXB		aid1806861	US11459308	Bowlin, TL; Moir, DT; Chandran, K; Dye, Jr., JM; Williams, JD; Aron, ZD; Barbor, JP; Lively, KN; Nash, PJ; Mills, DM; Basu, A	Microbiotix, Inc.; Albert Einstein College of Medicine; The Government of the United States as Represented by the Secretary of the Army	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574807	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Envelope+glycoprotein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574807&enzyme=Envelope+glycoprotein&column=ki&startPg=0&Increment=50&submit=Search			134588992	474497034							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1212051	CN(C1CCN(C)CC1)c1ccc(c(NC(c2ccccc2)c2ccccc2)c1)[N+]([O-])=O	InChI=1S/C26H30N4O2/c1-28-17-15-22(16-18-28)29(2)23-13-14-25(30(31)32)24(19-23)27-26(20-9-5-3-6-10-20)21-11-7-4-8-12-21/h3-14,19,22,26-27H,15-18H2,1-2H3	IGEOYTBDOUGUCV-UHFFFAOYSA-N	574815	US11459308, Compound 3741	Envelope glycoprotein			 10300							US Patent		10.7270/Q28G8PXB		aid1806861	US11459308	Bowlin, TL; Moir, DT; Chandran, K; Dye, Jr., JM; Williams, JD; Aron, ZD; Barbor, JP; Lively, KN; Nash, PJ; Mills, DM; Basu, A	Microbiotix, Inc.; Albert Einstein College of Medicine; The Government of the United States as Represented by the Secretary of the Army	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574815	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Envelope+glycoprotein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574815&enzyme=Envelope+glycoprotein&column=ki&startPg=0&Increment=50&submit=Search			134588681	474497042							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1212057	CN1CCN(CC1)c1ccc(c(NC(c2ccccc2)c2ccccc2)c1)[N+]([O-])=O	InChI=1S/C24H26N4O2/c1-26-14-16-27(17-15-26)21-12-13-23(28(29)30)22(18-21)25-24(19-8-4-2-5-9-19)20-10-6-3-7-11-20/h2-13,18,24-25H,14-17H2,1H3	RHCKSABVOKGXBN-UHFFFAOYSA-N	50223308	CHEMBL398481::N-benzhydryl-5-(4-methylpiperazin-1-yl)-2-nitrobenzenamine::US11459308, Compound PPZ-1	Envelope glycoprotein			 2300							US Patent		10.7270/Q28G8PXB		aid1806861	US11459308	Bowlin, TL; Moir, DT; Chandran, K; Dye, Jr., JM; Williams, JD; Aron, ZD; Barbor, JP; Lively, KN; Nash, PJ; Mills, DM; Basu, A	Microbiotix, Inc.; Albert Einstein College of Medicine; The Government of the United States as Represented by the Secretary of the Army	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50223308	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Envelope+glycoprotein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50223308&enzyme=Envelope+glycoprotein&column=ki&startPg=0&Increment=50&submit=Search			5206725	104095403		CHEMBL398481				ZINC04687377	1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1212059	C1CCN2CCN(CC2C1)c1ccc2ncn(C(c3ccccc3)c3ccccc3)c2c1	InChI=1S/C28H30N4/c1-3-9-22(10-4-1)28(23-11-5-2-6-12-23)32-21-29-26-15-14-24(19-27(26)32)31-18-17-30-16-8-7-13-25(30)20-31/h1-6,9-12,14-15,19,21,25,28H,7-8,13,16-18,20H2	VTHFHIDGTGGXJL-UHFFFAOYSA-N	574821	US11459308, Compound 4210	Envelope glycoprotein			 1800							US Patent		10.7270/Q28G8PXB		aid1806861	US11459308	Bowlin, TL; Moir, DT; Chandran, K; Dye, Jr., JM; Williams, JD; Aron, ZD; Barbor, JP; Lively, KN; Nash, PJ; Mills, DM; Basu, A	Microbiotix, Inc.; Albert Einstein College of Medicine; The Government of the United States as Represented by the Secretary of the Army	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574821	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Envelope+glycoprotein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574821&enzyme=Envelope+glycoprotein&column=ki&startPg=0&Increment=50&submit=Search			134589315	474497045							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1212062	CN1CCN(CC1)c1ccc2ncn(c2c1)C(C)(C)c1ccccc1	InChI=1S/C21H26N4/c1-21(2,17-7-5-4-6-8-17)25-16-22-19-10-9-18(15-20(19)25)24-13-11-23(3)12-14-24/h4-10,15-16H,11-14H2,1-3H3	GGCLIGXPEVGFQQ-UHFFFAOYSA-N	574823	US11459308, Compound 4212	Envelope glycoprotein			 530							US Patent		10.7270/Q28G8PXB		aid1806861	US11459308	Bowlin, TL; Moir, DT; Chandran, K; Dye, Jr., JM; Williams, JD; Aron, ZD; Barbor, JP; Lively, KN; Nash, PJ; Mills, DM; Basu, A	Microbiotix, Inc.; Albert Einstein College of Medicine; The Government of the United States as Represented by the Secretary of the Army	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574823	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Envelope+glycoprotein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574823&enzyme=Envelope+glycoprotein&column=ki&startPg=0&Increment=50&submit=Search			134589591	474497047							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1212064	CN(C)CCNc1ccc2ncn(C(c3ccccc3)c3ccccc3)c2c1	InChI=1S/C24H26N4/c1-27(2)16-15-25-21-13-14-22-23(17-21)28(18-26-22)24(19-9-5-3-6-10-19)20-11-7-4-8-12-20/h3-14,17-18,24-25H,15-16H2,1-2H3	HHJZPWQQAQZTCX-UHFFFAOYSA-N	574824	US11459308, Compound 4215A::US11459308, Compound 4251	Envelope glycoprotein			 2660							US Patent		10.7270/Q28G8PXB		aid1806861	US11459308	Bowlin, TL; Moir, DT; Chandran, K; Dye, Jr., JM; Williams, JD; Aron, ZD; Barbor, JP; Lively, KN; Nash, PJ; Mills, DM; Basu, A	Microbiotix, Inc.; Albert Einstein College of Medicine; The Government of the United States as Represented by the Secretary of the Army	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574824	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Envelope+glycoprotein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574824&enzyme=Envelope+glycoprotein&column=ki&startPg=0&Increment=50&submit=Search			134589587	474497048							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1212066	CN(C)CCCNc1ccc2ncn(C(c3ccccc3)c3ccccc3)c2c1	InChI=1S/C25H28N4/c1-28(2)17-9-16-26-22-14-15-23-24(18-22)29(19-27-23)25(20-10-5-3-6-11-20)21-12-7-4-8-13-21/h3-8,10-15,18-19,25-26H,9,16-17H2,1-2H3	FFPGMBMQIVMSGL-UHFFFAOYSA-N	574825	US11459308, Compound 4252	Envelope glycoprotein			 8620							US Patent		10.7270/Q28G8PXB		aid1806861	US11459308	Bowlin, TL; Moir, DT; Chandran, K; Dye, Jr., JM; Williams, JD; Aron, ZD; Barbor, JP; Lively, KN; Nash, PJ; Mills, DM; Basu, A	Microbiotix, Inc.; Albert Einstein College of Medicine; The Government of the United States as Represented by the Secretary of the Army	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574825	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Envelope+glycoprotein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574825&enzyme=Envelope+glycoprotein&column=ki&startPg=0&Increment=50&submit=Search			134589412	474497049							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1212068	CC(C)N(CCNc1ccc2ncn(C(c3ccccc3)c3ccccc3)c2c1)C(C)C	InChI=1S/C28H34N4/c1-21(2)31(22(3)4)18-17-29-25-15-16-26-27(19-25)32(20-30-26)28(23-11-7-5-8-12-23)24-13-9-6-10-14-24/h5-16,19-22,28-29H,17-18H2,1-4H3	BFRUDLITMGWGDG-UHFFFAOYSA-N	574826	US11459308, Compound 4253A	Envelope glycoprotein			 1850							US Patent		10.7270/Q28G8PXB		aid1806861	US11459308	Bowlin, TL; Moir, DT; Chandran, K; Dye, Jr., JM; Williams, JD; Aron, ZD; Barbor, JP; Lively, KN; Nash, PJ; Mills, DM; Basu, A	Microbiotix, Inc.; Albert Einstein College of Medicine; The Government of the United States as Represented by the Secretary of the Army	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=574826	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Envelope+glycoprotein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=574826&enzyme=Envelope+glycoprotein&column=ki&startPg=0&Increment=50&submit=Search			134605370	474497050							1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1212072	CN1CCN(CC1)c1ccc(c(NC(c2ccccc2)c2ccccc2)c1)[N+]([O-])=O	InChI=1S/C24H26N4O2/c1-26-14-16-27(17-15-26)21-12-13-23(28(29)30)22(18-21)25-24(19-8-4-2-5-9-19)20-10-6-3-7-11-20/h2-13,18,24-25H,14-17H2,1H3	RHCKSABVOKGXBN-UHFFFAOYSA-N	50223308	CHEMBL398481::N-benzhydryl-5-(4-methylpiperazin-1-yl)-2-nitrobenzenamine::US11459308, Compound PPZ-1	Envelope glycoprotein			 2300							US Patent		10.7270/Q28G8PXB		aid1806861	US11459308	Bowlin, TL; Moir, DT; Chandran, K; Dye, Jr., JM; Williams, JD; Aron, ZD; Barbor, JP; Lively, KN; Nash, PJ; Mills, DM; Basu, A	Microbiotix, Inc.; Albert Einstein College of Medicine; The Government of the United States as Represented by the Secretary of the Army	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50223308	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Envelope+glycoprotein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50223308&enzyme=Envelope+glycoprotein&column=ki&startPg=0&Increment=50&submit=Search			5206725	104095403		CHEMBL398481				ZINC04687377	1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
1212076	CN1CCN(CC1)c1ccc(c(NC(c2ccccc2)c2ccccc2)c1)[N+]([O-])=O	InChI=1S/C24H26N4O2/c1-26-14-16-27(17-15-26)21-12-13-23(28(29)30)22(18-21)25-24(19-8-4-2-5-9-19)20-10-6-3-7-11-20/h2-13,18,24-25H,14-17H2,1H3	RHCKSABVOKGXBN-UHFFFAOYSA-N	50223308	CHEMBL398481::N-benzhydryl-5-(4-methylpiperazin-1-yl)-2-nitrobenzenamine::US11459308, Compound PPZ-1	Envelope glycoprotein			 2300							US Patent		10.7270/Q28G8PXB		aid1806861	US11459308	Bowlin, TL; Moir, DT; Chandran, K; Dye, Jr., JM; Williams, JD; Aron, ZD; Barbor, JP; Lively, KN; Nash, PJ; Mills, DM; Basu, A	Microbiotix, Inc.; Albert Einstein College of Medicine; The Government of the United States as Represented by the Secretary of the Army	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50223308	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=1305&target=Envelope+glycoprotein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50223308&enzyme=Envelope+glycoprotein&column=ki&startPg=0&Increment=50&submit=Search			5206725	104095403		CHEMBL398481				ZINC04687377	1	MGVTGILQLPRDRFKRTSFFLWVIILFQRTFSIPLGVIHNSTLQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKDFFSSHPLREPVNATEDPSSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTIGEWAFWETKKNLTRKIRSEELSFTAVSNRAKNISGQSPARTSSDPGTNTTTEDHKIMASENSSAMVQVHSQGREAAVSHLTTLATISTSPQPPTTKPGPDNSTHNTPVYKLDISEATQVEQHHRRTDNDSTASDTPPATTAAGPLKAENTNTSKGTDLLDPATTTSPQNHSETAGNNNTHHQDTGEESASSGKLGLITNTIAGVAGLITGGRRARREAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYTEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVDKTLPDQGDNDNWWTGWRQWIPAGIGVTGVIIAVIALFCICKFVF	7SSQ,7SSR,7SWD,7TN9,8DPL,8DPM	Envelope glycoprotein	VGP_EBOZ5	P87666	Q6V1Q7						
