Report error Found 1194 Enz. Inhib. hit(s) with Target = 'Protein mono-ADP-ribosyltransferase PARP14'
TargetProtein mono-ADP-ribosyltransferase PARP14(Human)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 0.360nMAssay Description:Inhibition of PARP14 (unknown origin) incubated for 1 hr by ELISAMore data for this Ligand-Target Pair
Ligand Info
TargetProtein mono-ADP-ribosyltransferase PARP14(Human)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 0.420nMAssay Description:Inhibition of PARP14 (unknown origin) incubated for 1 hr by ELISAMore data for this Ligand-Target Pair
Ligand Info
TargetProtein mono-ADP-ribosyltransferase PARP14(Human)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 0.470nMAssay Description:Inhibition of PARP14 (unknown origin) incubated for 1 hr by ELISAMore data for this Ligand-Target Pair
Ligand Info
TargetProtein mono-ADP-ribosyltransferase PARP14(Human)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 0.75nMAssay Description:Inhibition of PARP14 (unknown origin) incubated for 1 hr by ELISAMore data for this Ligand-Target Pair
Ligand Info
TargetProtein mono-ADP-ribosyltransferase PARP14(Human)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 0.75nMAssay Description:Inhibition of PARP14 (unknown origin) incubated for 1 hr by ELISAMore data for this Ligand-Target Pair
Ligand Info
TargetProtein mono-ADP-ribosyltransferase PARP14(Human)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 0.950nMAssay Description:Inhibition of PARP14 (unknown origin) incubated for 1 hr by ELISAMore data for this Ligand-Target Pair
Ligand Info
TargetProtein mono-ADP-ribosyltransferase PARP14(Human)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 1nMAssay Description:Inhibition of PARP14 (unknown origin) incubated for 1 hr by ELISAMore data for this Ligand-Target Pair
Ligand Info
TargetProtein mono-ADP-ribosyltransferase PARP14(Human)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 1.70nMAssay Description:Inhibition of PARP14 (unknown origin) incubated for 1 hr by ELISAMore data for this Ligand-Target Pair
TargetProtein mono-ADP-ribosyltransferase PARP14(Human)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 2.20nMAssay Description:Inhibition of PARP14 (unknown origin) incubated for 1 hr by ELISAMore data for this Ligand-Target Pair
Ligand Info
TargetProtein mono-ADP-ribosyltransferase PARP14(Human)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 2.30nMAssay Description:Inhibition of PARP14 (unknown origin) incubated for 1 hr by ELISAMore data for this Ligand-Target Pair
Ligand Info
TargetProtein mono-ADP-ribosyltransferase PARP14(Human)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 2.40nMAssay Description:Inhibition of PARP14 (unknown origin) incubated for 1 hr by ELISAMore data for this Ligand-Target Pair
Ligand Info
TargetProtein mono-ADP-ribosyltransferase PARP14(Human)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 3nMAssay Description:Inhibition of human PARP14 by TR-FRET assayMore data for this Ligand-Target Pair
TargetProtein mono-ADP-ribosyltransferase PARP14(Human)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 3nMAssay Description:Inhibition of PARP14 (unknown origin) incubated for 1 hr by ELISAMore data for this Ligand-Target Pair
Ligand Info
TargetProtein mono-ADP-ribosyltransferase PARP14(Human)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 3nMAssay Description:Inhibition of PARP14 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
TargetProtein mono-ADP-ribosyltransferase PARP14(Human)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 3nMAssay Description:Inhibition of N-terminal hexahistidine-tagged human PARP14 (1611 to 1801 residues) catalytic domain extracted from Escherichia coli BL21-CodonPlus (D...More data for this Ligand-Target Pair
Ligand Info
TargetProtein mono-ADP-ribosyltransferase PARP14(Human)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 3nMAssay Description:Displacement of a biotinylated small molecule probe from human PARP14 catalytic domain incubated for 30 mins by TR-FRET assayMore data for this Ligand-Target Pair
TargetProtein mono-ADP-ribosyltransferase PARP14(Human)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 4nMAssay Description:Inhibition of PARP14 (unknown origin)More data for this Ligand-Target Pair
TargetProtein mono-ADP-ribosyltransferase PARP14(Human)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 5nMAssay Description:Inhibition of PARP14 (unknown origin) incubated for 1 hr by ELISAMore data for this Ligand-Target Pair
Ligand Info
TargetProtein mono-ADP-ribosyltransferase PARP14(Human)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 5.5nMAssay Description:Inhibition of PARP14 (unknown origin) incubated for 1 hr by ELISAMore data for this Ligand-Target Pair
Ligand Info
TargetProtein mono-ADP-ribosyltransferase PARP14(Human)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 9.20nMAssay Description:Inhibition of PARP14 (unknown origin) incubated for 1 hr by ELISAMore data for this Ligand-Target Pair
Ligand Info
TargetProtein mono-ADP-ribosyltransferase PARP14(Human)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Inhibition of PARP14 (unknown origin)More data for this Ligand-Target Pair
TargetProtein mono-ADP-ribosyltransferase PARP14(Human)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 19nMAssay Description:Inhibition of PARP14 (unknown origin)More data for this Ligand-Target Pair
TargetProtein mono-ADP-ribosyltransferase PARP14(Human)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 21nMAssay Description:Inhibition of PARP14 (unknown origin) incubated for 1 hr by ELISAMore data for this Ligand-Target Pair
Ligand Info
TargetProtein mono-ADP-ribosyltransferase PARP14(Human)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 29nMAssay Description:Inhibition of PARP14 (unknown origin) incubated for 1 hr by ELISAMore data for this Ligand-Target Pair
Ligand Info
TargetProtein mono-ADP-ribosyltransferase PARP14(Human)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 45nMAssay Description:Inhibition of PARP14 (unknown origin) incubated for 1 hr by ELISAMore data for this Ligand-Target Pair
Ligand Info
TargetProtein mono-ADP-ribosyltransferase PARP14(Human)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 54nMAssay Description:Inhibition of PARP14 (unknown origin) incubated for 1 hr by ELISAMore data for this Ligand-Target Pair
Ligand Info
TargetProtein mono-ADP-ribosyltransferase PARP14(Human)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 76nMAssay Description:Inhibition of PARP14 (unknown origin)More data for this Ligand-Target Pair
TargetProtein mono-ADP-ribosyltransferase PARP14(Human)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 132nMAssay Description:Inhibition of PARP14 (unknown origin) incubated for 1 hr by ELISAMore data for this Ligand-Target Pair
Ligand Info
TargetProtein mono-ADP-ribosyltransferase PARP14(Human)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 160nMAssay Description:Inhibition of full length recombinant His6-tagged PARP14 catalytic domain (unknown origin) expressed in Escherichia coli BL21(DE3) by fluorescence ba...More data for this Ligand-Target Pair
TargetProtein mono-ADP-ribosyltransferase PARP14(Human)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 160nMAssay Description:Inhibition of recombinant human His6-tagged PARP14 catalytic/WWE domain (1459 to 1801 residues) expressed in Escherichia coli BL21(DE3) preincubated ...More data for this Ligand-Target Pair
TargetProtein mono-ADP-ribosyltransferase PARP14(Human)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 160nMAssay Description:Inhibition of recombinant human His6-tagged PARP14 catalytic/WWE domain (1459 to 1801 residues) expressed in Escherichia coli BL21(DE3) preincubated ...More data for this Ligand-Target Pair
TargetProtein mono-ADP-ribosyltransferase PARP14(Human)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 270nMAssay Description:Inhibition of recombinant human His6-tagged PARP14 catalytic/WWE domain (1459 to 1801 residues) expressed in Escherichia coli BL21(DE3) preincubated ...More data for this Ligand-Target Pair
TargetProtein mono-ADP-ribosyltransferase PARP14(Human)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 275nMAssay Description:Inhibition of recombinant human His6-tagged PARP14 catalytic/WWE domain (1459 to 1801 residues) expressed in Escherichia coli BL21(DE3) preincubated ...More data for this Ligand-Target Pair
TargetProtein mono-ADP-ribosyltransferase PARP14(Human)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 300nMAssay Description:Inhibition of N-terminal MBP tagged/C-terminal PARP14 (unknown origin) expressed in Escherichia coli in presence of NAD+ by proximity enhanced assayMore data for this Ligand-Target Pair
TargetProtein mono-ADP-ribosyltransferase PARP14(Human)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 300nMAssay Description:Inhibition of PARP14 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
TargetProtein mono-ADP-ribosyltransferase PARP14(Human)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 310nMAssay Description:Displacement of [3H]NAD+ from GST-tagged PARP14 (unknown origin) incubated for 210 mins by radiometric assayMore data for this Ligand-Target Pair
TargetProtein mono-ADP-ribosyltransferase PARP14(Human)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 370nMAssay Description:Inhibition of recombinant human His6-tagged PARP14 catalytic/WWE domain (1459 to 1801 residues) expressed in Escherichia coli BL21(DE3) preincubated ...More data for this Ligand-Target Pair
TargetProtein mono-ADP-ribosyltransferase PARP14(Human)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 372nMAssay Description:Inhibition of recombinant human His6-tagged PARP14 catalytic/WWE domain (1459 to 1801 residues) expressed in Escherichia coli BL21(DE3) preincubated ...More data for this Ligand-Target Pair
TargetProtein mono-ADP-ribosyltransferase PARP14(Human)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 407nMAssay Description:Inhibition of recombinant human His6-tagged PARP14 catalytic/WWE domain (1459 to 1801 residues) expressed in Escherichia coli BL21(DE3) preincubated ...More data for this Ligand-Target Pair
TargetProtein mono-ADP-ribosyltransferase PARP14(Human)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 410nMAssay Description:Inhibition of recombinant human His6-tagged PARP14 catalytic/WWE domain (1459 to 1801 residues) expressed in Escherichia coli BL21(DE3) preincubated ...More data for this Ligand-Target Pair
TargetProtein mono-ADP-ribosyltransferase PARP14(Human)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 447nMAssay Description:Inhibition of recombinant human His6-tagged PARP14 catalytic/WWE domain (1459 to 1801 residues) expressed in Escherichia coli BL21(DE3) preincubated ...More data for this Ligand-Target Pair
TargetProtein mono-ADP-ribosyltransferase PARP14(Human)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 450nMAssay Description:Inhibition of recombinant human His6-tagged PARP14 catalytic/WWE domain (1459 to 1801 residues) expressed in Escherichia coli BL21(DE3) preincubated ...More data for this Ligand-Target Pair
TargetProtein mono-ADP-ribosyltransferase PARP14(Human)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 490nMAssay Description:Inhibition of fluorescently-labeled PARP14 (unknown origin) by small molecule microarray based analysisMore data for this Ligand-Target Pair
Ligand Info
TargetProtein mono-ADP-ribosyltransferase PARP14(Human)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 490nMAssay Description:Inhibition of PARP14 (unknown origin) expressed in bacterial expression system using histone substrate incubated for 60 mins by chemiluminescence ass...More data for this Ligand-Target Pair
TargetProtein mono-ADP-ribosyltransferase PARP14(Human)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataKd: 550nMAssay Description:Binding affinity to PARP14 MD2 (A994 to N1191 residues) (unknown origin) expressed in bacterial expression system by ITC assayMore data for this Ligand-Target Pair
TargetProtein mono-ADP-ribosyltransferase PARP14(Human)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 580nMAssay Description:Displacement of [3H]NAD+ from GST-tagged PARP14 (unknown origin) incubated for 210 mins by radiometric assayMore data for this Ligand-Target Pair
TargetProtein mono-ADP-ribosyltransferase PARP14(Human)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 610nMAssay Description:Inhibition of PARP14 (unknown origin)More data for this Ligand-Target Pair
TargetProtein mono-ADP-ribosyltransferase PARP14(Human)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 630nMAssay Description:Inhibition of PARP14 (unknown origin) using NAD+ as substrate incubated for 18 hrs by fluorescence based assayMore data for this Ligand-Target Pair
TargetProtein mono-ADP-ribosyltransferase PARP14(Human)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 650nMAssay Description:Inhibition of recombinant human His6-tagged PARP14 catalytic/WWE domain (1459 to 1801 residues) expressed in Escherichia coli BL21(DE3) preincubated ...More data for this Ligand-Target Pair
TargetProtein mono-ADP-ribosyltransferase PARP14(Human)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 650nMAssay Description:Inhibition of N-terminal MBP tagged/C-terminal PARP14 (unknown origin) expressed in Escherichia coli in presence of NAD+ by proximity enhanced assayMore data for this Ligand-Target Pair












3D Structure (crystal)



























