Report error Found 107 Enz. Inhib. hit(s) with Target = 'Protein arginine N-methyltransferase 7'
Ligand Info
Affinity DataIC50: 2.5nMAssay Description:Inhibition of full-length PRMT7 (unknown origin) expressed in Sf9 cells using biotinylated H2B as substrate incubated for 60 mins in presence of 3H-S...More data for this Ligand-Target Pair
Affinity DataIC50: 2.5nMAssay Description:Inhibition of full-length PRMT7 (unknown origin) expressed in Sf9 cells using biotinylated H2B as substrate incubated for 60 mins in presence of 3H-S...More data for this Ligand-Target Pair
Affinity DataIC50: 2.5nMAssay Description:Inhibition of PRMT7 (unknown origin) incubated for 1 hr in presence of 3H-SAM by topcount plate reader analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 2.5nMAssay Description:Inhibition of PRMT7 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 110nMAssay Description:Inhibition of recombinant human PRMT7 using GST-GAR as substrate by hotspot assayMore data for this Ligand-Target Pair
Affinity DataIC50: 220nMAssay Description:Inhibition of human full length recombinant his-tagged PRMT7 (2 to 692 residues) using GST-GAR as substrate incubated for 20 mins in presence of [3H]...More data for this Ligand-Target Pair
Affinity DataIC50: 226nMAssay Description:Inhibition of human full length recombinant his-tagged PRMT7 (2 to 692 residues) using GST-GAR as substrate incubated for 20 mins in presence of [3H]...More data for this Ligand-Target Pair
Affinity DataIC50: 294nMAssay Description:Inhibition of PRMT7 (unknown origin) assessed as reduction in HSPA8 methylationMore data for this Ligand-Target Pair
Affinity DataIC50: 320nMAssay Description:Inhibition of human full length recombinant his-tagged PRMT7 (2 to 692 residues) using GST-GAR as substrate incubated for 20 mins in presence of [3H]...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 410nMAssay Description:Inhibition of human full length recombinant his-tagged PRMT7 (2 to 692 residues) using GST-GAR as substrate incubated for 20 mins in presence of [3H]...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 540nMAssay Description:Inhibition of N-terminal/C-terminal His-tagged human recombinant full-length PRMT7 (2 to 692 residues) using histone GST-GAR as substrate and 3H-SAM ...More data for this Ligand-Target Pair
Affinity DataIC50: 550nMAssay Description:Inhibition of human full length recombinant his-tagged PRMT7 (2 to 692 residues) using GST-GAR as substrate incubated for 20 mins in presence of [3H]...More data for this Ligand-Target Pair
Affinity DataIC50: 555nMAssay Description:Inhibition of PRMT7 (unknown origin)More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 631nMAssay Description:Inhibition of human full length recombinant his-tagged PRMT7 (2 to 692 residues) using GST-GAR as substrate incubated for 20 mins in presence of [3H]...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of full-length PRMT7 (unknown origin) expressed in Sf9 cells using biotinylated H2B as substrate incubated for 60 mins in presence of 3H-S...More data for this Ligand-Target Pair
Ligand Info
Ligand Info
Affinity DataIC50: 1.68E+3nMAssay Description:Inhibition of human full length recombinant his-tagged PRMT7 (2 to 692 residues) using GST-GAR as substrate incubated for 20 mins in presence of [3H]...More data for this Ligand-Target Pair
Ligand Info
Ligand Info
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibition of PRMT7 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 2.30E+3nMAssay Description:Inhibition of PRMT7 (unknown origin)More data for this Ligand-Target Pair
Ligand Info
Ligand Info
Affinity DataIC50: 2.40E+3nMAssay Description:Inhibition of human PRMT7 using GST-GAR as substrate and SAM as cofactor by radiometric HotSpot assayMore data for this Ligand-Target Pair
TargetProtein arginine N-methyltransferase 7(Mus musculus)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 2.40E+3nMAssay Description:Inhibition of PRMT7 in mouse C2C12 cells assessed as reduction in HSP70 methylationMore data for this Ligand-Target Pair
Affinity DataIC50: 2.40E+3nMAssay Description:Inhibition of PRMT7 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibition of PRMT7 (unknown origin)More data for this Ligand-Target Pair
Ligand Info
Ligand Info
Ligand Info
Ligand Info
Ligand Info
Ligand Info
Ligand Info
Ligand Info
Ligand Info
Affinity DataIC50: 4.68E+3nMAssay Description:Inhibition of human full length recombinant his-tagged PRMT7 (2 to 692 residues) using GST-GAR as substrate incubated for 20 mins in presence of [3H]...More data for this Ligand-Target Pair
Ligand Info
Ligand Info
Ligand Info
Ligand Info
Affinity DataIC50: 5.60E+3nMAssay Description:Inhibition of N-terminal/C-terminal His-tagged human recombinant full-length PRMT7 (2 to 692 residues) using histone GST-GAR as substrate and 3H-SAM ...More data for this Ligand-Target Pair












































