Compile Data Set for Download or QSAR
Report error Found 32 Enz. Inhib. hit(s) with Target = 'Pendrin'
TargetPendrin(Human)
University of California San Francisco

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50653508BDBM50653508(CHEMBL6145989)
Affinity DataIC50: 480nMAssay Description:Agonist activity at rat CB2 receptor assessed as inhibition of forskolin-induced cAMP production by cell based assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/3/2026
Entry Details PubMed
TargetPendrin(Human)
University of California San Francisco

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50653507BDBM50653507(CHEMBL1416075)
Affinity DataIC50: 490nMAssay Description:Agonist activity at rat CB2 receptor assessed as inhibition of forskolin-induced cAMP production by cell based assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/3/2026
Entry Details PubMed
TargetPendrin(Human)
University of California San Francisco

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50653506BDBM50653506(CHEMBL1409977)
Affinity DataIC50: 650nMAssay Description:Agonist activity at rat CB2 receptor assessed as inhibition of forskolin-induced cAMP production by cell based assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/3/2026
Entry Details PubMed
TargetPendrin(Human)
University of California San Francisco

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50653509BDBM50653509(CHEMBL1897294)
Affinity DataIC50: 1.44E+3nMAssay Description:Agonist activity at rat CB2 receptor assessed as inhibition of forskolin-induced cAMP production by cell based assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/3/2026
Entry Details PubMed
TargetPendrin(Mouse)
University of California

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50512539BDBM50512539(CHEMBL4466170)
Affinity DataIC50: 3.10E+3nMAssay Description:Inhibition of mouse PDS stably expressed in FRT cells coexpressing EYFP-H148Q/I152L/F46L assessed as reduction in I-/Cl- exchange incubated for 10 mi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetPendrin(Human)
University of California San Francisco

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50653514BDBM50653514(CHEMBL6120880)
Affinity DataIC50: 3.10E+3nMAssay Description:Antagonist activity at human cloned vasopressin V2 receptor by cell based beta lactamase assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/3/2026
Entry Details PubMed
TargetPendrin(Mouse)
University of California

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50512543BDBM50512543(CHEMBL4546564)
Affinity DataIC50: 3.30E+3nMAssay Description:Inhibition of mouse PDS stably expressed in FRT cells coexpressing EYFP-H148Q/I152L/F46L assessed as reduction in I-/Cl- exchange incubated for 10 mi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetPendrin(Mouse)
University of California

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50512535BDBM50512535(CHEMBL4435424)
Affinity DataIC50: 3.30E+3nMAssay Description:Inhibition of mouse PDS stably expressed in FRT cells coexpressing EYFP-H148Q/I152L/F46L assessed as reduction in I-/Cl- exchange incubated for 10 mi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetPendrin(Human)
University of California San Francisco

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50653505BDBM50653505(CHEMBL1370459)
Affinity DataIC50: 4.10E+3nMAssay Description:Agonist activity at rat CB2 receptor assessed as inhibition of forskolin-induced cAMP production by cell based assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/3/2026
Entry Details PubMed
TargetPendrin(Mouse)
University of California

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50512536BDBM50512536(CHEMBL4446784)
Affinity DataIC50: 4.60E+3nMAssay Description:Inhibition of mouse PDS stably expressed in FRT cells coexpressing EYFP-H148Q/I152L/F46L assessed as reduction in I-/Cl- exchange incubated for 10 mi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetPendrin(Human)
University of California San Francisco

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50653510BDBM50653510(CHEMBL1404124)
Affinity DataIC50: 4.80E+3nMAssay Description:Antagonist activity at human cloned oxytocin receptor by cell based beta lactamase assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/3/2026
Entry Details PubMed
TargetPendrin(Human)
University of California San Francisco

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50653512BDBM50653512(CHEMBL1313061)
Affinity DataIC50: 5.00E+3nMAssay Description:Antagonist activity at human cloned vasopressin V2 receptor by cell based beta lactamase assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/3/2026
Entry Details PubMed
TargetPendrin(Mouse)
University of California

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50607937BDBM50607937(CHEMBL4515533)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of mouse Pendrin stably expressed in FRT cells with YFP assessed as inhibition of pendrin mediated Cl-/NO3- exchange by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetPendrin(Human)
University of California San Francisco

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50653511BDBM50653511(CHEMBL1544526)
Affinity DataIC50: 5.60E+3nMAssay Description:Antagonist activity at human cloned vasopressin V1a receptor by cell based beta lactamase assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/3/2026
Entry Details PubMed
TargetPendrin(Mouse)
University of California

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50512537BDBM50512537(CHEMBL4474736)
Affinity DataIC50: 6.60E+3nMAssay Description:Inhibition of mouse PDS stably expressed in FRT cells coexpressing EYFP-H148Q/I152L/F46L assessed as reduction in I-/Cl- exchange incubated for 10 mi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetPendrin(Human)
University of California San Francisco

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50512537BDBM50512537(CHEMBL4474736)
Affinity DataIC50: 7.00E+3nMAssay Description:Inhibition of human PDS stably expressed in FRT cells coexpressing EYFP-H148Q/I152L/F46L assessed as reduction in I-/Cl- exchange incubated for 10 mi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetPendrin(Human)
University of California San Francisco

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50653513BDBM50653513(CHEMBL6103470)
Affinity DataIC50: 8.20E+3nMAssay Description:Antagonist activity at human cloned vasopressin V1a receptor by cell based beta lactamase assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/3/2026
Entry Details PubMed
TargetPendrin(Mouse)
University of California

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50607937BDBM50607937(CHEMBL4515533)
Affinity DataIC50: 9.00E+3nMAssay Description:Inhibition of mouse Pendrin stably expressed in FRT cells with YFP assessed as inhibition of pendrin mediated Cl-/SCN- exchange by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetPendrin(Mouse)
University of California

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50512528BDBM50512528(CHEMBL4590521)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of mouse PDS stably expressed in FRT cells coexpressing EYFP-H148Q/I152L/F46L assessed as reduction in I-/Cl- exchange incubated for 10 mi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetPendrin(Mouse)
University of California

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50512529BDBM50512529(CHEMBL4436619)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of mouse PDS stably expressed in FRT cells coexpressing EYFP-H148Q/I152L/F46L assessed as reduction in I-/Cl- exchange incubated for 10 mi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetPendrin(Mouse)
University of California

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50607937BDBM50607937(CHEMBL4515533)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of mouse Pendrin stably expressed in FRT cells with YFP assessed as inhibition of pendrin mediated Cl-/HCO3- exchange by fluorescence assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetPendrin(Mouse)
University of California

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50512527BDBM50512527(CHEMBL4529094)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of mouse PDS stably expressed in FRT cells coexpressing EYFP-H148Q/I152L/F46L assessed as reduction in I-/Cl- exchange incubated for 10 mi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetPendrin(Mouse)
University of California

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50512542BDBM50512542(CHEMBL4445120)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of mouse PDS stably expressed in FRT cells coexpressing EYFP-H148Q/I152L/F46L assessed as reduction in I-/Cl- exchange incubated for 10 mi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetPendrin(Mouse)
University of California

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50512540BDBM50512540(CHEMBL4444793)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of mouse PDS stably expressed in FRT cells coexpressing EYFP-H148Q/I152L/F46L assessed as reduction in I-/Cl- exchange incubated for 10 mi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetPendrin(Mouse)
University of California

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50512541BDBM50512541(CHEMBL4571849)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of mouse PDS stably expressed in FRT cells coexpressing EYFP-H148Q/I152L/F46L assessed as reduction in I-/Cl- exchange incubated for 10 mi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetPendrin(Mouse)
University of California

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50512538BDBM50512538(CHEMBL4576357)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of mouse PDS stably expressed in FRT cells coexpressing EYFP-H148Q/I152L/F46L assessed as reduction in I-/Cl- exchange incubated for 10 mi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetPendrin(Mouse)
University of California

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50512534BDBM50512534(CHEMBL4578218)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of mouse PDS stably expressed in FRT cells coexpressing EYFP-H148Q/I152L/F46L assessed as reduction in I-/Cl- exchange incubated for 10 mi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetPendrin(Mouse)
University of California

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50512532BDBM50512532(CHEMBL4444063)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of mouse PDS stably expressed in FRT cells coexpressing EYFP-H148Q/I152L/F46L assessed as reduction in I-/Cl- exchange incubated for 10 mi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetPendrin(Mouse)
University of California

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50512533BDBM50512533(CHEMBL4575750)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of mouse PDS stably expressed in FRT cells coexpressing EYFP-H148Q/I152L/F46L assessed as reduction in I-/Cl- exchange incubated for 10 mi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetPendrin(Mouse)
University of California

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50512530BDBM50512530(CHEMBL4546431)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of mouse PDS stably expressed in FRT cells coexpressing EYFP-H148Q/I152L/F46L assessed as reduction in I-/Cl- exchange incubated for 10 mi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetPendrin(Mouse)
University of California

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50512531BDBM50512531(CHEMBL4577192)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of mouse PDS stably expressed in FRT cells coexpressing EYFP-H148Q/I152L/F46L assessed as reduction in I-/Cl- exchange incubated for 10 mi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetPendrin(Human)
University of California San Francisco

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50512537BDBM50512537(CHEMBL4474736)
Affinity DataIC50: 1.25E+4nMAssay Description:Agonist activity at rat CB1 receptor assessed as inhibition of forskolin-induced cAMP production by cell based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2026
Entry Details PubMed