Compile Data Set for Download or QSAR
Report error Found 12 Enz. Inhib. hit(s) with Target = 'Neuronal acetylcholine receptor subunit alpha-6/beta-2'
TargetNeuronal acetylcholine receptor subunit alpha-6/beta-2(Human)
Xiamen University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50621981BDBM50621981(CHEMBL5412811)
Affinity DataKi:  0.0600nMAssay Description:Binding affinity to nACh alpha6beta2 receptor (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-6/beta-2(Human)
Xiamen University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50481208BDBM50481208(CHEMBL594330)
Affinity DataIC50: 0.160nMAssay Description:Inhibition of alpha6beta2 nAChRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2020
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-6/beta-2(Human)
Xiamen University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50481207BDBM50481207(CHEMBL595286)
Affinity DataIC50: 0.260nMAssay Description:Inhibition of alpha6beta2 nAChRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2020
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-6/beta-2(Human)
Xiamen University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50621984BDBM50621984(CHEMBL5404578)
Affinity DataKi:  0.360nMAssay Description:Binding affinity to nACh alpha6beta2 receptor (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-6/beta-2(Human)
Xiamen University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50481206BDBM50481206(CHEMBL595311)
Affinity DataIC50: 0.390nMAssay Description:Inhibition of alpha6beta2 nAChRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2020
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-6/beta-2(Human)
Xiamen University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50621983BDBM50621983(CHEMBL5438932)
Affinity DataKi:  0.5nMAssay Description:Binding affinity to nACh alpha6beta2 receptor (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-6/beta-2(Human)
Xiamen University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50621985BDBM50621985(CHEMBL5430462)
Affinity DataKi:  0.670nMAssay Description:Binding affinity to nACh alpha6beta2 receptor (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-6/beta-2(Human)
Xiamen University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50621982BDBM50621982(CHEMBL5423438)
Affinity DataKi:  0.950nMAssay Description:Binding affinity to nACh alpha6beta2 receptor (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-6/beta-2(Human)
Xiamen University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50481209BDBM50481209(CHEMBL595047)
Affinity DataIC50: 0.950nMAssay Description:Inhibition of alpha6beta2 nAChRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2020
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-6/beta-2(Human)
Xiamen University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50481212BDBM50481212(CHEMBL609593)
Affinity DataIC50: 3nMAssay Description:Inhibition of alpha6beta2 nAChRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2020
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-6/beta-2(Human)
Xiamen University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50621986BDBM50621986(CHEMBL5404069)
Affinity DataKi:  77nMAssay Description:Binding affinity to nACh alpha6beta2 receptor (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-6/beta-2(Human)
Xiamen University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50481210BDBM50481210(CHEMBL609594)
Affinity DataIC50: 201nMAssay Description:Inhibition of alpha6beta2 nAChRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2020
Entry Details Article
PubMed