Compile Data Set for Download or QSAR
Report error Found 97 Enz. Inhib. hit(s) with Target = 'Glutamyl aminopeptidase'
TargetGlutamyl aminopeptidase(Human)
University of Paris

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50083386BDBM50083386(1-{[1-(2,3-Dicarboxy-pyrrolidine-1-carbonyl)-2-met...)
Affinity DataKi:  0.873nMAssay Description:Binding affinity against recombinant Aminopeptidase AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/13/2012
Entry Details Article
PubMed
TargetGlutamyl aminopeptidase(Mus musculus)
Quantum Genomics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50633859BDBM50633859(CHEMBL6101922)
Affinity DataIC50: 1nMAssay Description:Modulation of rat mGlu5 receptor assessed as calcium mobilization by cell based fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2026
Entry Details
PubMed
TargetGlutamyl aminopeptidase(Human)
University of Paris

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50083394BDBM50083394(1-{[1-(1,2-Dicarboxy-ethylcarbamoyl)-2-methyl-buty...)
Affinity DataKi:  3.20nMAssay Description:Binding affinity against recombinant Aminopeptidase AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/13/2012
Entry Details Article
PubMed
TargetGlutamyl aminopeptidase(Human)
University of Paris

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50083376BDBM50083376(3-Carboxy-1-{[1-(1,2-dicarboxy-ethylcarbamoyl)-2-m...)
Affinity DataKi:  3.60nMAssay Description:Binding affinity against recombinant Aminopeptidase AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/13/2012
Entry Details Article
PubMed
TargetGlutamyl aminopeptidase(Human)
University of Paris

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50083378BDBM50083378(1-{[1-(1-Carboxy-2-sulfo-ethylcarbamoyl)-2-methyl-...)
Affinity DataKi:  3.60nMAssay Description:Binding affinity against recombinant Aminopeptidase AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/13/2012
Entry Details Article
PubMed
TargetGlutamyl aminopeptidase(Human)
University of Paris

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50083385BDBM50083385(1-{[1-(2,3-Dicarboxy-pyrrolidine-1-carbonyl)-2-met...)
Affinity DataKi:  3.80nMAssay Description:Binding affinity against recombinant Aminopeptidase AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/13/2012
Entry Details Article
PubMed
TargetGlutamyl aminopeptidase(Mus musculus)
Quantum Genomics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50633836BDBM50633836(CHEMBL6091985)
Affinity DataIC50: 4nMAssay Description:Negative allosteric modulation of rat mGlu3 receptor assessed as calcium mobilization by cell based fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2026
Entry Details
PubMed
TargetGlutamyl aminopeptidase(Human)
University of Paris

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50083393BDBM50083393(1-{[1-(1,2-Dicarboxy-ethylcarbamoyl)-2-(4-hydroxy-...)
Affinity DataKi:  4.30nMAssay Description:Binding affinity against recombinant Aminopeptidase AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/13/2012
Entry Details Article
PubMed
TargetGlutamyl aminopeptidase(Human)
University of Paris

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50083390BDBM50083390(1-{[1-(1,2-Dicarboxy-ethylcarbamoyl)-2-methyl-buty...)
Affinity DataKi:  5.40nMAssay Description:Binding affinity against recombinant Aminopeptidase AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/13/2012
Entry Details Article
PubMed
TargetGlutamyl aminopeptidase(Mus musculus)
Quantum Genomics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50633862BDBM50633862(CHEMBL6091920)
Affinity DataIC50: 7nMAssay Description:Negative allosteric modulation of rat mGlu3 receptor assessed as calcium mobilization by cell based fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2026
Entry Details
PubMed
TargetGlutamyl aminopeptidase(Mus musculus)
Quantum Genomics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50633852BDBM50633852(CHEMBL6132685)
Affinity DataIC50: 9nMAssay Description:Modulation of rat mGlu5 receptor assessed as calcium mobilization by cell based fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2026
Entry Details
PubMed
TargetGlutamyl aminopeptidase(Mus musculus)
Quantum Genomics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50633858BDBM50633858(CHEMBL6078602)
Affinity DataIC50: 9nMAssay Description:Modulation of rat mGlu5 receptor assessed as calcium mobilization by cell based fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2026
Entry Details
PubMed
TargetGlutamyl aminopeptidase(Human)
University of Paris

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50083374BDBM50083374(1-{[1-(1-Carboxy-3-sulfo-propylcarbamoyl)-2-(4-hyd...)
Affinity DataKi:  9.30nMAssay Description:Binding affinity against recombinant Aminopeptidase AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/13/2012
Entry Details Article
PubMed
TargetGlutamyl aminopeptidase(Mus musculus)
Quantum Genomics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50633844BDBM50633844(CHEMBL6134529)
Affinity DataIC50: 10nMAssay Description:Modulation of rat mGlu5 receptor assessed as calcium mobilization by cell based fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2026
Entry Details
PubMed
TargetGlutamyl aminopeptidase(Mus musculus)
Quantum Genomics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50633857BDBM50633857(CHEMBL6141870)
Affinity DataIC50: 10nMAssay Description:Modulation of rat mGlu5 receptor assessed as calcium mobilization by cell based fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2026
Entry Details
PubMed
TargetGlutamyl aminopeptidase(Human)
University of Paris

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50083382BDBM50083382(1-{[1-(1,2-Dicarboxy-ethylcarbamoyl)-2-methyl-buty...)
Affinity DataKi:  12nMAssay Description:Binding affinity against recombinant Aminopeptidase AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/13/2012
Entry Details Article
PubMed
TargetGlutamyl aminopeptidase(Human)
University of Paris

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50083403BDBM50083403(3-Carboxy-1-{[1-(1,2-dicarboxy-ethylcarbamoyl)-2-m...)
Affinity DataKi:  13nMAssay Description:Binding affinity against recombinant Aminopeptidase AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/13/2012
Entry Details Article
PubMed
TargetGlutamyl aminopeptidase(Human)
University of Paris

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50457482BDBM50457482(CHEMBL4217064)
Affinity DataKi:  13nMAssay Description:Inhibition of APA (unknown origin) using GlubetaNA as substrate after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetGlutamyl aminopeptidase(Human)
University of Paris

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50083387BDBM50083387(1-{[1-(1-Carbamoyl-2-carboxy-ethylcarbamoyl)-2-met...)
Affinity DataKi:  15nMAssay Description:Binding affinity against recombinant Aminopeptidase AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/13/2012
Entry Details Article
PubMed
TargetGlutamyl aminopeptidase(Human)
University of Paris

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50083392BDBM50083392(1-{[1-(1,2-Dicarboxy-ethylcarbamoyl)-2-methyl-buty...)
Affinity DataKi:  15nMAssay Description:Binding affinity against recombinant Aminopeptidase AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/13/2012
Entry Details Article
PubMed
TargetGlutamyl aminopeptidase(Human)
University of Paris

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50083400BDBM50083400(3-Carboxy-1-{[1-(1,2-dicarboxy-ethylcarbamoyl)-2-m...)
Affinity DataKi:  16nMAssay Description:Binding affinity against recombinant Aminopeptidase AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/13/2012
Entry Details Article
PubMed
TargetGlutamyl aminopeptidase(Mus musculus)
Quantum Genomics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50633846BDBM50633846(CHEMBL6144468)
Affinity DataIC50: 18nMAssay Description:Modulation of rat mGlu5 receptor assessed as calcium mobilization by cell based fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2026
Entry Details
PubMed
TargetGlutamyl aminopeptidase(Human)
University of Paris

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50083384BDBM50083384(1-{[1-(1,2-Dicarboxy-ethylcarbamoyl)-2-methyl-buty...)
Affinity DataKi:  20nMAssay Description:Binding affinity against recombinant Aminopeptidase AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/13/2012
Entry Details Article
PubMed
TargetGlutamyl aminopeptidase(Mus musculus)
Quantum Genomics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50633861BDBM50633861(CHEMBL6102273)
Affinity DataIC50: 21nMAssay Description:Modulation of rat mGlu5 receptor assessed as calcium mobilization by cell based fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2026
Entry Details
PubMed
TargetGlutamyl aminopeptidase(Mus musculus)
Quantum Genomics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50633849BDBM50633849(CHEMBL6083014)
Affinity DataIC50: 21nMAssay Description:Modulation of rat mGlu5 receptor assessed as calcium mobilization by cell based fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2026
Entry Details
PubMed
TargetGlutamyl aminopeptidase(Mus musculus)
Quantum Genomics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50633848BDBM50633848(CHEMBL6142075)
Affinity DataIC50: 23nMAssay Description:Modulation of rat mGlu5 receptor assessed as calcium mobilization by cell based fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2026
Entry Details
PubMed
TargetGlutamyl aminopeptidase(Mus musculus)
Quantum Genomics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50633854BDBM50633854(CHEMBL6096566)
Affinity DataIC50: 24nMAssay Description:Modulation of rat mGlu5 receptor assessed as calcium mobilization by cell based fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2026
Entry Details
PubMed
TargetGlutamyl aminopeptidase(Mus musculus)
Quantum Genomics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50633851BDBM50633851(CHEMBL6145942)
Affinity DataIC50: 26nMAssay Description:Modulation of rat mGlu5 receptor assessed as calcium mobilization by cell based fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2026
Entry Details
PubMed
TargetGlutamyl aminopeptidase(Mus musculus)
Quantum Genomics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50633856BDBM50633856(CHEMBL6149319)
Affinity DataIC50: 26nMAssay Description:Modulation of rat mGlu5 receptor assessed as calcium mobilization by cell based fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2026
Entry Details
PubMed
TargetGlutamyl aminopeptidase(Human)
University of Paris

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50083395BDBM50083395(1-{[1-(1,2-Dicarboxy-ethylcarbamoyl)-2-(4-hydroxy-...)
Affinity DataKi:  27nMAssay Description:Binding affinity against recombinant Aminopeptidase AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/13/2012
Entry Details Article
PubMed
TargetGlutamyl aminopeptidase(Mus musculus)
Quantum Genomics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50633847BDBM50633847(CHEMBL6147420)
Affinity DataIC50: 27nMAssay Description:Modulation of rat mGlu5 receptor assessed as calcium mobilization by cell based fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2026
Entry Details
PubMed
TargetGlutamyl aminopeptidase(Mus musculus)
Quantum Genomics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50633853BDBM50633853(CHEMBL6078318)
Affinity DataIC50: 28nMAssay Description:Modulation of rat mGlu5 receptor assessed as calcium mobilization by cell based fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2026
Entry Details
PubMed
TargetGlutamyl aminopeptidase(Mus musculus)
Quantum Genomics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50633839BDBM50633839(CHEMBL6120447)
Affinity DataIC50: 29nMAssay Description:Modulation of rat mGlu5 receptor assessed as calcium mobilization by cell based fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2026
Entry Details
PubMed
TargetGlutamyl aminopeptidase(Mus musculus)
Quantum Genomics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50633863BDBM50633863(CHEMBL6114886)
Affinity DataIC50: 30nMAssay Description:Negative allosteric modulation of rat mGlu3 receptor assessed as calcium mobilization by cell based fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2026
Entry Details
PubMed
TargetGlutamyl aminopeptidase(Mus musculus)
Quantum Genomics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50633840BDBM50633840(CHEMBL6146273)
Affinity DataIC50: 39nMAssay Description:Modulation of rat mGlu5 receptor assessed as calcium mobilization by cell based fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2026
Entry Details
PubMed
TargetGlutamyl aminopeptidase(Human)
University of Paris

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50083398BDBM50083398((3R,4R)-3-ammonio-5-{[(1S)-1-carboxy-2-methylbutyl...)
Affinity DataKi:  40nMAssay Description:Binding affinity against recombinant Aminopeptidase AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/13/2012
Entry Details Article
PubMed
TargetGlutamyl aminopeptidase(Mus musculus)
Quantum Genomics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50633845BDBM50633845(CHEMBL6120664)
Affinity DataIC50: 41nMAssay Description:Modulation of rat mGlu5 receptor assessed as calcium mobilization by cell based fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2026
Entry Details
PubMed
TargetGlutamyl aminopeptidase(Mus musculus)
Quantum Genomics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50633860BDBM50633860(CHEMBL6083078)
Affinity DataIC50: 42nMAssay Description:Modulation of rat mGlu5 receptor assessed as calcium mobilization by cell based fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2026
Entry Details
PubMed
TargetGlutamyl aminopeptidase(Human)
University of Paris

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50083377BDBM50083377(1-{[1-(1,2-Dicarboxy-ethylcarbamoyl)-2-methyl-buty...)
Affinity DataKi:  50nMAssay Description:Binding affinity against recombinant Aminopeptidase AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/13/2012
Entry Details Article
PubMed
TargetGlutamyl aminopeptidase(Human)
University of Paris

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50083375BDBM50083375(3-[(1S,2R)-1-((S)-1,2-Dicarboxy-ethylcarbamoyl)-2-...)
Affinity DataKi:  51nMAssay Description:Binding affinity against recombinant Aminopeptidase AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/13/2012
Entry Details Article
PubMed
TargetGlutamyl aminopeptidase(Human)
University of Paris

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50083402BDBM50083402(1-{[1-(1,2-Dicarboxy-ethylcarbamoyl)-2-methyl-buty...)
Affinity DataKi:  53nMAssay Description:Binding affinity against recombinant Aminopeptidase AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/13/2012
Entry Details Article
PubMed
TargetGlutamyl aminopeptidase(Mus musculus)
Quantum Genomics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50633841BDBM50633841(CHEMBL6144088)
Affinity DataIC50: 54nMAssay Description:Modulation of rat mGlu5 receptor assessed as calcium mobilization by cell based fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2026
Entry Details
PubMed
TargetGlutamyl aminopeptidase(Mus musculus)
Quantum Genomics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50633855BDBM50633855(CHEMBL6091792)
Affinity DataIC50: 54nMAssay Description:Modulation of rat mGlu5 receptor assessed as calcium mobilization by cell based fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2026
Entry Details
PubMed
TargetGlutamyl aminopeptidase(Mus musculus)
Quantum Genomics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50633850BDBM50633850(CHEMBL6134712)
Affinity DataIC50: 61nMAssay Description:Modulation of rat mGlu5 receptor assessed as calcium mobilization by cell based fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2026
Entry Details
PubMed
TargetGlutamyl aminopeptidase(Human)
University of Paris

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50190112BDBM50190112(CHEMBL88808)
Affinity DataKi:  67nMAssay Description:Inhibition of APA (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetGlutamyl aminopeptidase(Human)
University of Paris

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50083399BDBM50083399(1-{[1-(1-Carboxy-3-sulfo-propylcarbamoyl)-2-(4-hyd...)
Affinity DataKi:  73nMAssay Description:Binding affinity against recombinant Aminopeptidase AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/13/2012
Entry Details Article
PubMed
TargetGlutamyl aminopeptidase(Human)
University of Paris

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50083380BDBM50083380(1-{[(1S,2R)-1-((S)-1,2-Dicarboxy-ethylcarbamoyl)-2...)
Affinity DataKi:  80nMAssay Description:Binding affinity against recombinant Aminopeptidase AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/13/2012
Entry Details Article
PubMed
TargetGlutamyl aminopeptidase(Human)
University of Paris

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50083389BDBM50083389(1-{[1-(1-Carboxy-2-sulfo-ethylcarbamoyl)-2-methyl-...)
Affinity DataKi:  83nMAssay Description:Binding affinity against recombinant Aminopeptidase AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/13/2012
Entry Details Article
PubMed
TargetGlutamyl aminopeptidase(Human)
University of Paris

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50083372BDBM50083372(1-{[1-(2,3-Dicarboxy-pyrrolidine-1-carbonyl)-2-met...)
Affinity DataKi:  110nMAssay Description:Binding affinity against recombinant Aminopeptidase AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/13/2012
Entry Details Article
PubMed
TargetGlutamyl aminopeptidase(Human)
University of Paris

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50457465BDBM50457465(CHEMBL4204736)
Affinity DataKi:  130nMAssay Description:Inhibition of APA (unknown origin) using GluNA as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
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