Compile Data Set for Download or QSAR
Report error Found 142 Enz. Inhib. hit(s) with Target = 'G protein-coupled receptor kinase 6'
TargetG protein-coupled receptor kinase 6(Human)
Ontario Institute For Cancer Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50566950BDBM50566950(CHEMBL4852125)
Affinity DataIC50: 3.5nMAssay Description:Inhibition of recombinant full-length human GRK6 using casein as substrate measured after 80 mins in presence of [gamma33P]ATP by radiometric scintil...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2022
Entry Details Article
PubMed
TargetG protein-coupled receptor kinase 6(Human)
Ontario Institute For Cancer Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50566949BDBM50566949(CHEMBL4877302)
Affinity DataIC50: 3.80nMAssay Description:Inhibition of human GRK6 using casein as substrate in presence of [gamma33P]ATP by radiometric hotspot kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2022
Entry Details Article
PubMed
TargetG protein-coupled receptor kinase 6(Human)
Ontario Institute For Cancer Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 130909BDBM130909(US8822500, Stauro- sporine | US9920060, Staurospor...)
Affinity DataIC50: 4.20nMAssay Description:Inhibition of human GRK6 using casein as substrate preincubated for 20 mins followed by [gamma-33P]-ATP addition and measured after 120 mins by radio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetG protein-coupled receptor kinase 6(Human)
Ontario Institute For Cancer Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50566953BDBM50566953(CHEMBL4860332)
Affinity DataIC50: 6nMAssay Description:Inhibition of recombinant full-length human GRK6 using casein as substrate measured after 80 mins in presence of [gamma33P]ATP by radiometric scintil...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2022
Entry Details Article
PubMed
TargetG protein-coupled receptor kinase 6(Human)
Ontario Institute For Cancer Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50566946BDBM50566946(CHEMBL4854871)
Affinity DataIC50: 7.20nMAssay Description:Inhibition of recombinant full-length human GRK6 using casein as substrate measured after 80 mins in presence of [gamma33P]ATP by radiometric scintil...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2022
Entry Details Article
PubMed
TargetG protein-coupled receptor kinase 6(Human)
Ontario Institute For Cancer Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50566949BDBM50566949(CHEMBL4877302)
Affinity DataIC50: 8nMAssay Description:Inhibition of recombinant full-length human GRK6 using casein as substrate measured after 80 mins in presence of [gamma33P]ATP by radiometric scintil...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2022
Entry Details Article
PubMed
TargetG protein-coupled receptor kinase 6(Human)
Ontario Institute For Cancer Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50566923BDBM50566923(CHEMBL4855000)
Affinity DataIC50: 10nMAssay Description:Inhibition of recombinant full-length human GRK6 using casein as substrate measured after 80 mins in presence of [gamma33P]ATP by radiometric scintil...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2022
Entry Details Article
PubMed
TargetG protein-coupled receptor kinase 6(Human)
Ontario Institute For Cancer Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50566951BDBM50566951(CHEMBL4875929)
Affinity DataIC50: 11nMAssay Description:Inhibition of recombinant full-length human GRK6 using casein as substrate measured after 80 mins in presence of [gamma33P]ATP by radiometric scintil...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2022
Entry Details Article
PubMed
TargetG protein-coupled receptor kinase 6(Human)
Ontario Institute For Cancer Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50566948BDBM50566948(CHEMBL4874424)
Affinity DataIC50: 16nMAssay Description:Inhibition of recombinant full-length human GRK6 using casein as substrate measured after 80 mins in presence of [gamma33P]ATP by radiometric scintil...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2022
Entry Details Article
PubMed
TargetG protein-coupled receptor kinase 6(Human)
Ontario Institute For Cancer Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50566947BDBM50566947(CHEMBL4847703)
Affinity DataIC50: 18nMAssay Description:Inhibition of recombinant full-length human GRK6 using casein as substrate measured after 80 mins in presence of [gamma33P]ATP by radiometric scintil...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2022
Entry Details Article
PubMed
TargetG protein-coupled receptor kinase 6(Human)
Ontario Institute For Cancer Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50566946BDBM50566946(CHEMBL4854871)
Affinity DataIC50: 18nMAssay Description:Inhibition of human GRK6 using casein as substrate in presence of [gamma33P]ATP by radiometric hotspot kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2022
Entry Details Article
PubMed
TargetG protein-coupled receptor kinase 6(Human)
Ontario Institute For Cancer Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50566922BDBM50566922(CHEMBL4876072)
Affinity DataIC50: 20nMAssay Description:Inhibition of recombinant full-length human GRK6 using casein as substrate measured after 80 mins in presence of [gamma33P]ATP by radiometric scintil...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2022
Entry Details Article
PubMed
TargetG protein-coupled receptor kinase 6(Human)
Ontario Institute For Cancer Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50657930BDBM50657930(CHEMBL6151486)
Affinity DataIC50: 20nMMore data for this Ligand-Target Pair
Ligand InfoPDB
In Depth
Date in BDB:
6/5/2026
Entry Details PubMed
TargetG protein-coupled receptor kinase 6(Human)
Ontario Institute For Cancer Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50640313BDBM50640313(CHEMBL5569207)
Affinity DataIC50: 22nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/5/2026
Entry Details PubMed
TargetG protein-coupled receptor kinase 6(Human)
Ontario Institute For Cancer Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50566939BDBM50566939(CHEMBL4871944)
Affinity DataIC50: 27nMAssay Description:Inhibition of recombinant full-length human GRK6 using casein as substrate measured after 80 mins in presence of [gamma33P]ATP by radiometric scintil...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2022
Entry Details Article
PubMed
TargetG protein-coupled receptor kinase 6(Human)
Ontario Institute For Cancer Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50566952BDBM50566952(CHEMBL4872426)
Affinity DataIC50: 27nMAssay Description:Inhibition of recombinant full-length human GRK6 using casein as substrate measured after 80 mins in presence of [gamma33P]ATP by radiometric scintil...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2022
Entry Details Article
PubMed
TargetG protein-coupled receptor kinase 6(Human)
Ontario Institute For Cancer Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50566940BDBM50566940(CHEMBL4870615)
Affinity DataIC50: 29nMAssay Description:Inhibition of recombinant full-length human GRK6 using casein as substrate measured after 80 mins in presence of [gamma33P]ATP by radiometric scintil...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2022
Entry Details Article
PubMed
TargetG protein-coupled receptor kinase 6(Human)
Ontario Institute For Cancer Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50566949BDBM50566949(CHEMBL4877302)
Affinity DataIC50: 30nMAssay Description:Binding affinity to FLAG-tagged GRK6 in human KMS11 cells incubated for 2.5 hrs by ITDR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2022
Entry Details Article
PubMed
TargetG protein-coupled receptor kinase 6(Human)
Ontario Institute For Cancer Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50657931BDBM50657931(CHEMBL6146311)
Affinity DataIC50: 32nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/5/2026
Entry Details PubMed
TargetG protein-coupled receptor kinase 6(Human)
Ontario Institute For Cancer Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 2579BDBM2579(CHEMBL388978 | Staurosporine, 8 | Staurosporin, 4 ...)
Affinity DataIC50: 32.9nMAssay Description:Inhibition of human GRK6 using casein as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetG protein-coupled receptor kinase 6(Human)
Ontario Institute For Cancer Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50657929BDBM50657929(CHEMBL6152550)
Affinity DataIC50: 33nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/5/2026
Entry Details PubMed
TargetG protein-coupled receptor kinase 6(Human)
Ontario Institute For Cancer Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50566947BDBM50566947(CHEMBL4847703)
Affinity DataIC50: 33nMAssay Description:Inhibition of human GRK6 using casein as substrate in presence of [gamma33P]ATP by radiometric hotspot kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2022
Entry Details Article
PubMed
TargetG protein-coupled receptor kinase 6(Human)
Ontario Institute For Cancer Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 79886BDBM79886(US20250388567, Compound 21)
Affinity DataIC50: 34nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2026
Entry Details PubMed
TargetG protein-coupled receptor kinase 6(Human)
Ontario Institute For Cancer Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 79878BDBM79878(US20250388567, Compound 14)
Affinity DataIC50: 36nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2026
Entry Details PubMed
TargetG protein-coupled receptor kinase 6(Human)
Ontario Institute For Cancer Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50566943BDBM50566943(CHEMBL4846282)
Affinity DataIC50: 40nMAssay Description:Inhibition of recombinant full-length human GRK6 using casein as substrate measured after 80 mins in presence of [gamma33P]ATP by radiometric scintil...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2022
Entry Details Article
PubMed
TargetG protein-coupled receptor kinase 6(Human)
Ontario Institute For Cancer Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50657925BDBM50657925(CHEMBL6164395)
Affinity DataIC50: 40nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/5/2026
Entry Details PubMed
TargetG protein-coupled receptor kinase 6(Human)
Ontario Institute For Cancer Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50657928BDBM50657928(CHEMBL6162335)
Affinity DataIC50: 40nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/5/2026
Entry Details PubMed
TargetG protein-coupled receptor kinase 6(Human)
Ontario Institute For Cancer Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50657934BDBM50657934(CHEMBL6164393)
Affinity DataIC50: 40nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/5/2026
Entry Details PubMed
TargetG protein-coupled receptor kinase 6(Human)
Ontario Institute For Cancer Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50566928BDBM50566928(CHEMBL4847311)
Affinity DataIC50: 41nMAssay Description:Inhibition of recombinant full-length human GRK6 using casein as substrate measured after 80 mins in presence of [gamma33P]ATP by radiometric scintil...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2022
Entry Details Article
PubMed
TargetG protein-coupled receptor kinase 6(Human)
Ontario Institute For Cancer Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50657927BDBM50657927(CHEMBL6161120)
Affinity DataIC50: 50nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/5/2026
Entry Details PubMed
TargetG protein-coupled receptor kinase 6(Human)
Ontario Institute For Cancer Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50657922BDBM50657922(CHEMBL6168617)
Affinity DataIC50: 60nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/5/2026
Entry Details PubMed
TargetG protein-coupled receptor kinase 6(Human)
Ontario Institute For Cancer Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50657926BDBM50657926(CHEMBL6151812)
Affinity DataIC50: 60nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/5/2026
Entry Details PubMed
TargetG protein-coupled receptor kinase 6(Human)
Ontario Institute For Cancer Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 2579BDBM2579(CHEMBL388978 | Staurosporine, 8 | Staurosporin, 4 ...)
Affinity DataIC50: 61.7nMAssay Description:Inhibition of human GRK6 using casein as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetG protein-coupled receptor kinase 6(Human)
Ontario Institute For Cancer Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50640321BDBM50640321(CHEMBL5574633)
Affinity DataIC50: 62nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/5/2026
Entry Details PubMed
TargetG protein-coupled receptor kinase 6(Human)
Ontario Institute For Cancer Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50566937BDBM50566937(CHEMBL4850937)
Affinity DataIC50: 70nMAssay Description:Inhibition of recombinant full-length human GRK6 using casein as substrate measured after 80 mins in presence of [gamma33P]ATP by radiometric scintil...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2022
Entry Details Article
PubMed
TargetG protein-coupled receptor kinase 6(Human)
Ontario Institute For Cancer Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50566941BDBM50566941(CHEMBL4849245)
Affinity DataIC50: 91nMAssay Description:Inhibition of recombinant full-length human GRK6 using casein as substrate measured after 80 mins in presence of [gamma33P]ATP by radiometric scintil...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2022
Entry Details Article
PubMed
TargetG protein-coupled receptor kinase 6(Human)
Ontario Institute For Cancer Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50566924BDBM50566924(CHEMBL4860927)
Affinity DataIC50: 100nMAssay Description:Inhibition of recombinant full-length human GRK6 using casein as substrate measured after 80 mins in presence of [gamma33P]ATP by radiometric scintil...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2022
Entry Details Article
PubMed
TargetG protein-coupled receptor kinase 6(Human)
Ontario Institute For Cancer Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50657924BDBM50657924(CHEMBL6161413)
Affinity DataIC50: 100nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/5/2026
Entry Details PubMed
TargetG protein-coupled receptor kinase 6(Human)
Ontario Institute For Cancer Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50657933BDBM50657933(CHEMBL6152245)
Affinity DataIC50: 110nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/5/2026
Entry Details PubMed
TargetG protein-coupled receptor kinase 6(Human)
Ontario Institute For Cancer Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50566921BDBM50566921(CHEMBL4876138)
Affinity DataIC50: 110nMAssay Description:Inhibition of recombinant full-length human GRK6 using casein as substrate measured after 80 mins in presence of [gamma33P]ATP by radiometric scintil...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2022
Entry Details Article
PubMed
TargetG protein-coupled receptor kinase 6(Human)
Ontario Institute For Cancer Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50566915BDBM50566915(CHEMBL4848826)
Affinity DataIC50: 120nMAssay Description:Inhibition of recombinant full-length human GRK6 using casein as substrate measured after 80 mins in presence of [gamma33P]ATP by radiometric scintil...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2022
Entry Details Article
PubMed
TargetG protein-coupled receptor kinase 6(Human)
Ontario Institute For Cancer Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50657932BDBM50657932(CHEMBL6145814)
Affinity DataIC50: 130nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/5/2026
Entry Details PubMed
TargetG protein-coupled receptor kinase 6(Human)
Ontario Institute For Cancer Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50566927BDBM50566927(CHEMBL4860406)
Affinity DataIC50: 140nMAssay Description:Inhibition of recombinant full-length human GRK6 using casein as substrate measured after 80 mins in presence of [gamma33P]ATP by radiometric scintil...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2022
Entry Details Article
PubMed
TargetG protein-coupled receptor kinase 6(Human)
Ontario Institute For Cancer Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50566925BDBM50566925(CHEMBL4860226)
Affinity DataIC50: 160nMAssay Description:Inhibition of recombinant full-length human GRK6 using casein as substrate measured after 80 mins in presence of [gamma33P]ATP by radiometric scintil...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2022
Entry Details Article
PubMed
TargetG protein-coupled receptor kinase 6(Human)
Ontario Institute For Cancer Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50566953BDBM50566953(CHEMBL4860332)
Affinity DataIC50: 170nMAssay Description:Binding affinity to FLAG-tagged GRK6 in human KMS11 cells incubated for 2.5 hrs by ITDR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2022
Entry Details Article
PubMed
TargetG protein-coupled receptor kinase 6(Human)
Ontario Institute For Cancer Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50566917BDBM50566917(CHEMBL4848792)
Affinity DataIC50: 180nMAssay Description:Inhibition of recombinant full-length human GRK6 using casein as substrate measured after 80 mins in presence of [gamma33P]ATP by radiometric scintil...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2022
Entry Details Article
PubMed
TargetG protein-coupled receptor kinase 6(Human)
Ontario Institute For Cancer Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50566916BDBM50566916(CHEMBL4858397)
Affinity DataIC50: 190nMAssay Description:Inhibition of recombinant full-length human GRK6 using casein as substrate measured after 80 mins in presence of [gamma33P]ATP by radiometric scintil...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2022
Entry Details Article
PubMed
TargetG protein-coupled receptor kinase 6(Human)
Ontario Institute For Cancer Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50657935BDBM50657935(CHEMBL6162930)
Affinity DataIC50: 190nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/5/2026
Entry Details PubMed
TargetG protein-coupled receptor kinase 6(Human)
Ontario Institute For Cancer Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50657923BDBM50657923(CHEMBL6159848)
Affinity DataIC50: 220nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/5/2026
Entry Details PubMed
TargetG protein-coupled receptor kinase 6(Human)
Ontario Institute For Cancer Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50566942BDBM50566942(CHEMBL4875743)
Affinity DataIC50: 230nMAssay Description:Inhibition of recombinant full-length human GRK6 using casein as substrate measured after 80 mins in presence of [gamma33P]ATP by radiometric scintil...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2022
Entry Details Article
PubMed
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