Compile Data Set for Download or QSAR
Report error Found 272 Enz. Inhib. hit(s) with Target = 'Cyclin-dependent kinase 2/G1/S-specific cyclin-E1/G1/S-specific cyclin-E2'
LigandChemical structure of BindingDB Monomer ID 50378304BDBM50378304(CHEMBL568080)
Affinity DataIC50: 0.0300nMAssay Description:Inhibition of Cdk2/cyclinEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50378288BDBM50378288(CHEMBL567434)
Affinity DataIC50: 0.0300nMAssay Description:Inhibition of Cdk2/cyclinEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50378289BDBM50378289(CHEMBL565705)
Affinity DataIC50: 0.0400nMAssay Description:Inhibition of Cdk2/cyclinEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50378290BDBM50378290(CHEMBL568310)
Affinity DataIC50: 0.0400nMAssay Description:Inhibition of Cdk2/cyclinEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50378291BDBM50378291(CHEMBL568302)
Affinity DataIC50: 0.0400nMAssay Description:Inhibition of Cdk2/cyclinEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50378319BDBM50378319(CHEMBL568303)
Affinity DataIC50: 0.0400nMAssay Description:Inhibition of Cdk2/cyclinEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50378305BDBM50378305(CHEMBL583417)
Affinity DataIC50: 0.0400nMAssay Description:Inhibition of Cdk2/cyclinEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50378292BDBM50378292(CHEMBL566106)
Affinity DataIC50: 0.0500nMAssay Description:Inhibition of Cdk2/cyclinEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50003691BDBM50003691(CHEMBL567624)
Affinity DataIC50: 0.0500nMAssay Description:Inhibition of Cdk2/cyclinEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50378293BDBM50378293(CHEMBL566550)
Affinity DataIC50: 0.0600nMAssay Description:Inhibition of Cdk2/cyclinEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50378294BDBM50378294(CHEMBL566972)
Affinity DataIC50: 0.0700nMAssay Description:Inhibition of Cdk2/cyclinEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50378295BDBM50378295(CHEMBL565490)
Affinity DataIC50: 0.0800nMAssay Description:Inhibition of Cdk2/cyclinEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50378296BDBM50378296(CHEMBL568510)
Affinity DataIC50: 0.0900nMAssay Description:Inhibition of Cdk2/cyclinEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50378297BDBM50378297(CHEMBL566105)
Affinity DataIC50: 0.0900nMAssay Description:Inhibition of Cdk2/cyclinEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50378298BDBM50378298(CHEMBL583421)
Affinity DataIC50: 0.0900nMAssay Description:Inhibition of Cdk2/cyclinEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50378299BDBM50378299(CHEMBL568079)
Affinity DataIC50: 0.0900nMAssay Description:Inhibition of Cdk2/cyclinEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50378301BDBM50378301(CHEMBL568311)
Affinity DataIC50: 0.100nMAssay Description:Inhibition of Cdk2/cyclinEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50378302BDBM50378302(CHEMBL583615)
Affinity DataIC50: 0.100nMAssay Description:Inhibition of Cdk2/cyclinEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50378303BDBM50378303(CHEMBL567208)
Affinity DataIC50: 0.100nMAssay Description:Inhibition of Cdk2/cyclinEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50378212BDBM50378212(CHEMBL575450)
Affinity DataIC50: 0.100nMAssay Description:Inhibition of Cdk2/cyclinEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50378300BDBM50378300(CHEMBL565930)
Affinity DataIC50: 0.100nMAssay Description:Inhibition of Cdk2/cyclinEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50378307BDBM50378307(CHEMBL566329)
Affinity DataIC50: 0.150nMAssay Description:Inhibition of Cdk2/cyclinEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50378311BDBM50378311(CHEMBL568301)
Affinity DataIC50: 0.200nMAssay Description:Inhibition of Cdk2/cyclinEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50378312BDBM50378312(CHEMBL578664)
Affinity DataIC50: 0.200nMAssay Description:Inhibition of Cdk2/cyclinEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50378313BDBM50378313(CHEMBL567626)
Affinity DataIC50: 0.200nMAssay Description:Inhibition of Cdk2/cyclinEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50378314BDBM50378314(CHEMBL578256)
Affinity DataIC50: 0.200nMAssay Description:Inhibition of Cdk2/cyclinEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50378308BDBM50378308(CHEMBL568509)
Affinity DataIC50: 0.200nMAssay Description:Inhibition of Cdk2/cyclinEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50378309BDBM50378309(CHEMBL568093)
Affinity DataIC50: 0.200nMAssay Description:Inhibition of Cdk2/cyclinEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50378310BDBM50378310(CHEMBL566971)
Affinity DataIC50: 0.200nMAssay Description:Inhibition of Cdk2/cyclinEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50378315BDBM50378315(CHEMBL578865)
Affinity DataIC50: 0.300nMAssay Description:Inhibition of Cdk2/cyclinEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50378316BDBM50378316(CHEMBL568291)
Affinity DataIC50: 0.300nMAssay Description:Inhibition of Cdk2/cyclinEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50378317BDBM50378317(CHEMBL565273)
Affinity DataIC50: 0.400nMAssay Description:Inhibition of Cdk2/cyclinEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50378318BDBM50378318(CHEMBL566539)
Affinity DataIC50: 0.400nMAssay Description:Inhibition of Cdk2/cyclinEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 7533BDBM7533(2,6,9-Trisubstituted purine deriv. 28 | (2R)-2-[[6...)
Affinity DataIC50: 0.520nMAssay Description:Inhibition of Cdk2/cyclinEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50378306BDBM50378306(CHEMBL567647)
Affinity DataIC50: 0.950nMAssay Description:Inhibition of Cdk2/cyclinEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50611455BDBM50611455(CHEMBL5286090)
Affinity DataKi:  1nMAssay Description:Inhibition of CDK2/cyclin E (unknown origin) assessed as inhibition constant incubated for 30 to 60 mins presence of dithiothreitol by Cheng-Prusoff ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
LigandChemical structure of BindingDB Monomer ID 370121BDBM370121(6-(difluoromethyl)-8-[(1R,2R)-2-hydroxy-2-methylcy...)
Affinity DataKi:  1nMAssay Description:Inhibition of CDK2/cyclin E (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMedPDB3D3D Structure (crystal)
LigandChemical structure of BindingDB Monomer ID 50139171BDBM50139171(Dinaciclib | MK-7965 | SCH-727965 | US11643396, Ex...)
Affinity DataKi:  1nMAssay Description:Inhibition of CDK2/cyclin E (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
LigandChemical structure of BindingDB Monomer ID 2579BDBM2579(CHEMBL388978 | Staurosporine, 8 | Staurosporin, 4 ...)
Affinity DataIC50: 1nMAssay Description:Inhibition of CDK2/cyclin E (unknown origin) after 40 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2016
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50299138BDBM50299138((S)-1-(4-(5-cyclopropyl-1H-pyrazol-3-ylamino)pyrro...)
Affinity DataIC50: 2nMAssay Description:Inhibition of CDK2/Cyclin E after 60 mins by fluorescence electrophoresisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50338873BDBM50338873(N-(5-Amino-1-(4-methoxybenzyl)-1H-pyrazol-4-yl)-5-...)
Affinity DataIC50: 2.13nMAssay Description:Inhibition of CDK2/cyclin EMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2013
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50193093BDBM50193093(RGB-286638)
Affinity DataIC50: 3nMAssay Description:Inhibition of CDK2/cyclin E (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
LigandChemical structure of BindingDB Monomer ID 50431360BDBM50431360(CHEMBL2347597)
Affinity DataKi:  3nMAssay Description:Inhibition of CDK2/cyclin E (unknown origin) assessed as inhibition constant incubated for 30 to 60 mins presence of dithiothreitol by Cheng-Prusoff ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
LigandChemical structure of BindingDB Monomer ID 50431360BDBM50431360(CHEMBL2347597)
Affinity DataKi:  3nMAssay Description:Inhibition of CDK2/cyclin E (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
LigandChemical structure of BindingDB Monomer ID 50615309BDBM50615309(CHEMBL5285888)
Affinity DataIC50: 4nMAssay Description:Inhibition of CDK2/cyclin E (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2024
Entry Details
PubMed
LigandChemical structure of BindingDB Monomer ID 50615312BDBM50615312(CHEMBL5287185)
Affinity DataIC50: 4nMAssay Description:Inhibition of CDK2/cyclin E (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2024
Entry Details
PubMed
LigandChemical structure of BindingDB Monomer ID 50615310BDBM50615310(CHEMBL5278558)
Affinity DataIC50: 4nMAssay Description:Inhibition of CDK2/cyclin E (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2024
Entry Details
PubMed
LigandChemical structure of BindingDB Monomer ID 50615311BDBM50615311(CHEMBL5288780)
Affinity DataIC50: 4nMAssay Description:Inhibition of CDK2/cyclin E (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2024
Entry Details
PubMed
LigandChemical structure of BindingDB Monomer ID 50593923BDBM50593923(CHEMBL5195030)
Affinity DataKi:  5nMAssay Description:Inhibition of CDK2/cyclin E (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
LigandChemical structure of BindingDB Monomer ID 5718BDBM5718(2,6,9-Trisubstituted purine deriv. 26 | 2-{[6-(ben...)
Affinity DataIC50: 5nMAssay Description:Inhibition of CDK2/cyclin E (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2024
Entry Details
PubMedPDB3D3D Structure (crystal)
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