BDBM50653426 Conivaptan

SMILES Cc1nc2c([nH]1)-c1ccccc1N(C(=O)c1ccc(NC(=O)c3ccccc3-c3ccccc3)cc1)CC2

InChI Key

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50653426   

TargetVasopressin V2 receptor(Human)
Gedeon Richter Plc

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50653426BDBM50653426(Conivaptan)
Affinity DataKi:  0.600nMAssay Description:Inhibition of BACE1 (unknown origin) by cell based assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/3/2026
Entry Details PubMed
TargetVasopressin V1a receptor(Human)
Gedeon Richter Plc

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50653426BDBM50653426(Conivaptan)
Affinity DataKi:  2.90nMAssay Description:Positive allosteric modulation of human mGlu4 receptor by cell based calcium mobilizationMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/3/2026
Entry Details PubMed