BDBM50666465 CHEMBL6163448

SMILES C=CC(=O)Nc1ccc(NC(=O)c2ccc(C)c(C#Cc3cnc4cccnn34)c2)c2ccccc12

InChI Key

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 5 hits for monomerid = 50666465   

TargetMast/stem cell growth factor receptor Kit(Human)
TU Dortmund University and Drug Discovery Hub Dortmund (DDHD)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50666465BDBM50666465(CHEMBL6163448)
Affinity DataIC50: 0.600nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/6/2026
Entry Details PubMed
TargetPlatelet-derived growth factor receptor alpha(Human)
TU Dortmund University and Drug Discovery Hub Dortmund (DDHD)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50666465BDBM50666465(CHEMBL6163448)
Affinity DataIC50: 1.80nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/6/2026
Entry Details PubMed
TargetMast/stem cell growth factor receptor Kit(Human)
TU Dortmund University and Drug Discovery Hub Dortmund (DDHD)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50666465BDBM50666465(CHEMBL6163448)
Affinity DataIC50: 198nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/6/2026
Entry Details PubMed
TargetPlatelet-derived growth factor receptor alpha(Human)
TU Dortmund University and Drug Discovery Hub Dortmund (DDHD)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50666465BDBM50666465(CHEMBL6163448)
Affinity DataIC50: 257nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/6/2026
Entry Details PubMed
TargetPlatelet-derived growth factor receptor alpha(Human)
TU Dortmund University and Drug Discovery Hub Dortmund (DDHD)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50666465BDBM50666465(CHEMBL6163448)
Affinity DataIC50: 305nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/6/2026
Entry Details PubMed